iupac (4R)-5,8-dichloro-N,2-bis(methylsulfanyl)-4-(3-phenylpropoxy)-6H-isochromeno[4,3-b]pyridine-3-carboxamide 2,3-dioxospiro[7H-benzo[a]phenalene-9,4'-piperidine]-1'-carboxylic acid (Z)-3-[4,5-dimethoxy-2-[(4-nitrophenyl)methylsulfanyl]phenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile N-(furan-2-ylmethyl)-N'-[1-[4-(2-phenylethoxy)anilino]ethenyl]propanediamide (E)-3-[6-[5-amino-4-fluoro-2-(trideuteriomethyl)phenyl]imidazo[1,2-a]pyridin-3-yl]but-2-enal 3-[3-(2,5-dimethylphenoxy)piperidin-1-yl]pyrazine-2-carbonitrile N-[(2-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-3-carboxamide;hydrochloride 1-[(4aS,8aS)-2-[[3-chloro-5-(trifluoromethyl)phenyl]methyl]-3,4,4a,5,7,8,8a-octahydro-1H-pyrido[4,3-d]azepin-6-yl]ethanone 3,5-diamino-6-methyl-1H-quinoxaline-2-thione 4-[6-amino-5-(4-phenoxycyclohexen-1-yl)pyrimidin-4-yl]oxypiperidine-1-carboxylic acid 1-(2,6-dimethylphenyl)-3-[1-[2-fluoro-4-(trifluoromethoxy)anilino]cyclopentanecarboximidoyl]urea 4-[3-chloro-5-(cyclohexylamino)sulfanylphenyl]sulfanylaniline N-[5-(azidomethyl)pyridin-2-yl]-4-fluorobenzenesulfonamide 1-butyl-3,4,5-trimethoxypyrazole (3R)-3-[7-chloro-5-(4-fluorophenyl)-2,2-dioxo-1H-pyrido[4,3-b][1,4]oxazin-8-yl]pyrrolidine-1-carbonitrile 6-amino-5-(3-ethoxybutanoyl)-1H-pyrimidine-2,4-dione 4-[5-[2,3-difluoro-6-(1-oxothian-4-yl)oxyphenyl]pyridin-3-yl]-N-methylbenzenesulfonamide 2-[4-[5-(dimethylamino)-6-fluoropyridine-3-carbonyl]-1,4-diazepan-1-yl]acetamide 2-amino-6-(1,3-thiazol-2-yl)phenol;6,9,13-trimethoxy-4-azatricyclo[10.4.0.02,7]hexadeca-1(12),13,15-triene N-(2,2-dimethoxyethyl)-3,7-dihydroxynaphthalene-1-sulfonamide 3-N,4-N-bis(4-methylphenyl)cyclohexa-1,5-diene-1,4-diamine 6-cyclohexyl-3-[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-1H-pyridin-2-one;N'-hydroxyheptanediamide 2-[(5S,10bR)-5-thiophen-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 5-(2,3-difluorophenyl)-1-methyl-4-methylidenepyridazine 2-[[2,5-bis(trifluoromethyl)phenyl]iminomethyl]-6-tert-butyl-4-sulfanylidenecyclohexa-1,3-dien-1-ol 3-(2-chlorophenyl)-5-[1-methoxy-6-(trifluoromethyl)cyclohexa-2,4-dien-1-yl]-N-[(Z)-prop-1-enyl]pyrazolo[1,5-a]pyrimidin-7-amine 2-(3-ethoxycyclobutyl)sulfonylpyridine 2-(3,5-dimethylphenyl)-4,4-difluoropiperidine 1-N,5-N,2,2-tetraphenyl-4,5,6,7,8-hexahydro-3H-quinoline-4,5-diamine 6-methyl-4-[3-[(1R)-2-piperidin-1-ylcyclopentyl]phenyl]pyridine-2,5-dicarboxylic acid 5-(aminomethyl)-3-cyclopropyl-4,7-difluoro-1-[4-(2,2,2-trifluoroethoxy)phenyl]sulfonylindole-6-carbonitrile 3-methyl-1,5-di(propan-2-yl)pyrazolo[3,4-c]pyridazine 3-ethoxycarbonyl-4-methylbenzoic acid (7S)-7-[4-(difluoromethoxy)phenyl]-N-(2,4-dimethylphenyl)-5-methyl-3-thiophen-2-yl-6,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide 4-(N-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-propan-2-ylanilino)butan-1-ol 2-amino-4-[3-chloro-4-(trifluoromethoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile 1-[6,6-dimethyl-5-(2-morpholin-4-ylethoxy)thieno[2,3-b]pyrrol-7-yl]ethanone 4-(2,4-dihydroxyphenyl)benzenecarboximidamide 5-(5,6-dichlorobenzimidazol-1-yl)-N-[2-(4-methoxyphenyl)ethyl]pentanamide N-(3-methylbutyl)-2,4,6-trinitro-N-octylaniline 4-(2-methoxyphenyl)-3,5,6,7-tetrahydrocyclopenta[d]pyridazine 2-methyl-4,6-bis[3-(1H-pyrazol-5-yl)anilino]phenol (NZ)-N-[[3-(4-bromophenyl)-4-oxo-1,3-thiazolidin-2-ylidene]methyl]benzenesulfonamide N-azido-4-(1,3-benzodioxol-5-yl)butanamide 3-[[2,4-bis(methylamino)pyrimidine-5-carbonyl]amino]propylcarbamic acid 4-azidooxy-2,3-dibromobenzaldehyde 5-[4-chloro-3-(1,3-dioxolan-2-yl)phenyl]-N-pyridin-2-yl-1H-pyrrole-3-carboxamide 3-[2-methyl-6-(4,5,8,10-tetrahydrothieno[3,2-d]azocine-6-carbonyl)phenyl]propanal [(2S,4S)-1-[2-[cyclopentylmethoxy(methyl)amino]acetyl]-4-fluoropyrrolidine-2-carbonyl]azanium;2-methylpropane 5-[3-[(2R)-2,6-dimethylmorpholine-4-carbonyl]phenyl]-6-oxo-1H-pyridazine-3-carboxylic acid N-[(E)-2-aminoethenyl]-N-(1,3-benzodioxol-5-yl)formamide;2-methoxyacetamide 5-amino-4-(3,4-dimethylphenyl)imino-2,2,6,6-tetramethylpyran-3-carbonitrile (3S,4R)-1-[5-fluoro-2-methoxy-4-(2-phenylsulfanylacetyl)phenyl]sulfonylpiperidine-3,4-dicarboxamide 3-bromo-5,7-diethylpyrazolo[1,5-a]pyrimidine N-cyclohexa-2,4-dien-1-yl-4-phenylbenzenesulfonamide 2-azido-N'-[(Z)-benzylideneamino]propanehydrazide 2-(cyclohexylamino)-5-[(4R,6S)-3,8-dimethyl-7-oxo-6-propan-2-yl-1-oxabicyclo[3.2.0]hepta-2,4-dien-7-yl]benzenesulfonamide 4-(2,3-dihydrothiophen-5-yl)thieno[3,2-b]pyrrole 2-[(3R,6S)-1-(cyclopropylmethylsulfonyl)-6-propan-2-ylpiperidin-3-yl]oxypyrazine 6-bromo-5,7-dihydroindolo[2,1-a]isoquinoline 7-methoxy-1-[(5R)-3,4,8-trihydroxy-5,6,7,8-tetrahydronaphthalene-2-carbonyl]-6,7-dihydroquinolin-4-one 2-[4-[1-(cyclohexylmethoxy)ethyl]phenyl]benzamide 2-[2-(3,5-difluorophenoxy)phenyl]propanoic acid (2R)-2-[[3-[4-[(3,5-dichlorophenyl)sulfanylamino]phenyl]-1H-pyrazolo[3,4-b]pyridine-6-carbonyl]amino]propanoic acid 1-(2,6-diphenylpyrimidin-4-yl)propan-1-one (5R)-7,8-dimethoxy-2,2,3,4-tetrahydropyrano[3,2-c]quinoline 4-fluoro-N-[(2R,3S)-2-methyl-1,1,1-trideuterio-5-hydroxy-4-oxopentan-3-yl]benzamide 1-azidooxy-2,3,4,5,6-pentafluoro-7-methylnaphthalene (1S)-3-azido-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine 1,3-bis(4-methoxyphenyl)propane-2,3-diamine 4-[2-(5-methyl-1,3-thiazol-2-yl)ethylsulfamoyl]benzoic acid 1-[(2,4-dimethylphenyl)methyl]-3,4-bis[2-(trifluoromethoxy)phenyl]-1,3,5-triazinan-6-one 3-[2-(2,6-dioxopiperidin-4-yl)-1-oxoisoquinolin-5-yl]oxypropanenitrile 1-chloro-4-(2,5,5-trifluoropentan-3-yl)benzene (1-aminocyclopentyl)-[4-(2,6-difluorophenoxy)piperidin-1-yl]methanone;hydrochloride 5-(3,6-dichlorocarbazol-9-yl)-2-fluorobenzoic acid 5-[[2,3-dimethoxy-6-(morpholine-4-carbonyl)phenyl]carbamoylamino]-1H-pyrrole-2-carboxamide 7,8-dichloro-2-oxopyrano[4,3-b]chromene-3-carbonitrile 2-(6,8-dimethylimidazo[1,5-a]pyridin-3-yl)-N-[5-hydroxypentanoyl]acetamide 4-(1,3-benzodioxol-5-yl)-5-chlorodithiol-3-one 6-ethyl-1,2-bis(2-methoxyphenyl)cyclohexa-3,5-diene-1,3-diamine 2-[4-(dimethylamino)-N-methylsulfonylanilino]propanoic acid 3-[5-cyano-4-(cyclobutylamino)pyridin-2-yl]-1-(4-formamidophenyl)-N,N-dimethylpyrazole-4-carboxamide 2-N,1-bis(4-fluorophenyl)-3-[4-(4-methylsulfonylpiperazin-1-yl)cyclohexa-2,4-dien-1-ylidene]propane-1,2-diimine 2-N-[3-(1H-imidazol-5-yl)propyl]-4-N-methyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-2,4-diamine;dihydrochloride [2-(4-acetylpiperazin-1-yl)-5-methoxyphenyl]azanide 1-[(E)-4,5-dimethoxypent-3-enyl]-4-propan-2-ylidenepyridine;ethane 1-(2,6-dimethylphenyl)-3-[(E)-4,8,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-11-ylideneamino]thiourea 4-(5,6-dimethylindazol-1-ium-2-yl)-3-methoxy-N'-[(Z)-3-(4-pyridin-3-ylpiperazin-1-yl)prop-1-enyl]benzenecarboximidamide N-[[2,6-dichloro-4-(trifluoromethyl)phenyl]methylideneamino]-1H-pyrazole-3-carboxamide 5-amino-2,4-dihydroxy-3-(oxolan-2-ylmethoxy)benzaldehyde 5-[4-[4-amino-6,7-dimethyl-2-(2H-tetrazol-5-yl)benzimidazol-1-yl]piperidine-1-carbonyl]pyrrolidin-2-one 5-[6-chloro-7-(oxan-4-ylmethoxy)quinolin-2-yl]pyrimidine-2,4-diamine 2-[3-methylbut-2-enyl(1,3-thiazol-5-yl)amino]propanoic acid 4-(4,6-dimethoxypyrimidin-2-yl)piperazine-1-carboxylic acid 1-[2-(cyclopropylamino)pyrimidine-5-carbonyl]-N-phenylazetidine-3-carboxamide 5-[2,4-diamino-6-(3,4-dimethylphenyl)pyrimidine-5-carboximidoyl]-N-pyridin-2-yl-1H-pyrrole-3-carboxamide N-(cyclopropylmethoxy)-4-[3-(1H-pyrazol-5-yl)phenyl]-2,3-dihydro-1,4-benzoxazine-6-carboxamide 1-(5,7-difluoroquinolin-4-yl)-N,N',2-trimethoxypropane-1,3-diamine (2R)-1-[4-[8-chloro-4-[4-methoxy-3,5-di(propan-2-yl)phenyl]imidazo[1,5-a]pyrazin-6-yl]piperazin-1-yl]-3-fluoro-2-hydroxypropan-1-one 1-(3-aminophenyl)indole-6-carboxylic acid 4-[1-(3,5-dichloropyridin-2-yl)pyrrolidin-3-yl]oxy-N-ethylpyrimidine-5-carboxamide 4-fluoro-1-(2-methylpropyl)-7-methylidene-8-[2-methyl-5-(trifluoromethyl)pyridin-3-yl]-6,9-dihydro-3H-pyrido[3,4-b]indole 4-fluoro-N-(5-pyridin-4-ylsulfanylpyrimidin-2-yl)benzamide 5-[2,6-difluoro-4-(2-methylpyridin-3-yl)phenyl]-1-[2,6-difluoro-3-(propanoylamino)benzoyl]-N-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide (E)-4,4,5,6-tetrachloro-2-[4-(difluoromethoxy)phenyl]hex-1-en-3-one 4-tert-butyl-5-[3-(4,6-diphenylpyrimidin-2-yl)benzenecarboximidoyl]-2,6-dimethoxyaniline (2S)-1-[3,4-bis(difluoromethoxy)benzoyl]-N'-[5-bromo-6-fluoro-7-[2-(trideuteriomethylamino)ethylcarbamoyl]naphthalen-2-yl]piperidine-2-carboximidamide 1-[4-(6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-2-yl)piperazin-1-yl]ethanone 1-[4-(ethylamino)-2-methylphenyl]-3-(N'-phenylcarbamimidoyl)urea 2-[3-(6,7-dihydro-5H-cyclopenta[b]pyridine-5-carbonyl)phenyl]propanoic acid 1-(4-azido-3-methoxyphenyl)sulfonylpiperidine N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-5-methyl-1H-pyrazole-3-carboxamide (1R)-2-[[(E,4S)-3-[6-[2,6-dimethyl-4-(2-methylpropoxycarbonylamino)phenyl]pyridine-3-carbonyl]oxy-1-oxohept-5-en-4-yl]amino]cyclopentane-1-carboxylic acid N-[2-(3-azidophenyl)ethyl]pyrimidine-4-carboxamide N'-(3-benzylsulfonyl-2,6-dinitrophenyl)ethane-1,2-diamine (4-aminophenyl)methyl-ethylamino-[4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl]azanium 4-tert-butyl-6-(2,3-dihydro-1H-inden-5-ylmethyl)pyrimidine N-[4-(difluoromethoxy)phenyl]-2-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine;1-(2,3-dihydro-1H-pyrrol-4-ylamino)propan-1-one N-[1,4-bis(6-methylpyrimidin-4-yl)cyclohexa-2,4-dien-1-yl]benzamide N-[(4-methoxyphenyl)methyl]-2-[(6S)-2-methyl-7-oxo-4,5,6,8-tetrahydrocyclohepta[d][1,3]thiazol-6-yl]acetamide 2,3-difluoro-N-(1H-imidazo[4,5-b]pyridin-6-yl)benzenesulfonamide 2-cyclohexylsulfanylethyl(diphenyl)phosphane;rhenium (3S)-3-[4-[5-chloro-2,6-difluoro-3-(1H-pyrazolo[3,4-b]pyridine-4-carbonylamino)phenoxy]piperidin-1-yl]butanoic acid [1-(2,3-dihydroindol-1-yl)-2H-naphthalen-1-ylidene]oxidanium 4-(6-bromo-2,3,4a,5,7,8,9,9a-octahydro-1H-pyrido[4,3-b]indole-1-carbonyl)benzonitrile N-[6-[(3R,5S)-3,4,5-trimethylpiperazin-1-yl]pyridazin-3-yl]acetamide 3-chloro-N-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]-5-methylbenzenesulfonamide 3-[4-(diethylaminomethyl)phenyl]-5-(1,2-thiazol-3-yl)furan-2-carboxamide;hydrochloride (1S)-2,3,4,5,6,10,11b-octahydrocyclopenta[b]quinolizine N-[(5R)-3-(5-oxo-2,4,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)-5-thiophen-2-yl-8-azatricyclo[7.4.0.02,7]trideca-1(9),10,12-trien-12-ylidene]benzenesulfonamide N-(3-chlorophenyl)-2-[7-ethyl-5-(4-methoxyphenyl)-6-(1,3-oxazol-2-yl)-9-oxo-1,2,6,11b-tetrahydrobenzo[b][1,4]benzoxazepin-10-yl]acetamide 1-(dimethoxyphosphorylmethyl)naphthalene 3-[(2S)-6-amino-5-oxo-2-phenylcyclopenten-1-yl]butanoic acid (1-aminocyclopentyl)-[4-methoxy-7-(4-propan-2-ylphenyl)-3,5-dihydro-2H-1,4-benzodiazepin-1-yl]methanone 4-(2,4-difluorophenyl)-N-[1-(5-ethylsulfanylpyridin-3-yl)-2-hydroxyethylidene]piperidine-1-carboxamide 5-methyl-1-phenyltetrazole (3R)-2,6-dioxopiperidine-3-carbohydrazide;5-hydroxy-4-[1-phenylethyl-[(4-phenylmethoxyphenyl)methyl]amino]pentanoic acid 1-(4-azidophenyl)-3,5-dimethylpyrazole 2-[2-[[1-(benzenesulfonyl)piperidin-4-yl]amino]pyrimidin-5-yl]-6-bromo-N,5-dimethylpyrrolo[3,2-d]pyrimidin-4-amine (6R)-N-benzyl-8,8-dimethyl-2-[4-[3-(trifluoromethoxy)phenyl]piperidine-1-carbonyl]-5,7,9,10-tetrahydro-4H-pyrazolo[3,4-b][1,7]naphthyridine-6-carboxamide 5-bromo-3,3a,4,5,6,7,8,8a-octahydroimidazo[2,1-c][1,4]oxazin-2-one 4-[(3R)-3,7-dimethyloct-6-enoyl]-1H-pyrrole-2-carboxylic acid 1-(4,6-dichloro-2-phenylpyrimidine-5-carbonyl)-3-methylimidazolidin-4-one 1-ethyl-N-(oxan-4-yl)pyrazole-3-carboxamide 2-[6,6-dimethyl-3-[4-(4-phenylpiperidin-1-yl)piperidine-1-carbonyl]-5,7-dihydro-4H-indazol-1-yl]-1-morpholin-4-ylethanone 4-azidooxy-5-[(2,3-dimethylbenzimidazol-5-yl)amino]pentanenitrile 5-(3,4-dichlorophenoxy)-1H-indole (5E)-2-(4-ethoxyphenyl)imino-5-[[1-(naphthalen-1-ylmethyl)indol-3-yl]methylidene]-1,3-thiazolidin-4-one 2-(2,6-dioxopiperidin-3-yl)-4-[[1-[1-(4-hydroxyphenyl)ethyl]piperidin-4-yl]methoxy]isoindole-1,3-dione;hydrochloride [(3S,5R)-4-[6-[4-fluoro-2-(trifluoromethyl)anilino]purin-9-yl]-3,5-dihydroxycyclohexyl]methylcarbamic acid (4S)-1,3-dimethyl-4-[2-methyl-5-(2-morpholin-4-ylethoxy)phenyl]-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one N-(2,6-dimethoxypyrimidin-4-yl)-4-[3-nitro-N-(1,3-thiazol-5-yl)anilino]benzenesulfonamide 3-cyclopropyl-N-[5,6-dichloro-1-(2-oxobut-3-enoxy)benzimidazol-2-yl]methanesulfonamide [2,3-bis(propanoylamino)phenyl]carbamic acid 1-(5-ethylsulfanylpyridin-3-yl)-7-methoxy-2H-quinoline 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]pyridine;6-methoxy-7-methyl-2-propan-2-ylidenechromene 4-chloro-2-fluoro-N-(3-methyl-1,3-benzothiazol-3-ium-6-yl)benzenesulfonamide 5-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)acetyl]cyclohexane-1-carboxylic acid (E)-5,5,5-trifluoro-4-hydroxy-1-[2-[4-[1-(1H-pyrazol-5-ylmethyl)piperidine-4-carbonyl]anilino]-1,3-thiazol-4-yl]pent-2-en-1-one 2-[(1S)-1-azido-5-methylhexyl]pyridine (2-hydroxy-1H-indol-3-yl)-oxomethanesulfonate 3-methyl-1-[1-methyl-3-[(2S)-6-methylideneoxan-2-yl]oxypyrrolo[3,4-c]pyridin-5-yl]pentan-3-amine 5-(4-phenylcyclohexyl)oxy-N,2-di(propan-2-yl)pyrimidine-4-carboxamide 5-(2,4-dimethoxyphenyl)-3-ethyl-6H-1,3,4-thiadiazin-2-one 2-[4-(4-benzoylphenyl)-1,3-thiazol-2-yl]-N'-hydroxypropanehydrazide 1-[2-fluoro-6-hydroxy-3-(methoxyamino)phenyl]ethanone 3-[4-[(E)-2-cyclopropylethenoxy]phenyl]-7,8-difluoro-6H-pyrrolo[1,2-a]pyrazine [2-(azidomethyl)phenyl]-(1H-indol-2-yl)carbamic acid N-[5-[3-[4-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-yl]butanamide 1-azido-4,5-bis(chloromethyl)-2-methoxybenzene 4-[1,3-dihydroisoindole-2-carbonyl(hydroxy)amino]-3-methylbutanamide;6,7,8-trimethoxy-5H-quinazolin-4-amine 3-[5-chloro-6-(hydroxymethyl)pyridin-2-yl]cyclohexane-1,3-dione 2-[4-bromobutan-2-yl-(8-hydroxy-6-sulfonaphthalen-2-yl)amino]decanoic acid N-[(4S)-3,4-dihydro-2H-chromen-7-yl]-5-methyl-1-(8-oxooctyl)triazole-4-carboxamide 1,3-dibromo-2-(chloromethyl)benzene;ethane 3-[(1,1-dioxothiolan-2-yl)methoxy]-N-ethylpyridine-4-carboxamide 4-(2,3-dichlorophenyl)benzo[h]quinazoline 3-[2-azidooxy-1-(4-pyridin-2-ylphenyl)ethoxy]propanenitrile (4Z)-2-methyl-4-[[5-[3-(1,3-oxazol-2-yl)propylamino]pyrazin-2-yl]methylidene]cyclohexa-1,5-dien-1-amine N-[2,3-bis(ethenyl)-5-methoxyphenyl]prop-2-ynamide [(2S)-4-(5,6,7,8-tetrahydronaphthalene-1-carbonylamino)butan-2-yl]carbamic acid 4-(3,5-dimethylphenyl)-2H-triazole 2-[(2E,5S)-3-methyl-4-oxo-2-(pentanoylhydrazinylidene)-1,3-thiazolidin-5-yl]benzoic acid (2S)-1-(3,5-difluorobenzoyl)-N-[4-[4-[[[cyclobutylidene(hydroxy)methoxy]amino]carbamoyl]phenyl]pyridin-3-yl]pyrrolidine-2-carboxamide 2-bromo-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N-hexadecanoylbenzamide (2R,3S)-3-amino-4-(3-fluorophenyl)-2-hydroxybutanoic acid 3-hydroxy-5,8-dimethyl-2-(4,7,8-trimethylnonanoyl)naphthalene-1,4-dione N-butanoyl-N-methylbenzamide 4-[(2E,4Z)-5-methoxypenta-2,4-dien-3-yl]-5-[4-[2-(4-prop-1-ynylphenyl)ethynyl]phenyl]-1H-imidazole 4-N,6-bis(cyclopropylmethyl)-3-(difluoromethyl)-1-N,2-N-dimethylbenzene-1,2,4-triamine (5E)-5-[(4-bromo-1,3-benzodioxol-5-yl)methylidene]-2-imino-1,3-thiazolidin-4-one 1-[5-[4-(difluoromethyl)pyrimidin-2-yl]oxy-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]-2,2-dihydroxy-4-oxobutan-1-one 6-cyclopropyl-N-methyl-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)quinoline-4-carboxamide 2-methoxy-3,4-disulfobenzoic acid (3S,4S)-1-cyclobutyl-4-[1-[[6-[2-methoxyethyl(methyl)amino]pyridin-3-yl]methyl]piperidin-4-yl]pyrrolidine-3-carboxylic acid;dihydrochloride 3-(2,6-dimethylphenoxy)-N-(1-hydroxybutan-2-yloxy)propane-1-sulfonamide 1-[(2S,4R)-5-bromo-3,4-dihydroxy-6-methoxyoxan-2-yl]pyrimidine-2,4-dione 2-[4-methoxy-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)anilino]decanoic acid N-[4-methoxy-2-(methylamino)phenyl]-3H-thiadiazole-2-carboxamide 1-(4,5-diethylthiophen-2-yl)sulfonylpiperidine 2-[(7-cyano-6-methyl-1,3-benzothiazol-2-yl)diazenyl]-5-[(4-ethoxynaphthalen-1-yl)sulfonylamino]benzoic acid 2-(4,5-difluorocyclohexa-1,3-dien-1-yl)oxyphenol N-cyclopropyl-4-[3-(2,6-dichloroanilino)pyridin-4-yl]benzenesulfonamide 2-cyclohexylethylphosphane;3-methylpentan-1-one;pentane;6-propylspiro[3H-chromene-2,4'-piperidine] N-methylsulfonyl-2-(3-nitro-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)acetamide;hydrochloride N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-octylacetamide N-[(5-methylpyrazin-2-yl)methyl]thieno[3,2-d]pyrimidin-4-amine 4-[(Z)-4,5-dihydroxy-1-phenylpent-3-enoxy]benzenesulfonamide 1-[4-(cyclobutylmethoxy)phenyl]pentan-2-one 2-benzylsulfanyl-4,5-dichlorothiophene;hydrochloride (E)-3-[5-hydroxy-4,6-dimethoxy-7-(4-nitrosophenoxy)naphthalen-2-yl]prop-2-enal (2R)-2-methyl-3,4-bis[4-(pyridin-2-ylamino)butyl]cyclohexan-1-one 1-[[2,4-difluoro-3-(trifluoromethyl)phenyl]methoxycarbonylamino]cyclopentane-1-carboxylic acid (3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-b]pyridin-8-yl)methanamine 4-[2,6-dimethyl-3-(prop-1-en-2-ylamino)phenyl]piperidine-1-carboxylic acid (3R)-4-[6-amino-8-(2,6-difluoro-4-hydroxyphenyl)purin-9-yl]pentane-1,3-diol (7S)-N,N-bis[(4-methoxyphenyl)methyl]-2,3-dimethyl-6-oxo-5-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyridazine-7-carboxamide 4-methyl-N,2-bis[(Z)-1H-pyrrol-3-ylmethylideneamino]-1,3-thiazole-5-carboxamide 4-[(2,5-dimethylfuran-3-carbonyl)amino]-N-propan-2-ylpiperidine-1-carboxamide 3-(2,6-dichlorophenyl)-7-[(5-methylsulfonylpyridin-2-yl)amino]-2H-pyrimido[5,4-e][1,3]thiazin-4-one 2-[(3-cyclopropylimidazol-4-yl)methyl-[4-methoxy-6-[[4-[5-(oxetan-2-yloxy)pyridin-2-yl]phenoxy]methyl]pyrimidin-2-yl]amino]ethanol 5-cyclopropyl-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-1,4,6-trimethyl-7H-pyrazolo[3,4-b]pyridine-4-carboxamide 2-(5,7-dimethyl-1H-indole-3-carbonyl)-6-phenyloxane-3,4-dione [1-methyl-3-(2-methylpropanoylamino)cyclobutyl]-[4-(pyridine-4-carbonyl)phenyl]borinic acid 3-[2-(4-methylpiperazin-1-yl)ethoxy]benzoic acid N-[4-[3-(5,7,10,11-tetrazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,8,11-hexaen-13-yl)phenyl]butyl]pyridine-4-carboxamide [3-(2,4-dichlorophenyl)-3-ethenylpentan-2-ylidene]cyanamide N-[1-(3,5-dimethylbenzoyl)-4,5-dihydroxypyrrolidin-2-yl]-2-methoxybenzamide 3-amino-6-fluoro-N'-(2-methylpyridin-4-yl)pyridine-2-carboximidamide N-[3-[(dimethylamino)methyl]phenyl]cyclohexanecarboxamide 4-(6-azidonaphthalen-1-yl)morpholine N-(2,4-dimethoxyphenyl)-1-[1-[(Z)-prop-1-enyl]indol-3-yl]-5-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide 2-methylpropane;2-methyl-5,6,7,8-tetrahydroquinoline;1-(6-methylpyridin-3-yl)-4-[3-(trifluoromethoxy)phenyl]piperazine (Z)-1,3-bis(4-methoxyphenyl)prop-2-en-1-one 4-(1,1-difluoroethyl)benzenethiol;ethane;N-[2-methoxy-5-methyl-6-(3-phenylpropylsulfanyl)pyridin-3-yl]acetamide (5R,6S)-2-amino-5-(4-propan-2-ylphenyl)cyclopentan-1-ol 3-[2-oxo-1-phenyl-7-(trifluoromethyl)pyrido[2,3-b][1,4]oxazin-8-yl]azetidine-1-carboxylic acid 5-amino-4-[(3,5-dichlorophenyl)methyl]-6-ethoxycarbonylpyridine-2-carboxylic acid 2-[2-(4-chlorophenyl)ethyl]-5-[2-methoxy-4-(trifluoromethyl)phenyl]thiophene 4-bromo-3,5-bis[(2,6-difluorophenyl)methoxy]benzaldehyde 2-(4-chlorophenoxy)-N-[6-[[5-methyl-3-(oxan-4-ylamino)cyclohexa-1,3-dien-1-yl]amino]pyridin-3-yl]acetamide N-(3-morpholin-4-ylsulfonylphenyl)-1-pentanoylpiperidine-3-carboxamide 3-azido-1,2,5-trifluoro-4-(1H-imidazol-5-yl)benzene N-[3-(2,6-dimethylpiperidin-1-yl)propyl]-2-hydroxy-5-nitrobenzamide 4-(3,7-dimethyl-2H-indazol-5-yl)piperazine-1-carboxylic acid N-(3,5-dimethylphenyl)-5,8-bis[2-(4-hydroxyphenyl)ethenyl]-4,7-dioxooctanamide N-(4-aminosulfanylphenyl)pyridine-2-carboxamide 3-(1H-indol-4-yl)-1H-thieno[2,3-d]imidazol-2-one 6-(2,5-dihydroxyphenyl)-4H-pyran-3-one;hydrobromide 4-[3-(2-aminoethylamino)propyl]-N-[1,2-dihydropyridazin-3-yl-[6-methoxy-5-(trifluoromethyl)pyridin-3-yl]carbamoyl]benzamide 2-N-azido-4-N,4-N-dipropylpyrimidine-2,4-diamine 2-[2,6-dioxo-3-[[4-(pyridin-4-ylmethyl)phenyl]methylideneamino]piperidin-1-yl]acetic acid 6-amino-2-(3,4-dihydroxyphenyl)-8-[2-[5-(1-hydroxypropan-2-yl)pyridin-3-yl]ethynyl]pyrido[2,3-d]pyrimidin-7-one 3-azidosulfanyl-5,6,7,8-tetrahydronaphthalene-1,4-dione (2R)-4,4-difluoro-1-[5-(6-hydroxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]piperidine-2-carboxamide 3-[(2-chlorobenzoyl)amino]-4-methoxycyclohexa-1,5-diene-1-carboxylate 4-[3,5-bis(trifluoromethyl)phenyl]sulfanyl-N-(4-chlorobutyl)aniline 5-methylsulfonyl-2-(3,4,5-trichlorophenyl)benzamide (1S,5R)-3-[4-methyl-6-oxo-2-[2-(2-phenylethynyl)pyridin-4-yl]-1H-pyrimidin-5-yl]-3-azabicyclo[3.1.0]hexane-1-carbonitrile 1-(4-chlorophenyl)pyrrolidine;N,3-dimethylbenzamide [(3R,4S)-1-[4-(2-ethoxyphenyl)benzoyl]-4-hydroxypyrrolidin-3-yl]-morpholin-4-ylmethanone 4-methoxy-5,10-dihydropyrimido[5,4-g]quinazolin-2-amine N-[3-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1]benzazepine-11-carbonyl)phenyl]-6-bromopyridine-3-carboxamide 4-[7-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)heptanoyloxymethyl]benzoic acid 1-[4-(dimethylamino)cyclohexyl]-2,3-dihydroindole-7-carbonitrile 2-(dimethylamino)ethyl-[1,1,1-trifluoro-3-[3-methoxy-4-[[2-[4-(4-methoxybutanoyloxy)phenyl]benzoyl]amino]phenyl]propan-2-yl]azanide 2-(N,4-diethoxycarbonylanilino)acetic acid 3-(1H-indol-2-yl)-N'-[[6-morpholin-4-yl-2-[(Z)-prop-1-enyl]pyrimidin-4-yl]methoxy]penta-2,4-dienimidamide N-methyl-1-[5-methyl-6-(2,3,4,7-tetrahydroazepine-1-carbonyl)pyridin-2-yl]piperidine-4-carboxamide (E)-2,2-dichloro-1-[5-ethyl-2-methoxy-4-(3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazol-2-yl)phenyl]pent-3-en-1-one;N-hydroxyformamide 5-[(2-methylphenyl)diazenyl]-1H-pyrazole-4-carbonitrile [(1S,6R)-6-hydroxycyclohex-2-en-1-yl]-phenylmethanone 4-amino-5-[2,6-dichloro-3-(4-hydroxybutyl)phenyl]-1H-pyrimidin-6-one N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-2-imino-5H-1,3,4-thiadiazin-6-amine 2-[1-cyclopropylethenyl(methyl)amino]propanal;N-(2,5-dimethoxyphenyl)sulfanylformamide 2-[(1R)-5,6-dichloro-1H-inden-1-yl]acetaldehyde N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)propyl]butanamide 2-(3,5-dibromophenyl)benzenethiol;ethane 3-[2-(1,5-dimethylpyrazol-4-yl)-7-oxo-3-phenylpyrazolo[1,5-a]pyrimidin-6-yl]benzenesulfonamide 6-[2-(methylamino)pyrimidin-5-yl]-N-[3-(2-methylimidazol-1-yl)phenyl]pyridine-3-carboxamide N-ethenyl-2,4-bis(trifluoromethyl)aniline;N'-[3-fluoro-5-[3-[(6R)-7-oxa-1,3-diazabicyclo[4.1.0]heptan-3-yl]propylsulfamoyl]phenyl]ethane-1,2-diamine 3-(2,4-dichlorophenyl)sulfinyl-N-[3-fluoro-5-methyl-1-[6-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-4-ylidene]propanamide 2-(dipropylamino)quinoline-6-carboxamide 1-[(2S)-5,12-dimethyl-11-[1-(3-methylidenecyclopenten-1-yl)piperidin-4-yl]-6H-indolo[2,3-b]quinolin-6-yl]ethanone N-[(5-tert-butylpyridin-2-yl)methyl]spiro[4,7-dihydrotriazolo[1,5-a]pyrazine-6,3'-pyrrolidine]-1'-carboxamide;2,2,2-trifluoroacetic acid 2-(4-chlorophenyl)-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one N-(2,3-dihydro-1H-inden-5-yl)-2-[4-oxo-2-[(E)-[(2-piperidin-1-ylacetyl)hydrazinylidene]methyl]imino-1,3-thiazolidin-5-yl]acetamide 5-(1,2-dihydroisoquinolin-5-yl)-N-[(4-fluorophenyl)methyl]-3H-pyrrole-2-carboxamide N-[4,5-bis(4-methylphenyl)cyclohexa-1,3-dien-1-yl]-N-[4-methoxy-2-(4-oxoquinazolin-3-yl)phenyl]propanamide [3-(2,6-difluoroanilino)pyrido[2,3-b]pyrazin-6-yl]-(4-methoxypiperidin-1-yl)methanone 2-(2,3-dihydrofuran-4-yl)-1H-indole-7-carboxamide 2-(furan-3-yl)-4-phenyl-1H-pyrimidin-6-one (2S)-N-[2-hydroxy-3-(3,4,5-trimethoxyphenyl)propyl]piperidine-2-carboxamide 3-chloro-N'-hydroxy-5,6-dimethylpyridazine-4-carboximidamide 2-(2,6-dioxopiperidin-3-yl)-5-[1-(1-propanoylazetidin-3-yl)pyrazol-4-yl]isoindole-1,3-dione 5-(2,6-diphenylpyridin-4-yl)-3-ethynyl-1H-indazole 1-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-5,10-bis(4-fluorophenyl)anthracen-9-one;methanol 1-(3,5-dihydroxyphenyl)-2-[5-(hydroxymethyl)cyclohexa-1,4-dien-1-yl]ethanone (3R,4S)-1-[5-chloro-1-(3-methylsulfonylpropyl)benzimidazole-2-carbonyl]-N-(2-hydroxyethyl)-3-methoxypiperidine-4-carboxamide 2-[(5R)-5-cyclopropyl-4,5-dihydro-1,3-thiazol-2-yl]phenol [3-(4-fluorophenyl)oxetan-2-yl]oxy-phenylmethanediol (2-cyclobutyloxypyridin-3-yl)-[4-(5,6,7,8-tetrahydroquinazolin-4-yl)piperazin-1-yl]methanone 4-[4-(4,7-difluoronaphthalen-1-yl)-2,3-bis(trifluoromethoxy)phenyl]piperidine 7-amino-5-(4-fluorophenyl)-1,3,6-trimethylpyrido[2,3-d]pyrimidine-2,4-dione (4S)-3-[3-fluoro-5-methoxy-4-(trifluoromethylsulfanyl)phenyl]-1,4,6,7,8,9-hexahydropyrazolo[4,3-c]quinoline 4-N,6-diethyl-2-N-[(E)-[4-hydroxy-3,5-bis(sulfanylidene)cyclohexa-1,4-dien-1-yl]methylideneamino]pyrimidine-2,4-dicarboxamide N-cyclopentyl-2,3-dimethoxybenzamide;5-(2-ethylimidazo[1,2-a]pyridin-6-yl)-3H-pyrrole-2-carboxamide 3-chloro-N,5-dimethyl-4-[4-[1-(2-pyridin-3-ylphenyl)ethylidene]piperidin-1-yl]sulfanylaniline 6-bromospiro[1,3-dihydroisoquinoline-4,1'-cyclopropane] 2-N,6-N-bis[(4-methylphenyl)methylideneamino]-1,3,5-triazine-2,4,6-triamine N-(3,4-difluorophenyl)-3-[1-hydroxyethyl(2-methoxyethyl)amino]-N'-[6-[4-(trifluoromethoxy)phenyl]pyrimidin-4-yl]propanimidamide N-[2-(4-chlorophenyl)ethyl]-6-fluoro-5,8-dihydroxy-7,8-dihydronaphthalene-1-carboxamide;methanol 1-[5-tert-butyl-2-(4,6-dimethoxypyrimidin-2-yl)pyrazol-3-yl]-3-(4-hydroxyphenyl)urea 1-[2-methyl-4-(trifluoromethoxy)phenyl]pentane-2,3-dione 4-(3,5-dichloro-2,6-dimethoxyphenyl)-N-[1-(1H-indol-2-yl)ethylideneamino]-1,3,5-triazin-2-amine 4-fluoro-5-methyl-2-(4-methylphenyl)-1,3-dihydroisoindole 1-[2-[[4-(5-fluoropyrimidin-2-yl)morpholin-3-yl]methoxy]ethyl]imidazolidine-2,4-dione 7-[1,2-bis(4-fluorophenyl)ethylidene]-3-methyl-10-oxa-2,7-diazaspiro[4.6]undecan-9-one 2-ethyl-5-[(3E)-4-pyridin-4-ylbuta-1,3-dien-2-yl]thiophene (3S,4R)-5-methyl-1-[6-oxo-4-(trifluoromethyl)-1H-pyrimidin-2-yl]piperidine-4-carboxylic acid N-[4-(aminomethyl)phenyl]-2-azidoacetamide 3-cyclobutyl-N,2-dimethoxybenzamide 2-azido-6-[1-[4-(trifluoromethoxy)phenyl]piperidin-4-yl]pyrazine 1-[2-(dimethylamino)ethyl]-N-[4-fluoro-3-(trifluoromethoxy)phenyl]cyclopropane-1-carboxamide 2-methyl-4-[3-(4-methylphenyl)sulfonylpropoxy]naphthalene 2-[1,5-bis(4-chlorophenyl)penta-1,4-dienyl]sulfanylethanethial ethane;1-(4-fluorophenyl)-N-[(6R,8S)-8-(methoxymethyl)-6-thiophen-2-yl-9-azatricyclo[5.3.0.02,7]deca-2(7),10-dien-12-ylidene]piperidine-4-carboxamide [4-(cyclohexa-1,3-dien-1-ylmethoxy)phenyl]urea (2S)-2-(4-bromophenyl)-N,3-dimethylhexanamide [(3R)-3-benzylpyrrolidin-1-yl]-[4-(2H-quinolin-1-yloxymethyl)phenyl]methanone 1-azidooxysulfanyl-2,4-dichlorobenzene 5-[3-(3,4-dimethylphenyl)buta-1,3-dien-2-yl]-2-methylidene-3H-indene 4-amino-1-(1,3-dihydroxypropan-2-yl)-2-phenylcyclohexane-1-carboxylic acid 1-[1-(2,3-dihydroindol-1-yl)ethyl]naphthalene-2,3-dithiol 2-[[4-(2-iodophenyl)phenyl]methylidene]propanedinitrile 4-[3-amino-6-(2,5-dimethylphenyl)pyrazin-2-yl]phenol 2-[(4-fluorophenyl)methyl]-8-hydroxyquinazoline-7-carboxamide ethene;N-[4-fluoro-3-(1H-pyrazol-5-ylmethyl)phenyl]formamide 5-phenyl-9H-fluorene-4,6-diol 1-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzoyl]piperidine-4-carboxylic acid 1-[4,5-dimethoxy-2-(3-oxobutanoylamino)phenyl]cyclopropane-1-carboxylic acid 2-(5,7-difluoro-1H-indole-3-carbonyl)-N'-[2-(methylamino)ethyl]propanehydrazide;hydrochloride 3-[3-(2,6-dimethylpyridin-4-yl)oxyphenyl]oxirane-2,2-dicarbonitrile [2-chloro-4-[(E)-2-[6-methyl-5-(trifluoromethoxy)pyridin-3-yl]ethenyl]phenyl]phosphane 4-chloro-5,6-dimethoxy-2-(trifluoromethyl)pyrimidine 4-[7-[3-(tert-butylamino)propoxy]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-2-yl]phenol 1-[(4S)-3,4-dihydro-2H-chromen-4-yl]pyrrolidine (2R)-3-[[4-(1-ethenyl-5-methyltriazol-4-yl)-6-methoxyquinoline-7-carbonyl]amino]-N,2-dimethylpropanamide 5-bromo-2-(chloromethyl)-6H-benzo[h]chromene 3-(4-chlorophenyl)sulfonylpropyl-diphenoxyphosphinic acid 4-(3,5-dimethoxyphenyl)butylphosphane 4-[1,3-difluoro-6-(2-fluorooctoxy)naphthalen-2-yl]phenol 1-(2,2-difluoroethyl)-N-[5-methyl-3-[(E)-6-methylhept-3-en-4-yl]pyridin-2-yl]-7H-pyrazolo[3,4-c]pyridazine-4-carboxamide 2-[4,6-bis(ethenyl)triazin-5-ium-1-yl]-N-tert-butylacetamide N-[4-(2-hydroxyethylamino)phenyl]-3,5-dimethylbenzohydrazide;hydrochloride 1-[4,5-di(cyclopropyl)pyridin-3-yl]-N'-methoxyethane-1,2-diimine 3-methoxy-4,5-bis(phenylsulfanyl)benzenecarboximidamide N-[2,4-difluoro-3-[5-(2-methoxypyrimidin-5-yl)imidazo[1,2-a]pyrimidin-6-yl]phenyl]butanamide 3-[3,4,5-trimethoxy-N-(2-oxopropyl)anilino]butanoic acid 6-methyl-4,9-diphenyltetracyclo[6.6.2.02,7.011,15]hexadeca-1(14),2,4,6,10,12,15-heptaen-8-one (4-aminophenyl)-(3-iminobutyl)azanium (4aS,12bS)-9-(benzenesulfonylmethyl)-8-phenyl-2,3,4,4a,5,6,10b-octahydropyrano[3,2-c]quinoline 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]-5-hexoxypyridine N-methyl-2-[1-(pyridine-4-carbonyl)piperidin-3-yl]-N-(2,2,2-trifluoroethyl)acetamide 4-azido-2-(3-cyclopropylphenoxy)pyrimidine 5-[(4-chlorophenyl)methylamino]-2,3-dihydroinden-1-one;hydrochloride 4-[3-(difluoromethyl)phenyl]iminobutanoic acid 4-[(1R)-2-(cyclohexylamino)-1,2-dihydroxyethyl]benzoic acid 1-methyl-2,3-dihydroanthracene-9,10-dione 5-(4-chlorophenyl)-N-methyl-3,6-dihydro-1H-pyrrolo[2,3-c]pyrrole-2-carboxamide;methane 2-ethyl-4-[(5-methoxy-3,4-dihydroisoquinoline-1-carbonyl)amino]thiophene-3-carboxylic acid 2-[N-(4-bromobutan-2-yl)-2,6-dichloro-4-nitroanilino]ethanol (2S)-1-[1-tert-butyl-4-hydroxy-6-oxo-5-(2-phenylethynyl)pyrimidin-2-yl]pyrrolidine-2-carboxylic acid 2-[5-(4,4-dimethylpiperazine-1-carbonyl)pyridin-3-yl]acetic acid (E)-3,7-dihydroxy-1-[3-methyl-2-(4-phenylphenyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-yl]hept-2-en-4-one 2-[(3,4-dimethoxyphenyl)methyl]cyclohexane-1,5-dione 2,4-dibromo-6-[3-[(4R)-6-fluoro-7-hydroxy-1H-1,3-diazonin-4-yl]phenyl]benzonitrile 7,8-difluoro-1H-[1]benzothiolo[3,2-b]pyridine 2,4-dimethyl-1-(2-phenylpentanoyl)pyrrolidine-3-carboxamide (2S)-3-[2-(trifluoromethyl)phenyl]cyclopropane-1,2-diamine 2-methyl-4-(3-naphthalen-1-ylpropoxy)pyridine [4-(5-amino-2H-triazolo[4,5-b]pyridin-7-yl)phenyl]-piperidin-1-ylmethanone 6-methylsulfanyl-1',3,7-triphenylspiro[5H-pyrrolo[2,3-d]pyrimidine-4,1'-cyclopentane]-2-one (3S)-4-azido-1'-(2,6-dichlorophenyl)spiro[1H-indole-3,3'-pyrrolidine]-2-one 2,6-difluoro-N-[(3S)-3-hydroxybutyl]benzamide;1-fluoro-4-(1H-inden-5-yl)benzene 2-[(4-tert-butylphenyl)methoxy]benzenethiol 5-methyl-2,3-diphenyl-3H-1,4-benzodiazepine 3-(2,4-dichlorophenyl)sulfonyl-N-methyl-5-piperazin-1-ylpyrrolo[2,3-b]pyrazin-6-amine (2R)-2-benzyl-N,N-diethylpyrrolidine-1-sulfonamide 3-benzyl-7-(cyclohexanecarbonyl)-2-methylsulfanyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-one N-[3-[3-(diethylamino)propoxy]-4-methoxyphenyl]propanamide 5-(2,3-dimethoxyphenyl)-7-[1-(4-hydroxybutyl)piperidin-4-yl]pyrrolo[2,1-f][1,2,4]triazin-4-amine 1-butyl-3-[(4-fluorophenyl)methoxy]benzene 6-bromo-3-chloro-1,8a-dihydroimidazo[1,2-a]pyridine N-(2-benzamidoethyl)-1-[6-[(3,5-dichlorophenyl)methylamino]pyrimidine-4-carbonyl]piperidine-4-carboxamide (2R,3S)-N-[(2,4-difluorophenyl)methyl]-2-(1-methylpyrazol-4-yl)oxane-3-carboxamide 3-[5-(4-chlorophenyl)furan-2-yl]butanal 6-tert-butyl-3-iodo-9,9-dimethylfluoren-4-amine N-[4-[2,5-dimethyl-3-(trifluoromethoxy)phenyl]-1H-pyrrol-3-yl]methanimine 2-(3,4-dichlorophenyl)-N-[(5S,7R)-8-fluoro-5-methyl-6-oxo-1,2,4,5-tetrahydropyrano[3,4-c]isoquinolin-3-yl]acetamide N-methyl-1-[4-(2-nitrosoethoxy)phenyl]propan-2-amine 2-[(2Z,5S)-2-[(Z)-1-(4-methoxyphenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 6-bromo-2-[1-(difluoromethyl)imidazol-4-yl]thieno[3,2-b]pyridine;methanol 4-[[2,3-difluoro-5-(2,2,2-trifluoroethoxy)phenyl]methylamino]cyclohexan-1-one 2-(4-cyano-N-[4-[2-fluoro-4-[(E)-prop-1-enyl]phenyl]-3-methoxybenzoyl)anilino)acetamide;cyclopentane 2-methyl-5-[1-(3-methylphenyl)ethenyl]thiophene N-[(3R,4S)-1-[2-(4-chlorophenyl)ethyl]-4-(3-methoxypyrrolidin-1-yl)piperidin-3-yl]cyclopropanecarboxamide;hydrochloride 2-(4,6-diphenyl-1H-1,3,5-triazin-2-yl)phenol [(3R,4S)-1-ethyl-4-propan-2-ylpyrrolidin-3-yl]-[4-methylsulfonyl-5-(trifluoromethoxy)pyridin-2-yl]methanone 2-ethylimino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one [1-amino-2-[3,5-bis(trifluoromethyl)phenyl]ethylidene]azanium 2-amino-4,6-dichloro-5H-pyrrolo[3,4-d]pyrimidine-7-carboxylic acid 2-benzyl-6-[(3R)-1,3-dimethylpiperidin-4-yl]oxy-1H-isoquinoline N-(2,4-dimethylphenyl)-3-(6-methoxypyridin-3-yl)aniline 4-[2-methoxypropanoyl(pentyl)amino]-N,3-dimethyl-5-[(Z)-(5-methylpyrazolidin-3-ylidene)amino]thiophene-2-carboxamide 4-cyclopropyloxy-3,6-difluoro-N'-hydroxypyridine-2-carboximidamide [3-(1-methylindol-2-yl)pyrrolidin-1-yl]-pyridin-4-ylmethanone 5-chloro-1-[[3,4,5-trifluoro-2-(2-iodophenyl)phenyl]methyl]imidazole 2,7-diaminopyrrolo[3,4-c]pyridine-1,6-disulfonic acid;hydrochloride [4-(2,3-dihydroxypropoxy)phenyl]-methylazanium 2-methylsulfanyl-5,6-dihydropyrrolo[3,4-d]pyrimidine-7-carboxylic acid N'-azido-1-(5,6-diethylthieno[2,3-d]pyrimidin-4-yl)butane-1,4-diamine 5-(4,7-difluoro-2-methylbenzimidazol-1-yl)pyridine-2-carboxylic acid [(3aR,6aS)-5-(5-bromothiophene-2-carbonyl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]-(cyclopropylmethyl)methanone;2,2,2-trifluoroacetic acid 2-[(1R)-3-methylcyclohexyl]pyridine;yttrium 1-[1-(4,4-dimethylpentoxy)butan-2-yl]-4-(trifluoromethyl)benzene 2-[1-(3,5-dichlorophenyl)sulfonylpiperidine-4-carbonyl]oxyethylazanide 5-N-[3-amino-1-(2,6-dimethylphenyl)-4H-pyridazin-4-yl]isoquinoline-1,5-diamine 1-azidooxy-4-(2,3-diphenylphenoxy)naphthalene 3-[2-(2-ethoxyphenoxy)butanoylamino]propylazanium 2-[[8-(3,4-dihydroxyphenyl)quinoline-6-carbonyl]amino]benzoic acid 1-[(2S)-4,5-diamino-3-[4-[3-(trifluoromethoxy)phenyl]piperazine-1-carbonyl]piperidin-2-yl]ethanone 6-fluoro-1-phenyl-7H-pyrazolo[3,4-d]pyrimidine 2-[[4-[6-[(3R)-3-(2,5-dimethylpyrazol-3-yl)-1,2-oxazolidin-2-yl]pyridin-3-yl]piperidin-1-yl]oxymethyl]pyrazine N-(5,6-diphenylpyridazin-3-yl)-5-methylpyridine-2-carboxamide (1R)-N,1-diphenyl-2-[3-[3-(trifluoromethyl)phenyl]imidazo[4,5-b]pyridin-2-ylidene]ethanamine 4-azido-5-bromo-2,3-dimethoxypyridine 6-chloro-4-[3-(2,5-difluorophenyl)phenyl]-2-sulfanylidene-1H-pyrimidine-5-carbonitrile N-[2,4-dimethyl-5-(1-methylindazol-7-yl)pyrazol-3-yl]hydroxylamine 4-(1-cyclopropylethenylamino)naphthalene-1,5-disulfonic acid (3-bromophenyl)methyl-[3-methoxy-4-[4-(5,6,7,8-tetrahydronaphthalene-2-carbonylamino)butanoyl]oxybutyl]oxidanium 2-(2,3-dihydro-1H-inden-5-ylmethoxy)-4-ethoxypyrimidine 3-(4-benzylpiperazin-1-yl)-6-[2-(5-fluoropyridin-2-yl)pyrrolidine-1-carbonyl]-7H-pyrazolo[1,5-a]pyrimidin-5-one 1-(5-bromo-2,3-dihydroindol-1-yl)ethanone (3-azidophenyl)-[4-[2-fluoro-5-(2,2,2-trifluoroethoxymethyl)benzoyl]piperazin-1-yl]methanone 5-methyl-8-(2-methylphenyl)-7,9-dihydrobenzo[c]fluorene (2R,3S)-N,2-dimethyloxane-3-carboxamide;7H-pyrrolo[2,3-d]pyrimidin-4-amine 1-(2-hydroxyethyl)-N,2-dimethylpiperidine-3-carboxamide;N-[5-[3-(6-methoxypyridin-3-yl)prop-1-ynyl]pyridin-3-yl]formamide 1-(oxan-2-yl)indazole-6,7-diol [2-(2,6-diethylphenyl)-4-fluorophenyl]phosphane 1-[(2R)-2-amino-4,4-difluoropyrrolidin-1-yl]-3-[5-methoxy-7-(trifluoromethyl)pyrazolo[1,5-a]pyridin-2-yl]propan-1-one N'-[(3S)-1,2-dimethylpyrrolidine-3-carboximidoyl]-4-fluorobenzenecarboximidamide (2S)-2-[3,5-difluoro-4-(oxan-2-yloxy)phenyl]morpholine 5-[1-(3,4-dimethylphenoxy)propan-2-yl]-2-iminopyrrolidin-3-one 1-(dimethylamino)-3,4-dihydronaphthalene-2-carboxylate 5-benzyl-3,6-dichloro-1,2-dihydropyrazine 2-chloro-1-(3,4-dihydro-2H-pyridin-1-yl)ethanone;7-chloro-6-fluoro-1-oxo-3,4-dihydroisoquinoline-2-carboxylic acid 3-(2,4-dihydroxy-5-propanoylphenyl)-N-ethyl-N-(4-methoxy-6-methylpyrimidin-2-yl)-1H-pyrazole-5-carboxamide 4-amino-5-fluoro-3,6-dimethylbenzene-1,2-disulfonic acid 2-[6-chloro-5-(4,5-dihydrocyclopenta[d]imidazol-1-yl)pyridin-3-yl]acetamide 1-(1,1-dioxothiazinan-2-yl)-N-[6-[4-fluoro-3-(trifluoromethoxy)phenyl]pyridazin-3-yl]cyclopropane-1-carboxamide 4-[[5-methoxy-2-(4-methoxyphenyl)-1,3-benzoxazol-6-yl]sulfonyl-(thiophen-2-ylmethyl)amino]-N-(2-methylsulfonylethylidene)butanamide (2Z)-3-ethyl-2,5,8-trimethyl-6,7-dihydro-5H-naphthalene 1-(4,5-dibromo-2-hydroxyphenyl)cyclopropane-1-carboxamide 1-benzyl-3-[(Z)-(4,6-dioxocyclohexa-2,5-dien-1-ylidene)methyl]thiourea 2-[[[(3S,4R)-1-methyl-4-phenylpyrrolidine-3-carbonyl]amino]carbamoyl]benzoic acid (3R,4S)-1-benzyl-4-[(5Z,7E,9Z)-2,3-dimethylideneundeca-5,7,9-trienoyl]piperidine-3-carboxylic acid (2-methylphenyl)-(4-propan-2-ylphenoxy)borinic acid 3-(4-chlorophenyl)sulfanyl-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]propanamide 6-[6-(2,5-dichlorophenyl)pyridin-3-yl]oxy-4H-1,3,5-triazin-2-amine N'-(4-chlorophenyl)-2-methyliminobutanediamide 1-cyclopropyl-7-[6-(4,4-difluoropiperidine-1-carbonyl)pyridin-3-yl]-8,9-dimethoxy-5-oxo-2H-pyrazolo[4,3-c]quinoline-3-carboxamide 6-(2,5-dimethoxyphenyl)-3-methyl-1-propan-2-ylideneindol-1-ium 2-(4-anilinophenyl)acetamide 4-chloro-N-[(3Z)-2,2-dimethylpenta-1,3-dien-3-yl]-5-ethyl-6-phenylpyridazine-3-carboxamide [1-[1,3-benzodioxol-5-ylmethyl(ethyl)amino]-2-hydroxypropan-2-yl]carbamic acid 3-(1,5-dimethylpyrazol-4-yl)-N-[2-(4-methylpiperazin-1-yl)ethyl]benzenesulfonamide;hydrochloride 4-[(2S)-1-(dimethylamino)pentan-2-yl]-N-[1-[5-[[4-ethyl-3-(trifluoromethyl)phenyl]carbamoylamino]pyrazin-2-yl]piperidin-4-yl]piperazine-1-carboxamide 4-[2,6-difluoro-3-(propoxymethyl)phenyl]-2,2-difluoro-5H-1,3-oxazole 4-[2-(4,6-dimethylpyrimidin-5-yl)ethyl]-3-[(1R)-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]piperazin-2-one 5-bromo-2,6-dichloro-3-(3,4,5-trimethylphenyl)pyrimidin-4-one (4Z)-4-[[5-(2,3-dihydroindole-1-carbonyl)furan-2-yl]methylidene]-1-phenylpyrrolidine-2,5-dione 3-[4-(5,6-dimethylpyrazin-2-yl)phenyl]propanoic acid;hydrochloride [4-(5,5-dimethylhexanoyl)piperazin-1-yl]-naphthalen-2-ylmethanone 4-amino-6-[[(2S)-3,5-dihydroxyoxan-2-yl]methyl]-1H-1,3,5-triazin-2-one 4-[4-[(2R)-2-azidopropyl]piperazin-1-yl]sulfonylphenol 3-azido-1-[(2,5-difluorophenyl)methyl]pyrrolidine 5-benzylsulfanyl-N'-hydroxypyrazine-2-carboximidamide 2-(3,4-dimethoxyphenyl)acetic acid;N,2-dimethylquinazolin-5-amine (3S)-1-[(5-bromo-2-ethylsulfanylimidazo[4,5-b]pyridin-3-yl)methyl]pyrrolidine-3-carbonitrile 3-butyl-5,7,8-trifluoro-2-(4-fluorophenyl)naphthalene 2-cyclopentyl-4-methoxybenzoic acid;5,6,7,8-tetrahydroquinoline (3-azido-5,6,7,8-tetrahydronaphthalen-2-yl)methanamine 1-(5-chlorothiophen-2-yl)sulfonylpiperidine (1Z)-2,4-dimethylpenta-1,3-diene;N'-[[2-ethoxy-5-[4-(N'-hydroxycarbamimidoyl)piperazin-1-yl]phenyl]methyl]-2-oxopropanimidamide N-[3-(methoxymethyl)morpholin-4-yl]sulfonyl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-3-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-2-chloroacetamide;3-[1-(4-chlorophenyl)-4-methoxypyrazol-3-yl]-7-hydroxy-6H-pyrrolo[3,4-b]pyridin-5-one 4-(2,6-dimethoxyphenyl)-3-ethyliminobutanenitrile 3-chloro-5-[6-(2,7-diazaspiro[4.4]nonan-2-yl)pyridazin-3-yl]oxybenzonitrile ethane;methane;(3E,5Z)-N-[(Z)-2-[6-(1-methylpyrazol-4-yl)-3H-imidazo[4,5-c]pyridin-2-yl]but-2-enylidene]hepta-1,3,5-triene-3-sulfonamide 2-(2-aminoethylamino)-6,7,8,9-tetrahydrofuro[3,2-g]chromene-5,11-dione 3-methyliodanuidyl-2-[4-(1,4-oxazepane-6-carbonylamino)phenyl]propanoic acid 4-(2-bromo-N-(5,8-dichloroquinoxalin-6-yl)anilino)butan-1-ol 5-chloro-6-fluoro-3,10-dimethylanthracene-9,10-dione (7S)-8-tert-butyl-N-[(1R,2S)-2-methoxycyclopentyl]-11-oxo-6,7-dihydropyrido[1,2-d][1,4]benzoxazepine-10-carboxamide 1-(9H-fluoren-2-yl)-4,5,6,7-tetrahydroindazole 3-[5-amino-6-(6,7-dihydro-1H-indazol-4-yl)pyrazin-2-yl]cyclobutan-1-ol 1-[4-[(2R)-2,3-dihydroxypropoxy]-3-fluorophenyl]ethanone 6-[5-(2,3-dihydro-1H-inden-4-yl)-1,3,4-thiadiazol-2-yl]-7-ethyl-8a-methyl-4a,9,10,10a-tetrahydrobenzo[c]chromene 4-[1,3-benzothiazol-2-yl(3,3-dimethoxypropyl)amino]butan-1-ol N-[[(3R,4S)-1-(2-hydroxyethyl)-4-(5-methoxypyridin-2-yl)pyrrolidin-3-yl]methyl]oxane-4-carboxamide;dihydrochloride (6R,8S)-8-(4-bromophenyl)-6-[3-chloro-5-fluoro-2-[hydroxy(methoxy)phosphoryl]oxyphenyl]-2,6,7,9-tetrahydro-1H-pyrazolo[3,4-b]quinolin-5-one 1-(4,5-dihydrothiophen-2-yl)benzimidazole N-[4-[2-(6,7-dimethoxyquinazolin-4-yl)ethynyl]phenyl]propanamide (3S,4R)-1-[2-chloro-4-(trifluoromethyl)phenyl]sulfonyl-4-(triazolo[1,5-a]pyridin-7-yloxy)pyrrolidine-3-carboxylic acid 2-[2,4-dichloro-5-(hydroxymethyl)phenyl]ethanol 4-[1,2-diphenylethenyl(pyridine-2-carbonyl)amino]butanoic acid 4-[(2-chloroacetyl)-(2,2-diethoxyethyl)amino]benzenesulfonic acid 2-(1H-indol-3-ylmethylideneamino)phenol 1-(4-chlorophenyl)-3-[2,6-dimethyl-5-(2-propan-2-ylbenzoyl)pyrazin-4-ium-3-carbonyl]indole-6-carboxylic acid 2-[4-(1H-indol-3-yl)piperidin-1-yl]-N-methylethanamine 4-[(4,6-dimethoxypyrimidin-2-yl)sulfamoyl]piperidine-1-carboxylic acid N-methyl-1-[2-(3,4,5-trimethoxyphenyl)imidazol-1-yl]butan-1-imine [4-(1H-indole-2-carbonylamino)benzoyl]-oxoazanium 2-chloro-4-(4-propylphenyl)benzenethiol 4-[2-(3,5-dichlorophenyl)-1-[(2Z,4E,6Z)-5-ethyl-3-methylideneocta-2,4,7-trienoxy]propan-2-yl]benzenesulfonic acid 3-[5-[(E)-2-[4-[2-fluoroethyl(methyl)amino]phenyl]ethenyl]-1H-pyrazol-3-yl]benzenesulfonamide 2-(3-methylbut-1-enoxycarbonyl)benzoate 4-[6-[2-(5-fluoropyridin-3-yl)ethynyl]pyridazin-1-ium-3-yl]thieno[3,2-d]pyrimidine 2-amino-4-[[3,5-difluoro-2-(trifluoromethoxy)phenyl]carbamoyl-propylamino]butanoic acid N-[(2S)-3-hydroxy-1-oxo-1-(1,2,4-triazol-1-ylamino)propan-2-yl]thiophene-2-carboxamide 2-[(3S)-4-azido-3-benzylpiperazin-1-yl]ethanol N-cyclopropyl-7,8-dimethoxy-2-(3-methylsulfanylphenyl)quinoline-4-carboxamide ethane;(3Z,5E)-hepta-1,3,5-triene;(2R)-4-hydroxy-6-[4-hydroxy-3-(hydroxymethyl)phenyl]-N,2-dimethylhexanamide N-[[3-[2-(dimethylamino)ethoxy]-5-(trifluoromethylsulfonylamino)phenyl]methyl]-2-oxo-1H-pyridine-4-carboxamide N-[3-fluoro-2,6-di(propan-2-yl)phenyl]-1H-pyrrole-3-carboxamide 4-chloro-N-[(3S)-1-ethylpiperidin-3-yl]quinoline-2-carboxamide 3-(4,7-dimethyl-1H-indole-2-carbonyl)-4H-1,2,4-oxadiazol-5-one N-[2-(dimethylamino)ethyl]-2-nitropyridine-3-carboxamide 2-amino-9-(oxan-4-yl)purine-8-carboxamide 6-[(2R,4S)-2-methyloxan-4-yl]-1-phenylpyrazolo[3,4-d]pyrimidine (3S,5R)-2-[6-chloro-8-fluoro-7-[(5-methyl-1H-indazol-4-yl)oxy]quinazolin-4-yl]-5-(dimethylamino)piperidine-1-carboxylic acid 4-fluoro-N-[3-(2-methoxyethylamino)pentan-2-yl]benzamide 4-(5-fluoropyridin-3-yl)-N,2-dimethylaniline;formic acid 6-[[1-(dimethylamino)cyclopropyl]amino]-2,3-dihydronaphthalene-2-carboxamide N-[(1R)-1-cyclohexylethyl]-2-phenyl-5,6-dihydro-4H-imidazo[1,5-a]imidazole-7-carboxamide 2-[(1R,3S)-3-ethylcyclopentyl]oxy-5-nitropyridine N-[1-(2,4-dichlorophenyl)ethyl]-6-methylidene-5H-benzo[b][1,4]benzothiazepine-3-carboxamide N-[4-hydroxy-1-(3-phenylpropanoyl)piperidin-4-yl]butanamide 2-[4-(2,6-dimethoxyphenyl)piperazine-1-carbonyl]-5H-thieno[3,4-b]pyrazin-6-one 6-chloro-3-(4-hydroxy-3,5-dimethylphenyl)pyrazolo[1,5-a]pyrimidine-2-carboxylic acid 2-[3-(4-methylphenyl)pyrrolidin-1-yl]propanamide 4-[(E)-2-[4-amino-5-methoxy-2-[(E)-(pyridin-2-ylhydrazinylidene)methyl]phenyl]ethenyl]phenol 4-(4-fluorophenyl)-N-[1-(2,2,3,3,3-pentafluoropropanoyl)piperidin-4-yl]butanamide 2-[4,6-dichloro-5-(3-cyclobutylbenzenecarboximidoyl)pyrimidin-1-ium-2-yl]sulfanylethanamine 2-ethenylimino-5,6-dimethoxy-1H-pyridine-3-carboxylic acid;propane 2-(benzenesulfonamido)-N-[4-[4-[3-[acetyl(oxan-4-ylmethyl)amino]propoxy]phenyl]pyridin-2-yl]acetamide 2-[2-(azetidin-1-yl)ethyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide 6-(1-cyanopropyl)-N-[4-methoxy-3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]-7-propan-2-ylidene-5,10b-dihydro-4aH-benzo[g]quinoline-9-carboxamide N-(2,4-dichloropyrimidin-5-yl)-N-naphthalen-1-ylethenesulfonamide 1-[2-methyl-5-(oxolan-3-yl)pyrazol-3-yl]azepane N-[5-[3-(1H-indol-2-yl)-2,7,8-trimethylimidazo[4,5-b]quinoxalin-5-yl]pentyl]formamide 2-(5-bromothiophen-2-yl)-N-[(3,4-dihydroxyphenyl)methylideneamino]propanamide ethane;1-(7-methoxynaphthalene-2-carbonyl)piperidin-4-one 1-[1-(2,4-difluorophenyl)cyclopentyl]-N-[5-methoxy-2-[6-(trifluoromethyl)pyridazin-3-yl]pyrazole-3-carbonyl]methanesulfonamide 4-[3-(methoxymethyl)phenyl]benzohydrazide 1-[4-(difluoromethoxy)phenyl]ethanol;methanamine 3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethylpyrido[3,4-b]pyrazin-8-one 3-N,2-dimethyl-4-oxo-2H-1-benzofuran-5-carboxamide 5-[(2Z)-2-[4-(3,4-dichlorophenyl)butylidene]hydrazinyl]-N-(oxan-4-ylmethyl)-6-oxohexanamide 5-tert-butyl-N-[2,6-dimethyl-4-(1,3-oxazol-2-yl)phenyl]thiophene-2-carboxamide 7-azidooxy-2,3,4a,5,6,7,8,9,10,11,11a-decahydrocyclopenta[b]fluorene (1S)-2-[3-fluoro-N-methyl-4-(piperidine-4-carbonylamino)anilino]cyclohexane-1-carboxylic acid (3S)-1-[4-methyl-6-[(5-methyloxolan-2-yl)methoxy]pyrimidin-2-yl]piperidine-3,4-diamine [4-(2,5-dioxopyrrolidin-1-yl)oxyphenyl]-phenylmethanone;3-[6-fluoro-1-(pyridin-4-ylmethyl)indol-3-yl]-N-hydroxypropanamide [(2-aminopyridine-3-carbonyl)amino]carbamodithioic acid 2-cyclobutyl-N-(3,4-dihydro-2H-chromen-8-ylmethoxy)-1,3-thiazole-5-carboxamide 2-(dimethylamino)ethyl-[1-(2,5-dimethylphenyl)cyclopentanecarbonyl]-methylideneazanium 4-(4-tert-butylphenyl)sulfanylpiperidine N-azido-4-(4-bromophenyl)-N,3-dimethylbutanamide 4-[3-(2-chloroethyl)-5-oxo-1,2,4-oxadiazol-4-yl]benzonitrile 2-[[6-(3,4-dichlorophenyl)-5-methylpyridine-2-carbonyl]amino]propanoic acid 3-azido-4-(1,2,5-oxadiazol-3-yl)butan-1-ol 1-[4-[2-chloro-5-(trifluoromethyl)pyridin-3-yl]cyclohexen-1-yl]-N-ethanimidoylmethanesulfonamide N-[(2S,3R)-5-[(4-chlorophenyl)methyl]-1-formyl-2-hydroxyindol-3-yl]iminopyridine-3-carboxamide 2-amino-N-[4-methyl-3-(sulfanylcarbamoyl)phenyl]benzamide 5-[1-(4-fluorophenyl)cyclopropyl]furan-2-carboxamide 1-ethyl-N-[(4R,5S)-3-methoxy-5-(2-oxopropylcarbamoylamino)cycloheptyl]pyrrole-3-carboxamide 3-[1-azido-2-(2,6-difluorophenyl)ethyl]sulfonylaniline 2-[5-(4,4,5,5-tetramethyloxaborolan-2-yl)indol-1-yl]ethanamine 4-[1-(oxan-2-yloxy)butyl]benzoate 3-(4-chlorophenyl)-7,8-dimethoxy-2H-thiochromene 3-[2,5-difluoro-4-[3-(1H-pyrazol-5-yl)cyclobutyl]oxyphenyl]-5-propan-2-yl-1,2,4-oxadiazole N-[(E)-1-[4-(dipropylamino)phenyl]ethylideneamino]-6-methylcyclohexa-2,4-diene-1-sulfonamide (3R)-3-[2-chloro-5-[4-[(1R,2S)-2-hydroxycyclohexyl]phenyl]pyridin-3-yl]cyclopentan-1-one 2-[1-(6-aminopyridine-3-carbonyl)piperidin-4-yl]-5,6,7,8-tetrahydrocinnolin-3-one 3-(N-[4-(N,2-dimethylanilino)phenyl]anilino)propanal 3-(2,6-dichlorophenyl)-7-[4-(2,5-dimethylpyrazole-3-carbonyl)piperazin-1-yl]sulfanyl-8H-[1,2,4]triazolo[4,3-a]pyrimidin-5-one 6-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-2H-pyrrolo[1,2-a]pyrazin-1-one 2-[(3,4-dichlorophenyl)sulfanylamino]-5-hydroxy-1,7a-dihydroindole-6-carbonitrile N-[(Z)-(5-bromo-2-hydroxyphenyl)methylideneamino]-2-(4-chlorophenyl)acetamide 2-(6-chloroindol-1-yl)-N-[3-(pyridin-4-ylmethoxy)phenyl]propanamide 2-amino-4-(2-methoxyphenyl)-1-(2-methylsulfonylethyl)piperazine-2-carboxylic acid 7-methoxy-6,8-dihydro-5H-[1]benzofuro[2,3-d]pyrimidine 2-[4-amino-6-chloro-5-(4-fluorophenyl)pyrimidin-1-ium-2-yl]oxyethanol;chloride 1-(2,4,5-trifluorophenyl)sulfanyl-3H-indol-2-one [4-(2,5-dihydrotetrazol-1-yl)phenyl]methanamine;hydrochloride 2-[3,5-bis(trifluoromethyl)phenyl]sulfanylpyrimidine N-[(3S,4R)-1-cyclopentyl-3-(oxetan-3-ylmethylcarbamoyl)piperidin-4-yl]-5-(2,6-difluorophenyl)-1,2-oxazole-3-carboxamide 4-ethoxy-1,5-dimethyl-2-[3-(trifluoromethyl)phenyl]imidazole 2-chloro-1-(4,4-difluoropiperidin-1-yl)-6-methoxyisoquinoline (2R)-N-[4-[5-chloro-3-fluoro-6-[1-methyl-3-(trideuteriomethoxy)pyrazol-4-yl]pyridin-2-yl]phenyl]pyrrolidine-2-carboxamide 3-amino-1-(4-chlorophenyl)pyrrolidin-2-one;ethane 6-(2,5-difluorophenyl)-1H-pyrimidine-2,4-dione 4-azidooxy-N,N-dimethylbenzenesulfonamide 2-[4-(1H-benzimidazol-2-yl)phenoxy]hexanoic acid 4-(2,3,6,7,8,9,10-hexahydro-1H-[1]benzoxepino[2,3-b]pyridin-8-yl)-N-methylsulfonylbutanamide 1-[4-(5-nitropyridine-2-carbonyl)piperazin-1-yl]ethanone 2-(4-ethenylcyclohexa-1,3-dien-1-yl)oxy-N-(5-fluoropyridin-2-yl)benzamide 1-(2,3,4a,5,6,7,8,9,9a-octahydrobenzo[d]azepin-1-yl)-3-methyl-2-[1-[5-methyl-2-(trifluoromethyl)phenyl]ethoxymethyl]butan-1-one (3S,4R)-1-benzyl-3-(3-phenylpropanoylamino)piperidine-4-carboxylic acid 5-azidonaphthalene-1,3-dicarboxylate N'-[(Z)-3,6-dimethyl-2H-indazole-5-carbonyl]-N'-methyl-1-azabicyclo[4.1.0]heptane-3-carbohydrazide 4-[(Z)-[(2,6-dichlorophenyl)methylhydrazinylidene]methyl]-3-nitrobenzene-1,2-diol 2-chloro-5-fluoro-4-[(3S)-1,3,4-trimethyl-3H-pyrrol-2-yl]pyrimidine 2-[5,6-diphenyl-4-(1H-pyrrol-2-yl)thieno[3,2-d]pyrimidin-7-ylidene]propanedioic acid 1-azido-N-(3,5-dichloropyridin-4-yl)piperazine-2-carboxamide (1S)-2,3-dihydro-1H-indene;(Z)-2-phenyl-4-sulfanylpent-2-enal 1-azidooxy-3,4,6,7-tetrachloroquinolin-2-one 3-(2,4-dichlorophenyl)-N'-hydroxypyridazine-4-carboximidamide 5-(4-butylphenyl)-1,3-difluoronaphthalene 2-bromo-5-[1,4-bis(trifluoromethyl)-5,6-dihydropyrazolo[3,4-h]quinazolin-8-yl]phenol ethane;3-[2-methyl-6-(trifluoromethyl)phenyl]pyridine 2-[(3R)-1-azabicyclo[2.2.0]hexan-3-yl]-N-methylaniline 1,2-bis(4-methylphenyl)piperazine 5-[(5E)-4,4-dimethylhepta-1,5-dien-2-yl]-3-phenyl-1,3-oxazolidine 2-(N-(4-nitrophenyl)anilino)acetonitrile N-[4-(hydroxymethyl)oxan-4-yl]benzamide 2-[(4R)-1-acetyl-6,8-dimethoxy-4H-[1,2]oxazolo[5,4-c]quinolin-4-yl]-N-benzylacetamide 3-[7-(2,3-dimethylbutan-2-yl)-1H-indole-3-carbonyl]heptanenitrile 6-bromo-2-(5,7-difluoroquinolin-3-yl)-4H-1,8-naphthyridin-3-one 6-[4-(4,5-dimethyl-1H-imidazole-2-carbonyl)piperazin-1-yl]pyridine-3-carboxamide 1-azido-2,3-dimethyl-9H-fluorene 4-[2,3-bis(ethenyl)phenyl]benzonitrile;ethane;1-methyl-4-propan-2-ylbenzene 5-[5-cyclopropyl-3-(1,1,2,2,2-pentafluoroethyl)pyrazol-1-yl]sulfanyl-N'-hydroxypyridine-2-carboximidamide 4-(2,3-dihydro-1H-isoindole-5-carbonyl)-N'-hydroxypyridine-2-carboximidamide 6-chloro-N-(2-pyrrolidin-1-ylethyl)-8-[4-(trifluoromethoxy)phenyl]quinolin-2-amine (2R,3S)-3-[4-(benzimidazol-1-yl)butanoylamino]-N'-hydroxybutanediamide 1-[3-[4-(8-amino-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)phenyl]pyrrolidin-1-yl]-2,2-dimethoxyethanone 3-[4-(2-cyclopropylethoxy)phenyl]-5-methyl-1,2,4-oxadiazole (2R,3S)-2-N-[1-(3-chloro-4-fluorophenyl)ethenyl]-1,4-dioxane-2,3-diamine N-[(1R)-3-amino-6-(6-chloropyridin-2-yl)iminocyclohexa-2,4-dien-1-ylidene]hydroxylamine 3-[4-(difluoromethoxy)phenyl]-5-[2,6-dimethyl-1-(naphthalene-2-carbonyl)indol-3-yl]pentanoic acid N-(cyclohexylmethoxy)-1,6-dimethylpyrazolo[3,4-d]pyrimidine-7-carboxamide (E)-4-[3,5-dichloro-N-[(2R)-4-[[2-(methanesulfonamido)pyridine-4-carbonyl]amino]-2-propan-2-ylpentyl]anilino]but-1-enylcarbamic acid (2R)-5-[4-(1,1-difluoroethyl)phenyl]-3-methoxy-2-methylpentanamide;ethane 5-(3,4-dichlorophenyl)-2H-triazolo[4,5-b]pyridin-7-one 2-[(3R,4S)-3-cyclopropyl-4-[[4-(2,6-dichloro-3-methoxyphenyl)pyrimidin-2-yl]amino]pyrrolidin-1-yl]acetamide 5-bromo-2-[3-(4,5-difluoro-1H-benzimidazol-2-yl)propoxy]-N'-methylpyridine-3-carbohydrazide;2-prop-1-en-2-ylthiophene 5-tert-butyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid 4-[2-[(5E,7Z)-3-methylnona-5,7-dienoyl]benzimidazol-1-yl]benzoic acid 3-[(4-tert-butylphenoxy)methyl]-1,3-oxazolidine N-[2,6-di(propan-2-yl)phenyl]butanamide;3-methylsulfanylbutane;uranium(2+) N-[2-(azepan-1-yl)phenyl]-N'-methoxypyridine-4-carboximidamide (5Z)-2-[(2,3-dichlorophenyl)methylsulfanyl]-5-[[4-[(2,6-difluorophenyl)methoxy]phenyl]methylidene]-1,3-thiazol-4-one 3-[(3,5-dichloro-2-ethylsulfonylphenyl)methylidene]piperazine-1,4-dicarboxylic acid 1-(5,7-dimethylindazole-1-carbonyl)piperidine-4-carboxylic acid (E)-3-amino-N-[5,6-dimethoxy-2-(4-pyridin-3-ylpiperidine-1-carbonyl)pyrimidin-4-yl]prop-2-enamide 2-(4-azidopyridin-3-yl)sulfanylethanol 6-methyl-4,7-dioxabicyclo[3.2.0]heptane;4,5,9,10-tetrahydropyrene 1-[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,5,6,7-tetrahydroindazol-5-yl]pyrrolidine-2,5-dione 4-[(Z)-2-cyano-3-oxoprop-1-enyl]-N',N'-dimethylbenzohydrazide N-cyclopentyl-4,6-dimethoxyquinoline-3-carboxamide (2Z)-6,8-dichloro-N'-[[2-hydroxyethyl(methyl)amino]methyl]-3-methanimidoylisoquinoline-1,7-dicarboximidamide N-[(1R,2S)-2-(3-chlorophenyl)cyclopropyl]-4-methoxypyrimidine-5-carboxamide N-[4-(3,5-dimethylpiperidine-1-carbonyl)phenyl]-4-phenylpiperidine-1-carboxamide 1-(2,6-dichlorophenyl)-3H-indol-2-one 4-[2-ethoxy-4-(trifluoromethyl)anilino]-N-hydrazinylidene-3,5-dinitrobenzenecarboximidamide 5-(2,4-dimethyl-1H-benzimidazol-5-yl)-N-[4-[1-(difluoromethyl)pyrazol-3-yl]phenyl]-3-methoxypyridine-2-carboxamide 4-[[2,3-dihydroxypropyl(methyl)amino]methyl]-N'-hydroxypyridine-2-carboximidamide [1-[6-chloro-5-(methylsulfonylmethoxy)pyridin-2-yl]benzimidazol-4-yl]methanol 5-[(1,3-dimethylindazol-6-yl)amino]-1H-pyrazole-4-carboxamide 3-[2,4-dimethyl-5-(trifluoromethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile [2-amino-5-(4,4-difluorocyclohexyl)oxyphenyl]methanol ethane;1-[4-(trifluoromethoxy)phenyl]azepane N-(4-methylpyrimidin-5-yl)-2,3,3a,5,6,7,7a-octahydrofuro[3,2-b]pyridine-3-carboxamide;hydrochloride 3-ethoxy-2,6-difluorobenzenesulfonic acid (2S,4R)-N-[(2-amino-1H-imidazol-5-yl)methyl]-4-hydroxypyrrolidine-2-carboxamide;dihydrochloride N-[5-(3,4-dimethoxyphenyl)pyridin-2-yl]-1H-pyrazole-5-carboxamide 4-(3-bromo-1H-pyrrolo[2,3-b]pyridin-5-yl)cyclohexan-1-amine 2-(3,4-dimethoxyphenyl)sulfanylbenzoic acid 4-[3,5-dimethyl-1-(2-methylphenyl)pyrazole-4-carbonyl]piperazine-1-carboxylic acid 2-hydroxy-4,6-diphenylbenzenecarboximidate;1-methyl-3-(2,4,4-trimethylpentan-2-id-2-yl)benzene;oxido-oxovanadium 2-[(4,5-dichlorothiophen-3-yl)sulfonylamino]-N-pyridin-3-ylbenzamide N-[1-cyclopropyl-3-(4-fluorophenyl)pyrazol-4-yl]-7H-purine-6-carboxamide 1,5-dimethyl-3-[(4-pyrazol-1-ylphenyl)methylidene]indol-2-one 2-methyl-7,10-dihydrophenoxazine 6-[(Z)-1-ethoxy-4,4,4-trifluorobut-2-enyl]-N-methyl-5H-cyclopenta[b]pyridine-3-carboxamide N-(3,4-dihydropyridin-5-yl)-N',2-dimethoxybenzenecarboximidamide;ethane 3-methyl-N-[6-(2-nitrophenyl)pyridazin-3-yl]-N-propan-2-ylbut-1-en-2-amine 1-[3-hydroxy-5-[(4-methoxyphenyl)diazenyl]thiophen-2-yl]naphthalene-2,7-disulfonic acid (4-hydroxy-5-nitrofuran-2-yl)-morpholin-4-ylmethanone 2-(3,4-dichlorophenyl)sulfanyl-7-[3-[3-(5-methoxy-1H-indol-3-yl)propyl]piperidine-1-carbonyl]cyclohepta-2,6-diene-1-carboxylic acid 2-(3-chlorophenyl)-2-[1-[4-[5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl(quinolin-8-ylsulfanyl)amino]butyl]piperidin-4-ylidene]acetic acid 5-(3,4-dimethoxyphenyl)-2,4-dimethyl-1H-pyrimidin-6-one 6-(3-acetylphenyl)-8-chloro-2-[4-(trifluoromethoxy)phenyl]-1H-imidazo[1,2-a]pyridin-7-one 4-[(Z)-[2-oxo-3-[3-(trifluoromethoxy)phenyl]-1,5-naphthyridin-1-yl]iminomethyl]benzonitrile 2-(4-methylpiperidin-1-yl)-5-(thiophen-3-ylmethoxymethyl)pyridine 5-[6-[(1S)-1-[4-chloro-2-ethyl-5-methoxy-3-(morpholine-4-carbonyl)phenyl]ethyl]thieno[3,2-d]pyrimidin-4-yl]-5-azaspiro[2.4]heptan-7-one 2-(azidomethyl)-7-[[4-(4-methoxyphenoxy)phenyl]methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine 3-[4-amino-2-(oxan-4-yl)pyrimidine-5-carbonyl]-1H-quinoxalin-2-one 4-[(E)-2-[7-cyclopropyl-8-methoxy-5,6-dihydroquinolin-4-yl]ethenyl]benzaldehyde N-(3,4-dimethylphenyl)-2-[3-ethoxy-4-hydroxy-5-(2H-tetrazol-5-yl)phenyl]acetamide [4-(cyclohexylmethoxy)phenyl]carbamic acid (5Z)-1,3-bis[2,6-dichloro-4-(trifluoromethyl)phenyl]imino-5-[(E)-3-(4-nitrophenoxy)prop-1-enyl]pyrrolidine-2-thione 4-[(5S)-2-[(3,4-dimethoxyphenyl)methyl]-8-(2-hydroxyethyl)-2,8-diazaspiro[4.5]decan-3-yl]phenol 4-[1-(cyclohexanecarbonyl)piperidin-3-yl]-2-methyl-1H-pyrimidin-6-one N-azido-2,3-dihydroindole-1-carboxamide N-cyclohexa-1,5-dien-1-yl-3,6,11-triazatetracyclo[10.7.0.02,6.07,11]nonadeca-1(19),2,4,7(11),8,12,14,16,18-nonaen-16-amine 7-(3,5-difluorophenyl)sulfinyl-2-(2-methyl-1H-indol-4-yl)pyrido[1,2-a]pyrimidin-4-one 1-benzyl-4-methoxypyrrolidine;2,3-diaminoanthracene-9,10-dione 5-methyl-3-[(Z)-[2-(4-phenyl-N-[4-(2,2,2-trifluoroethoxy)phenyl]anilino)acetylidene]amino]thiophene-2-carboxylic acid N-(4-azidopyridin-2-yl)cyclopentanecarboxamide N-butyl-1-phenylethanimine 3-[1-[4-(1,2-dihydroquinolin-6-yl)pyrimidin-2-yl]piperidin-4-yl]-N,N-diethylpropan-1-amine N-(4-hydroxybutyl)-N-[2-[[5-[(dimethylamino)methyl]furan-2-yl]methylamino]ethyl]butanamide 5-[(3Z)-3-ethylidene-2,4-dimethylhexa-1,5-dien-2-yl]-1,2-thiazole 5-(3,4-difluorophenyl)-N-methyl-2-[1-(oxan-3-ylmethyl)piperidin-4-yl]pyridine-3-carboxamide N-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)-3,4-dihydro-1H-isoquinoline-2-carboxamide N'-[(3R,5S)-2-oxo-1-pyridin-4-ylpyrrolidin-3-yl]oxamide N-[2-fluoro-4-methoxy-3-(1,3-oxazol-5-yl)phenyl]propanamide 2,4-bis(5-chloropyridin-3-yl)pentan-1-amine 2,5-dimethyl-1,3-thiazole;3-[4-(8-methoxyquinolin-7-yl)phenyl]propanoic acid 4-(azidomethyl)-2,3-dibromobenzenesulfonic acid 1-(5,6,7,8-tetrahydroquinolin-2-yl)piperazin-2-one 1-azido-6,8,9,10-tetrahydrobenzo[c]chromene N-[(3Z,5E)-hepta-1,3,5-trien-2-yl]-6H-benzo[c]isochromene-8-carboxamide 1-(4-chlorophenyl)-N-[3-[(dimethylamino)methyl]cyclobuta-2,4-dien-1-ylidene]-5-methoxy-2H-quinazolin-4-amine N-[3-[1-[4-(4-chloroanilino)phenyl]-2,3-dihydro-1H-indene-5-carbonyl]oxyphenyl]pyridine-4-carboxamide N-(3,5-ditert-butylphenyl)-2,3-dioxopiperazine-1-carboxamide 7-[(2,6-dichlorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one (2S)-1,2-diphenyl-4-[1-[[4-(trifluoromethyl)phenyl]methoxycarbonylamino]cyclopropanecarbonyl]piperazine-2-carboxylate N-[(4-fluorophenyl)methyl]-3,5-dihydroxybenzamide (4S,5R)-2-[3-chloro-6-[(E)-2-methylbut-1-enoxy]pyridin-2-yl]sulfanyl-4-methyl-5-(2-oxoimidazolidin-1-yl)oxolan-3-one N'-(4,6-dimethylpyrimidin-2-yl)-5-ethoxypyridine-3-carbohydrazide (3-aminopyrrolidin-1-yl)-[2-[4,5-bis(ethenyl)imidazol-1-yl]-6-morpholin-4-ylpyridin-3-yl]methanone 2-[(1R)-4,5-dimethoxycyclohexa-2,4-dien-1-yl]-2-hydroxyacetamide 1-[(2R,3S)-4-[4-(cyclopropylmethoxy)phenyl]-3-hydroxybutan-2-yl]-5-hydroxy-3H-2,1-benzoxaborole [4-amino-2-(3,5-dichloropyridin-2-yl)iminocyclohexa-1,3-dien-1-ylidene]methylideneazanide N-[4-[4-amino-7-methyl-5-(2-methylpyridin-3-yl)pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]prop-2-enamide 4-[2-(3,5-dichlorophenyl)ethynyl]pyridine 4-(4-aminopiperidine-1-carbonyl)-2-(3,5-dimethylpyrazol-1-yl)benzonitrile;hydrochloride 2-(1,3-dioxoisoindol-2-yl)-5-methoxy-N-[4-(1,3-thiazol-2-yl)cyclohexa-1,5-dien-1-yl]pentanamide 4-[1-(2,6-dihydroxy-3-methoxyphenyl)cyclooctyl]benzene-1,3-disulfonic acid 2-amino-N-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)benzamide 1-methylsulfonylpyrazole;platinum(2+);triphenylphosphane N'-[(2R)-5-acetyl-6,15-dibromo-4-oxo-14-oxa-5-azatricyclo[9.3.0.02,7]pentadeca-1(11),2,4,6,12-pentaen-3-yl]-N,N-dimethylmethanimidamide;ethane N-cyclohexyl-3,3-dimethyl-2H-indole-1-carboxamide;ethane 3-ethoxy-1-(4-methylphenyl)sulfinylpyrrolo[2,3-b]pyridine 7-cyclopentyl-2-[(3,5-dimethoxyphenyl)methylsulfanyl]-N-hydroxypyrrolo[2,3-d]pyrimidine-6-carboxamide 2-(5,8,8-trimethyl-6,7-dihydronaphthalen-2-yl)benzaldehyde 3-[4,5-dimethoxy-2-(propylamino)phenyl]-3-(1H-indol-2-yl)propanoic acid 2-(4-azidophenoxy)-N-[3-[4-[5-chloro-6-(difluoromethyl)pyridin-3-yl]piperazin-1-yl]propyl]-4-(trifluoromethoxy)benzamide 2-ethylsulfanyl-1-(4-fluorophenyl)-4-methyl-5,6-dihydrobenzimidazole N-(4,5-dimethyl-2H-pyridin-1-ium-1-ylidene)benzenecarboximidate 6-[(3,4,5-trimethoxyphenyl)methyl]quinoline 4-[6-(2-hydroxyethylamino)pyridin-3-yl]benzaldehyde 6-[(3R)-4-(cyclopropanecarbonyl)morpholin-3-yl]-2,2-diphenylhexanamide 3-[(4-oxo-6-propan-2-ylpyran-3-carbonyl)amino]hexanoic acid 3,5-bis(2-methoxyphenyl)-1H-indole 3-chloro-N-[2,4-difluoro-5-[6-methyl-7-oxo-1-(2-oxo-1H-pyridin-3-yl)quinolin-4-yl]phenyl]benzenesulfonamide (6S,9R)-8-oxo-4-[2-(pyridin-3-ylamino)phenyl]-5-thia-1,7-diazatricyclo[7.4.0.02,6]trideca-2(6),3,10-triene-11-carbonitrile 4-[2-(2,3-dihydroindol-1-yl)pyrimidin-5-yl]-N-phenylsulfanylbenzamide 4-[2,5-difluoro-3-[(6-methylpyridin-3-yl)methoxy]phenyl]-8-[[3-(hydroxymethyl)oxetan-3-yl]amino]quinoline-3-carbonitrile N-[[4-(difluoromethoxy)phenyl]methyl]-7H-purin-2-amine 1-azido-3-[(4-fluorophenyl)methyl]pyrrolidine (3S)-1,4'-dimethylspiro[2H-isoindole-3,5'-imidazolidine]-2'-one 6-(3-hydroxypropyl)-2-[4-methoxy-1-(pyridine-4-carbonyl)piperidin-4-yl]pyridazin-3-one 4-N-[(2E)-3,7-dimethylocta-2,6-dienoxy]-1H-quinazoline-2,4-diamine 1-[2-fluoro-3-(1H-indole-3-carbonyl)phenyl]pentane-1,4-dione 3-(1H-indol-2-yl)quinoxalin-2-amine 5-methyl-7-nitro-N-[[(1S,2R)-2-pyridin-3-ylcyclopropanecarbonyl]amino]pyrazolo[4,3-d]pyrimidine-3-carboxamide N-(4-nitrophenyl)-N-(2,4,6-trichlorophenyl)methanesulfonamide 1-[[4,5-bis(ethenyl)furan-2-carbonyl]amino]-3-(2,6-dimethoxyphenyl)urea N-[4-(ethylamino)phenyl]sulfanyl-1,3-thiazol-2-amine 1-(2,4-dichloro-5-methylphenyl)-N-[(3S)-1,6-dihydroxyhexan-3-yl]cyclopropane-1-carboxamide 1-[2-(5-chloro-1,3-benzoxazol-2-yl)piperidin-1-yl]ethanone 4-fluoro-6-[(2S)-3-hydroxy-1,1,1-triphenylpropan-2-yl]oxypyridine-2-carboxamide N-[(3R,4S)-1-(2-cyano-6-fluorophenyl)sulfonyl-4-methoxypyrrolidin-3-yl]-3,3,5-trimethylhexanamide;hydrochloride 4-[5-(3,5-dibromopyridin-2-yl)oxypentoxy]-4-oxobutanoate 2-N,1-bis(4-fluorophenyl)-5-iodoiminopyrazolidine-3,4-diimine (2S)-2-[(2-chlorophenyl)methyl]-3,4-dihydro-1H-benzo[h]quinoline-8-carboxylic acid 7-azidooxy-N,5-diphenylheptanamide 2-[(5S)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-5-carbonyl]-3H-quinazolin-4-one 4-(3,5-dichlorophenyl)iminopyrrolidine-2-carboxylic acid 2-[(3S)-3-(3,4-dihydro-1H-isoquinoline-2-carbonylmethyl)pyrrolidin-1-yl]benzamide N-methoxy-6,8-dinitroquinoline-3-carboxamide 6-(3,4-dichlorophenyl)-8-methyl-11-methylidenepyrido[2,3-b][1,4]benzothiazepine 1-[2,3-bis(chloromethyl)cyclopropyl]oxy-4-nitrobenzene 2-[4-(1,3,7,10-tetrazatricyclo[6.4.0.02,6]dodeca-2(6),7,9,11-tetraen-12-yl)piperidine-1-carbonyl]-5H-imidazo[1,2-a]quinoxalin-4-one 2-(2,6-dichlorophenyl)sulfonylquinoline 1-(3,5-dimethylphenoxy)pyrrolidine;4-[[4-fluoro-2-(trifluoromethoxy)phenyl]methylamino]butanamide 4-methyl-1,2-bis(5-phenylpyridin-2-yl)pyridin-1-ium;trifluoromethanesulfonate 1-(4-iodo-2-methoxybutan-2-yl)oxy-4-nitrobenzene N-azido-2-(4,6-dimethoxypyrimidin-5-yl)thieno[3,2-b]pyridin-7-amine N-[4-(2,5-difluorophenyl)-2-[(1S)-4-fluorocyclohexa-2,4-dien-1-yl]-3-oxobutan-2-yl]acetamide 2,4-dichloro-N-(4,5-dimethylcyclohexa-1,3-dien-1-yl)-N-propan-2-ylaniline N-(6-oxo-2,3,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridin-1-yl)-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide 2-fluoro-6-methoxy-N-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamide 3-bromo-6-(4,4-difluorocyclohexyl)pyridine 2-[1-(dimethylamino)heptan-3-yl]benzoic acid N-[4-(dimethylamino)phenyl]-2-[(1R,3S)-3-hydroxycyclohexyl]propanamide (3E)-4-amino-3-[[4-methoxy-2,6-dimethyl-N-[(3,4,5-trifluorophenyl)methyl]anilino]methylidene]azete-2-thione N-methyl-4-(5-nitrothiophene-3-carbonyl)morpholine-2-carboxamide 1-[(4S)-3,9-diazatricyclo[6.2.0.02,7]dodeca-2(7),3,5-trien-4-yl]ethanone N-(cyclohexylmethyl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-3-carboxamide 5-(4-methylphenyl)-2,2-diphenoxy-3H-1,3-oxazole 2-[2-(5-fluoropyridin-3-yl)quinolin-8-yl]oxypropanoic acid 4-tert-butyl-5-iodotriazole 1-(3,4-dichlorophenyl)-2,5-dimethylpiperazine N-[2,4-di(propan-2-yl)phenyl]-3-[1-[2-(2-methoxyethylamino)ethylcarbamoylamino]cyclohexyl]naphthalene-2-carboxamide 3-(1,3-benzothiazol-2-ylsulfanyl)-N-[4-[ethyl(propyl)amino]butyl]propanamide 1-methyl-4-[2-(3-methyl-2H-indazol-5-yl)ethynyl]piperidine-4-carbonitrile N-[[3-(5-acetamidoindol-1-yl)phenyl]methyl]benzamide (7R)-7-amino-3-[5-chloro-2-(4,5-dihydropyrimidine-2-carbonyl)phenyl]-1-(2,6-difluorophenyl)-4H-pyrimido[4,5-d]pyrimidin-2-one N-[(4-azidophenyl)methyl]prop-2-ynamide 3-[4,6-dimethyl-1-[(4-methylphenyl)methyl]indol-2-yl]phenol (2S,3S)-2-(9H-fluoren-9-ylmethoxycarbonylamino)-3-hydroxybutanoic acid 3-(3,5-dimethylphenyl)sulfanyl-N'-hydroxypyrazine-2-carboximidamide 4-methyl-2-[(2R)-2-(5-pyridin-3-ylthiophen-2-yl)propoxy]pyrimidine 4-[(2S)-1-(1-hydroxyethylamino)propan-2-yl]phenol 6-ethyl-2,3,4a,5-tetrahydrobenzo[h]chromene 7-(3,5-dimethylphenyl)-2-[(E)-pent-3-enoxy]thieno[3,2-d]pyrimidine N-[3-(cyclopropylmethoxy)-1H-indazol-5-yl]-4,7-dioxo-2,3-dihydro-1H-pyrano[2,3-c]pyridine-6-carboxamide 2-[4-ethoxycarbonyl-N-(3-methylbutyl)anilino]decanoic acid (4-iodophenyl)methylazanide 1-phenylmethoxy-2,4-bis(prop-2-enyl)benzene 1-[(2,4,6-trimethylphenyl)sulfonylamino]thiourea 1-[4-chloro-3-(trifluoromethyl)phenyl]-6,7-dihydroxy-8-methoxyquinazoline-2,4-dione (1S)-N',4-dihydroxy-N-[2-oxo-5-phenyl-3-[[4-(trifluoromethylsulfanyl)phenyl]methoxy]pentanoyl]benzohydrazide 5-[4-[(3S)-3-methylpiperazine-1-carbonyl]phenyl]-11,13-dihydroindolo[2,1-c][1,4]benzodiazepin-6-one 2-[(4-acetamidophenyl)methyl]-7,8-dihydro-3H-[1]benzofuro[3,2-d]pyrimidine-6-carboxylic acid [(3aS,8bS)-1-[(4-fluorophenyl)methyl]-2,3,3a,5,6,7,8b-octahydropyrrolo[3,2-b]azepin-8-ylidene]carbamic acid 3-(4-chlorophenyl)-5,7-dimethoxychromen-2-one N'-methyl-3-[(Z)-3-(propan-2-ylideneamino)prop-1-enyl]pyridine-4-carboximidamide N-[1-(dimethylamino)cyclohexyl]-4-fluoro-2,3-bis(trifluoromethyl)benzenesulfonamide 2-(4-fluorophenyl)-N-[3-(6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-ylamino)propyl]acetamide;dihydrochloride 2-methylsulfanyloxycarbonylnaphthalene-1,4-dicarboxylic acid 5-[2-[4-[[1-(hydroxymethyl)cyclopropanecarbonyl]amino]phenyl]iminoethylideneamino]-1,3-dihydroindol-1-ium-2-one 3-(1H-imidazol-2-yl)-N-[(4S,5R)-4-(hydroxymethyl)piperidine-1-carbothioyl]propanamide (3R)-4-[2-hydroxy-3-(3-methylbutoxy)propyl]-3,5-dihydro-2H-1,4-benzoxazepine-9-carboxamide 2-[(2E)-2-[(Z)-(3,4-dimethoxyphenyl)methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 3-[2,4-dihydroxy-6-(propan-2-ylcarbamoyl)phenyl]-5-(4-methoxynaphthalen-1-yl)-N-(2-piperazin-1-ylethyl)benzamide;ethane 1,2-difluoro-4-[4-[(Z)-2-ethenylpent-3-enoxy]cyclohexa-2,4-dien-1-yl]benzene 3-[1-(1,2-dimethyl-4H-[1,2,4]triazolo[5,1-c][1,4]benzoxazin-7-yl)ethylideneamino]piperidine-2,6-dione [(2R,4S)-1-acetyl-5-hydroxy-2-methoxypiperidin-4-yl]-[3-(4-carbamimidoylanilino)benzoyl]azanium 1-[4-chloro-6-(5-cyclopropyl-3,4-dihydropyrazol-2-yl)pyrimidin-2-yl]piperidine-4-carbonitrile N-[(5R,7S)-3-chloro-1,4-dimethyl-6-oxo-5,7-dihydro-2H-pyrazolo[3,4-b]pyridin-5-yl]-2-methoxybenzamide 4-methoxy-6,7,8,9-tetrahydropyrimido[2,1-c][1,4]benzodiazepine 2-[(3S)-piperidin-3-yl]oxy-1,3-benzothiazole 6-[2-hydroxyethyl(propan-2-yl)amino]-N'-hydroxypyridine-2-carboximidamide 3-(2,4-diethylphenyl)furan 5-bromo-3-methylthieno[2,3-b]pyridine 3-(1H-indol-4-yl)-2,7-naphthyridine 3-[4-(1,3,5-triazin-2-ylamino)naphthalen-1-yl]propan-1-ol N-[(1E)-3-aminobuta-1,3-dienyl]-4-[[4-(3,5-dimethoxyphenyl)-2,6-dioxopiperidin-3-ylidene]methyl]benzamide 2-[(E)-3-(2,6-dimethoxyphenyl)prop-2-enoyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidine-8-carboxamide 3-cyclopropyl-5,6-dimethoxy-2-(4-thiophen-3-ylpiperazin-1-yl)pyridine N-[5-(2,3,5-trifluoroanilino)sulfanylpyridin-2-yl]acetamide ethane;1-(6-methyl-3,4-dihydronaphthalen-2-yl)-N-pentan-3-ylpropan-1-imine [5-fluoro-2-methoxy-4-[1-(trideuteriomethyl)piperidin-3-yl]phenyl]-methylidene-[2-oxo-1-(1,3-thiazol-2-yl)ethyl]azanium 2-[1-azidoethyl(naphthalen-1-ylmethoxycarbonyl)amino]acetic acid N-[5-(2,3-difluorophenyl)sulfanyl-1H-indazol-3-yl]cyclopropanecarboxamide 6-chloro-3,3-difluoro-1H-thieno[2,3-b]quinolin-8-one 3-[(4-azidopyridin-2-yl)amino]-1H-pyridin-2-one 2-[3,5-dichloro-4-[(5-hydroxy-6,7-dimethyl-8,9-dihydropyrimido[4,5-b]azepin-4-yl)amino]phenoxy]acetic acid N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-methoxy-3-(2-morpholin-4-ylethoxy)benzenecarboximidate 5-[2,6-difluoro-4-(3-propylhexoxy)phenyl]-1,3-difluoro-2-isothiocyanatobenzene 4-chloro-1H-imidazo[4,5-c]quinoline;N-[(2S)-2-[4-(3,4,5-trifluorophenyl)piperazin-1-yl]propyl]formamide 3-[2-(3,5-dimethyl-1H-pyrazole-4-carbonyl)benzimidazol-1-yl]pyrrolidin-2-one 1-[(5S,7R)-5-azido-7-methyldecan-2-yl]-4-propoxybenzene N-[(5Z)-5-[(4,4-dimethyl-2-nitrophenyl)hydrazinylidene]cyclohexa-1,3-dien-1-yl]-6-methoxypyridine-3-carboxamide N-[1-(2-chloro-6,7,8,9-tetrahydropyrido[3,4-b]indolizin-5-yl)ethylidene]hydroxylamine N-(2,6-dibromopyridin-4-yl)-N-phenylbenzamide (E)-2-(3,4-difluorophenyl)-N-[1-(furan-2-ylmethoxy)ethenyl]propanamide 1-[4-chloro-2,6-di(propan-2-yl)phenyl]ethylcarbamic acid (E,2S)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N'-[(6-methoxyquinolin-3-yl)methyl]but-3-enediamide 5-[(Z)-[4-fluoro-2-oxo-1-(4-propylphenyl)quinolin-3-ylidene]methyl]-6-hydroxy-1,3-di(propan-2-yl)pyrimidine-2,4-dione 2-[4-[1-(3,5-dichloropyridine-4-carbonyl)piperidin-4-yl]butoxymethyl]pyrimidin-4-amine 4-[2,6-dimethyl-5-(trifluoromethyl)-1H-indol-3-yl]benzonitrile 2-tert-butyl-6-[(3,4-dimethoxyphenyl)sulfonylamino]benzoic acid 2-azido-6,7,8,9,10,11-hexahydropyrido[1,2-a]azocine 5-[2-methyl-4,6-bis(trifluoromethoxy)phenyl]-N-(1-phenylethylideneamino)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 2-[2,3-bis(ethenyl)phenoxy]ethanethiol 1-[3,5-bis(trifluoromethyl)phenyl]-3-[3-chloro-2-(4,5-dihydroazepin-7-ylidenemethyl)indol-6-yl]-5-ethoxycarbonylpyrazole-4-carboxylic acid 2-[[3-(dimethylamino)phenyl]diazenyl]phenol 1-[(4R)-2,4-dimethyl-5-propan-2-ylidenepyrrolidin-3-yl]-6-fluoro-4-morpholin-4-ylbenzimidazole N-methyl-1,3-bis(2-phenylphenyl)imidazol-2-imine;nickel(2+) 3-[2-azido-6-[(3S)-1-benzylpyrrolidin-3-yl]-4,5,7,8-tetrahydrothieno[2,3-d]azepine-4-carbonyl]benzonitrile 4-[2,4,7-tris(sulfanylidene)-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidin-5-yl]benzoic acid 2-[(2E)-2-[(1-ethylpyrazol-4-yl)methylidene]hydrazinyl]-6,7-dihydroquinazolin-8-one 2,4-difluoro-3-(4-methylthiophen-2-yl)-6-phenylbenzamide 4-chloro-N-[2-(2,5-dimethoxyphenyl)ethyl]cyclohexa-1,3-diene-1-sulfonamide N-ethylsulfonyl-4-nitrobenzenesulfonamide [5-(1-azidooxy-4,4,4-trifluorobutyl)pyridin-2-yl]methanamine 1-[(2-chloro-3,6-difluorophenyl)methyl]pyrazole-4-carboxamide (2Z)-3-[1-(cyclopropylmethyl)piperidin-4-yl]oxy-2-(6,7-dihydronaphthalene-2-carboximidoyl)penta-2,4-dienal N-[2,4-difluoro-3-(3-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridine-5-carbonyl)phenyl]propane-1-sulfonamide 4-(2,3-difluoro-4-isothiocyanatophenyl)benzoic acid 3-(3,5-dibromo-4-hydroxyphenyl)-2H-[1]benzofuro[3,2-g]chromen-7-one 1-[3-(azidomethyl)-2,6-dichlorophenyl]pyrrole 6-chloro-2-(4-bromophenyl)imidazo[1,2-a]pyrimidine 2-[(5S)-3-benzyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ium-1-carbonyl]prop-2-enedioate 2-[3-(4,5-dimethylpyrimidin-2-yl)piperidine-1-carbonyl]-5-ethylsulfonylbenzaldehyde 2-amino-N-[(2S)-1,1-bis(4-chlorophenyl)butan-2-yl]acetamide 2-[(4-cyclopentyloxycarbonyl-1,3-thiazol-5-yl)sulfonyl]-2-methylbutanoic acid 1-[4-(6,7-dihydrobenzo[a]quinolizin-5-ium-10-yl)cyclohexa-2,4-dien-1-ylidene]guanidine [4-[[5,6-dimethyl-3-(5-methylcyclohexa-1,5-dien-1-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]piperidin-1-yl]-phenylmethanone N-[(3R,4S)-1-tert-butyl-2-oxopyrrolidin-3-yl]-5-methoxypyridine-3-carboxamide 2-[4-(4,5-dihydrotriazol-1-yl)phenyl]-6,7-dimethoxy-3H-quinazolin-4-one [2-[3-(3,4-dichlorophenyl)propyl]morpholin-4-yl]-quinolin-6-ylmethanone N-[1-amino-3-(4-methoxyphenyl)propan-2-yl]carbamate 1-[(4aS,9aR)-1,3,4,4a,5,6,7,8,9,9a-decahydropyrido[2,3-b]azepine-2-carbonyl]pyrazole-3-carboxylic acid 2-amino-4-[3-(dipropylamino)phenyl]-6-methylbenzene-1,3-dicarbonitrile 6-[2-methylpropanoyl(1,3-thiazol-5-yl)amino]pyridine-4-sulfonic acid 4-[6-amino-5-(cyclopropylmethoxy)pyridin-3-yl]-7-fluoro-2H-phthalazin-1-one N-[1-(2,6-dichlorophenyl)ethenyl]-5-fluoro-4-methoxypyrimidin-2-amine 6-[1-amino-2-(2,3,4-trifluorophenyl)ethyl]-N-[[4-(difluoromethoxy)phenyl]methyl]pyrimidine-4-carboxamide;hydrochloride N-(2,3-dichloro-4-nitrophenyl)-2,5-dimethyl-N-phenacylbenzenesulfonamide 2-[4-[2,3,4,5-tetrafluoro-6-(1-methylpyrrolidin-2-yl)phenyl]piperidin-1-yl]ethanol N-[4-fluoro-3-(trifluoromethyl)phenyl]pyrrolidine-2-carboxamide 1-chloro-4-[2,3,3,5,6-pentadeuterio-4-fluoro-5-(trideuteriomethyl)phenyl]-2-phenylbenzene 4-[[(Z)-2-amino-3,3-dimethylbut-1-enyl]sulfanylmethyl]benzenecarboximidamide N-(2,5-difluorophenyl)-5-[3-[(Z)-4-imino-4-methylpent-2-enimidoyl]phenyl]pyrimidin-2-amine N-[3-(5-methyl-1,2-dihydrotriazol-3-yl)phenyl]pyrazolo[1,5-a]pyridine-6-carboxamide 1-[1-(2,2,3,3,4,4,5,5,6,7,8,9,10-hexadecafluorodecyl)cyclohexyl]triazole 4-(3,5-dimethylphenyl)-N'-hydroxy-2-(4-methoxypiperidin-1-yl)butanimidamide 1-[4-(6,7,8,9,10,11-hexahydrocycloocta[b]pyran-2-yl)piperazin-1-yl]ethanone 3-[3-(4,5-dimethyl-1H-imidazol-2-yl)phenoxy]butan-2-one 1-cyclopropyl-3-[4-(difluoromethoxy)phenyl]pyrazolo[3,4-c]pyridine N-[(3-ethoxy-1H-pyrazol-5-yl)methyl]-2-(9H-fluoren-2-yloxy)benzamide 2-[(E)-5,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl]quinoline-8-carbonitrile (E)-3-[4-[5-[2-(cyclopropylamino)pyrimidin-4-yl]-1,6-dihydropyrrolo[2,3-b]pyridin-4-ium-3-yl]phenyl]prop-2-enenitrile N-(2,3-dimethylphenyl)-3-(4-methoxyphenyl)pentanamide 6-hydroxy-5,9b-dimethyl-6H-benzimidazolo[1,2-a]quinoxaline 2-methyl-3,4-diphenyl-9H-carbazole [(2S)-2,4-dimethylpentoxy]methylbenzene 1,5-bis[(4-tert-butylphenyl)methoxy]pentan-3-one 1-phenyl-4-piperidin-2-ylpyrazolo[3,4-b]pyridine 2-[3-(6,7-dimethoxyquinazolin-4-yl)sulfanylphenyl]butylcarbamic acid 2-hydroxy-6-oxo-N-[1-(4-phenylphenyl)-2-pyrrolidin-1-ylethyl]piperidine-3-carboxamide;hydrochloride 2-cyclopropyl-6-[[(1R)-4,5-difluoro-2,3-dihydro-1H-inden-1-yl]oxy]-1-[(6S)-2,2-dimethyl-4,5,6,7-tetrahydro-1,3-benzodioxol-5-yl]indole 3-azido-4-(2,6-dichlorophenyl)-5-methyl-1,2-oxazole 1-methyl-2-[4-(trifluoromethoxy)phenyl]benzimidazole N-[3-bromo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]formamide 2-[4-(3,5-dimethylphenoxy)phenyl]-6-oxo-1H-pyrimidine-5-carboxylic acid 1-azido-2,6-ditert-butyl-4-(3-phenylphenyl)benzene 3-[2-(1,3-dimethylpyrazol-4-yl)ethoxy]-5,8-bis(2-methylpropyl)pyrido[2,3-b]pyrazin-6-one 2-(3,4-dihydro-1H-isochromen-1-yl)-5-[(3R,4S)-3-methoxypiperidine-4-carbonyl]-7,8-dihydro-6H-pyrazolo[1,5-a][1,4]diazepin-4-one 3-(1,5-dimethylpyrazol-4-yl)-6-[4-hydroxy-2-[[2-methoxyethyl(methyl)amino]methyl]phenyl]-8-methoxypyrido[3,4-d]pyrimidin-4-one 4-(3-bromophenyl)sulfanyl-2-methoxybenzaldehyde 2-[(2R,6S)-4-butoxy-6-methyloxan-2-yl]ethylcarbamic acid (3R)-2,6-diamino-4-[(1R)-1-phenylpropyl]hexanoic acid 1-(benzenesulfonyl)-3-[4-(furan-2-ylmethylideneamino)butanoyl]urea 6-bromo-N-(2,6-dimethylphenyl)-3-iodoimidazo[1,5-b]pyridazin-8-amine N-cyclohexyl-6,7-dimethoxy-1-methylquinolin-4-imine;(E)-3-methylideneoct-5-enal 2-ethoxy-N,N-dimethyl-4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)aniline 5-[3-(4-chlorophenoxy)propyl]-7-methoxy-2,3-dihydro-1H-benzotriazole 4-[(4,5-dimethyl-1H-imidazole-2-carbonyl)amino]hexanedioic acid 3-[5,6-diamino-2-(2-methoxyethyl)pyrimidin-4-yl]phenol 2-(azepan-1-yl)-4,6-dichloropyrimidine 4-[3-[(2E,4Z)-hepta-2,4-dien-6-yn-2-yl]imidazo[1,2-a]pyridin-7-yl]-N'-hydroxybenzenecarboximidamide 4-[(Z)-3-fluoropent-1-enyl]-6-methoxyquinoline N-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]propanamide 7-benzyl-2-chloro-3,6,8,9-tetrahydro-1H-pyrido[4,3-e][1,5]diazecine (5S,8R)-N-[2-methyl-1-(oxan-4-yl)piperidin-3-yl]-5-phenyl-7-(trifluoromethyl)-4,5,6,8-tetrahydropyrazolo[1,5-d][1,4]diazepine-2-carboxamide 3-[2,5-dioxo-4-[4-(N'-phenylmethoxycarbamimidoyl)phenyl]imidazolidin-1-yl]propanamide N-[(4,5-dimethyl-1H-imidazol-2-yl)methylideneamino]pyridine-3-carboxamide N-[4-(diethylamino)phenyl]-3-methoxy-10-phenylacridin-9-imine 4-amino-3,5,6-trichloropyridine-2-carboxylate 5-bromo-N-[(E)-(4-ethoxy-2,6-difluorophenyl)methylideneamino]pyrimidine-2-carboxamide N-[3,5-dibromo-2,6-bis(hydroxymethyl)phenyl]-4-oxochromene-2-carboxamide 1-(4,6-dichloropyrimidin-5-yl)imidazole N'-[5-(2,6-dichlorophenyl)furan-3-yl]-N-hydroxyimidazole-1-carboximidamide 2-(4-fluorophenyl)-2-[(3S,7R)-11-hydroxy-12-methoxy-8-oxa-14,15-diazatetracyclo[7.6.0.02,7.010,14]pentadeca-1(9),2,4,6,13-pentaen-5-yl]acetic acid N-[(4S,5S)-3,3-difluoro-7-oxabicyclo[2.2.0]heptan-6-yl]-2-(5,8-dihydroxyquinolin-2-yl)acetamide 2-(2,4-diaminophenyl)sulfanylnaphthalen-1-ol 2-[3-(1,4-diazepan-1-yl)propyl]-5-hydroxy-6-methoxy-3H-isoindol-1-one 1-(2-methylphenyl)-4-(6-phenoxycyclohexa-2,4-dien-1-ylidene)piperidine 3-[1-(2,4-difluorophenyl)cyclobutyl]oxy-5-[2-[2-methylsulfonylethyl(propyl)amino]pyrimidin-5-yl]pyridine-2-carboxamide N-[(3S,4R)-1-cyclopentyl-3-(dimethylsulfamoylamino)piperidin-4-yl]-5-phenyl-1H-pyrrolo[2,3-b]pyridine-4-carboxamide 5-(2,6-difluorophenyl)-N-ethenylpyridine-3-carboxamide 3-(2,6-dichlorophenyl)-7-[4-ethyl-1-methyl-5-(piperazine-1-carbonyl)pyrazol-3-yl]-8H-1,8-naphthyridin-4-one 3-[2-bromo-4-(trifluoromethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile [5-methyl-6,7-bis(2-methylpropoxy)naphthalen-1-yl]-phenoxyphosphane 2-[6-(7-chloroquinolin-4-yl)oxynaphthalen-1-yl]-N',N'-diethylpropanediamide 4-amino-N-methyl-1-(1,2,3,5,6,7-hexahydropyrrolizin-8-yl)pyrazolo[3,4-d]pyrimidine-3-carboxamide 4-cyclopentylsulfanyl-N',N'-dimethylbenzohydrazide (E)-5-[2-hydroxyethyl(methyl)amino]pent-4-enal;2-methyl-3-(propan-2-ylideneamino)but-1-ene-1,4-diol;4-oxo-4-pyridin-4-ylbutanenitrile (2-methyl-1,3-oxazol-4-yl)-[7-(2-phenylethynyl)furo[3,2-b]pyridin-5-yl]methanone N-(4-chlorophenyl)-N-prop-2-enylhexadecanamide 2-[N-(benzenesulfonyl)-4-methoxyanilino]decanoic acid 2-[(3-methylphenyl)methylamino]-N'-(4-propan-2-ylphenyl)ethanimidamide 3-cyclohexyl-4,5-dimethoxybenzamide 5-[7-(difluoromethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-3-yl]furan-3-carboxylic acid;2,2,2-trifluoroacetic acid 4-[2,3-difluoro-4-(trifluoromethoxy)phenyl]cyclohexan-1-ol 4-amino-1,2,5-tris(sulfanyl)anthracene-9,10-dione 2-[4,4-difluoro-5-[(5E)-4,8,10-trimethylundeca-3,5,7,9-tetraenyl]cyclohexa-1,5-dien-1-yl]-5-octoxypyrimidine N-(1,2-benzothiazol-6-yl)-2-(4-chlorophenyl)acetamide;ethane [2-methoxy-5-(3,4,5-trifluorophenyl)-1,3-dihydroinden-2-yl]carbamic acid 6-chloro-N-ethylnaphthalen-2-amine 5-[4-chlorobutyl(2,3-dihydroxypropyl)amino]-N-(4-methylpyrimidin-2-yl)-1H-pyrrole-3-sulfonamide N-[5-methyl-2-(4-oxo-1-phenyl-5H-pyrazolo[3,4-d]pyrimidin-6-yl)pyrazol-3-yl]naphthalene-2-carboxamide 1-N',2-N'-bis[(4-fluorophenyl)methyl]butanedihydrazide 6-[4,5-dibromo-1-(4-ethylphenyl)-3-hydroxypyrazol-2-ium-2-yl]oxy-7-fluorochromen-2-one N-[4-amino-3-[(Z)-prop-1-enyl]phenyl]cycloheptanecarboxamide 1-[4-(4-bromophenoxy)phenyl]piperazine (E)-2-ethyl-3-(methylideneamino)-4-phenylbut-1-en-1-ol N-[3,5-bis(trifluoromethyl)phenyl]-2-chloro-1-propyl-9H-fluorene-9-carboxamide [(2R,6S)-6-methylmorpholin-2-yl]-phenylmethanol;hydrochloride 7-[5-(6,8-dimethyl-2H-quinolin-1-yl)pentanoyl]-9H-fluorene-1-sulfonic acid 2-[5-(3,5-dichlorophenyl)thiophen-2-yl]acetamide 2-[[3,5-dichloro-4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-ylamino)phenyl]methyl-ethylamino]acetic acid 3-[2,4-dimethyl-5-(methylamino)phenyl]-N-[2-[2-hydroxyethoxy-(4-methylphenyl)sulfonylamino]ethyl]benzamide 1,3-dichloro-4-cyclohexylbenzene;ethane (6S)-6-[5-cyclopropyl-3-fluoro-2-(methoxycarbonylamino)phenyl]-1,4-oxazepane-4-carboxylic acid 1-(3-chlorophenyl)-2,5-dimethylcyclohepta-3,5-diene-1,4-dione;4-(3-formylbenzene-6-id-1-yl)butanenitrile;uranium(2+) N-(cyclopropylmethyl)-5-[4-[4-(2,3-dihydroindol-1-ylsulfanyl)phenyl]pyrazol-1-yl]pentanamide 2-[[4-(6-methoxyquinolin-4-yl)cyclohexyl]amino]pyridine-3,5-dicarboxamide [4-(3,5-dimethylpyrazol-1-yl)phenyl]-phenylmethanone 2-amino-N-[1-(1-methylpyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyridine-3-carboxamide 5-[6-bromo-2,3-difluoro-4-(oxiran-2-ylmethoxy)phenyl]-1H-imidazole N-[4-methyl-3-(2-morpholin-4-ylethoxy)phenyl]carbamate 2-(9H-fluoren-9-ylmethoxycarbonylamino)butanoic acid 2-(4,5-dichloroindol-1-yl)-N-[3-fluoro-6-[1-(methanesulfonamido)ethenylamino]pyridin-2-yl]acetamide N-(5,6-difluoroindol-1-yl)formamide 3-[4-(3,5-dimethylpyrazol-1-yl)anilino]-1-phenylpropan-1-one 5-(2,3-dihydrothiophen-4-yl)-N-[1-[2-[3-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide (2Z,4Z)-7-[3-(4-tert-butylphenyl)-6-methylidenecyclohexa-1,4-dien-1-yl]-5-chlorohepta-2,4-dienenitrile N-[[4-(3,4-dimethoxyphenyl)cyclohexyl]methyl]imidazo[1,2-a]pyrazine-8-carboxamide N-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)ethynyl]cyclopropanecarboxamide [2-[(1R)-1-(4-bromophenyl)ethyl]-7-methoxyspiro[3,9-dihydro-1H-pyrido[3,4-b]indole-4,3'-pyrrolidine]-1'-carbonyl]carbamic acid 3-bromo-2,4,5,6-tetrachlorobenzoic acid N-[1-(2,4-dichlorophenyl)ethyl]-1-[[(E)-3-methylidene-6,7-dihydro-5H-pyrazolo[5,1-c][1,2,4]triazol-6-yl]methyl]piperidine-4-carboxamide 3-methyl-1-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)pyrrolidine-1-carbonyl]cyclobutan-1-ol;hydrochloride 2-(5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carbonyl)benzoic acid 5-[2-hydroxy-4-(3-methylbutanoyl)phenyl]iminopyrazolidine-3-thione 1-(2,6-difluorophenyl)-4-[2-[[3-(trifluoromethyl)benzoyl]amino]ethyl]pyrazole-3-carboxamide 7-[(5R)-2,2-dimethyl-4,5-dihydro-1H-1-benzazepin-5-yl]-N'-ethylimidazo[1,2-a]pyridine-6-carboximidamide 3-(2,2-diethoxyethyl)-N-(3-methylbutyl)aniline (2R)-3-cyclobutyl-N,2-dihydroxypropanamide;1,4-difluorobenzene;1-(3-methoxy-6-azabicyclo[3.1.0]hexan-6-yl)-3-phenylpropan-1-one 1-(3,5-dichlorophenyl)sulfanylpiperidine [(2S)-1-chloro-4,4-difluoro-2-hydroxy-3-oxobutyl]-[6-[5-fluoro-7-methoxy-6-(piperazin-1-ylmethyl)pyridin-2-yl]-2-phenylpyrimidin-4-yl]carbamic acid 5-chloro-2,4-bis(trifluoromethyl)pyridine-3-carboxylate 3-(2,4-dimethylcyclohexen-1-yl)oxy-2-fluorobenzaldehyde N-(5,6,7,8-tetrahydronaphthalen-1-ylmethyl)propan-2-amine [2-(4-chlorophenyl)cyclopropyl]-[2,3-dihydroindol-1-ylmethylamino]methanol (2S)-2-[3-chloro-5-[5-[3,4-difluoro-6-(1H-indol-2-yl)cyclohepta-1,3,6-trien-1-yl]-2,4-dimethoxyphenyl]-1-methylsulfonylindole-7-carbonyl]pyrrolidine-1-carboxylic acid 2-[4-(benzoylsulfamoyl)-N-hexadecylanilino]acetamide N-[4-(2,6-dimethoxyphenoxy)-3-(3-propan-2-ylpyridin-1-ium-1-yl)phenyl]pyridine-2-carboxamide;2-[[5-[3-(furan-3-yl)-1H-indol-5-yl]-2-oxo-1,3-oxazolidin-3-yl]methyl]pyridine N'-[3-cyano-5-(6,7-difluoroquinolin-4-yl)pyridin-2-yl]-1H-pyrrole-2-carboximidamide 1-[2,6-bis(phenylmethoxy)-3,4-dihydronaphthalen-1-yl]ethanone 2-(4,5-dimethyl-1H-pyrazol-3-yl)-7-methoxy-6-methylsulfanyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine (2S)-N-[[1-(4-chlorophenyl)cyclohexyl]methyl]-1-[6-oxo-3-(trifluoromethyl)pyridazin-1-yl]pyrrolidine-2-carboxamide 3-benzylsulfanyl-N'-hydroxypyrazine-2-carboximidamide 2-[5,6-dimethoxy-1-[4-[(E)-3-phenylprop-2-enyl]piperidine-1-carbonyl]indol-3-yl]acetic acid 1-[2,4-difluoro-3-(trifluoromethyl)phenyl]-N-piperidin-4-ylmethanimine 3-[(4Z,8E)-9-fluoro-10-hydroxy-11-imino-8H-naphtho[1,2-b][1]benzazepin-5-yl]benzonitrile 2-bromo-3-chloro-6-methoxypyridine 1-[4-[3-(2,6-difluorophenyl)-1H-pyridazin-2-yl]cyclohexa-2,4-dien-1-ylidene]azepane N-[4-amino-5,6-diethoxy-7-(1H-pyrazol-5-yl)quinazolin-2-yl]propanamide (E)-N-hydroxy-3-[2-(3,4,5-trichlorophenyl)-1H-imidazol-5-yl]prop-2-enamide 4-azido-3,5-dimethylbenzoic acid (5Z)-4-benzyl-1-ethenyl-2,3-dihydroindene 4-bromo-5-phenyl-2H-isoindole N'-[(Z)-(2-hydroxynaphthalen-1-yl)methylideneamino]-N-(3,4,5-trimethoxyphenyl)oxamide 4-cyclohexyl-2-methyl-5,6-diphenylpyrimidine (1E,3Z)-2-amino-5-[9-(2-methylphenyl)dibenzothiophen-1-yl]penta-1,3-dien-1-amine 2-[4-(1,3-benzodioxol-5-yl)phenyl]-N-(3,6-dihydro-2H-pyridin-1-ylsulfonyl)acetamide [3-[[3-(trifluoromethyl)phenyl]carbamoylamino]azetidin-1-ium-1-ylidene]oxidanium 3-bromo-2-ethylpyrido[1,2-a]pyrimidin-4-one (2S)-1,4-dioxan-2-amine;2-[3-(4-fluorophenyl)prop-1-en-2-yl]phenol 2-bromo-7-cyclobutyloxyimidazo[1,5-a]pyridine 1-N',2-N'-bis[3-(2-ethylimidazol-1-yl)propyl]hexanedihydrazide 4-[5-(6,7,8-trimethoxyquinazolin-4-yl)-1H-pyrazol-3-yl]phenol N-[3-(4,5,6,7-tetrahydrobenzimidazol-1-ylmethyl)phenyl]hydroxylamine 1-[2,3-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyridine-4-carbonyl]azetidine-3-carboxylic acid N-(2,6-diethyl-4-propanoylphenyl)acetamide;2-methoxycarbonylcyclobutanedioic acid [(5R,7S)-2,5,7-trimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carbonyl]carbamic acid N-[4-(2,5-dimethylphenyl)butanoyl]-6-oxo-1H-pyridine-3-carboxamide ethane;3-fluoro-2-[6-(4-morpholin-4-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]aniline 1-[5-(2,3-dihydro-1H-inden-4-yl)pyrazin-2-yl]-3-methylidene-2-N-phenylsulfanylpiperazine-2,6-diimine 3-[3-(aminomethyl)phenyl]-2-[4-hydroxybutyl(propanoyl)amino]benzoic acid (1S)-1'-methyl-6,8-diphenylspiro[3H-furo[2,3-f]chromene-3,4'-cycloheptene] [6-[3-amino-2-(hydroxymethyl)phenyl]imidazo[1,2-a]pyridine-7-carbonyl]oxidanium 3-[4-[2-(2,3-dihydroxypropoxy)ethoxy]phenoxy]propanal [2-(benzylamino)thieno[3,2-c]pyridin-4-yl]-(2-cyclohexylphenyl)methanone 1-phenyl-3-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-7-yl)imidazol-1-yl]propan-1-one 3,4-bis(ethenyl)naphthalene;ethane 2-(5-chloroquinolin-8-yl)oxy-N-[4-(5,6-dimethylbenzimidazol-1-yl)-3-fluorophenyl]pentanamide 5-(6-fluoroquinolin-4-yl)spiro[1H-2,3-dihydro-benzofuran-3,4'-piperidine] 4-(3-fluoropropyl)-2-[6-methoxycarbonyl-5-[(1R)-1-phenylethoxy]pyridin-3-yl]morpholine-4-carboxylate 2-(4-amino-3,5-dichlorophenyl)-N-tert-butylsulfonyl-1H-benzimidazole-4-carboxamide 5-[(E)-2-phenylprop-1-enyl]-4H-pyridine 3-[3-methylbutyl-(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid N-[(Z)-1H-indol-3-ylmethylideneamino]-2-[5-(4-methoxyphenyl)-2,4-dioxopyrimidin-1-yl]acetamide 3-(7H-purin-6-yl)benzenethiol N-[3-(1H-benzimidazol-2-yl)phenyl]-4-methoxybenzamide N-[4-fluoro-5-(5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-ylamino)pyridin-2-yl]ethanesulfonamide 4-[2-[[(3E)-hexa-1,3,5-trien-3-yl]amino]pyrimidin-4-yl]-N-[4-methoxy-3-(morpholine-4-carbonyl)phenyl]furan-2-carboxamide 1,2-diamino-4-[4-bromo-3-(2-nitrophenyl)sulfanylphenyl]-6-oxopyridine-3,5-dicarbonitrile 3,6-diphenyl-1H-[1]benzofuro[2,3-d]pyrimidine-2,4-dione 7-(2,5-dimethylcyclohexen-1-yl)-N'-hydroxyisoquinoline-1-carboximidamide 6-[5,6-dideuterio-2-(trifluoromethyl)pyridin-3-yl]-4-N-propan-2-ylpyrimidine-2,4-diamine 5-(2-chloro-6-cyclopropylbenzoyl)pyridine-3-carboxylic acid 2-[3,5-bis(trifluoromethyl)phenyl]ethanethiol;methoxymethane N-[[4-[(4,5-dihydro-1H-imidazol-2-ylamino)methyl]phenyl]methyl]-4-formylbenzamide [(2R)-1-[4-[2-chloro-4-fluoro-N-[[5-(trifluoromethyl)pyrimidin-2-yl]amino]anilino]cyclohexyl]pyrrolidin-2-yl]carbamic acid 4-[5-bromo-2-(1H-indol-3-yl)phenyl]sulfanylbenzenecarboximidamide (6S)-7-acetyl-3-butylsulfanyl-6-(3,4,5-trimethoxyphenyl)-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one [2-(5,6-dichlorocyclohexa-1,3-dien-1-yl)hydrazinyl]-phenylmethanol 2-amino-9-(1,3-benzodioxol-5-ylmethyl)-6-(5-hydroxypyridin-2-yl)-7H-purin-8-one 2-N,4-N,4-trimethyl-6-[(1-methylpiperidin-3-yl)methoxy]pyridine-2,3,4-triamine (1S,5R)-3-[4-chloro-3-(trifluoromethyl)phenyl]-7-[5-ethynyl-6-(1,2,3,6-tetrahydropyridin-4-ylmethyl)pyrimidin-4-yl]oxy-8-azabicyclo[3.2.0]heptane N-[2-(3,4-dichlorophenyl)-1-hydroxyethyl]-3-propan-2-yloxypyridine-4-carboxamide (2E,4Z)-N'-(3H-benzimidazol-5-ylmethyl)-6-(N-ethenylanilino)-2-ethylidenehexa-3,5-dienimidamide 3-(4-iodophenyl)sulfanyl-1-naphthalen-2-ylpyrrolidine 2-(4,5-dihydrotriazol-1-yl)-N-[(6-methoxypyridin-3-yl)methyl]pyrimidin-4-amine 1-[4-[[2-(cyclopropylmethoxy)-5-fluorophenyl]methylamino]piperidin-1-yl]ethanone 3-[(1E)-2-(4,5-dimethylpyrazol-1-ium-1-ylidene)ethoxy]benzonitrile;tetrafluoroborate 4-[1-(2,5-dimethylphenyl)ethenoxy]benzonitrile 4-N,6-diethyl-2-N-[1-(3-methoxyphenyl)ethylideneamino]pyrimidine-2,4-diamine 2-[4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]acetic acid 2-[6-[(4-methoxyphenyl)methyl]pyridin-3-yl]-5H-pyrido[3,2-b]indole 2-[4-(4-methylpentoxy)phenyl]ethanimine 5-[(E)-2-amino-1-[(6Z,8E)-6-propan-2-ylidene-9H-pyrido[3,4-b]indolizin-5-yl]ethenyl]pyrazin-2-amine (5-chlorothiophene-3-carbonyl)azanium;[4,6-diamino-5-[2-(furan-2-ylmethylcarbamoyloxy)ethyl]pyrimidin-2-yl]-formamidoazanide 5-[2,4-bis(trifluoromethyl)phenyl]furan-3-carboxylic acid 4-(2,3-diethoxyphenyl)-1H-indene 4-[1,2-difluoro-2-(3-fluorophenyl)ethenyl]-N'-methanimidoyl-2-methoxybenzenecarboximidamide 2-(3-azido-1,4-diphenylbutyl)-1H-imidazole 2-[5-(ethylamino)-4-oxoquinazolin-3-yl]acetic acid (E,2S)-N-cyclopropyl-5-[4-methoxy-3-(trifluoromethoxy)phenyl]-1-(prop-2-enoxyamino)pent-4-en-2-amine 2-[N-(4-hydroxybutyl)-3-nitroanilino]octanoic acid [(2R,3S)-1-methyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]carbamic acid 7-hydroxy-N,2-dimethyl-6-(4-phenylpiperazin-1-yl)imidazo[1,2-a]pyridine-3-carboxamide 2-[(4S,5R)-4,6-bis(benzylsulfanyl)-1,3-dimethyl-3-propyl-2H-pyrazin-5-yl]ethanol 1-(2,3-dihydrofuran-5-yl)-N-[(2S)-4-ethylhexan-2-yl]-N'-methylimidazole-4-carboximidamide N-azido-3-[2,6-dibromo-4-[(2R)-1,1,1-trifluoropropan-2-yl]oxyphenyl]propane-1-sulfonamide N-cyclopentylformamide;3-[2-(cyclopropylamino)pyrimidin-4-yl]-5-ethynyl-1H-pyrrolo[2,3-b]pyridine-7-carboxamide (3S)-N,N'-diamino-3-[5-chloro-2-fluoro-4-methyl-3-[(E)-pent-1-enyl]phenoxy]pyrrolidine-1-carboximidamide 3-(4,5-dimethylfuran-2-yl)-1-[2-[4-(trifluoromethoxy)phenyl]ethynyl]pyrrolo[2,3-b]pyridine 2-(4-bromophenyl)-N-[(Z)-[4-(naphthalen-1-ylmethoxy)phenyl]methylideneamino]acetamide 1-[[4-(2,5-difluorophenyl)pyridin-3-yl]methyl]-N-ethylpiperidine-4-carboxamide 1,2-dimethyl-3-(4-propylphenyl)benzene;ethane 3-[4-(3,5-dichloroanilino)-7-methoxyquinazolin-6-yl]oxypropan-1-ol 2-[4-methyl-1-oxo-1'-(pyridin-3-ylmethyl)spiro[indole-3,4'-piperidine]-5-yl]acetamide;2,2,2-trifluoroacetic acid 3-[2-(6-methylpyridin-3-yl)ethenyl]phenol 1-[2-ethyl-4-(trifluoromethoxy)phenyl]ethanone 2-(1H-benzimidazol-2-yl)quinolin-7-ol 2-[6-fluoro-5-(3-methylbutanoyl)pyridin-3-yl]oxybutanedioic acid N-[4-(ethylideneamino)phenyl]benzamide 6-[2-[4-(dimethylamino)phenyl]-4,5-bis[[1-(oxiran-2-ylmethoxy)naphthalen-2-yl]oxy]phenoxy]hexan-3-one 5-ethoxy-6,7,8-trimethylquinoline 4-[1-(dimethylamino)propan-2-yl]-N,3-dihydroxybenzamide;ethane 6-methyl-1-phenylindole-3-carboxylic acid 1-benzyl-3-(2-fluorophenyl)imidazolidine 2-(N-hexadecanoylanilino)acetic acid (2S)-4-[(2S)-1-hydroxypropan-2-yl]oxy-1-methyl-3H-2,1-benzoxaborole 2-[4,6-dimethyl-1'-(pyridine-3-carbonyl)spiro[2H-indole-3,4'-piperidine]-1-yl]acetic acid;2,2,2-trifluoroacetic acid 4-[2-(2,6-difluoro-3,5-dimethoxyphenyl)imidazol-1-yl]pyridine 1,3-difluorobenzene;3-[(E)-2-(5-fluoropyridin-3-yl)ethenyl]pyridine (3,4-difluoro-2-methylphenyl)-[5-hydroxy-8-(trifluoromethoxy)quinolin-2-yl]methanone 1-[(Z)-3,4-dihydro-2H-naphthalen-1-ylideneamino]piperidin-3-ol 3-(hydroxymethyl)-2,4-bis(2-phenylethynyl)phenol 4-(2-azidooxyethyl)benzonitrile N-[(2-methylphenyl)methyl]-1-[4-(trifluoromethoxy)phenyl]ethanamine 1-[4-(3,4-difluorophenyl)sulfanyl-2,6-bis(methoxymethyl)phenyl]-N'-ethenylpropane-1,3-diamine (4S)-N,4-dimethyl-3-[6-propanoyl-2-(trifluoromethoxy)pyridin-3-yl]imidazolidine-1-sulfonamide 4-[6-(5-fluoro-2,3-dihydroindole-1-carbonyl)imidazo[1,2-b]pyridazin-3-yl]benzenesulfonamide 4-(1,2-dimethylcyclohexa-2,5-dien-1-yl)-N-[3-[(E)-pent-1-enyl]phenyl]naphthalen-1-amine 3-[(2-cyanophenyl)methyl]-4,5-dihydroimidazole-1-carboxamide 4-[3-hydroxy-2-(4-methoxyphenyl)prop-1-enyl]phenol N-[(3-propoxyphenyl)methyl]pyridine-2-carboxamide 2-(5-hydroxy-9,10-dioxoanthracen-1-yl)oxyacetic acid 1-[5,8-bis(trifluoromethyl)quinoxalin-2-yl]piperidine-4-carbonitrile [2-amino-6-(4-phenylmethoxy-1H-pyrrolo[3,2-c]pyridin-7-yl)pyridin-3-yl]-(4-azidopiperazin-1-yl)methanone 2-[4-cyano-3-(trifluoromethyl)phenyl]-8-methoxy-N,N-dimethyl-8-propanoyl-2,8-diazaspiro[4.5]decane-3-carboxamide 4-(5-amino-2-butoxyphenyl)-6,7-dihydropyrido[3,2-b]indole-5-carbonitrile 1-[(3-fluorophenyl)methyl]-4-(2H-indazol-6-yl)piperidine-3,4-diol 1-ethyl-N,6-dimethoxy-4-oxocinnoline-3-carboxamide 4-[3-(2,4-dichlorophenoxy)propyl]piperazine-1-carboxylic acid N-[(3R,4R)-1-methyl-4-propan-2-ylpyrrolidin-3-yl]-2-(8H-[1,2,4]triazolo[4,3-a]pyridin-7-ylidenemethyl)benzamide 2-[2-(1H-imidazol-5-yl)ethyl]-7,9-dihydropurin-8-one 4-amino-1-[2,3-difluoro-5-(2H-tetrazol-5-yl)phenyl]-2-[6-methyl-4-(trifluoromethoxy)pyridin-2-yl]butan-2-ol N-[5-(4-chlorophenyl)sulfonyl-3a,7a-dihydro-1H-indol-3-yl]-2-(oxolan-2-yl)acetamide 4-[2-(aminomethyl)-3-fluoroprop-2-enoxy]-N-propan-2-ylbenzamide N-[2-methyl-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]cyclopentanecarboxamide (5S,7R)-N-[1-(2-methylpyrazol-3-yl)pyrrolidin-3-yl]-1-propanoyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carboxamide 5-[[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]methoxy]-8-hydroxynaphthalene-1,7-disulfonic acid 1-[(4-tert-butylphenyl)methyl]-3,6-diethyl-2-methylindole;N-methylformamide (Z)-3-[4,6-bis(ethenyl)pyridin-2-yl]-1-(3,5-dimethoxyphenyl)prop-2-en-1-one N-(2,5-difluorophenyl)-2-[1-hydroxy-4-oxo-6-(2-phenylethylamino)-7H-pyrazolo[3,4-d]pyrimidin-5-yl]acetamide 5-[4-methyl-3-(2,2,2-trifluoroethoxy)phenyl]sulfinyl-2H-triazole-4-carboxylic acid 5-methylsulfonylsulfanyl-2-propoxybenzoic acid N-[2-(6,7-dimethoxyquinazolin-4-yl)oxypyridin-3-yl]ethanesulfonamide;N'-methyl-1-phenylpropan-1-imine N-[4-(2,6-difluorophenyl)cyclohexyl]-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide;hydrochloride 2-[5-fluoro-3-(5-phenylpyrimidin-4-yl)indol-1-yl]-N,N-dimethylethanamine 7-[(Z)-1-amino-3-iminoprop-1-en-2-yl]-N'-butan-2-yl-5-methylidene-6,10-dihydroanthracene-2-carboximidamide 1-(cyclopropylmethylamino)-3-[[5-(4-ethoxyanilino)thiophen-2-yl]sulfonylamino]thiourea 2-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)pyrazol-1-yl]acetamide 4-methyl-2-[5-(1,3-thiazol-2-yl)hexanoylamino]pentanoic acid 3-[4-(9,10-dioxoanthracen-2-yl)oxyphenyl]-2-methylprop-2-enoate 1-(3-azidophenyl)-4,5-dihydroimidazole N-ethenylmethanamine;methoxy-(2-phenylphenyl)phosphane N-[(1R,2S)-1-amino-3-methylbutan-2-yl]-7,8-dihydronaphthalene-1-carboxamide;1,4-diamino-3-hydroxypent-4-en-2-one [5-cyano-6-(cyclopropanecarbonylamino)pyridin-3-yl]azanide 2-(cyclohexylmethoxy)-4-(1H-indole-5-carbonyl)benzoic acid 2-cyclopentyloxy-3-[4-(trifluoromethyl)phenyl]phenol N-(5,6-dimethyl-2-phenylpyrazolo[1,5-a]pyrimidin-7-yl)-3-oxobutanamide 5-(3,4-difluorophenyl)-2-methylpyrimidine 5-N,8-diaminonaphthalene-2,7-disulfonamide 1,4-dioxonaphthalene-2-sulfonate 5-[3,4-dihydroxy-5-(2-phenylethyl)oxolan-2-yl]oxy-3-methylpentanoic acid (3S)-1-[6-amino-5-(4-chlorobenzenecarboximidoyl)pyrimidin-4-yl]piperidin-3-ol 1-(5-azidooxypentan-2-yl)anthracene (Z)-1-N',1-diethyl-1-N-methylidenebut-2-ene-1,1-diamine;4-(1H-indol-3-ylmethyl)benzaldehyde N-[4-(furan-2-carbonyl)phenyl]-2,5-dimethylpyrazole-3-carboxamide 4-(5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-2-yl)benzene-1,3-diol 5-[2-(2,4,6-trichlorophenyl)ethynyl]pyrimidine 3-[4-methyl-2-(2,4,6-trimethoxyphenyl)cyclohexa-1,5-dien-1-yl]propanamide 7-chloro-5-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-2-ethylpyrazolo[1,5-a]pyrimidine 1-(2,6-dichlorobenzoyl)-N-[4-(dimethylamino)phenyl]-2H-quinoline-3-carboxamide N'-hydroxy-1,3-dimethylpyrrolo[2,3-c]pyridine-5-carboximidamide 6-[4-(1H-imidazol-5-yl)butoxy]-3-[3-[2-(trifluoromethyl)pyridin-4-yl]propanoylamino]furo[3,2-b]pyridine-2-carboxylic acid N-[5-tert-butyl-2-methoxy-3-(phenylsulfanylamino)phenyl]formamide 4-[6-(1-adamantyl)pyridin-3-ylamino]-N'-cyclohexylbenzenecarboximidamide (3R)-1-[4-(4-methylsulfonylphenyl)-2-piperazin-1-ylquinoline-6-carbonyl]pyrrolidine-3-carbonitrile ethane;2-[1-(4-methoxyphenyl)sulfonylpiperidine-3-carbonyl]oxy-2-methylpropanoic acid (2R)-2-[(1R)-3,4-dihydroxycyclohexyl]oxy-N-(5-phenylpentan-2-yl)propanamide (3aR,7aS)-4-(2,5-dimethylbenzoyl)-1-(thiophen-2-ylmethyl)-3,3a,6,7,7a-hexahydroimidazo[4,5-c]pyridin-2-one;formic acid N-[(3R)-1-cyclopentylpiperidin-3-yl]-5,6-dimethoxypyridine-3-carboxamide 4-azido-N-(1,3-benzodioxol-5-ylmethyl)cyclohexan-1-amine 2-[[4-methoxy-3,5-bis(phenylsulfanyl)thiophen-2-yl]carbamoyl]cyclopropane-1-carboxylic acid 5-methylsulfonyl-2,3-dihydropyrido[4,3-b]indole 4-[(2,5-dioxopyrrol-1-yl)methyl]-N-[3-fluoro-4-(trifluoromethyl)phenyl]benzamide 1-[4-[(5-chloropyridin-2-yl)methoxy]piperidin-1-yl]-3-cyclohexylpropan-1-one N-[(E)-[4-(diethylamino)phenyl]methylideneamino]-5-ethyl-1H-pyrazole-3-carboxamide (2R,4S)-2-[5-(4-fluorophenyl)-1H-imidazole-2-carbonyl]piperidin-4-ol 2,3-difluoro-1-[4-(triazol-1-ylmethyl)phenyl]sulfonylpiperidine 5-(4-methylpiperazine-1-carbonyl)-2-[[5-(3,4,5-trifluorophenyl)pyridin-3-yl]amino]benzonitrile 3-[(E)-2,5-dimethyloct-4-en-3-yl]sulfonylphenol 4-[5-(cyclohexylmethoxy)pyrimidin-2-yl]-N-ethylsulfanylaniline;1,3-thiazol-4-one N-[4-(2,3-dihydro-1H-indene-1-carbonylamino)cyclohexyl]furan-2-carboxamide N-[3,5-difluoro-4-(trifluoromethyl)phenyl]-1-[1-(6H-cyclohepta[d]pyrimidin-2-yl)piperidin-4-yl]azetidine-3-carboxamide 4-(3-fluorophenyl)-5,6,7,8-tetrahydronaphthalene-2-carbonitrile 4-[[3-(4,6-dimethoxypyrimidin-5-yl)-2H-1,2-oxazol-3-ium-5-yl]methylidene]morpholine 4-(2,3-dihydro-1H-inden-5-yl)-6,8-bis(trifluoromethoxy)quinoline 2-(azidomethyl)-1,3,5-tripropoxybenzene (3R,4S)-4-benzyl-N-(cyclopropylmethoxy)pyrrolidine-3-carboxamide;hydrochloride 2-chloro-N-[3-(dimethylamino)propyl]benzenesulfinamide 2-ethoxy-3,5-diiodobenzoic acid (4E)-2-cyclopentyl-4-[[3,5-dichloro-4-[(3-fluorophenyl)methoxy]phenyl]methylidene]-1H-imidazol-5-one N-[(Z)-1H-indol-3-ylmethylideneamino]-2,4-dinitrobenzenesulfonamide 4-(2,3-dihydro-1H-indole-5-carbonyl)-2,5-dimethyl-1,4-benzothiazin-3-one (3R)-2,4-diamino-5-[6-(tert-butylcarbamoylamino)purin-9-yl]pentanoic acid (E)-2-ethoxycarbonyl-3-[5-(4-methoxyphenyl)thiophen-2-yl]prop-2-enoic acid (4Z)-2-cyclopentyloxycarbonyl-3,4-dimethylidene-5-phenylpyrazole-1-carboxylic acid 4-[(5S)-2-[5-chloro-3-[(4-methylphenyl)sulfonylamino]pyridin-2-yl]imino-1,3-thiazolidin-4-yl]butanoic acid [3-fluoro-5-(trifluoromethyl)phenyl]boronic acid 2-(4-anilino-N-methylsulfonylanilino)benzenesulfonic acid 3-N-[5-(difluoromethyl)-1,2,4-oxadiazol-3-yl]-6-morpholin-4-ylpyridine-2,3-diamine (2S)-1-[3,4-bis(methylsulfanylmethoxycarbonyl)phenoxy]propane-2-carboxylic acid 3-(2,5-dimethylphenyl)-6-(4-hydroxyphenyl)-7-iodo-1H-quinazoline-2,4-dione N-[5-(2,4-dichlorophenyl)sulfonylpyridin-2-yl]propanamide 2-(1,3-dihydroisoindol-2-yl)-N'-hydroxypyrimidine-4-carboximidamide 2-methyl-N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-7-yl)phenyl]sulfanyl-1H-indole-5-carboxamide;dihydrochloride [4-(2-phenylpyrazolo[1,5-a]pyrimidine-6-carbonyl)morpholin-3-yl]carbamic acid (2S)-1-[3,5-dimethyl-4-(2,2,2-trifluoroethylsulfonylamino)phenyl]pyrrolidine-2-carboxamide 3-[7-(5-chlorothiophen-2-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-[5-(cyclohexylmethyl)pyridin-3-yl]-2H-pyrazolo[3,4-b]pyridine N-[4-(aminomethyl)phenyl]-1,3,5,9-tetrahydropyrrolo[2,3-b]quinolin-8-imine 1-[4-(3,6-dihydro-2H-pyran-5-ylmethoxy)pyridin-2-yl]-N-[7-methoxy-8-(trifluoromethyl)quinolin-4-yl]piperidine-4-carboxamide N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)spiro[2.3]hexane-5-sulfonamide (1S)-3-methyl-N,N'-bis[2-methyl-4-(trifluoromethyl)phenyl]sulfanylbenzohydrazide N-(3-hydroxypropyl)-5-[(E,3Z)-3-[3-methoxyimino-4-oxo-6-(2,4,6-trimethylphenyl)hexan-2-ylidene]-2-methylpiperidin-1-yl]pyridine-3-carboxamide 3,3-dimethyl-2-[[3-(pyrimidine-5-carbonyl)-7,8-dihydro-6H-1,4-diazepin-5-yl]methyl]butanoic acid 4-(1,2-dihydrotriazol-3-yl)-N-[4-(1H-pyrazol-5-yl)pyridin-2-yl]piperazine-1-carboxamide 3-[(E)-1H-benzimidazol-2-yliminomethyl]chromene-4,8-dione (5R)-4-amino-2,2-dimethyl-7-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-5-(1H-pyrrolo[2,3-b]pyridin-4-yl)decanoic acid 2-[(2S)-1-cyclohexa-1,5-dien-1-ylpyrrolidin-2-yl]oxy-4-methoxy-N-phenylpyridine-3-carboxamide 4-[3,5-difluoro-2-(trifluoromethyl)phenyl]piperazine-1-carboxylate 5-[[4-(hydroxymethyl)pyrimidin-2-ylamino]methylideneamino]-1H-indazole-3-carboxamide 6-[5-(oxolane-2-carbonyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile 1-azido-4-(2-bromoethylsulfonyl)benzene 3-(4-bromophenyl)-2-[5-(4-methylsulfanylphenyl)thiophen-2-yl]prop-2-enenitrile N-(azidomethyl)-2-bromo-N-[2,4-difluoro-6-(propanoylamino)phenyl]benzamide N-butylsulfanyl-3,5-difluoroaniline 2-[1-(5-azidopentyl)-4-methoxynaphthalen-2-yl]oxythiophene 2-[6-chloro-4-(4-morpholin-4-ylpiperidin-1-yl)quinazolin-7-yl]oxyethanol 2-N,4-N-bis(3,5-dimethylphenyl)-1,4-dihydropyrimidine-2,4-diamine 2-[3-(7-methyl-4,5-dihydroimidazo[1,2-a]pyrimidine-8-carbonyl)phenyl]acetamide 2-(4-methoxyphenyl)-6,8-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,4,7-tetraene N-[2-(1-aminoethenyl)-1,3-dihydroinden-2-yl]-4-[(3Z)-hexa-1,3,5-trien-2-yl]cycloheptan-1-amine (6S)-5-oxo-N,9-diphenylnonanamide 2,3-dihydroxy-1,4-bis(phenylmethoxy)anthracene-9,10-dione N-[[2,6-diethoxy-4-(2-methylpropanoylamino)phenyl]carbamothioyl]cyclobutanecarboxamide 5-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)pyrido[4,3-b]indole 1-[(4S)-2,7-dimethylheptan-4-yl]sulfonylpyrazole N-(3,4-dihydro-2H-chromen-7-ylsulfonyl)oxane-4-carboxamide 3-[(4-chlorophenyl)methyl]-2-methylsulfanyl-6-oxo-1H-pyrimidine-5-carbonitrile 3-[4-chlorobutyl(hexyl)amino]phenol N-[(3S)-6-cyano-3,4-dihydro-2H-chromen-3-yl]-1-(furan-2-carbonylamino)cyclobutane-1-carboxamide 3-bromo-5,8-dimethylquinoline;ethane 6-(3,4-dimethoxyphenyl)imino-2H-benzo[de]isoquinoline-1,3-dione 2-[4-(3,5-dichlorophenyl)piperazine-1-carbonyl]-N-propan-2-ylbenzenesulfonamide 1-(4-fluorophenyl)-5,6-dihydrocyclopenta[b]pyridine-2,3-dione 5-[(4S)-7,8-dichloro-1,3-dimethyl-2,4-dihydropyrimido[4,5-d]pyrimidin-4-yl]-6-nitro-1,3-benzoxazol-2-amine N-(3,5-dichlorophenyl)-2-[4-[6-(2H-tetrazol-1-ium-1-yl)pyridine-3-carbonyl]piperazin-1-yl]acetamide N-[2,6-di(propan-2-yl)phenyl]-2-(3-methylcyclohexa-1,5-dien-1-yl)-6-oxo-1H-pyrimidine-4-carboxamide N-[2,4-difluoro-3-(8-methylquinazolin-6-yl)phenyl]acetamide 2-[(1R,3S)-3-aminocyclopentyl]oxy-5-bromobenzonitrile 5-(2,4-difluorophenyl)-7,8-dihydroisoquinolin-6-ol 5-[3-(difluoromethoxy)phenyl]-2,3-dihydro-1H-imidazole 1-N',3-N'-diphenylpropanedihydrazide 2-[6,7-dimethoxy-4-(3-pyrrolidin-1-ylphenyl)quinazolin-2-yl]phenol 4-[8-(3,4-difluorophenyl)-2-imino-1-propan-2-ylimidazo[4,5-c]quinolin-7-yl]cyclohexane-1-carboxylic acid 6-ethyl-2-methoxy-5,6-dihydrobenzo[h]quinazoline N-(2,4-difluorophenyl)-5-methyl-7-nitro-2,3-dihydroindole-1-carboxamide N-[3-[amino(hydroxy)methyl]phenyl]-4-chlorobenzamide 4-[2,6-dichloro-3-[(7,9-dimethyl-6H-pyrrolo[3,2-h]quinoxalin-8-yl)oxy]phenyl]-1,3-oxazolidine N-[1-(2,3-dihydro-1H-inden-5-yl)-6-ethoxypiperidin-3-yl]formamide ethane;4-(3-methylphenyl)-1,2-dihydronaphthalene N-(3,4-dihydroxyphenyl)-6-methylpyridine-3-carboxamide 3-[2-(2,4-dimethoxyphenyl)ethynyl]-5,6-dimethyl-1H-pyrrolo[2,3-b]pyridine 2-(2,3-dihydro-1H-inden-2-yl)-4,5-bis(4-propan-2-ylphenyl)oxadiazole 4-(3,5-difluorophenoxy)-1H-triazole-5-carboxylic acid N-[3,5-bis(trifluoromethyl)phenyl]-2,5-dichloro-4-methoxybenzamide (4R,5S)-3-[1-hydroxy-6-methyl-2-(propan-2-ylideneamino)hexyl]-7-oxo-4,5-dihydrothieno[3,2-c]pyran-6-carbonitrile [(4S,5R)-2,2-dimethyl-1,3-dioxolan-4-yl]oxymethylsulfanylbenzene 2-chloro-N,5-dimethyl-1-[(3S)-oxan-3-yl]pyrrole-3-carboxamide 7-N-[(2S)-1-methylpyrrolidin-2-yl]-8-nitroisoquinoline-3,7-diamine [5-cyclopropyl-2-[4-(3,5-difluorophenyl)-1H-imidazol-5-yl]phenyl]hydrazine (3S,4R)-1-[3-[8-amino-1-methyl-5-[(E)-pent-2-enimidoyl]imidazo[1,5-a]pyrazin-3-yl]propyl]piperidine-3,4-diol;ethane 1-[5-[(2R)-3-amino-1,1,1-trifluoropropan-2-yl]oxypyrazine-2-carbonyl]-N'-ethylpiperidine-4-carbohydrazide (2S,3R)-2,5-diamino-1-methyl-7-[4-methyl-6-oxo-5-[(E)-prop-1-enyl]-1H-pyrimidin-2-yl]-3-phenylazepane-2,4-diol 5-chloro-1-methylpyrazolo[3,4-d]pyrimidine;ethane 5-[(1Z)-buta-1,3-dienyl]-2-ethenyl-6-methylbenzene-1,4-disulfonic acid 1-methylspiro[1,2,4-triazol-3-one;nickel(2+);dichloride 4-(2,6-dimethylphenoxy)-3-[(E)-1H-imidazol-5-ylidenemethyl]-1H-indole 5-[[(3R,4S)-4-azidooxolan-3-yl]amino]pyrazine-2-carbonitrile (2S,3R)-3-methyl-1-[4-[(7-morpholin-4-ylquinoxalin-5-yl)amino]pyrimidin-2-yl]pyrrolidine-2-carboxamide 2-(4,5-dimethylthiophene-3-carbonyl)propanedioate 2-[6-chloro-1,3-dihydroisoindole-2-carbonyl(propyl)amino]-4-methylpentanoic acid N-butanoyl-2,6-dichlorobenzamide N-[3-(2,4-dimethylphenyl)-1H-indazol-5-yl]-5-(methoxymethyl)furan-3-carboxamide N-[(1R,2S)-2-aminocyclohexyl]-4-oxo-3H-quinazoline-6-carboxamide 6,8-dichloro-1-(3-fluorophenyl)-4H-isoquinoline [3-(1,4-dioxepan-6-ylmethyl)-6H-benzo[b][1]benziodol-5-ylidene]hydrazine 4-[(Z)-1-amino-2-(benzenecarboximidoyl)-3-hydroxyprop-2-enyl]phenol 3-[2-(9H-fluoren-1-yl)-5-methoxyphenyl]propanoic acid N-[3-(tert-butylamino)sulfanylphenyl]formamide 4-methoxycarbonyl-1-nitrosulfonylnaphthalene-2,3-dicarboxylic acid 7-chloro-1-(4,5-dihydro-1H-imidazol-2-ylmethoxy)-2-ethylimidazo[4,5-c]quinolin-4-amine N'-[(3S)-1-azidopyrrolidin-3-yl]-N'-[[4-methoxy-3,5-bis(trifluoromethyl)phenyl]methyl]oxamide 2-chloro-6-fluoro-5,8-dimethylthieno[3,2-g]chromene 4-[3-(2,5-dimethoxyphenyl)propyl]morpholine 4-(5,6-dihydroxypyridin-2-yl)benzonitrile 4-(6,7-dimethoxyquinolin-4-yl)sulfanyl-N-diazobenzenesulfonamide 4-(azidomethyl)-N,3-dimethoxyaniline 6-ethoxy-2-[(4-fluorophenyl)methyl]-5H-pyrazolo[1,5-b][2,3]benzodiazepine N-[1-[4-[2-[(6-methylpyridine-3-carbonyl)amino]ethyl]phenyl]cyclopropanecarboximidoyl]pyrimidine-5-carboxamide 6,7-dibromospiro[2H-furo[3,4-b]pyridine-3,1'-cyclopentane] 2-[(4R,5S)-2-benzylsulfanyl-4,5-diphenyl-4,5-dihydroimidazole-1-carbonyl]oxyethyl-trimethylazanium;chloride (2E)-2-[1-(3,4-dihydroquinoxalin-6-yl)-2-hydroxyethylidene]tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaen-6-ol N-[2,5-dioxo-4-(6-phenoxyhexanoyl)imidazolidin-1-yl]benzamide 6-(4-chlorophenyl)-N-(1H-pyrrolo[3,2-c]pyridin-5-ylmethyl)pyrazin-2-amine 1-[4-[[(E)-3-aminoprop-2-enyl]amino]butan-2-yl]pyrimidine-2,4-dione 2-bromo-5,6-dimethoxythieno[2,3-d]pyrimidine 4-[[4,5-bis(ethenyl)imidazol-1-yl]methyl]benzonitrile 4-N-[(E)-2-fluoroethenyl]-6-methyl-1,3,5-triazinane-2,4-diimine 3-(5,6-dihydro-1H-pyrrolo[2,3-b]pyridine-7-carbonyl)bicyclo[1.1.0]butane-1-carboxylic acid [4-[[7-[3-(dimethylamino)propoxy]quinolin-2-yl]amino]phenyl]azanide 3-(1H-indol-2-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 4-N,4-N-dimethyl-2-N-[5-(1H-pyrrol-3-yl)pyridin-3-yl]pyrimidine-2,4-diamine 6-cyclohexa-1,3-dien-1-yl-3-(5,6,7,8-tetrahydronaphthalen-2-yl)-4H-benzo[h]chromene N-[5-[4-[4-(1-cyclopentyloxyethenyl)piperidin-1-yl]phenyl]-3-[3-(dimethylaminosulfanyl)anilino]-2,6-naphthyridin-7-yl]cyclopropanecarboxamide (4R,5S)-3-[(2E,4E)-5-ethenylhexa-2,4-dienoyl]-4-methyl-5-(1-methylpyrrol-2-yl)-1,3-oxazolidin-2-one;N-methylformamide 3-[4-(4-chlorophenyl)phenyl]oxirane-2,2-dicarbonitrile 2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]cyclohexan-1-one N-methyliodanuidyl-2-phenylaniline N-[3-(3-fluorophenoxy)-4-methylphenyl]-2-methoxyethanesulfonamide 3,5-dimethylbenzamide;5-(4-methoxyphenyl)-1-[1-[2-(oxan-4-ylamino)ethyl]piperidin-4-yl]pyrrolidin-2-one 1-cyclopentyl-4-ethenylbenzene;3-methoxy-5-methylbenzoic acid (5Z)-2-(3,4-dichlorophenyl)imino-5-[(7-fluoro-1H-indol-3-yl)methylidene]-1,3-thiazolidin-4-one (4Z)-4-[(3,5-diethoxy-4-propoxyphenyl)methylidene]-2-methyl-1,3-oxazol-5-one 4-[1-(1H-imidazol-5-ylmethylamino)-2,3-dihydro-1H-inden-5-yl]benzoic acid [2-hydroxyimino-1-(9H-xanthen-9-yl)ethylidene]oxidanium 4-(2,3-dihydropyridine-5-carbonyl)-1H-pyrazole-5-carboxylic acid 1-(5-fluoro-2,3-dihydro-1-benzofuran-4-yl)-6-methoxy-N-[6-(4-methylpiperazine-1-carbonyl)pyridin-3-yl]-3H-indol-2-imine 4-(2-methoxyphenyl)sulfonyl-N-[(Z)-[4-(trifluoromethylsulfanyl)cyclohexa-1,3-dien-5-yn-1-yl]methylideneamino]piperazine-1-carboxamide N-(3-aminopropyl)-2-[(4-phenyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine-2-carbonyl)amino]butanamide N-[(2S)-1-[4-(2-aminoethylsulfanylmethyl)anilino]-3-methyl-1-oxobutan-2-yl]-4-fluorobenzamide N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-4-(2,5-difluorophenyl)pyrrolidine-2-carboxamide 1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonyl)piperidin-3-one 1-(3-azidopropyl)-4-[2-(3,4-dichlorophenyl)ethenoxy]piperidine 4-[2,5-dichloro-3-(methylideneamino)phenyl]sulfanylbenzonitrile N-[3,4-difluoro-2-(3-fluorophenyl)phenyl]-3,5-dimethylbenzamide;ethane 4-[3-methylbut-2-enyl(1,3-thiazol-5-yl)amino]benzenesulfonamide (4R)-1,2-diphenyl-3a,4-dihydrobenzimidazole N-[1-(2,4-difluorophenyl)ethyl]formamide;1-[2-(dimethylamino)pyridine-3-carbonyl]pyrrolidine-3-carboxamide N-(2,5-dichlorophenyl)-N-ethylsulfonylbutanamide 4-(1-aminoethyl)-2-ethyl-3,5-dihydroxybenzoic acid 2-(cyclopentylamino)-5,6,7,8-tetrahydro-3H-pyrido[4,3-d]pyrimidin-4-one 4-[(2E,3Z)-1-chloro-2-ethylidenehexa-3,5-dienyl]-7-methoxy-2,5-dihydro-1H-benzo[e]indole 2-(3-bromopropyl)benzene-1,3,5-tricarboxamide 2-[(4R,5S)-3-fluoro-7-methyl-6-oxo-1,3-diazonan-4-yl]isoindole-1,3-dione N-[3-(1,3-dioxolan-2-yl)phenyl]-1-methoxycyclobutane-1-carboxamide 3-ethyl-N,2-dimethyl-1-[4-(propan-2-ylideneamino)oxybutyl]pyrrolo[2,3-c]pyridin-7-amine 2-chloro-4-N,6-N-diphenylpyrimidine-4,6-diamine 2-[1-(2,4-difluorophenyl)ethylimino]imidazolidine-4,5-dione 4-[2-(azetidine-1-carbonyl)pyrrolidine-1-carbonyl]benzonitrile;5,6-difluoro-N'-hydroxypyrazine-2-carboximidamide 7-[1-(4-ethenylphenyl)but-3-yn-2-ylidene]cyclohepta-1,3,5-triene;(2Z)-N'-methyl-N-[1-(3-propan-2-ylphenoxy)butan-2-yl]penta-2,4-dienimidamide (2E,4Z)-1-[2-[3-[4-[[5-[(4R)-2,6-dioxopiperidin-1-yl]pentoxy]methyl]piperazine-1-carbonyl]phenoxy]ethylamino]hepta-2,4-diene-4-thiol;ethane 2-azido-3,4-dibromopyridine 2-azido-6,11-dihydrobenzo[c][1]benzoxepine (2S,4R)-N-[(3-fluorophenyl)methyl]-1-[6-(hydroxyamino)pyridine-2-carbonyl]-4-methoxypyrrolidine-2-carboxamide N-[4-(3,5-dichloropyridin-2-yl)oxyphenyl]-3-hydroxypropanamide 2-bromo-6,7-diethoxy-1H-quinolin-4-one (2R)-N-methyl-3-phenyl-1,4-dioxaspiro[4.5]decane-2-carboxamide 4-[(3R)-3-azidopyrrolidin-1-yl]sulfonylbenzonitrile 3-[4-(2,3-dihydroindol-1-yl)anilino]-1H-pyrazin-2-one 3-[2,4-bis(trifluoromethyl)phenyl]-5-methyl-1H-pyrazole 4-(benzenesulfinyl)-1,2,3,5,6,7-hexahydro-s-indacen-1-ol 2-chloro-5,6-dimethylquinoline-4-carboxylic acid 5-cyclopropyl-4,6-dihydrothieno[2,3-b]pyrrole-2-carboxamide [4-(2,3-dimethoxyphenyl)piperazin-1-yl]-[5-methylsulfonyl-2-(oxan-4-yl)phenyl]methanone N-[5-(2,3-dimethylimidazo[1,2-a]pyridine-7-carbonyl)-4-[(4-fluorophenyl)methoxy]-2-oxopentanoyl]-2-methylprop-2-enamide 2-[(4R)-2-[(3,5-dibromophenoxy)methyl]-8-oxo-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-N-propan-2-ylacetamide 3-(2,6-difluorophenyl)benzenecarboximidate 1-[4-(5,7-dichloro-2H-azepine-3-carbonyl)piperazin-1-yl]-2-(methylamino)ethanone 1-(4-fluorophenyl)sulfanylpyrrolidine;(3R,5R)-5-methoxy-N-[(4-oxo-3H-quinazolin-2-yl)methyl]piperidine-3-carboxamide 2-[4,5-bis(ethenyl)-3,6-dihydroxypyridin-2-yl]acetaldehyde 3-[4-(4,5-dimethylimidazol-1-yl)-1H-indol-2-yl]-5-pyridin-4-yl-1H-pyrazolo[4,3-b]pyridine N-(6-methoxypyridin-3-yl)-1H-indazole-4-carboxamide N-[(3,5-dimethylpyridin-2-yl)methylidene]benzamide (3-fluorophenyl)methyl-[6-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]carbamic acid 1-(2,2-difluoropropyl)indazole-3-carboxamide 2-[3-(4-fluorophenyl)sulfanylpropylamino]-8-methoxyquinazoline-7-carbonitrile 1-(azidomethoxy)naphthalene ethane;(3R)-1'-(2,5,7-trimethylquinolin-6-yl)spiro[1H-indole-3,4'-5,7-dihydropyrazolo[3,4-b]pyridine]-2,6'-dione N-(6-oxo-1H-pyrimidin-4-yl)-3,4-dihydro-2H-1,4-benzothiazine-7-carboxamide N-[2-(1,1,1,3,3,3-hexafluoropropan-2-yl)-6-methoxypyridin-4-yl]-5-[4-iodo-2-methyl-5-[[5-methyl-2-(trideuteriomethyl)pyrazol-3-yl]carbamoylamino]phenyl]furan-2-carboxamide N-[2-(4-aminophenyl)ethyl]-2-methyloxane-3-carboxamide 2-[6-(2-azidoethoxy)naphthalen-1-yl]acetic acid 1-[4-amino-2-(oxan-2-yl)pyrimidin-5-yl]ethanethiol 1-azido-2-(methoxymethyl)naphthalene 1-(4,6-dimethoxypyrimidin-2-yl)azepan-3-amine;hydrochloride 1-[2-azido-6-methyl-4-(trifluoromethoxy)phenyl]piperidine N-[(4-chlorophenyl)methyl]-1,4,2-trioxo-3-thiophen-2-yl-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxamide N-azido-6,7-dimethoxyquinazoline-2-carboxamide N'-hydroxy-2-[3-(methylsulfonylmethyl)phenoxy]pyridine-4-carboximidamide 4-methylsulfanyl-2-nitrobenzenesulfonic acid N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]-4-(4-methylphenyl)piperazine-1-carbothioamide 1-azidosulfanyl-2,3-dimethoxybenzimidazole [(1R,2S)-1-[4-chloro-5-fluoro-2-methyl-3-[[(2E,4Z)-6-(methylideneamino)hexa-2,4-dien-3-yl]carbamoyl]phenyl]-3-oxo-1-phenylbutan-2-yl]carbamic acid N-[3-chloro-4-[(1R,5S)-2-(2-fluorophenyl)-6-(trideuteriomethyl)-3-azabicyclo[3.1.0]hexan-3-yl]phenyl]benzamide 2-[(2-hydroxy-6-methylnaphthalen-1-yl)diazenyl]-4-methoxy-N,N-diphenylbenzamide 3-amino-N-[(1R)-2-oxo-1,3-dihydroimidazo[1,2-a]benzimidazol-1-yl]benzenesulfonamide N-[2-amino-1-(4-ethynylphenyl)ethyl]formamide;6-N,3,5-tribenzamidohexane-1,4,6-tricarboxamide (E)-1,2-difluorobut-2-ene;ethane;5-[3-methylpenta-1,3-dien-2-yloxymethyl(oxetan-3-yl)amino]-N-[(4-propan-2-ylphenyl)methyl]pentanamide 7-(1H-indole-2-carbonyl)-2,5,6,8-tetrahydroimidazo[1,2-a]pyrazin-3-one 2-[1-(4-chlorophenyl)ethyl]naphthalene 1-(4-chlorophenyl)-2,2-dimethylpentan-3-one 2-[3-(2,6-dimethylphenyl)-5-(3-hydroxypropylsulfanyl)-1H-pyrazol-4-yl]-N'-pyrimidin-2-ylpropanehydrazide 3-[[6-(4-fluorophenyl)sulfonylpyridine-2-carbonyl]amino]propanoic acid N-cyclohexyl-N-methyl-1,1-dioxo-3,4-dihydro-2H-thiochromene-7-sulfonamide 1-(4,5-diamino-2-chlorophenyl)ethanone 7-[(3S)-4,8b-dimethyl-1,2,3a,8b-tetrahydrocyclobuta[c]quinoline-3-carbonyl]-6,8-dimethoxy-2-phenylchromen-4-one 1-(azidooxymethyl)-3,4-dichloro-2-[(4-methoxyphenyl)methyl]benzene 5-chloro-1,3,3a,4,9,10,10a-octahydrophenanthro[9,10-d]imidazol-2-one;ethane 5-chloro-3-(2,6-difluorophenyl)imidazo[1,2-a]pyridine 3-[2-(4,6-dimethylcyclohexa-1,5-dien-1-yl)sulfonyloxyphenyl]-N-[2-(ethylideneamino)ethyl]propanamide (E)-1,2-difluorobut-2-ene;3-[4-[(2,6-difluorophenyl)methoxy]phenyl]-5-[3-[methyl(propanoyl)amino]phenyl]thiophene-2-carboxamide N-(4-chlorophenyl)-2,7-bis[(Z)-prop-1-enyl]-9H-fluoren-4-amine (4R,6S)-4,5,6-trimethyl-3-(2-propan-2-yloxypyrimidin-4-yl)-1,3-oxazinan-2-one 1-benzyl-5-(4,6-dihydropyrrolo[3,4-c]pyrazol-2-ylmethyl)triazolo[4,5-b]pyridine;2,2,2-trifluoroacetic acid [5-(1,3-benzothiazol-2-yl)-6-methoxypyridin-3-yl]-[4-[2-[4-(2-hydroxyethylamino)phenyl]hydrazinyl]piperidin-1-yl]methanone 5-[(6S)-7-[2-chloro-4-fluoro-3-[[[1-hydroxy-3,3-bis(methylamino)propylidene]amino]methyl]phenyl]-6-methyl-4,5-dihydrothiepin-3-yl]pyrimidine-2-carboxylic acid ethane;3-fluoro-4,5-bis(methoxycarbonyl)benzoate ethane;4-(5-fluoro-2,3,8,8a-tetrahydro-1H-indolizine-7-carbonyl)benzonitrile 3-(4,6-dimethylquinazolin-2-yl)sulfanylpropanenitrile (2R)-2-[amino-(5,6-dichloro-1H-benzimidazole-2-carbonyl)carbamoyl]oxyazetidine-1-carboxylate 2-amino-9-[(4S,5R)-3,3-dimethyl-1-phenyl-6-oxabicyclo[3.2.0]heptan-7-yl]-1H-purin-6-one N-[4,5-dibromo-2-(trifluoromethyl)phenyl]-2-hydroxyacetamide 2-chloro-N-methylsulfonyl-4-nitrobenzenecarboximidate 5-[3,4-dihydroxy-5-(2H-tetrazol-5-yl)phenyl]thiophene-3-carboxylic acid (5Z)-2-(4-bromophenyl)imino-5-[(1,5-dimethylpyrrol-3-yl)methylidene]-1,3-thiazolidin-4-one 7-(2,5-dihydropyrazin-1-ium-1-yl)thieno[3,2-c]quinoline 2-[4-[(1R)-1,7b-dimethyl-4aH-naphtho[2,1-b][1]benzofuran-10-yl]phenyl]pyridine [4-(6-phenylpyridazine-3-carbonyl)piperazin-1-yl]-pyrrolidin-2-ylmethanone 1-(5-nitrocyclohexa-2,4-dien-1-yl)-3-[(E)-3-phenylprop-1-enoxy]propan-1-ol 4-[2-(5,6-dihydroquinazolin-2-yl)but-3-yn-2-yl]morpholine 2-[8-(5-bromo-1,3-thiazol-2-yl)purin-9-id-9-yl]ethanol 2-[N-(benzenesulfonyl)-4-nitroanilino]benzoic acid 1-(3,4-dichlorophenyl)-2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethanesulfonate N-[3-(4,5-dihydropyrimidin-2-yl)phenyl]-7-methylpyrazolo[1,5-a]pyridine-3-carboxamide 2-[1-(5-fluoropyrimidine-4-carbonyl)piperidin-3-yl]-4-pyridin-2-yl-1H-pyrimidin-6-one 2-methylsulfanyl-7-(1H-pyrazol-5-yl)quinoline N-(2,3-dihydro-1H-benzimidazol-4-yl)propanamide (2R)-2,3-diamino-1-[4-(5-methoxypyridin-3-yl)piperazin-1-yl]propan-1-one;methoxyethane 3-[2-(4-chlorophenyl)-1,3-dioxolan-2-yl]phenol 1-cyclohexyl-6-[(3-ethoxyphenyl)methyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one 6,7-difluoro-2-(trifluoromethyl)quinoline-4-carboxylic acid (Z)-1,3-diamino-N'-[(3E)-6-fluorohexa-1,3,5-trien-3-yl]oxy-2-iminopropanimidamide;3-(dimethylsulfamoylamino)thiophene 3-[2,6-difluoro-4-(5-hexoxypyrimidin-1-ium-2-yl)phenyl]-1,8-difluoro-7-propoxyisoquinoline 2-[(3-cyclopentyloxyphenyl)methyl]propanedinitrile 1-(6-chloronaphthalen-2-yl)-3,4-dihydro-1H-isoquinoline (NE)-N-[1-(3,4-dichlorophenyl)-2,2,2-trifluoroethylidene]hydroxylamine 6-methoxy-1,7-dimethylindole 3-[5-[4-(trifluoromethyl)phenyl]thiophen-2-yl]-1,2-thiazole 5-[2-chloro-4-(trifluoromethoxy)phenyl]-3,6,6a,7,8,9,10,11,11a-octahydrobenzo[b][1,4]diazepin-6-one (7S)-6,8,9,10-tetrahydroxy-1H-naphtho[2,3-f]isochromene-2,7-dione 4-[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]benzaldehyde 5-bromo-N'-hydroxy-4-(pyrrolidine-1-carbonyl)pyridine-2-carboximidamide 1-[4,6-bis(ethenyl)pyridin-3-yl]ethenamine;ethane (2S)-2,3-bis[4-(diethylaminomethylideneamino)phenyl]propanoic acid 5-[2,3-dihydroxypropyl(prop-2-enyl)amino]naphthalene-2-sulfonic acid 4-azidooxy-3,7-dimethylpurine 4-methoxy-2-(pyrrolidin-1-ylmethyl)benzamide (3S)-2,6-diamino-5-methyl-N'-[2-oxo-1-[4-(trifluoromethylsulfanyl)phenyl]pyrimidin-4-yl]hexanediamide 5-(2,6-difluorophenyl)-1-[(4R,7S)-7-fluoro-3-methyl-10-oxa-2,13-diazatricyclo[12.4.0.02,6]octadeca-1(18),14,16-trien-12-yl]pentan-1-one 2-(4-chlorophenyl)sulfanyl-N'-hydroxypyridine-3-carboximidamide 2-[[3-chloro-5-(trifluoromethyl)phenyl]carbamoylamino]butanoic acid N-methyl-2-(3-nitrophenoxy)butanamide N'-[5-chloro-2-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)phenyl]methanimidamide 3-[(6-chloroimidazo[1,2-a]pyridine-7-carbonyl)amino]-2H-furan-5-carboxylate 3-[[5-chloro-6-(trifluoromethyl)pyridine-2-carbonyl]amino]piperidine-1-carboxylate 1-[3-(4-ethenyl-2,6-dimethoxyphenyl)propyl]piperidine 4-(1H-imidazol-5-ylmethyl)-2-[(Z)-(3-oxo-5-phenylsulfanyl-1,2-oxazol-4-ylidene)methyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione 3,5-dimethyl-7-(4,4,6,6-tetramethylcyclohexa-1,5-dien-1-yl)quinoline 1-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-(5-ethoxypyridin-2-yl)butane-1,4-dione;hydrochloride 1-cyclopropyloxy-4,5-difluoro-3-(2,3,6-trichlorophenyl)pyrazole 4-amino-2,6-dichloroquinazoline-7-carboxylic acid 5-azido-N-(cyclohexylmethyl)pyridin-3-amine 3-methyl-2-[[2-methyl-4-(piperidine-1-carbonyl)phenyl]carbamoylamino]pentanoic acid 5-N-[4-(azetidin-1-ylmethoxy)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)phenyl]-6-ethanimidoyl-3-N-methylpyridine-3,5-dicarboxamide 2-methoxy-1,2-bis(methylperoxy)-9H-fluorene [4-(dimethylamino)phenyl]sulfonyl-[1-(2,5-dimethylpyrazole-3-carbonyl)pyrrolidin-3-yl]carbamic acid 5-(3,4-difluorophenyl)-2-methyl-1H-pyrrole 2,4-dichloro-6-[(E)-methoxyiminomethyl]pyridine-3-carboxylic acid N-[(2S)-1-(dimethylamino)-3-phenylpropan-2-yl]sulfamate 6-N-[2-(4-aminoanilino)ethyl]-4,5-dimethyl-3H-2,1-benzoxazole-3,6-disulfonamide 2-[1-(3,4-difluorophenyl)sulfonylpyrrolidin-2-yl]-7-pyridin-3-yl-3H-imidazo[5,1-f][1,2,4]triazin-4-one 4-[[8-(1-cyclobutylpiperidine-3-carbonyl)-6,11-dihydrobenzo[c][1]benzoxepin-2-yl]oxymethyl]benzonitrile [3-(methoxyamino)phenyl]-[4-[1-(1,2,4-triazol-4-yl)propan-2-yloxy]piperidin-1-yl]methanone N-[1-(5,6-dichloro-3-ethylpyridine-2-carbonyl)piperidin-4-yl]acetamide N-(2,6-dichlorophenyl)formamide;N-[4-fluoro-3-(trifluoromethyl)phenyl]formamide N-[1-amino-2-[4-(trifluoromethyl)pyrimidin-2-yl]ethylidene]acetamide;1,3-diaminocyclobutane-1-carbonitrile 1-[4-(azidooxymethyl)phenyl]piperidine 1-[(4aR,8aS)-3-oxo-4a-(pyrrolidine-1-carbonyl)-4H-quinoxalin-2-yl]-N-(furan-2-ylmethyl)piperidine-4-carboxamide 5-[(2R,6S)-2-methyl-6-phenylmorpholine-4-carbonyl]-1H-pyrimidine-2,4-dione 5-amino-4-(4-methoxyanilino)-1H-pyrimidin-6-one 4-(2-methylpyridin-3-yl)-6,7,8a,9,10,11,12b-octahydrobenzo[a]quinolizin-1-amine N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-(furan-2-yl)pyrazol-3-yl]-2-thiophen-2-ylacetamide 2-bromo-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine;5,6-dimethoxy-2-(4-pentan-3-ylphenyl)-1H-benzimidazole 2-(4,5-dimethyl-3,6-dihydro-2H-pyridine-1-carbonyl)indene-1,3-dione 2-[1-(6,7,8,9,10,11-hexahydrocycloocta[b]indole-5-carbonyl)piperidin-4-yl]oxyacetic acid N-[4-[2-(4,5-dichlorocyclohexa-1,3-dien-1-yl)ethoxy]phenyl]quinoline-8-carboxamide 1-(6,11-dihydrobenzo[c][1]benzoxepin-11-yl)piperidine (Z)-3-[4-[(E)-2-(1H-indazol-6-yl)ethenyl]phenyl]but-2-en-2-amine 2-(1H-indazol-6-ylmethylamino)-4,5,6,7-tetrahydroisoindole-1,3-dione N-[4-methyl-5-oxo-2,3-bis(sulfanyl)imidazolidin-1-yl]-3-phenylbenzamide 1-azido-4-[2,3-bis(trifluoromethyl)phenyl]piperazine 2-azidooxy-4,5-dinitrobenzenesulfonic acid 2-hydroxyimino-3-oxo-3-[4-(trifluoromethyl)phenyl]propanoate 3-(3,5-dichloro-4-hydroxyphenyl)-1H-pyrazole-5-carboxylic acid 2-[1-(3,4-dimethoxyphenyl)-5-[3-[4-(dipropylcarbamoylamino)phenyl]-2H-furo[3,2-b]pyridin-6-yl]pyrrol-2-yl]acetamide N-(4-aminophenyl)-2-[3-chloro-6-ethyl-5-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-9-oxoacridin-10-yl]acetamide 2-methyl-5-(6-piperazin-1-ylpyridin-3-yl)oxybenzamide (E)-N-[4-(4-methoxyphenyl)piperazin-1-yl]-2-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]but-2-enamide N-[(3,4-dichlorophenyl)methyl]-9-methyl-2-(1H-pyrazolo[3,4-b]pyridin-4-ylamino)purine-8-carboxamide (3R)-6,6-dimethyl-4-pyridin-2-ylhexan-1-ol 2-tert-butyl-1'-[(6-chloropyridin-3-yl)methyl]spiro[5,6-dihydrocyclopenta[d]pyrimidine-7,4'-piperidine];formic acid 1-[2,6-di(propan-2-yl)phenyl]-3-[(E)-(2-hydroxynaphthalen-1-yl)methylideneamino]thiourea 3-[4-methyl-6-oxo-2-(1,3-thiazol-2-yl)-1H-pyrimidin-5-yl]propanoic acid [4-(azidomethyl)piperidin-1-yl]-[5-chloro-6-[3-[3,5-difluoro-4-[(2S)-3-hydroxy-2-methoxypropoxy]phenyl]butanoylamino]pyrimidin-4-yl]methanone 4-[1-[5-(dimethylamino)naphthalene-2-carbonyl]-3,6-dihydro-2H-pyridin-4-yl]butanoic acid 2-methylpropan-1-ol;N-[3-(trifluoromethoxy)phenyl]oxane-4-carboxamide (5S)-5-[(2,4-dichlorophenyl)methyl]-2-(furan-2-ylmethylidenehydrazinylidene)-1,3-thiazolidin-4-one 2-[3-(1H-benzimidazol-2-ylmethyl)-4,5,6,7-tetrahydroindazol-2-yl]acetamide 4-[(2Z,5E)-6,7,8,10-tetrahydroazecine-3-carbonyl]benzonitrile 1-[(2,6-difluorophenyl)methyl]-4-fluoroindazole 2-[(1-aminocyclopropyl)methoxy]-N'-hydroxypyridine-4-carboximidamide 1,2-difluoro-4-(3-methylbutan-2-yl)benzene 4-[3,5-bis(trifluoromethyl)phenyl]-1-ethylpiperidine 1-[4-bromo-5-fluoro-2,6-di(propan-2-yl)pyrimidin-1-ium-1-yl]piperidine N-[2,4-difluoro-3-(4-pyridin-4-ylpyrazole-1-carbonyl)phenyl]-2-fluorobenzenesulfonamide 7-fluoro-3-(2-thiophen-2-ylpyrrolidine-1-carbonyl)chromen-2-one 2-[[2,5-dichloro-4-(1H-indole-6-carbonyl)phenyl]methyl]propanedioate 1-(2,3-dihydropyridine-5-carbonyl)-4-phenylpiperidine-4-carbonitrile 2-[4-(3-bromopropoxy)phenyl]pyridine 2-chloro-N-[(3S)-1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl]-5-methanimidoylpyrimidine-4-carboxamide 2-[2-chloro-5-(methylideneamino)-N'-(1,3-thiazol-4-ylmethyl)anilino]acetic acid 1-[4-(cyclopenten-1-yl)piperidine-1-carbonyl]pyrazole-3-carboxylic acid N-[(2R)-4,5-dihydroxy-6-methyl-3-nitrosohexan-2-yl]-8-fluoro-7-methoxyquinoline-2-carboxamide 6-amino-4-(5-cyano-1H-indol-3-yl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 3-[4-(1H-imidazol-5-ylmethoxy)phenyl]-5-[5-(2-phenylethynyl)thiophen-3-yl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one 4-[6-[2-(dimethylamino)ethoxy]pyridin-3-yl]benzaldehyde 2-N-(4-azidopiperidin-1-yl)-1,3,5-triazine-2,4-diamine N-[2-[4-(3,4-difluorophenyl)piperazin-1-yl]ethylsulfanylmethyl]quinoline-8-carboxamide;propane [5-amino-1-(3-methoxy-4-morpholin-4-ylphenyl)pyrazol-4-yl]-[6-chloro-5-(2,2-difluoroethoxy)-1H-inden-2-yl]methanone 2-cyclohexyl-1H-quinoline 2-(azidomethyl)-5,6,7,8-tetrahydronaphthalene 3-chloro-4-hydroxybenzaldehyde;2,5-dimethylbenzonitrile;7-(3-pyrrolidin-1-ylpropoxy)spiro[3,5-dihydrochromene-2,4'-piperidine] N-[3,4-dimethyl-5-(2-nitrophenyl)-1H-pyrrol-2-yl]pyrimidine-4-carboxamide 2-(4-azidophenyl)-6,7,8,9-tetrahydro-5H-carbazole 1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]sulfinyl-N-pyridin-2-ylpiperidine-4-carboxamide 4-(2,6-dihydroxyphenyl)-3-[2-methyl-5-[(E)-2-(6-methylpyridin-2-yl)ethenyl]anilino]sulfanylbenzoic acid N-butanoyl-4,5-dichloropyridine-2-sulfonamide 2-N,6-N-dicyclopropylpyrimidine-2,4,6-triamine 4-[3-(diethylamino)propyl]thiophene-2-sulfonamide N-(4,5-dimethylpyrimidin-2-yl)-4-[ethylsulfonyl(pyridin-3-yl)amino]benzenesulfonamide 3-[1-(1H-benzimidazol-2-yl)ethyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine 5-bromo-2-(8-methylnonan-5-ylideneamino)benzonitrile 1-[3-(2,4-dimethylphenoxy)propyl]-4-(pyridine-2-carbonyl)piperazin-2-one N-[2-(3,4-dimethoxyphenyl)ethyl]-5-hydroxy-6H-benzo[c]chromene-8-sulfonamide 2-methyl-6-[5,5,7,7-tetrafluoro-4-(trifluoromethyl)heptanoyl]pyridazin-3-one 4-methyl-7,8-dihydropurino[9,8-a]pyridine 2-(4-methylpiperidine-1-carbonyl)benzohydrazide 6-(5-fluoropyridin-3-yl)-2,7-dimethoxynaphthalen-1-amine 6-[(3,5-dichlorophenyl)methyl]-2-propan-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-[(3-chloropyridin-2-yl)methylamino]-1H-pyrimidin-6-one 2-bromo-1-[4-[[1,3-di(ethyl)pyrazol-4-yl]methyl]-6-oxo-3,7,11-trithiatricyclo[6.3.0.02,6]undeca-1(8),2(6),4,9-tetraen-5-yl]ethanesulfonic acid 4-[4-(5-chloropyridin-2-yl)phenyl]sulfonylmorpholine 2-[5,6-dimethoxy-7-(1H-pyrazol-4-yl)-1H-indole-3-carbonyl]propanedinitrile (3S)-5,7-dimethyl-1'-(quinoline-2-carbonyl)spiro[1H-indole-3,4'-5,8-dihydropyrazolo[4,3-g]quinazoline]-2,6'-dione 2-amino-N'-[(3E)-2-methylhexa-1,3,5-trien-3-yl]pyridine-4-carboximidamide 6-amino-2,4-bis(5-methylhexan-3-yl)-1H-pyrimidine-2,5-diol 5-methyl-N-[4-(oxan-2-yl)pyrimidin-2-yl]thieno[2,3-d]pyrimidine-6-carboxamide 6,7-dibromo-4-(cyclopropanecarbonyl)-3-[2-ethoxy-5-[(Z)-(4-hydroxyphenyl)methylideneamino]phenyl]sulfonyl-1H-quinoxaline-2-thione N-[(1S)-2-hydroxycyclohexyl]-7-(methylamino)-5-[(2R,3R)-3-methyl-4-(6-methylpyridine-3-carbonyl)morpholin-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 1-azidooxy-2,3-dimethyl-5-phenoxybenzene N-(1-cyanobutan-2-yl)benzamide N-cyclopentyl-2-[3-(1,5-dimethylpyrazol-4-yl)propanoyl]-2-azaspiro[4.4]nonane-4-carboxamide 3-[4-[2-fluoro-5-(trifluoromethyl)phenoxy]phenyl]-N-hydrazinylidenepropanimidamide N-[4-amino-3,5-bis(trifluoromethyl)phenyl]-3-[2-chloroethyl(propanoyl)amino]piperidine-1-carboxamide 3,6-dimethyl-5-(2-phenylethoxy)pyrimidin-4-one 1,3-diphenylpropylazanide 3-[(1R)-3,4,6-trihydroxy-2-methylcyclohex-3-en-1-yl]benzene-1,2-diol 5-[3-azido-2,6-difluoro-4-(methanesulfonamido)phenyl]-N-benzylpyridine-2-carboxamide 4-(8,14-dioxapentacyclo[11.7.0.02,10.03,8.015,20]icosa-1(13),2(10),3(8),4,6,11,15,17,19-nonaen-9-ylmethoxy)aniline 3-chloro-N-methyl-4-[(2S)-pyrrolidine-2-carbonyl]benzenesulfonamide 1-[2,4-bis(trifluoromethyl)phenyl]-3-[4-methanimidoyl-5-(4-piperidin-1-ylanilino)pyridin-2-yl]urea 6-(2-tert-butylphenyl)-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione N-[3-ethylsulfonyl-4-(1,2,3,6-tetrahydropyrazin-4-ium-5-yl)phenyl]-5-(trifluoromethyl)pyridine-2-carboxamide N-[4,6-di(propan-2-yl)pyridin-3-yl]-2,7-bis(ethenyl)-1,5,10-triazatricyclo[7.3.0.03,7]dodeca-9,11-diene-12-carboxamide 5-(3,4-difluorophenyl)sulfanyl-2H-triazole 3,4,5-trichloro-1-(3-ethenylnaphthalen-2-yl)-6-methoxybenzimidazol-2-one N-[(2S)-4,4-difluoropyrrolidin-2-yl]-3-fluoro-4-hydroxybenzamide;hydrochloride N-[4-(2,2,3,3a,5,6,7,7a-octahydroindol-1-yl)phenyl]-4-chlorobenzenesulfonamide 2-bromo-N-(4-hydroxybutyl)-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]benzamide 3-hydroxy-2,4-di(piperazin-1-yl)benzaldehyde N-[1-azido-2-[4-(difluoromethoxy)phenyl]ethyl]-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine [2-(4-tert-butylcyclohexen-1-yl)pyridin-4-yl]methanimine 3-chloro-4-[1,2-dihydroxypropyl(methoxycarbonyl)amino]benzoic acid 5-cyclopropyl-N'-(2-methoxyethylsulfonyl)-3-propan-2-yloxypyridine-2-carboximidamide 2-cyclopropyloxy-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]benzamide [(2S,4S)-1-acetyl-4-methoxypyrrolidin-2-yl]-piperazin-1-ylmethanone;2-bromopyridine N-[4,6-bis(sulfanyl)pyrimidin-2-yl]acetamide 2-(4-chlorophenyl)-1,1-dioxo-5H-[1,3]thiazolo[5,4-d]pyrimidine 2-(4-bromophenyl)-N,1-dimethylpiperidine-3-carboxamide 3-[5-(1H-benzimidazol-2-yl)thiophen-2-yl]-4-(3,5-difluorophenyl)pyridin-2-amine N-(2,5-dichlorophenyl)-N-prop-2-enylethanesulfonamide N-cyclobutyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide 6-[(3R)-4-[2-fluoro-5-(6-methoxy-1,3-benzothiazol-2-yl)phenyl]-3-(hydroxymethyl)piperazine-1-carbonyl]pyridine-3-carbonitrile 1-[2-[4-(3-chlorophenyl)piperidine-1-carbonyl]morpholin-4-yl]ethanone N-[(E)-3-methoxybut-1-enyl]-5,6-dihydronaphthalene-2-carboxamide N-methyl-1'-[6-(4-methylpiperazin-1-yl)pyridine-3-carbonyl]spiro[5,6-dihydroimidazo[2,1-c][1,4]oxazine-8,4'-piperidine]-6-carboxamide;2,2,2-trifluoroacetic acid N-[4,5-bis(methoxymethyl)-1H-pyrazol-3-yl]-2-pyrimidin-5-ylacetamide N-[2-(dimethylamino)ethyl]-3-pyridin-4-yl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carboxamide 3-(N-[2-(1H-indol-3-yl)ethyl]anilino)butanoic acid 2-amino-4-(4-fluoro-3,5-dimethylphenyl)-6-[2-oxo-1-[4-(2,2,2-trifluoroethoxymethyl)cyclohexyl]piperidin-3-yl]pyridine-3-carbonitrile N-[(1R,2S)-2-hydroxycyclopentyl]-3-iodopyridine-4-carboxamide [2-methyl-1-oxo-3-[(Z)-2,3,6,7-tetrafluorohept-2-en-4-ylidene]inden-5-yl]boronic acid [3-(3,5-dimethoxyphenyl)piperidin-1-yl]-(2H-triazolo[4,5-b]pyridin-7-yl)methanone 2-[(1R,3S)-3-ethyl-5-methoxycyclohexyl]ethynylbenzene 1-[(Z)-ethylideneamino]-N',2-dimethylindole-3-carboximidamide 1-[(2,6-dichlorophenyl)methyl]-4-(2-fluorophenyl)benzene 4-[(2R)-3-(3,5-difluorophenyl)-4,4,4-trifluoro-1-phenylbutan-2-yl]benzenesulfonic acid 3-[2-(1,4-dioxan-2-yl)ethoxy]-N'-hydroxypyridine-2-carboximidamide (2R)-3-(diphenylphosphorylmethoxy)butan-2-ol N-[6-methyl-2-(4-propan-2-ylpiperazine-1-carbonyl)pyrimidin-4-yl]acetamide [2-amino-4-oxo-5-(pyridine-3-carboximidoyl)-1,6-dihydropyrimidin-7-yl]methylideneazanium (2E)-1,3-diamino-N'-(naphthalene-1-carbonyl)penta-2,4-dienediamide;ethane 5-tert-butyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,2]oxazepine 2-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-prop-2-enylamino]decanoic acid 2-[(4-chlorophenyl)methylamino]pyridine-3-carboxylate N-(3-methylsulfonyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl)-1H-pyrazole-4-carboxamide 2-(3,5-ditert-butyl-4-hydroxyphenyl)ethanimidate 2,4-diethoxy-N-[6-[1-(3-phenylpropyl)piperidin-4-yl]pyridin-2-yl]benzamide 1-(4-azidooxybutylsulfonyl)-2,3,6,7-tetrachloronaphthalene 1-[6-[3-(3-aminopropanoyl)indol-1-yl]-2,3-dihydroindol-1-yl]ethanone 4-hydroxy-3,5-dimethylsulfonyl-N-propan-2-ylbenzamide 2-(azidomethyl)benzo[g][1,3]benzoxazole 1-(1,2-diphenylpropyl)naphthalene N-[2-(5,6-dihydronaphthalen-1-yl)ethyl]-3-fluoroaniline (1R,2S)-3-methylsulfonyl-1,2,4a,5,6,7,8,9-octahydronaphthalene-2-carboxamide 2-[2,5-difluoro-4-(4-pentylcyclohexyl)phenyl]-6-ethoxy-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 2,6-dichloro-N-[(5E)-3,4-dihydro-1H-diazocin-2-yl]aniline 4-bromo-5-[2-(diethylamino)ethoxy]-1,3-dimethylimidazol-2-one 3-(2,5-dimethylpyrazol-3-yl)-5-[(2E,4Z)-hexa-2,4-dien-3-yl]-1H-pyrazolo[4,3-b]pyridine [(3S,5R)-1-[2-[[3-acetamido-6-ethyl-8-[(4-fluorophenyl)methylamino]-7H-pyrrolo[2,3-c]azocin-9-yl]amino]-2-oxoethyl]-2-oxopyrrolidin-3-yl]carbamic acid 3-[5-bromo-2-hydroxy-1-(2-phenylethyl)indol-3-yl]imino-N,2-dimethylindole-6-carboxamide (5S)-2,4-dimethyl-5-(phenylsulfanylmethyl)-1H-imidazole N-(4-azidophenyl)benzenesulfonamide 1-[1,2-bis(methoxymethyl)anthracen-9-yl]oxypropan-2-ol N-(5-methylpyridin-3-yl)-4-[4-[[1-(oxetan-3-yl)piperidin-4-yl]methoxy]phenyl]-1,3-thiazol-2-amine 2-(3-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 5-(4-chlorophenyl)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]-2,5-dihydro-1H-2-benzoxepine 1,4-dihydroxynaphthalene-2,3-disulfonic acid 4-chloro-3,5-dimethyl-N-[(2E)-penta-2,4-dien-2-yl]benzamide 3-(1-benzofuran-2-yl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole N-[3-[(6Z)-6-[(4-methoxy-2,5-dimethylphenyl)methylidene]-7H-purin-8-ium-2-yl]phenyl]cyclopropanesulfonamide 3,5-dichloro-N'-[4-(N-methylanilino)cyclohexyl]benzohydrazide N-(2,3-dihydrofuro[2,3-b]pyridin-5-ylmethyl)-1-propan-2-yl-4H-pyridazine-6-carboxamide 3-(1-methylimidazol-2-yl)-4H-pyrido[1,2-a]pyrimidine 3-[(4-chlorophenyl)methyl]-2-(2-cyclohexa-1,5-dien-1-ylethenyl)-5-methoxyquinoxaline N-[2-(1H-indol-3-yl)ethyl]-4-nitro-N-octylbenzamide 2,2-dichloro-N-(4-chloro-3-pyridin-2-ylphenyl)cyclopropane-1-carboxamide N-[1-(2,3-dimethylanilino)-1-oxo-3-phenylpropan-2-yl]-N-[4-[2-(dipropylamino)ethoxy]-3-fluorophenyl]benzamide [(1R,2S)-5-oxo-2-phenylcyclohexyl]methylazanide [1-(2,4-dimethylphenyl)cyclopropyl]-(3-pyridin-4-ylpiperazin-1-yl)methanone N-[1-(3,5-dichlorophenyl)-2-imidazol-1-ylethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 4-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]benzoic acid (2R)-2,4-bis[(4-fluorophenyl)methoxy]pentanal;methylsulfane 5-methyl-6,7,8,9-tetrahydroimidazo[1,2-a][1,3]diazepine;(Z)-pent-2-ene 5-[4-(5,6-dimethoxypyridin-3-yl)phenyl]-2-methylidenepentanoic acid 4-[3,5-bis(2,6-dimethylpyridine-4-carbonyl)phenyl]-1H-indazole-3-carbonitrile N-[(2R)-4,6-diaminohexan-2-yl]-5-fluoropyridine-3-carboxamide 2-[4-[3,3a-dihydro-1H-pyrrolo[2,3-b]pyridine-5-carbonyl(methyl)amino]phenyl]acetic acid 2-(1H-indol-6-yl)benzo[g]isoquinoline 2-(7-chloro-9H-pyrido[3,4-b]indol-1-yl)acetic acid;hydrochloride 4-[N-(benzenesulfonyl)-2,5-dichloroanilino]benzoic acid 1-(7,8-dimethyl-5H-[1]benzofuro[3,2-b]pyridin-9-ium-2-yl)-N-phenylazethenamine 6-[(5-amino-3-methylcyclohepta-1,4,6-trien-1-yl)oxy]-2-tert-butylpyridine-3-carboxylic acid N-[(3R)-1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-3-yl]-6-fluoro-5-methoxypyridine-3-carboxamide 6-fluoro-5,8-dimethyl-N-(3-methylphenyl)-[1]benzothiolo[2,3-d]pyrimidin-4-amine 1-amino-N',2-dimethylbutane;6-chloro-5-(4,6-dichloropyridin-3-yl)pyridine-2-carboximidamide N'-(2,6-dimethylphenyl)-1H-pyrrolo[3,2-b]pyridine-7-carboximidamide (2S,3R)-4-cyclopropyloxy-N-(2-methoxyethylsulfonyl)-1,2,3,5-tetrahydro-1,4-benzodiazepine-3-carboxamide 1-[(4aR)-8a-ethyl-3,5,6,8-tetrahydro-2H-pyrano[3,2-b]pyrrol-1-yl]-2-(4-pyrazol-1-ylphenyl)ethanone N-(1H-imidazol-2-ylmethoxy)naphthalene-1-carboxamide 3-azido-N,N-dimethyl-2-propan-2-ylidenebutanethioamide 1,2-dihydroxyxanthen-9-one [4-(2,6-dimethoxyphenyl)thiophene-3-carbonyl]carbamic acid 2,5-dichloro-N-(3-morpholin-4-ylpropyl)-N-octylaniline N-[2,6-dimethyl-4-(4-sulfamoylphenyl)-3H-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]ethanone;ethane 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]pyrimidine 5-(2,3,4-triethoxyphenyl)imidazolidine-2,4-dione N-[1,2-dihydropyrimidin-6-yl(phenyl)methyl]ethanimine;fluorobenzene N-(7,8-difluoro-5-methyl-1-oxo-2H-isoquinolin-3-yl)pyrazine-2-carboxamide 2-[(E)-3-(4,6-dimethoxycyclohexa-1,5-dien-1-yl)prop-2-enoyl]chromene-4-thione (2S)-1-[3-(tert-butylcarbamoylamino)azetidine-1-carbonyl]oxy-3,4,6-trimethyl-2H-pyridine-2-carboxylic acid (7S)-3-benzylsulfanyl-5-methylidene-4,6,7,8-tetrahydrothieno[2,3-c]azepine 3-N-[(Z)-2,5-dihydroxyhex-3-enyl]-1-N-methyl-4-methylidenepyrrolo[2,3-c]pyridine-1,3-dicarboxamide N-[3,5-dimethyl-2-(4-methylanilino)phenyl]ethanesulfonamide 3-chloro-4-methoxyiminocyclohexa-1,5-diene-1-carbonitrile;4-fluorobenzaldehyde N-(2-aminoethyl)-1-[1-[6-(4-chloro-3,5-dimethoxyphenyl)thieno[3,2-d]pyrimidin-4-yl]piperidin-4-yl]formamide (2R,3R)-4,4-bis(phenylmethoxy)-5-[(E)-3-phenylprop-2-enoxy]pentane-1,2,3-triol (4Z)-5,6-dimethylhepta-1,4,6-trien-3-amine;ethane;7-fluoro-2-[4-(trifluoromethyl)phenyl]isoquinolin-1-one (2R)-3,4,7-trimethylsulfanyl-1-[(Z)-propylideneamino]-2H-pyrimido[5,4-e][1,3]oxazin-6-one 3-bromo-1-(2,4-difluorophenyl)-5-iodopyridin-4-one 2-(3,4-dichlorophenyl)-1-[2-[methyl-[(1S)-1-piperidin-4-ylethyl]amino]pyrimidin-5-yl]butan-1-one 6-N,2-diethyl-4-N-(3H-imidazo[1,5-a]pyridin-4-ium-8-yl)pyrimidine-4,6-diamine [4-(4-ethylphenyl)piperidin-1-yl]-(2,3,6-trifluorophenyl)methanone (3S)-1-[2,4-dichloro-6-[methyl-[1-[(3S)-pyrrolidin-3-yl]piperidin-4-yl]amino]pyrimidin-5-yl]sulfonylpyrrolidine-3-carboxylic acid 2-[[5,7-dichloro-6-(2H-tetrazol-5-yl)isoquinolin-3-yl]carbamoylamino]-4-fluorobenzamide (5Z)-2-[5-[[1-(4-bromophenyl)-3,5-dimethylpyrazol-4-yl]methylideneamino]pyridin-2-yl]imino-5-[(E)-4-hydroxybut-2-enylidene]-1,3-thiazolidin-4-one 1,2-diamino-4-(3,5-dibromophenyl)-6-oxopyridine-3,5-dicarbonitrile 2-[3-(methoxyamino)phenyl]benzenesulfonic acid N-methyl-6,7-diphenyldibenzofuran-3-amine 3-butan-2-yloxy-N'-hydroxybenzenecarboximidamide 2-[1-amino-2-(3-bromophenyl)ethyl]phenol 4-[8-amino-3-(1-oxo-2,9a-dihydro-6H-pyrazino[1,2-b]pyridazin-7-yl)imidazo[1,5-a]pyrazin-1-yl]-N-ethylbenzamide (2R,3S)-2-N-[1-[[5-chloro-4-(6-pyrrolidin-1-ylpyridin-3-yl)thiophen-2-yl]methylamino]ethenyl]butane-2,3-diamine 4-[4-(1,3-benzodioxol-5-yl)phenyl]benzamide N-[4-(benzylamino)phenyl]-1-azidopiperidine-3-carboxamide 3-[(4-tert-butylphenyl)methoxy]-N'-hydroxypyrazine-2-carboximidamide [3-(3,5-ditert-butylphenyl)-2,4-bis(methoxycarbonyl)benzoyl]azanium N-[(E)-(2,4-dihydroxyphenyl)methylideneamino]-3-methoxybenzamide 4-[2-azidooxy-6-[(3,5-dichlorophenyl)methylsulfanyl]pyrimidin-4-yl]morpholine 2,5-dibromo-N-(4-chlorobutyl)-N-(4-nitrobenzoyl)benzamide 1-(6,7-dimethoxyquinolin-4-yl)-3-[5-propan-2-yl-1-(2,2,2-trifluoroethyl)pyrazol-3-yl]urea 1-amino-4-(2,3-dimethylanilino)anthracene-9,10-dione (2S)-N'-(3,5-dimethylphenyl)sulfonyl-4-ethoxy-1,2-dimethylpyrrolidine-2-carbohydrazide 3-[(4,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)amino]-4-propanoyloxybutanoic acid 1-[(2R)-4,4-difluoro-2-[3-methyl-6-(trifluoromethoxy)indole-1-carbonyl]pyrrolidin-1-yl]prop-2-en-1-one 2-amino-4,6-dimethylbenzenesulfonic acid N-[5-(4-methylpentanoyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]cyclopropanecarboxamide 4-fluoro-3-[7-(5-methylthiophen-2-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-pyrimidin-5-yl-1H-pyrazolo[3,4-c]pyridine N-[(1R)-2-methoxy-3-oxocyclopentyl]-5-[2-propan-2-yl-6-(trifluoromethyl)pyridin-4-yl]naphthalene-2-carboxamide 3-(2,4-dichlorophenyl)sulfonylpyrrolidine;ethane 4-benzyl-1,3-diphenylpiperazine-2,5-dione 3-[4-(5,6-dihydronaphthalene-1-carbonyl)phenyl]propanoic acid (5E)-2-(4-bromo-3,5-dimethylphenyl)imino-5-[(1R)-1-(2,3,4-trichlorophenyl)ethoxy]imino-1,3-thiazolidin-4-one N-(4-nitrophenyl)-4-oxo-2-propanoyl-1,3-oxazolidine-3-carboxamide 1-[5-chloro-2,3-diethyl-4-(5-fluoro-6-oxo-1H-pyridine-3-carbonyl)phenyl]-3-[2-fluoro-4-(trifluoromethoxy)phenyl]urea 4-[4-(6-methylcyclohexa-2,4-dien-1-yl)sulfonylpiperazin-1-yl]aniline 4-amino-N-[2-[[6-(4-methyl-3,5-dihydropyrazole-1-carbonyl)pyridin-3-yl]oxymethyl]phenyl]thieno[3,2-d]pyrimidine-7-carboxamide N-[(1R,2S)-2-(dimethylamino)cyclopentyl]-4-nitro-5-pyrrolidin-1-yl-6H-cyclopenta[d]pyrimidin-7-amine 2-(2-aminoanilino)-1,3-dihydroindene-5-carboxylic acid;dihydrochloride 3-(azidomethyl)-5-phenylmethoxy-1H-indole 5-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N-[(3R,4S)-4-fluoropyrrolidin-3-yl]pyridine-2-carboxamide 1-(2,4-dimethylphenyl)-N-[4-[(6,7-dimethylquinazolin-4-yl)amino]butyl]triazole-4-carboxamide 3-[4-(2-bromoethoxy)phenyl]-1H-pyrrolo[2,3-c]pyridine 3-amino-1-(2-cyanopyridin-4-yl)piperidine-3-carboxamide;4-[cyclopropylmethoxy-[4-(1,3-oxazol-5-yl)phenyl]methyl]morpholine [4-(2,3,5,6-tetradeuteriopyridine-4-carbonyl)piperazin-1-yl]methanol 3-chloro-N-(2,4-dioxospiro[1H-quinoline-3,4'-piperidine]-6-yl)benzamide 5-[(E)-[3-methyl-1-(4-phenoxybenzoyl)piperidin-4-ylidene]methoxy]pyridine-2-carboxamide N-[4-(cyclopropylmethoxy)phenyl]oxazinane-2-carboxamide 5-[5-azidooxy-4-chloro-2-(difluoromethyl)pyrazol-3-yl]-1H-imidazole 6,7-dimethoxy-4-[4-(morpholine-4-carbonyl)piperazin-1-yl]-N-pyridin-3-ylquinoline-2-carboxamide;hydrochloride 2-ethyl-1-[4-(1H-pyrazole-5-carbonylamino)phenyl]cyclopropane-1-carboxylic acid (6R)-6-(2,4-dimethoxyphenyl)-3-propanoylsulfanyl-7-pyridin-1-ium-1-yl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one [3-ethylsulfonyloxy-5,6-difluoro-1-(4-fluorophenyl)indol-2-yl]boronic acid ethane;1-methyl-2-[3-(4-methylphenyl)propyl]benzene 3-[(2E)-2-[(4-hydroxyphenyl)methylidene]hydrazinyl]benzoic acid (2R,4S)-1-[2-[3-(2,6-dimethoxyphenyl)propyl]-3H-pyrrole-5-carbonyl]-4-fluoropyrrolidine-2-carboxylic acid N-cyclohexyl-6-ethyl-4,5-dihydrothieno[2,3-d][1]benzazepine-2-carboxamide 1-azidooxy-2,4-ditert-butylbenzene N-[5-(2,3-difluorophenyl)sulfinyl-1H-indazol-3-yl]-4-[4-[4-(3-pyrrolidin-1-ylpropanoyl)piperazin-1-yl]piperidin-1-yl]benzamide 4-[N-(2,3-dihydroxypropyl)-2-methoxyanilino]-2-nitrophenol 4-(1,3-benzothiazol-2-yl)-N-benzyl-5-methoxy-N-[2-oxo-2-(propan-2-ylamino)ethyl]thiophene-3-carboxamide;ethane 4-(3,5-dimethylphenyl)sulfonylmorpholine 3-methyl-4-[2-oxo-2-(6-pyrrolidin-1-ylpurin-9-yl)ethoxy]benzaldehyde 1-(3-azidophenyl)-2,4-dimethyl-5-pyridin-2-yl-6-thiophen-2-ylbenzimidazole 2-(3,6-dimethylcarbazol-9-yl)-4-N-[4-(5-pyrrolidin-1-ylpentoxy)phenyl]pyrimidine-4,6-diamine 1-[6,8-bis(ethenyl)-2-phenyl-5H-pyrido[4,3-d]pyrimidine-7-carbonyl]pyrrolidine-3-carboxamide 7-fluoro-8-methyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxylic acid 4-(3,5-dihydroxyphenyl)benzamide [4-(2,5-dimethylphenyl)piperazin-1-yl]-(7H-purin-6-ylamino)methanol 1-[4-(5,7-dihydropyrrolo[3,4-b]pyridin-6-ylsulfonyl)phenyl]ethanone 1-(4-bromobutoxy)-6,7-difluoronaphthalene 3-(3,6-dihydro-2H-pyridin-1-ylmethylideneamino)-N-[(4R)-7-fluoro-2-oxo-1-[5-(trifluoromethoxy)pyrimidin-2-yl]piperidin-4-yl]thiophene-2-carboxamide 2-amino-6-ethoxy-4-[3-methyl-5-(oxolan-2-ylmethoxy)phenyl]-4H-pyran-3,5-dicarbonitrile N-(3-iodophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 3-(3,5-dimethylpyrazol-1-yl)-6-methylpyridine;hydrochloride 5-[2-(4-chlorophenyl)ethenyl]pyridine-2-carboxylic acid (2S)-5,7-dimethoxy-2-[4-[3-(2-oxopyrrolidin-1-yl)azetidine-1-carbonyl]pyrazol-1-yl]-N,N'-bis(pyridin-4-ylmethyl)heptanediamide 2-amino-N'-[3,6-dichloro-5-(trifluoromethyl)pyridin-2-yl]sulfanylpropanimidamide 5-chloro-4-[1-(3,4-dimethoxyphenyl)ethylamino]-1H-pyrimidin-6-one 1-[(2,6-difluoro-4-methoxyphenyl)methyl]-3-ethenyl-2-methylidenepyridine 2-(methylamino)-N-[(1S,3R)-3-[(6-oxo-4-propyl-1H-pyrimidin-2-yl)amino]cyclohexyl]benzamide 1-[3-fluoro-5-[[2-(trifluoromethyl)pyridin-4-yl]amino]piperidin-1-yl]ethanone 3-[3-(6,7-dihydro-1H-inden-2-yl)phenyl]propanoic acid [4-[4-(hydroxymethyl)anilino]phenyl]azanide 1-[2-(3,5-ditert-butylphenyl)ethoxy]propan-2-ol 5-[3-[4-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl]pyrimidine-4,6-diamine 3-(1,2-difluoroethyl)-5-[4-[(E)-2-nitroethenoxy]phenoxy]-N-(1,3-thiazol-4-ylmethylsulfonyl)thiophene-2-carboxamide 2-[(E)-4-bromobut-3-enyl]anthracene 5-methyl-N-[[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methyl]pyrazine-2-carboxamide N-(4,4-difluorocyclohexyl)-2,6-dimethylbenzenesulfonamide 3-chloro-1,5-dimethylpyrazolo[4,3-b]pyridine (4R)-3-[5-[5-[(2,6-dichlorophenyl)methoxy]pyridin-1-ium-2-yl]-7-fluoro-1H-indazol-3-yl]-4-ethyl-1,3-oxazolidine 1-(6,7-dimethoxyquinolin-4-yl)-N,N,3-trimethylpyrrolidin-3-amine 4-[4-[(4R)-1-cyclohexyl-3,3-difluoropiperidin-4-yl]phenyl]sulfonylbenzonitrile N-(3,5-difluoropyridin-2-yl)-5,6-dimethoxypyrimidin-4-amine;1,1,1-trifluoroethane N-[2-(2,3-dihydroindol-1-yl)ethyl]-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepine-3-carboxamide;hydrochloride N-[3,5-bis(difluoromethyl)pyrazol-1-yl]-1-prop-2-enoylazetidine-2-carboxamide ethane;1-methylspiro[2H-indole-3,9'-xanthene] 5-[(4,6-dichlorotriazolo[1,5-a]pyridin-2-yl)methoxy]-3-(difluoromethyl)-N-ethyl-4-methylidenepyrimidin-2-imine 2-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenoxy]acetonitrile 3-(4-methoxyphenyl)-2,9-dihydrobenzo[f]chromen-1-one 5-cyclobutyl-4-(cyclopropanecarbonyl)-3-ethylsulfanyl-1,2-oxazole-6-carboxylic acid 2-[(4,5,7-trimethyl-1H-indole-6-carbonyl)amino]benzoic acid 2-[(5-methylfuran-3-carbonyl)amino]-9-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)nonanoic acid 3-(1H-benzimidazol-2-ylmethylidene)-4,6-dichloro-1H-indol-2-one 2-[4-amino-3-[2-(dimethylamino)ethylimino]-4,5,6,8-tetrahydroimidazo[4,5-c]azepin-7-yl]-1-phenylethanone;ethane 1-azidosulfanyl-2,3,4,5-tetrafluorobenzene (Z)-2-(1,3-benzothiazol-2-yl)-4-[(5-nitropyridin-2-yl)amino]sulfanyl-3-oxidobut-2-enal 3,6-dibromo-9H-carbazole ethane;4-(6-methoxynaphthalen-2-yl)sulfonylmorpholine 1-(2,4,5,6-tetrahydropyrimidine-1-carbonyl)indole-5-carboxylic acid 6-[4-(dimethylamino)phenyl]-1,5,7,8-tetrahydropyrimido[4,5-d]pyrimidine-2,4,9-trithione N-butyl-6,7-difluoroquinoline-3-carboxamide N-[4-(2,5-dimethoxyphenyl)pyridin-3-yl]-1-ethylpyrrolidine-2-carboxamide 4-[(5-acetamido-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-2-carbonyl)amino]benzamide 3-(6-piperidin-4-yl-1H-benzimidazol-2-yl)benzene-1,2-diol;dihydrochloride (5Z)-3-[2,6-dichloro-4-[2-hydroxy-2-(methylamino)ethoxy]phenyl]-5-[(4-fluorophenyl)methylidene]-1,3-thiazolidine-2,4-dione 6-chloro-4,5,7-trideuterio-2,9-dimethylcarbazole (2S)-1-(3,4-dimethylphenyl)pentane-2-sulfonic acid 1-[2-(furan-2-yl)ethylamino]-3-octoxypropan-2-ol 4-[4-[(E)-3-[4-[2-(5,5-dimethylcyclohexa-1,3-dien-1-yl)ethenyl]phenyl]prop-2-enoyl]phenyl]sulfonylbenzoic acid 4-(3-bromophenyl)-2-[[ethyl(methoxycarbonyl)amino]methyl]piperidine-1-carboxylic acid (2R)-1-acetyl-N-[(Z)-1H-indol-3-ylmethylideneamino]pyrrolidine-2-carboxamide (5E)-2-(3,4-dichlorophenyl)imino-5-[[4-(3,4-dimethoxyphenyl)furan-2-yl]methylidene]-1,3-thiazolidin-4-one 2-[3,5-bis(trifluoromethyl)phenyl]-N-[6-cyclopropyl-4-fluoro-3-(pyridin-2-ylcarbamoylamino)pyrazolo[1,5-a]pyridin-7-yl]acetamide (3S,4R)-4-[(1R,5S)-3-(4-chlorophenyl)sulfanyl-6-bicyclo[3.2.0]hept-2-enyl]piperidine (2Z)-N'-[(3,5-dimethylphenyl)methoxy]-3-[4-ethoxy-3-(trifluoromethyl)phenyl]-2-hydroxyiminopropanimidamide 3-methyl-2,4,5-tris(trifluoromethoxy)benzaldehyde (2E,5Z)-5-[(4-chlorophenyl)methylidene]-2-[1-[4-(diethylamino)-2-nitrophenyl]-2,5-dioxopyrrolidin-3-ylidene]-1,3-thiazolidin-4-one 2-hydroxy-6-nitroindole-1,3-dicarboxylic acid N-methylethanamine;4-(methylaminosulfanyl)-1H-pyrrolo[2,3-b]pyridine-5-carbonitrile (1S,3R)-2,2-dichloro-N'-[4-cyano-2-[2-fluoro-3-[1-methyl-5-[[methyl-[[5-(trifluoromethyl)pyrimidin-2-yl]amino]methyl]pyrazole-4-carbonyl]phenyl]phenoxy]-6-fluorophenyl]-N-cyclopropylethanehydrazide 3-N,5-N,7-N-trimethyl-2-piperidin-1-ylquinoxaline-2,7-diamine N-but-1-en-2-yl-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-imine 3-amino-6,7-difluoroquinoxaline-2-carboxylic acid 7-(difluoromethyl)-6-[1-[2-oxo-2-[4-(trifluoromethoxy)phenyl]ethyl]pyrazol-3-yl]imidazo[1,5-a]pyridine-3-carboxylic acid (2Z)-N-[3-(4-formylphenoxy)propyl]-6,11,12-trihydroxytetracene-5,10-dicarboxamide 3-[1-(2-aminoethylamino)ethenyl]-5-chloro-N'-[[7-fluoro-4-methyl-6-(1-methylpyrazol-4-yl)quinazolin-2-yl]methyl]-2-(methylideneamino)benzenecarboximidamide 4-N,2-dimethylbenzene-1,4-disulfonamide 2-(5,6-dihydroxybenzimidazol-1-yl)acetic acid N-(2-chloropyrimidin-4-yl)-3-methoxypropanamide N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide 2-[(3S)-1-(4-chlorophenyl)sulfonylpyrrolidin-3-yl]-7,8-dimethoxy-N-methyl-[1,2,4]triazolo[1,5-a]pyridine-6-carboxamide [6-(3,4-dimethylphenyl)sulfanylpyridin-2-yl]-methylideneazanium 1-[(E)-[amino-[4-(5,6-difluoroindol-1-yl)anilino]methylidene]amino]-3-(2-phenylpropanoyl)thiourea 1-[1,2-bis(ethenyl)anthracene-9,10-diyl]piperidine 2-[(3S)-1-[2-[cyclopropylmethyl-[4-(4,5-dichlorothiophen-2-yl)sulfanylbutyl]amino]acetyl]pyrrolidin-3-yl]-N-ethyl-N-prop-1-en-2-ylacetamide (2S,4R)-1-[5-amino-7-fluoro-3-(trideuteriomethyl)pyrazolo[4,3-d]pyrimidine-1,6-diium-1-carbonyl]-N,4-diphenylpyrrolidine-2-carboxamide 4-N-(5-bromonaphthalen-1-yl)benzene-1,4-diamine (6S)-2,5-bis[4-(dimethylamino)phenyl]cyclopentene-1,3-disulfonic acid;buta-1,3-diene 6-[4-(trifluoromethyl)phenoxy]naphthalene-1,3-dicarboxylic acid 4-[(3S)-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione;2-methoxyethanol 2-[7-(4,6-dimethylcyclohexa-1,3-dien-1-yl)oxyheptyl]isoindole-1,3-dione 2-amino-4-methoxy-N-[(3S)-5-methylsulfanyl-1-oxopentan-3-yl]benzamide;hydrochloride 2-[[2-[3-(4,5-dimethyl-1H-imidazol-2-yl)phenoxy]acetyl]amino]propanoic acid 2-[4-(1H-pyrazol-4-yl)phenyl]-3-pyridin-4-ylquinoline 3-(2,4-dimethylphenyl)-1-ethylazetidine;2,3-bis[4-fluoro-2-(trifluoromethoxy)phenyl]-N'-hydroxypropanimidamide 2-N,3-N-bis(4-methoxyphenyl)acenaphthylene-1,2,3-triimine N-[4-[2-(cyclopropylmethylamino)ethoxy]phenyl]hydroxylamine 2-[2-[5-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]ethoxy]-N,N-diphenylpyrimidine-4-carboxamide 2,6-difluoro-N'-[2-(4-hydroxyphenoxy)acetyl]benzohydrazide 2-(3,4-difluorophenyl)-N-[4-(2-methylpropoxymethyl)phenyl]propanamide 2-[3-(4-chlorophenyl)sulfonylpropyl]isoindole-1,3-dione N-[(5S)-3-(4-methoxyphenyl)sulfonyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-7-en-9-yl]benzamide 4-[3-(2,5-dimethylphenyl)imidazo[1,5-a]pyridin-8-yl]-7H-pyrazolo[1,5-a]pyrazine 1-[(Z)-3-aminobut-2-enimidoyl]-8-chloro-6,7-dimethoxy-2H-quinoline-4-carboxylic acid 2-[4-(azidomethyl)piperidin-1-yl]-N-benzyl-2-phenylacetamide N-[2,5-difluoro-4-[(4-methylsulfanylphenyl)methoxy]phenyl]-6-oxo-2-pyrimidin-2-yl-1H-pyrimidine-5-carboxamide [6-(3,5-dimethylpyrazol-1-yl)pyridin-3-yl]-[4-[(E)-hydroxyiminomethyl]piperidin-1-ium-1-yl]methanone 1-[3-methyl-4-(pyridine-2-carbonyl)piperazin-1-yl]prop-2-en-1-one 2-(benzenesulfonylmethyl)-N,5-dimethylaniline (2-methylpropanoylamino)urea;4-[6-(1H-pyrazole-5-carbonylamino)pyridin-3-yl]oxybenzamide [(4aR,8aS)-6-[2-(5-methyl-1H-indol-3-yl)ethyl]-1,2,3,4,4a,5,7,8,8a-octahydropyrido[3,4-b]pyrazin-9-yl]-pyridin-3-ylmethanone;dihydrochloride 1-[3-(4-azidopiperidine-1-carbonyl)thiophen-2-yl]ethanone 2-[3-(cyclopropanecarbonyl)phenyl]propylurea 1-[(6S)-3-hydroxy-2,6-dimethylpiperidin-4-yl]-3-(8-methoxyquinoxalin-5-yl)urea 5-(azidomethyl)-3-[4-bromo-3-(trifluoromethoxy)phenyl]pyridine 4-[3-(aminomethyl)-5,6-dihydronaphthalen-2-yl]-N-pyridin-2-yl-1,3-thiazol-2-amine 1-[5-chloro-2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)phenyl]-N,N'-dimethylmethanediamine [(2S)-3-chloro-1,2-dihydroxypropyl]-triphenylphosphanium;bromide 1-(3,4,6,7,8,9,10,11-octahydro-2H-pyridazino[1,2-a]benzimidazol-4-yl)propan-1-one 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-(6-sulfonaphthalen-1-yl)amino]decanoic acid 4-[1,2-diamino-3-(4-bromophenyl)iminoprop-1-enyl]phenol 7,8-dimethyl-3,6,7,9-tetrahydro-2H-furo[2,3-h]quinoline;propanoic acid 3-(3,4-diethoxyphenyl)-5-[2-(methylamino)pyrimidin-4-yl]imidazo[1,2-a]pyridine-8-carbonitrile 2-(1,3-thiazol-5-yl)pyridine-4-carbohydrazide (4S,5R)-2-(3,4-dimethoxyphenyl)-8-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-methoxy-2,8-diazaspiro[4.5]decane;formic acid (Z)-4-[2-acetamidoethyl-(3,4,5-trifluorophenyl)sulfonylamino]-N-hydroxy-3-methylbut-3-enamide 3-[3-(2-methylpropyl)phenyl]cyclohexan-1-amine N-(1-cyanocyclopropyl)cyclobutanecarboxamide;5,6-difluoro-3H-isoindol-1-amine;(2S)-1-[4-(7-methoxyisoquinolin-1-yl)piperazin-1-yl]propan-2-ol 1-(2,4-dichlorophenyl)sulfonyl-2-methylbenzene;5,6-dihydroxy-7-[(5E)-3-hydroxyocta-5,7-dienoxy]-2-methylidenechromene-3-carbonitrile 2-(4-azidophenyl)sulfanylbenzoic acid 1-[(4-methoxyphenyl)methyl]-3-(methylamino)urea N-(2,4-difluorophenyl)sulfonyl-3-ethoxy-4-methoxybenzenesulfonamide 2-[(3S)-2,6-dioxopiperidin-3-yl]-4-methoxyisoindole-1,3-dione 2-[(3aR,7aS)-2-[2-cyanoethyl(methyl)amino]-1,3,4,5,6,7,7a-octahydroisoindol-3a-yl]-N-(furan-2-ylmethyl)acetamide 2-[(1,3,3-trimethylindol-2-ylidene)methyl]furan-3-carboxamide 4-[2,6-difluoro-N-(1,3-thiazol-5-yl)anilino]butan-1-ol (1S,3R)-N-[5-cyano-6-(triazol-2-yl)pyridin-3-yl]-3-(dimethylamino)cyclopentane-1-carboxamide 3-(7-bromo-5-tert-butylbenzimidazol-1-yl)propan-1-ol 2-(N-[2,4-dioxo-1H-pyrimidin-5-yl)-2-methoxyanilino]acetonitrile 6-(2,3-dihydro-1H-inden-5-ylamino)-1'-propanoylspiro[5H-pyrazolo[3,4-d]pyrimidine-4,3'-piperidine]-7-one N-[2,5-dimethoxy-4-(1H-pyrazolo[3,4-c]pyridin-4-yl)phenyl]methanimine (E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]-N-methoxyprop-2-enamide ethane;3-[4-(2-propan-2-ylimidazol-1-yl)anilino]cyclobutan-1-ol [2-[(dimethylamino)methyl]morpholin-4-yl]-[(2R,3S)-2-phenyloxolan-3-yl]methanone (3S,4R)-3-N,1-dibenzyl-4-N-methylpyrrolidine-2,3,4-tricarboxamide N-(2,3-dihydro-1H-inden-5-yl)-7-methoxy-2-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1]benzazepine-4-carboxamide 5-(azidomethyl)-1,3-dichlorobenzene 1-cyclohexyl-2,3-difluorobenzene;7H-purin-6-amine 7-(1,3,2-dioxatriazet-4-yl)-8a-benzyl-4a,5,6,8-tetrahydro-[1]benzofuro[3,2-d]pyrimidine-2,4-dione 4-(2,6-dimethylphenoxy)carbonylbenzoate N-[[(2S,4R)-1-acetyl-2-phenylpiperidin-4-yl]methoxy]-1-azidocyclobutane-1-carboxamide 4-bromo-2,3-dihydro-1H-isoindole-1-carboxamide;N-methylhydroxylamine 4-[(1R)-2,2-dimethyl-3-phenylcyclopropyl]butanoic acid ethane;methanamine;methanol;N-[(2Z,4E)-4-methoxyhepta-2,4,6-trienyl]-5-[3-[7-(1H-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]phenyl]pentanamide 1-(2,6-difluorophenyl)-4-[5-(4-methoxyphenyl)-3-(trichloromethyl)pyrazol-1-yl]sulfonylpiperazine 2-bromo-N-(1,3-thiazol-5-yl)-N-[4-(thiophen-2-ylsulfamoyl)phenyl]benzamide 3-amino-1-[(3R)-2-(4-methylbenzoyl)pyrrolidin-3-yl]pyrazole-4-carboxamide 4-[1-(methylamino)ethenyl]-N-phenylaniline 1,4-dichloro-2-(2-methylphenyl)benzene 2-[4-(6-nitroquinoxalin-2-yl)oxypiperidine-1-carbonyl]butanoic acid N-[3-methyl-4-(2,2,2-trifluoroethoxy)pyridin-2-yl]-4-oxopiperidine-1-carboxamide 2-[4-[7-amino-5-[4-(3,6-dihydro-2H-pyridin-1-yl)cyclohexa-1,3-dien-5-yn-1-yl]pyrazolo[1,5-a]pyrimidin-2-yl]phenyl]-N'-methanimidoylbutanediamide 6-cyclopentyloxy-N,N'-dimethylpyridine-2-carboximidamide 2-[(1Z,3E)-4-aminobuta-1,3-dienyl]-5-methyl-3-phenylquinazolin-4-one 2-azido-5-[2,6-difluoro-4-(trifluoromethoxy)phenyl]thiophene N-[4,6-diamino-5-(2-azidoethylsulfanyl)pyrimidin-2-yl]acetamide 4-[2,2,3,5-tetrafluoro-5-(trideuteriomethyl)heptoxy]-N-(1,3,4,9-tetradeuterio-6-isocyano-7-methylidene-10H-anthracen-2-yl)benzenesulfonamide 1-ethyl-6,7-dimethoxy-4-(3-nitroanilino)quinolin-2-one 4-[3,5-bis(trifluoromethyl)phenyl]-N'-methylpiperidine-1-carboximidamide (5S)-1,5-dibenzylimidazolidine-2,4-dione 2-(4-chlorophenyl)-N-methylbutanamide;1-[5-ethynyl-6-[methoxy(propyl)amino]pyridine-3-carbonyl]piperidin-4-ol 2-[(3R)-4-benzylsulfanylbutyl]-6-iodopyridine 2-[4-(6-chloropyridazin-3-yl)piperazine-1-carbonyl]-2,3-dihydroinden-1-one 3-(1,2-benzothiazol-6-yl)-5-fluoro-6-morpholin-4-yl-7H-imidazo[1,2-b]pyrazole-2-carboxylic acid (Z)-3-hydroxy-1,2-diphenylprop-2-en-1-one (E)-N-[2,3-dihydroxypropyl(methyl)amino]sulfanyl-2,3-dihydroindene-1-carboxamide;ethane 5-(2,6-dichlorophenoxy)-1H-pyrazole 2-[4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]ethanol 5-(1,1,2,2,2-pentafluoroethoxy)-3-[6-[methyl-(7-oxopyrrolo[3,4-b]pyridine-6-carbonyl)amino]spiro[3.3]heptan-2-yl]oxy-2H-indazole-6-carboxylic acid 3-chloro-2-(dibenzylamino)benzoate 5-[(3,5-difluorophenyl)methylamino]-4H-1,2,5-oxadiazol-3-one 2-[4-(1H-benzimidazol-2-yl)butanoylamino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid (2R)-N',N',2-trimethyl-3-naphthalen-1-ylpropanehydrazide 3-[4-(2-phenylethyl)piperazine-1-carbonyl]cyclobutane-1-carboxylic acid 6-[1-methyl-2-oxo-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-b]pyridazine-8-carboxylic acid 1-butan-2-yl-5-[4-methoxy-3,5-bis(sulfanylidene)penta-1,4-dienyl]-6-methylindole-3-carbonitrile (E)-2-cyano-3-[3,5-dimethyl-4-oxo-6-[3-(trifluoromethoxy)phenyl]thieno[3,2-d]pyrimidin-7-yl]-N-(2-morpholin-4-ylethyl)prop-2-enamide 4-azidooxy-1,2-diphenylbutan-1-one N-[4-(4-azidooxy-2,5-dichlorophenyl)pyridin-3-yl]pyridine-2-carboxamide 5-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-3-(1H-pyrrolo[2,3-c]pyridin-2-ylmethyl)-1H-pyrazolo[3,4-b]pyridine 2-(3,5-dimethylpyrazol-1-yl)-N-[1-(pyridin-4-ylmethoxy)propan-2-ylidene]acetamide 2-azido-4-methylsulfanylnaphthalene N-[2,4-difluoro-3-(1H-indazole-5-carbonylamino)phenyl]-6-fluoro-2H-azepine-8-carboxamide (5S)-2-[2-hydroxyethyl(methylamino)amino]-N,5-diphenylcyclohexa-1,3-diene-1-carboxamide 2-[(1,5-dimethylpyrazol-3-yl)carbamoylamino]-N-ethoxyacetamide 6-(3,5-difluorophenyl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]sulfonylpyrazolo[1,5-a]pyridine-4-carboxamide N-[3,5-difluoro-4-(2-sulfanylidene-1H-pyridin-6-yl)phenyl]acetamide 2-[4-(azidomethyl)phenyl]-5-ethoxyfuran N-azido-1-(2,6-dichlorophenyl)methanamine 2-[3-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]-1-phenylethanone;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide 4-(benzenesulfonyl)-5H-benzo[e]indole N-[4-(difluoromethoxy)phenyl]sulfonyl-6-(2,3-dihydropyrrolo[2,3-b]pyridine-1-carbonyl)pyrazolo[1,5-a]pyridine-3-carboxamide 1-(3-bromophenyl)sulfonyl-2-methylbenzimidazole 6-amino-3-bromo-7,8,9,10-tetrahydrobenzo[h]quinoline-2-carboxylate 2-fluoro-3-[1,1,1,2,3,3,4,5,6,7,8,9,10,10,11,12,12a-henicosacyclononaene-2,15-diyl-(2-methoxyphenyl)carbamoyl]benzoic acid N-[(2R)-butan-2-yl]-4-fluorobenzenesulfonamide 1-phenylmethoxycarbonylpiperidine-3-carboxylic acid 2-[4,7-bis(ethenyl)naphthalene-1-carbonyl]oxyacetic acid N-[[3-fluoro-5-[2-(5-pyridin-4-yl-1H-pyrazolo[3,4-c]pyridin-3-yl)-1H-imidazo[4,5-b]pyridin-7-yl]phenyl]methyl]methanesulfonamide 4-N-azido-5,6-dimethylpyrimidine-2,4-diamine N-[1-(3,4-difluorophenyl)-2-methylpropan-2-yl]-7-(2-methoxypyridin-4-yl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine;ethane 3-[(Z)-2-ethoxy-1-fluoro-2-[3-methyl-6-oxo-5-(trifluoromethyl)pyridazin-1-yl]ethenyl]benzonitrile 2-chloro-N'-cyclohexylbenzohydrazide 3-[5-(3,5-dichlorophenyl)-4-methylfuran-2-yl]piperidine 4-[8-amino-1-(2,6-dichlorophenyl)imidazo[1,5-a]pyrazin-3-yl]cyclohexane-1-carboxylic acid 2-[4-(2,5-dioxoimidazolidin-1-yl)phenyl]piperazine-1-carboxylate 2-cyclopropyl-4-(2,5-dimethoxyphenyl)-6-[3-(4-ethylpiperazin-1-yl)azetidine-1-carbonyl]-7H-pyrrolo[3,4-b]pyridin-5-one 6-[[3,5-difluoro-4-(1H-pyrazol-5-yl)phenyl]methyl]-7,8-dihydropyrazino[2,3-b]pyrazine 5-(3,4-difluorophenyl)sulfanyl-2,6,7,8-tetrahydro-1H-pyrazolo[4,3-g]quinazoline 2-[(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanyl]-N-(2,4,5-trifluorophenyl)propanamide 7-(furan-2-yl)-5-thiophen-3-yl-[1,2,4]triazolo[1,5-a]pyrimidine N-[(2S)-5,7-dimethyl-1-[6-oxo-4-(trifluoromethyl)-1H-pyrimidin-2-yl]pyrrolidin-3-yl]-2-methoxy-N-phenylacetamide (E)-2-[4-[4-fluoro-N-methyl-3-(trifluoromethoxy)anilino]piperidine-1-carbonyl]-4,4-dihydroxybut-2-enenitrile 2-(4-chlorophenoxy)-N-[(1R,3S)-3-[2-(5-fluoropyrimidin-2-yl)oxypropanoylamino]cyclopentyl]acetamide 3-cyclopentyloxy-N-[4-(2,4-dimethoxyphenyl)piperazin-1-yl]benzamide 4-chloro-3-methoxy-N-[(2S)-1,1,1-trifluoropropan-2-yl]benzenesulfonamide 2-[4,6-bis(phenylmethoxy)-1H-inden-2-yl]ethanol;ethane 4-benzyl-1,2,3,5-tetrafluorobenzene 2-[3-hydroxy-1-(hydroxymethyl)piperidine-3-carbonyl]benzonitrile N-[2-(benzenesulfonamido)ethyl]-6-oxo-1H-pyrimidine-4-carboxamide 4-benzylsulfanyl-2,6-ditert-butyl-3,5,7-trimethoxynaphthalene 2-[N-ethyl-4-(thiophen-3-ylsulfamoyl)anilino]octanoic acid [[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methylideneamino]carbamic acid 2-cyclopropyl-6-[(2,3-dichlorophenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S,2R,5S)-5-methoxy-2-propanoylcyclohexyl]methanesulfonamide 2-[7-(cyclohexylmethoxy)-1,2,3,4-tetrahydronaphthalen-2-yl]butanal 2-chloro-N-(2-nitrophenyl)-N-propylacetamide (2-methylpyridin-4-yl)-[3-[4-(2-phenylimidazo[1,2-a]pyrazin-3-yl)piperidine-1-carbonyl]pyrrolidin-1-yl]methanone N-benzyl-5-(trifluoromethoxy)spiro[1,3-dihydroindene-2,4'-piperidine]-1'-carboxamide 6-methyl-2,3,5,7,8,9-hexahydrofuro[4,3-h]isoquinoline 2-(2-phenylmethoxycarbonylpiperazin-1-yl)benzoic acid 2-[(2,6-dichlorobenzoyl)amino]-3-[5-[4-[4-(7-hydroxy-3-oxooctoxy)phenyl]piperazine-1-carbonyl]pyridin-2-yl]propanoic acid 6-(4,5-dimethylcyclohexa-1,3-dien-1-yl)pyridine-2-carboxamide 6-(4,5-dihydropyrimidin-2-yl)naphthalene-1,3,4-triamine 2-[5-[[4-chloro-1-methyl-6-(trifluoromethyl)indole-2-carbonyl]amino]pyridin-3-yl]sulfonylacetic acid (4R)-2,4-diphenyl-1,3-thiazole-5-carboxylic acid 4-amino-5,7-dimethyl-2-[1-(methylideneamino)ethyl]-6H-thieno[3,2-c]pyridin-3-one 4-[3,5-bis(trifluoromethyl)anilino]-6-methoxyquinoline-2-carboxamide 2-methyl-4-(3,3,5-trimethyl-2H-indole-1-carbonyl)benzonitrile 2-[4-[(3R)-1-[6,7-dimethyl-8-[[(1S)-1-phenylethoxy]carbonylamino]octyl]pyrrolidin-3-yl]piperidin-1-yl]pyridine-3-carboxylic acid 2-amino-5,7-dimethyl-4-oxothiochromene-3-carboxylic acid 1-methyl-3-(1,4,5,8-tetramethoxynaphthalene-2-carbonyl)imino-1,3a,7a-trihydropyrrolo[3,4-c]pyridine-4-carbonitrile (4R)-6,7,8-trifluoro-N,N,1-trimethyl-2,3-dihydrobenzo[g]thiochromene-4-carboxamide 3-(4,5-dichlorothiophen-2-yl)-4-hydroxy-6-methylpyran-2-one 1-benzyl-2,3-dimethoxybenzene (1S,3R)-3-[[7-cyclopropyl-2-(3H-pyrrol-4-yl)quinoline-4-carbonyl]amino]cyclohexane-1-carboxylic acid 3-[4-(2-hydroxyacetyl)piperazin-1-yl]benzenesulfinamide 5-azido-1,4-dimethylnaphthalene 2-[N'-methyl-N-(oxolan-3-yl)carbamimidoyl]sulfanylpyrimidine-4,6-diamine 4-[(1S)-5,7-difluoro-3,4-dihydro-1H-isoquinoline-2-carbonyl]-5,6-bis(methylsulfanyl)pyridine-2-carboxylic acid [2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-ylmethylamino)-1H-pyridin-4-ylidene]methanol N-(4-bromophenyl)-6-methyl-7H-pyrimido[5,4-b][1,4]oxazin-2-amine ethane;(4R)-2,6-dimethyl-5,7-dihydro-4H-thieno[2,3-c]pyridine [2-chloro-5-fluoro-4-(triazol-1-yl)phenyl]methanol 2-(3,4-dichlorophenyl)-1H-imidazole;propane 3-[5-cyclopropyl-2-(ethylamino)phenyl]-1,6-dimethoxybutan-1-ol;2,3-difluoro-N-methylaniline N-benzyl-4-ethenyl-N,2,5-trimethylaniline N-[4-(2-methoxyphenyl)-2,3-dihydro-1H-inden-5-yl]imidazo[1,2-a]pyridine-8-carboxamide (1R,2S)-N'-[[2-[3-[(2-chloroacetyl)amino]propoxy]phenyl]methyl]spiro[1,3-dihydroindene-2,4'-piperidine]-1'-carboximidamide;dihydrochloride 2-[2-methyl-4-(1-tritylpyrazole-3-carbonyl)piperazine-1-carbothioyl]-6-oxa-2,9-diazaspiro[4.5]decane-8,10-dione 6-bromo-N-[(5,7-dimethyl-1H-indol-4-yl)methylideneamino]-8-(2,2,2-trifluoroethoxy)quinoline-5-carboxamide [(4aR,7aS)-6-(1-methylcyclohexanecarbonyl)-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazin-4-yl]-(furan-2-yl)methanone 5-methyl-6-(oxan-4-yloxy)pyridine-3-carbohydrazide (2S)-3-[4-[3,5-difluoro-2-(propylamino)phenyl]phenyl]-N-methoxy-1,1,1-trifluorobutan-2-amine N-[(5R)-3,3-difluoropiperidine-4-carbonyl]benzamide 4-(1,3-benzothiazol-2-yl)benzene-1,3-diol;2,7-dichlorocyclohepta-1,3,5-triene [4-(N-methylanilino)phenyl]-naphthalen-1-ylazanium 5-[(3S)-1-benzylsulfonylpyrrolidin-3-yl]-2-pyrimidin-5-yl-4H-pyrazol-3-one 5-[[2,6-difluoro-4-[2-(3-methyloxetan-3-yl)ethynyl]phenoxy]methyl]-1H-pyrazole 2-(dimethylamino)-1-[4-[4,6-bis(trichloromethylsulfanyl)pyrimidin-5-yl]phenyl]ethanol N-[1-[2-(1H-imidazol-5-yl)acetyl]piperidin-4-yl]-N,3,3-trimethylbutanamide (1R)-2,2,3-trimethyl-5-phenyl-1H-indene 1,2-dimethoxy-9H-fluorene 2-cyclopropyl-N-[(6-fluoropyridin-3-yl)methyl]oxane-3-carboxamide (4-cyclopentylpiperazin-1-yl)-[4-(3,5-dimethylpyridin-2-yl)oxy-3-fluorophenyl]methanone 6-[(3R)-1,1-dioxothiolan-3-yl]oxy-5-ethyl-N'-hydroxypyridine-2-carboximidamide 1-chloro-2,4,5-triphenylbenzene 1-[(5Z)-5-[[4-(furan-2-ylmethoxy)phenyl]methylidene]-2,3,4,8a-tetrahydro-[1,3]thiazolo[3,2-a]pyridin-7-yl]ethanone 3-[[4-chloro-N-(2,2,2-trifluoroethyl)anilino]methoxy]benzoate 6-[(E)-1-amino-3-methyliminoprop-1-en-2-yl]-4-(2,3,5-trifluorophenyl)pyrazolo[1,5-a]pyridine-3-carbonitrile 1-(2-ethylsulfonylpyridine-3-carbonyl)azetidine-3-carboxamide 3-(cyclohexatrienyl)-1,5,7-trimethoxybenzo[g]indole (E)-3-[4-(dihydroxymethyl)phenyl]-1-[4-[(Z)-2-(5-fluoro-1H-imidazol-4-yl)ethenyl]phenyl]prop-2-en-1-one 3-azido-1,5-bis[(2S)-butan-2-yl]pyrrolo[2,3-b]pyridine (4-chlorophenyl)sulfonyloxymethanide 4-fluoro-N-[[3-(6-methoxypyrimidin-4-yl)oxyphenyl]carbamothioyl]benzamide 1-[4-[5-(aminomethyl)-6-[2-(dimethylamino)ethoxy]-7-fluoro-1H-indol-3-yl]phenyl]cyclopropane-1-carbonitrile;hydrochloride ethane;7-(1H-indol-2-yl)thianthren-2-ol N-(3,5-dichlorophenyl)-2-[4-[6-methyl-7-(pyrrolidine-1-carbonyl)quinolin-4-yl]oxycyclohexyl]propanamide N'-[3-(4-fluorophenyl)propyl]-1,2,3,5,6,7-hexahydropyrrolizine-8-carbohydrazide;hexane 3-amino-N-[5-methyl-7,10,12-trioxo-2-(propan-2-ylamino)-6H-naphtho[1,2-g]quinazolin-8-ylidene]benzamide N-[3-chloro-4-(pyridine-2-carbonyl)phenyl]-1-(4,5-dimethylfuran-2-carbonyl)pyrrolidine-2-carboxamide;hydrochloride N-[1-[(3S,5S)-3,5-dimethylpiperidin-4-yl]pyrazol-4-yl]acetamide 2,4-dimethyl-5-[1-(1-propan-2-ylazetidin-3-yl)pyrazol-4-yl]pyridazin-3-one 2-[3-(4-azidooxybutyl)phenyl]ethanamine 2-[4-(1,3-dioxoisoindol-5-yl)phenyl]acetamide (5-chloro-2,4-dimethoxyphenyl)-[2-(1H-indol-3-yl)ethyl]azanium 2-chloro-4,6-dimethylpyrimido[1,2-a]indole 1-[4-(3,5-difluorophenyl)triazol-1-yl]pyrrolidine;hydrochloride [(4E)-4-[5-chloro-1-[3,3-difluoro-2-hydroxy-3-(3-methylphenyl)propyl]-6,7-dihydro-4H-indazol-3-yl]hepta-4,6-dienoyl]azanium N-[5-fluoro-3-(1H-pyrrolo[2,3-c]pyridine-2-carbonyl)cyclohexa-1,5-dien-1-yl]-1-benzofuran-5-sulfonamide 1-[4-[2-(3,4-dimethoxyphenyl)ethyl]piperidin-4-yl]ethanone 4-azido-N,3-dimethyl-1H-benzo[g]indole-7-carboxamide N-methyl-1,2,3,4-tetrahydronaphthalene-2-carboxamide 4-(3,6-dihydro-2H-pyran-5-yl)-N,N-dimethylthieno[2,3-d]pyrimidine-7-carboxamide (5S)-N-(2-methoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 3-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)-1H-pyridazin-6-one N-[1-[2-(4-methylpiperazin-1-yl)ethoxy]isoquinolin-6-yl]-3,5-dihydro-2H-1,4-benzothiazepine-7-carboxamide 3-[4-[(E)-2,3,3a,9a-tetrahydro-1H-cyclopenta[b]naphthalen-5-ylmethylideneamino]oxybutyl-methylamino]-1-phenylpyrrolidine-2,5-dione 3-[[2-(7-chloroquinolin-4-yl)sulfanylacetyl]amino]-N-(4-phenoxyphenyl)benzamide (E)-3-[4-amino-7-methyl-6-[2-[1-(1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]ethynyl]pyrrolo[2,3-d]pyrimidin-5-yl]prop-2-enoic acid 4-[2-(dimethylamino)ethoxy]-N'-hydroxypyridine-2-carboximidamide 4-ethenyl-2-(5-fluoro-1,3,4-oxadiazol-2-yl)phenol [3-[4-(aminomethyl)phenyl]piperidin-1-yl]-cyclopentylmethanone 1-[4-[[6-chloro-2-(methylamino)pyrimidine-4-carbonyl]amino]cyclohexyl]azetidine-3-carboxylic acid 6-[(E)-2-amino-1-iodoprop-1-enyl]-4-(5,8,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-13-ylamino)pyridine-3-carboxamide 3-[(Z)-1H-indol-6-ylmethylideneamino]-2-sulfanylidene-6-thiophen-2-yl-4,5-dihydro-3H-azepin-7-one ethane;2-[[4-[4-(methoxymethyl)phenyl]piperidin-1-yl]sulfanylamino]pentanedioic acid 3-(4,5-diphenyl-1H-imidazol-2-yl)-9-phenylcarbazole N-[5-(2,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-6-[2-[4-(dimethylamino)piperidin-1-yl]ethoxy]pyrimidine-4-carboxamide 4-[2,6-dichloro-N-(3-methylbutyl)-4-nitroanilino]butan-1-ol 2-[3,5-dimethoxy-4-(morpholin-4-ylmethyl)phenyl]ethanol 2-[[4-(3,5-dichloropyridine-4-carbonyl)piperazin-1-yl]methyl]benzonitrile (2R)-4-azido-N',3-dihydroxy-2-[1-[4-(oxan-4-ylmethoxymethyl)phenyl]cyclopropyl]butanehydrazide 2-(3,5-dimethylpyrazol-1-yl)-N'-hydroxy-6-methylpyridine-4-carboximidamide 2-[(4-ethoxyphenyl)methylideneamino]benzoic acid 2-(9H-fluoren-1-yl)-4,5-dihydro-1H-imidazole 2-[[2-(6,7-dimethoxyisoquinolin-1-yl)oxyphenoxy]methylidene]cyclopropane-1,3-dione 5-[4-(2-methoxyethyl)piperazine-1-carbonyl]thiophene-3-carbonitrile (Z)-2-[2,6-bis(trifluoromethylsulfonyloxy)phenyl]-3-[1,4-dimethyl-5-(trifluoromethyl)pyrazol-3-yl]prop-2-enoate 1-[(2S)-3,3-dimethylbutan-2-yl]-N-naphthalen-2-ylcyclopropane-1-carboxamide N-[(2,4-dihydroxyphenyl)methylideneamino]furan-3-carboxamide 6,7-diethyl-1H-indene 3-[7,10-difluoro-1-methyl-5-(2-phenylethynyl)-4H-imidazo[4,5-c][1]benzazepin-8-yl]propanal 1-(4-ethylphenyl)-3-(2H-tetrazol-5-ylmethoxy)-6,7-dihydroindazole 4-azidooxy-6,7-dichloroquinazoline (3E)-4-amino-3-[(2,5-dimethoxyphenyl)methylidene]azete-2-thione N-[1-(3,4-dichlorophenyl)ethenyl]-6-methylidene-2-pyridin-3-ylcyclohexa-2,4-diene-1-carboximidate (2S)-N-[2-cyclopentyl-5-(4-iodopiperidine-1-carbonyl)phenyl]pyrrolidine-2-carboxamide [4-(2,3-dihydro-1H-benzimidazole-5-carbonyl)morpholin-2-yl]-pyrrolidin-1-ylmethanone 5-[1,3-dimethyl-4-(3-nitropyridin-2-yl)pyrazolo[3,4-b]pyridin-6-yl]oxycarbonylpyrrolidine-2-carboxylic acid 3-(diphenylphosphanylmethylamino)propanenitrile N-[4-[(3,5-dimethylphenoxy)methyl]thiophen-2-yl]propanamide 2,2-bis(4-hydroxyphenyl)-3-[2-(4-methylphenoxy)acetyl]propanedioic acid 7-(2,6-dimethylpyridin-4-yl)oxy-1,3-dihydroimidazo[4,5-b]pyridin-2-one 4-chloro-7,8,9,10-tetrahydrobenzo[h]quinazoline (4-fluorophenyl)-[3-hydroxy-2-oxo-8-(trifluoromethyl)chromen-5-yl]carbamic acid 2-[4-[(3Z,5E)-6-chloro-3-methoxyhepta-1,3,5-trien-4-yl]phenyl]-N-propan-2-ylideneacetamide (2S,3R,4R)-2-[[cyclopropyl-[2-(dimethylamino)ethyl]carbamoyl]oxymethyl]-1-(3-phenoxypropanoyl)-4-phenylpiperidine-3,4-dicarboxylic acid 6-azidooxy-2,3-dichloropyridine (1R)-2,4-difluoro-3-methylsulfonyloxybenzenecarboperoxoic acid 3-amino-4-cyano-5-[2-methoxy-6-(trifluoromethyl)phenyl]-1H-pyrrole-2-carboxamide 2-cycloheptylacetamide;3,6-dimethyl-4H-1,2,4-benzothiadiazin-7-ol 3-[4,5-bis(ethenyl)furan-2-yl]chromene-2,2-diol;ethane 1-[4-[2-(3,5-dimethylcyclohexa-1,5-dien-1-yl)oxyethoxy]-2-propan-2-yloxyphenyl]sulfonylpiperidine 3-[6-(2,4-difluorophenoxy)-8-methyl-7H-purin-2-yl]imidazo[1,2-a]pyridine N-[3,4-dioxo-1-(3-phenylphenyl)butan-2-yl]-5-fluoro-5-(methylaminomethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-2-carboxamide N-[3-(4-azidooxyphenyl)propyl]acetamide 6,11-dihydrobenzo[c][1]benzoxepine;2-methylpiperidine;4-methylmorpholine 1-(3,4-dihydro-2H-chromen-8-yloxy)-3-(3,5-dimethylpiperidin-1-yl)propan-2-ol;formic acid N-methyl-2,3-bis[(4-methylphenyl)sulfonyl]benzamide 4-[(6-fluoroquinolin-7-yl)methoxy]pyrrolidine-2-carboxylic acid 4-[[3,5-bis(trifluoromethyl)phenyl]methoxymethyl]benzaldehyde 3-amino-4-cyano-5-[3,4-difluoro-2-(trifluoromethoxy)phenyl]-1H-pyrrole-2-carboxamide (2S)-2-hydroxy-N-[[3-methylsulfanyl-5-[4-methylidene-6-(1,2,4-triazol-1-yl)-3H-quinazolin-7-yl]phenyl]methyl]propanamide 4-(1,3-thiazol-2-yl)-6-[[2-[2-(trifluoromethoxy)phenyl]sulfonylpyridin-4-yl]amino]cyclohexa-1,5-diene-1-carboxamide 4-(3-hydroxypropyl)-3,6-dimethoxy-7-propan-2-yloxychromen-2-one 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-hydroxypyrimidine-4-carboximidamide 3-[4-(1,6a-dihydrocyclopropa[a]inden-5-ylamino)piperidin-1-yl]-2H-furan-3-ol;ethane 1-(4,5-dihydropyrimidin-2-yl)indole;ethane 1,3-dimethylpyrrolidine;6,8-dimethoxy-2-(4-methylcyclohexa-1,5-dien-1-yl)quinoline 2-[(E)-1-chloroethenyl]-5-fluoro-6,11-dihydropyrido[3,2-c][1,5]benzodiazepine 1-(4-bromophenyl)sulfonyl-3,3a,4,5,6,7,8,9,10,11,12b-undecahydrocycloocta[d]imidazole 1-butyl-4,5-bis(ethenylamino)-3-[2-(methylamino)-6-oxopyran-4-yl]imidazol-2-one;ethane N-(2,4-difluorophenyl)-2-(2-iodoanilino)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 6-bromo-2,3,4,9-tetrahydropyrano[2,3-b]indole 6-cyclopropyl-3-[[1-(2-thiophen-3-ylacetyl)piperidin-4-ylidene]methyl]quinazolin-4-one N-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]butanamide 1-[3-(3,4-dihydro-1H-isoquinolin-2-yl)azetidin-1-yl]-2-(4-phenoxyphenyl)ethanone;propane 5-[4-(1,1-difluoroethyl)anilino]-2-ethoxyphenol N-(4,6-dimethyl-2H-pyrazolo[3,4-c]pyrazol-3-yl)-1,3-benzoxazol-5-amine (5S,6S)-1',3'-dimethylspiro[6H-pyrrolo[2,1-c][1,2,4]triazole-8,4'-piperidine] 2,2-dichloro-3-[4-ethoxy-5-(7-oxo-6,8-dihydro-5H-1,8-naphthyridin-4-yl)thiophen-2-yl]cyclopropane-1,1-dicarbonitrile N-[2-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1H-pyridazin-5-yl]-1,3-benzothiazol-6-amine N-[3,5-difluoro-2-(hydroxymethyl)phenyl]-N'-ethyl-1H-indazole-3-carboximidamide N-benzyl-2-hydroxy-3-[(E)-2-[1,3,4-thiadiazol-2-yl(phenyl)methoxy]ethenyl]-N-propan-2-ylnaphthalene-1-carboxamide 2-methylsulfanyl-N-[5-(pyridin-3-ylamino)pyridin-2-yl]thieno[2,3-c]pyrazole-4-carboxamide N-[(1Z,3E)-1-[4-cyclopropylidene-8-hydroxy-6-(trifluoromethyl)chromen-2-yl]-5-cyclobutyl-4-methylhepta-1,3-dienyl]ethanesulfonamide 2-[[(E)-3,5-dihydroxypent-1-enyl]amino]benzoic acid 3-amino-4-cyano-5-(2,6-difluoro-4-hydroxyphenyl)-1H-pyrrole-2-carboxamide 2-[4-(aminomethyl)-3,5-difluorophenyl]-1H-indol-6-amine N-(4-acetamidophenyl)-2,3-dioxo-1H-indene-5-carboxamide 6-[(3,4-dimethoxyphenyl)methyl]-2-pyridin-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 1,2-diethyl-4-(3-methylsulfinylpropoxy)benzene 2,3-dichloro-1,4,5-triphenyl-4H-indeno[1,2-b]pyrrole 1-[(1S)-2,3-dihydro-1H-inden-1-yl]-3-pyrrolidin-1-ylpropan-2-ol 2-cyclopentyl-5-iodo-4-methyl-1H-pyrimidin-6-one 3-[2-hydroxyethyl(methylsulfonyl)amino]propanoic acid;(1Z,4E)-1-[2-[(Z)-hydroxyiminomethyl]phenyl]penta-1,4-dien-3-one 3-(1,2-dimethylcyclopropyl)-4-[5-[2-fluoro-3-(2H-tetrazol-5-yl)phenyl]pyridin-2-yl]-N'-propan-2-ylidenebenzenecarboximidamide 2,3-dimethylpentane;(1R)-N-[4-ethyl-5-[2-(ethylideneamino)-4,5-difluorophenyl]-2,6-dimethylpyridin-3-yl]-2-hydroxy-2-methoxycyclohexane-1-carboxamide 3-[6-(2,4-dichlorophenyl)pyridazin-3-yl]propanal 2-[5-(1-chloroisoquinolin-4-yl)oxypyrimidin-2-yl]-4-methylpiperazine-1-carboxylic acid [3-(4-fluorophenyl)-5,7-dimethyl-2,3-dihydro-1H-furo[3,2-c]pyridin-6-yl]-pyrrolidin-1-ylmethanone;2-hydroxy-N-[2-(3,4,5-trimethoxyphenyl)ethyl]acetamide (3Z)-2,6-dimethylhepta-1,3,5-triene;1,4,7,8-tetramethylnaphthalene 3-[8-(trifluoromethyl)quinoline-2-carbonyl]piperidine-1-carboxylic acid (2R)-1,3-diamino-N',2-bis[2,6-di(propan-2-yloxy)phenyl]propane-2-carbohydrazide 1-(1,3-benzodioxol-5-yl)-N-[4-methanimidoyl-6-morpholin-4-yl-2-(piperidin-4-ylamino)pyridin-3-yl]cyclopropane-1-carboxamide [4-(2-azidoethynyl)phenyl]sulfonylcarbamodithioic acid (2E)-3,7-dimethylocta-2,6-dienamide;[2-hydroxy-4-(4-methoxyphenyl)phenyl]-(7-oxooctyl)azanium 2-(4,5-diaminoimidazol-1-yl)ethanesulfinate 3-[4-(benzenesulfonyl)piperidine-1-carbonyl]-6H-cyclohepta[b]pyran-2,5-dione N-(4-methylphenyl)-N-[2-oxopropyl(phenylmethoxy)phosphanyl]hydroxylamine (3R)-3-[3,4-bis(phenylmethoxy)phenyl]-2,5,9b-trimethyl-1-phenylsulfonyl-3H-pyrrolo[2,3-g]indol-6-one N-[2,3-difluoro-4-(4-methylpyridin-1-ium-1-yl)phenyl]-6-(3-fluoropiperidine-1-carbonyl)imidazo[1,5-a]pyridine-8-carboxamide 6-(4,5-dichloro-2-ethoxyphenyl)-3-methylsulfanylpyrazine-2-carbonitrile 6-(2-morpholin-4-ylethoxy)pyridin-3-amine 1-[4-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylcarbamoylamino)sulfanylphenyl]azetidine-3-carboxylic acid (3-methylpiperidin-1-yl)-[(2S,4R)-6-nitro-4-[8-[4-(trifluoromethyl)phenoxy]octoxy]oxan-2-yl]methanone 5-(2,3-dichlorophenyl)-1,3-benzothiazole 1-[(4aS,7aS)-1-methyl-2,3,4,4a,5,7,7a-octahydropyrrolo[3,4-b]pyridin-6-yl]-2-cyclopropylideneethanone;3,6-difluoropyridine 5-amino-3-[4-fluoro-2,6-dimethyl-3-(trifluoromethyl)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile 1-azidooxy-2,3-dichlorobenzene ethane;1-[(4Z)-3-methylidenehepta-4,6-dienyl]-9H-fluorene 3-[4-(1,2,4-triazol-1-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 4-[(2-benzylphenoxy)methyl]-N'-hydroxypyridine-2-carboximidamide 2-methyl-1,3,8-triazatricyclo[7.4.0.03,7]trideca-9,12-diene 5-[2-(4-ethenoxyphenyl)ethynyl]-1,3-difluoro-6-isothiocyanato-2-propylnaphthalene 1-[(E)-3-ethenyliminobut-1-enyl]-6,7-dimethoxy-2,3-dihydro-1H-isoindole [4-(2-chlorophenyl)piperazin-1-yl]-[6-(3,4-dimethoxycyclohexa-2,4-dien-1-ylidene)-2-fluorocyclohexa-2,4-dien-1-yl]methanone 2-(3,4-dichlorophenyl)-N-[2-[methyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]-2-oxoethyl]sulfanylacetamide 1-[4-(2,2,2-trifluoroethoxy)pyridine-3-carbonyl]piperidine-3-carboxylic acid 2,6-diamino-N'-[[2-fluoro-5-(trifluoromethyl)phenyl]methyl]benzenecarboximidamide 2,5-dimethyl-3-[[1-(4-phenylphenyl)ethylamino]methyl]phenol N-[2,3-dihydro-1H-inden-4-yl(oxetan-3-yl)methyl]but-2-ynamide 5-(azidooxymethyl)-1,3-dichloronaphthalene 3-[6-(5,5-dimethylhexylamino)-1H-benzimidazol-2-yl]-4-[(3,3-diphenylpropanoylamino)methyl]-5-hydroxynaphthalene-1-carboxamide 1-N',3-N'-bis[(Z)-pyridin-2-ylmethylideneamino]benzenedihydrazide;butane 4-[(2R)-1-hydroxypropan-2-yl]sulfanyl-3-methoxyphenol 5-[3-(4-azidophenoxy)propoxy]-2H-tetrazole 4-[4-amino-3-(methoxyiminomethyl)phenyl]-2,6-dichlorophenol 2-[3-amino-4-(2,5-difluorophenyl)butanoyl]-N-[1-[3-[(Z)-hydroxyiminomethyl]thiophen-2-yl]ethylidene]-6-methoxy-7-methyl-3,4-dihydro-1H-isoquinoline-6-carboxamide N-(3,5-dimethoxyphenyl)-1H-pyrrole-2-carboxamide (5R)-N-(2,4-dimethylphenyl)-2-[(3S,6S)-3,5-dihydroxypiperidin-1-ium-1-ylidene]-4-oxo-1,3-thiazinane-5-carboxamide 2-(3,6-dichloro-9H-xanthen-1-yl)-5-nitrobenzoic acid 6-azidooxy-7,8,9,10-tetrahydrophenanthridine 1-[(Z)-3-aminobut-2-enimidoyl]oxycarbonyl-5-chloronaphthalene-2,6-dicarboxylic acid N-[3-(5-oxo-1,4-dihydropyrazol-3-yl)phenyl]-2-propan-2-yl-1,3-thiazole-5-carboxamide 4-azidooxy-3-(4-fluorophenyl)sulfanyl-1H-pyrrole 6-[2-(trifluoromethyl)phenyl]sulfonylquinoline (3S)-N,2-dimethyl-4-[(6R,11R)-7-oxa-1,5,10-triazatricyclo[8.4.0.03,8]tetradeca-10,13-dien-12-yl]-3-[3-oxo-3-[[3-(trifluoromethyl)phenyl]sulfonylamino]propanoyl]piperazine-1-carboxamide N-[(3R)-1-(3-cyanoazetidine-1-carbonyl)piperidin-3-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carboxamide N-(azidomethyl)-3,5-dichloro-N-ethylaniline 7-bromo-2-(4-methylphenyl)-3H-quinazolin-4-one 1-(2,6-dimethylphenyl)-3-[(Z)-(4-hydroxy-3-iodo-5-methoxyphenyl)methylideneamino]urea 2-amino-N-(1H-imidazol-5-ylmethyl)thieno[3,2-d]pyrimidine-4-carboxamide [2-(3,5-dimethylpyrazol-1-yl)pyridin-4-yl]-[3-fluoro-3-(hydroxymethyl)pyrrolidin-1-yl]methanone 4-methyl-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-yl)thiophene-3-carboxamide 3-chloro-2,5,6-trimethoxybenzoic acid N-butanoyl-2-methyl-N-(3-morpholin-4-ylpropyl)benzamide 1-butyl-2,3-dimethyl-5-nitrobenzene 4-bromo-2,6-dichloropyridin-3-amine 2-(3,4-dichlorophenyl)sulfonylacetic acid (2S)-2-[[4,6-dichloro-5-(3,4-dihydro-1H-isoquinoline-2-carbonyloxymethyl)pyridine-2-carbonyl]amino]-3-phenylpropanoic acid 5-[(4-fluorophenyl)methyl]-4,6-dioxothieno[2,3-d]pyrimidine-2-carboxylic acid 2-[(1S,3aR)-5-hydroxy-6-propyl-1,3a-dihydrocyclopenta[c]chromen-4-ylidene]propanedioic acid 2-(4-bromophenyl)pyridine;ethane 1-[4-(2,6-dimethylmorpholine-4-carbonyl)cyclohexen-1-yl]-3-pyridin-2-ylurea 3-[(2E)-3,7-dimethylocta-2,6-dienoxy]-4-hydroxybenzoic acid 2-(4-azidooxyphenoxy)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine 6-cyclopropylsulfonyl-N,2-dimethoxypyridine-3-carboxamide 2-(3-oxobutanoyl)benzoic acid [4-azidooxy-6-methylsulfanyl-5-(trifluoromethyl)pyridin-2-yl]hydrazine (2R)-2-[[3,5-bis(trifluoromethyl)phenyl]carbamoylamino]-N'-hydroxypropanediamide (1-methoxybenzo[f]indol-2-yl)methanamine (2S)-2-[2,5-difluoro-4-(N'-hydroxycarbamimidoyl)phenoxy]propanoic acid 3-chloro-N-(5,6-diethoxypyridin-2-yl)benzamide 4-[(4S)-5-methylidene-4,8b-dihydro-1H-cyclohepta[c]pyrazol-4-yl]benzenesulfonamide [1-[3,4-bis(trifluoromethyl)benzoyl]piperidin-2-yl]carbamic acid (6S,9R)-N-(2,4-difluorophenyl)-8-oxo-3,5,6,7,9,10,11-hexazatricyclo[7.4.0.02,6]trideca-1(13),2,4,10-tetraene-12-carboxamide 5-ethyl-2,4-diiodothiophene N-(6,7-dihydrobenzo[e][1]benzothiol-4-yl)-2-pyridin-3-ylacetamide 4-[azido(phenyl)methyl]-2,3-dihydroinden-1-one 3-[(1S)-1-(4-ethylsulfonylphenyl)-2,2,2-trifluoroethoxy]-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine (2S)-4-[3-chloro-7-(thiophen-2-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]oxy-N,1-dimethylpyrrolidine-2-carboxamide N-[2-fluoro-5-(trifluoromethyl)phenyl]formamide;1-[2-hydroxy-4-(1H-pyrazol-4-yl)phenyl]ethanone 2-(azidomethylsulfanyl)-6-bromo-1H-benzimidazole (5R)-N-(2,4-dimethylphenyl)-4,7-dioxo-2-propan-2-ylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-[[(3S)-4-oxo-1-phenylazetidine-2-carbonyl]amino]piperidine-1-carboxylic acid (E)-1,3-diphenylpent-1-en-2-ol 6-[2-(4,5-dihydro-1H-imidazol-2-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile N-[(2S)-1-(3,5-dihydroxyphenyl)propan-2-yl]acetamide 2-(4,5-ditert-butyl-2-hydroxyphenyl)acetic acid N-[5-(2,4-difluorophenyl)sulfonyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-3-yl]pyridine-2-carboxamide 2-amino-4-(3,5-dinitrophenyl)-6-methylbenzene-1,3-dicarbonitrile 2-[1-(cyclopropanecarbonyl)piperidin-4-yl]-6-[(2,4-difluorophenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-[1-(6-chloropyridazin-4-yl)piperidine-4-carbonyl]benzonitrile 2-[3-[4-(8,9-dihydropyrido[2,3-b]indol-6-yl)phenyl]phenyl]pyrido[1,2-a]pyrimidine 5-[(1E,3Z)-2,4-difluorohexa-1,3,5-trienoxy]-2-[6-[1-ethyl-3-methylidene-5-(2,2,2-trifluoroethoxymethyl)pyrazol-2-yl]pyridin-3-yl]-N'-hydroxybenzenecarboximidamide N-[3-methyl-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yloxy)phenyl]pyridine-4-carboxamide N-[1-(2,4-dimethoxyphenyl)ethyl]-7-methoxyquinoline-3-carboxamide 1-[(2R,3S)-3-methoxybutan-2-yl]-N-phenylazetidine-2-carboxamide 4-bromo-2,3-di(propan-2-yl)pyridine 2-[3-[5-(1-bicyclo[1.1.0]butanyl)pentoxy]benzoyl]-7-chloro-N,4-dihydro-1H-isoquinoline-5-sulfonamide 2-azidooxy-1,3,5,6-tetrachloronaphthalene 3-(1,4-dioxaspiro[4.5]decan-8-yl)-4-phenylbenzoic acid 4-(2-bromophenyl)-N'-(5,6-dihydronaphthalen-1-ylmethyl)benzohydrazide 3-(azidomethyl)-5-[4-chloro-2-methoxy-6-(trifluoromethyl)phenyl]-1,2,4-oxadiazole 4-[(3R)-1-azidopyrrolidin-3-yl]oxy-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid 4-[3,4,7-trihydroxy-5-(methylamino)naphthalen-2-yl]benzene-1,3-diol 3-[4-(3-fluorophenyl)-1H-pyrrolo[2,3-c]pyridin-2-yl]-5-pyrazin-2-yl-1H-pyrazolo[4,3-b]pyridine 2-bromo-N',N'-bis(4-propan-2-ylbenzoyl)benzohydrazide 3-bromo-N-(2,6-difluorophenyl)-4-methylbenzamide;ethane 2-[4-(2,6-dimethoxypyrimidin-4-yl)phenyl]-N-hydroxypropanamide 1-[(4S)-4,8-dimethyl-2-piperidin-1-yloctoxy]-3-ethylbenzimidazol-3-ium;bromide N-cyclohexylsulfonyl-1-(3,4-dichlorophenyl)-5-methylimidazole-2-carboxamide 1-[(E)-1H-indol-3-ylmethylideneamino]-2-nitroguanidine 4-tert-butyl-2-(3,5-dimethylphenyl)-1H-pyrimidin-6-one (4Z,5E)-2-(4-methylphenyl)-3-oxo-1,4-diazepane-6-carbonitrile (2-azidopyrimidin-5-yl)-(1,6-dimethylindol-4-yl)methanone N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]prop-2-enamide N-[(E)-[4-hydroxy-3-nitro-5-(trifluoromethyl)phenyl]methylideneamino]pyridine-2-carboxamide N-butan-2-yl-1'-(thiophene-3-carbonyl)spiro[5,6,8,8a-tetrahydro-[1,3]oxazolo[3,4-a]pyrazine-1,4'-piperidine]-7-carboxamide [[5-chloro-6-(2,6-difluoroanilino)pyridin-3-yl]amino]thiourea (5S)-3-[3,5-bis(trifluoromethyl)phenyl]-5-(diethoxyphosphorylmethylidene)-1,4-dihydroxy-2H-pyrrole N'-[(1Z,3E)-2-[6-(trifluoromethyl)pyridin-3-yl]penta-1,3-dienyl]ethane-1,2-diamine 6-azidonaphthalene-1,3-dicarboxylic acid 3-[(1R)-5,6-difluorocyclohepta-2,4,6-trien-1-yl]-7-(methoxyamino)-2H-quinazoline-2-carboxylic acid 6-bromo-3-methyl-2,4-dihydro-1H-pyridine;N-[(E)-2-hydroxypent-2-en-4-ynyl]-5-methoxypyridine-3-carboxamide 2-(4-methoxyphenyl)-5-(trifluoromethylsulfanyl)pyrazole-3-carboxylate 3,6-dimethoxy-N'-[[5-methyl-2-(1H-pyrazol-4-yl)phenoxy]methylsulfonyl]pyridazine-4-carboximidamide 4-[(2,5-difluorophenyl)methoxy]-3-ethylpyridine 2-cyclohexa-1,5-dien-3-yn-1-yl-4-[(E)-2-[4-[6-hydroxy-2-(oxan-4-yl)indazol-5-yl]oxyphenyl]ethenyl]-1,2,4-triazol-3-one N-[4-(methylamino)phenyl]-2-propan-2-yloxyacetamide 6-[[(2S,4R)-4-methoxypyrrolidine-2-carbonyl]amino]pyridine-3-carboxamide ethane;N-[2-methyl-5-(6-methylidenecyclohexa-1,3-dien-1-yl)phenyl]formamide 3-[(4-chlorophenyl)methyl]-1-[(E)-2-hydroxypropylideneamino]thiourea 2-methoxy-1,4-bis[3-(trifluoromethyl)phenyl]benzene 1-(2,3-dimethoxyphenyl)-2-methylcycloheptane 1,2-bis(2-cyclohexylethoxy)-10H-phenothiazine 3-[5-(2-methoxypyrimidin-4-yl)-1,2-dihydrotriazolo[4,5-b]pyridin-1-ium-3-yl]propanamide 5-methyl-1,3-diphenylpyrazolo[4,3-c]pyridazine 3-[4-(2,6-difluorophenyl)pyrrolidin-1-yl]oxy-5-ethynylpyridine 2-aminooxycarbonyl-3-(4-methylsulfonylphenoxy)benzoic acid [2-(1,3-benzodioxol-5-yl)pyridin-4-yl]methanamine 2-[(E)-1,3-benzodioxol-5-ylmethylideneamino]oxy-N-[(Z)-(4-hydroxy-3-nitrophenyl)methylideneamino]acetamide (5S)-2-benzylsulfanyl-4,7-dioxo-N-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide (4R)-1',7'-dihydroxyspiro[6H-furo[2,3-f]chromene-8,3'-indole]-2'-one 3-cyclohexylpropanoic acid;N-[4-[(E)-2-(1H-indol-5-yl)ethenyl]-6-methylpyridin-2-yl]formamide 2-tert-butyl-5-(4-propan-2-ylphenyl)-1H-pyrrole N-[(1R,3S)-3-(6-chloroimidazo[1,2-a]pyridin-5-yl)cyclopentyl]-4-methoxypyrimidine-2-carboxamide 2-(1-phenylethylamino)-4,5-dihydropyrimidine-6-carboxamide 2-(2,6-dimethylpyridin-4-yl)-3H-thieno[3,2-d]pyrimidin-4-one 1-(4,5-dimethylcyclohexa-1,3-dien-1-yl)sulfonylbenzimidazole (Z)-3-[4-(diethylamino)phenyl]-2-[6-fluoro-5-methyl-1-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzimidazol-2-yl]prop-2-enenitrile 2-(4-aminophenoxy)-N-[6-(3,5-dimethylphenyl)-1,8a-dihydroimidazo[1,2-a]pyridin-7-ylidene]acetamide ethane;(2S)-N-hydroxy-6,8,12,13,14,15,16,17-octahydrocyclopenta[a]phenanthrene-2-carboxamide 7-methylsulfanyl-3,4-dihydroquinoline 7-azidooxy-3,4-dichloro-1H-quinolin-2-one 3-[3,5-bis(trifluoromethyl)phenyl]propanamide 1-azido-3-(4-tert-butylphenyl)benzene 4-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-N-[2-[(6S)-6-ethenoxy-1,5-dioxospiro[2.5]octane-7,4'-piperidine]-1'-yl]pyridine-3-carboxamide 3-[4-chloro-3-(trifluoromethyl)phenyl]-1,2-dihydrobenzimidazole 3-chloro-4-[[2-(cyclopropylmethyl)-1,3-thiazol-5-yl]sulfonylamino]benzoic acid 1-[2,4-dimethyl-5-(3-naphthalen-2-ylpropyl)phenyl]ethanone (2S,3R)-1-(5-chloropyrimidine-4-carbonyl)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-N-(oxetan-3-ylsulfamoyl)-2-pyridin-3-ylpyrrolidine-3-carboxamide 5-[[4-hydroxy-1-(1,2,3,4-tetrahydroquinoline-2-carbonyl)piperidin-4-yl]methyl]-1H-pyridin-2-one 2-amino-4-(4-chlorobenzoyl)-N-[1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl]-6-fluorobenzamide N-ethylacetamide;2,3,4,5,6-pentachloroaniline 4-methyl-6-[5-(4-phenylimidazol-1-yl)thiophen-2-yl]pyrimidine (2R)-4,7-dihydroxy-N-[1-(5-methylfuran-2-yl)ethyl]-6-oxospiro[2.5]octane-2-carboxamide 4-[[2,5-difluoro-3-(methylamino)phenyl]sulfamoyl]thiophene-2-carboxamide 3-methyliodanuidylisoquinoline N-[(4,5-dimethylthiophen-2-yl)methylideneamino]pyridine-3-carboxamide [4-[(4-aminophenyl)diazenyl]cyclohexa-1,5-dien-1-yl]-methoxy-oxoazanium 1-[4-(2,5-dimethylbenzimidazol-1-yl)-6-propan-2-ylpyrimidin-2-yl]azepane 3-chloro-N-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]pyridine-2-carboxamide 2-[(3-hydroxy-7-methyl-1H-indol-2-yl)diazenyl]-5-nitrobenzoic acid N-[2,3-dimethyl-4-(6-oxo-1H-pyrimidine-4-carbonyl)phenyl]-2,2-dimethoxycyclopropane-1-carboxamide [(4aS,7aS)-1-[(2-methylphenyl)methyl]-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b]pyridin-6-yl]-pyrimidin-5-ylmethanone;2,2,2-trifluoroacetic acid (2S)-N,4-dimethyl-1-[3-(trifluoromethoxy)benzoyl]pyrrolidine-2-carboxamide 1-methyl-2,6-di(propan-2-ylidene)-5H-imidazo[4,5-b]pyridine 2-(7,8-difluoro-3-pentylnaphthalen-1-yl)-5-methoxypyridine 1-[4-(2,3-dimethylbutan-2-yl)phenyl]sulfanylnaphthalene N-[4-cyano-3-(trifluoromethyl)phenyl]-2-ethoxybenzamide (4S)-3-[3-methoxy-5-oxo-6-[2,4,6-trideuterio-1-(trifluoromethyl)indol-3-yl]pyrazin-2-yl]-4-methyl-N-(2,2,2-trifluoroethyl)-1,3-oxazolidine-5-carboxamide 4-cyclopropyl-6,8-bis[(5-methoxy-1H-indol-3-yl)methyl]quinazolin-7-ol 7-azido-5,7-dimethyl-2-[(4-methylphenyl)methyl]-1H-imidazo[4,5-b]pyridine (5E)-2-imino-5-[(1-methylpyrazol-4-yl)methylidene]-3H-pyran-4-one 3-[2,4-difluoro-5-(propylcarbamoyl)anilino]sulfanylbenzoic acid 5-[2-(4,6-diphenylpyrimidin-2-yl)-3H-1,2-benzothiazol-7-ium-3-yl]benzimidazolo[1,2-a]quinazoline ethane;N-[1-[3-(4,6,7-trimethoxyquinazolin-2-yl)phenyl]sulfonylpyrrolidin-3-ylidene]acetamide 4-(dimethylcarbamoyl)-3,5-bis[2-(trifluoromethoxycarbonylamino)ethyl]benzoic acid [7-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl]carbamic acid N-[(3,4-difluorophenyl)methyl]-2-methoxy-6-(piperidin-1-ium-1-ylideneamino)pyrimido[5,4-d]pyrimidin-8-amine 4-(2-propan-2-ylbenzimidazol-1-yl)aniline 3-(9H-fluoren-1-yl)-2-nitrobut-2-enenitrile 5-bromo-2-[3-[(1R)-1-cyclopropylethoxy]pyridin-4-yl]-N,N-dimethylaniline 2-azido-4,5-diphenyl-1H-imidazole 2-(azidomethyl)-7-chloroquinoline 6-(4,5-dihydrothieno[3,2-b]pyrrol-2-yl)hexanamide N-[4-chloro-3-(trifluoromethyl)phenyl]-2-methoxy-5-(pyridin-4-ylmethylamino)sulfonylbenzenesulfonamide 4-N-(7,8-dihydronaphthalen-1-yl)benzene-1,4-diamine N-(2,5-dimethoxyphenyl)-6-ethyl-1-[(4S)-3-methylideneoxan-4-yl]pyrazolo[3,4-d]pyrimidine-4-carboxamide 2,4-dimethyl-5-[[6-[(3R)-oxolan-3-yl]oxypyrazin-2-yl]amino]benzenesulfonamide 2-cyclobutyloxy-5-[4-(2,3-difluorophenyl)piperazine-1-carbonyl]benzonitrile 6-amino-5-[[(4S,8aR)-3,4,4a,5,7,8,8a-octahydro-2H-pyrano[3,4-b]pyrazin-1-yl]methyl]pyridine-3-carbonitrile N-[2-[4-(9H-fluoren-1-ylsulfonylamino)phenyl]ethyl]benzenesulfonamide 4-hydroxy-2,5-di(propanoyl)benzonitrile 1-cyclopropylsulfonyl-4-(3,5-dimethoxyphenyl)piperazine 4-[5-(2,6-difluorophenyl)-1H-imidazol-2-yl]-3-(3-methoxyphenyl)-1H-pyridin-2-one 2-(4,5-dimethylheptanoyl)benzenesulfonamide 2,3-dimethyl-6-[(1Z)-3-methylidenepenta-1,4-dienyl]pyrazolo[5,1-c][1,2,4]triazole N'-(6-methylpyridin-2-yl)-1,3-thiazole-4-carbohydrazide 2-bromo-6-(1,1,1,2,3,3,4,4,4-nonafluorobutan-2-yl)-1H-indole 2,3-dihydro-1H-inden-4-yloxymethanol;6-(trifluoromethyl)-1-benzofuran 5-[(4E)-4-butylidene-2,5-dimethylphenyl]sulfanyl-4H-pyrimidine 5-[4-(9,9'-spirobi[fluorene]-2'-yl)phenyl]imidazolidine-2,4-dione N-[1-(3-bromo-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl)-2-methoxyethylidene]hydroxylamine N-[2-(dimethylamino)ethyl]-5,6-difluoro-3-iodopyrazine-2-carboxamide 5-(1,3-benzodioxol-5-yl)imidazolidine-2,4-dione 3-azido-1-ethylsulfonyl-2,5-dimethoxybenzene 2-[6-(4-chloro-2-methoxyphenoxy)-1-methylindazol-3-yl]propanamide 5-(3,4-dichlorophenyl)imino-1-[2-(methylamino)ethyl]imidazolidine-2,4-dione 2-(4,5-dihydro-1H-imidazol-2-yl)-1-methoxyindole 4-(1H-pyrrolo[2,3-b]pyridin-5-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 2,3-dimethylbutane;6-(3-ethylphenyl)-7-methylidene-1-methylidene-5H-imidazo[4,5-g]quinoline (2R)-N-[(1S)-1-[2-[4-cyano-3-(trifluoromethyl)anilino]-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]propyl]pyrrolidine-2-carboxamide 2-[2-(5-aminothiophen-3-yl)ethynyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-6H-benzo[h]quinoline-9-carboxamide (1S)-N-[6,7-difluoro-2-methyl-4-[[3-(trifluoromethoxy)phenyl]methylamino]quinazolin-5-yl]-8-azaspiro[4.5]decane-8-carboxamide 3-[1,2-dimethyl-5-(trifluoromethoxy)indol-3-yl]propanal N-[2-(ethylideneamino)phenyl]propanethioamide 3-azidosulfanyl-2-butylfuran N-[2-(4-bromophenyl)ethyl]-N',N'-dimethylpropane-1,3-diamine;oxalic acid 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]piperazine-1-carboxamide N-[5-[[3-(2-azidopropyl)-1H-indol-4-yl]oxymethyl]pyridin-2-yl]acetamide N-(1H-indazol-6-yl)-2-methyl-N'-[(3E,5Z)-octa-3,5-dien-4-yl]propane-1,3-diamine 1-[2-(3,4-dimethoxyphenyl)ethyl]-6-hydroxy-5-[(1R)-2-[(4S)-oxepan-4-yl]-1-pyridin-4-ylpropyl]pyrimidine-2,4-dione 2-[5,8-difluoro-6-(2-methoxyethyl)naphthalene-2-carbonyl]-3-ethylsulfonyloxy-3,4,7,9-tetrahydro-1H-pyrido[4,3-b]indole-5-carboxylic acid 1-bromoethane;ethane;N'-(4-methoxyphenyl)sulfonyl-N,N'-diphenylpropanediamide 3-[2-methylsulfonyl-5-(trifluoromethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 2-[4,6-bis(4-methylpiperazin-1-yl)pyrimidin-5-yl]benzoate N-[2-(4,5-diphenylthiophen-3-yl)ethyl]-2-pyridin-2-ylpyridine-4-carboxamide N-(2-hydroxyethyl)-3-[5-methoxy-4-oxo-6-[4-(2H-triazol-1-ium-1-yl)anilino]-7H-pyrrolo[2,3-d]pyrimidin-3-yl]benzamide N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]-3-hydroxybenzamide 4-[2,6-dimethyl-3-(trifluoromethyl)phenyl]-N-pyrimidin-5-ylpyrimidin-2-amine N-[(2S)-1-cyclohexyl-3-pyridin-4-ylpropan-2-yl]pyrrolidine-1-carboxamide (2R,4S)-1-[(3-azidophenyl)methyl]-2-(cyclopropylmethoxy)piperidine 2-[6-(ethoxymethyl)-3,5-dimethylpyridin-2-yl]-5-hydroxypyran-4-one 2-(4-fluorophenyl)-5,6-dimethyl-1H-pyrrolo[3,2-c]imidazole 6-(cyclopropanecarbonyl)-3-[2-hydroxy-4,5-bis(phenylmethoxy)phenyl]thieno[3,2-d]pyrimidin-4-one 4-[[5-(aminomethyl)-1,2-oxazol-3-yl]diazenyl]benzene-1,2-disulfonic acid (3S,4R)-2-[5-[6-(4-chlorophenoxy)pyridin-3-yl]pyridin-3-yl]-1-oxo-N'-propan-2-ylpyrazolidine-4-carboximidamide 1-[[3-(3,5-dimethylpiperidine-2-carbonyl)phenyl]methyl]pyrazole-4-carboxylic acid 4-(2,6-difluoro-3,5-dimethoxyphenyl)butanoate 3-[2-methylpropyl(1,3-thiazol-5-yl)amino]butanoic acid (2S,4S)-N-[5-chloro-3-fluoro-1-hydroxy-7-(trifluoromethyl)-3H-2,1-benzoxaborol-6-yl]-4-hydroxy-4-(2-methoxyethyl)pyrrolidine-2-carboxamide 1-(5,7-dibromobenzo[g][2]benzoxepin-3-yl)pyrrolidine;hydrochloride 3-cyclopropylsulfonyl-2,4,6-trimethylpyridine 3-[4-(furan-2-ylmethylamino)phenyl]benzamide 1-[4-methyl-3-[5-(3,6,6-trimethylcyclohexen-1-yl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]-2,3,4,4a,5,6-hexahydroquinoline-8-carbonitrile 4-[[1-ethylsulfonyl-3,5-dimethyl-2-(trifluoromethoxy)-2H-imidazole-4-carbonyl]amino]pyridine-2-carboxylic acid 4-[2-(3,5-dichloro-4-fluorophenyl)cyclohexyl]butanoic acid 4-(5,6-dimethyl-2,3-dihydro-1H-indene-2-carbonyl)-N-[2-[3-fluoro-4-(pyrrolidine-1-carboximidoyl)phenyl]propan-2-yl]piperazine-1-carboxamide 5-(2,4-dichlorophenyl)-1H-pyrazole 1-[[(5R,6S)-3-methyl-7,8-dioxo-2,4,5,6,9-pentazatricyclo[7.4.0.02,6]trideca-1(13),3,10-tetraene-12-carbonyl]amino]pyrazole-3-carboxylic acid 4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-pyridin-2-one N-[(E)-(5-bromo-2,3-dihydroxyphenyl)methylideneamino]benzamide;nickel(2+);(E)-oxido-oxidoimino-oxido-oxidoazanium 1-[(2S,4R)-4-hydroxy-2-methylpiperidine-1-carbonyl]-N,N-dimethylpyrazole-3-sulfonamide 1,2-diamino-6-oxo-4-(3,4,5-trifluorophenyl)pyridine-3,5-dicarbonitrile (1Z,3E)-2-methylsulfanyl-4-phenoxybuta-1,3-diene-1,4-diamine N-[2,5-dimethyl-4-(6-methylcyclohexa-1,3-dien-1-yl)pyrazol-3-yl]-2H-pyridine-1-carboxamide 1-[1-(2,4,5-trifluorophenyl)ethyl]pyrrolidine 5-ethyl-1,3-dimethyl-2-[(4-phenylpiperazin-1-yl)methyl]-6H-pyrazolo[4,3-d]pyrimidin-7-one 3-(2,4-difluorophenyl)-N-[5-methyl-1-(oxan-2-yloxy)pentan-3-ylidene]cyclobutane-1-carboxamide 4-[(6R)-7-(3,4-dichlorobenzoyl)-2-[3-methyl-5-(1H-pyrazole-4-carbonyl)phenyl]-3-oxo-6-(trifluoromethoxy)-6,8-dihydro-5H-imidazo[1,5-a]pyrazin-1-yl]-N-ethylbenzamide 1-[2-amino-3-(4,5-dimethoxycyclohexa-1,3-dien-1-yl)-6-methanimidoylphenyl]ethanone 6-methoxy-7-pentyl-4H-chromene 2-[3-(difluoromethoxy)phenyl]-N,6-dimethyl-1H-imidazo[4,5-b]pyridin-7-amine 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-hydroxypyrimidine-4-carboximidamide 1-ethylsulfonyl-4-[4-(trifluoromethoxy)anilino]-7-(trifluoromethylsulfanyloxy)quinolin-2-one 2-[(6,7-dichloro-4-oxo-3H-quinazolin-2-yl)methoxy]-N'-hydroxybenzenecarboximidamide 4-[5-ethoxycarbonyl-1-(4-fluorophenyl)pyrazole-3-carbonyl]piperazine-1-carboxylic acid 5-[(2R)-6,15-dibromo-13-chloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl]-N-[(1S)-1-hydroxyethyl]pyridine-3-carboxamide 3-(2,3-dihydro-1H-inden-2-yl)-N'-[(E)-prop-1-enyl]-5-[1-(3-pyrimidin-4-ylanilino)ethylideneamino]penta-1,3-diene-2-carboximidamide (1S,2R)-N-[8-amino-6-(4-benzylphenyl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 6-[4-(1,3,5-trimethylpyrazol-4-yl)phenoxy]pyridine-2-carboxamide 1-N',2-N'-diethyl-3-methoxy-1-N,2-N'-bis[(4-methoxyphenyl)methylidene]propane-1,1,2-tricarbohydrazide N-(2-acetamidoethyl)-N-[4-(dimethylsulfamoyl)phenyl]-2-methoxyacetamide 3-chloro-4-hydroxybenzamide;6-methylspiro[1H-indole-3,2'-cyclopropane]-2-one N-[[4,5-bis(ethenyl)-1H-pyrrol-2-yl]methyl]-4-bromoaniline 5-[4-(1H-indol-2-yl)pyridin-3-yl]-1,6-dimethoxynaphthalen-2-ol (3R,4S)-4-(1H-indol-2-yloxymethyl)pyrrolidine-3-carboxylic acid (4S,5R)-5-[2,6-dimethyl-4-[5-phenyl-3-(trifluoromethyl)pyrazol-1-yl]phenoxy]-4-hydroxypentanamide 4-[[(2S)-3-ethyl-1-hydroxypentan-2-yl]carbamoylamino]benzamide 6-bromo-8-(1H-imidazol-2-yl)-2-methylimidazo[1,2-a]pyridine 5-(2,4-difluorophenyl)-N'-hydroxypyrazine-2-carboximidamide (3S)-1,3-diamino-4-[2-methyl-5-(1H-pyrrol-2-yl)phenyl]butan-2-one 3-methyl-4-[3-(oxolane-2-carbonylamino)piperidin-1-yl]benzoic acid N-(2-cyclohepta-1,4,6-trien-1-ylethyl)-3-methoxy-5-phenylpyrazine-2-carboxamide 4-chloro-2,6-diphenyldiazenylphenol 6-amino-1H-indazole-3-carboxamide;5-methyl-3-phenyl-2H-pyrazolo[3,4-c]quinolin-4-one 1-[(2Z,4E)-5-fluorohepta-2,4,6-trienyl]-6-(3-methoxyphenyl)imidazo[4,5-c]pyridine 3-[2-(diethylamino)propoxy]benzenediazonium 2-(4-chlorophenyl)-1-[2-(4-methylpiperazin-1-yl)ethoxy]cyclohexa-3,5-diene-1,3-dicarboxylic acid 4-[3-fluoro-2-(1H-pyrazolo[4,3-b]pyridin-5-yloxymethyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile (2R)-2-methyl-3-[6-[(1S,4R)-4-(trifluoromethoxycarbonylamino)cycloheptanecarbonyl]naphthalen-2-yl]propanoic acid 3-ethyl-4-propoxybenzaldehyde N-(1-bromoethyl)-N,4,5-trimethyl-2-nitroaniline 7-tert-butyl-N-diazoindole-1-sulfonamide 2-[(4-methoxyphenyl)methyl]-1,2,3,4-tetrahydroquinoline 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethanimine 4-benzyl-N-[[3-(oxan-2-yl)-1H-pyrazol-5-yl]methyl]piperazine-1-carboxamide N-[(1R)-1-(2,6-difluorophenyl)ethyl]-2-(5-pyridin-4-yl-1H-pyrrolo[3,2-b]pyridin-2-yl)acetamide 1-[3-[4-(6,7-dimethoxyquinolin-4-yl)pyrazol-1-yl]-2-hydroxypropyl]cyclohexan-1-ol 4-[(2R)-1-methoxybutan-2-yl]oxybenzamide 3-azidosulfanyl-5-methylsulfonylthiophene 1-(azidomethyl)-4-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfonylpiperazine N-[(2S)-3-amino-1-phenylbut-3-en-2-yl]benzamide N-[(1S)-1-cyclohexyl-2,4,6,7-tetramethyl-5-propan-2-ylnaphthalen-2-yl]acetamide 4-[2,3-dihydroxypropyl(hexadecanoyl)amino]benzenesulfonic acid 5-(dibutylamino)-3-[(2R,3S,4R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]sulfanyl-6H-triazolo[4,5-d]pyrimidin-7-one N-(1,3-thiazol-5-yl)-2,4,6-triazin-5-amine 2-[2,6-dichloro-4-(4-methylcyclohexa-1,3-dien-5-yn-1-yl)phenoxy]acetaldehyde 4-[(3-chloro-2,5-dimethoxyphenyl)sulfamoyl]benzoate 1-[4-(6,8-dihydro-5H-imidazo[5,1-c][1,4]oxazin-3-ylmethyl)-2,3-difluorophenyl]-N-methyl-1,2,4-triazol-3-amine N-cyclopropylsulfanyl-4-[[3-(1,2,3,6-tetrahydropyridin-4-yl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]methyl]benzamide N-(3-methoxypyridin-2-yl)-4,5-dihydro-1H-imidazole-2-carboxamide 5-[4-(furan-2-yl)phenyl]pyrimidine 3-[(2S)-1-aminopyrrolidin-2-yl]-5-azidooxyaniline 2-[4-(6-cyanopyridin-3-yl)oxy-3,5-difluorophenoxy]-N,N-dimethylpropanamide 1-[2-(dimethylamino)phenyl]heptan-3-ol (3-ethoxyphenyl)-[4-(7-fluoro-2,5-dimethylpyrazolo[1,5-a]pyridin-6-yl)piperazin-1-yl]methanone 2-[4-(2,3-dihydro-1H-pyrrole-2-carbonyl)phenoxy]acetic acid 4-[2-(6-hydroxy-3,7-dimethyloctoxy)phenoxy]butanenitrile 2-fluoro-N-[6-methyl-5-(4-propan-2-ylpyridin-3-yl)oxypyrimidin-4-yl]benzamide 4-[4-(2,3-dihydro-1H-inden-5-yl)-6-[2-(2-propoxyethoxy)ethoxy]pyridin-2-yl]morpholine 1-[2-[6-fluoro-7-(2-fluorophenyl)quinazolin-4-yl]pyrrolidin-1-yl]propan-1-one;hydrochloride 1-[4-[[2-(3,4-dichlorophenyl)quinolin-4-yl]amino]butyl]piperidine-2,6-dione 1-[4-bromo-2,5-dimethyl-N-(2H-tetrazol-5-yl)anilino]propan-2-one 3-methyl-6-methylidene-11H-benzo[c][1]benzoxepine 2-[3-cyclopropyl-5-(methylamino)anilino]phenol [(3S)-3-hydroxy-1-oxo-1,2-thiazolidine-2-carbonyl]oxy-diphenylsulfanium [(2S,4R)-1-acetyl-4-[2-[4-methoxy-3-(3-methoxypropylsulfonylamino)phenyl]imidazol-1-yl]pyrrolidin-2-yl]carbamic acid 2-[(4-aminopiperidin-1-yl)methyl]-3H-thieno[3,2-d]pyrimidin-4-one;dihydrochloride 3-[2-hydroxyethyl(methoxy)amino]oxycarbonyloxybenzoic acid 2-[[(3S)-6,8-dichloro-1-methyl-4H-chromeno[4,3-c]pyrazole-3-carbonyl]amino]acetic acid 2-[4-(3,5-difluoropyridin-2-yl)piperazin-1-yl]-N'-hydrazinyl-6-oxo-1H-pyrimidine-4-carboximidamide 1-[5-amino-4,6-bis(ethenyl)pyridin-3-yl]-3-(2H-tetrazol-5-yl)urea 6-[(Z)-1-amino-2-pyridin-4-ylethenoxy]-N-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-ylmethyl)pyrazin-2-amine (3R)-4-methyl-3-[(2,4,6-trihydroxyphenyl)sulfonylamino]pentanamide 6-azidooxy-4-(2-piperidin-1-ylethoxy)quinoline 1-[3,5-dichloro-4-(1H-indole-2-carbonyl)phenyl]propan-1-one 2-[1,3-bis(2,4,6-trimethylphenyl)imidazolidine-2-thioyl]cyclohexane-1-carboxylic acid [6-bromo-2-chloro-3-(methylamino)phenyl]-[4-(1,1,1-trifluoropropan-2-yl)piperazin-1-yl]methanone;butane;ethene 3-[5-fluoro-2,6-dimethyl-4-(3-phenylpropoxy)phenyl]-1-morpholin-4-ylbutan-1-one 6-bromo-N-(2,6-dimethylphenyl)naphthalene-1-carboxamide 3,4-diamino-N'-(6-phenylhexyl)benzenecarboximidamide 1-[(2S)-2-[[4-(2-aminoethylsulfonyl)piperazin-1-yl]methyl]pyrrolidine-1-carbonyl]-7-chloroisoquinoline-6-carboxamide;dihydrochloride 3-[2-(2,6-dichloro-4-nitrophenyl)pyrazol-3-yl]oxy-N,N-dimethylpropan-1-amine 4-hydroxy-2,6-dioxo-1H-pyrimidine-5-sulfonamide 2-[6-[4-(methylamino)butoxy]naphthalen-2-yl]acetaldehyde 1-N',3-N'-bis(ethenyl)-5-fluoro-2-methoxybenzene-1,4-diamine [3-(2,5-difluorophenyl)phenyl]-pyrrolidin-1-ylmethanone;ethane 2-ethyl-4,5-dimethoxybenzamide 2-(1-aminoethyl)-N,N-dibutyl-3H-benzimidazole-5-sulfonamide 2-[(6S)-2-(4-chlorophenyl)-5-oxo-4,6-dihydroimidazo[1,2-b]pyrazol-6-yl]-N-(3,4-dimethoxyphenyl)acetamide 2-[[3-[[4-(difluoromethoxy)phenyl]sulfonylamino]benzoyl]amino]butanedioic acid 3-(4,5-difluoro-2-methoxyphenyl)-3-oxopropanenitrile 1-(cyclopropylmethylamino)-3-(5,8-difluoroquinolin-4-yl)oxypyrrolidine-2,5-dione (6S)-2,3,10-trimethoxy-6H-cyclopenta[c]chromene ethane;2-(7-fluoro-1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carbonyl)cyclohex-2-en-1-one 1-[(3-methylthiophen-2-yl)methylamino]hexan-2-one (2Z)-3-[4,5-bis(ethenyl)furan-2-yl]-N-methyl-3-hydroxyimino-2-phenylpropanamide 3-(4,5-dimethoxy-2-nitrophenyl)cyclopropane-1,1,2,2-tetracarbonitrile N'-[4-(3-bromophenoxy)pyridin-2-yl]-N,N'-dimethylethane-1,2-diamine N-ethyl-N-methyl-3,4-dihydro-2H-chromene-3-carboxamide 2-[2-(cyclobutylmethoxy)-5-fluorophenyl]-4H-1,3,4-oxadiazin-5-one 6-[2-[6-(4-methoxybutyl)pyridin-3-yl]ethynyl]-1,3-benzothiazol-2-amine [3-(3,5-diamino-6-bromopyrazin-2-yl)-5-phenylmethoxyphenyl]methanol 1-[4-(2-hydroxyphenyl)piperazine-1-carbonyl]piperidine-3,6-dicarboxylic acid 1-(3,4-dimethylphenyl)sulfonyl-N-[2-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl]piperidine-3-carboxamide (5-chloro-3-methylpyridin-2-yl)-pyrrolidin-1-ylmethanone 1-[2-(3,4,5-trimethoxyphenyl)cyclopropanecarbonyl]pyrrolidine-2-carboxylic acid N-[4-[3-(2,6-difluorophenoxy)azetidine-1-carbonyl]phenyl]-5-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide 1-methyl-6-oxo-N-[(2S)-3,3,5,7-tetrahydroxyheptan-2-yl]pyridazine-3-carboxamide 3-[4-(2,6-difluorophenyl)-5-hydroxytetrazol-1-yl]cyclopentane-1-carboxylic acid 3-[(4,5-dimethyl-1H-pyrazol-3-yl)methylidene]azete (5R)-2-[(2-chlorophenyl)methylsulfanyl]-5-(4-ethoxyphenyl)-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione N-[2-(6,7-dimethoxyquinolin-4-yl)ethyl]-3-[1-[(Z)-methylideneamino]oxyethenyl]benzamide (3E,5Z)-6-amino-2-[7-(difluoromethyl)imidazo[1,2-a]pyridin-3-yl]nona-3,5,7-trienoic acid 5-[6-azido-4-(4-fluorophenyl)-3,5-dimethylpyridin-2-yl]-1H-indazole N-[(2S)-1,3-dihydroxypropan-2-yl]-3,3a,4,9b-tetrahydrofuro[3,4-c]chromene-1-carboxamide N-[2,4-difluoro-3-(triazol-1-yl)phenyl]-4-fluorobenzamide;ethane N-(2,3-dihydro-1H-inden-5-yl)-4-methoxy-2-[(E)-2-nitroethenyl]benzamide N-[4-(cyclopropylamino)pyridine-2-carbonyl]propanamide (5R)-3-[2,6-dimethyl-4-[(E)-[4-oxo-2-sulfanylidene-1-(thiophen-2-ylmethyl)azetidin-3-ylidene]methyl]phenyl]-5-methylimidazolidine-2,4-dione 3-amino-4-(2-azidoanilino)butanal N-cyclopropyl-3-[6-(4,4-difluoropiperidin-1-yl)pyridin-3-yl]-4-methoxybenzamide N-[3-[(1R)-6,8-dichloro-2-methyl-9b-(4-phenylmethoxyphenyl)sulfonyl-2,3a,4-trihydro-1H-pyrano[2,3-b]indole-3-carbonyl]phenyl]methanesulfonamide 1-[2-(dimethylamino)pyrimidin-4-yl]-N-piperidin-3-ylindazole-5-sulfonamide;hydrochloride 3-[(5-methylthiophene-2-carbonyl)amino]-N-(1-pyrazin-2-ylazetidin-3-yl)benzamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]benzonitrile 2-[4,5-bis(ethenyl)-1H-imidazol-2-yl]pyridine;methanamine 2-[5-[(3,4-diethylphenyl)methoxy]piperidin-2-yl]ethanol 3,4-dichloro-N-(5-chloro-2-pyrrolidin-1-ylphenyl)-2-nitrobenzenesulfonamide 6-chloro-N-[3-(difluoromethoxy)phenyl]quinoline-8-carboxamide 2-(4-chlorophenyl)-1-[(3S,4R)-3-methylpiperidin-4-yl]-N-(oxan-2-yloxy)indole-5-carboxamide 3-[2-(6-cyclopropylpyridazin-3-yl)-1,3,3a,4,5,7,8,8a-octahydropyrrolo[3,4-d]azepine-6-carbonyl]benzonitrile 3-(2,2,4,6,7,8-hexamethyl-1H-naphthalen-1-id-5-yl)-N-phenylaniline;uranium(2+) 2-bromo-5,6-dimethoxy-1H-carbazole 2-[4-(methylamino)naphthalen-1-yl]oxyacetic acid 4-(cyclopropanecarbonylamino)pyridine-3-carboxamide N-[4-(2,6-difluorophenyl)-5-[2-(dimethylamino)ethoxy]pyridin-2-yl]hydroxylamine [7-amino-3,5-bis(4-hydroxyphenyl)pyrazolo[1,5-a]pyrimidin-6-yl]methylidene-pyridin-2-ylazanium [3-azido-1,5-dimethyl-6-(4-phenylbutoxy)indol-2-yl]-(4-chlorophenyl)methanone N-azido-1-ethylindazole-3-carboxamide [(2S,3R)-6-oxo-8-[5-(trifluoromethylsulfanyl)pyridin-2-yl]oxy-7H-purin-1-ium-2-yl]hydrazine 3-[2,6-bis(2,4-dimethylpentanoyloxy)phenyl]propanoic acid 4-[(2,5-dichloropyrimidin-4-yl)amino]benzoic acid 2-[(4-chloropyridin-3-yl)methyl]-5-methoxypyridazin-3-one 3-amino-2,6-dichloro-N'-(4-methoxyphenyl)benzenecarboximidamide;5-aminosulfanyl-6-chloro-3-ethyl-1H-benzimidazol-2-one 3-[(1R,2S)-2-pyridin-4-ylcyclopropanecarbonyl]benzenesulfonamide 1-(3-azidopropoxy)-4-chlorobenzene 1-[2-[2-(4-methoxyphenyl)imidazol-1-yl]propanoyl]pyrrolidine-3-carboxylic acid 7-hydroxy-1,8-dimethyl-3H-purine-2,6-dione N-[(1S)-2,3-dihydro-1H-inden-1-yl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide (Z,2S)-4-[3-chloro-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]oxybut-3-en-2-amine [2-(3,5-dimethyl-1,2-oxazol-4-yl)pyridin-4-yl]methanamine;ethane (3S,4R)-1-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-N,2-dimethylpyrrolidine-3-carboxamide 2-(dimethylcarbamoylamino)-N-[3,5-bis(trifluoromethyl)phenyl]acetamide 2-[[(3R,5S)-1-acetylpiperidine-3-carbonyl]amino]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid 4-[(1-ethylpyrazol-3-yl)methylamino]-6-[3-oxo-3-(phenylmethoxyamino)propyl]pyridine-2,5-dicarbonitrile [3-amino-6-(3,4-dihydroxyphenyl)pyrazin-2-yl]-piperidin-1-ylmethanone N'-(3,4-dimethylphenyl)pentanimidamide;ethane 2-[7-amino-3-(4-chlorophenyl)imino-4,5-dihydropyrazolo[1,5-a]pyrimidin-5-yl]phenol 2-[(4-azidonaphthalen-1-yl)oxymethyl]-1,3-thiazole 3-amino-4-cyano-5-(2-fluoro-6-methoxyphenyl)-1H-pyrrole-2-carboxamide N-methyl-1'-pyridin-3-ylspiro[4,5-dihydrothieno[2,3-c]pyran-7,4'-piperidine]-2-carboxamide N-[2-[(2Z)-3,7-dimethylocta-2,6-dienoxy]propan-2-yl]pyridin-4-amine (2-azidooxyphenyl)sulfanium 5-[1-(4,6-diphenylpyrimidin-2-yl)cyclohexa-2,4-dien-1-yl]benzimidazolo[1,2-a]quinoline N-[(1R)-2,3-dihydro-1H-inden-1-yl]-6-(2-methoxypyrimidin-5-yl)pyridine-3-carboxamide 2-(3-methylbutanoyl)benzenesulfonic acid 2,2-dimethyl-N-[3-(1H-pyrazol-4-yl)phenyl]cyclopropane-1-carboxamide 3-chloro-N-[4-(4,5-dihydroimidazol-1-yl)-2,6-difluorophenyl]benzamide (5E)-2-(4-methoxyphenyl)imino-5-[[1-(3-nitrophenyl)pyrrol-2-yl]methylidene]-1,3-thiazolidin-4-one (4S)-1,3-dimethyl-4-[2-methyl-5-(trifluoromethyl)phenyl]-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one (1E,4Z)-1-(6-aminopyridin-2-yl)-5-fluoropenta-1,4-dien-3-one 1,3-bis[2-(dimethylamino)ethyl]-4H-pyrimido[5,4-d]pyrimidine-2,7-dione;trihydrochloride 5-azido-2-(3,5-dichlorophenoxy)quinoline 2-[(4-azidopiperazin-1-yl)methyl]-7,8-dihydrofuro[3,2-e]benzimidazole (1S,3R)-N-[(2R)-1-(4-methoxyanilino)-3-naphthalen-2-ylpropan-2-yl]-3-[5-oxo-3-phenyl-6H-1,2,4-triazin-6-yl]cyclohexane-1-carboxamide 5-amino-7-(3,4-dimethylphenyl)-8H-[1,2,4]triazolo[4,3-c]pyrimidine-3-thione 5-chloro-6-(dimethylamino)-N'-hydroxypyridine-2-carboximidamide 5-methoxy-1'-[2-(4-oxo-3H-quinazolin-2-yl)acetyl]spiro[1,3-dihydroindene-2,4'-piperidine]-1-one 1-[1-(4,6-dimethylpyrimidin-2-yl)azetidin-3-yl]-N-[(2,5-dimethylpyrazol-3-yl)methyl]cyclobutane-1-carboxamide (4R)-N-[1-(4-chlorophenyl)cyclopropyl]-6-[3-(1,2,5-oxadiazol-3-yl)pyrazol-1-yl]-3,4-dihydronaphthalene-2-carboxamide 3-[3,5-dimethyl-1-(4-methylsulfanylphenyl)pyrazol-4-yl]-1H-pyrrolo[2,3-b]pyridine 2-[(3R)-4,4-difluoropiperidin-3-yl]oxy-5-methylsulfonylbenzamide N-[2-[3-(dimethylamino)propoxy]-4,5,6,7-tetrahydro-1-benzothiophen-3-yl]formamide (2-amino-1,3-dihydroisoindol-4-yl)-[4-[[5-fluoro-2-(methylamino)phenyl]methyl]piperazin-1-yl]methanone 3-chloro-1H-indole-2,7-disulfonic acid 3-(1H-indole-2-carbonylamino)propanoic acid;1,4-xylene 5-chloro-2-[4-(chloromethyl)phenyl]pyridine 2-benzylsulfanyl-4-[(E)-4,5-dihydroxypent-3-enyl]-6-pyridin-3-ylpyridine-3-carbonitrile 2-(3,5-dimethoxyphenyl)-N'-[6-(4-fluorophenyl)-8H-pyrido[3,2-d]pyrimidin-7-yl]ethanimidamide 2-(6-methylpyrazolo[4,3-c]pyridine-1-carbonyl)spiro[5H-furo[3,4-b]pyridine-7,4'-piperidine]-4-one 2-[4-(5,6-dihydrobenzo[h]quinazolin-7-ylamino)cyclohexanecarbonyl]benzoic acid N'-hydroxy-4-[2-[3-(2H-tetrazol-5-ylmethoxy)propylamino]ethylsulfanyl]pyridine-2-carboximidamide 2-chloro-4-[6-fluoro-1-[(2E,3Z)-2-hydroxyiminohexa-3,5-dienyl]indol-3-yl]phenol [3-(4-aminoanilino)cycloheptyl]methanol [5-amino-1-(2-butylphenyl)pentan-3-ylidene]azanium 6-hydroxy-5-(2,3,4-trifluorophenyl)-3H-2-benzofuran-1-one 1-[5-(cyclopropylmethoxy)-6-[4-methoxy-2,3-bis(trifluoromethoxy)phenyl]pyridine-2-carbonyl]pyrrolidine-3-carboxylic acid 2-[(6-bromopyridin-3-yl)methoxy]ethanol 4-N,6-diethyl-2-(5-phenylpyrazin-2-yl)pyrimidine-4,5-diamine;propane 4-[(1,3-dimethyl-6-nitrobenzimidazol-2-ylidene)amino]phenol 7-(4-bromophenyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine [2-fluoro-6-methyl-4-(8,12,12-trimethyltridecoxymethyl)phenyl]methanol N-(2-aminoethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide [4-(hydroxymethyl)piperidin-1-yl]-[5-(methoxymethyl)furan-2-yl]methanone N-[4-fluoro-3-(trifluoromethyl)phenyl]-1-(2-methoxyethyl)-6-(1,3-oxazol-5-yl)pyrazolo[3,4-b]pyridine-4-carboxamide N-[2,3-bis(methylimino)propanoyl]-4-(ethoxyamino)benzamide 4-azidooxy-N'-phenylbenzenecarboximidamide 5-(2-methylpyridin-4-yl)-3-[6-(trifluoromethyl)pyridin-2-yl]oxypyrazolo[1,5-a]pyrimidine (4-aminophenyl)sulfonyliminomethylideneazanide 2-(2,6-diethylphenoxy)-1H-indene;ethane 1-(3,5-dichloro-4-hydroxyphenyl)-N-[6-(dimethylamino)pyridin-2-yl]ethanesulfonamide 2-[1-(3,4-difluorobenzoyl)piperidin-4-ylidene]propanoic acid 3-amino-4-[5-(2,6-diphenylpyrimidin-4-yl)cyclohepta-1,4,6-trien-1-yl]benzoic acid N-[2,3-dimethyl-5-(2-methylpropoxy)phenyl]formamide N'-[amino(sulfamoyl)methylidene]benzenecarboximidamide (7E)-2-[2-[(1,3-dioxoisoindol-4-yl)amino]ethoxy]imino-7-(3,3-dimethoxypropylidene)chromene-4-carboxylic acid 1-(2,2-difluorobutyl)-N'-(6-ethynylpyrimidin-4-yl)-3H-pyrazolo[3,4-c]pyridine-6-carbohydrazide 2-[3,5-bis(trifluoromethyl)phenyl]-1-diazenylguanidine 2-(2,4-difluorophenyl)sulfanyl-N'-hydroxypyridine-4-carboximidamide (Z)-2,3-bis[[5-(furan-2-yl)thiophen-2-yl]methylideneamino]but-2-enoic acid 3-(4,5-dichloro-2-hydroxyphenyl)-1H-pyrazole-5-carboxylic acid 4-[(2R)-1-aminopentan-2-yl]oxy-6-cyclopropylpyridine-3-carboxamide 4-[(2-butyl-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-4-yl)oxy]aniline N'-(6,7-dichloro-2H-chromene-3-carbonyl)thiophene-3-carbohydrazide 5-[(2R)-2,4-dimethylpentoxy]-3-[6-fluoro-1-methyl-2-[(2S)-oxolan-2-yl]indol-3-yl]pyrazin-2-amine N-[6-(3,4-dihydro-2H-chromen-7-ylamino)pyrimidin-4-yl]methanesulfonamide 5-ethyl-4,6-dimethoxypyrimidine;5-[2-(6-hydroxy-7H-pyrrolo[3,2-d]pyrimidin-4-yl)thiophen-3-yl]pentanenitrile 4-N,6-N-bis[(Z)-(2-ethoxyphenyl)methylideneamino]pyrimidine-2,4,5,6-tetramine (2S,3R)-N,1-diethyl-5-oxo-N-propanoyl-3-[[(1E,3Z)-4-pyridin-4-ylbuta-1,3-dienoxy]methyl]pyrrolidine-2-carboxamide 3-[6,7-dihydroxy-2-(4-methoxyphenyl)chromen-4-ylidene]piperidine-2,4-dione 5-chloro-N-methyl-1,2-dihydrophenazine-2-carboxamide 3-(1,3-benzothiazol-6-ylamino)cyclobutan-1-ol 2-ethyl-5-[1-(2,3,4-trifluorophenyl)propan-2-yl]pyridine 2-[(1R)-2,3,4,6-tetrahydropyrrolo[3,4-c]pyrrole-5-carbonyl]pyridine-3-carboxylic acid;hydrochloride 3-[[4-chlorobutyl(naphthalen-1-yl)amino]methyl]phenol 1-azidooxy-3-(4,5-dimethyl-2-phenylmethoxyphenyl)propan-2-ol (3R)-2-[(4,6-dimethylpyrimidin-2-yl)carbamoylamino]-N'-[6-[4-(trifluoromethoxy)phenyl]pyridazin-3-yl]pentanediamide 3-methoxy-4-[[2-methyl-1,6-di(piperidin-4-ylidene)hexan-3-yl]oxymethyl]benzoic acid (5S)-1-ethyl-2-oxo-3,4,6,7-tetrahydropyrimido[2,1-c][1,4]oxazine-10-carboxamide 1-[2,6-difluoro-4-(2H-pyridin-1-ylmethoxy)phenyl]pyrrolidine-3-carboxamide 3-(3,5-dichlorophenyl)-N-[(3R,4S,6S)-3-methyl-2,3,4,9-tetrahydro-1H-carbazol-1-yl]propanamide N-ethylsulfonyl-3-(4-methoxyphenyl)-2-[8-oxo-2,7-bis(prop-1-en-2-ylsulfanyl)purin-9-yl]propanamide 2-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-5-N-methylpyridine-2,5-dicarboxamide N-(3,4-dichlorophenyl)-2-(1H-imidazol-5-ylmethylidenehydrazinylidene)propanamide 2-chloro-6-[3-[(4-fluorophenyl)methyl]benzimidazol-5-yl]pyridine-3-carboxylic acid N-[(4S)-1,3-oxazolidin-4-yl]-5-[3-(trifluoromethoxy)phenyl]naphthalene-2-sulfonamide 2-[5-(3,4-dimethoxyphenyl)thiophen-2-yl]-N-[[1-hydroxy-3-(4-nitrophenyl)propan-2-ylidene]amino]acetamide 4-ethenyl-5-methoxy-N,6-diphenylpyridine-3-carboxamide 2-[azido(phenyl)methyl]-3-bromo-1H-indole N-(6-bromo-1H-indazol-3-yl)formamide;2,4,5-trimethyl-1,3-oxazole 2-[(E)-[1,3-dihydroxy-4-oxo-2-sulfanyl-6-(trifluoromethoxy)anthracen-9-ylidene]methyl]naphthalene-1,5-disulfonic acid 1-(2,4-dichlorophenyl)-3-methylazetidine 1-(cyclopropylmethyl)-3-[(4-methoxyphenyl)methylamino]thiourea (3aR,6aS)-5-cyclobutyl-2-[3-(3-methoxyphenyl)pyrazole-1-carbonyl]-3a,4,6,6a-tetrahydropyrrolo[3,4-d][1,3]oxazol-7-one 6-(1H-indol-3-yl)-2-[2-(4-pyrrolidin-1-ylphenyl)ethyl]pyrimidin-4-amine 2-(diaminomethylideneamino)-N-ethyl-N'-[4-(trifluoromethyl)phenyl]butanimidamide 1-cyclohexyl-3-(2,4-difluorophenyl)urea 2-[1-(4,5-dihydrobenzo[g]indol-1-yl)propan-2-ylideneamino]guanidine;tetrahydrochloride 3-[4-(1H-pyrazol-5-yl)piperidine-1-carbonyl]benzonitrile 3-[(E)-3-[4-hydroxy-5-(7-methoxyquinolin-2-yl)furan-2-yl]prop-2-enoyl]piperidine-1,6-dicarboxylic acid N-benzyl-4-methoxy-6-(3,3,3-trifluoropropoxy)pyridine-2-carboxamide 7-[(1-azidonaphthalen-2-yl)oxymethyl]phenanthrene-9,10-dione 5-[2-(4-fluorophenyl)ethynyl]-N-hydroxypyridine-3-carboxamide 2-[(E)-3-[(5R)-3,5-dimethyloxan-4-ylidene]prop-1-enyl]-1H-indole 1-(azidomethyl)-3,6,7-trichloropyrazolo[4,3-c]pyridine 2-[(3Z,5E)-hepta-1,3,5-trien-4-yl]oxy-N-pyridin-4-ylpyridine-3-carboxamide (5R)-2-[(Z)-(3,4-dimethoxyphenyl)methylidenehydrazinylidene]-5-propan-2-yl-1,3-thiazolidin-4-one N-[2,4-difluoro-3-[2-(4-iodoanilino)thieno[3,2-d]pyrimidine-7-carbonyl]phenyl]pyrrolidine-1-sulfonamide 5-[4-(4-cyclopropylpiperazin-1-yl)-2-methoxyphenyl]-3-(2,6-dichloro-4-iodoanilino)-1-methylpyrazin-2-one 4-[(2R)-2,3,3a,8b-tetrahydro-1H-cyclopenta[b][1]benzofuran-6-yl]pyrimidine 2-(methylcarbamoyl)-3,4,5,6-tetrahydro-1H-pyrrolo[3,4-b]pyrrole-4a-carboxylic acid 4-(4-chloro-3,5-dimethylphenoxy)-2,6-dioxopyrimidine-1-carbonitrile ethane;3-(5-fluoro-1H-indol-2-yl)-6,8-dimethoxy-7-methylchromen-4-one 4-(2,3-difluorophenyl)-N,1,5-trimethylpyrazole-3-carboxamide N-(3,4-difluorophenyl)-5-(6,8-dimethyl-7-oxopteridin-2-yl)-6-hydroxynaphthalene-1-carboxamide 2-[4-(6-methyl-1,3-benzothiazol-2-yl)piperidine-1-carbonyl]benzamide 2-(4,5-dimethylpyridin-3-yl)-6-[3-[(2R)-pyrrolidin-2-yl]propoxy]-1H-benzimidazole N-[4-chloro-2-(trifluoromethyl)phenyl]-2-[3-(5,6-dioxo-1H-pyrazine-3-carbonyl)phenyl]acetamide 3-bromo-2-hydroxybenzenesulfonate 2-(5,6-difluoroindol-1-yl)ethanethiol 2-tert-butyl-1,9-dihydropurin-6-one N-[2-(6-chloro-7-fluoroimidazo[1,2-a]pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carboxamide 4-(3-aminophenyl)-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-2-amine 1-azido-3-methyl-N-[3,4,5-trifluoro-2-(2,2,2-trifluoroethoxy)phenyl]pyrrolidine-3-carboxamide (E)-3-[4-(3,5-ditert-butylphenyl)sulfanyloxy-3-methyl-2-nitrobenzoyl]oxyprop-2-enoic acid 1-[[6-(3,4-dichlorophenyl)pyrimidine-4-carbonyl]amino]-N-(2-morpholin-4-ylethoxy)pyrazole-3-carboxamide (E)-4,8-dihydroxy-6-methylidene-3-phenylnon-5-enal;N-[3-(ethylaminosulfanyl)phenyl]-2,7-bis(4-methoxyphenyl)quinazolin-4-amine 4-[1-(3-ethoxypropyl)piperidin-4-yl]-2-pyridin-4-yl-1,3-thiazole;dihydrochloride 5-(3,4-difluorophenyl)-N'-[4-(2-methylsulfanylpyrimidin-4-yl)phenyl]pentanehydrazide N-[2,5-dimethyl-4-(3-methyl-2H-indazol-6-yl)phenyl]cyclohexa-1,3-diene-1-sulfonamide 3-[(1,6-dibenzylpiperidin-4-ylidene)methyl]-2-hydroxybenzoic acid ethane;3-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]isoquinoline 2-methyl-4-(1,3-thiazol-5-yl)benzenesulfonamide 7-[5-fluoro-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]pyrrolo[2,1-f][1,2,4]triazin-4-amine 4-[(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)amino]benzonitrile;1,3-thiazole 3-hydroxy-N'-methylbenzohydrazide (1E)-4,6-diamino-8-[6-(2,3-dihydro-1H-inden-5-yl)pyrazin-2-yl]-7-methyl-1-propan-2-ylidenedecan-10-one 2-azido-5-pyridin-3-ylpyrazine N-ethyl-2-[4-(quinolin-8-ylsulfonylamino)phenoxy]acetamide 2-(5-chloro-1H-indol-3-yl)benzo[g][1]benzofuran 1-[3-(azetidin-1-yl)-1,2-oxazol-5-yl]-6-chloro-7,8-difluoro-4-oxoquinoline-3-carboxylic acid 6-(6-cyclobutyloxypyridine-3-carbonyl)-N,N-dimethyl-6-azaspiro[2.5]octane-8-carboxamide 2-[6-methoxy-5,10-dioxonaphtho[1,2-g][1]benzofuran-2-ylidene]propanedinitrile 4-azidooxy-7-methoxyquinoline (E)-3-(3,5-dimethoxyphenyl)-1-[4-(1H-indole-2-carbonyl)piperazin-1-yl]prop-2-en-1-one 5-[(2,4-difluorophenyl)methyl]-N-(1H-indazol-3-ylsulfonyl)-1,3,4-thiadiazol-2-amine 1-ethyl-5-methoxybenzimidazole;5-hydroxy-3,4,6-triiodobenzene-1,2-dicarbonitrile 2-[(2,3,4-trihydroxyphenyl)methylideneamino]-1,6-naphthyridine-5-carbonitrile 4-[1,4-dihydroxy-2-(3-phenylmethoxycyclobutyl)ethyl]benzonitrile 1,3-dicyclopentyl-N-[(4R)-4-methoxyoxolan-3-yl]indole-5-carboxamide 1-[4-(cyclopentylmethoxy)phenyl]-2-pyridin-4-ylethanone 1-[5-ethylsulfonyl-6-[7-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]pyridin-3-yl]cyclopropane-1-carbonitrile 3-chloro-4-(dimethylamino)-N'-hydroxypyridine-2-carboximidamide 2,4-ditert-butyl-6-[(E)-2-(1H-imidazol-5-ylmethylsulfanyl)ethenyl]benzaldehyde 3-(5,6-difluoropyridin-2-yl)-6-methyl-1-pyridin-4-ylindole 2-[4-(aminomethyl)phenyl]-N-carbamoylacetamide 2-[4-chloro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-8-ethoxy-1-methylimidazo[1,2-a]pyrazine 2-[6-(4-hydroxyphenyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]phenol N-ethyl-5-(3-methoxypyridine-2-carboximidoyl)-4-piperidin-1-ylpyrimidin-2-amine 3-(4-bromophenyl)sulfonyl-2,2,6-trimethylmorpholine 1-[5,7-difluoro-2-(4-fluorophenyl)-3-methylquinolin-6-yl]-N-methoxy-1-phenylmethanimine 6-[4-(3,5-dimethylbenzenecarboximidoyl)piperazin-1-yl]-N-(3,4-dimethoxyphenyl)pyrimidin-4-amine 3-[4-(2,3-dichlorophenyl)butanoyl]piperidine-1-carboxylate 5-(2,6-dimethoxyphenyl)-4,8-bis[(3R)-pyrrolidin-3-yl]oxyquinoline 4-[2,6-dimethyl-3-(6-oxo-1H-pyridazin-3-yl)anilino]piperidine-1-carboxylic acid (4-iodo-1H-indol-2-yl)urea 3-[(4,5-dimethylimidazol-1-id-2-yl)methoxy]propanamide;palladium(2+);triphenylphosphane 3-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N-[3-chloro-4-[4-(pyrrolidine-1-carbonyl)piperazin-1-yl]phenyl]benzamide 3-(9H-fluoren-1-yloxy)cyclohexan-1-one 2-[(2,5-dimethylphenyl)sulfonylamino]-N-[(Z)-(3-ethoxy-4-hydroxyphenyl)methylideneamino]benzamide 3-amino-5-(3,4-dichlorophenyl)-2-methylhexanoic acid 3-(5-methoxy-2,4-dimethylphenyl)propanoic acid ethane;(3S)-N-ethyl-7,9-dihydroxy-2-imino-6-methoxy-1-oxo-3H-benzo[f]isoindole-4-carboxamide N-[6,7-dichloro-1-(hydroxymethyl)isoquinolin-5-yl]acetamide N-(6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-ylmethyl)propanamide 2-[4-(3,5-dimethoxyphenyl)-1H-benzimidazol-2-yl]-7-(furan-3-yl)-5-methyl-1H-imidazo[4,5-b]pyridine N-(3-aminopropyl)-2-[4-benzamido-5-ethyl-3,6-bis(ethenyl)cyclohexa-1,3-dien-1-yl]acetamide 5-[5-(azidomethyl)naphthalen-2-yl]oxypyridine-3-carbonitrile 2-[4-[(5R)-4,5-bis(hydroxymethyl)-1,3-oxazolidin-3-yl]-2-fluorophenyl]sulfanyl-4-methyl-1H-pyrimidin-6-one N'-hydroxy-2-[4-(1H-pyrrol-3-ylmethylideneamino)phenyl]-2,3-dihydro-1H-indene-5-carboximidamide 1,4-difluorobenzene;N-(3,5-dimethoxyphenyl)sulfonylformamide 6-cyclopropyloxy-N,3-dimethylpyrazolo[1,5-a]pyridine-2-carboxamide 2-amino-7-[4-(trifluoromethoxy)phenyl]pyrrolo[1,2-b]pyridazine-3-carboxylic acid 3-[5-oxo-2-(trifluoromethyl)-4H-thiochromeno[3,4-c]pyrazole-3-carbonyl]-1-(3-pyrrolidin-1-ylpropyl)pyridin-2-one 6-methyl-4-(5-propan-2-ylpyridin-3-yl)pyrido[3,2-b][1]benzazepine 4-(4-methylphenoxy)benzoic acid;propane (2Z)-N',N'-diethyl-1-[3-(trifluoromethyl)phenyl]penta-2,4-dienimidamide 1-(4,4-difluorocyclohexyl)-6-[[(3R)-5-hydroxy-1-pyridin-2-ylsulfonylpyrrolidin-3-yl]methoxy]imidazo[4,5-b]pyridine-7-carboxamide 2-(difluoromethyl)-4,6-bis(3-fluorophenyl)pyrimidine 1,5-bis[4-(dimethylamino)-2-(4-hydroxyphenyl)butyl]-3-iodopyrazole-4-carbonitrile 2-[6-[(1S,3R)-3-[methyl-(6-oxo-7H-purin-8-yl)amino]cyclopentanecarbonyl]pyridin-2-yl]benzoic acid [5-tert-butyl-4-methoxy-2-(3-oxo-1,2-oxazol-5-yl)phenyl]carbamic acid N-benzyl-4,7-diphenylpyrrolo[2,3-d]pyrimidin-2-amine N-[3-[5-(cyclohexylmethoxy)pyrimidin-2-yl]phenyl]methanesulfonamide (1S)-3,4,4-trimethyl-2-(2-phenoxyethoxycarbonyl)cyclopentane-1-carboxylic acid 2-N-[(3Z)-4-(propan-2-ylamino)hepta-1,3-dien-2-yl]-5-(trifluoromethyl)pyridine-2,4-diamine 4-fluoro-3-[4-(4-methylphenyl)butoxy]aniline 3-[2-(1,1-dimethylcyclopropanecarbonyl)oxyethyl]benzoic acid (2S)-1-[4-chloro-3-[(1R,5Z,7E)-7,8-difluorocycloocta-1,5,7-trien-1-yl]sulfonylanilino]propan-2-ol [4-[[5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazol-4-yl]methoxy]piperidin-1-yl]-(1H-indol-2-yl)methanone 1,3-diethyl-5-phenylpyrazol-4-ol 4-(2,3-dimethylphenyl)butanamide 6-(3,4-difluorophenyl)-2-[4-(1H-pyrrolo[2,3-b]pyridin-5-ylamino)piperidine-1-carbonyl]pyridazin-3-one (NE)-N-[1'-[2-[4-chloro-5-(trifluoromethyl)pyrimidin-2-yl]oxyethyl]spiro[cyclopropane-1,3'-pyrrolo[2,3-c]pyridine]-2'-ylidene]hydroxylamine 3-cyclohexylsulfonylaniline 5-(2,3-dimethylquinoxaline-6-carbonyl)-2-[(4S)-3,3-difluoro-1-methylpiperidin-4-yl]oxypyridine-3-carbonitrile 7-(3,4-dimethoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine 3-[2,6-di(propan-2-yl)phenyl]-1H-indole 5-[[(5S)-3,4-diazabicyclo[3.2.0]heptan-5-yl]methoxy]-6-fluoro-1H-quinolin-2-one 2-hydroxy-6-[(4-methylphenyl)sulfonylamino]benzoic acid 1-methyl-N-(4-phenoxybutan-2-yl)cyclopropane-1-sulfonamide 2-azidooxy-1,3,4-trinitrobenzene 5-amino-N-[2-chloro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyrazine-2-carboxamide 2-[2,4-dichloro-6-(furan-3-ylmethyl)phenyl]acetaldehyde N-[2,4,5-trichloro-3-(trifluoromethyl)phenyl]acetamide 2-[(5R,10bS)-7-methoxy-5-pyridin-3-ylsulfanyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-chlorophenol (2S)-N-[1-amino-4-(3,5-dichlorophenyl)-1,1-dioxothian-4-yl]-2-azido-2-benzamidoacetamide (4R)-4-[[2,3-difluoro-6-(3,5,6-trimethylpyrazin-2-yl)phenyl]methoxy]pyrrolidin-2-one 2-chloro-4-(4,4-dimethylazetidine-1-carbonyl)benzonitrile 5-[6-(2,4-difluorophenyl)pyridin-2-yl]-N-methoxy-1H-pyrazole-3-carboxamide 4-[(2S)-4,6-dihydroxyoxan-2-yl]-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 1-azidooxy-N,4,5-trimethyl-3-phenylpyrazole-3-carboxamide 4-[(Z)-3-(3,6-dimethoxycyclohexa-1,5-dien-1-yl)-2-pyridin-4-ylprop-2-enoyl]benzaldehyde 1-[5-[[(2R,3S)-2-(1H-pyrazol-4-yl)oxolan-3-yl]methoxy]pyridin-2-yl]pyrrolidin-2-one 7-(2,4-dimethylphenyl)pyrrolo[1,2-a]pyrazine 3-(cyclopropylmethoxy)-N'-hydroxypyridine-4-carboximidamide 5-[2-(4,6-dihydroxy-3-oxo-1H-isoindol-2-yl)ethoxycarbonyl]thiophene-3-carboxylic acid 6-(4-bromophenyl)sulfonyl-2,3-dihydro-1H-azepine 3-[2,6-dimethyl-4-(trifluoromethyl)phenyl]-1-[[7-[4-(morpholine-4-carbonyl)anilino]pyrazolo[3,4-d]pyrimidin-4-yl]amino]propan-2-one 2-[(6R)-3-ethylsulfanyl-6-thiophen-2-ylthieno[2,3-b]pyridine-4-carbonyl]oxyacetic acid N-(1H-benzimidazol-2-ylmethyl)-7-hydroxy-6-(5-thiophen-3-ylfuran-2-yl)-4,7-diazaspiro[2.5]octane-4-carboxamide;2,2,2-trifluoroacetic acid (2E)-N-[5-(3,4-dichlorophenyl)sulfonylpyridin-2-yl]-4-iminopenta-2,6-dienamide N-[(Z)-1H-indol-3-ylmethylideneamino]-2-methoxyquinoline-4-carboxamide 3-[2,4-bis(phenylmethoxy)phenyl]pentanenitrile [(3R)-5-[6-chloro-2-[4-(2-cyclohexylethynyl)phenyl]quinolin-4-yl]-1,3-dimethylpiperidin-3-yl]methanamine 1-[(2R)-3,4-bis(phenylmethoxy)butan-2-yl]-5-pyridin-4-yl-2H-pyrazine N-[1-(3,5-dichlorophenyl)cyclobutyl]azetidine-3-carboxamide N-azido-3,4-dichlorobenzohydrazide 3-aminooxy-N-[(1R,2S)-2-hydroxycyclopentyl]benzamide (4R)-1-[(2S)-butan-2-yl]-4-(3,5-difluorophenyl)azetidin-2-one 6-[6,7-dimethoxy-2-(4-propan-2-ylphenyl)cyclohepta-1,3,5-trien-1-yl]pyridine-2-carboxamide N-[3-(1,6-dihydropyrrolo[2,3-c]pyridine-5-carbonyl)phenyl]pyrrolidine-1-carboxamide 5-butyl-N-[1-(2,3-dihydroindole-1-carbonyl)piperidin-4-yl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide N-[4-(3-bromophenyl)-2,6-dimethyl-5-oxopyrazin-1-yl]benzamide N-ethyl-2-[3-fluoro-5-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1H-indole-6-carboxamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-methoxypyridine-2-carboxamide 2-(9H-fluoren-1-yl)-7,8-dimethoxychromen-4-one 2-[[3-chloro-5-(trifluoromethyl)pyridine-4-carbonyl]amino]ethanesulfonic acid (2S)-3-[6-(6,7-dimethoxyquinolin-4-yl)oxypyridin-3-yl]sulfanyl-N'-[[4-(trifluoromethyl)phenyl]methyl]butanehydrazide;ethane N-(6-chloro-3-nitropyridin-2-yl)nitramide 2-ethylsulfanyl-4-(trifluoromethoxy)benzaldehyde 3-[2-[ethyl(oxolan-2-ylmethyl)amino]ethyl]-1-(4-hydroxyphenyl)pyrrolidine-2,5-dione (5S,7R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-5-(furan-2-yl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide [5-(5,6-dichlorobenzimidazol-1-yl)thiophen-2-yl]-phenylmethanone (5Z,6E)-1-[2-chloro-5-fluoro-4-(4-nitrophenyl)phenyl]-5-ethylidene-6-prop-2-enylidenepyridine-2-thione 3-[(3R)-3,5-dihydroxypentyl]-7,9,9a-trimethyl-2H-cyclopenta[c]chromen-1-one 5-(2,4-dihydroxy-3-propanoylphenyl)-N-[2-methyl-4-(morpholine-4-carbonyl)phenyl]-1,2-oxazole-3-carboxamide N-(4,4-difluorocyclohexyl)-1H-indazole-3-carboxamide 1-(2,4-dichlorophenyl)-5-[[[4-methoxy-6-[[3-(trifluoromethyl)phenyl]methoxy]cyclohepta-1,4,6-trien-1-yl]amino]methyl]-N-methylpyrazole-3-carboxamide 5-methoxy-N-[2,3,4-trifluoro-6-(tetrazol-1-yl)phenyl]pyrimidin-4-amine 4-[(3aR,7aS)-2-[(1S)-1-phenylethyl]-1,3,3a,4,6,7,7a-octahydropyrano[3,4-c]pyrrol-5-yl]pyridine-2-carbonitrile N-[1-(4-chlorophenyl)pyrrolidin-3-yl]-2-ethoxypyridine-3-carboxamide 1-[(3S,4R)-3-hydroxyoxan-4-yl]pyrazole-4-carboxamide;5-[[(1E)-1-(methylideneamino)buta-1,3-dien-2-yl]amino]-7H-pyrrolo[2,3-d]pyrimidine-6-carbonitrile N-(6,7-dihydro-4H-pyrano[3,2-d][1,2]oxazol-3-ylmethoxy)-6-pyrazol-1-ylpyridine-2-carboxamide 1-(3-bromophenyl)nonane-1,6-dione (3Z)-N,2-diethylhexa-1,3,5-trien-3-amine;4-methanimidoyl-N'-[(3Z,5E)-6-[5-(trifluoromethyl)pyridin-3-yl]octa-3,5-dienyl]benzenecarboximidamide 1-azido-3,7-dimethyl-5-propan-2-ylnaphthalene 3-(2,6-dimethoxyphenyl)-7-[3-fluoro-4-(3-propylpiperazin-1-yl)anilino]-2H-pyrimido[5,4-e][1,3]oxazin-4-one 3-chloro-4,5-dimethoxybenzonitrile;2-[6-(1H-pyrazol-4-yl)pyridin-3-yl]acetamide [3-(2,2-dimethylpropanoyl)phenyl]azanium 1-[3,5-bis(trifluoromethyl)phenyl]-N-(2-fluoro-6-methoxyphenyl)sulfanylmethanamine;ethane 2-(5-cyclopropylpyrimidin-2-yl)-5,7-difluorophthalazin-1-one 2,5-dimethyl-3-(4-phenoxyphenyl)-6H-1,3,4-oxadiazine N-[3-(4-benzylpiperidine-1-carbonyl)phenyl]furan-2-sulfonamide 3-(2,6-difluorophenyl)-1-(2,4-dimethylphenyl)-6-(4-pyrrolidin-1-ylbutoxy)-6H-cyclohepta[d]imidazole 5-(3,4-dichlorophenyl)sulfanyl-1H-pyrrolo[2,3-b]pyridine 4-(7-methoxyquinolin-8-yl)-N,1-dimethylpiperidine-3-carboxamide N-[4-(6-methoxy-3-propanoylfuro[2,3-b]pyridin-2-yl)phenyl]acetamide (3E)-6,10-dichloro-5-methoxy-3-[(2Z)-penta-2,4-dienylidene]-1H-2-benzoxocine;ethane (2S)-1,2,3,5-tetramethyl-4-[4-phenyl-6-(3-propan-2-ylpyridin-2-yl)pyridin-2-yl]-2H-benzimidazole 4-methoxy-1-[(E)-3-phenylprop-2-enoyl]piperidine-4-carboxamide [4-(2,3-dimethylindole-1-carbonyl)piperazin-1-yl]-phenylmethanone [(2R,3S)-2-[(4-methoxyphenyl)methyl]-3-pyridin-3-ylmorpholin-4-yl]-(5,6,7,8-tetrahydroquinolin-8-yl)methanone 3-chloro-2,6-diiodopyridine 1-(1H-benzimidazole-2-carboximidoyl)naphthalen-2-ol 2-[4-(5,7-dimethyl-1H-indol-4-yl)piperazin-1-yl]-6-ethoxy-1,3-benzothiazole 3-(cyclohexylmethoxy)thiophene N-[1-(3,4-dichlorophenyl)ethyl]-2-[(6S)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]acetamide 2-[2,6-difluoro-4-(1-pyridin-3-ylpyrazol-4-yl)benzoyl]oxyacetic acid 1-(6,7-dimethoxyquinazolin-4-yl)piperazine 4-[(3R)-3-methylpyrrolidine-1-carbonyl]benzamide 6-chloro-3-(2,6-dichlorophenyl)pyridine-2-carbonitrile N-[5-(2,3-dichlorophenyl)-1H-pyrazol-4-yl]-3-methylpyridine-4-carboxamide N-[4-(hydroxycarbamoylamino)phenyl]octanamide 2-[3,5-dimethyl-1-(4-methylphenyl)sulfonylpyrrol-2-yl]-5,7-difluoro-1,3-benzoxazole N-butanoyl-N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-3,3,4,4,5,6-hexadeuteriopiperidine-1-carboxamide (6R)-7-[[2-(8-chloro-4-oxochromen-2-yl)acetyl]amino]-3,4-dihydro-2H-azocine-1-carboxylic acid 2-amino-1'-[5-(benzylcarbamoyl)-1H-imidazole-4-carbonyl]spiro[7,8-dihydro-3H-pyrrolo[2,1-c][1,4]oxazine-6,3'-pyrrolidine]-3-carboxamide;2,2,2-trifluoroacetic acid 5-cyclopropyl-N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]pyrazine-2-carboxamide 3-[[(2S)-5-(4-chlorophenyl)morpholin-2-yl]methoxy]benzoate N-[(2,4-dichlorophenyl)methyl]-6-[3-[(dimethylamino)methyl]pyrrolidin-1-yl]pyridazine-3-carboxamide 4-[2-(cyclopropylmethoxy)-5-methylsulfonylphenyl]butanamide 2-[(4-benzylbenzoyl)amino]-N-hydroxybutanamide 5-[2-amino-3-chloro-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-N,N-dimethylpyrazine-2-carboxamide N-[2,4-dioxo-1-(5-propan-2-ylsulfanylpyridin-3-yl)pyrrolidin-3-yl]acetamide 2-(1,3-benzothiazol-2-yl)-5-chloro-4H-pyrazol-3-one N-(7-azido-3-bromoimidazo[1,2-a]pyridin-8-yl)butane-2-sulfonamide 4-[3-[[4-(trifluoromethyl)phenyl]carbamoylamino]propoxy]butanoic acid 5-azido-3-(2,4-difluorophenyl)-1H-indole 4-(2,3-dihydro-1H-inden-5-yloxy)-5,6-dimethoxypyrimidine 5-bromo-2,6-dimethyl-4-[(E)-2-nitroethenyl]pyridine 2-[5,6-dimethoxy-1-(4-propan-2-ylphenyl)sulfonylindole-3-carbonyl]piperidine-3-carboxylic acid ethane;(E)-1,2,3,4-tetramethylpent-1-ene;1,5,7,8-tetramethylnaphthalene N-[(4S)-6-chloro-3,4-dihydro-2H-chromen-4-yl]butane-1-sulfonamide N-[1-(furan-3-yl)ethenylamino]formamide;3,5-dimethoxy-4-[(E)-pent-2-enoxy]benzaldehyde 5-cyclobutyl-2,4-diethoxypyrimidine 3-[4,5-bis(ethenyl)-3H-pyrrol-2-yl]propanoic acid 6-methylsulfanylquinazoline;hydrobromide 3-(4-chlorophenyl)sulfanyl-N'-(6-oxo-1,7,8,9-tetrahydropurin-2-yl)propanehydrazide N-[4-(3,4-dihydro-2H-1,5-benzodioxepine-7-carbonyl)phenyl]-1-propan-2-ylpyrrolidine-2-carboxamide 7-(dimethylamino)-3-hydroxynaphthalene-2,8-disulfonic acid;manganese(2+) 3-[4-(2,6-diphenylphenyl)-1,4-dihydropyrimidin-5-yl]-1H-imidazole-2-thione (1R,3S)-3-N,3-N-bis[2-(2-pyridin-4-ylethenyl)-6-thiophen-2-ylpyrimidin-4-yl]cyclopentane-1,3-diamine 2-methoxy-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine [5-(5,6-dihydronaphthalen-2-yl)furan-3-carbonyl]azanium;2,2,2-trifluoroacetate 2-[3,4-diamino-5-(trifluoromethyl)phenyl]-6,7-dihydro-3H-furo[3,4-c]pyridin-1-one 2-amino-N,N'-bis[4-(3-phenylquinoxalin-6-yl)phenyl]pentanediamide 2-(3,5-dimethylbenzoyl)-10,10-difluoro-7-oxa-9-azaspiro[4.6]undecan-11-one 2-[3,5-bis(trifluoromethyl)phenyl]-1,8-dioxaspiro[4.6]undecane N-[1-[4-(aminomethyl)phenyl]cyclobutyl]-2,5-dichlorobenzamide 4-(3,4-dihydrochromen-2-ylidene)-1-[5-methyl-6-(2,4,6-trichlorophenyl)furo[2,3-d]pyrimidin-3-yl]piperidine-3-carboxylic acid 3-[(4,5-diphenyl-1H-pyrazol-3-yl)amino]propanoic acid 4-(1H-indole-2-carbonyl)-N-pyridin-3-ylpiperazine-1-carboxamide N-[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]sulfanylbut-1-en-2-amine 1-[2,4,6-trimethyl-5-(3-oxobutanoyl)phenyl]pentane-1,4-dione N-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethyl)-2-(4-methyl-1,4-thiazepan-5-yl)acetamide N-[(2S,4R)-1-acetyl-2-(3-chlorophenyl)piperidin-4-yl]-5-methoxypyridine-3-carboxamide 3-[(2,4-dihydroxyphenyl)methyl]-5-ethoxycarbonylcyclohexane-1-carboxylic acid N-(3,3-dimethylbut-1-en-2-yl)-5-[3-[7-(4-fluorophenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-amine 1-(4-bromophenyl)sulfonyl-2,3-dihydropyrazolo[1,5-a]pyridin-8-ol 2-[[[4-(dimethylamino)pyridin-3-yl]amino]methyl]-N'-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-N,N,5-trimethylbenzenecarboximidamide N-[1-(5,6-dihydroquinoline-2-carbonyl)piperidin-3-yl]cyclopropanecarboxamide (4R)-5-(3,4-dimethoxyphenyl)-3,7,7-trimethyl-1-propan-2-yl-6,8-dihydroquinoline-4-thione 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(2-fluoropropan-2-yloxy)azetidin-3-yl]acetamide N-[[2,4-bis(trifluoromethyl)phenyl]methyl]-5-[3-(dimethylamino)propanoyl]-1H-imidazole-2-carboxamide [4-[5-(2,6-difluorophenyl)-1H-imidazol-3-ium-2-yl]pyridin-2-yl]methanamine N-(4,5-dimethylpyridin-2-yl)-3-[4-fluoro-2-(5-methyl-1H-indol-3-yl)phenyl]-4H-quinazolin-2-amine 1-(3,4-dichlorophenyl)-N'-hydroxy-2-[(5R)-4,7,8-trimethyl-3,6-dioxooctyl]imidazole-4-carboximidamide 2-tert-butyl-7-(3,5-dichlorophenyl)-1H-purine 2-[[5-(4,7-dimethylquinolin-2-yl)pyridine-3-carbonyl]amino]acetic acid 3-[4-[2-(6-butylpyridin-3-yl)ethynyl]phenyl]propanal;N,4-dimethyl-5-(trifluoromethyl)furan-2-sulfonamide 2-[N-(4,5-dimethylpyrimidin-2-yl)-3-nitroanilino]acetonitrile 7-(1H-indazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-2-carboxamide 4-[5-(3-chloro-2H-indazol-6-yl)pentyl]morpholine (2S)-2-[1-benzyl-5,6-diethoxyindol-3-yl]-2-sulfanylidenepropanedioic acid N-[3-(2-fluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-7-yl]-2-methoxybenzenesulfonamide N-[(5Z)-3-tert-butyl-2,6-dioxo-1-[(4-nitrophenyl)methyl]-4H-pyrimidin-5-yl]formamide 3-methyl-2,4-bis(phenylmethoxy)piperidine 1-(3-acetylthiophen-2-yl)ethanone;N'-[6-methoxy-7-(4-morpholin-4-ylbutoxy)quinazolin-4-yl]cyclopropanecarboximidamide N-(2-morpholin-4-ylethoxy)benzenecarboximidate 6-chloro-N-[1-(1,3-dimethylpyrazol-4-yl)piperidin-3-yl]pyridazin-3-amine 2-[3-(3,4-dimethoxyphenyl)propanoyl]-5,5-difluorocyclohexan-1-one 1-(6-aminopyrimidin-4-yl)indole-5-carboxylate (3R,4S)-1-[[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]methyl]-4-(1-methylimidazol-2-yl)pyrrolidine-3-carboxamide 4-[2-[[(1S)-1-[6-(3,5-dimethylpyrazol-1-yl)-3-fluoropyridin-2-yl]ethyl]amino]pyrimidin-5-yl]-6-morpholin-4-ylpyridine-3-carbonitrile [(2S)-1-azidooxy-4,4-difluorobutan-2-yl]benzene 2-(3,4-dihydro-1H-isoquinolin-2-yl)-6-(oxan-4-ylamino)pyridine-3-carbonitrile 2-azido-N-[(4,5-dimethylthiophen-3-yl)methyl]acetamide N-[4-(8,9-dihydrodibenzothiophen-2-yl)phenyl]-N'-[(E)-1,3-di(propan-2-ylideneamino)prop-1-enyl]propane-1,3-diamine 2-methylsulfinyl-1,3-benzothiazole 1-(azidomethyl)-4,6-dimethyl-2,3-dihydroindole 3-(2-chlorophenyl)-1-[(4R,6S)-6-(3-methoxy-4-propan-2-yloxyphenyl)-8-oxo-5,6-dihydrobenzo[h]quinazolin-2-yl]piperidine-2-carboxylic acid 2-[4-(6,7-dihydro-1H-indazole-3-carbonyl)piperazin-1-yl]benzonitrile (2S,3R)-3-azido-N'-benzylpyrrolidine-1-carboximidamide N-(azidomethyl)-1-(4-chlorophenyl)-N'-[3-(dipropylamino)propyl]ethane-1,2-diamine 4-[5-(azetidin-1-ylmethyl)-6,7-dihydronaphthalene-2-carbonyl]benzonitrile N-[2,5-dimethyl-4-(3-oxo-1H-isoindol-2-yl)phenyl]-6,7-dihydronaphthalene-2-carboxamide 4-methyl-5-(trifluoromethyl)-1H-indole-2-carboxylic acid N-[1-[(2S)-2-amino-3,3-dimethylbutanoyl]azetidin-3-yl]benzenesulfonamide 1-[(2S,4R)-4-chloro-2-methyl-3,4-dihydrochromen-7-yl]pyrrole-3-carboxylic acid 5-chloro-3-methyl-N-[1-(2,4,6-trifluorophenyl)ethenyl]penta-1,3-dien-2-amine (5-phenyl-1,3-thiazol-2-yl)-[2-[(Z)-1-pyridin-2-ylprop-1-enyl]pyrrolidin-1-yl]methanone 4-(2-cyclopropylethoxy)pyridine;(Z)-3,4,6-trihydroxyhept-5-en-2-one 2-benzylsulfanyl-1H-benzimidazole 5-[3-fluoro-4-(6-methylpyridin-2-yl)oxyphenyl]imidazolidine-2,4-dione 2-[(3R)-3-(4,5-dimethyl-1H-imidazol-2-yl)pyrrolidine-1-carbonyl]-1,3-thiazole-4-carboxylic acid (Z,3Z)-3-[[2-ethyl-4-[5-methoxy-1-(4-methylphenyl)sulfonylindole-7-carbonyl]piperazin-1-yl]imino]prop-1-en-1-ol N-[3,5-bis(trifluoromethyl)phenyl]-3-[3-(cyclobutylmethoxy)-4-[2-oxo-2-[[(1S)-1-pyridin-3-ylethyl]amino]ethoxy]phenyl]propanamide [7-(3,4-dimethoxyphenyl)-3H-inden-1-yl]-trihydroxyphosphanium N'-[(2S)-4,5,6-trimethyl-2H-1,3-thiazin-3-yl]thiophene-2-carbohydrazide [(2S)-1-[[4-(aminomethyl)phenyl]methoxycarbonyl]pyrrolidine-2-carbonyl]oxidanium 4-[(2S,3S)-2-methyl-1-azabicyclo[2.2.2]octan-3-yl]-3-[[6-methyl-5-(5-methylpyridin-3-yl)oxypyridazin-3-yl]amino]benzoic acid (2R)-N-(1,3-benzodioxol-5-ylmethyl)-4-(2-chlorophenyl)-2,3-dihydrochromene-7-sulfonamide;hydrochloride 3-(diethylamino)-4-[6-[4-(3,5-dimethyl-1,2-oxazol-4-yl)phenyl]pyrazin-2-yl]benzoate 2-amino-6-methyl-4-(3,4,5-trihydroxyphenyl)sulfanylbenzenesulfonic acid (2S)-N-[4-[4-chlorobutyl(4-hydroxybutanoyloxymethyl)carbamothioyl]phenyl]sulfonylpyrrolidine-2-carboxamide 5-[4-fluoro-3-(4-pyridin-4-yl-1H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]-N,N-dimethylpyridin-3-amine 4-[3-[2-(4-chlorophenyl)ethyl]piperidine-1-carbonyl]-N-hydroxybenzamide 6-cyclopropyl-N'-hydroxy-3-[4-(methoxymethyl)-1,3-thiazol-2-yl]sulfanylpyridazine-4-carboximidamide N-(7-chloro-1H-indazol-3-yl)pyridine-4-carboxamide 2-(5-methylsulfanylpyridin-3-yl)oxypyrimidine 2-[4-(aziridin-1-yloxy)phenyl]-N,N'-dimethylpyridine-4-carboximidamide 2-[6-(3-chlorophenyl)imidazo[1,2-a]pyridin-5-yl]benzonitrile 2-[[1-(4,6-dimethylpyrimidin-5-yl)sulfonylpyrrolidin-3-yl]-ethylamino]ethanol 3,5-dimethoxy-4-[(Z)-1-(1H-pyrrolo[2,3-b]pyridin-4-yl)prop-1-enyl]phenol [4-(azidomethyl)phenyl]sulfonyl-[2-[4-chloro-3-[6-[(2R,5S)-2,5-dimethylpiperazin-1-yl]pyridin-3-yl]anilino]pyrimidin-4-yl]carbamic acid [2-(6-azido-1,3-benzodioxol-5-yl)cyclohexen-1-yl]-phenylmethanone 1-methyl-3,5-bis(trifluoromethoxy)benzene;4-[(E)-prop-1-enyl]benzonitrile (2R)-3,6-dioxo-1,2-bis(5H-pyrrolo[3,4-b]pyrazine-7-carbonyl)piperazine-2-carboxylic acid 3-azidooxy-1-chloronaphthalene 4-cyclohexylsulfonyl-N-[(3S)-1-methylpyrrolidin-3-yl]-2,5-diphenylfuran-3-carboxamide 4-[(1R,2S)-2-aminocyclohexyl]-2-[3-(cyclopropanecarbonylamino)phenyl]-1H-indole-7-carboxamide 5-butoxy-2-[4-(difluoromethyl)phenyl]-1,3-dioxane 2-(7,8,9,10,11-pentamethyldodeca-3,6-dienyl)naphthalene [4-(aminomethyl)-3-methoxyphenyl]-[2-chloro-6-(hydroxymethyl)-1,3-benzothiazol-5-yl]methanone 6-[(2Z)-3,3-dimethyl-4-naphthalen-1-ylpenta-2,4-dien-2-yl]-10-methoxy-1,2-dihydrophenazine 4-methyl-3-(trifluoromethoxy)benzoic acid 3-N-tert-butyl-1,1,4-trioxothiane-3,5-dicarboxamide;6-methoxy-1,2,3,4-tetrahydronaphthalene N-[(2S)-4-methyl-1-oxo-1-(pyridin-3-ylmethoxy)pentan-2-yl]benzamide N-(2,3-dichlorophenyl)-6-methylquinazoline-8-sulfonamide 6-[(4-tert-butylphenyl)methylsulfanylamino]-5H-pyrazolo[1,5-b][1,2,4]triazole-4-carboxamide N-[4-[4-(dimethylamino)-6-[(3R)-3,4-dihydroxybutoxy]pyridin-2-yl]phenyl]acetamide 1-ethyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)piperidine-1-carbonyl]pyrrolidin-2-one 2-bromo-7,9-dichloro-1H-pyrrolo[3,4-b]quinoline (1S)-2-azido-4,5,7-trifluoro-N-(4,6,6-trimethylcyclohexa-2,4-dien-1-yl)-3H-1,3-benzothiazol-2-amine 1-butyl-5-ethylsulfanyltetrazole [1-(4-methoxyphenyl)cyclopropanecarbonyl]-methylideneazanium 3,4-dichloro-N-[(Z)-4-[5-fluoro-6-[2-hydroxyethyl(methyl)amino]pyridin-2-yl]but-1-enyl]benzamide 2-(4-bromophenyl)sulfanyl-1-methoxyethanesulfonic acid 2-[4-(1-aminocyclopropyl)anilino]pyrimidine-5-carboxylic acid N-methyl-3-phenyl-2,4-dihydrobenzo[h]chromene-2-carboxamide [3,4-bis(1H-inden-2-yl)phenyl]methanamine 4-[2-(2,6-difluorophenyl)-7H-pyrrolo[3,2-d]pyrimidin-4-yl]morpholine 3-(3-ethylsulfonylphenyl)-4,5-dimethyl-1H-pyridazin-6-one 5-ethyl-2,3-dimethoxy-6-nitrobenzoic acid [5-methylsulfanyl-2,3-di(propan-2-yl)imidazol-4-yl]methanimine 2-[1-(6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)pyrrolidin-3-yl]-N-methoxyacetamide N-[5-(2,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-6-(2-pyrrolidin-1-ylethoxy)-2-(piperidin-4-ylamino)pyridine-3-carboxamide N-[5-chloro-2-(2,6-difluorophenoxy)phenyl]ethanesulfonamide 4-chloro-2-[1,3-thiazol-2-yl(sulfanyl)methoxy]benzoic acid (3E,5Z)-N-[1-cyclopropylidene-2-[5-methyl-4-(2-piperidin-1-ylethoxy)pyridin-3-yl]ethenyl]-6-fluoro-2-methylhepta-3,5-dienamide 4-chloro-2,6-difluoro-N-[(1R)-5-methyl-2,3-dihydro-1H-inden-1-yl]benzamide 4-(azidomethyl)-1-cyclopentyltriazole N-(2-hydroxyphenyl)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide (5Z)-5-[[3-[[3,4-bis(difluoromethoxy)phenyl]methyl]cyclobutyl]methylidene]imidazolidine-2,4-dione N-cyclopropylsulfanyl-2,3-dimethoxyaniline;3-[(E)-hex-1-enyl]-7H-purin-6-imine [1-[(4-fluorophenyl)methyl]triazol-4-yl]urea [4-[2-(7,8-dimethoxy-3H-imidazo[1,5-c]quinazolin-2-yl)ethynyl]phenyl]-morpholin-4-ylmethanone 3-[1,4-dimethyl-2-(6-methylcyclohexa-1,5-dien-1-yl)-9H-carbazol-3-yl]-N,N-dimethylaniline N-[(5S)-3,4-dihydro-2H-chromen-7-yl]-1-(4-methylsulfonylphenyl)pyrazole-3-carboxamide N-[5-(2,3-dihydrothiophen-5-yl)pyrimidin-4-yl]hydroxylamine 2-bromo-1,3-difluoro-5-nitrobenzene 7-[(5-ethylsulfonylpyridin-2-yl)methyl]-5-methyl-4H-pyrrolo[3,2-d]pyrimidine 2-bromo-N-(5-bromonaphthalen-1-yl)sulfonylacetamide (2S)-N-[6-methyl-1-(4-nitrophenyl)sulfonylpyrrolo[3,2-b]pyridin-2-yl]piperidine-2-carboxamide 4-[(Z)-2,3-diaminoprop-1-enyl]-N-methylbenzamide;4-piperidin-1-ylquinazoline (3S)-5-(4-cyano-2,6-difluorophenyl)sulfonyloxy-N-[(3R,5S)-5-fluoropyrrolidin-3-yl]-1-(quinoline-7-carbonyl)piperidine-3-carboxamide [(3R)-1-(7,8-dihydronaphthalen-2-ylmethoxy)-5-(trifluoromethyl)piperidin-3-yl]carbamic acid 4-[3,5-bis(trifluoromethyl)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one [3-(2-azidoethoxy)phenyl]-morpholin-4-ylmethanone (1-azidooxyisoquinolin-7-yl)oxy-(dimethylamino)methanol 2-[4-(4-tert-butylphenoxy)phenyl]quinoline 1-N'-[(3-chlorophenyl)methyl]cyclopropane-1,1-dicarboxamide 2-[[4-chloro-3-(trifluoromethyl)phenyl]methoxycarbonyl-methylamino]-5,6,7,8-tetrahydro-1H-isoquinoline-4-carboxylic acid 1-(4-azidooxyphenoxy)-3,5-dichlorobenzene N-(2,3-dihydroxypropyl)-1H-indole-5-carboxamide N-[(2-ethylphenyl)methyl]-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide 1-amino-3-[4-(5-fluoropyrimidin-2-yl)oxypiperidine-1-carbonyl]cyclobutane-1-carbonitrile N-[(2S)-1-[1-(cyclopropylmethylcarbamoyl)cyclopentanecarbonyl]pyrrolidin-2-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide 2-[(1-aminoisoquinoline-5-carbonyl)amino]-N,3-dimethylbutanamide 5-methyl-2-[2-(1H-pyrrol-2-yl)ethenyl]-3,4-dihydro-1H-isoquinoline N-[2-(2,4-dichlorophenyl)ethyl]-2-hydroxy-2-[3-methoxy-5-(methylideneamino)phenyl]-N',N'-bis(pyridin-2-ylmethyl)propanediamide 3-(5,6-difluorocyclohexa-1,3-dien-1-yl)-2-methoxyquinoline 5-[3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-1H-pyrimidine-2,4-dione 3-[2,4-dioxo-5-(2-phenylethyl)pyrimidin-1-yl]propanoate 1-[(E)-2,3-bis(3,4,5-trimethoxyphenyl)prop-2-enyl]-2-(1H-imidazol-5-ylmethylideneamino)guanidine 2-(4-methylphenyl)sulfanyl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole 2-(3,5-dimethylphenyl)-4-[3-(7H-purin-6-ylamino)phenyl]phenol N-[2,3-dioxo-6-phenyl-5-(trifluoromethyl)piperidin-1-yl]propanamide (Z)-1,4-diamino-5-[4-(2-aminophenoxy)-3-methoxyphenyl]pent-4-en-2-one 1-azidooxy-2,3,4,5-tetramethylbenzene 2-[(4R)-3,4-dihydro-2H-chromen-4-yl]-1-[3-(6-methoxy-7H-cyclopenta[b]pyridin-3-yl)butyl]-3-propan-2-ylpyrrolo[3,2-c]pyridine 5-[[[(Z)-1H-indol-3-ylmethylideneamino]carbamothioylamino]carbamoyl]furan-2-carboxylic acid 3-fluoro-2-N,4-N-bis(methylaminosulfanyl)benzene-1,2,4,5-tetramine 1-[4-(2,2-dimethylpropanoyl)phenyl]ethanone 2-[6-methyl-5-(6-piperidin-1-ylpyridin-3-yl)oxy-1H-indazol-4-yl]acetamide 1-(3,5-dimethoxyphenyl)sulfonyl-2-[2-(1H-indole-3-carbonylamino)ethyl]piperidine-4-carboxylic acid (6S)-10-bromo-3-methylsulfanyl-7-propanoyl-6-[5-(trifluoromethyl)pyridin-2-yl]-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 4-methyl-5-propan-2-yloxycarbonylbenzene-1,3-disulfonic acid 4-(8,14-dioxapentacyclo[11.7.0.02,10.05,9.015,20]icosa-1,3,5(9),6,10,12,15(20),16,18-nonaen-14-yloxymethyl)benzenethiol 2-[(E)-3,4-dimethyl-1-[6-oxo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,7,11b-triazatricyclo[10.4.0.04,9]hexadeca-1(12),3,8,13,15-hexaen-14-ylamino)hexoxy]pent-3-en-2-yl]guanidine 5-[(2E,4Z)-1-methoxyhepta-2,4-dien-3-yl]-N'-propan-2-ylthiophene-2-carbohydrazide 2-[4-[3,5-difluoro-4-(trifluoromethyl)phenyl]cyclohexyl]-1,3-difluoro-7-propoxynaphthalene 6-[(2,4,4a,5,7,8,8a-octahydropyrido[3,4-b][1,4]oxazin-6-ylamino)methyl]-2H-benzotriazole-4-thiol 5-[(2S,4R)-2-methyloxan-4-yl]oxy-1H-indazole 2-[3-cyclohexyloxy-5-(6,7-dihydro-1H-indole-2-carbonyl)phenyl]benzoic acid 3-[4-(azidomethyl)-3,5-difluorophenyl]benzonitrile [3-(4-chlorobenzoyl)-4,5-dioxopyrazolidin-1-yl]oxymethylphosphonic acid 5-azido-3-chloro-2,4-dimethoxythiophene 1,2-bis(chloromethyl)-4-(trifluoromethoxy)benzene 1-[2,5-difluoro-4-(trifluoromethyl)phenyl]hexan-3-one (2Z)-N',1',5,7-tetramethylspiro[3H-1-benzazepine-4,3'-cyclopentene]-6-carboximidamide 4-[2,3-bis(hydroxymethyl)phenyl]-5,8,11-trioxatetracyclo[7.6.0.02,6.010,12]pentadeca-1,3,6,9,13-pentaen-14-one (1Z,3E)-5-[2-methoxy-4-(3,5,7-triazatricyclo[6.3.1.04,12]dodeca-1,3,8(12),9-tetraen-2-yl)phenyl]penta-1,3-diene-1,3-diamine 2-[(4E,5Z)-4-ethylidene-1H-cyclopenta[b]pyridin-3-yl]pyridine-4-carboxylic acid 4-(4-bromophenyl)-2,6-bis[3-(trifluoromethyl)phenyl]pyrimidine 4-bromo-1,6-dimethylindazole 2-[4-(4,4-dimethylpiperidine-1-carbonyl)anilino]-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine-4-carbonitrile (3E)-4-amino-3-[[2,3-difluoro-5-(trifluoromethyl)phenyl]methylidene]azete-2-thione 3-(2,4-difluorophenoxy)-N-methyl-1,6-naphthyridine-5-carboxamide N-[2-(2,4,5-trimethyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carboxamide;hydrochloride 2-[7-(diethylamino)-3,4-dihydronaphthalene-1,5-disulfonate 5-[(6-aminopurin-9-yl)methyl]-4-ethylsulfonyl-2-methoxybenzoic acid (5E)-5-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-2-(2,4-dimethylphenyl)imino-1,3-thiazolidin-4-one 6-[5-bromo-3-(4-methylpiperazin-1-yl)sulfonylindol-1-yl]hexanoic acid (E)-3-[2,5-dimethyl-1-[4-methyl-3-(propan-2-ylideneamino)phenyl]pyrrol-3-yl]prop-2-enamide N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]prop-2-enamide 2-[[4-methoxy-3,5-bis(trifluoromethyl)phenyl]carbamoyl]pyrrolidine-1-carboxylate 3-ethyl-2-methoxy-5,6,7,8-tetrahydroisoquinoline;3-(4-fluorophenyl)-1H-pyrrolo[2,3-b]pyridine N-[(Z)-2-(3,5-dimethoxyphenyl)-3-(2-ethylhydrazinyl)but-1-enyl]-2-propan-2-ylidene-4H-cyclopenta[a]acenaphthylen-1-imine;(E)-N-(2,2-dimethylpropyl)dec-2-ene-1,6-diamine 1-[2-(2-ethylphenyl)quinolin-4-yl]oxypyrrolidine-2-carboxamide;dihydrochloride N-[2,3,5-trifluoro-6-(phenylcarbamoylamino)phenyl]formamide 2-azido-N,5-dimethyl-1H-indole-3-carboxamide 2,4-dimethyl-6-oxo-N-(oxolan-2-yl)-1H-pyrimidine-5-carboxamide 2-[4,4-bis(3-aminophenyl)butanoyloxy]-2-(1H-indol-6-ylmethylsulfanyl)acetic acid 2-chloro-4,6-dimethylbenzenethiol;ethane;formaldehyde;4-(1,3-thiazol-5-ylsulfanyl)benzaldehyde 4-[6-amino-5-(1,2,3,4-tetrahydroisoquinolin-7-yl)pyridazin-3-yl]phenol 7-chloro-2-(2-methylpropoxy)-5-[4-[2-[(3S)-oxolan-3-yl]ethynyl]phenyl]-1,3-benzoxazole 1-azidosulfanyl-3,4-dimethyl-5-phenyl-2-(trifluoromethyl)benzene 3-[2-amino-4-(benzylamino)phenyl]-1H-pyrazole-5-carbonitrile;ethane 2-chloro-N-(4-ethylphenyl)-9,9-dimethyl-N-[3-(trifluoromethyl)phenyl]fluoren-1-amine 2-[6-[[3-(1,4-dioxaspiro[4.5]decan-8-yl)phenoxy]methyl]pyridin-2-yl]benzenethiol [(2R,4S)-6-azido-1-methylsulfonyl-4-phenylhexan-2-yl]benzene 6-[(2S,4R)-2-[[5-chloro-2-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)pyrimidin-4-yl]amino]-4-methoxypyrrolidin-1-yl]pyridazine-3-carbonitrile 2-(1,3-benzodioxol-4-yl)-N-[6-[4-[(3S)-oxolan-3-yl]oxyphenyl]pyridin-3-yl]cyclopropane-1-carboxamide 3-[(2R,6S)-1-methyl-5-oxo-2-phenylmorpholin-4-yl]propanenitrile ethane;4-[5-(oxan-2-yloxymethyl)furan-3-yl]benzenesulfonamide 2-amino-9-[(Z,3E)-3-hydroxyiminopent-1-enyl]-1H-purine-6-thione 6-methyl-2,3-di(pyrimidin-2-yl)quinoxaline 4-chloro-2-[3-(methoxymethyl)morpholine-4-carbonyl]phenol N-[(4,5-diethylcyclohexa-1,3-dien-1-yl)methyl]-2,6-dimethoxybenzamide 7-(2,4-difluorophenyl)-8-methoxy-3H-pyrazolo[1,5-a]quinazoline 3-[3-(2-chlorophenoxy)phenyl]oxirane-2,2-dicarbonitrile (2Z)-1-ethylsulfonyl-3,4,5-trifluoro-6-methoxy-2-[(2E)-3-sulfanylpenta-2,4-dienylidene]naphthalene 3-[1,6-dimethyl-4-[2-(2-methylpropoxy)ethoxy]pyrrolo[2,3-c]pyridin-7-ium-3-yl]azetidine-1-carboxylate (3,5-ditert-butylphenyl)methanethiol 1-[(3,4-difluorophenyl)methyl]-2-pyridin-4-yl-N-pyrimidin-5-ylindole-5-carboxamide N-(3,3-difluorocyclobutyl)-4-phenylpyrimidine-5-carboxamide 3-[[3,5-bis(trifluoromethyl)phenyl]carbamoylamino]-N-diazo-2,4-difluorobenzenesulfonamide 7-(azidomethyl)-6,8-difluoroquinoline 2-(azetidin-1-yl)-4,8-dimethylquinoline N-(2,6-dibromopyridin-4-yl)-N-(3-nitrophenyl)butanamide (6S)-3-ethylsulfanyl-6-[4-[2-(1H-indol-5-ylmethoxy)phenyl]phenyl]-7-(2H-tetrazol-5-yl)-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one N-[4-(4,5-dimethylimidazol-1-yl)pyridin-3-yl]-2-(2H-pyridin-1-yl)pyrimidine-4-carboxamide 7-chloro-2-iodoquinoline;ethane 2-(4-methoxyphenyl)-5-[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]-7-(trifluoromethyl)-3H-pyrido[2,3-d]pyrimidin-4-one 3-methyl-4,5-diphenylimidazole 6-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(hexadecyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 1-[(3aR,7aS)-1-(4-fluorophenyl)-2,2-dimethyl-3,3a,5,6,7,7a-hexahydropyrrolo[3,2-b]pyridin-4-yl]ethanone;2,2,2-trifluoroacetic acid 3-[(E)-hydroxyiminomethyl]-5,6-dihydrobenzo[h]quinoxaline-2-carboxamide 5-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrimidine-2,4-diamine 4-[(2E)-2-ethylidenehydrazinyl]-N-(5-fluoro-6-methoxypyridin-3-yl)-7-[3-(4-hydroxypiperidine-1-carbonyl)phenyl]-6,8-dihydro-5H-1,7-naphthyridine-2-carboxamide 1-[2,3-difluoro-6-(5-methylpyrimidin-4-yl)phenyl]-7,9-dihydro-6H-pyrido[4,3-b]azepine 2-[(1S)-1-azido-2,3-dihydro-1H-inden-5-yl]acetic acid 7-fluoro-8-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-9-oxa-1,3-diazatricyclo[6.3.0.02,6]undeca-2(6),4,7-triene 4-(2,3-dihydropyridine-6-carbonyl)-1-cyclopentyl-N-methyl-5-[2-[(1R)-1-[3-(trifluoromethoxy)phenyl]ethyl]pyrazol-3-yl]pyrrole-2-carboxamide 3-[1-(2,4-difluorophenyl)cyclohexyl]-5-methyl-6H-triazolo[4,5-d]pyrimidin-7-one 4-[1-azido-2,2-dimethyl-3-(propanoylamino)propoxy]benzoic acid 5-(azidomethyl)-2,3-dichloropyridine (3-chloro-4-methylphenoxy)boronic acid 1-[1-(2,4-difluorophenyl)ethyl]piperidine 6-N,5-N-bis(4-chlorophenyl)-1H-indole-2,3,5-triamine 2-(benzylideneamino)-N,3,5-triphenylaniline 1-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-5-oxopyrrolidine-2,4-dicarboxamide 2-(4-chloro-5-methoxy-2-nitrophenyl)acetonitrile 4-[7-methyl-1,3-dioxo-6-(1,2,5-thiadiazol-4-yl)isoindol-2-yl]piperidine-2,6-dione 2-(3,4-dimethoxyphenyl)-N'-hydrazinylbenzohydrazide 2,3-diethyl-1-phenylmethoxyazetidine 2-(3,4-dichlorophenyl)-5-methoxy-6H-[1]benzoxepino[3,4-d]pyrimidine N-(3-tert-butylphenyl)-4-(4,4-dimethoxy-2-methylidenepentanoyl)benzamide 2-azidooxy-1,3-difluoro-5-(trifluoromethyl)benzene 4-[1-(2,6-dichlorophenyl)sulfonylpiperidin-3-yl]-2H-triazole [4-(1,3-benzoxazol-2-ylsulfanyl)phenyl]azanide N-[5-(1-methylpyrazol-4-yl)pyrimidin-2-yl]spiro[3,4-dihydrochromene-2,1'-cyclopropane]-4-amine N-butanoyl-2-methoxybenzamide 1-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-ethoxypyrazole 1-[4-(4-chlorophenyl)buta-1,3-dien-2-yl]-2,6-dimethoxynaphthalene 7-[(2,6-difluorophenyl)methyl]-2-propan-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 1-(1,4-dimethylcyclohexa-2,4-dien-1-yl)-N-(4-methoxyphenyl)cyclopropane-1-carboxamide 1-azido-3-methylindole-2-carboxylic acid 3-[[4-(1H-indole-2-carbonylamino)cyclohexyl]amino]-6-methylthieno[2,3-b]pyridine-2-carboxylic acid 1-[(E)-6-fluoro-3,4-dihydro-2H-chromen-8-yl]ethanone;methanesulfonic acid 2-methyl-5-[(6R)-6-pyrrolidin-1-ylheptan-3-ylidene]-1H-imidazole N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-2-[2-[(4,5-dimethyl-6-oxopyrimidin-1-yl)methoxy]phenyl]benzamide 1-methyl-6,7,8,9,10,11-hexahydro-5H-cycloocta[d]pyridazine 6-[3-(azidomethyl)phenyl]-2,5-difluoro-1H-benzimidazole 2-hydroxy-N,N'-diphenylpropanediamide 6-methyl-5,11-dihydrocyclohepta[c]chromene 3-[(6,7-dimethoxyquinazolin-4-yl)amino]-1-ethylpiperidin-2-one 2-[[4-(3,5-dichloroanilino)thieno[3,2-c]quinoline-7-carbonyl]amino]acetic acid N-cyclopentyl-1,2-dihydrotriazolo[4,5-d]pyrimidine-6-carboxamide N-[6-(2,3-dimethoxyphenyl)-5-fluoropyridin-3-yl]ethanethioamide N-(6-chloropyridin-2-yl)-N-methoxy-5-methylpyridine-3-carboxamide 5-[2-(1,3-benzothiazol-6-yl)acetyl]-2-[[2,6-difluoro-4-(methanesulfonamido)benzoyl]amino]thiophene-3-carboxylic acid 6-chloro-3,3-diethyl-2H-1-benzofuran;hydrochloride 4-[1-(2,5-dimethylphenyl)propoxy]aniline [3-(cyclobutylmethoxy)azetidin-1-yl]-naphthalen-2-ylmethanone 3-cyclopentyloxy-2-(3,4-dichlorophenoxy)-N'-hydroxypyridine-4-carboximidamide ethane;3-(8-methoxy-[1,2]thiazolo[4,5-c]quinolin-4-yl)aniline N-(3,4-difluorophenyl)-7-ethoxy-6-methoxyquinazolin-2-amine N-[4-methyl-3-(tetrazolo[1,5-b]pyridazin-6-ylamino)phenyl]-2,2-di(propan-2-yloxy)acetamide 1,4-dimethyl-2-[(E)-3-methylsulfanylprop-2-enimidoyl]aniline 4-[[2-[[4-(difluoromethyl)phenyl]carbamoylamino]phenoxy]carbonylamino]-3,5-bis[difluoro(iodo)methyl]benzoate 4-(1,3-benzodioxol-5-yl)pyridine;6-bromo-1H-pyrrolo[2,3-b]pyridine (1S,3R)-N-[6-(4-methoxyphenyl)pyridazin-3-yl]-2,2,3-trimethylcyclopropane-1-carboxamide 5-(1,3-benzodioxol-4-yl)-N'-methanimidoylpyrazine-2-carboximidamide 6-[4-(6-butoxypyridine-3-carbonyl)piperazin-1-yl]pyridazine-3-carboxylic acid 2-amino-N-(3,4-dihydro-1H-isoquinolin-2-yl)acetamide;N-[6-ethylsulfanyl-5-fluoro-2-(trifluoromethyl)pyridin-3-yl]-3-formamidobenzamide 4-methyl-N'-[[4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperazin-1-yl]methoxymethyl]pyridine-2-carboximidamide 1-[5-(4,4-dimethylcyclohexen-1-yl)-2-methoxyphenyl]-N-(piperidine-1-carbothioylamino)formamide;ethane 2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)quinoline 1-(1,3-benzodioxol-5-ylmethoxy)butan-2-one 4-hydroxy-3-(6-morpholin-4-ylhexyl)pyran-2-one 5-[(E)-1,2-bis(4-hydroxyphenyl)pent-1-enyl]benzene-1,3-diol [(Z,2E)-2-ethylidene-5-methylhept-3-enyl]benzene N-(4-chlorophenyl)-4,5-dimethylpyridine-3-carboxamide 2,6-diamino-N-azido-5-ethylsulfanylpyrimidine-4-carboxamide 4-[[[3,5-bis(trifluoromethyl)phenyl]sulfanylamino]methyl]benzenethiol 1-[6,11-diamino-3-(3H-benzimidazole-5-carbonyl)-9-hydroxy-8,10-dihydro-7H-pyrido[2,3-c]azecin-7-yl]pyrrolidine-2,3-dione 7-(3,4-dimethoxyphenyl)-6-N-[3-[2-(ethylamino)ethoxy]phenyl]-5-methyl-3H-pyrido[2,3-d]pyrimidine-4,6-diamine 1-(3,4-dimethylphenyl)-6-hydroxy-5H-pyrazolo[3,4-d]pyrimidin-4-one 3-[2-(1H-indol-4-yl)ethyl]-5-methyl-2,6-dihydropyrazolo[4,3-d]pyrimidin-7-one 1-(4-chlorophenyl)-3,5-dimethylcyclohexa-2,4-diene-1,4-dicarboxylic acid 4-azido-3,5-dichloro-6-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyridazine N-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-7-ylmethyl)-2-(trifluoromethoxy)benzamide 5-tert-butyl-2-hydroxy-N,3-dimethoxybenzamide 3-[(3,4-dihydroxyphenyl)methylamino]benzenesulfonic acid 2-methylsulfonyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridine N-[4-[(6-chloro-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)sulfonyl]phenyl]acetamide 3-[2-[3,4-bis(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-1H-pyrrole-2-carboxylic acid 2-[(3,4-dimethoxyphenyl)carbamoyl]pentanedioic acid 5-bromo-N-[2-(2,4-difluorophenyl)ethyl]-4-methoxy-1H-indole-3-carboxamide 1-[2,6-difluoro-4-(7-pyridin-3-ylimidazo[5,1-b][1,3]thiazol-3-yl)phenyl]-N-methylpiperidine-4-carboxamide 5-[3-amino-4-(aminomethyl)phenyl]-N-(2,6-difluorophenyl)-1-(4-propan-2-ylsulfanylphenyl)pyrazole-3-carboxamide N-[3-(N-azidoanilino)phenyl]-4-fluorobenzenesulfonamide 7-chloro-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole 2-(4,6-difluorocyclohexa-1,5-dien-1-yl)benzamide;6-methoxy-N'-(4-phenylbut-1-ynyl)hexanehydrazide 3-[2-(benzylamino)pyridin-4-yl]-N-phenylpropanamide 3-methyl-2-[(E)-3,4,6-trimethylhept-5-enyl]pyridine 1-[1-(3,4-dihydro-2H-pyran-2-yl)propan-2-yl]-7-ethoxy-6-fluoroquinolin-4-one 1-[3-hydroxy-2-[(1E,5Z)-7-methylocta-1,5,7-trienyl]pyrido[1,2-a]benzimidazol-9-yl]ethanone 2-[3-(4-carbamimidoylanilino)propylamino]-6-(2,2-difluoroethoxymethoxy)-N-[5-(hydroxymethyl)pyridin-2-yl]pyridine-3-carboxamide 3-[(2R)-2,4-dihydroxy-5-(5-methylsulfonyloxypentoxy)cycloheptyl]-6-fluoropyrazolo[1,5-a]pyridine-7-carboxylic acid (2-ethylpyrrolidin-1-yl)-[4-[3-phenyl-4-(thiophen-2-ylmethoxy)phenyl]sulfonylphenyl]methanone N-[2,4-difluoro-3-[[6-[4-[1-(methylamino)cyclobutanecarbonyl]piperidin-1-yl]pyrimidin-4-yl]carbamoyl]phenyl]-5-fluoroquinoline-8-carboxamide 2-[3-(oxan-4-yl)propylamino]pyridine-4-carboxylic acid [3-(2,3-dihydro-1H-indene-4-carbonyl)pyrrolidin-1-yl]-[6-(2-methoxyethoxy)pyridin-3-yl]methanone 2-[3-(1H-imidazole-5-carbonyl)phenyl]acetic acid N-[3-(4-chloro-1H-pyrrolo[2,3-b]pyridin-5-yl)cyclohexa-2,4-dien-1-yl]-2-methoxybenzenesulfonamide 7-[5,6-difluoro-1-(4-methylcyclohexyl)benzimidazole-2-carbonyl]-8a-methyl-1,5,6,8-tetrahydro-[1,3]oxazolo[3,4-a]pyrazin-3-one N-[5-(1,2-benzothiazol-3-yl)-4-chlorothiophen-2-yl]sulfanyl-4-ethoxy-6-methylpyrimidin-2-amine [(3R)-1-[6-amino-5-[(2E,4Z)-hepta-2,4,6-trien-3-yl]pyridine-3-carbonyl]piperidin-3-yl]carbamic acid (2S)-6-N,2-bis[(3-methoxyphenyl)methyl]-8-N-methyl-9-(oxolan-3-yl)purine-2,6-diamine 6-amino-4-(5-chloro-2,3-difluorophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide N-(1-cyanocyclopropyl)formamide;7,8-dichloro-4,10-dihydro-1H-thieno[3,2-a]quinolizine 5-fluoro-2-N-[4-(1,3-thiazol-2-yl)cyclohexa-1,5-dien-1-yl]pyrimidine-2,4-diamine N-[4-[7'-(3-hydroxypropyl)spiro[8H-anthracene-9,2'-pyrrolidine]-1'-yl]butyl]pyridine-4-carboxamide 3-bromo-4,5-dimethyl-N-(3-propanoylphenyl)thiophene-2-carboxamide [3-(aminomethyl)azetidin-1-yl]-[4-[7-fluoro-2-[2-[2-(methylsulfanylamino)ethoxy]phenyl]furo[3,2-c]pyridin-5-yl]piperidin-1-yl]methanone;dihydrochloride 4-[5-(2,3-dimethylfuran-4-yl)-1H-pyrazol-3-yl]-6-ethoxypyrimidine (E)-3-[2,4-bis[(E)-2-(6,8-dimethyl-1,7-naphthyridin-5-yl)ethenyl]phenyl]prop-2-enoic acid (3S)-2,3-dimethyl-7-(trifluoromethyl)-4H-pyrido[1,2-a]pyrimidine 4-[2,6-di(propan-2-yl)phenyl]-1H-inden-1-ide;ethanethiolate;zirconium(4+) [2-[[4-(N-phenylanilino)cyclohexa-1,3-dien-1-yl]methyl]phenyl]boronic acid 5-azido-6,7,8-trimethylnaphthalene-1-thiol 3-(3,6-dimethoxycarbazol-9-yl)cyclohexan-1-one 3-[6-(1,2-dimethylbenzimidazol-5-yl)naphthalen-2-yl]oxypropane-1-thiol (2R)-2-[2-amino-5-bromo-4-[1-[(4,6-difluorocyclohepta-1,3,6-trien-1-yl)methyl]piperidin-4-yl]pyridine-3-carboximidoyl]pentan-1-ol 4-(methylamino)benzenesulfinic acid;6-[(2S,5R)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-quinolin-2-one 3-[4-(2,6-difluorophenyl)imidazol-1-yl]piperidine;dihydrochloride (2E,4Z)-5-[6-[4-(1-ethylsulfanylethenylamino)phenyl]quinolin-4-yl]penta-2,4-dienoic acid 3-[2,4-difluoro-N-(2-methylpropanoyl)anilino]butanoic acid 2-hydroxy-5,6-dimethoxy-3-nitroso-N-phenylbenzamide (2-benzamidoimidazo[1,2-b]pyridazin-6-yl)methylidenehydrazine 2-amino-1-(4-chloro-2,5-dimethylphenyl)-N'-hydroxy-3-pyrrolidin-1-ylpyrrolo[2,3-b]pyridine-6-carboximidamide 6-[2-(3,4-dimethoxyphenyl)ethyl]-7,8-dihydropyrido[3,2-d]pyrimidine 1-(4,5-dibromothiophen-2-yl)-N-methylideneethanesulfonamide 2-[4-(5,6-dihydro-1H-benzimidazol-2-ylmethoxy)phenoxy]acetamide 3-bromo-5-[4,6-bis(phenylsulfanyl)-1H-triazin-2-yl]benzamide N-[4-[(1Z)-3-(dimethylamino)buta-1,3-dienyl]phenyl]-2-(5-fluoropyrimidin-2-yl)-N'-pyridin-2-ylethanimidamide 2-(hydroxymethyl)-1,3-dioxoisoindole-5-carboxylic acid N'-(2,6-dichlorophenyl)-2-[2-(methylideneamino)phenyl]iminoacetohydrazide 2-[3-(5-bromopyridin-2-yl)propanoyl]-N,4-dimethyl-3,6-dioxocyclohexa-1,4-diene-1-carboxamide 3-methoxy-2,6-diphenylphenol N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)formamide;N-methyl-1-[(Z)-pent-3-en-2-ylideneamino]ethenamine N'-ethyl-N'-[4-fluoro-2,6-di(propan-2-yl)phenyl]-N-(1H-indol-3-ylmethylideneamino)-1-phenylmethanediamine N-[(2S)-3,4-dioxobutan-2-yl]-5-phenylpentanamide [(2-cyclohexylacetyl)amino]carbamodithioic acid;rhodium N-[1-(3,4-dichlorophenyl)ethenyl]-2-fluoro-6-methoxyaniline 1-[(E)-3-azidobut-2-enyl]sulfonyl-4-chlorobenzene N-(diaminomethylidene)-3,4-bis[2-(3,4,5-trimethoxyphenyl)ethyl]benzamide 2-[(6S)-1-acetyl-4,8-dimethyl-3,5,7,10-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),4,8,11-tetraen-3-yl]-N-benzylacetamide 2-(4-aminobutyl)imidazo[5,1-f][1,2,4]triazin-4-amine (5R)-3,3,4-trideuterio-4-[7-[bis(2-fluoroethyl)amino]-1-oxo-3H-isoindol-2-yl]piperidine-2,6-dione 3-[(2E,4Z)-4-methylhexa-2,4-dien-3-yl]oxybenzenethiol 5-[(3R)-1-[3,4-difluoro-2-(trifluoromethyl)phenyl]pyrrolidin-3-yl]oxy-N-[(Z)-pent-1-enyl]pyridine-2-carboxamide 3-amino-5-(3,4-dimethylcyclohexa-1,5-dien-1-yl)benzamide N-[2-chloro-5-methoxy-4-(3,3,3-trifluoropropyl)phenyl]benzenesulfonamide 3-methyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]butan-2-one 2-[(1S)-4,5,5-trimethylcyclohepta-2,6-dien-1-yl]naphthalene 3-[(3R,4R)-1-(cyclopentylmethyl)-4-pyridin-2-ylpyrrolidin-3-yl]-5-methyl-6H-triazolo[4,5-d]pyrimidin-7-one 2,4-dichloro-1-(1-phenylethenyl)benzene 2-chloro-4-(2,2-difluoroethylamino)benzoate N-[6-(3,4-dichlorophenoxy)pyridin-2-yl]benzenesulfonamide 3-(2,4-dichlorophenyl)imino-N-ethenyl-1,1,2-trimethylinden-5-amine 2-[4,5-bis(2,6-dimethylphenyl)imidazol-1-id-2-yl]ethanol;osmium(2+);trihexafluorophosphate 3-[(4E)-2,6-dimethylocta-2,4-dien-4-yl]pyridine 3-[2,6-difluoro-4-(4-propylcyclohexyl)phenyl]-7-ethoxy-1,8-difluoro-5,6,7,9-tetrahydroisoquinoline 1-[6-(difluoromethoxy)pyridin-3-yl]-4,5-bis[4-(trideuteriomethoxy)phenyl]-2H-pyrimidine 1-[4-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)piperazin-1-yl]ethanone 4-[2-(3,5-dichlorophenyl)pyridin-1-ium-1-yl]butanoic acid 1-(4-chlorophenoxy)heptane-2,6-dione (2R)-4-amino-1-(1H-benzimidazole-2-carbonyl)pyrrolidine-2-carboxylic acid 3-[(2R)-1,4-bis(4-chlorophenyl)butan-2-yl]oxy-N-diazobenzenesulfonamide 2-[(4R)-8-acetyl-3,4-dimethyl-7-oxooctyl]isoindole-1,3-dione 5-chloro-2-[[(3S)-1-(4,4-dimethylcyclohexanecarbonyl)piperidin-3-yl]amino]-4-methoxybenzamide N-[1-[(2S,4R)-2-amino-4-hydroxypyrrolidin-1-yl]-3-naphthalen-2-yl-1-oxopropan-2-yl]-4-chlorobenzenesulfonamide;hydrochloride (4-bromophenyl)-[6-hydroxy-2-[3-methylbutyl(propanoyl)amino]naphthalen-1-yl]azanium (3-benzylphenyl)methanol;ethane 3-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]-N-methylpiperidine-1-carboxamide 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-(4-phenoxyphenyl)aniline 5-chloro-2-[(2S)-1-hydroxypropan-2-yl]oxybenzonitrile [1-(2-chlorophenyl)sulfonyl-5,6-dihydropyrrolo[3,4-b]pyrrol-4-yl]methanol 6-(difluoromethyl)-N-[4-[4,5-bis(ethenyl)imidazol-1-yl]phenyl]pyridin-2-amine 1-[2,6-dimethyl-4-(pyrrolidine-1-carbonyl)phenyl]-3-methylurea N-(4-butanoylphenyl)-6,7,8,9-tetrahydropyrido[1,2-a]indole-5-carboxamide 7-(3,4-dimethoxybenzoyl)-1-azaspiro[2.5]octane-6-carboxylic acid N-(1,5-dimethylcyclohexa-2,4-dien-1-yl)-N'-[(E)-3-phenylprop-2-enoyl]oxamide 2-[(3R)-3-methylmorpholine-4-carbonyl]-1,3,4,5-tetrahydropyrido[4,3-b]indole-8-carboxylic acid 2-chloro-N-[4-(6-methyl-1H-indol-3-yl)butan-2-yl]acetamide 2-[1-(6-chloro-1,3-benzothiazol-2-yl)ethylamino]-N-[5-(trifluoromethyl)pyridin-2-yl]acetamide 1-cyclopropyl-6-fluoro-7-(2H-tetrazol-5-yl)quinolin-4-one N-(3,5-dimethylphenyl)-2-[[6-oxo-4-(propan-2-ylidenehydrazinylidene)-1H-pyrimidin-2-yl]sulfanyl]butanamide (3S)-N,1'-ditert-butyl-5-[4-(trifluoromethoxy)phenyl]spiro[2H-indole-3,3'-pyrrolidine]-1-carboxamide N-(5-benzamidopentyl)-1-oxothiane-4-carboxamide 3-[4,5-bis(ethenyl)-1H-imidazol-2-yl]benzenethiol;dichloromethane 1-[(3-propan-2-yl-7H-purin-6-ylidene)amino]ethanethiol 2-chloro-N-(5-methylpyrazin-2-yl)spiro[3.4]octane-2-carboxamide (2R,3S)-1-[4-(2-azidophenyl)-5-chloropyridin-3-yl]-2,3-dimethoxy-N,N-dimethylpyrrolidine-1-carboxamide (1-azidonaphthalene-2-carbonyl)oxidanium (3R,4R)-1-benzyl-2-tert-butylpyrrolidine N-[3-(3,5-dimethylpyrazol-1-yl)propyl]quinoline-4-carboxamide (6-amino-2-pyridin-4-ylpyrimidin-4-yl)-methylideneazanium (E)-1-[4-(cyclopropylmethoxymethyl)phenyl]ethylidenehydrazine 4-N,4-N-dimethyl-2-N-[1-[2-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)ethyl]pyrrolidin-3-yl]pyrimidine-2,4-diamine 1-[(E)-1-cyclopentylprop-2-enyl]-4-ethynylbenzene;(3R)-5-(2,6-difluorophenyl)-7-methylspiro[2H-furo[2,3-c]pyridine-3,1'-cyclobutane] 2-hydroxy-3,3-diphenylpropanoic acid 2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-(4-fluoroanilino)-6H-pyrimido[4,5-d]pyridazin-5-one 1-azido-4,5,7-trifluoroisoquinoline N-(2,3-dihydroindol-1-yl)-2-[4-methoxy-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylacetamide N-[(2S)-3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-hydroxypropyl]methanesulfonamide 1-(4-bromophenyl)sulfonyl-3-methylpiperidine 7-[(4-fluorophenyl)methyl]-6-hydroxy-8-methoxy-3-(5-methylhexanoyl)pyrano[2,3-f]chromen-9-one 2-[5-(cyclopropylcarbamoyl)-1H-pyrazol-3-yl]benzamide [(E)-7-[2-[2-methyl-3-(piperidine-1-carbonylamino)phenyl]ethoxy]hept-5-enoyl]oxidanium 7-(1,4-dichlorocyclohexa-2,4-dien-1-yl)oxychromen-2-one N-[3,5-di(propan-2-yl)phenyl]sulfanylmethanamine;1,4-dioxane 2-ethyl-1,4-di(propan-2-yl)naphthalene N-[(E)-1H-indol-3-ylmethylideneamino]-5-methoxy-6,7-dihydroquinoline-8-carboxamide (2S,3R)-N,N-dimethyl-2-[1-oxo-8-(trifluoromethylsulfonyloxy)phthalazin-2-yl]oxolane-3-carboxamide 1-(4,6-dimethyl-2-oxopyran-3-yl)sulfonylpyrrolidine-3,4-dione N-[2-oxo-3-[(E)-3-phenylprop-1-enyl]cyclopentyl]furan-3-carboxamide 2-[4-(1,3-diethylimidazol-1-ium-2-yl)pyridin-1-ium-1-yl]ethanesulfonic acid;bromide 2-(4-azidooxyphenyl)sulfonyl-4,6-ditert-butylphenol 5-bromo-4,7-difluoro-2,3-bis(trifluoromethyl)benzimidazole 2-(1H-imidazol-5-yl)-6,7-dimethoxy-3-[(4-propylphenyl)methyl]chromene-2,4-dione N-(2,5-difluorophenyl)-6-hydroxy-7-methoxy-1'-oxospiro[4H-isoquinoline-3,3'-azetidine]-2-imine N-[(1R)-6,7-dichloro-2-oxo-3,4-dihydro-1H-quinolin-5-yl]-5-methyl-6-oxo-1,4-dihydropyridazine-3-carboxamide 4-[(2E,4Z)-5-[2-aminoethyl-[[3-methoxy-4-(trifluoromethyl)phenyl]methyl]carbamoyl]hepta-2,4,6-trien-2-yl]-N-methylpyridine-2-carboxamide;propane ethane;3-methylpiperidine;1-(4-piperidin-4-yloxyphenyl)pyrrolidin-2-one [3-(1-benzothiophene-2-carbonylamino)-5,6,7,8-tetrahydronaphthalen-2-yl]methylcarbamic acid 1-(1-azidoethyl)benzo[f]quinazoline 4-[3-(2,6-dioxopiperidin-3-yl)-1,2-benzoxazol-5-yl]-N',N'-dimethylpiperidine-1-carboximidamide 1-[3-(2,4-dimethylpyrazol-3-yl)azetidin-1-yl]sulfonyl-3,4-dihydro-2H-quinoline 5-N-[1-(2,6-dimethylphenyl)ethylideneamino]-3-N-methylpyrazolo[1,5-a]pyrimidine-3,5-diamine N-[(5S,7R)-7-chloro-5-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-3-fluorobenzamide 1-(3,4,6,7,8,9-hexahydropyrazino[2,1-c][1,4]oxazin-1-yl)-4-phenylbutane-1,4-dione 4-(2,3,5,6-tetrachloropyridin-4-yl)-1H-pyrazole 2-[2,3-bis(trifluoromethyl)phenyl]-N-(4-cyclohexa-1,5-dien-1-ylbut-1-ynylsulfanyl)-1,3-thiazole-5-carboxamide 2-[4-(1,3-benzodioxol-5-yl)phenyl]-2-imino-1-[(2R,4S)-4-methoxypyrrolidin-2-yl]ethanone 1-[2-(4-bromo-N-(8-hydroxynaphthalen-1-yl)-3,5-dimethoxyanilino)ethyl]piperidine-4-carboxylic acid 7-methoxy-3,4,6,9,10,10a-hexahydro-2H-phenanthrene 1-(azidomethylsulfonyl)-4-chlorobenzene 2-[(5R,10bS)-7-methoxy-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 5-[(4S)-3,8-dimethyl-4,7-dihydro-1H-pyrazolo[3,4-b]isoquinolin-4-yl]-2-propan-2-ylidenepyrrole-3-carbonitrile 1-[3,5-bis(trifluoromethyl)phenyl]-2-[4-chloro-6-oxo-5-[(3R)-oxolan-3-yl]pyridazin-1-yl]ethanone 2-(4-amino-1,3,5-triazin-2-yl)sulfanyl-1-phenylethanone (Z)-2-hydroxy-3-(4-methylphenyl)-N-phenylprop-2-enamide (4-fluorophenyl)-[3-(1H-pyrrolo[2,3-b]pyridin-5-ylamino)piperidin-1-yl]methanone 1-[(2,4-dichlorophenyl)methyl]-3-[(1S)-2-(dimethylamino)cyclopentyl]urea (2R,3S)-N'-[1-(4-fluorophenyl)-5-methylpyrazole-4-carbonyl]-2-[4-[4-(trifluoromethoxy)phenoxy]phenyl]oxane-3-carbohydrazide 2-[(1R,5S)-3-[6-[(Z)-hydroxyiminomethyl]pyridin-2-yl]oxycyclohexyl]acetic acid N-(3,4-dichlorophenyl)-2-[6-methoxy-5-(4-morpholin-4-ylpiperidine-1-carbonyl)indol-1-yl]acetamide [3-cyclopropyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl(hydroxy)methyl]phosphonic acid 2-[7,8-difluoro-6-(trideuteriomethoxy)naphthalen-1-yl]-5-(4-pentoxyphenyl)pyrimidine 2-[(3R,4S)-4-hydroxypyrrolidin-3-yl]-N-(4-piperidin-1-ylpyridin-3-yl)acetamide 2-(3,5-dibromo-4-cyanophenyl)sulfonyl-N-phenylbenzamide N-[(3,4-difluorophenyl)methyl]-5-hydroxy-2,6-dimethylpyrimidine-4-carboxamide N-[3-[2-(4-ethylphenyl)imino-3,6-dihydro-1,3,4-thiadiazin-5-yl]phenyl]methanesulfonamide N-butyl-2-[4-(ethylaminomethyl)phenyl]sulfanyl-5,6,7,8-tetrahydroquinazolin-4-amine N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-fluorobenzenesulfinamide;ethane 1-[5-chloro-2-(difluoromethoxy)phenyl]ethylphosphane 2-[(5-tert-butylthiophene-3-carbonyl)amino]-4-[2,6-dichloro-4-(1-oxopentan-2-yloxymethyl)phenyl]butanoic acid 2,4-dinitro-6-[5-(oxolane-3-carbonyl)cyclohepta-1,3,6-trien-1-yl]sulfanylbenzaldehyde (2R)-N-[5-chloro-4-methyl-1-[3-(trifluoromethoxy)phenyl]sulfonylpyrazol-3-yl]-2-hydroxy-N,3-dimethylbutanamide 4-(6,8-dihydro-5H-imidazo[2,1-c][1,4]oxazin-3-ylsulfamoyl)-N,N-dimethylbenzamide N-[3,5-bis(trifluoromethyl)phenyl]-2-[4-oxo-6-[2-(4-piperidin-1-ylpyrrolidin-1-yl)pyridin-3-yl]pyrido[2,3-d]pyrimidin-3-yl]acetamide 2-[5-carbamoyl-9-[(4-methylphenyl)methyl]carbazol-4-yl]-2-hydroxyacetic acid (3R)-2-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxylic acid 2-amino-3-[4-chloro-7-hydroxy-6-(2-hydroxyethyl)naphthalen-1-yl]oxypropanoic acid 1-azido-2,3-bis(benzenesulfonyl)guanidine (2-azidopyridin-4-yl)methanol 2-[(1Z,3E)-4-aminohexa-1,3,5-trienyl]benzonitrile N-[2,6-dichloro-4-(1H-pyrazol-5-yl)phenyl]-3,3-bis(hydroxymethyl)cyclobutane-1-carboxamide 2-hydroxy-4-methylsulfanylanthracene-9,10-dione 5-cyclopentylsulfanylpyrimidine-4-carboxylic acid 1-(2,4-dichlorophenyl)-2-imino-4,5-dihydropyrano[3,2-c]chromene-3-carbonitrile N-(2,3-dimethoxyphenyl)-4-iminopentanamide (3S)-N-methyl-1-[6-[(E)-prop-1-enyl]cyclohexa-2,4-dien-1-ylidene]-5-pyridin-2-ylsulfonylpyrrolidine-3-carboxamide 6-bromo-1'-[2-(dimethylamino)-4-propan-2-yloxybenzoyl]spiro[3H-chromene-2,4'-piperidine]-4-one;hydrochloride 1,3-bis(4-ethenylcyclohexyl)benzene 2-(cyclohexylamino)-5-fluoro-6-[(3S,4S)-3-hydroxy-1-methylpiperidin-4-yl]pyridine-3-carboxamide 3-[4-(2,3-dihydro-1H-inden-2-ylamino)quinazolin-6-yl]-5-methoxyphenol 6-(2,4,5-trimethylphenyl)-[1]benzofuro[3,2-c]pyridine N-methyl-4-(trifluoromethyl)aniline;hydrochloride 2-[(E)-(4-hydroxyphenyl)methylideneamino]oxybenzoic acid 3-[2-chloro-5-(trifluoromethyl)phenyl]-1H-indole 5-amino-3-[2-(difluoromethoxy)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile 2-(4,4,4-trifluoro-2-methoxybutanoyl)oxybenzoate 1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxy-3-methylbenzene (1R)-N-[1-[4-[2-ethyl-5,6-dimethoxy-3-[(E)-2-nitroethenyl]phenyl]sulfonylpiperazin-1-yl]-3-hydroxy-1-oxopropan-2-yl]-1-[4-fluoro-3-(trifluoromethyl)phenyl]cyclopropane-1-carboxamide (Z)-3,7-diethyl-6-hydroxynon-5-en-4-one;5-[(2-methylpropan-2-yl)oxycarbonyl]furan-2-carboxylic acid N-[5-(2,6-dichlorophenyl)-3H-pyrrol-4-yl]-1-methylazepane-4-carboxamide 6-[3-(cyclopentylmethoxy)phenoxy]-2,2,4-trimethylquinoline 7-[5-(2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-3-yl]quinolin-8-ol N-[(3S)-1,2,5-trioxopyrrolidin-3-yl]naphthalene-1-sulfonamide (2R)-N-[3-chloro-4-(difluoromethylsulfanyl)phenyl]-6,6,8,8-tetraethyl-5,7-dihydronaphthalene-2-carboxamide 3-ethylsulfanyl-6-(3-fluorophenyl)-4H-1,2,4-triazin-5-one 7-[2-(4,5-dihydrobenzo[g]quinolin-2-yl)hydrazinyl]-6-methoxychromen-4-one 5-N-[(3R)-oxolan-3-yl]-7H-pyrrolo[2,3-d]pyrimidine-4,5-diamine 2-chloro-7-(3,5-difluorophenyl)thieno[3,2-d]pyrimidine;ethane 2-methylsulfonyl-4-[2-oxo-3-(pyridin-3-ylmethyl)imidazolidin-1-yl]benzoic acid 2-(2,4,6-trifluorophenyl)pyrimidine [[2-amino-3,4-bis(trifluoromethyl)phenyl]-(1,3-dihydropyrazol-2-yl)methylidene]azanium 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3H-1,3-benzothiazole N'-hydroxy-4-[(1,3,3-trimethylcyclobutyl)amino]pyridine-2-carboximidamide 5-tert-butyl-2,3-diphenyl-1H-pyrrole;ethane 2-[(2S)-4-(1,3-dihydroisoindole-2-carbonyl)pyrrolidin-2-yl]-7-ethoxy-3H-quinazolin-4-one 3-methyl-N,4-diphenylaniline 4-[2-[5-(3,6-dihydro-2H-pyridine-1-carbonyl)-4-methyl-2-oxo-1H-pyridin-3-yl]-3H-benzimidazol-5-yl]piperazine-1-carboxylate 2-[6-(3,5-dimethoxyphenyl)pyridin-2-yl]-N-(2,4,5-trifluoro-3,6-dihydro-1H-pyridin-4-yl)acetamide;ethane 1-[(2S,5R)-4-[4-chloro-6-[(3-fluoropyridin-4-yl)methoxy]quinolin-7-yl]sulfonyl-2,5-dimethylpiperazin-1-yl]prop-2-en-1-one 2-chloro-N-[3,5-bis(trifluoromethyl)phenyl]quinoline-6-carboxamide 4-methyl-N-[1-(3-methylbutyl)pyrrolidin-3-yl]pyrimidine-5-carboxamide 3-[1-(3,4-dimethoxyphenyl)butan-2-ylamino]propanal 3-(1,3-benzothiazol-2-yl)-5-[[4-(hydroxymethyl)phenyl]diazenyl]-1H-pyrazole-4-carbonitrile 4-[4-chlorobutyl(2,3-dihydroxypropyl)amino]benzenesulfonic acid 3-methyl-N-(2,5,5-triphenylcyclopenta-1,4-dien-1-yl)aniline 4-[6-fluoro-2,3-dimethyl-5-[4-(trifluoromethoxy)phenyl]benzimidazol-1-ium-1-ylidene]butanenitrile 7,8-dimethoxy-6-(4-methylsulfinylphenyl)pyrido[2,3-d]pyrimidine 2-(2,5-diethoxyphenyl)benzene-1,4-diol 1-cyclopropyl-N-[4-methoxy-2-(2-oxoimidazolidin-1-yl)phenyl]triazole-4-carboxamide N-[2,3-dihydroxypropyl(hexadecanoyl)amino]benzamide 6-(2,5-difluorophenyl)sulfanyl-3H-thieno[3,2-d]pyrimidin-4-one 1-(2-azido-2-methoxyethyl)-4-[3-[4-(trifluoromethyl)phenyl]prop-2-enoyl]piperazine-2,5-dione 5-bromo-4,6-difluoro-2-pyrimidin-2-yl-1H-benzimidazole 1-[(3S,4R)-1-[(5-methylpyridin-2-yl)methyl]piperidin-4-yl]triazole-4-carboxylic acid 2-azidooxy-1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]ethanone 3-butyl-6,8-dichloroimidazo[1,2-b]pyridazine 2-[4-(3,5-dimethylpyrazole-1-carbonyl)piperazin-1-yl]pyridine-4-carbonitrile 3-(4-methylphenyl)sulfonylaniline [1-[(Z)-2-aminoethenyl]piperidine-3-carbonyl]-methylidene-[4-(5,7,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),2,4,8,10-pentaen-13-ylsulfonyl)phenyl]azanium [2-bromo-5,6-dichloro-4-(1H-indole-3-carbonyl)phenyl]chloranium 4-[4-[(2S,3R)-1,5-dioxo-2-phenylpyrrolidine-3-carbonyl]piperazin-1-yl]benzaldehyde (5-chloro-2,3-dihydro-1H-inden-4-yl)azanide;dimethoxyethane;yttrium(3+) ethane;3-methoxy-2,5,6-triphenylphenol 4-[1-(4-hydroxyphenyl)-1-[4-(trifluoromethyl)phenyl]ethyl]phenol N-[2-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]ethoxy]-4-fluorobenzamide 3-[4-[(5-chloropyridine-2-carbonyl)amino]pyrazol-1-yl]pyrrolidine-1-carboxylate 3-chloro-5-[(Z)-2-(4-ethoxyphenyl)-2-hydroxyethenyl]-1,3,4-oxadiazole-2-thione 4-[[7-(1H-indazol-6-ylamino)quinazolin-2-yl]amino]cyclohexan-1-ol 4-[[2,6-dibromo-4-(trifluoromethoxy)phenyl]iminomethyl]benzene-1,3-disulfonic acid 1-(5-bromo-2,3-dihydroindole-1-carbonyl)pyridin-4-one 4-(1,3-benzodioxol-5-yl)-N'-[4-[N-cyclohexa-2,4-dien-1-ylidenecarbamimidoyl]phenyl]piperidine-1-carboximidamide (2S,3R)-N-hydroxy-1-[4-[[5-(4-isocyano-2-phenylmethoxyphenyl)pyrimidin-2-yl]amino]benzoyl]pyrrolidine-2-carboxamide 2,3-dichloro-N'-(4,5-dimethylfuran-2-carbonyl)benzohydrazide [1-(2,5-dihydroxyphenyl)cyclopentyl]azanium 5-(4-azidooxyphenyl)-7,8-dihydro-6H-pyrido[2,3-d]pyrimidine 5-[5-(5,6-dimethylpyrazin-2-yl)furan-2-yl]imidazolidine-2,4-dione 4-(5,7,10,12-tetrazatricyclo[6.3.0.02,6]undeca-1(8),9-dien-11-ylsulfanylmethyl)oxan-4-ol [2-(aminomethyl)pyrrolidin-1-yl]-[2-methanimidoyl-3,4-dimethoxy-5-(trifluoromethylsulfanyl)phenyl]methanone 4-[(1Z,3E)-4-(3-ethyl-5-methoxyphenyl)buta-1,3-dienyl]morpholine 5-methoxy-4-methyl-2-[2-(trifluoromethyl)pyridin-4-yl]-1H-pyrimidin-6-one 1-[4-(6,11-dihydrobenzo[c][1]benzazepine-5-carbonyl)-3,6-dihydro-2H-pyridin-1-yl]ethanone 2-(aminomethyl)-6-bromo-3H-thieno[3,2-d]pyrimidin-4-one 1-(6-bromopyridin-2-yl)-3,5-dimethylpyrazole-4-carboxamide N-benzyl-2-[4-(4-bromophenyl)sulfanyloxyphenyl]acetamide 1-(4-aminobutyl)quinoline-2,3,4-trione N-[2,6-di(propan-2-yl)phenyl]-N-ethylcarbamate 3-(cyclopropylmethylamino)-N'-[3-[4-(ethylideneamino)phenyl]-1,2-oxazol-5-yl]pyrazine-2-carboximidamide 2-methoxy-6-(6-methylpyrazin-2-yl)pyridine 2-(2,6-dichloro-N-cyclohexyl-4-nitroanilino)propanoic acid 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-[[(Z)-(2-hydroxynaphthalen-1-yl)methylideneamino]carbamothioyl]propanimidamide 3-[5-(1,2,4-triazol-1-ylmethyl)furan-2-yl]pyrazine-2-carbonitrile 1-[4-bromo-2,5-dimethyl-N-(2-phenylethyl)anilino]propan-2-one 2-[1-(4-bromobenzoyl)-3,6-dihydro-2H-pyridin-5-yl]acetic acid (Z)-2,6-dimethoxyhex-3-ene;1-methyl-4-phenylcyclohepta-1,3,5-triene N-(4-azidophenyl)-2,2-dimethylpropanamide N-[4-(2,6-dimethoxyphenyl)-5-(5-oxo-1H-pyrazol-3-yl)-1,2,4-triazol-3-yl]cyclohexanecarboxamide 6-[(Z)-1-amino-3-iminoprop-1-en-2-yl]-N-[4-(difluoromethoxy)phenyl]imidazo[1,2-a]pyridine-2-carboxamide (E)-N',2-diamino-3-[5-[4-(6-chloropyridin-2-yl)piperazine-1-carbonyl]-2-methoxyphenyl]prop-2-enimidamide 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-4-[1-(methoxymethyl)cyclopentyl]-1H-1,2,4-triazol-5-one 4-N,6-N-bis(2-chloroethyl)-4-N,8-N,8-N-trimethylquinazoline-4,7,12-triamine 1-methoxy-2,4,6-triiodo-3,5,8-tris[(Z)-prop-1-enyl]naphthalene 2-amino-4-(3,5-dichlorophenyl)-4H-pyran-3,5-dicarbonitrile 1-[(2R,4S)-2-tert-butyl-4-hydroxypiperidin-1-yl]-2-(4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl)ethanone 5-[2-(3,4-dichlorophenyl)ethyl]-2,6,9-trimethyl-8H-pyrimido[4,5-e][1,4]diazepine 2-methylsulfonyloxyethoxy-(3-phenylprop-2-enoylamino)borinic acid 2-[(5Z)-3-hydroxy-6,7-dimethylocta-5,7-dien-2-ylidene]-6,8-bis(3-methoxyphenyl)-4a,8a-dihydronaphthalen-1-one 7-amino-2-hydroxyacridine-1,8-dicarboxylic acid (3E,5Z)-N,4-dimethyl-6-(8-methylnaphtho[2,1-b][1]benzofuran-9-yl)hexa-1,3,5-trien-3-amine 1-(4-bromophenyl)sulfonyl-3-ethoxybenzimidazol-2-one 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)cyclopentan-1-one (7R)-N,3-dimethyl-5-oxo-6,7-dihydro-4H-[1,2]oxazolo[5,4-c]pyridine-4-carboxamide 4-(3,6-dihydro-2H-pyran-5-yl)-2-methylquinoline;7H-pyrrolo[2,3-d]pyrimidin-4-amine [1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-6-carbonyl)pyrrolidin-3-yl]methanesulfonamide 3-(6-chloro-5-cyanopyridin-2-yl)-N,N,4-trimethyl-1H-pyrrole-2-carboxamide N-(1,3-benzodioxol-5-ylmethyl)-2,4-dichloroaniline N-[5-(1H-indol-3-yl)-2-methoxyphenyl]-N',N',N'-trimethylethane-1,2-diamine 3-fluoro-5-(1H-indole-2-carbonyl)benzaldehyde 5-(4-benzylpiperazin-1-ium-1-ylidene)-2,3-dimethyl-1,2-benzothiazole 1-[4-methylsulfonyl-2,6-di(propan-2-yl)phenyl]imidazole 4-[[1,3-dihydroisoindol-2-ylmethoxy(1H-indol-6-yl)phosphoryl]amino]cyclohexan-1-ol (2R)-3-(6,7-dimethoxyisoquinolin-1-yl)sulfonyl-N'-hydroxy-4-(methanesulfonamido)butanimidamide 1-(3,4-difluorophenyl)-5,6-dimethoxy-2H-indole 2-(4-fluorophenyl)-1,5-dimethylpiperidine;4-formylbenzenesulfonic acid 1-[(Z)-2-cyano-3-[4-(diethylamino)phenyl]prop-2-enoyl]pyrrolidine-3-carboxylic acid 1-[4,4-bis(4-methylphenyl)but-2-en-2-yl]-6-hydroxycyclohepta-3,5-diene-1,3-dicarboxylic acid 1-[2-amino-4-(2,5-difluorophenyl)-6-[2-methyl-5-(4-methylpiperazin-1-yl)phenyl]phenyl]ethanone 2-[5-[3,4-bis(ethenyl)pyridin-2-yl]-6,7-dihydro-1H-indazol-3-yl]propan-2-ol 1-methyl-3-propan-2-ylbenzene;6-(methylideneamino)pyrimidine-4,5-dione N-[(3R,4S)-1-benzyl-4-methoxypyrrolidin-3-yl]-N-(3-phenylpropyl)acetamide;hydrochloride 6-[2,5-difluoro-4-[2-(3-methylazetidin-1-yl)ethoxy]phenyl]pyridine-2-carboxamide 5-[(2S,3R)-1-ethyl-4-oxoazetidin-2-yl]-8-fluoro-1H-pyrrolo[3,2-b]quinoline-2-carbonitrile N-azido-4,6-diphenylpyridin-3-amine N-(2,4-dichloropyrimidin-5-yl)-N-[4-(pyridin-2-ylsulfamoyl)phenyl]benzamide N-[(2S)-3-chloro-1-hydroxypropan-2-yl]benzamide;N,2-dimethoxyaniline (1E,4Z,8Z)-2-bromo-7,12-diazatricyclo[6.3.0.02,5]undeca-9,11-dien-8-ol 3-fluoro-6-iodoquinoline 2-chloro-6-(3,3-difluorocyclohexyl)oxypyridine 1-[(4-nitrophenoxy)methyl]-3-undecylurea 4-[6-(N-aminoanilino)pyridin-2-yl]-1,2-dihydronaphthalene-1,3-diol 6-(azetidin-1-yl)-3,4-dihydrochromen-2-one 6-[2-(2-aminopyridin-4-yl)oxyethyl]pyridazine-3,4-diamine 4-(2,3-dichlorophenyl)sulfonyl-N-[3-fluoro-4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]piperidine-1-carboxamide N-methylsulfonyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide N'-[4-cyano-2,6-di(propan-2-yl)phenyl]-2,5,7,8-tetramethylnonanehydrazide 1-[(2S,3R)-2-methyl-3-phenylbutanoyl]pyrrolidine-2-carboxamide (4S)-1,3-dimethyl-4-[2-(trifluoromethoxy)phenyl]-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one N-(3,3a,4,5,6,7,7a-octahydro-1H-2,6-benzodioxazol-5-ylmethyl)-2-phenylimidazo[2,1-b][1,3]thiazole-6-carboxamide (2S,4R)-1-acetyl-N-[(3-chlorophenyl)methyl]-4-hydroxy-4-methoxypyrrolidine-2-carboxamide 5-[[6-(trifluoromethoxy)-1,3-benzoxazol-2-yl]amino]benzenesulfonamide 1-[2,5-dichloro-4-(3,3,3-trifluoropropyl)phenyl]ethanone 5-bromo-4,6-dimethylbenzene-1,2,3-tricarboxylic acid N-cyclopropyl-5-methoxy-4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]pyridine-2-carboxamide 1-[3-(4-methylphenoxy)phenyl]ethanamine 5-[(1R)-2-azidocyclohexyl]oxy-1H-indazole N-[3-chloro-4-[[(5Z)-4-oxo-5-[[2,4,6-trifluoro-3-(tetrazol-1-yl)phenyl]methylidene]-1,3-thiazolidin-2-ylidene]amino]phenyl]acetamide N-[1-amino-3-(2,4-difluorophenyl)-3-oxopropan-2-yl]pyrimidine-5-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]sulfanylpropanamide;3-(4-propan-2-ylcyclohexa-1,3-dien-1-yl)-6-[4-[2-(triazol-1-yl)ethoxy]piperidin-1-yl]pyridazine 2-[N-(4-bromobutan-2-yl)-3,5-dichloroanilino]ethanol 3-(6-methyl-2-oxo-1,3-benzoxazol-3-yl)pyrrolidine-2,5-dione N-methoxy-N,5-dimethyl-2-(4-phenyl-1,3-thiazol-2-yl)pyrazole-3-carboxamide N-[3,4-bis(ethenyl)phenyl]-2-chloro-4-methanimidoyl-5H-1,3-thiazol-4-amine 4-(3,7-dimethyloctanoyloxy)phthalic acid 1-benzyl-2,3,4a,5-tetrahydropyrido[2,3-b]quinoxaline 2-chloro-4-[(E)-3-(diethylamino)prop-1-enyl]aniline;ethane 6-[4-fluoro-3-(trifluoromethoxy)phenyl]-N,8,8-trimethyl-2-sulfanylidene-5,7-dihydropyrimido[4,5-d]pyrimidine-7-carboxamide (2S,3S)-1-azido-3-[[4-(4-methoxyphenyl)butanoylamino]methyl]-N-methylsulfonylpyrrolidine-2-carboxamide 3-[(1S)-1-azidoethyl]-N-methylbenzamide [(5E)-1,3-bis(3-chlorophenyl)octa-5,7-dienyl]phosphane 4-[[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]methylideneamino]benzenethiol;4-hexan-2-ylmorpholine 1-[(E)-4-[4-methanimidoyl-3-[[5-methoxy-7-(morpholin-2-ylmethoxy)quinazolin-4-yl]amino]phenyl]but-3-en-1-ynyl]cyclopropane-1-carbonitrile 1-[1-(2,5-difluorobenzenecarbothioyl)piperidin-4-yl]-3H-imidazo[4,5-c]pyridin-2-one 4-N-[(2R)-6,7-dimethoxy-2-[[4-(1H-pyrazol-5-yl)benzoyl]amino]heptanoyl]cyclohexane-1,4-dicarboxamide (1Z,3E)-3-[5-amino-6-(4-fluorophenyl)pyrazine-2-carboximidoyl]penta-1,3-dien-1-amine 2-(3,5-dimethylanilino)-N'-hydroxypyridine-4-carboximidamide 3-[1,1-difluoro-2-(4-fluorophenyl)ethyl]-6-(5-methoxypyrazin-2-yl)-[1,2,4]triazolo[4,3-a]pyridine 1-(1H-indole-3-carbonyl)-2,3,4,6-tetrahydropyrrolo[3,4-c]pyrrole-5-carboxylic acid 2-[(Z)-[amino-[6-methyl-3-propan-2-ylidene-4-(pyridin-3-yloxymethyl)pyrazin-2-yl]methylidene]carbamoyl]benzoic acid 1-[4-methyl-3-(trifluoromethoxy)phenyl]pentan-2-amine 5-[3-[[(1S,2R)-2-aminocyclohexyl]iminomethyl]-1H-indol-6-yl]-N-cyclohexylthiophene-2-carboxamide [3-(3,5-dimethylpyrazol-1-yl)phenyl]urea 2-[5,6-dichloro-1-(2-pyridin-3-yloxyacetyl)indol-3-yl]benzoate 2-[4,5-bis(ethenyl)-3,6-dimethylidenecyclohexa-1,4-dien-1-yl]-1,5-dimethoxynaphthalene 2-[5-bromo-1-(3,4,5-trimethoxyphenyl)sulfanylindol-3-yl]ethylphosphonic acid 1-(2,4-dichlorophenyl)heptan-3-one (3S)-1-methyl-5-oxo-N-[(2,4,6-trifluorophenyl)methyl]pyrrolidine-3-carboxamide 1,3-di(propan-2-yl)pyrrole-2-carbothioate;triethylazanium N-cyclopropyl-3,5-bis(4-methoxyphenyl)-1H-pyrazole-4-carboxamide N-(azidomethyl)-2,6-dichlorobenzenesulfonamide 5-(4-methoxyphenyl)-2-[4-[3-[3-(4-methylpiperazin-1-yl)propyl]pyrrolidin-1-ium-1-ylidene]cyclohexa-2,5-dien-1-ylidene]thieno[3,2-d]pyrimidine N-[3-[[(2S)-5-[[4-[6-(dimethylamino)pyridin-3-yl]oxycyclohexanecarbonyl]amino]-1,2,3,4-tetrahydronaphthalene-2-carbothioyl]amino]phenyl]furan-2-carboxamide 2-(3-azidopiperidin-1-yl)benzonitrile 3,5-ditert-butyl-4-[2-(2,4-difluorophenyl)propan-2-yl]aniline 4-[5-(azidomethyl)furan-2-carbonyl]piperazine-1-sulfonamide 2-[3-(4,4-dimethylpentoxy)phenoxy]-6-methyloxane (2R)-1-ethoxycarbonyl-6,7-dimethyl-3-phenyl-2H-benzimidazole-5-carboxylic acid 2-benzyl-N,3-dimethoxyaniline 4-(3,5-dibromophenyl)-2-(4-iodophenyl)-6-(2-methylprop-1-enoxy)pyridine 3,4-dibromo-5-[2-(1,2,4-oxadiazol-3-yl)-5-phenylthieno[2,3-d]pyrimidin-6-yl]benzaldehyde 4-methoxy-3,5,6-tri(propan-2-yl)aniline N-(1-bicyclo[2.2.2]octanyl)benzamide N-[1-(4-methyl-6,7,8,9-tetrahydrocyclohepta[b]pyridine-2-carbonyl)piperidin-4-yl]ethenesulfonamide 1-[4-(3,3-dimethylpentyl)phenyl]azetidine 2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridine-5-carbonyl)azetidine-1-carboxylic acid 4-[[4-(cyclohexanecarbonylamino)phenyl]sulfonylamino]benzoic acid 1-[5-tert-butyl-2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(thiophen-2-ylmethyl)urea 1,2-bis(chloromethyl)naphthalene N-(1,3-benzothiazol-2-yl)-4-[5-methyl-4-(methylideneamino)-6-oxopyridazin-1-yl]butanamide N-[3-(4-bromophenyl)propyl]benzamide;ethane 2-(3-methoxy-4-nitrophenyl)sulfonylacetic acid 3-(2,4-difluorophenyl)sulfanylfuran (2S,3R)-N'-cycloheptyl-1-ethoxycarbonyl-N,2-dimethylpiperidine-3-carbohydrazide;(Z)-3-[methyl-[4-(trifluoromethyl)phenyl]hydrazinylidene]but-1-ene (5E)-5-[(2,4-difluorophenyl)methylidene]-1-(4-phenoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione 2-(4,5-dimethyl-1H-pyrazol-3-yl)-1-(4-propoxypiperidin-1-yl)ethanone 4-[[(2R)-1,4-dioxan-2-yl]methoxy]-5-fluoro-6-(2,2,3,3,4,4,5,5,6,7,8,9,9-tridecafluorodecoxy)pyrimidine N-(2,6-dimethoxypyrimidin-4-yl)-4-[ethenylsulfonyl(propyl)amino]benzenesulfonamide (6S)-2,5-dimethyl-4-(3-nitrophenyl)-1,6-dihydropyridazine 3-(1H-benzimidazol-2-yl)-4-fluorobenzamide 2-(3,6-dihydro-2H-pyran-5-yl)benzenesulfonamide 2-[N-[(3-fluorophenyl)methyl]-4-phenoxyanilino]propanoic acid [3-[(2Z)-2-ethenylpenta-2,4-dienoxy]phenoxy]boronic acid 3-chloro-6-[(E)-2-(4,5-dimethylimidazol-1-yl)ethenyl]-7-fluoroquinoline (1S,2R)-3-[4-hydroxy-5-(2,3,6-trifluorophenyl)pentanoyl]oxy-2,3-dihydro-1H-indene-2-carboxylic acid N-[(Z)-1-amino-3-(methylamino)prop-2-enylidene]-3-cyano-4-ethylbenzamide 4-[4-[5,6-diamino-8-(2H-pyrrol-2-yl)purin-9-yl]phenoxy]butanamide (Z)-3,7-bis[(4-methoxyphenyl)methyl]-6-methylnon-5-ene-1-sulfonate (3S,5R)-N-[2-(4-aminophenoxy)ethyl]-7-methoxy-1-(pyridine-3-carbonyl)-5-pyridin-4-yl-2-thiophen-3-yl-2,3-dihydro-1H-imidazo[1,2-a]benzimidazole-8-carboxamide 6-[4,5,9-trimethyl-7-(oxan-2-yloxy)pyrrolo[1,2-a]quinoxalin-10-ylidene]-7H-imidazo[5,1-c][1,4]thiazine (2S)-3-[4-chloro-3-[(1,3-dioxoisoindol-2-yl)methyl]phenyl]-2-(9H-fluoren-9-ylmethoxycarbonylamino)propanoic acid 3-[5-(1,2,3,4,6,7-hexahydroisoquinolin-7-yl)-1H-indazol-3-yl]-1-[1-(2-morpholin-4-ylethyl)piperidin-4-yl]-1-phenylurea 4-[2-(4-methylpiperazin-1-ium-1-ylidene)ethyl]phenol 5-fluoro-3,8-dimethoxy-1-trityl-2H-quinoline 2-(3,5-dimethylphenyl)-7-[4-[(1R)-1-hydroxybutyl]piperidine-1-carbonyl]-9H-pyrimido[4,5-b]indole-8-carbonitrile (3-bromo-2,4-dichlorophenyl)boronic acid 2-[(3S)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-3-yl]oxypyridine-4-carbonitrile 1-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-yl)-6-methoxy-2H-indazol-3-one N-[1,2,3,5,6,7-hexahydro-s-indacen-4-yl(sulfamoyl)methylidene]hydroxylamine N-(2,3-dihydro-1H-imidazo[1,2-b]pyrazol-7-ylmethyl)-4-fluorobenzenesulfonamide 5-[1-(3,4-dihydro-2H-chromene-6-carbonyl)piperidin-3-yl]-3H-1,3,4-oxadiazol-2-one N'-[2,3-difluoro-5-[(1R)-1-[4-(trideuteriomethoxy)phenyl]ethyl]phenyl]oxamide 2-[1-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)piperidin-4-yl]acetonitrile N-[1-(2,3-dimethoxyphenyl)ethyl]-6-methylimidazo[4,5-b]pyridine-3-carboxamide 5-(1,3-benzodioxol-4-yl)-7-ethoxy-2H-pyrido[4,3-d]pyrimidine N-[5-fluoro-4-[2-(hydroxymethyl)-6,7-dimethoxyquinoxalin-5-yl]oxy-2-nitrophenyl]methanesulfonamide 4-bromo-2,3-dimethylnaphthalene-1-carboxamide 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-7-(trideuteriomethoxy)quinoline 2-[3,5-dichloro-4-(3-methylsulfonylphenyl)sulfanyloxyphenoxy]propanoic acid ethane;4-(2,3,7,10-tetramethoxyanthracene-9,10-diyl)benzaldehyde N-(4-anilinophenyl)-N-(3,5-dichlorophenyl)sulfonylbenzamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-methoxy-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide 2-[4-[(E)-3-[4-[5-[3-cyano-1-(cyclopropylmethyl)indol-6-yl]pyridin-2-yl]piperazin-1-yl]-3-oxoprop-1-enyl]phenyl]guanidine 2-[4-(4-amino-7,8-dihydropyrimido[5,4-f][1,3]benzoxazol-6-yl)phenyl]ethanamine 1-[[(E)-3,5-dimethoxybut-2-enyl]amino]-7-phenylheptane-1,3-dione 5-bromo-3,4-dimethoxy-N-[2-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)cyclohexyl]thiophene-2-carboxamide 5-chloro-4,6-dideuterio-2,3,7-trideuterio-8-[[6-fluoro-1-(oxetane-3-carbonyl)indol-5-yl]amino]quinoline-8-carbonitrile 3-[4-(benzoylsulfamoyl)-N-cyclohexylanilino]butanoic acid 2-(3,5-dimethylphenyl)-5H-chromeno[4,3-c]pyridazine-1,9-dione 2-benzylsulfanyl-4-(8,9,10,11-tetrahydronaphtho[3,2-e]indol-7-yl)aniline 1-(3,4-dimethylphenyl)sulfonyl-5-fluoroindole-2-carboxylic acid 6-[(3S)-1-(4-chlorobenzoyl)piperidin-3-yl]oxy-5-cyclopropylpyridine-2-carboxylic acid 4-[(4-ethenylcyclohexyl)methyl]benzenecarboximidamide 6-chloro-N-[5-(3-cyclobutyloxyphenyl)pyridin-2-yl]pyridazine-4-carboxamide N-[3-[4-(methylideneamino)-2-propylphenyl]prop-1-en-2-yl]-6-morpholin-4-ylpyridine-3-carboxamide [4-(5-chloro-6-methoxypyrimidin-4-yl)piperazin-1-yl]-[2-fluoro-3-(trifluoromethyl)phenyl]methanone N-(4-fluorophenyl)sulfanyl-2,6-dimethoxy-4-(1H-pyrazol-5-yl)aniline 2-(2,3-dihydro-1H-inden-2-yl)-5-(9-methylidenefluoren-4-yl)pentanoic acid 1-[4,6-bis(4-chlorophenyl)-3-methylthieno[2,3-b]pyridine-5-carbonyl]piperidine-4-carboxylic acid 3-methyl-1-[4-[4-(propan-2-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]phenoxy]butan-2-one 2-[N-(1,3-thiazol-5-yl)anilino]benzoic acid N-[(2E,4Z)-5,6-diamino-3-[(cyclopropylmethylcarbamoylamino)methyl]-7-methoxyocta-2,4,7-trien-2-yl]-1H-indole-5-carboxamide N-[(3S)-1,1-dioxothiolan-3-yl]-5-fluoro-3,4-dihydroisoquinoline-2-sulfonamide N-[(2,4-dimethoxyphenyl)methyl]-N-(3-pyrrolidin-1-ylpropyl)acetamide (6R)-7-(3,4-dichlorobenzoyl)-2-[4-(trifluoromethoxy)anilino]-N-[3-(trifluoromethyl)phenyl]-3-(3,3,3-trifluoropropanoylamino)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-1-carboxamide 4-[2-fluoro-5-(3-phenylphenyl)phenyl]pyridine N-[(1S)-4,6-dichloro-2,3-dihydro-1H-inden-1-yl]carbamate 5-(3,3-difluoropyrrolidine-1-carbonyl)-N'-hydroxypyridine-2-carboximidamide 2-(2,6-difluorophenyl)-1H-pyrazole;N-(3,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl)formamide 2-[4-azido-3-[4-(1,2,5-triazepane-1-carbonyl)phenyl]pyrazol-1-yl]-N,N-dimethylacetamide N-(2,4-dichloropyrimidin-5-yl)-N-[3-(trifluoromethoxy)phenyl]benzenesulfonamide 4-[2,3-bis(ethenyl)phenoxy]-6,7-dimethoxy-1-propan-2-ylquinolin-2-one [(1S,2R)-2-hydroxy-1-(4-methoxyphenyl)propyl]iminocarbamic acid 4-[(7S)-8-cyclopropyl-9-methoxy-5,6,11-trioxo-1H-pyrazino[2,3-b][1,4]benzodiazepin-2-yl]-N'-diazenylpiperidine-1-carboximidamide N-(2-aminoethyl)formamide;2-[4-tert-butyl-1-[[4-[4-(2,3-dimethylphenyl)piperazin-1-yl]phenyl]methyl]pyrrolidin-3-yl]acetaldehyde 1-N',2-N'-dimethylethene-1,1,2,3-tetracarbohydrazide;4-(3-methylbutan-2-yl)-5H-[1,3]thiazolo[4,5-b]azepine 6-[(3R)-3-aminopyrrolidine-1-carbonyl]-4H-1,4-benzoxazin-3-one 4-amino-3-(2,4,5-trihydroxyphenyl)-1H-1,2,4-triazole-5-thione 2-[[5-(3-methylbutanoyl)thiophene-2-carbonyl]amino]pentanedioic acid [5-(4-fluorophenyl)-2-methyl-1,3-oxazol-4-yl]methanimine (4-hydroxyphenyl)methyl-[2,3,5,6-tetrafluoro-4-(trifluoromethoxysulfanyloxy)phenyl]carbamic acid N-azido-2,3-dichloro-5-(trifluoromethoxy)aniline 2-(4-fluorophenyl)-6-propan-2-ylpyridine 4-[4-(3,5-diphenyl-2,4-dihydrotriazin-1-yl)phenyl]dibenzofuran 1-(5-azido-2-methoxyphenyl)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline 2-[(3-methoxyphenyl)methyl]-4-propanoyl-1,3,4,5-tetrahydropyrrolo[1,2-a]quinoxaline-8-carbonitrile N-[(Z)-1H-benzimidazol-2-ylmethylideneamino]-6-chloro-3,5-dihydro-2H-1,4-benzothiazepine-7-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]butan-2-one;cyclobutane 2-[6-(4,5-dimethylcyclohexa-1,3-dien-1-yl)oxyhexyl]isoindole-1,3-dione 6-[[5-(3,4-dichlorophenyl)furan-2-yl]methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 1-(4-butylphenyl)sulfonyl-4-methyl-3,6-dihydro-2H-pyridine N-[3-(2,4-dichlorophenyl)sulfanylpropyl]formamide 2-(4,4-dimethylcyclohexen-1-yl)-N-[4-(3,5-dimethylpyridin-2-yl)butan-2-yl]acetamide [4-(dimethylamino)phenyl]iodanium (2Z,4E)-5-[6-(benzylideneamino)pyrimidin-4-yl]hexa-2,4-dien-1-amine [(1S,3R)-3-hydroxycyclopentyl]-[2-(pyridin-4-ylmethoxymethyl)-6-azaspiro[3.4]octan-6-yl]methanone (1S)-N'-methyl-1,2,3,4-tetrahydronaphthalene-1-carboximidamide;dihydrochloride (2S,3R)-3-[4-(4-fluorophenyl)benzoyl]oxy-1,5-dihydroxy-5-methylpiperidine-2-carboxylic acid (5R)-2-azido-1,3,9,11,13-pentazatetracyclo[8.7.0.03,8.012,16]heptadeca-2,4,6,10,12,14,17-heptaene 2,5-dichloro-4-[[(1S)-4-cyclopropyl-6-[3-(trifluoromethyl)phenyl]cyclohexa-2,4-dien-1-yl]methoxy]benzonitrile 3-[4-[5-(6,8-difluoro-2H-quinolin-1-yl)pyridin-2-yl]oxyphenyl]azetidine-1-carboxylic acid [(Z)-3-[1-methoxyethyl(methyl)amino]-1-phosphonopent-2-enyl]phosphonic acid;naphthalene-1,6-disulfonic acid 3,5-dibromo-4-[(6R)-3-(4-methoxyphenyl)-5-oxo-4H-1,2,4-triazin-6-yl]benzenesulfonamide N-[2-chloro-4-fluoro-5-[3-(trifluoromethyl)pyrazole-1-carbonyl]phenyl]-4,6-difluorobenzenesulfonamide (1R)-3-[[4,5-bis(ethoxycarbonylaminomethyl)cyclohexanecarbonyl]amino]-2-[6-methyl-8-(trifluoromethyl)quinolin-7-yl]cyclopropane-1-carboxylic acid 3-(4-aminophenoxy)-5-methylphenol 7-[4-hydroxy-3,5-bis(trifluoromethyl)phenyl]heptanoic acid 6-amino-4-(4-fluorophenyl)-1H-pyridine-2-thione 1-[2,6-dibromo-4-(trifluoromethyl)phenyl]hexan-1-one 2-(3,5-dichlorophenyl)sulfanyl-N'-hydroxypyridine-4-carboximidamide 5-chloro-1,2,4-trimethoxybenzene;2-chloro-N-[(3-oxocyclopentyl)methyl]pyridine-4-carboxamide 4-fluoro-3-(4-methoxyphenyl)sulfanylpiperidine 2-[3-(azidomethyl)phenoxy]-N-ethylacetamide N'-(3,5-dichlorophenyl)-2-oxoethanimidamide;hydrochloride 2,4-dichloropyrido[3,4-d]pyrimidine 5-chloro-2-(4,7-dihydroxy-3-oxoxanthen-9-yl)benzoic acid N-[3,5-bis(trifluoromethyl)phenyl]-N'-[4-(2,6-dimethoxyphenyl)pyridin-3-yl]-1H-imidazo[4,5-b]pyridine-7-carboximidamide (2S,3R)-1-azido-5-[4-(difluoromethoxy)phenyl]-3-(trifluoromethyl)piperidine 2-(4,6-dichloropyrimidin-5-yl)sulfanyl-N'-hydroxypyridine-4-carboximidamide 1-[(3S,5R)-4-acetyl-3,5-dimethylpiperazin-1-yl]-2-azidoethanone 2-[(3Z,5E)-5-acetyloxyhepta-1,3,5-trien-2-yl]oxy-4,6-dimethylpyridine-3-carboxylic acid N'-[2,3-bis(ethenyl)phenyl]-2-methoxybenzenecarboximidamide;ethane 1-methyl-N-[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)ethyl]indole-4-carboxamide 1-[(2R,4S)-5-[4-(3-methoxypropylamino)benzoyl]-2-phenylpiperidin-4-yl]ethanone 2-(3,5-dichlorophenyl)-N-ethyl-3-[(Z)-1H-indol-3-ylmethylideneamino]-4,6-dioxocyclohexene-1-carboxamide N-[2-(4-chlorophenyl)ethyl]-1,3,5-triazin-2-amine 4-bromo-3-methylsulfonylpyridine 1-methoxy-3-(2-methylphenyl)-4-propan-2-ylidenepiperidine 5-methyl-3-(2-methylpyrazol-3-yl)imidazo[1,2-a]pyridine 2-[3-(diethylamino)phenyl]-1H-benzimidazole-4,5-dicarboxylic acid 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-hydroxy-6-methylpyrimidine-4-carboximidamide N-[(5-ethylsulfanylpyridin-2-yl)methyl]spiro[1,4-dihydroquinoxaline-3,4'-thiane]-2-imine N-(5-cyclopropyl-1,2-oxazol-3-yl)-4-[(2S,4R)-2-methyl-4-[[2-[(2-methylpyrazole-3-carbonyl)amino]pyrimidin-4-yl]methyl]piperidin-1-yl]benzamide N-[5-cyano-4,6-dimethyl-3-(trifluoromethyl)pyridin-2-yl]acetamide;ethane 2-[3,4-difluoro-5-(trifluoromethyl)phenyl]sulfanylpropanenitrile N-[3-[2-azido-5-(trifluoromethyl)phenyl]propyl]benzamide N-[(2S)-3-cyclohexyl-1-oxo-1-piperidin-4-ylidenepropan-2-yl]furan-3-carboxamide 2-(3,4-dimethoxyphenyl)-N-[2-[[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]amino]pyrimidin-5-yl]acetamide N-[(Z)-(5-bromo-2-hydroxyphenyl)methylideneamino]-4-morpholin-4-ylbenzamide N-[5-tert-butyl-2-methoxy-3-(trifluoromethyl)phenyl]sulfanyl-1-(cyclopropylmethyl)pyrazol-4-amine 4-[2,6-di(propan-2-yl)phenyl]-3H-1,3-thiazol-2-one 3-(2,4-dihydroxyphenyl)-N-[(Z)-1H-indol-6-ylmethylideneamino]-1H-pyrazole-5-carboxamide 4-tert-butyl-1H-naphtho[2,3-h]quinoline 2-[1,3-bis(4-methoxyphenyl)pyrazol-4-yl]-N-(cyclobutylcarbamoyl)cyclopropane-1-carboxamide 3-[(1R)-2,2,2-trifluoro-1-(8-nonylnaphthalen-2-yl)ethoxy]cyclobutan-1-ol 4-[2-(5,7-dihydropyrrolo[3,4-b]pyridin-6-yl)ethyl]morpholine;ethane N-[3-(dimethylamino)propyl]-4-[2-[(4,6-dimethylpyrimidin-2-yl)amino]-4,5-bis(ethenoxy)phenyl]benzamide 2-[3,5-bis(trifluoromethyl)phenyl]-N-(4,6-dichloropyrimidin-5-yl)acetamide 4-chloro-3-[[1,3-dioxo-2-(trifluoromethyl)isoindol-5-yl]amino]-2-ethanimidoylbenzoic acid (1R)-4-amino-N',N'-dimethylcyclohexane-1-carbohydrazide;1-[(2S)-2-(3,4-dichlorophenyl)propanoyl]pyrrolidine-2-carboxylic acid N-[5-chloro-1-(3,4-difluorophenyl)sulfonylpiperidin-3-yl]-2-methoxyethanesulfonamide N-[5-[(Z)-3-amino-1,2-diaminoprop-1-enyl]pyridin-2-yl]-2-cyanobutanamide [6-(2,3-dichlorophenyl)sulfanyl-5-(methylaminomethyl)pyrimidin-4-yl]methylphosphonic acid 1-[4-bromobutan-2-yl(pyridin-3-yl)amino]propan-2-one 2-(4-hydroxyphenyl)-N-methylimidazo[1,2-a]pyridine-3-carboxamide 6-chloro-7-methoxy-1,4,4,9b-tetrahydroindeno[2,3-c]pyridine-5-carboxylate (2R)-1-[4-azidooxy-3,5-bis(trifluoromethyl)phenyl]sulfonylpyrrolidine-2-carboxylic acid 5-bromo-4-N-[(2R)-1,2,3,5,6,7-hexahydropyrrolizin-8-ylideneamino]pyrimidine-4,6-diamine (2-iodophenyl)-methyl-[[(2R,3S)-3-methyloxolan-2-yl]methyl]azanium 2-(2-cyclohexylethyl)-6-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazole-2-carboximidoyl)phenol 1-[3,5-bis(trifluoromethyl)phenyl]-4-[[dimethoxyphosphanyl(2,3,4,5,6-pentafluorophenyl)methylidene]amino]butane-1,4-dione;cyclohexa-1,3-diene [(1R)-3,4-dihydro-1H-isochromene-1-carbonyl]carbamic acid 4-[(E)-2-[3,5-difluoro-6-[(E)-pent-3-enyl]naphthalen-2-yl]ethenyl]benzonitrile 4-[[1,2-dimethyl-6-oxo-4-(pyridin-3-ylamino)pyrimidin-5-yl]methyl]-N-ethynylbenzamide 4-[(8-chloro-7-hydroxyquinazolin-4-yl)amino]cyclohexane-1-carboxamide 4-[2-bromo-N-(1,3-thiazol-5-yl)anilino]-N-quinoxalin-2-ylbenzenesulfonamide N-[3,6-bis(ethenyl)pyridin-2-yl]propanamide 1-[2,4-dichloro-3-(isoquinoline-6-carbonyl)phenyl]propan-2-one;ethane 2-[(3S)-2-oxo-1,3,4,5-tetrahydropyrido[2,3-e][1,4]diazepin-3-yl]acetic acid;hydrochloride 4-methyl-3-(quinolin-6-ylamino)phenol 1-(2,4,5,6-tetrabromocyclohexa-1,3-dien-1-yl)sulfonylnaphthalene 1-(2-hydroxyphenyl)-3,5-dimethyl-2H-pyrido[2,3-e][1,4]diazepine-7-carboxamide N-[(2R)-1-oxo-3-phenyl-1-(pyridin-2-ylamino)propan-2-yl]naphthalene-2-carboxamide 7-phenyldec-1-en-2-ol (3aR,6aS)-5-[(1R,2S)-2-(1H-indazol-6-ylamino)cyclopentanecarbonyl]-3,4,6,6a-tetrahydro-1H-furo[3,4-c]pyrrole-3a-carboxylic acid;formic acid (Z)-3-[5,7-difluoro-2-methyl-4-(morpholine-4-carbonyl)indol-1-yl]prop-2-enal 2-amino-7-[(3S,4R)-3,4-dihydroxypyrrolidin-1-yl]-5-methylpyrido[2,3-d]pyrimidine-6-carboxylic acid 2-[1,1-difluoro-3-(5-methoxycarbonylthiophen-3-yl)oxypropan-2-ylidene]-1,4-thiazine-6-carboxylic acid (2R,3S)-4-[5-(3-chlorophenyl)-1H-imidazol-2-yl]-2-methoxy-N-[(E)-pent-2-en-2-yl]pyrrolidine-3-carboxamide 2-[(2E)-2-[[5-(4-bromophenyl)thiophen-2-yl]methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 2-[3-ethylsulfonyl-5-(trifluoromethoxy)pyridin-2-yl]-7-[3-(isocyanomethoxy)phenyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one 4-[(2R)-3,4-dimethylpentan-2-yl]oxy-3-propan-2-ylpyridazine (Z)-3-chloro-N'-ethyl-2-(methylideneamino)but-2-enediamide;4-[7-(6-chloropyridazin-3-yl)-8-oxo-5-thia-1,7-naphthyridin-3-yl]benzaldehyde N-(2,5-diethylpyrazol-3-yl)-1H-indole-7-carboxamide 4-[3,5-bis(trifluoromethyl)phenyl]-2-[[4-hydroxy-1-[(1R)-3-pyridin-3-ylcyclohexanecarbonyl]piperidin-4-yl]methyl]-N,N-dimethylpentanamide 5-methylsulfanyl-6,7-dihydrocyclopenta[f]indazole 1-amino-3,5,6,9-tetramethylpyrazolo[4,3-h]quinazoline-2,8-dione 6-[1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]pyridazine-3,5-diamine 2-[2-methylpropanoyl(1,3-thiazol-5-yl)amino]guanidine N-azidooxy-1-benzyl-4,5-dimethoxycyclohexa-2,4-dien-1-amine 2-(3,4-dimethylphenyl)-7H-imidazo[5,1-c][1,2,4]triazole-3,6-dione [3-amino-5,6-bis(methylamino)pyridin-2-yl]methanol [4-(difluoromethoxy)phenyl]sulfonylmethanamine 2-[1-[4-(6-hydroxy-5-methylheptanoyl)benzoyl]piperidin-4-yl]propanamide 4-(1H-indol-5-ylmethylidene)-3-(2-morpholin-4-ylethylamino)cyclohexa-2,5-dien-1-one 6-(3,4-difluorophenyl)-2-[5-ethylsulfonyl-1-methoxy-2-(3,3,3-trifluoropropylamino)pyridin-1-ium-4-yl]-7H-pyrrolo[3,4-b]pyridin-5-one 3-(2,2-difluoroethylamino)benzaldehyde;N-[1-[5-(4-methylimidazol-1-yl)pyridin-2-yl]ethenyl]methanimine N-(1H-benzimidazol-2-ylmethylideneamino)naphthalene-1-carboxamide N-[(4S)-6,8-diethyl-1,2,3,4-tetrahydronaphthalen-2-yl]benzamide 3-(4,5-dihydro-1H-imidazol-2-yl)-N-ethoxyaniline [3-(4,5-dimethylfuran-2-carbonyl)azetidin-1-yl]-[4-(oxolan-3-yloxy)pyridin-2-yl]methanone 2-[2,5-bis(trifluoromethyl)phenyl]iminoacetonitrile;3-ethylhexane 2-tert-butyl-4-methyl-6-(oxan-2-yloxy)pyrimidine (2R)-N-[[4-[4-amino-6-(ethylaminomethyl)pyrimidine-5-carboximidoyl]phenyl]methyl]-1-(6,7-dihydrothieno[3,2-d]pyrimidin-4-yl)pyrrolidine-2-carboxamide 1-(3,4-difluorophenyl)-2-ethylhexane-1,3,5-trione 4-[3-(5,6-dichlorobenzimidazol-1-yl)piperidin-1-yl]thieno[3,2-d]pyrimidine N-(3,5-dichloropyridin-4-yl)-2-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]oxyacetamide N-[4-(2,6-dimethylmorpholin-4-yl)phenyl]-5-fluoroquinazolin-3-ium-7-amine 5-methyl-1,4-bis[(2-nitrophenyl)methoxy]cyclohexa-3,5-diene-1,3-dicarboxylic acid N-cyclohexyl-5-fluoro-4-(3-methoxyphenyl)pyrimidin-2-amine N-(1,3-benzothiazol-2-yl)-4-[1-methylidene-5-oxopyrrolidin-1-ium-2-carbonyl]piperazine-1-carboxamide 2-[[(2S)-1-methylpyrrolidin-2-yl]methoxy]-4-phenyl-7,8-dihydropyrido[4,3-d]pyrimidine 2-methyl-2-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]propanal 2,3-dichloro-N-diazonaphthalene-1-sulfonamide 6-N-(3-methylbutyl)-7H-purine-2,6-diamine 4-[(5R)-3-azido-6,6-difluoro-2,4-dihydropyrrolo[2,1-c][1,4]oxazin-9-yl]aniline 4-(3,5-dimethoxyphenyl)imino-2,3-dihydrochromene-8-carboxamide 4-(3-methylpyridin-2-yl)benzenesulfonamide (2S)-5-chloro-N-[4-fluoro-3-(methanesulfonamido)phenyl]spiro[2H-indole-3,1'-cyclohexane]-1-carboxamide 4-[2-aminoethyl(methylamino)amino]-N'-ethylbenzenecarboximidamide 5-(1-cyclopentylpiperidin-4-yl)oxypyridine-2,3-diamine 1-[2-fluoro-4-(methanesulfonamido)phenyl]cyclopropane-1-carboxamide 2-[3-(3,5-difluorophenyl)phenyl]acetamide 4-[5-(2-chlorophenyl)-3,6-dimethylpyridine-2-carbonyl]benzoic acid 5-(1,2-dimethoxypropan-2-yl)naphthalene-2-carboxylic acid 2-(1-cyclopentyl-5,6-dihydrobenzimidazol-2-yl)-5-(4-pyridin-3-ylpiperazine-1-carbonyl)phenol [5-(2,4-difluorophenyl)-1,3,4-oxadiazol-2-yl]methanamine;hydrochloride 2-(4,6-diphenylpyrimidin-2-yl)-3-[4-(9H-fluoren-1-ylsulfanyl)phenyl]sulfonylbenzenethiol 2,6-ditert-butyl-4-[(E)-[[5-(3,5-dichloro-4-fluorophenyl)furan-2-carbonyl]hydrazinylidene]methyl]phenolate;nickel(2+) N-[(3S,7R,8aS)-3-(2-hydroxyethyl)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-5-methoxy-2-propan-2-ylbenzamide 5-[4,5-bis(ethenyl)-2,3,6-trifluorophenoxy]pyrimidine;2-ethenoxypropane 1-[3-(dimethylamino)propyl]-N,N'-diethylpyridine-4-carboximidamide;ethane 5-(3,4-dichlorophenyl)-7H-pyrrolo[2,1-f][1,2,4]triazin-4-amine N-[[2-(furan-3-yl)phenyl]methoxy]acetamide 2-(3,4-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine 2-(8,8-dimethyl-7H-benzo[c]fluoren-10-ylidene)propanedinitrile 2-[N-(1-carboxypropan-2-yl)-3,5-dichloroanilino]octanoic acid [(3S)-1-(5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carbonyl)pyrrolidin-3-yl]azanide 4-[2-(3,5-diphenylphenyl)ethoxy]piperidine 4-(2,3-dihydro-1H-inden-5-yl)-N'-hydroxypyridine-2-carboximidamide N-[(1R)-2,3-dihydro-1H-inden-1-yl]pyrimidine-5-carboxamide 1-[4-[5-(2-iodopropan-2-yl)pyridin-3-yl]oxyphenyl]pyrrolidin-2-one 3-bromo-4,5-dimethoxybenzenecarboperoxoic acid 5-[5-methyl-2-(1,3-oxazol-4-yl)thiophen-3-yl]pyridine-3-carboxamide (7S)-2-[[1-[(4-chlorophenyl)methyl]pyrazol-3-yl]amino]spiro[5H-pyrido[2,3-d]pyrimidine-6,3'-pyrrolidine]-7-carboxylic acid 1-[(4-aminophenyl)methyl]-3-[2-[4-(4-ethoxy-5,6,8,10-tetrahydrothieno[3,2-d]azocine-7-carbonyl)phenoxy]ethyl]urea 4-methyl-2-[3-(7H-purin-6-ylsulfanyl)cyclopenten-1-yl]pyrimidine 4-amino-1-[[5-(methanesulfinamido)naphthalen-2-yl]sulfonyl-[(3S)-piperidin-3-yl]amino]-6,7-dihydropyrrolo[2,3-d]pyrimidine-5-carboxamide 4-(cyclohexylmethyl)-N'-diazenyl-5-nitrobenzenecarboximidamide N-[1-[3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]ethyl]prop-2-enamide 4-(3,5-ditert-butyl-2-hydroxyphenyl)-3,8a-dihydroanthracene-9,10-dione (Z)-3-hydroxy-N'-[2-(trifluoromethyl)phenyl]prop-2-enimidamide (E)-N-ethyl-2-[(4-formylphenyl)methylideneamino]but-2-enamide N-[[4,5-bis(ethenyl)-1H-imidazol-2-yl]methyl]-2-cyclohexyl-6-(4-propan-2-ylidenepiperidin-1-yl)pyrimidin-4-amine (4S)-2,5-diamino-5-[4-(3-methoxyphenyl)-1,3-thiazol-2-yl]-4-methylpentanoic acid N-cyclopropyl-1'-(2,6-dioxopiperidin-3-yl)spiro[2H-indole-3,4'-piperidine]-5-carboxamide 3-(4,5-dihydroimidazol-1-yl)-N-ethyl-2-(6-methoxynaphthalen-2-yl)propanamide 1,4-bis(4-aminophenyl)-3-[[2-(3-methylbutoxy)pyridin-4-yl]methyl]imidazolidin-2-one 5-[(1R)-2,3-dihydro-1H-indene-1-carbonyl]-N-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide 3,5-dichloro-4-fluoroaniline;1-methylnaphthalene 3-chloro-5-[1,6-dimethyl-4-[(4-nitrophenyl)methoxy]cyclohexa-2,4-dien-1-yl]pyridine 1,1-bis(2,3-dihydrothiophen-4-yl)-N'-ethylmethanediamine 4-[2,3-diamino-5-(4-chlorophenyl)phenyl]benzene-1,2-disulfonic acid (3R,5S)-2,4-ditert-butyl-6-methoxycarbonyl-3,5-bis[phenyl-[2-(trifluoromethyl)pyridin-4-yl]methylidene]cyclohexa-1,4-diene-1-carboxylate 6-(1H-indole-3-carbonyl)naphthalen-2-ol 6-(6-chlorospiro[3,4-dihydrochromene-2,4'-piperidine]-1'-yl)-5H-cyclopenta[d]pyrimidin-4-amine (1-ethylpyrrolidin-2-yl)-[3-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)piperidin-1-yl]methanone 2-methyl-1-[4-(trifluoromethoxy)phenyl]butan-1-one 2,4-diaminopyrimidine-5-carbonitrile;3-ethyl-8-(2-fluoro-6-methoxyphenyl)-2-[1-(1H-indazol-6-yl)ethyl]isoquinolin-1-one 4-(5-azidoindol-1-yl)cyclohexan-1-ol 2-[(1S,5R)-3,9-diazabicyclo[3.3.1]nonane-9-carbonyl]-4,6-dimethyl-1H-pyridin-8-one;dihydrochloride ethane;2-methylbutanal;6-[5-(propanoylamino)pentan-2-ylideneamino]pyridine-3-carboxamide 6,7-dimethyl-10-[2-(oxiran-2-ylmethoxy)phenyl]spiro[4H-acridine-9,1'-cyclopropane] [2-[2-(2,3-dihydrofuran-5-yl)ethynyl]-6,7-dimethoxyquinolin-4-yl]urea 1-[4-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalene-2-carbonyl]piperazin-1-yl]-2-[ethoxy(methyl)amino]-2-methylpropan-1-one 2-(4-bromophenyl)ethylazanium (3,4-dimethoxyphenyl)-(8-imidazol-1-yl-9H-pyrido[2,3-b]indol-6-yl)methanone 5-(3,4-dimethoxyphenyl)-2-(2-ethyltriazol-4-yl)-N'-hydroxypyrimidine-4-carboximidamide (4S)-2,5-dimethoxy-N-[[3-[2-oxopropyl(1,2,4-triazol-4-yl)amino]phenyl]methylideneamino]-4-phenylpentanamide 6-tert-butyl-3H-benzo[f]chromene 3-[[(2R,3S)-1-ethyl-5-oxo-2-pyridin-4-ylpyrrolidine-3-carbonyl]amino]-3-(6-methoxy-5-methylcyclohexa-2,4-dien-1-yl)propanoic acid 4-azido-2,3-bis(ethenyl)quinoxaline 5-[2,4-difluoro-3-[(2E)-5-methylocta-2,6-dienoyl]anilino]-1H-pyrazole-4-carboxylic acid 4-chloro-3-(4,5-dimethylthiophene-2-carbonyl)-1H-indole-7-carbonitrile 2-methoxy-4-[3-(6-pyridin-2-ylthieno[2,3-d]pyrimidin-4-yl)propyl]benzoic acid N-[3,5-bis(trifluoromethyl)phenyl]-3-cyano-4-(2,6-dichloropyridin-3-yl)oxybenzamide;3,4-dihydro-2H-chromene;ethanamine (2E,3Z)-1-fluoro-4-methylidene-2-propylimino-3-[[5-[4-[2-(trifluoromethyl)phenyl]phenyl]furan-2-yl]methylidene]pyrrolidine 4-chloro-3-(2,5-dimethylpyrazol-3-yl)benzamide 3-(5-azido-2-chlorophenyl)pyridine 3-(2,5-dimethylpyrrol-1-yl)sulfonyl-N'-hydroxybenzenecarboximidamide 3,6-diaminopyridine-2-sulfonate 2-amino-6-[4-chloro-3-(trifluoromethoxy)phenyl]-4,4-dimethoxy-3-azabicyclo[3.1.0]hex-2-ene-1,5-disulfonate 4-[2,3-bis(sulfanyl)phenyl]-N,1-dimethylpyrazole-3-carboxamide N-[3-(1H-imidazol-2-yl)propyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-4-carboxamide;dihydrochloride 2-methyl-5-(3-methylphenyl)quinazoline 4-(3,5-dimethylphenyl)-2-[(E)-2-[6-methyl-1-[(3Z)-3-propylidene-1H-pyrrol-2-ylidene]azepine-2-carbonyl]but-2-enyl]-3,4-dihydroisoquinolin-1-one 2-[2-(1H-imidazol-5-yl)propanoylamino]propanedioic acid 2-(6,7-dihydropyrazolo[1,5-a]pyrimidine-3-carbonylamino)-4-methoxybenzoic acid (3R)-2-amino-1-[(6S,11R)-9-methoxy-11-(2H-triazol-4-yl)-6,8-dihydro-5H-pyrido[2,3-b][1]benzazepin-7-yl]-3-phenylsulfanylbutan-1-one N-[(Z)-(3-bromo-2-hydroxyphenyl)methylideneamino]-4,5-dinitrofuran-2-carboxamide (3R,4S)-1-[5-cyclopropyl-2-(cyclopentylmethoxy)phenyl]pyrrolidine;2,2,2-trifluoroacetic acid 5-bromo-4-cyclopropyl-2-(1,3-thiazol-4-yl)-1H-pyrimidin-6-one 2-[3-(4-fluorophenyl)pentanoyl]cyclohexane-1,3-dione N-(3-fluorophenyl)-2-[4-(trifluoromethyl)phenoxy]acetamide 7-[3-[(4,5-dichloro-2-ethylphenoxy)methyl]phenyl]-9H-fluorene [2-[(Z)-but-1-enyl]-5-methoxyphenyl]-dimethylsulfanium N-[2,4-difluoro-3-(6H-pyrrolo[3,4-c]pyrazol-1-yl)phenyl]methanesulfonamide 2-(4-chlorophenyl)-6,8-dimethoxyquinazoline 2-[4-[[(5R)-3,9-diazaspiro[5.5]undecan-9-yl]sulfonyl]pyrazol-1-yl]acetic acid 2-[4-[6-(methoxyamino)imidazo[1,2-b]pyridazin-3-yl]phenyl]propanamide N-[5-(azidomethyl)-1,3-thiazol-2-yl]-6-(trifluoromethoxy)pyridine-3-carboxamide 2-amino-N-(1,3-benzothiazol-5-ylmethyl)-4-methoxybenzamide 2-[4-(4-butylcyclohexyl)phenyl]-6,7-difluoronaphthalene 5-[6-[2-(2,4-dichlorophenyl)ethylamino]pyridin-3-yl]-1H-imidazole-4-carboxylic acid 1-(2,4-dimethylpentyl)-N-[3-ethoxy-4-(1H-pyrazol-4-yl)phenyl]benzimidazole-5-carboxamide 2-[4-bromobutan-2-yl(1,3-thiazol-5-yl)amino]phenol 2-chloro-N-[5-cyano-4-(3-methoxypropylsulfanyl)-1,3-thiazol-2-yl]-5-nitrobenzenesulfonamide 1-[(E)-(2,4-dihydroxyphenyl)methylideneamino]-3-[2-(4-methoxyphenyl)ethyl]thiourea 2-azidooxy-3,4,5-trimethylfuran (3Z,5E)-3,5-dimethylhepta-1,3,5-triene;N-ethyl-4-methoxybenzamide;2-formamido-2-methylpropanoic acid 4-benzyl-N-[5-cyano-4-(2,6-dimethoxyphenyl)-1H-imidazol-2-yl]piperidine-4-carboxamide 1-(1,3-benzodioxol-4-yl)-3-(5-methoxy-2-nitroanilino)propan-2-one 6-(4-bromo-2-fluorophenyl)-5,7-dihydropyrrolo[3,4-b]pyridine 1-[6-(3,5-dichlorophenyl)-4-[3-fluoro-4-(3-methoxypyridin-2-yl)sulfanylanilino]quinolin-3-yl]ethanone (1S,2R)-N-[6-amino-5-(5,6-dihydroxypyridin-3-yl)pyridin-3-yl]-2-cyclopentylcyclopropane-1-carboxamide [(2S,4R)-4-azidooxy-1-butylpiperidin-2-yl]methanol N-[2,4-bis(trifluoromethyl)phenyl]-5-fluoro-1,3-dihydroindol-2-imine N-[[3,5-bis(trifluoromethyl)phenyl]methyl]acetamide 6-methyl-2-[(4-nitrophenyl)carbamoyl]cyclohexane-1,3-dicarboxylic acid (2S)-N-[3-(2,4-dichlorophenyl)propyl]-1-(2-hydroxy-2-methylpropanoyl)pyrrolidine-2-carboxamide (5R)-1-(2,6-difluorophenyl)-3-[4-[4-(morpholine-4-carbonyl)anilino]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]-2-oxoimidazolidine-4,5-dicarbonitrile 2-[2,6-dimethoxy-4-(piperidine-1-carbonyl)phenyl]-4,5-dihydroimidazol-1-amine 1-[4-(2,5-dichloropyrimidin-4-yl)morpholin-2-yl]ethanol 3-[(3R)-3-(dibenzylamino)cyclohexyl]-2H-imidazole-4-carboxamide 4-[2-(ethylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzaldehyde 1-[4-amino-3-(trifluoromethyl)phenyl]-2-hydroxyethanesulfonic acid N-(cyclohexylmethyl)-6-(2,5-difluorophenyl)-1,4-oxazepane-4-carboxamide;ethane N-[(2R,3S)-2-methyloxolan-3-yl]-1H-pyrrole-3-carboxamide 2-[4-(3,5-difluorophenyl)-1H-pyrrole-2-carbonyl]-5-methoxy-6a,7-dihydropyrrolo[1,2-c]quinazolin-4-one 4-[(1,5-dimethylpyrazole-3-carbonyl)amino]-2-phenoxybutanoic acid 4-[(3S)-1-(4,5-dimethylpyrimidine-2-carbonyl)piperidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-6-one [3-(dimethylamino)-2-[3-[1-ethyl-4-[1-[5-fluoro-6-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)pyridin-3-yl]ethenyl]piperidin-4-yl]propyl]phenyl]methanol N-[6-(dimethylamino)pyridin-3-yl]-2-hydroxy-3-oxobutanamide (2S,4R)-4-methoxy-5-phenylmethoxy-1-pyrimidin-2-ylpentan-3-one 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzimidazolo[1,2-a]quinoline 2-[[5-(1H-indole-3-carbonyl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl]amino]acetic acid N-[3-(5,7-difluoroquinolin-6-yl)-4-methylphenyl]pyrrolidine-1-carboxamide N-cyclopentyl-3-[2-(cyclohexylamino)quinazolin-6-yl]benzenesulfinamide 6-(3,4-dichlorophenyl)-N-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]quinazolin-2-amine 1-[2,6-di(propan-2-yl)phenyl]-3-(N'-hydroxycarbamimidoyl)urea 4-[[(1R,2S)-6-chloro-8-hydroxy-2,3,4,9-tetrahydro-1H-carbazol-2-yl]oxy]oxan-2-ol N-[4-fluoro-3-(1H-indazol-5-yl)phenyl]-2,5-dimethoxybenzenesulfonamide N-(3,4-dihydro-2H-1,5-benzothiazepin-7-ylmethyl)-6-methoxypyrimidine-4-carboxamide 3-[(3R)-2-benzylsulfonyl-1,3-dihydropyrazol-5-yl]pyridine [(E)-5,6-dimethylhept-4-enoxy]methylbenzene 4-[3-(cyclopropylmethoxy)-5,6,7,8-tetrahydronaphthalen-2-yl]-5,5,5-trifluoropentanenitrile 6-[4-(4-ethenylcyclohexyl)phenyl]-1,2,3-trifluoronaphthalene 3-[4-(azetidin-1-yl)cyclohexyl]-5-methoxy-N-(oxan-4-ylmethyl)-1H-indole-2-carboxamide 1-(2-nitroethenyl)-4-pentan-3-ylbenzene (5-bromo-3-chlorothiophene-2-carbonyl)-cyclopropylazanium (3S)-4,7-dibromo-1,2,3,3a,8b-tetrahydrocyclopenta[b]indol-6-one 2-[(5S,10bS)-5-thiophen-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 7-bromo-5-nitropyrrolo[2,1-f][1,2,4]triazin-4-amine N-[3,5-dimethyl-4-(piperidine-1-carbonyl)thiophen-2-yl]methanesulfonamide 4-[(2,6-dichlorophenyl)methyl]cyclohexane-1-carbonitrile 4-(4-methylphenyl)sulfonyloxypiperidine-2-carboxylic acid 2-[4-[3-(2-fluorophenyl)propyl]piperazin-1-yl]-N,N-dimethylpyrimidin-5-amine 4-[3-[1,7-dihydroxy-6-(2-piperidin-1-ylethoxy)naphthalen-2-yl]-4,5-bis(prop-2-enoxy)phenyl]benzoic acid 2-(6,6-difluoroheptyl)-4-nitrophenol 2-[[5-[1-(4-fluorophenyl)cyclohexyl]tetrazol-1-yl]methyl]quinoline N-[2-(5-bromopyrimidin-4-yl)oxyethyl]acetamide 1-ethyl-2,4,5-tris(2-methoxyethoxy)benzene 3-[(2-amino-5-methoxyphenyl)diazenyl]-N,4-dimethylaniline 2-[3-(4,6-dichloropyridin-3-yl)oxyphenoxy]-N-(4-ethoxyphenyl)propanamide 4-[7-[(E)-1-amino-3-iminoprop-1-enyl]thieno[3,2-b]pyridin-5-yl]-N-(4-ethoxybutyl)benzamide [4-hydroxy-4-(phenylsulfanylmethyl)piperidin-1-yl]-[3-methoxy-5-(2,2,2-trifluoroethoxy)pyridin-4-yl]methanone 2-(4-chlorophenyl)-7,7a-dihydro-1H-indazole (E)-3-[6-[2-methylsulfanyl-4-(trifluoromethoxy)phenyl]pyrimidin-4-yl]-N'-propanoylbut-2-enehydrazide 2-methyl-4-(5-pyrimidin-5-ylpyrimidin-2-yl)morpholine (2R)-3-chloro-N-cyclopropyl-2-[3-fluoro-4-(trifluoromethoxy)phenyl]-1,5-dihydropyrazole-5-carboxamide (2S)-1-[(2S,4S,5R)-3-hydroxy-9-oxa-7-azatricyclo[6.4.0.02,4]dodeca-1(12),8,10-trien-7-yl]propan-2-ol N'-[(4,6-dimethylpyrimidin-2-yl)iminomethyl]-1-[3-methoxy-5-(trifluoromethyl)phenyl]-N'-methylethane-1,2-diamine 2-[4-(6-methoxypyrimidin-4-yl)piperazin-1-yl]pyridine-3-carbonitrile 2,2-dimethyl-7-nitro-9H-fluorene 4-[1,3-bis(2,6-dimethylphenyl)imidazol-2-ylidene]-5H-pyrazol-3-one;ruthenium(2+);chloride 4-azido-2-ethyl-5-phenylmethoxypyrimidine 1-[4-(3,5-dimethylphenyl)piperazine-1-carbonyl]piperidine-2-carboxamide 2,4-dibromo-3-cyclopentyloxy-N-[(1S)-1-phenylethyl]benzamide 4-[(4-hydroxyphenyl)diazenyl]benzenesulfonic acid 4-[(E)-3-hydroxybut-1-enyl]-2-methoxyphenol;methane;1,4-xylene 3-(cyclopropanecarbonylamino)-4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-ylmethoxy)ethylamino]butanoic acid;hydrochloride 2-[1,3-dioxo-7-[[4-(trifluoromethoxy)phenyl]methylamino]isoindol-5-yl]-N-ethylidenepropanamide 6-(2-cyclopropylethoxy)-1H-quinazoline-2,4-dione 2-azido-5-chloro-N,N-dimethyl-6-[4-(trifluoromethyl)phenyl]pyrimidin-4-amine [2-[6-(4-cyclopropyl-1,3-thiazol-5-yl)pyrimidin-4-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-pyridin-3-ylmethanone N-[4-chloro-3-(1,2-oxazol-5-yl)phenyl]sulfanylmethanamine [3-(diethylamino)propoxy]sulfonyl-[4-[2-[[8,8-bis(trifluoromethyl)quinolin-4-yl]amino]ethyl]phenyl]azanide 5-hydroxy-2-methylbenzoic acid;N,1,4-trimethylpyridin-1-ium-2-sulfonamide ethane;3-methoxy-N-methyl-4-(3-methylsulfanylanilino)benzamide 5-fluoro-N'-methyl-2-[1-[4-(trifluoromethoxy)phenyl]ethylideneamino]benzenecarboximidamide [4-[(E)-2-methyl-3-[3-[1-[5-(6,7,8,9-tetrahydro-1H-pyrrolo[2,3-c]azepine-2-carbonyl)pyridin-2-yl]piperidin-4-yl]phenyl]prop-2-enoxy]cyclohexa-2,4-dien-1-ylidene]cyanamide 4-[5-(1-methylindazol-6-yl)imidazo[2,1-b][1,3]oxazol-8-yl]morpholine 4-[[3-(2,6-dimethylmorpholin-4-yl)quinoxaline-2-carbonyl]amino]butanoic acid N-butyl-4-[1,3-bis(2,6-dimethoxyphenyl)propan-2-yl]aniline (2S,4R)-4-[4-chlorobutyl(ethylsulfonyl)amino]-N-hydroxy-2-[(3-phenylphenyl)methoxycarbonyl]pyrrolidine-1-carboximidate 1-(2,6-dichlorophenyl)-2H-quinoline 3-hydroxy-5,7-dinitroanthracene-2-carboxylic acid 3-[(4-tert-butylphenyl)methylamino]-4H-1,2,4-triazin-5-one N-[5-[3-(2-methylpyrimidin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]pyridin-2-yl]acetamide N-[1-amino-4-methyl-3-(methylamino)pentylidene]-2-(3,5-dichlorophenyl)quinoline-8-carboxamide (5Z)-5-[[4-fluoro-2,6-dimethyl-3-(trifluoromethyl)phenyl]methylidene]imidazolidine-2,4-dione [(2R,3S)-2-(1-methylimidazol-2-yl)oxan-3-yl]-pyrrolidin-1-ylmethanone 5-[(2-methylphenyl)diazenyl]naphthalene-1,7-disulfonate [4-[[1,3-dimethyl-5-(4-phenylphenoxy)pyrazole-4-carbonyl]amino]cyclohexanecarbonyl]-methylidene-oxidoazanium N-[4-chloro-3-(trifluoromethyl)phenyl]-2,2-dimethylpropanamide 3-[5-(4-fluorophenyl)-1,2-dihydrotriazol-3-yl]-N-[5-methyl-6-[3-(propan-2-ylideneamino)phenoxy]pyridin-3-yl]benzamide 1-[4-[6-(4-chlorophenyl)-3,5-difluoropyridin-2-yl]piperazin-1-yl]propan-1-one (2Z,4E)-7-(3-ethoxypyrrolidine-1-carbonyl)-5-methyl-N-[2-oxo-2-(4H-1,2,5-oxadiazol-5-ylamino)ethyl]octa-2,4-dienamide N-(4,5-dimethylpyrimidin-2-yl)oxy-2,3-difluoropropanamide 2-azido-5-bromo-4,6-dimethylpyrimidine (2S)-N-ethylsulfonyl-3-[8-fluoro-6-methoxy-1-oxo-7-(3,4,5-trifluorophenyl)isoquinolin-2-yl]-2-(tritylamino)propanamide 3-[3-(5,6-diamino-2H-pyrimidine-1-carbonyl)phenyl]propanenitrile (2-ethyl-6-phenylpyridin-3-yl)methanol 2-(azidooxymethyl)-3,4,5-tribromopyridine [(2S,4R)-1-[3-(benzylideneamino)-6-(trifluoromethyl)pyridin-2-yl]-4-hydroxypyrrolidin-2-yl]-morpholin-4-ylmethanone 4-(4-chlorophenyl)-5,6-difluoro-3H-1,3-oxazin-2-one 1-(6-bromothieno[2,3-d]pyrimidin-4-yl)piperidin-4-ol;ethane [3-(4-chlorobenzoyl)phenyl]phosphonic acid 3-[(1-methyl-2,6-dioxopiperidin-3-yl)methylideneamino]-4-(oxan-4-ylsulfamoyl)benzenecarboximidamide (3S,4R)-3-azido-1-[(2-bromophenyl)methyl]piperidine 2-[(4-oxo-5,6,7,8-tetrahydrochromene-3-carbonyl)amino]-1H-benzimidazole-4-carboxamide 2-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]acetic acid 6-(4-chlorophenyl)-9-ethyl-8-(2,4,5-trimethoxyanilino)-2H-furo[3,2-f]chromene-7-thione 1-(2-iodopropan-2-yl)-5,6-dimethoxybenzimidazole 3-methoxy-4-nitro-1H-benzimidazole-2,5-dione 5-methoxy-2-(4-methoxyphenyl)-6-phenyl-2,3-dihydro-1H-quinoline 5-[2,3-bis(propanoylamino)phenyl]iminopenta-1,3-diene-2,4-diol 2-[4-[(E)-4,5-dihydroxypent-3-enyl]phenoxy]-1-pyrrolidin-1-ylethanone 1-amino-2,3-dichloroanthracene-9,10-dione 1-(7,8-dihydronaphthalene-2-carboximidoyl)-4-imino-5-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]imidazolidin-2-one 2-methoxy-4-[(E)-3-methylbutan-1-ylideneamino]sulfanylaniline 7-(2-bromoethyl)-6-methoxynaphthalene-2-sulfonic acid 2-hydroxy-N,3-dimethyl-4-oxo-3H-naphthalene-1-carboxamide 2-(4-chlorophenyl)-3-fluoroquinoline 5-[4-[bis(prop-2-enyl)amino]piperidine-1-carbonyl]-4,4-dimethyl-3H-thieno[2,3-c]chromen-10-one 1-[4-(diethoxyphosphorylmethyl)phenyl]-5-(2,6-difluoropyridine-3-carbonyl)pyrrolidin-2-one 1-[2,4-dichloro-3-(3-methylbutoxy)benzoyl]piperidine-4-carboxylic acid N-[(3S,7S,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-5-methoxypyrimidine-2-carboxamide 4-[1,4-bis(ethenyl)imidazol-2-yl]butanenitrile 2-benzyl-N-(8-bromoquinoxalin-5-yl)pentanamide 2-[3-[4-(dimethylamino)quinazolin-6-yl]oxypyrrolidine-1-carbonyl]-N,4-dimethylpyrrolidine-1-sulfonamide 3-azido-7-chloro-5-phenyl-1H-1,4-benzodiazepine 1,2-difluoro-6-propylnaphthalene N-(2,3,4,9b-tetrahydro-1H-chromeno[3,4-c]pyrrol-7a-yl)-3-fluoro-6-methoxypyridazine-4-carboxamide;2,2,2-trifluoroacetic acid N-[(6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl)methyl]-N'-propan-2-ylthiomorpholine-4-carbohydrazide 1-(cyclobutylmethoxy)-4-[3,3,5,5-tetradeuterio-4-fluoro-2-(trifluoromethyl)pentan-2-yl]benzene (2R)-6,7-dimethyl-4-[(E)-3-phenylprop-2-enoyl]oxyoctane-2-sulfonic acid 6-(2,3,5-trifluorophenyl)sulfanylcyclohexa-1,4-diene-1,5-diol 2-[(4Z)-5,6-dimethylhepta-1,3,5-trien-2-yl]oxyaniline (3R)-N-[2,6-difluoro-4-[5-(trideuteriomethyl)-1H-imidazol-2-yl]phenyl]piperidine-3-carboxamide N-[(2R)-1,1,3,3-tetramethyl-2H-inden-5-yl]propanamide 1-(5,6-dichloropyridin-3-yl)-N-[4-methoxy-6-(trifluoromethylsulfonyl)pyrimidin-2-yl]-3-[methyl(methylamino)amino]piperidine-3-carboxamide 2-benzyl-6-(1,4-diazepane-1-carbonyl)-5H-pyrazolo[3,4-d]pyrimidin-4-one 2-methylsulfanyl-5,6,7,8-tetrahydro-3H-quinazolin-4-one 3-(N-(2-bromophenyl)anilino)propanoic acid 2-(2-aminoethyl)-3,7-dimethylbenzo[f]isoindole-1,5-dione 2-[2-(4,5-dihydroimidazol-1-yl)phenyl]-3H-pyrido[2,3-d]pyrimidin-4-one 1-[4-chloro-5-(3,4,5-trimethoxyphenyl)thiophen-2-yl]ethanone 1-[6-(4-cyanophenyl)pyridin-2-yl]-3-ethoxyurea 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidin-4-one;ethane 5-(1H-indol-2-yl)benzene-1,3-diol ethane;3-[(4-ethoxyphenyl)methyl]-8H-pyrano[3,2-g]quinazolin-3-ium [(3S)-1-(4-aminobenzoyl)pyrrolidin-3-yl]urea N-[(E)-(3,4-dihydroxyphenyl)methylideneamino]-5-phenyl-1H-pyrazole-3-carboxamide 2-[3,5-dichloro-N-(2,2-diethoxyethyl)anilino]acetamide 5-(3,4-dihydronaphthalene-2-carbonylamino)-2,6-dimethylcyclohexa-1,5-diene-1-sulfonic acid 4-azidooxy-3-butylbenzoic acid 2-[(2S)-4,4-difluoro-1-iodocarbonylpyrrolidin-2-yl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 1-[(4-methoxyphenyl)methyl]-3,6-bis(sulfanylidene)piperazine-2,5-dione N-benzyl-N-[(Z)-1H-indol-3-ylmethylideneamino]-5,6,7,8-tetrahydroquinolin-8-amine 2-[2,6-diethoxy-4-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8,11-pentaen-4-yl)phenyl]acetaldehyde 3-methyl-1,9b-dihydrooxireno[2,3-b]indole-6-carboxylic acid 3-amino-5-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)cyclohexa-2,4-dien-1-one;ethane 3-(2,5-difluoro-4-methylanilino)furo[3,4-b]pyrazine-1,5-dione 1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)pyrrolidine-4-carboxamide N-[2-azidooxy-1-(4-benzylphenoxy)ethoxy]hydroxylamine 4-[2-(4,4-difluoropiperidine-1-carbonyl)phenyl]-5H-pyrido[3,2-b]indole-7-carboxamide [4-(3,6-dihydro-2H-pyran-4-yl)-1-(4-fluorophenyl)pyrazol-3-yl]urea 4-(2,6-dichlorophenyl)-N'-hydrazinyl-7H-pyrrolo[2,3-d]pyrimidine-5-carboximidamide 2-(3-fluorophenyl)-6-methoxyphenol N-butyl-3-[2,4-difluoro-6-(trifluoromethyl)phenyl]sulfanylpropanamide 2-(4-chlorophenyl)sulfonyl-3,5-dihydropyrrolo[3,2-d]pyrimidine N-methyl-2,5-dioxopyrrole-1-sulfonamide;2-[6-(4-phenylphenoxy)hexanoylamino]acetic acid N-[(E)-3-amino-1-(4-methylphenyl)-2-oxoprop-1-enyl]azetidine-3-carboxamide 4-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]-N-(2,6-difluorophenyl)benzamide 4-[5-(6,7,8,9-tetrahydropyrido[3,2-b]indolizine-5-carbonyl)thiophen-2-yl]piperidine-1-carboxylic acid 3-[2,6-difluoro-4-(propylsulfanylmethyl)phenyl]cyclopentane-1-carboxylic acid 3-(2,6-dichlorophenyl)sulfanyl-N'-hydroxypyrazine-2-carboximidamide 2-(N-(2,4-dichloropyrimidin-5-yl)-3-hydroxyanilino)propanoic acid (3,4-dichlorophenyl)methylsulfanium 2-(4-chlorophenyl)ethyl-[4-(5,6-dimethylbenzimidazol-1-yl)-3-isocyano-6-morpholin-4-ylpyridin-2-yl]azanium 1-[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]pyrazole-4-carboxylic acid 1-(benzenesulfonyl)-3,4-dihydropyrrolo[2,3-b]pyrazin-6-one N-[2-(6-ethoxypyridin-3-yl)-3,4-dihydro-1H-isoquinolin-7-yl]-5-fluoropyridine-2-carboxamide 2-[[4-[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]-3-fluorophenoxy]methyl]benzonitrile 3-[2-(dimethylamino)ethoxy]-N-ethylsulfonyl-1,5-naphthyridine-4-carboxamide 1-(3,5-dimethylphenyl)-4-[4-[4-[[4-[2-(2H-tetrazol-1-ium-1-yl)phenyl]phenyl]methoxy]-1H-benzimidazol-2-yl]phenyl]butan-2-one [(1R,2S)-3-[4-(cyclopropanecarbonylamino)phenyl]sulfonyloxy-6-oxocyclohexyl]carbamic acid 5-bromo-4-(3,5-dimethylanilino)-1H-pyrimidin-6-one (E)-3-[5-chloro-2-fluoro-4-[(E)-2-(1H-indazol-3-yl)ethenyl]phenyl]prop-2-enoic acid 2-aminooxycarbonylbenzenesulfinate 2-amino-3,5-bis(2-ethylhexoxy)benzaldehyde 4-(2,3-dichlorophenyl)sulfonyl-N-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperazine-1-carboxamide 1-(5,7-dimethylpyrazolo[3,4-d]pyrimidin-2-yl)-6,8-dihydro-5H-imidazo[2,1-c][1,4]oxazine [2-(difluoromethyl)pyrrolidin-1-yl]-[3-propan-2-yl-5-(trifluoromethyl)pyridin-4-yl]methanone (3S)-6,8-dimethyl-1-propanoyl-2,3,4a,5,7,8,8a-octahydro-[1,4]dioxino[2,3-c]pyrrole-3-carboxamide 5-benzyl-6-chloro-1H-pyrimidine-2,4-dione;ethane 5-[(4-chlorophenyl)methoxy]-2-[1-[4-[6-(ethylamino)pyridin-3-yl]-3-fluorophenyl]ethyl]pyran-4-one N-[2-(3,5-dimethoxyphenyl)ethyl]-N-ethyl-4-methylcyclohexa-1,5-dien-1-amine 2-chloro-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]-N-propylacetamide N-[6-(4-iodopiperazin-1-yl)pyridin-3-yl]-5,7-dihydropyrrolo[2,3-d]pyrimidin-4-amine (4-hydroxy-3-phenylsulfanylphenyl)-piperazin-1-ylmethanone 6-hydroxy-1,4,5-trimethylnaphthalene-2-carboxylate 3-(2-tert-butylphenyl)-4-methoxycarbonylpiperazine-1-carboxylate 5-chloro-4,7-dimethyl-2-propan-2-ylisoquinolin-1-one;3,6-diaminopyrazine-2-carboxamide 2-(4-azidophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine 2-methylsulfonyl-1,3,8-triazaspiro[4.5]deca-6,9-diene 4-(3,4-dichlorophenyl)sulfanyl-5-[(2S,4R,6S)-2,6-dimethoxyoxan-4-yl]sulfanyl-N'-hydroxypyridine-2-carboximidamide 4-(2,3-dihydropyridine-5-carbonyl)-N-[1-oxo-1-[[4-[5-(trifluoromethyl)-1H-imidazol-2-yl]phenyl]methylamino]propan-2-yl]benzamide (2S)-2-methyl-4,4-bis(phenylmethoxy)butanamide 2-ethyl-6,7-dimethoxyphenanthrene 2-[4-chloro-3-(2H-tetrazol-5-yl)phenyl]acetamide N-[2,4-difluoro-3-[5-(morpholin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]propanesulfonamide N-[(2E,4Z)-6-methylideneocta-2,4-dien-3-yl]-2-phenylbenzamide N-[(3-ethylthiophen-2-yl)methyl]-4-[(5-oxopyrrolidin-3-yl)amino]cyclohexane-1-carboxamide 3-(3,4-dihydroacridin-1-yl)propane-2,1-diol 4-(5-benzylpyridine-3-carbonyl)morpholine-2,6-dione 5-[(1Z,3E)-4-aminobuta-1,3-dienyl]-2-[5-(methoxymethyl)-1H-pyrazol-3-yl]phenol (2S)-1-[3-[1,5-dimethyl-2-[4-(trifluoromethoxy)phenyl]-6H-azulen-7-yl]propanoyl]pyrrolidine-2-carbonitrile 5-tert-butyl-N-[(4S)-2-formamido-3,3,3-trifluoro-1,2-oxazolidin-4-yl]thiophene-2-carboxamide;2-methoxypyridine (2E)-N,3-dimethyl-1-thiophen-2-ylhexa-2,5-dien-1-imine 3-[[2-(aminomethyl)morpholin-4-yl]-hydroxymethyl]-2,6-dichlorobenzamide 2-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]cyclohexan-1-one 1-[2,6-difluoro-4-(2-pentoxyethyl)phenyl]-5,5-dimethylpyrazolidin-3-one 2-[[4-fluoro-3-(trifluoromethyl)phenyl]carbamoyl]benzoate 6-(5,8-dioxa-14-azatricyclo[15.2.1.03,12]henicosa-1(20),3(12),4,6,13,19-hexaen-18-yl)hexan-1-ol [5-[3-(4,4-diphenylpiperidin-1-yl)propoxy]-2-methylpyridin-3-yl]carbamic acid N-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-6-[4-hydroxy-2-(trifluoromethoxy)phenyl]-5H-pyrrolo[3,4-b]pyridine-7-carboxamide 2-[(3R)-1-(cyclopentylmethyl)piperidin-3-yl]oxypyrimidine (2S)-4-[(3R,6S)-1-benzyl-5-oxopyrrolidine-3-carbonyl]piperazine-2-carboxylic acid (4S)-4-amino-5-[2-fluoro-3-(5-morpholin-4-ylpentanoyl)anilino]-5-oxopentanoic acid 1-[4,6-bis(2-methoxyphenyl)-1H-pyrimidin-2-ylidene]-3-[3-tert-butylsulfanyl-5-(methanesulfonamido)pyridin-2-yl]urea 2-[1,1-difluoro-3-(4-methylphenyl)propoxy]pyridine 2-(3-bromoquinolin-7-yl)oxypropanoic acid 4-[(4-fluorophenyl)sulfonylamino]piperidine-1-carboxylic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxy-4-phenylbutanamide (2Z,4E)-2-ethenyl-3,6-dimethylhepta-2,4,6-triene;1-fluoro-4-[(3S)-pentan-3-yl]benzene 2-[3-fluoro-4-(trifluoromethyl)phenyl]acetamide 4-[(4-azidopyrimidin-2-yl)amino]cyclohexan-1-ol 2,4-difluoro-1-methoxybenzene;3,3-difluoro-5-[(E)-2-phenylethenyl]-2H-1,2,4-oxadiazole 2-amino-3-[4-hydroxybutyl(methoxycarbonyl)amino]benzoic acid 5-azido-1-(2,6-dimethylmorpholin-4-yl)benzimidazole N-[(3S)-1-(6-bromopyridin-3-yl)piperidin-3-yl]-2,4-dimethylpyrimidine-5-sulfonamide (2R)-2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-N-methyl-N-(oxan-4-yl)propanamide 2-(4-tert-butylphenyl)-3H-pyrrolo[1,2-a]pyrazine 3-(2,5-dichloro-N-propylanilino)butanoic acid N-(4-methoxy-2,3,5,6-tetramethylphenyl)cyclobutanecarboxamide 3-methyl-1,2-dioxo-N-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-5-yl)-3H-isoindole-4-carboxamide [4-[3-[(4-cyclopropylpiperazin-1-yl)methyl]phenyl]-5-fluoropyridine-2-carboximidoyl]iminoazanium 2-amino-3-[4-(9H-fluoren-1-yl)piperazin-1-yl]propanoic acid (4S)-2'-amino-6-[3-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]spiro[2H-indole-3,9'-xanthene]-1-one;2,4-diaminopyrimidine-5-carbonitrile 1-[2,4-bis(5-methylthiophen-2-yl)buta-1,3-dien-2-yl]-4,5,6,7,8,9-hexahydrocycloocta[d]imidazole 3-methylsulfanyl-N-[5-(3,4,5-trimethoxyphenyl)-1H-pyrazol-3-yl]propanamide 2-(5,6-dimethylpyridine-3-carbonyl)-7-oxa-2,10-diazaspiro[4.6]undecan-9-one 1-phenyl-3,5-dihydropyridazino[4,3-b]indole N-[2-(5-chlorocyclohexa-1,3-dien-1-yl)propan-2-yl]-4-cyanobenzamide N-[4-fluoro-5-(2-morpholin-4-ylpyrimidin-5-yl)-2-piperidin-1-ylphenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide 3-amino-4-cyano-5-[2,6-difluoro-4-(trifluoromethoxy)phenyl]-1H-pyrrole-2-carboxamide 2-[5-[(4-fluorophenyl)methyl]thiophen-2-yl]-3H-benzimidazole-5-carboxamide 4-(2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl)piperazine-1-carboxylic acid 5-(2,4-dichlorophenoxy)carbonyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid 6-bromo-1-methylpyrrolo[2,3-b]pyridine 4-[5-(3,5-dimethylpyridin-2-yl)heptanoyl]benzoic acid N-[3-(dimethylamino)propyl]-4-(2-methoxyphenyl)-7-oxothieno[3,2-b]pyridine-6-carboxamide N-(3,4-dimethoxyphenyl)-6-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-7,8-dihydro-5H-pyrido[3,4-b]pyrazine-2-carboxamide (3E)-4,6-dimethyl-1-[2,2,4-trimethyl-5-(5-phenylmethoxypyridin-3-yl)-4H-pyran-3-yl]hepta-3,7-dien-2-one 4-[3,5-bis(trifluoromethyl)phenyl]-2-(4,6-dihydrotriazolo[1,5-a]pyrazin-7-ylidene)thiomorpholine 1-amino-4,6-dibromo-9H-fluorene-3-carboxylic acid 2-(4-methylphenyl)sulfinyloxybenzoate N-[1-(3,5-dimethylpiperidin-4-yl)ethenyl]-6-fluoropyridin-2-amine;ethane (2Z,5E)-3,4-diethyl-1-hydroxy-7-methyl-5-phenylhepta-2,5-dien-4-amine 1-[4-(4,5-diphenylimidazolidin-3-ium-1-yl)butoxy]ethanethiol 1-[7,8-difluoro-6-(3-methoxyphenyl)naphthalen-2-yl]ethanamine N-[(1,4-dimethylpyrrolidin-3-yl)methyl]-5-(2-fluoro-6-methoxyphenyl)pyridine-2-carboxamide 5-methylspiro[2H-indole-3,8'-7,9-dihydropyrrolo[1,2-a][1,4]diazepine] 2-(1,4-dimethylpyridin-1-ium-3-yl)-6-fluoro-7-(1H-pyrazol-5-yl)-[1]benzofuro[2,3-b]pyridine N-[3-(1,4-diazepane-1-carbonyl)phenyl]-2-piperidin-1-ylpyridine-4-carboxamide [4-[(3,5-dimethylpyrazol-1-yl)methyl]phenyl]boronic acid 2,6-ditert-butyl-4-[(Z)-[1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]ethylidenehydrazinylidene]methyl]phenol 4-[3-(2,6-dimethoxyphenyl)piperazin-1-yl]-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine 3-[4-(3-phenylphenyl)phenyl]pyridine 5-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N'-hydroxypyrazine-2-carboximidamide N-[2-amino-3-(cyclohexylmethoxy)propoxy]-4-[[6-(trifluoromethyl)pyridine-3-carbonyl]amino]benzamide [(2S,4R)-1-benzylpiperidin-4-ol 1-[(3E)-4,8-dimethylocta-3,7-dienyl]pyrazole-3-carboxylic acid 3-methylbut-1-ene;7,15-trimethoxytetracyclo[10.2.0.02,5.06,11]pentadeca-1(14),6,8,10-tetraen-12-one 5-chloro-2-[(5S)-4,8-diazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3-trien-11-yl]phenol N-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]acetamide [(2S,3R)-2-[1-(2-methoxyethyl)imidazol-2-yl]oxolan-3-yl]methanol N-(2-hydroxyethyl)-N,N'-dimethyl-N'-[(3R,4S)-4-(pyridin-3-ylmethoxy)oxolan-3-yl]ethane-1,2-diamine 2-[3-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydropyrimido[4,5-c]azepine N-[5-(3,4-dichlorophenyl)sulfonylhexyl]isoquinoline-5-sulfonamide N-[[3,4-dioxo-2-(trifluoromethyl)cyclobuten-1-yl]amino]benzamide N-[(1R,2S)-2-[4-[5-chloro-6-(trifluoromethyl)pyridin-3-yl]phenyl]cyclopropyl]propanamide 2-[(1R)-1-phenylethyl]piperidine-4,6-dione (3R)-1-[6-chloro-5-[4-(4,4-dimethylpiperidine-1-carbonyl)phenyl]-1H-indol-2-yl]-N',N-dimethylpyrrolidine-3-carboximidamide 1-(7-methylnaphthalen-2-yl)-3-pentoxybutan-2-one 5-chloro-6,7-diethyl-3-phenyl-4H-triazolo[1,5-a]pyrimidin-8-one [(7R)-4,8-dimethyl-2-[[1-[[6-(trifluoromethyl)pyridin-3-yl]methyl]pyrazol-4-yl]amino]-5,7-dihydropteridin-6-ylidene]-hydroxyazanium 7-[3-(hydroxymethyl)piperidin-1-yl]chromen-2-one (NZ)-N-[2-(3,4-dihydrocarbazol-9-yl)ethylidene]hydroxylamine 1-[(2,6-dimethylphenyl)methylamino]-3-(1H-inden-5-ylmethyl)urea 1-[4-(2,3-dihydrofuran-5-ylmethoxy)phenyl]propane-2-thiol 1-(2,5-dimethylthiophene-3-carbonyl)-N-(3-oxo-4H-1,4-benzothiazin-7-yl)piperidine-3-carboxamide N-[5,7-difluoro-6-(3-methylpyrazol-1-yl)-1H-indazol-4-yl]-2-(oxolan-3-yl)acetamide 2-bromo-1,5-difluoro-3-methoxybenzene;ethane 2-(3-ethoxypropyl)isoindole 2-[1-acetyl-5-chloro-3-(2,6-dimethoxyphenyl)-4-oxoquinazolin-2-ylidene]propanedinitrile [5-chloro-4-[(2,4-difluorophenyl)methoxy]-1H-indazol-3-yl]-(4-methylpiperazin-1-yl)methanone 6,7-dimethoxy-2-methylsulfanylquinazoline;ethane (3aR,7aS)-2-[(6R,8S)-8-(furan-3-ylmethyl)-6-phenyl-1,4,7,7a-tetrahydropyrano[3,4-c]pyrazol-3-yl]-5-methyl-1,3,3a,6,7,7a-hexahydropyrrolo[3,4-c]pyridine 1-[6-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]pyridazin-3-yl]-N-[(3R)-5,5-difluoropiperidin-3-yl]azetidine-3-carboxamide 4-bromo-N-(2-methylphenyl)pyridine-3-carboxamide 2-(4-methoxyphenoxy)sulfonylphenolate 3-(7,8-dihydro-[1]benzothiolo[2,3-b]pyrazin-6-yl)aniline (5S)-2-[(3,4-dimethylphenyl)methylsulfanyl]-N-naphthalen-1-yl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-ethoxy-6-[(3S,4R)-1-[(2R)-2-hydroxypropanoyl]-4-methylpyrrolidin-3-yl]pyridine-3-carbonitrile N'-(4-chlorobenzoyl)-3,3,5-trimethylcyclohexanecarbohydrazide 4-amino-5-(3,4-dimethylphenyl)imino-1,2-thiazol-3-one N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-methylpropanamide 5-bromo-N-[3-(2-chloro-6,7-dihydro-1H-indol-4-yl)phenyl]-2-methoxypyridine-3-carboxamide 1-ethyl-N-[[5-fluoro-2-methoxy-4-(triazol-2-yl)phenyl]methyl]-N-[1-[[3-[2-fluoro-6-hydroxy-5-(morpholine-4-carbonyl)cyclohexa-1,3-dien-1-yl]imidazo[1,2-a]pyridin-7-yl]methyl]piperidin-4-yl]-5-methylpyrazole-4-carboxamide 5-[(E)-2,3-dimethylbut-1-enyl]-6-[(2S,4R)-4-methoxyoxan-2-yl]naphthalen-2-ol (2S)-2-[3-[4-methyl-N-(2,2,2-trifluoroethyl)anilino]propyl]hexanamide 4-(2,3-difluorophenyl)-1-[2-hydroxy-6-methyl-5-[4-(trifluoromethoxy)phenyl]hexanoyl]piperidine-4-carbonitrile (3-azido-2,4-dimethylphenyl)methanol 1-(3,4-difluorophenyl)sulfonyl-2-(methoxymethyl)pyrrolidine-2-carboxylic acid 2-[3,5-dichloro-4-(3-cyanophenoxy)phenyl]-1,1,1,3,3,3-hexafluoropropane-2-sulfonic acid N-(3-chlorophenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide;hydrochloride 2-[(E)-2-carboxyethenyl]sulfonyloxybenzenesulfonate 7-[(2R)-1-cyclopentylpropan-2-yl]-4-methoxyquinoline 5-[1,1-bis(sulfanyl)ethoxy]-2-methoxybenzoic acid 1,3-difluoro-5-[4-[2-(4-pentylphenyl)ethynyl]phenyl]benzene;ethane 4-[(Z)-2-methyl-3-phenylprop-1-enyl]aniline N-cyclohexyl-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-3H-pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide 2-methyl-N,N-bis[(4-methoxyphenyl)methyl]pentan-1-amine 4-(benzenesulfonyl)-2-(1H-inden-1-yl)thiophene (2Z,5S)-3-(2-methylphenyl)-4-oxo-2-[(Z)-1-phenylethylidenehydrazinylidene]-1,3-thiazinane-6-carboxylic acid N-(5,6-difluoro-1H-indol-3-yl)-2-(methoxymethyl)-1H-indole-6-sulfonamide 3-[[1-(3,5-difluorophenyl)-2-hydroxyethyl]amino]-N-methylpyrrolidine-1-carboxamide 2,2-bis(3,4,5-trimethoxyphenyl)acetic acid (2S,4S)-N-[6-chloro-3-nitro-1-(oxan-2-yl)pyrazolo[4,3-b]pyridin-5-yl]-7-methoxy-2,4-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide 5-(1,3-benzodioxol-4-yl)-6-[ethyl(methylsulfonyl)amino]-2-methylpyridine-3-carboxylic acid N-[(2S,3R)-5-amino-2-hydroxyhexanoyl]pyridine-4-carboxamide 4-[(2S)-3-phenylbutan-2-yl]phenol 1-[(3-cyclopropyl-2,5-dimethoxyphenyl)methyl]-N,4-dimethylpiperidine-4-carboxamide;formic acid 4-methoxy-1,3-dimethylpyrazolo[4,3-b]quinoline 3-fluoro-N-[4-(2-methoxyphenyl)-5H-cyclohepta[d]imidazol-7-yl]benzamide 4-[[(6S)-9-chloro-1,5-dimethyl-5H-chromeno[3,4-c]pyridine-8-carbonyl]amino]butanoic acid (3R)-1,2,3,4,5,9b-hexahydrobenzo[e]isoindole (2-azidopyrrolidin-1-yl)-[3-phenylmethoxy-4-(trifluoromethyl)phenyl]methanone N-(2,5-dimethylphenyl)sulfanyl-2-methylaniline (2S)-4,6-dimethyl-8-propanoyl-7-(pyridine-3-carbonylamino)octanoic acid (Z)-N'-[2,5-dimethoxy-4-[(6R)-1,3,10-trihydroxyundec-8-enyl]phenyl]prop-1-ene-1,3-diamine N-[2-(4-methoxyphenyl)-3H-benzimidazol-5-yl]-3,5-bis(trifluoromethyl)benzamide 4-azidooxy-3,6-dimethylquinoline 3,5-dimethyl-2-(1H-pyrrolo[2,3-b]pyridin-2-yl)benzoic acid (2R)-1-[4,5-bis(4-fluorophenyl)-3-methyl-1H-pyrrol-2-yl]propan-2-amine;hydrochloride [3-(2,4-difluorophenoxy)-2,5-bis(trifluoromethyl)phenyl]methanamine 1-[(4aR,8aS)-8a-hydroxy-5-methyl-2,3,4,4a,9,10,10a-octahydropyrano[3,2-c]chromen-6-yl]-3-(4-fluoro-3-nitrophenyl)urea 5-[2,3-bis(hydroxyimino)indol-1-yl]-1,6-dihydropyrazolo[4,3-d]pyrimidine-7-thione 6-[2,3-bis(ethenyl)phenyl]dibenzofuran 2-[1-(3,5-dichlorophenyl)ethyl]-8-methoxyquinoline (2S)-N-[(1R)-3,4-dihydro-1H-isochromen-6-yl]-2-methoxy-N'-[5-[5-(trifluoromethyl)pyridin-2-yl]-1,3,4-thiadiazol-2-yl]propanediamide 3-(5,6,7,8-tetrahydronaphthalen-2-yl)oxirane-2,2-dicarbonitrile (3aR,7aS)-5-[(4-fluorophenyl)methyl]-1,2,3,3a,6,7,7a-octahydropyrano[3,4-b]pyrrole;2,2,2-trifluoroacetic acid N-[6-(2,3-dihydro-1H-inden-4-yl)pyridin-2-yl]acetamide 4-[3-[(1Z)-buta-1,3-dienyl]-2-methylidenepyrrol-1-yl]benzoic acid;ethane (4S)-1-(2,6-dimethylphenyl)-3-methyl-4-(4-propan-2-yloxybenzoyl)-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 3-[(3R)-2,7,9-trimethyl-1,10-dioxo-3H-benzo[f]chromen-3-yl]propanal 4-amino-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxylic acid 1-[(3R,4S)-4-hydroxypyrrolidin-3-yl]-6-oxo-N-[(2-propan-2-ylphenyl)methyl]-5H-benzo[b][1,4]benzoxazepine-3-carboxamide N-(4-bromophenyl)-2,6-dichloro-N-octylaniline N-[(5-bromopyridin-3-yl)methoxy]-1H-indazole-3-carboxamide 1-(6,7-dimethoxy-3,4-dihydro-2H-quinolin-1-yl)propan-2-one 4-[(E)-3-(furan-2-yl)prop-1-enyl]-N,N-dimethylaniline (3R)-7',8'-dichlorospiro[2H-isoindole-3,1'-naphthalene]-1-one N-[2-(azidomethyl)phenyl]pyridine-3-carboxamide 3-[(5R)-6-amino-1,2,4-triazin-3-yl]piperidine-1-carboxylate N-(1,2-dihydropyrimidin-6-yl)-3,5-dimethylpyridine-2-carboxamide 4-[2,2-dimethoxyethyl(hexadecanoyl)amino]benzenesulfonic acid 3-[(3R,4S)-1-(cyclohexanecarbonyl)-4-methoxypyrrolidin-3-yl]-1-ethylimidazo[4,5-b]pyridin-2-one 2-ethoxy-6-[(4E,5Z)-4-ethylidenenona-1,5-dienyl]benzonitrile 2-[3-(8-hydroxyquinolin-7-yl)oxypropyl]benzoic acid 1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]benzimidazole-5-carboxamide 1,7-dibromoheptane;formaldehyde;(5Z)-3-methyl-2-[4-methyl-3-(morpholine-4-carboximidoyl)phenyl]-N-propan-2-ylideneocta-5,7-dienamide 4-[3-(azetidin-1-yl)propylamino]-2-propan-2-yl-1H-pyrimidin-6-one N-azido-2,5-dichloropyrimidin-4-amine 6,7-dihydro-5H-cyclopenta[c]pyridin-3-yl(pyridin-4-yl)methanamine 4-[4-(aminomethyl)phenyl]sulfonyl-1,2,5-trimethylpyrrole-3-carboxylic acid 2-[(Z)-2-aminoethenyl]-5-(2,3-dihydro-1H-indol-6-ylmethyl)cyclohexane-1,3-dione N-azido-1-(2,5-diethylphenyl)methanesulfonamide N-[2-(4,6-dimethylpyridin-2-yl)propan-2-yl]formamide ethane;2-fluoro-4-[(E)-[(3Z)-3-[methyl-(5,6,7,8-tetrahydronaphthalen-1-ylamino)hydrazinylidene]pentan-2-ylidene]amino]phenol 1-[1-(4-methoxyphenyl)propyl]pyridin-2-one (E)-1-[4-[2-amino-5-(5-chloropyridin-3-yl)-6-ethanimidoyl-1H-indole-3-carbonyl]piperazin-1-yl]-4-(dimethylamino)but-2-en-1-one (3R,4S)-1-[6-(2-cyclopropylpyrazol-3-yl)pyridazin-3-yl]-4-fluoropiperidin-3-amine 1-ethyl-4,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-9,11-diene 4-[4-(3,5-dichloropyridin-4-yl)piperazin-1-yl]sulfonylbenzoic acid 2,2-dimethyl-3-[4-(2-methylbutan-2-yloxycarbonyl)benzoyl]cyclopropane-1-sulfonate [4-(3,5-dimethoxyphenyl)sulfonylmorpholin-2-yl]-pyrrolidin-1-ylmethanone 3-(3,4-dimethoxyphenyl)-1H-indole 6-methoxy-N-[4-(1,3-oxazol-5-yl)phenyl]quinoline-8-carboxamide 2-[4-azido-5-(2,3,4-trifluorophenyl)furan-2-yl]pyridine 1-(2,5-dimethylfuran-3-carbonyl)-N-[4-[[2-oxo-6-(trifluoromethyl)-3H-pyridin-5-yl]amino]cyclohexyl]piperidine-2-carboxamide 2-N-[3-(1,1-difluoroethyl)-5-[4-(3,3-dimethoxypropoxy)phenyl]thiophen-2-yl]benzene-1,2,3,4,5-pentamine 2-[N-(cyanomethyl)-4-[2,4,6-trichloro-N-(2-phenylethyl)anilino]anilino]acetonitrile [4-(2,5-dimethylanilino)pyrimidin-5-yl]methanol;propane 1-[4-(5-cyclopropylpyrazole-1-carbonyl)phenyl]imidazolidin-2-one 6-chloro-N-[4-methylsulfanyl-3-(trifluoromethoxy)phenyl]quinazolin-2-amine 3-(4-chlorophenyl)-1,6-dimethyl-2,7-dihydropyrazolo[3,4-d]pyrimidine 2-[2-(dimethylamino)ethyl]-4-nitrophenol 6,7-dihydro-4H-thieno[3,2-c]pyridine;5-(oxan-4-yl)imidazo[1,5-a]pyrazin-8-one 2-(3,5-dimethoxyphenyl)pyridine 2-(3-chloropropyl)-5,5,10b-trimethyl-8-phenylmethoxy-1,2,3,4,4a,6-hexahydropyrido[3,4-b]indole 1-ethyl-3-[4-[(6R)-8-methoxy-6,7-dihydro-5H-quinazolin-2-yl]phenyl]urea 1-amino-3-[[4,5-bis(4-chlorophenyl)-1H-imidazole-2-carbonyl]amino]thiourea N-[(3R)-1-[4-(6-chloropyridin-2-yl)phenyl]pyrrolidin-3-yl]-6-methoxy-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine [(3R)-1-[6-(2,2,4,4-tetramethylpentanoylamino)naphthalene-2-carbonyl]piperidin-3-yl]carbamic acid N-[(2S,4R)-1-(3-cyanoazetidine-1-carbonyl)-4-fluoropyrrolidin-2-yl]-5-[3-[4-fluoro-6-(trideuteriomethylamino)pyridin-3-yl]phenyl]-1-methylimidazole-2-carboxamide 3,5-di(propan-2-yl)pyrrolo[2,1-c][1,4]benzodiazepine N-[4-(3,5-difluorophenyl)-1-hydroxy-3-methoxybutan-2-yl]acetamide N-(3,5-difluorophenyl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxamide 3-[6-(ethyliminomethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl]thiophene-2-sulfonic acid 1-(4,6-dimethyl-2H-pyrazolo[3,4-c]pyrazol-3-yl)ethanone N-(1H-indol-4-ylmethyl)propanamide N-(3,4-dimethoxyphenyl)-2-[3-(1H-imidazol-5-yl)anilino]-6-morpholin-4-ylpyrimidine-4-carboxamide 1-methyl-3-[5-(4,4,5,5-tetramethyloxaborolan-2-yl)pyrazin-2-yl]urea N-(4,5-dimethylpyrimidin-2-yl)-4-[hexyl-(2-oxo-2-propoxyethyl)amino]benzenesulfonamide (1S)-N-[5-chloro-6-methoxy-2-(trifluoromethyl)pyridin-3-yl]-2,3-dihydro-1H-indene-1-carboxamide 2-[(1Z)-1-(ethylideneamino)buta-1,3-dienoxy]-N-methylaniline 1-[(4-ethenylphenyl)methylamino]ethenol (2R)-2,3-diaminopropanal;6-methyl-N-[(4-methylphenyl)sulfanylmethoxy]naphthalene-2-carboxamide 3-[2,4-bis(prop-1-en-2-yl)phenyl]-N-ethenyl-5,7-dimethyl-2-prop-1-ynylpyrazolo[1,5-a]pyrimidin-6-amine 1-chloro-5-(4-ethoxyphenyl)cyclohexa-2,4-diene-1-sulfonic acid 7-[5-(5-fluoropyridin-2-yl)-1H-imidazol-4-yl]-N,N-dimethylimidazo[1,5-a]pyrazin-8-amine 2-[[3-cyclohexyl-1-(3-phenylpropanoyl)azetidine-3-carbonyl]amino]propanoic acid 4-(1,5-dimethylpyrazole-3-carbonyl)-11-phenyl-1-oxa-4,11-diazaspiro[5.6]dodecan-12-one 2-[(2R,5S)-1-[3,4-difluoro-2-(trifluoromethyl)benzoyl]-5-methoxypyrrolidin-2-yl]-N-methylacetamide 1-azidosulfanyl-2,3-dimethoxybenzene 1-[(2R)-4,4-difluoro-2-methylpyrrolidin-1-yl]-6-[(1S)-1-pyridin-3-ylethoxy]isoquinoline 3-(cyclopenten-1-yl)-4,5-difluoroaniline 2-fluoro-4-[[(3S)-1-[2-methyl-6-oxo-5-(propanoylamino)hexan-2-yl]piperidine-3-carbonyl]amino]benzoic acid 1-N',3-N'-dimethyl-4-(3,3,5,5,6-pentamethylcyclohexen-1-yl)benzene-1,3-dicarboximidamide [(E)-3-amino-1-phenylbut-2-enylidene]azanium 2-[4-(2,5-difluorophenyl)phenyl]bicyclo[1.1.1]pentane 2-[7-[5-(azidomethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-3-yl]propan-2-ol 6,7-diphenyl-2-(4-pyridin-4-ylpiperazine-1-carbonyl)pyrrolo[3,2-d]pyrimidin-5-one N-[4,5-dimethyl-3-(1-methylindol-2-yl)-5H-1,2,4-triazin-6-yl]acetamide 1-(2-azidoethyl)-6,7,8-trimethoxyimidazo[4,5-c]quinoline 2-(3,5-diaminophenyl)benzoic acid 2-chloro-N-[5-(6,7-dimethoxyquinolin-4-yl)sulfanyl-1,3,4-thiadiazol-2-yl]acetamide 3-[(2S)-butan-2-yl]-4-oxo-1H-pyridine-2-carboxamide N-azido-3,4-difluoronaphthalene-1-carboxamide N-[3-amino-6-(5-fluoropyridin-2-yl)pyridazin-4-yl]spiro[2.3]hexane-5-carboxamide 3-(2,4-dimethylphenyl)-8-fluorospiro[chromene-2,1'-cyclobutane]-4-one 3-[(4-methoxyphenyl)methylamino]-N'-methylthieno[2,3-b]pyridine-2-carboximidamide 2-[4-methyl-3-[5-(methylamino)-1H-pyrrol-2-yl]phenyl]benzoic acid (NE)-N-[[2,6-dimethyl-4-(trifluoromethyl)phenyl]-[5-ethoxy-2-(methylamino)phenyl]methylidene]hydroxylamine 3-N,4-dimethyl-1-N,1-N-bis(prop-2-enylidene)benzene-1,3-disulfonamide 5-(6,7-dimethoxyquinolin-4-yl)-2H-isoindole 1-(2,3-dihydro-1H-inden-5-yloxy)-N-ethylpropan-2-amine 1-methoxy-2-[4-(trifluoromethyl)phenyl]piperazine 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-4-[4-hydroxy-1-[(6R)-6-phenyloxan-2-yl]butyl]-1H-1,2,4-triazol-5-one 4-[3,5-bis(trifluoromethyl)phenyl]-N-[2-(cyclopropylamino)ethoxy]cyclohexane-1-carboxamide 1,6-bis(3-hydroxypropyl)-10H-anthracen-9-one 2-[(1S,3R)-3-azidocyclohexyl]benzamide 4-[2-(3,5-dimethylphenyl)propan-2-yl]benzenesulfonamide 4-(2,2-dimethylpropoxy)carbonylbenzenesulfonic acid 2-(1H-indol-3-yl)-2,7-diazaspiro[4.5]decane 7-hydroxy-6,11-dihydrobenzo[c][1]benzoxepine N-[4-[3-methylbutyl(2H-tetrazol-5-yl)amino]phenyl]sulfonylbenzamide 4-fluoro-1-(3-methylbutoxy)-2,5-diphenylbenzene 5-benzylimino-4,4-dimethylpyrazolidin-3-one 2-N-[4-(3,5-dichlorophenyl)sulfonylcyclohexyl]-5-fluoropyrimidine-2,4-diamine 4-[(2-hydroxycyclopentyl)amino]-N-pyrimidin-5-ylpyrrolo[1,2-b]pyridazine-3-carboxamide 2-[3,5-dichloro-4-[(5-oxo-1,6,8-triazatricyclo[7.2.0.02,7]trideca-3,6,9,11-tetraen-12-yl)oxy]phenyl]-6-oxa-2,4-diazaspiro[3.4]octan-7-one 2-(3-methylbutanoyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-3-carboxamide 4-[5-(2,6-difluorophenyl)-1H-pyrazol-3-yl]-1-pyridin-4-ylbutan-1-one N-[2-bromo-4-(1,1-difluoropropyl)phenyl]-5-methoxy-3H-indole-2-carboxamide 4-amino-6-[(2,3-dihydroxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-[4,5-dimethyl-3-[(E)-2-phenylethenyl]pyrazol-1-yl]-N-phenylacetamide 2-[azido(cyclopentyl)methyl]sulfanylnaphthalene 2-(3,5-dimethylpyrazol-1-yl)-N-[4-[1-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)pyrrolidin-3-yl]phenyl]acetamide (2S)-N,5-dimethyl-1-[4-[methyl(3-phenylpropanimidoyl)amino]benzoyl]pyrrolidine-2-carboxamide;ethane 5-[4-(dimethylamino)phenyl]-3,6-bis(propylsulfanyl)cyclohexa-2,4-dien-1-one N-[3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]cyclohexyl]-7-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide (2Z,5S)-2-[(Z)-(3-bromophenyl)methylidenehydrazinylidene]-5-propan-2-yl-1,3-thiazolidin-4-one 1-azido-2-(4-ethoxyphenyl)-3,5-difluorobenzene 3-chloro-2,4,6-tris(trifluoromethyl)pyridine (4R,5S)-2-chloro-4-ethenyl-1-methyl-3-phenyl-4,5-dihydroimidazol-3-ium 4-(5,8-dibromoquinolin-6-yl)-3-methoxybenzaldehyde 2-[(E)-2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethenyl]isoindole 2-[(3,4,5-trimethoxyphenyl)methyl]aniline [(2R)-1-[(6,8-dichloro-4-oxochromene-2-carbonyl)amino]pentan-2-yl]-triphenylphosphanium [(3aS,4R,8bS)-5-methyl-2,2-diphenyl-1,3a,4,8b-tetrahydrocyclopenta[a]inden-3-yl]azanium (4S)-1-[4,6-dichloro-5-(trifluoromethyl)pyrimidin-2-yl]-4-hydroxypiperidine-3-carboxylic acid 5-(3,4-dichlorophenyl)pyridine-2,6-diamine 6-chloro-4-(3,5-dimethylphenyl)-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 1-[(2R)-1-hydroxypropan-2-yl]indole-7-carboxamide (4S)-1,3-dimethyl-4-thiophen-2-yl-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one 3-[3-methoxy-5-(trifluoromethyl)phenyl]-1,3-diazaspiro[4.5]decane 2-[(6S)-5-chlorospiro[3,4-dihydrochromene-2,1'-cyclohexane]-7-yl]oxyethanethiol N-[4-(4,7-dimethylquinazolin-2-yl)sulfanylphenyl]-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)butanamide [5-(1,1-difluoroethyl)-2-[3-(methylsulfanylamino)but-3-enoxy]phenyl]-(4-methylpiperidin-1-yl)methanone (2S)-1-azidooxy-4-methylsulfanyl-3-[2-(trifluoromethyl)phenyl]butane-2-thiol 2-[[3-(4-methoxyphenoxy)piperidin-1-yl]sulfonylamino]acetamide 5-[1-(cyclopropylmethylamino)buta-1,3-dienyl]-2-N-ethyl-4-N-[6-fluoro-5-(pyridin-3-ylmethoxy)-1H-benzimidazol-2-yl]pyrimidine-2,4-diamine 2,5-dimethyl-4-nitro-N'-[2-(4-phenylphenyl)ethanimidoyl]benzenecarboximidamide 5-chloro-4-[2-(1-methylpyrrolidin-3-yl)ethoxy]pyridine-2-carboxylic acid 2-(7-fluoro-3,4-dihydroisoquinolin-6-yl)-N,N'-dimethylacetamide 4-[[2,5-dimethoxy-1-(4-phenylbutyl)indol-3-yl]methylidene]cyclohexa-1,5-diene-1-carboxylic acid 2-fluoro-4,5-dimethoxybenzenethiol 2-[[3,5-difluoro-4-(trifluoromethyl)phenyl]methylamino]-1H-pyrimidine-2,4-diamine 2-[2,6-dimethyl-4-(3-oxomorpholin-4-yl)anilino]-N-(oxan-4-ylsulfonyl)-1-oxoisoquinoline-7-carboxamide 5-[[4-(3-fluoro-2,6-dimethoxyphenyl)-5-iminotetrazole-1-carbonyl]amino]pyrazolo[1,5-a]pyridine-7-carboxylic acid 7-amino-6-fluoro-8-iodo-1-[3-(4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl)cyclobutyl]-4H-quinoxaline-2,3-dione ethane;2-[2-fluoro-4-(6-methylimidazo[1,5-a]pyrazin-3-yl)phenoxy]ethanamine N-methoxy-4-[2-(3,3,5-trimethylpiperidin-1-yl)-5H-pyrrolo[3,2-d]pyrimidine-6-carbonyl]benzamide 2-[3-(methyldisulfanyl)phenyl]acetic acid 2-chloro-4-[3-cyclopentyl-4-(methoxyamino)phenyl]benzenethiol 2-(4-acetylphenyl)-N,N-diethylbutanamide;[7-chloro-1-[1-[(E)-3-hydroxyprop-1-enoxy]ethenylsulfamoyl]indol-4-yl]boronic acid 3-methylsulfanylpropane;6,7,8-trifluoro-2-[2-(4-fluorophenyl)ethynyl]-1-benzothiophene 3-azido-5,7-dichloropyrazolo[4,3-d]pyrimidine 1-(4-fluorophenyl)sulfanyl-3-methoxy-5-[2-(6-methoxypyridin-3-yl)ethynyl]indole N-cyclohexyloxy-2,4-dimethoxybenzamide 6-amino-4-[4-(2,4-dichlorophenoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 2-(benzenesulfonyl)butanoic acid 4-[4,7-bis(ethenyl)-1H-benzimidazole-2-carboximidoyl]aniline 2-cyclopropyl-N'-[(E)-[4-(2,3-dihydro-1H-inden-5-ylmethoxy)phenyl]methylideneamino]acetohydrazide 1-[2,6-dimethyl-4-(morpholine-4-carbonyl)phenyl]-3-(3-methoxy-5,6,7,8-tetrahydroisoquinolin-4-yl)urea (5E)-2-(2,3-dichlorophenyl)imino-5-[(7-fluoronaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one 1-[(3R)-4-amino-2,3-dihydrofuran-5-yl]-2H-quinoline-6-carbonitrile N-(4-chloro-2-methylphenyl)-4-oxopentanamide N-methyl-3-(1,2,3,4-tetrahydronaphthalen-2-yl)propanamide 2,3-diamino-6-chloro-N'-[1-[(3-methylphenyl)methyl]pyrazol-4-yl]pyridine-4-carboximidamide 6-azidooxyisoquinoline 5-(3,4-dichlorophenyl)-3,9-bis[[4-(methylsulfonylcarbamoylamino)phenyl]methoxy]pyrido[2,1-f][1,2,4]triazine-4,6-dione 1-azidooxy-3-cyclohexyloxybenzene 6-N-(3,4,5-trimethoxyphenyl)pyrido[2,1-f][1,2,4]triazine-4,6-diamine 5-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-methylsulfonylamino]naphthalene-2-sulfonic acid 3-benzyl-1H-indole-5-carbonitrile 2-cyclopropylimino-5-[(3,4-diethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 4-[(Z)-(7-chloro-2,3,4,5-tetrahydropyrido[3,2-b][1,4]oxazepin-9-yl)iminomethyl]phenol 1-[4,5-dimethyl-7-(trifluoromethyl)-4H-1,2-benzoxazin-3-ylidene]-N'-ethylpropane-1,3-diamine;dihydrochloride 3-methoxy-4,5,6-trimethylpyridine-2-sulfonamide 3-amino-1H-pyrrole-2,5-disulfonic acid 3-[2-(2-acetylphenyl)-6-chlorophenyl]-4H-1,2,4-oxadiazol-5-one 2-azidooxy-3,4-dichloro-6-[[2,4-bis(trifluoromethyl)phenyl]methoxy]pyridine 2-[(3R)-1-ethylsulfonylpiperidin-3-yl]oxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 3-methyl-4,5-diphenyl-1H-imidazol-2-one 2-[6,6-dimethyl-3-(trifluoromethoxy)cyclohexa-1,4-dien-1-yl]-5-propan-2-yloxybenzoic acid 2-(4,5-dimethyl-N-propylsulfonylanilino)acetamide 1-(2,3-dimethylphenyl)-6-propan-2-ylidene-4-[[4-[4-(trifluoromethoxy)phenoxy]phenyl]methyl]-5H-cyclopenta[d]pyrimidin-7-one 1-[(2R)-3,4-bis(phenylmethoxy)butan-2-yl]-2-diazohydrazine 4-benzyl-7-(1H-imidazole-2-carbonyl)-1,4,10-triazacyclododecane-3,5,8,11-tetrone 1-[(4aS,10bS)-7-ethoxy-4a-methyl-2,3,4,9b-tetrahydroindeno[2,1-b][1]benzofuran-8-yl]butan-1-one 2-[4,7-bis(carboxymethoxy)quinolin-2-yl]acetate 1-(4-aminophenyl)-3,7-diethylnaphthalen-2-ol 6-(5,7-difluoroquinolin-4-yl)oxy-2,3-dihydroindole-1-carboxylic acid [(1R,2S)-4,7-dichloro-2-hydroxy-5-oxocycloheptyl]methylcarbamic acid 2-[[4-(bromomethyl)phenyl]methylsulfanyl]-N-(1,3-thiazol-5-yl)acetamide 3-(2,4-difluorophenyl)-2H-1,2-benzothiazine (7S)-7-[3-bromo-4-[2-(trifluoromethyl)phenoxy]phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine N-[3-(5-chloro-2,4-dihydroxyphenyl)-1H-indazol-6-yl]pyridine-4-carboxamide 2-[(1S,5R)-3-[[4-cyano-3-(trifluoromethyl)phenyl]carbamoyl]-3-azabicyclo[3.1.0]hexan-6-yl]acetic acid 2-(6-chloropyridin-3-yl)-5-(1H-imidazol-5-ylmethylideneamino)pyridin-4-ol 4-[4-[4-(1-cyclobutylideneethyl)piperazine-1-carbonyl]phenyl]benzonitrile 3-[2-oxo-1-(7H-purin-6-yl)pyrrolidin-3-yl]benzenecarbothioamide 4-[2-(2-fluorophenyl)propanoylamino]-1-methylpyrrole-3-carboxylic acid 4-[2-methylpropanoyl-(2,4,6-trimethylphenyl)sulfonylamino]benzoic acid [4-chloro-6,7-bis(ethenyl)quinolin-3-yl]methanol N'-[2-(4-ethylpiperazin-1-yl)ethyl]-N-[7-hydroxy-8-(2,3,5-trifluorophenyl)quinazolin-6-yl]butanediamide N-ethyl-2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-4-phenylpyrimidine-5-carboxamide 7-[(4-fluorophenyl)methyl]-3-methylidene-2,8-dihydro-1H-furo[2,3-e]indole 4-(2,5-dioxo-3-phenylpyrrolidin-1-yl)benzoic acid 1,3-dimethyl-6-(6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepin-2-yl)pyrazolo[3,4-b]pyridine 4-(3,5-dimethyltriazol-4-yl)-N-[2-methoxy-1-methyl-3-[(E)-2-phenylethenyl]cyclohexa-2,4-dien-1-yl]benzamide 7-azido-4,6-dimethyl-1-(2-pyrrolidin-1-ylethyl)imidazo[4,5-c]pyridine (2R,3S)-N-[(5-ethylsulfanylpyridin-2-yl)methyl]-2-(1H-pyrazol-4-yl)oxolan-3-amine (3R,4S)-N,6-dihydroxy-2-oxo-1-[2-[2-phenylethyl(propanoyl)amino]acetyl]-3,4-dihydroquinoline-4-carboxamide 2-(3,4-dichlorophenyl)ethanamine;hydrochloride 4-(4,6-dimethylpyrimidin-2-yl)sulfanylbenzenethiol 4-bromo-5,8-dimethoxychromene-2-thione 1-[(2E,4Z)-hepta-2,4,6-trien-3-yl]sulfanyl-2-phenoxybenzene N-(2,6-difluorophenyl)-N-phenacylhexadecanamide N-[5-tert-butyl-3-[1-cyclohexyl-4,6-dioxo-2-(propanoylamino)pyrimido[5,4-d]pyrimidin-8-yl]-2-methoxyphenyl]-3-fluorobenzenesulfonamide 1-[4-methyl-2-(triazol-2-yl)phenyl]pentan-1-one (3Z,5E)-N-[[2,6-difluoro-4-(trifluoromethoxy)phenyl]methyl]-N-ethyl-5-(5-methylidene-1,3,4-thiadiazol-2-yl)hepta-1,3,5-trien-2-amine N-(4-chloro-5-propanoylpyridin-2-yl)acetamide 4-amino-3,5,6-trichloro-N-phenylpyridine-2-sulfonamide 2-chloro-1-[4-(6,8-dihydro-5H-1,7-naphthyridine-7-carbonyl)piperidin-1-yl]ethanone 3-[4-[2,6-difluoro-N-[(3-nitrophenyl)methyl]anilino]butylamino]propane-1,2-diol 2-[6,8-dimethyl-3-(3,4,5-trifluorophenyl)imidazo[1,2-a]pyrazin-7-yl]piperazine-1-carboxamide;ethane 3-[4-[2,6-diamino-8-(furan-2-yl)purin-9-yl]-3-methoxyphenyl]propanoic acid 7-azidooxy-4,5-difluoro-1H-indole N-[6,7-bis(2-chloroethoxy)quinazolin-4-yl]-1-benzofuran-5-carboxamide N-[2,4-difluoro-3-[(1,2-thiazol-3-ylamino)carbamoyl]phenyl]quinoline-7-carboxamide 2-(3,4-dimethoxyphenyl)-N-(1H-indazole-6-carbonyl)cyclopropane-1-carboxamide 3-cyclopentyl-N,N-diethyl-1-[5-(4-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine-2-carboxamide (3R)-2,5-dihydroxypentanamide;1-[(Z)-5-iminopent-1-enyl]-7-methoxy-6-propanoylquinolin-4-one ethane;1,3-dimethyl-6-(4-methylpiperazin-1-yl)pyrazolo[3,4-b]pyridine N-[(Z)-1,3-diaminoprop-2-enylidene]-2-[4-(trifluoromethoxy)phenyl]acetamide 2-[3,4-di(cycloheptyl)phenyl]pentanedioate (3R,4S)-N-[2-amino-5-(4-fluorophenyl)pyrimidin-1-ium-4-yl]-2-methylpiperidine-4-carboxamide (3S,6R)-2-amino-6-[4-(benzylamino)phenyl]oxane-3,4-diol;N-[(1R)-2-hydroxy-1-phenylethyl]acetamide 4-(methylideneamino)-6-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,7,9,11-pentaen-4-yl)naphthalene-2-carboxylic acid 3-[2-bromo-4-(2-hydroxypropan-2-yl)phenoxy]-N,1,7-trimethylpyrrolo[3,2-c]pyridine-2-carboxamide N'-hydroxy-3-[(1-methylpyrrolidin-2-yl)methoxy]pyridine-4-carboximidamide 1-[(3S)-3-(cyclohexen-1-ylmethoxy)pyrrolidin-1-yl]-2-naphthalen-1-ylethanone 1-methyl-4-[3-(7,9,11-trimethyldodeca-6,8,10-trienoxy)phenyl]piperazine 2-chloro-4-(3,5-difluorophenoxy)-6-methylpyrimidine 4-[4-(dimethylamino)benzoyl]-N,3-dimethylpiperazine-1-carboxamide 2-amino-4-ethoxycarbonylbenzoic acid 2-bromo-1-[3-(difluoromethyl)phenyl]pyrrole [2-(2,5-difluorophenyl)pyrrolidin-1-yl]-[6-methoxy-4-[2-[1-methanimidoyl-3-(oxetan-3-ylamino)cyclobutyl]pyridin-4-yl]oxypyrazolo[1,5-a]pyridin-3-yl]methanone 3-[(2Z,4E)-6-aminohepta-2,4,6-trienyl]-N-[1-[2-chloro-5-fluoro-4-[1-methyl-7-(piperidine-1-carbonylamino)-6,8-dihydro-5H-naphthalen-2-yl]phenyl]ethenyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide 6-amino-N-[4-fluoro-5-(6-morpholin-4-ylpyridine-3-carboximidoyl)-2,3-dihydro-1H-inden-1-yl]pyrazine-2-carboxamide (5R)-N-benzyl-5-methoxy-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-b]pyridine-3-carboxamide 2,6-dichloro-N-(5-methoxy-1H-indazol-3-yl)benzamide N-(3,5-dichlorophenyl)sulfonyl-2-methyl-1,3-thiazole-4-carboxamide (1S)-2,2-difluorocyclopentan-1-amine;N-[1-[5-(4-methylpiperidine-1-carbonyl)pyridin-3-yl]pyrazolo[3,4-c]pyridin-6-yl]acetamide 1,3-difluorobenzene;4,6-dimethyl-2-[(E)-1-phenylprop-1-en-2-yl]pyridine 1-chloro-2-fluorobenzene;(3R)-3,4-dimethylcyclohexan-1-ol;N-[6-(trifluoromethoxy)-5-[4-[(E)-pent-3-enyl]piperazin-1-yl]pyridin-3-yl]formamide N'-(2,3-dihydro-1H-inden-5-ylmethoxy)benzohydrazide 3-[2-amino-5-(4-chlorophenyl)phenyl]cyclopentan-1-ol;ethane 1-(2,4-dichlorophenyl)-6,7-dimethoxy-4-oxoquinoline-3-carboxylic acid N-[1,3-benzodioxol-5-yl(pyridin-3-yl)methyl]-2-bromopropanamide 3-(4,6-diphenylpyridin-2-yl)-11-azapentacyclo[10.7.0.02,10.04,8.013,18]nonadeca-1(12),2(10),4(8),5,13(18),14,16-heptaene N-[1,3-benzothiazol-6-yl(cyclobutyl)methylidene]hydroxylamine 1-[4-methyl-2,6-di(propan-2-yl)phenyl]imidazole 2-[(2S)-1-[4,5-dimethyl-6-(4-methylpiperidine-1-carbonyl)pyridine-3-carbonyl]pyrrolidin-2-yl]-7-[(2-fluorophenyl)methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one (NZ)-N-[6-[5-[4-[2-(4-propan-2-yloxyphenyl)ethynyl]piperidine-1-carbonyl]pyridin-3-yl]-3H-inden-2-ylidene]hydroxylamine 2-(2-aminopyridin-4-yl)-N-[(3S,6R)-6-[[2-[4-[4-(dimethylcarbamoyl)cyclohexanecarbonyl]piperidin-1-yl]acetyl]amino]oxan-3-yl]-1,3-thiazole-5-carboxamide 3-fluoro-2-(1H-indol-5-yl)benzonitrile 1-(4-benzoylpiperazin-1-yl)-2-[4-fluoro-5-(8-methoxyquinolin-4-yl)oxy-2,3-dihydroindol-1-yl]ethanone 3-cyclohexa-1,5-dien-1-ylprop-2-ynoxybenzene (Z)-3,7-diethyl-8-hydroxynon-5-en-4-one;1-[5-(2,6-dimethoxyphenyl)pyrrolo[2,3-b]pyrazin-1-yl]ethanone;ethane 5-[(1,3-diphenylpyrazol-4-yl)methylidene]-3-(2-methoxyethyl)-2-sulfanylidene-1,3-thiazolidin-4-one 2-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-5-[(R)-phenylsulfinyl]-4H-pyrazol-3-one 6-(2,4-dimethoxyphenyl)imidazo[1,5-b]pyridazine;hydrobromide 2-(3,4-dichlorophenyl)-N'-[(E)-pyridin-2-ylmethylideneamino]ethanimidamide;hydrochloride N-[4-(2,3,4a,5-tetrahydronaphthalene-1-carbonyl)phenyl]ethenesulfonamide 2-[N-(benzenesulfonyl)-4-fluoroanilino]propanoic acid 3-(2,4-difluorophenyl)imino-N'-hydroxybutanimidamide N-(cyclopropylmethyl)-6-[4-(2-phenylethoxy)piperidin-1-yl]pyrimidine-4-carboxamide;2,2,2-trifluoroacetic acid N-[5-(difluoromethyl)-1H-pyrazol-4-yl]-2-methoxyquinoline-3-carboxamide 4-[2,6-dimethyl-5-(4-oxospiro[3H-chromene-2,1'-cyclopentane]-7-carbonyl)phenyl]imino-N'-hydrazinylidenebut-2-enimidamide 5-[4-(4,5-diphenyl-1H-imidazol-2-yl)naphthalen-1-yl]-3H-oxadiazole 2-chloro-5-(3,4-dimethylpiperidine-1-carbonyl)oxybenzamide 3-cyclopropyl-2-[(1-methoxy-3H-pyrrolo[2,3-b]pyridin-6-yl)amino]benzamide 3-[2-(4,5-dihydro-1H-imidazol-2-ylmethyl)-6,7,8,9-tetrahydropyrido[2,3-b]indol-7-yl]benzoic acid 5-(4-chlorophenyl)-N-methylspiro[1,3-dihydropyrrole-2,4'-pyridine]-7'-carboxamide 2-[(4-methyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]acetic acid 2-[[(Z)-3-amino-1-hydroxypropan-2-yl]amino]-N'-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-ylmethyl)ethane-1,2-diamine N-[3-(aminomethyl)-5-fluorophenyl]-3-methylbutanamide (3Z)-2,3-dimethylidene-6,7-dihydro-5H-cyclopenta[c]pyridazine;ethane 1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)pyrrolidine-3-carbonitrile 7-chlorospiro[1H-3,1-benzoxazine-4,4'-piperidine] 1-[(2S)-3,4-dimethylpentan-2-yl]-3-fluorobenzene 1-(3,5-dimethyl-4H-pyrazol-1-yl)-2-(2-pyrrolidin-2-yl-3H-benzimidazol-5-yl)propan-2-ol (Z)-3-(2-fluorophenyl)-1,1-dioxo-5-[4-(1,3-thiazol-5-ylmethoxy)phenyl]pent-4-en-2-one 2-[(3R)-1-[6-[2,4-difluoro-N-methyl-5-(trifluoromethoxy)anilino]pyridine-3-carbonyl]pyrrolidin-3-yl]acetamide N-[1-(2,6-difluorophenyl)cyclopropyl]-3-[(4-methoxyanilino)sulfamoyl]benzamide 6-(2,5-dimethylthiophene-3-carbonyl)-N'-hydroxypyridine-2-carboximidamide 5-(2,3-dichlorophenyl)-4-methyl-1H-pyrimidin-6-one 4-[3-azido-1-(3,5-dimethoxyphenyl)propyl]-2H-triazole 4-[2-(3,5-dimethylphenyl)ethynyl]pyridine 4-(aminomethyl)-N-[1-(2,5-dihydroxyphenyl)ethylideneamino]benzenesulfonamide N-[4-chloro-3-(6,7-dihydro-1H-benzimidazole-2-carboximidoyl)phenyl]-1-methylpyrazole-4-carboxamide 2-[4-(3,5-dichlorophenoxy)phenyl]sulfonylphenol ethane;2-methylpropyl-[3-phenylmethoxy-5-(trifluoromethoxy)pentyl]phosphane 4-amino-6-[(3-bromo-5-ethoxy-2,4-dihydroxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-[(3-chlorophenyl)methyl]-N,N-diethylaniline;4-(1H-indol-5-yloxy)-6-methoxyquinazolin-7-amine 2-(4-ethylphenoxy)carbonylpropanoic acid 2-[4-(2-methylbenzotriazol-5-yl)phenoxy]acetic acid 1-(2,4-dichlorophenyl)-2-imidazol-1-ylbutan-1-one N-(1,5-dimethylpyrazol-3-yl)-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]acetamide 2-(4-tert-butylphenyl)-6-(5,5,8,8-tetramethyl-6,7-dihydronaphthalene-2-carbonyl)benzaldehyde 3-(5,8-dihydronaphthalen-2-ylsulfanyl)-N'-[ethyl(methyl)amino]propanehydrazide 2-(6-hydroxyhexyl)terephthalic acid 5-hydroxy-N-[(1R)-3,4,7-trihydroxy-6-phenylmethoxy-2,3-dihydroinden-1-ylidene]pentane-1-sulfonamide 4-hydroxy-N-[(E)-4-iminopentanoyl]benzamide (2S)-1,3-dimethyl-N-[5-methyl-4-[(1Z,3E)-penta-1,3-dienyl]-6-oxo-1H-pyrimidin-2-yl]pyrrolidine-2-carboxamide 1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl)cyclohexane-1-sulfonamide N-(4-bromophenyl)sulfonyl-6,7-dichloroquinoline-3-carboxamide 2-[2-(1,3-dioxolan-4-yl)ethoxy]-6-methoxy-5-phenylpyridine 5-amino-1-[[4-(2-oxopiperidine-1-carbonyl)phenyl]methyl]pyrazole-3-carbonitrile 2-[4-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)phenyl]-N-hydroxyacetamide 6-[(2,4-difluorophenyl)methyl]-1-hydroxycyclohepta-2,4-dien-1-ol 4-[(2E,4Z)-hepta-2,4-dien-3-yl]-N-phenylaniline 2-cyclopropyl-N-[6,7-dimethoxy-4-(4-methylpiperazin-1-yl)quinazolin-2-yl]thieno[3,2-d]pyrimidin-4-amine N-[(2S)-4-methyl-1-oxo-1-[3-(trifluoromethyl)anilino]pentan-2-yl]thiophene-2-carboxamide 4-N,6-N-dimethyl-4-N-(4-methylcyclohexa-1,5-dien-1-yl)-2-[3-(2-pyrrolidin-1-ylethoxy)phenyl]pyrimidine-4,6-diamine 6-(3,4-dimethylphenyl)-2-[2-(pyridine-2-carbonylamino)ethyl]quinoline-4-carboxylic acid;trihydrochloride 1-[4-(2,4,6-trimethylphenyl)pyrimidin-2-yl]piperidine-3-carboxylic acid 7-(2,6-dimethoxyphenyl)-1-[4-(1-piperidin-1-ylpentan-3-ylamino)cyclohexyl]pyrido[2,3-d]pyrimidine-2,4-dione 1-[2,6-dimethyl-3-(2-methylprop-2-enoxy)phenyl]ethanone N'-[3-chloro-4-[3-(dimethylamino)pyrrolidine-1-carbonyl]phenyl]-5-oxopentanimidamide 2-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]aniline N-[(Z)-1H-benzimidazol-2-ylmethylideneamino]-1,3-benzothiazol-2-amine 4-methylsulfanyl-2-(trifluoromethyl)pyridine (2R)-2-[(4-chlorophenyl)methoxy]piperidine N-[4-(3,5-ditert-butylphenyl)cyclohexen-1-yl]methanimine 1-N,2-N-dimethyl-4-(3-quinolin-6-ylpropyl)pentane-1,2-diamine 5-amino-6-[2,3-dihydroindole-1-carbonyl-(2-ethoxynaphthalen-1-yl)amino]-N-methylidenepyridine-3-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]-4-methoxy-2,6-dinitrobenzene 2-[(3,4,5-trimethoxyphenyl)methylidene]butanedinitrile (7R,9aS)-7-[4-(2,5-dioxopyrrolidin-1-yl)phenyl]-6-methoxy-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazine-2-carboxylic acid 2-[2-(4,6-dihydroxypyridin-1-ium-3-yl)oxyethoxy]acetic acid 4-[1,3-benzodioxol-5-yl(hydroxy)methyl]benzonitrile 3-(3,5-dimethoxyphenyl)-3-[2-fluoro-4-[2-(5,6,7-trifluoronaphthalen-2-yl)ethynyl]phenyl]propanoic acid 2-[5-azido-3-(4,6-difluoropyridin-3-yl)indol-1-yl]ethanol 2-(4-cyclohexylphenyl)-N,N-dimethylcyclopropan-1-amine 2-[3-chloro-4-(1,2,3,5,6,7-hexahydropyrrolizin-8-ylmethoxy)phenyl]acetate [3-(methoxymethyl)pyrrolidin-1-yl]-pyridin-4-ylmethanone N-[(Z)-(5-bromo-2-hydroxy-3-methoxyphenyl)methylideneamino]-2-[2,6-dichloro-4-nitro-N-(2-phenylethyl)anilino]acetamide 4-methylsulfanyl-3,6,8,9-tetrahydropyrimido[4,5-g]quinoline-7-thione 2-(1H-benzimidazol-2-yl)-3-[4-hydroxy-3,5-di(propan-2-yl)phenyl]-3-oxopropanoic acid N-(2,4-dinitrophenyl)-N-ethylsulfonylhexadecanamide 2-(3,6-difluorocarbazol-9-yl)acetic acid (NE)-N-[1'-[3-[4-[(Z)-[2-(4-chlorophenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]phenoxy]propyl]spiro[3H-chromene-2,4'-piperidine]-4-ylidene]hydroxylamine 6-[2-(4-chlorophenyl)sulfanylpropyl]-1,3,5-triazine-2,4-diamine 2-fluoro-N,N-dimethyl-4-[2-[4-(1,3-thiazole-4-carbonyl)piperazin-1-yl]ethoxy]benzamide 1,2-diamino-4-[3-methoxy-4-(trifluoromethyl)phenyl]-6-oxopyridine-3,5-dicarbonitrile 5-(4-benzylpiperazine-1-carbonyl)pyridine-2-carbonitrile 4-[5,6-dioxo-1-(3,4,5-trifluorophenyl)-7H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-1-carboxylic acid (5R)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-methyl-1,3-thiazolidin-4-one 3-(azidomethyl)-2,4-bis(difluoromethoxy)phenol 2-(4-chlorophenyl)-1-[4-(6-fluoroquinolin-4-yl)cyclohexa-1,3-dien-5-yn-1-yl]ethanone 1-[4-(difluoromethyl)phenyl]-3-methoxypyrazolo[4,3-b]pyridine 2-[6,7-dimethoxy-3-(4-morpholin-4-ylphenyl)quinoxalin-2-yl]guanidine 1-benzyl-5-hydroxyspiro[3H-indole-2,4'-piperidine] 2-[[5-(ethoxymethyl)-4-(4-fluorophenyl)-1,3-thiazol-2-yl]amino]benzenesulfinic acid 2-[4-fluoro-5,6-bis(4-methylphenyl)pyrimidin-2-yl]pyridine-3-carbonitrile 1-(5,5,5-trifluoro-4,4-dimethylpentanoyl)-2,3,3a,4,6,7,8,9,9a-octahydrobenzo[g]indole-8a-carboxylic acid 2-[N-(carboxymethyl)-4,5-dimethoxyanilino]acetic acid 4-methyl-2-(4-methylidenehept-6-enyl)phenol 4-[5-[4-[(3R)-1-methylpyrrolidin-3-yl]oxyphenyl]-2,6-dihydropyrrolo[3,4-c]pyrrole-1-carbonyl]benzonitrile 2-methyl-3,3a,4,5-tetrahydropyrrolo[1,2-a]quinoline-1,8b-dione N'-hydroxy-3-methyl-6-[methyl(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)amino]pyridazine-4-carboximidamide [4-methoxy-1-(2-methyl-6,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carbonyl)pyrrolidin-2-yl]-morpholin-4-ylmethanone 4-[2-(3,5-difluorophenyl)-1-[5-(6-ethylquinolin-8-yl)pyridin-2-yl]ethenyl]morpholine 1,2-dimethyl-4-(3,7,11-trithiatricyclo[6.3.0.02,6]undeca-1(8),2(6),4,9-tetraen-4-yloxy)piperidine;ethane [3-methyl-2-[[4-phenyl-4-(trifluoromethyl)cyclohexa-1,5-dien-1-yl]amino]butanoyl]azanide 3-chloro-5,6-dimethylimidazo[2,1-b][1,3]thiazole;(Z)-5-[5-(chloroamino)-2,4-bis(phenylmethoxy)phenyl]pent-4-enal 5-[4-fluoro-3-[7-(furan-3-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-amine 2-[[1-(azetidine-3-carbonyl)piperidin-4-yl]methoxy]benzonitrile 4-[3,5-dimethyl-2-(2H-pyrrol-5-yl)phenyl]butanoic acid 4-[2-(trifluoromethoxy)phenyl]benzenesulfonamide 1-[3-(4-chlorophenyl)-5,6,7,8-tetrahydroimidazo[2,1-b]purin-9-yl]-4-methoxypentan-2-one 1-[3-(4-cyanophenoxy)phenyl]ethylcarbamic acid N-(3-bromophenyl)-2,4-dichloroquinazoline-7-sulfonamide N-[(4,5-difluoro-2-phosphanylphenyl)methyl]pyridine-3-carboxamide 2,5-dibromo-4-phenylmethoxyquinoline 5-[1-azido-2-(3,4-difluorophenyl)ethyl]pyridine 5-bromo-2-(4,7-difluoro-1H-indol-3-yl)-6,7-dimethoxy-1-[(3R)-oxolan-3-yl]benzimidazole 3-[(2E)-4,5-dimethoxyhexa-2,4-dien-2-yl]-N-methylpyridine-2-carboxamide 1-azidooxynaphthalene (1-azidopiperidin-2-yl)-phenylmethanone ethane;[1-(2-methoxy-4-methylphenyl)-2-(oxiran-2-yl)butan-2-yl]hydrazine 6-(4-nitrophenoxy)-N-[2-(oxan-3-yloxy)ethyl]pyrimidine-4-carboxamide 5-[(6R)-7-bromo-2,3,4a,5,6,8,9,10,11,11a-decahydro-1H-pyrido[3,4-b]acridin-10-yl]pyrimidine-2,4-diamine 2-(1H-benzimidazol-2-yl)-3,4-dichlorophenol 2-amino-N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]acetamide [3-fluoro-4-(2H-quinolin-1-yl)phenoxy]boronic acid 4-(azidomethyl)-2,6-diphenylpyridine 6,8-dihydroxy-7H-naphthalene-1,3,5-tricarboxylic acid 2-[3-[[1-(cyclohexylmethyl)piperidin-4-ylidene]methoxy]phenyl]acetic acid (2Z,5R)-5-benzyl-2-[(Z)-(3-ethoxyphenyl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one 7-ethoxy-6,8-difluoro-3-(4-hexylphenyl)-1,2-dihydronaphthalene 4-[3-(cyclopropylmethoxy)phenyl]-6-methylpyridine-2-carboxamide 5-ethoxycarbonyl-6,7,8-trifluoronaphthalene-2-sulfonic acid 2-(cyclopropylmethoxy)-N'-(4,5,6,7-tetrahydrothieno[3,2-d]pyrimidin-2-yl)benzenecarboximidamide [4-(2,3-dichlorophenyl)piperazin-1-yl]-(6-methoxypyridin-2-yl)methanone 3-chloro-2,6-difluoro-N-(1-methylpyrazol-4-yl)benzamide N-[4-(6,11-dihydrobenzo[c][1]benzazocin-5-yl)butyl]cyclopropanecarboxamide 2-(3,4-dichlorophenyl)-N'-hydroxyethanimidamide 3-[(2,4-dichloropyrimidin-5-yl)-ethylamino]propan-1-ol 2-[(E)-1,3-diamino-3-oxoprop-1-en-2-yl]-N-(4-propan-2-ylphenyl)-1H-benzimidazole-4-carboxamide 1-(3,4-difluorophenyl)-2-[[2-(6-methoxynaphthalen-2-yl)acetyl]amino]cyclopropane-1-carboxamide 2-[2,4-dimethyl-5-(6-phenylpyridin-3-yl)-1H-pyrrol-3-yl]acetamide 5-[6-[(3S)-3-methylpyrrolidine-1-carbonyl]pyridin-2-yl]oxynaphthalene-1-carboxylic acid 2-azido-N,N-dimethylaniline 4-[[(3S)-2,2-difluoro-3-hydroxy-4-methylpentanoyl]amino]naphthalene-1-carboxamide [2-(4,6-dimethoxypyrimidin-2-yl)-1,3,3a,4,5,7,8,8a-octahydropyrrolo[3,4-d]azepin-6-yl]-quinoxalin-6-ylmethanone;formic acid 1-[[6-(3,5-dimethoxyphenyl)pyrimidin-4-yl]methylamino]-2-(dimethylsulfamoyl)propan-2-olate (E)-2-[(Z)-1,3-bis(4-hydroxyphenyl)prop-2-enylideneamino]-N,4-diethylpent-2-enamide 6-bromo-2,3-bis(ethenyl)naphthalene-1,4-dione 3-[(4R)-5-[1-hydroxyethyl(2,2,2-trifluoroethyl)amino]-1-propanoylpiperidine-4-carbonyl]chromen-2-one N-(2,4-dichloropyrimidin-5-yl)-N-naphthalen-1-ylacetamide 6-bromospiro[2H-1,4-benzodioxine-3,5'-imidazolidine]-2',4'-dione N-[1,3-bis(2,4,6-trimethylphenyl)imidazolidin-2-ylidene]nitramide N-[1-(3,5-difluorobenzoyl)azetidin-3-yl]-2-oxo-1H-pyridine-4-carboxamide (1R,2S)-N-[2-(4-methylpiperazine-1-carbonyl)phenyl]cyclopentane-1-carboxamide 1-(6-tert-butylpyridazin-3-yl)piperidin-4-ol 3-(dimethylamino)-2-hydroxy-N,N-bis(naphthalen-1-ylmethyl)propanamide 4-[(8R,9S)-13-hydroxy-12-iodo-2-tricyclo[7.3.1.05,13]trideca-1,5,7,9(13)-tetraenyl]benzonitrile 1-[5,6-difluoro-2-[4-(trifluoromethyl)phenyl]benzimidazol-1-yl]propan-2-one;pyrrolidine [2-chloro-6-(cyclopropylmethylamino)pyridine-3-carbonyl]urea [5-(4-chlorophenyl)sulfanyl-1H-pyrazol-3-yl]methanediol 2-(4-acetyloxyphenoxy)benzoic acid N-[(2S)-4-aminosulfanyl-1,1,1-trifluorobutan-2-yl]-8-chloronaphthalene-1-carboxamide 7-[(2R,4S)-2-(3,5-difluorophenyl)-4-fluoropyrrolidin-1-yl]-5-methoxypyrazolo[1,5-a]pyrimidine 2-[2-[4-[bis(2,2,2-trifluoroethyl)amino]phenyl]imidazol-1-yl]-N-cycloheptylacetamide 2-chloro-1-[3-(dimethylamino)phenyl]ethanone 7-(2-butylheptoxy)-3,4-dihydro-1H-quinazolin-2-one 3-(1,5-dimethylcyclohexyl)benzonitrile [3-(2,5-diphenylpyridine-4-carbonyl)oxyphenyl]azanium 4-(3,4,5-trimethoxyphenyl)-6-[2,3,5,6-tetrafluoro-4-(1,1,1-trifluoropropan-2-ylsulfanylamino)phenoxy]pyrimidine-5-carbonitrile 5-(2,4-difluorophenyl)sulfanyl-N'-hydroxypyrazine-2-carboximidamide [4-[(2,4-dimethoxypyrimidin-5-yl)-hydroxymethyl]-3-iodopyridin-2-yl]carbamic acid 2-[(2Z)-4-oxo-2-(2-phenylpropylidenehydrazinylidene)-1,3-thiazolidin-5-yl]acetic acid N-[[1-(3,5-dimethylcyclohexyl)triazol-4-yl]methyl]-2,8-diazaspiro[4.5]decane-4-carboxamide;hydrochloride (5S)-1,3-dimethyl-7-[4-methyl-3-(5-methylidenepyrrolo[2,3-d]pyrimidine-6-carbonyl)phenyl]-8,9-dihydro-6H-quinolizin-5-ium-4-one 1-chloro-4-methylbenzene;N-(3,5-dimethoxyphenyl)-3,7-diethynyl-1,2,4,5-tetrahydro-3-benzazepine-6-carboxamide (5Z)-2-(4,5-dimethyl-1H-imidazol-2-yl)imino-5-[(3-hydroxy-4,6-dimethylpyridin-2-yl)methylidene]-1,3-thiazolidin-4-one 5-[2-(1,3-benzodioxol-5-yl)ethynyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 2-[(3R,4S)-1-[1-(cyclopropylmethyl)pyrazole-4-carbonyl]-4-hydroxypyrrolidin-3-yl]-N-methylacetamide 2-[3-(6-oxocyclohexa-1,4-dien-1-yl)prop-2-ynoxy]ethoxy-[4-[2-(sulfamoylamino)ethylcarbamoyl]phenyl]phosphinic acid [3-methylsulfanyl-6-(2,4,5-trifluorophenyl)imidazo[1,2-b]pyridazin-8-yl]hydrazine 4-[(5R,9S)-7-chloro-2-(oxetan-3-yloxymethyl)-8-oxo-3,4,6,11b-tetrahydro-1H-pyrazino[2,1-a]isoindol-9-yl]benzonitrile N-[2-[cyclohexyl(methoxy)amino]phenyl]sulfonylbenzamide N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-4,4,4-trifluorobutanamide 4-(3,5-dimethylphenyl)-2,3-dihydro-1H-indene 4-[5-cyclohexyl-1,2-dimethyl-3-(2-oxopropyl)pyrrole-2-carbonyl]piperazine-1-carbonitrile 2-[(7R,9aS)-8-[1-(cyclopropanecarbonylamino)ethenyl]-4-oxo-3-phenyl-5,6,7,9a-tetrahydro-[1,3]thiazolo[5,4-b]quinolin-2-yl]acetic acid [2-chloro-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonylamino)phenyl]boronic acid 1-[5-methyl-2-(triazol-1-yl)phenyl]propan-2-one (2-azido-3,5-dibutylphenyl)methanol 4-methyl-N-[2-(5-methylsulfanyl-1,3,4-oxadiazol-2-yl)phenyl]benzenesulfonamide 3-azido-5-(2-methoxypyrimidin-4-yl)benzonitrile N-(3,4-difluorophenyl)-3-(5-methylthiophen-2-yl)quinoxaline-6-carboxamide 1-bromo-6,8-dimethylbenzo[b]carbazole (1R,2R)-N-[8-amino-6-(4-methylpyridin-3-yl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 2-[azidooxy-(4-ethoxyphenyl)methyl]naphthalene 2-[6-(2,3-dichlorophenyl)sulfonyl-4-oxopyrido[1,2-a]pyrimidin-9-yl]acetic acid 4-(aminomethyl)-2-[(3,5-difluorophenyl)methylsulfanyl]-1H-pyrimidin-6-one 2-(4,6-dimethyl-1H-benzimidazol-2-yl)naphthalen-1-ol 2-[(3R,4R)-1-benzylpiperidin-3-yl]-6-methoxy-1H-benzimidazole 4-[(6E)-3,7-bis(benzenesulfonylmethyl)deca-1,6-dienyl]-N,N-dipropylaniline 3-[2,4-bis(prop-1-en-2-yl)phenyl]-1-benzoxepine 3-[4-(2,6-dimethylanilino)piperidine-1-carbonyl]pyridine-2-carbonitrile 3-methyl-1-[4-[2-[(2S)-6-(5-propan-2-ylpyridazin-3-yl)oxyspiro[3.3]heptan-2-yl]oxyethoxy]pyridine-2-carbonyl]piperidine-4-carboxylic acid (E)-N,6-dimethyl-N-[(3Z)-2-methylidenehexa-3,5-dienyl]-4-pyridin-2-yloct-8-enamide 5-chloro-4-[6-fluoro-2-(2-methoxyethylsulfanyl)quinazolin-7-yl]pyridine-3-carbonitrile 4-N-[(3S,5R)-1-butanoyl-5-methylpiperidin-3-yl]-2-N-methylidene-6-(oxan-4-yloxy)pyridine-2,4-dicarboxamide 4-[5-fluoro-6-(2,2,2-trifluoroethoxy)pyridine-3-carbonyl]-1,4-oxazepane-6-carboxamide 5-(diethylamino)-2,4-dinitrobenzoic acid N-[1-(2,5-dichlorophenyl)piperidin-3-yl]-5-(4-methylpiperazine-1-carbonyl)thiophene-2-sulfonamide 5-ethyl-4,10-dihydrothieno[3,2-c][1]benzazepine (4R)-N'-[(3S)-3,4-dihydro-2H-chromene-3-carbonyl]-5-methyl-1-(pyridine-2-carbonyl)azepane-4-carbohydrazide (1R,3S)-N'-[4-chloro-3-[(4-methylphenyl)carbamoyl]phenyl]-2,2-difluorocyclopropane-1-carbohydrazide 2-amino-4-(5-bromo-3,6-dihydro-2H-pyridin-1-yl)benzoic acid N-[(4-azidophenyl)methyl]oxolane-3-carboxamide 2-[5-chloro-4-(trifluoromethyl)pyridin-3-yl]-1H-indole (3R)-7-fluoro-9,10-dimethyl-3-[2-(3-phenylpropanoylamino)ethyl]-1,4,7,12-tetrazatricyclo[6.3.0.02,5]undeca-9,11-diene-12-carboxamide N-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-5-pyrrolidin-2-ylthiophene-2-sulfonamide;hydrochloride 1-chloro-3,6,8-trimethylpyrene 6-(2,5-difluorophenyl)-3-[4-(6H-quinolin-8-id-7-yloxy)butyl]imidazo[1,2-b]pyridazine;uranium(2+) 1-[4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)-1,3-oxazol-5-yl]butan-1-one 1-[2-(4-fluorophenyl)ethylamino]-3-hexan-2-ylthiourea (2R)-1-[[5-[3-chloro-4-[(3R)-3-methylmorpholin-4-yl]phenyl]furan-2-carbonyl]amino]cyclopentane-1-carboxylic acid 2-[3-chloro-4,5-dimethoxy-N-methyl-6-(pyrimidin-5-ylamino)pyridin-2-yl]-1H-indole-6-carbonitrile 2,6-dichloro-4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoylamino]benzoic acid 1-[4-azidooxy-3,5-di(propan-2-yl)phenyl]ethane-1,1-disulfonic acid 2-[1-(3-chlorophenyl)propan-2-yl]-1,5-dimethylpiperazine 5-hydroxy-4-methoxycarbonyl-7,8-dihydronaphthalene-2,3-dicarboxylic acid N-[3,4-difluoro-2-(5-fluoropyridin-3-yl)phenyl]hydroxylamine;formamide (E)-3-[4-[(2,5-dimethylphenyl)methoxy]-3-iodophenyl]-2-sulfanylprop-2-enoic acid 1-[4-azido-3,5-di(propan-2-yl)phenyl]ethenesulfonic acid 7-(2,3-dihydro-1H-inden-5-yl)-3H-pyrrolo[2,3-d]pyrimidin-4-one;dihydrochloride 1-(3-chlorophenyl)sulfinylpyrrolidine (2S,3S)-4-[(1R)-1-azido-2-phenylethyl]-2,3-dimethoxybutane-2,4-diol (2S)-3-methyl-2-[(6-phenylpyridine-3-carbonyl)amino]butanoic acid (4-azidooxyphenyl)-cyclopentylmethanone 1-N-[1-(2,6-dichlorophenyl)ethyl]naphthalene-1,5-disulfonamide N-[3-(2-methylpropoxy)propyl]-4-oxopyrido[1,2-a]pyrimidine-2-carboxamide N-(6-methylpyridin-2-yl)quinoline-3-carboxamide 3-[4-[3-methylbutoxy(phenyl)phosphoryl]oxy-2,3-dihydroindol-1-yl]propanoic acid 5-[(6R)-6-[4,4-difluoro-2-(trifluoromethyl)butanoyl]-6-hydroxy-3-azabicyclo[4.1.0]heptan-3-yl]quinoxaline-8-carboxamide 5-(5-bromopyridin-3-yl)pentanoic acid 2-chloro-3-[[3,5-difluoro-4-(pyridine-2-carbonylamino)benzoyl]amino]-5-methylbenzoate (2R)-N-[2-azido-1-(3,5-difluorophenyl)ethyl]pyrrolidine-2-carboxamide 4-fluoro-2-[4-(5,6,7,8-tetrahydroisoquinolin-1-ylmethoxy)phenyl]benzenethiol 2-[(6R)-6-methyl-3-bicyclo[4.1.0]hepta-1,3,5-trienyl]-4H-isoquinoline-1,3-dione 4-[[2-chloro-6-(methoxymethyl)benzoyl]amino]oxane-3-carboxylic acid [(3S,5R)-4-hydroxy-1-oxa-9-azaspiro[4.6]undecan-9-yl]-(2-methylpyrazol-3-yl)methanone;2,2,2-trifluoroacetic acid 2-[3-(aminomethyl)piperidin-1-yl]-4,5-difluoro-9H-pyrimido[5,4-b]indole-8-carboxylic acid;hydrochloride 3-(3,4-dimethoxyphenyl)-2H-benzo[g]chromene 7-[4-(2,4,6-trimethylphenyl)-1,3-thiazol-2-yl]quinazoline N-cyclopentyl-2-[5-[3-(4,6-dichloropyridin-3-yl)propyl]tetrazol-1-ium-2-yl]acetamide [4-(1,1-difluoroethyl)phenyl]-dimethylborane N-methyl-3-[5-[4-(2,2,6,6-tetramethylpiperidin-4-yl)oxyanilino]pyridin-2-yl]benzamide 2-[3-[4-(diaminomethylideneamino)butanoyl-propylcarbamothioyl]-2,5-dihydroindol-1-yl]acetic acid N'-(2,2-dimethylpropoxy)-3,4-difluoro-N'-hydroxybenzenecarboximidamide 1-azidooxy-3,5-dichloro-2-ethenylbenzene 2-(1,3-benzodioxol-5-yl)-N'-[3,4-bis(phenylmethoxy)benzoyl]propanehydrazide N-[(3,4-dichlorophenyl)methyl]-2-[1-[2-(2-hydroxyethoxy)ethylamino]propan-2-ylideneamino]acetamide 2-(7-cyclohexyl-8-ethenylsulfanylimidazo[1,5-a]pyrazin-3-yl)acetamide 3-amino-6-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-N-[1-(propanoylamino)cyclohexyl]-5-(1H-pyrrole-2-carboximidoyl)pyrazine-2-carboxamide 4-[2-[(5S)-3-[(E,3R)-5-(1H-indazol-6-ylamino)-2-oxopent-4-enoyl]-2-oxo-1,3-oxazolidin-5-yl]ethynyl]benzoic acid 3-[7-(6-methoxypyridin-3-yl)furo[3,2-c]pyridin-2-yl]-1-phenylpentan-1-one 2-ethyl-3,4,5-tris(3,4,5-trimethoxyphenyl)phenol 1-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]piperidine-4-carbonitrile (4-chlorophenyl)sulfonylbenzene 4-[2-azidoethyl(methyl)amino]-1H-pyrimidin-6-one 2-bromo-5-[2,6-di(propan-2-yl)phenyl]-4-methoxyaniline 2,2-dimethylpropanoic acid;ethane;5-[5-[3-(morpholin-4-ylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-2-yl]-2-(oxolan-2-yloxy)benzonitrile 2-methylsulfonyl-4-(trifluoromethoxy)aniline 3-[(1,4-dioxonaphthalen-2-yl)amino]benzoic acid 3-[(1R)-1-(3-azidoazetidin-1-yl)butoxy]pyridine 6-chloro-4,8-dimethyl-3H-pteridine-2,5-dione 3-methyl-4-[2-(trifluoromethoxy)phenyl]sulfonylpiperazine-1-carboxylic acid 4-[(6-methoxypyridin-3-yl)methyl]-2-phenylpyrimidine (Z)-N'-[2,3-bis(ethenyl)naphthalen-1-yl]but-2-enediamide 5-[3-(2,4-difluorophenyl)cyclobutyl]-1H-pyrazole (3-methyl-2,6,7,8-tetrahydroquinolin-1-yl)-[5-(pyridin-2-ylamino)pyrazin-2-yl]methanone 2,3-bis(3-methylcyclopentyl)-5-propan-2-yloxyphenol N-[(2S)-1,1-bis(4-chlorophenyl)-3-oxobutan-2-yl]formamide 6-fluoro-2-(1-methoxypropan-2-yl)-3H-quinazolin-4-one 6-[4-(1,3-diphenylpropoxy)piperidine-1-carbonyl]pyridine-2-carbonitrile 4-azido-1,3-dibromo-5-nitro-2-(trifluoromethyl)benzene [[2-(aminomethyl)-5,6-dihydro-4H-cyclopenta[b]thiophen-3-yl]-[1-(2-fluorophenyl)piperidin-4-yl]oxymethylidene]azanium N-[2,4-bis(2-methylbutan-2-yl)phenyl]-1H-imidazole-5-carboxamide (2S,3R)-1-azido-3-benzylpiperidine N-(5-chloropyridin-2-yl)-3-[ethyl(hexyl)amino]propanamide 5-(3,4-dichlorophenyl)-N-[2-methylsulfanyl-1-[1-[2-oxo-2-[4-(1H-1,2,4-triazol-5-ylamino)anilino]ethyl]cyclopentanecarbonyl]piperidin-4-yl]-1,3,4-oxadiazole-2-carboxamide 2-(4,5,6-trimethylpyrimidin-1-ium-2-yl)sulfanylethanol 1-(3,5-difluorophenyl)sulfonylpiperidine 3-[4-(2-carboxyethenyl)phenyl]propanedioic acid 4-[5-(6,8-dichloronaphthalene-2-carbonyl)oxynaphthalen-1-yl]sulfonylcyclohexane-1-carboxylic acid (1R,3S)-3-[2-methyl-6-[1-methyl-5-oxo-4-(phenylcarbamoylamino)-1,2,4-triazol-3-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid 6-fluoro-1-phenyl-2H-isoquinoline [4-[(3-iodopyridin-2-yl)oxymethyl]piperidin-1-yl]-[3-(methoxymethyl)oxetan-3-yl]methanone 3-(4-azidophenoxy)-2,3-dimethylbutan-2-amine 6-(3,5-dimethylphenyl)-5H-pyrrolo[2,1-a]isoindole 1-(2,4-dimethylphenyl)sulfonyl-2-methylbenzene;ethane 2,6-bis(5-methylfuran-2-carbonyl)cyclohexa-1,3-diene-1-carbonitrile 1-[4-[6-amino-5-[(Z)-methoxyiminomethyl]pyridin-3-yl]phenyl]sulfonylpiperazine-2,6-dione 4-hydroxy-3,5-bis(trifluoromethyl)benzenesulfonate (E)-3-amino-1,2-difluoro-N'-[4-[(E)-2-oxoethoxyiminomethyl]phenyl]but-2-enimidamide 5-amino-3-[2-hydroxy-5-(trifluoromethyl)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile 2-[(3-aminopropylamino)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine 4-[[4-[(5-fluoropyridin-2-yl)amino]-6,8-dihydro-5H-pyrano[3,4-d]pyrimidin-2-yl]amino]benzonitrile 2-[4-[(5-methoxy-1H-indol-3-yl)methyl]piperazin-1-yl]ethanamine 1-(2,5-dimethoxyphenyl)sulfonyl-3-[[4-(2,6-dipyrrolidin-1-ylpyrimidin-4-yl)phenyl]methyl]urea [1-(4-cyclopropylphenyl)pyrazolo[3,4-d]pyrimidin-6-yl]methanol (E)-1-[2,4-bis(phenylmethoxy)phenyl]-3-phenylprop-2-en-1-one 2-[4-(cyclopropanecarbonylamino)butanoylamino]-N-(2,6-dioxopiperidin-3-yl)pyridine-4-carboxamide N-azido-3,5-dimethoxyaniline 3-(1,3-benzothiazol-2-yl)-4H-[1,2]oxazolo[5,4-b]pyridine-5,6-dione 4-(4-fluorophenyl)-2,5-dimethylfuran (3-cyano-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonyl)-methylideneazanium 5-(4,7-dioxo-3H-thieno[3,2-d]pyrimidin-6-yl)pentanoic acid 3-(4,6-dihydrotriazolo[1,5-a][2]benzazepine-5-carbonyl)-5-ethyl-8,9-dimethoxy-2H-imidazo[4,5-c]quinolin-1-one 3-N,4-dimethyl-1-N-[[(2R)-oxolan-2-yl]methyl]benzene-1,3-diamine 2-(2,4-difluorophenyl)-6,7-bis[3-methylbutoxy(propan-2-yl)phosphanyl]-N-(4-propan-2-ylpyridin-2-yl)quinazolin-4-amine 2-[4-[(3,5-difluorophenyl)methyl]piperidin-1-yl]-N-(2,6-dimethoxypyridin-3-yl)acetamide [4-(cyclohexylamino)-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-2-yl]cyanamide 2-[[1-(4,6-dimethoxypyrimidin-5-yl)sulfonylpiperidin-3-yl]methoxy]pyridine 4-(6-ethoxypyridine-3-carbonyl)morpholine-2-carboxylic acid 1-[4-[4-amino-2-(methoxymethyl)pyrrolidin-1-yl]pyrimidin-2-yl]piperidin-3-ol 4-bromo-5-(4-chlorophenyl)-1,3-benzodioxole N'-cyclobutyl-N-phenylpropanediamide;ethene 1-[2-(2,3-dihydro-1H-inden-5-yloxy)ethyl]piperazine;oxalic acid 1-N',2-N',3-N'-tetrabutylcyclopropanedi1,1-dicarboxamide;rhodium(3+);tris(4-fluorophenyl)phosphanium 6,9-difluorobenzo[g]pteridine 1-[2-[4-amino-5-(4-morpholin-4-ylcyclohexa-2,4-dien-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]ethoxy]propan-1-ol 3-(1-aminoethyl)-6-methoxyisochromen-1-one 3-[(1R)-3,3-dimethylbutyl]-6-hydroxy-2H-indazole-5-carboxylic acid 3-[2-(4,4-difluorocyclohexyl)acetyl]-6-(furan-2-yl)-1H-benzimidazol-2-one 4-azidooxy-1,2-dichloro-3-methylsulfanylbenzene [4-(3-chlorophenyl)piperazin-1-yl]-(1,2,6-trimethylindol-5-yl)methanone;hydrochloride N-[2-amino-4-(1H-pyrrole-3-carbonyl)phenyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carboxamide 2-[(3R)-5-azidopyrrolidin-3-yl]oxyquinoxaline 2-[1,4-bis(hydroxymethyl)naphthalen-2-yl]oxyacetic acid 2-(4-tert-butylphenyl)pentanoic acid 7-methyl-6-phenylsulfanyl-2H-1,4-benzoxazin-3-one 3-[(4R)-2,8-dimethyloctoxy]-1-ethylpyridin-1-ium;iodide 2-[(1,3,5-trimethylpyrazole-4-carbonyl)amino]quinoline-4-carboxylic acid 2-azido-4,5,6-trichloropyrimidine 3-(3,4-dimethoxyphenyl)-2H-1,5-benzothiazepine N-(4-chlorophenyl)-N-[1-methyl-2,6-dioxo-3-(2-phenylethylamino)pyrimidin-5-yl]methanimidamide (2-fluorophenyl)methyl-[1-(pyridine-4-carbonyl)pyrrolidin-3-ylidene]azanium 2-[1-(2,3-difluorophenyl)pyrrolidin-3-yl]oxypyrazine 3-[[2,4-bis(phenylmethoxy)-5-propan-2-ylbenzoyl]amino]benzoic acid 2,4-dimethyl-N-[3-(5H-pyrrolo[3,4-b]pyridine-7-carbonylamino)phenyl]pentanimidate [(4S)-4-(aminomethyl)-1,2-oxazol-3-yl]-[(2R)-2-phenylpyrrolidin-1-yl]methanone N-[2-hydroxy-2,5,6,7-tetramethyl-3-(4-propoxyphenyl)chromen-4-ylidene]hydroxylamine 2-[5-(1,1-difluoroethyl)thiophen-2-yl]-7-[4-(dimethylsulfamoyl)anilino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-4-carboxamide N-(6,7-dihydroquinolin-5-yl)-2-fluorobenzamide 5-[1-(2,4-dichlorophenyl)-3-methylbutyl]thiophene-3-carboxylic acid N-[(3S,4R)-1-cyclohexyl-3-(hydroxymethyl)piperidin-4-yl]-2,6-difluoro-3-[[4-methoxy-2-(trifluoromethyl)phenyl]sulfonylamino]benzamide 4-[3,5-bis(trifluoromethyl)phenyl]-N-cyclopenta-2,4-dien-1-ylidenenaphthalene-1-carboxamide N-[(4-azidosulfonylphenyl)methyl]acetamide 2,5-ditert-butyl-N-(3-chloro-1-pyridin-4-ylpyrazol-4-yl)benzenesulfonamide 1-[2,3-bis(4-methylphenyl)naphthalen-1-yl]ethanone 3-[4,6-bis(2,5-dimethoxyphenyl)pyridin-2-yl]-6-N,1-diethylindole-2,6-dicarboxamide N-[(5-aminopyridin-3-yl)methyl]-2,4,6-trifluoro-3-hydroxybenzamide 4-[1-(4-fluorobenzoyl)piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one 2-[4-(2,5-dimethylcyclohexa-1,3-dien-1-yl)phenyl]sulfanylnaphthalene 3-[4,5-bis(hydroxymethyl)furan-2-yl]-2,6-dihydro-1H-[1,3,5]triazino[1,2-a]benzimidazole-9,11-dione 3-[5-(4-chlorocyclohexa-2,4-dien-1-yl)pyrazol-1-yl]-N-[4-[2-hydroxyethoxy(methyl)phosphoryl]phenyl]benzamide 3-[3-(2,2-dimethylpropanoyl)phenyl]-N-(2H-triazol-4-yl)prop-2-enamide N-[4-[(Z)-3-amino-2-iminopropylidene]piperidin-1-yl]sulfonyl-6-chloro-5-fluoropyridine-3-carboxamide 2-(azidosulfanylmethyl)-5-chloropyrimidine 1-[2,4-difluoro-5-[[(3S)-pyrrolidin-3-yl]sulfamoyl]phenyl]indole-7-carboxylic acid 3-[4-[(Z)-N'-[amino(methyl)amino]carbamimidoyl]phenyl]propanamide 5-methylsulfonyl-1,3-benzothiazol-2-amine 4-[4-(4-methoxyphenyl)-2,3,6,7-tetrahydroazepine-1-carbonyl]piperazin-2-one 7-(2,3-dihydroxypropoxy)chromen-4-one N-[1-(2,4-dimethylphenyl)ethenyl]-2,6-difluoroaniline 1-(1H-imidazol-5-ylmethyl)-2-[2-(trifluoromethoxy)phenyl]piperazine N-[2-(3-ethylpyridin-2-yl)-1,3,4-thiadiazol-5-yl]-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine-2-carboxamide 2-[(6S)-6,7-dihydro-5H-1,3-benzothiazol-6-yl]-1-[4-[3-methoxy-4-[4-(trifluoromethyl)phenyl]anilino]piperidin-1-yl]ethanone (5R)-2-benzylsulfanyl-N,N-dibutyl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide N-(3,4-dimethylphenyl)-5-methyl-2-(4-piperidin-1-ylsulfonylanilino)pyrimidine-4-carboxamide 4-(2,6-difluorophenyl)-3-[(1R)-1-(dimethylamino)ethyl]-1H-pyrrole-2-carboxylic acid N-azido-3,4,6-trichlorobenzenesulfonamide (3R,5S)-1-benzyl-N,5-dimethoxypiperidine-3-carboxamide N-(1,3-benzodioxol-5-ylmethyl)-4-cyclopentyloxy-5-methyl-2-propan-2-ylaniline 2-(4,4-dimethylcyclohexen-1-yl)-7-methylidenepyrido[2,3-b]pyrazine 6-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-1H-pyridin-2-one 2-(5,6-dichloropyridin-3-yl)oxyethanamine 2-[3,5-dichloro-4-[(6-oxo-1H-pyridazin-3-yl)oxy]anilino]acetic acid 3-[4-(2-ethylhexoxy)phenyl]propanoic acid N-(3,4-dihydroxyphenyl)octadecanamide (1Z,3E)-4-chloropenta-1,3-dien-1-amine;1-cyclopentyl-2-[5-(4-methoxyphenyl)pyrimidin-2-yl]ethanone 2-N-[(3R,4S)-1-cyclopropylsulfonylpiperidin-3-yl]-4-N-methylpyrimidine-2,4-diamine;hydrochloride 2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]propanoic acid (E)-3-phenyl-N-[1-[4-[2-(propanoylamino)ethyl]phenyl]piperidin-4-yl]prop-2-enamide ethane;6-(4-fluorophenyl)-2,3-dimethylimidazo[1,2-b]pyridazine 2-(4-chlorophenyl)-N,N-dimethylpiperidin-1-amine 4-amino-3-methylsulfonylbenzaldehyde N-[2,3-dihydroxypropyl(naphthalen-1-yl)methylidene]benzenesulfonamide 2-(4-anilinophenoxy)-N-[(Z)-1H-indol-3-ylmethylideneamino]acetamide 2-amino-4-(4-cyanophenyl)-6-methylbenzene-1,3-dicarbonitrile 4-[(1R)-2,3-dihydro-1H-inden-1-yl]benzenesulfonamide (2S)-2-[[4-[5-chloro-3,4-bis(phenylmethoxy)anilino]-1,2,5-oxadiazol-3-yl]amino]butanoic acid 4-(2,3-dihydro-1H-indol-6-ylmethoxy)benzenesulfonic acid N-[(Z)-1H-indol-3-ylmethylideneamino]-4-pyridin-2-ylbenzamide 2,5-difluoro-4-hydroxybenzenesulfonamide N-(3,4,5,6-tetrafluoropyridin-2-yl)sulfonyl-1H-pyrrolo[2,3-b]pyridine-2-carboxamide (E)-3-[4-(2,5-diaminophenyl)sulfanyloxyphenyl]prop-2-enoic acid 5-[(2E)-3,7-dimethylocta-2,6-dienoxy]pyridine-2-carbonitrile N-[(4,6-dimethoxy-2-methylpyridin-3-yl)methyl]-1-ethyl-2-oxoquinoline-5-carboxamide 2-[6-(cyclopropylmethoxy)-5,7,8,9-tetrahydrocarbazol-3-yl]acetamide 2-methyl-3,5-dinitrobenzoate N-[(2E,3Z)-2-ethylidenehexa-3,5-dienyl]-2-piperidin-1-ylacetamide;ethane 2-ethyl-4-(3-methoxyanilino)-6,7-dihydropyrrolo[3,4-d]pyrimidin-5-one 1-[(E)-3-(4-tert-butylcyclohexa-1,5-dien-1-yl)prop-2-enoxy]-6-ethylnaphthalene N'-ethyl-2,2-difluorobutanehydrazide;(5Z)-4-methylidene-1-[4-(6-phenylhexoxy)benzoyl]-3,5-bis(propan-2-yl)-3H-pyrrole-2-carbonitrile (5E)-2-(3,4-dichlorophenyl)imino-5-[(1-ethylindol-6-yl)methylidene]-1,3-thiazolidin-4-one 2-(4-methylpyrazol-1-yl)-3H-quinazolin-4-one 2-[4-[(E)-3-fluoroprop-1-enyl]phenoxy]ethanol 1-azido-3-(3,4-dichlorophenyl)azetidine 4-(dibutylamino)-N'-hydroxypyridine-2-carboximidamide 2-[3-fluoro-4-(methanesulfonamido)phenyl]acetic acid 2-(4-chloro-6-methylcyclohexa-2,4-dien-1-ylidene)acetonitrile;1,3-dihydroisoindole (5Z)-2-(4-bromo-3,5-dimethylphenyl)imino-5-[(E)-3H-1,3]thiazolo[5,4-b]indol-6-one 4-[(2S)-4-hydroxy-5-oxo-2-[[4-phenoxy-3,5-di(propan-2-yloxy)phenyl]methylideneamino]pentanoyl]benzoic acid N-[3-(7,9-dihydro-6H-[1,2,4]triazolo[3,4-f]purin-5-yl)phenyl]-2,6-dimethoxybenzamide N-[4-(3-aminophenyl)-2,6-dimethylcyclohexa-1,3-dien-1-yl]ethanesulfonamide 1-ethenyl-2,4,5-trifluoro-3-(2-methoxyphenoxy)benzene 3-(4,5-dihydro-1H-imidazol-2-ylamino)-2-hydroxybenzoic acid N-[2,4-dichloro-5-(dimethylaminosulfanyl)phenyl]-3-(1-hydroxyethylideneamino)-2-methoxybenzamide N-[1-(4-methylphenyl)sulfonylpiperidin-3-yl]-2-propan-2-ylsulfanylacetamide 1-methoxybutane;6-[3-(4-nitrophenyl)oxiran-2-yl]naphthalene-2-carboxylic acid (5Z)-2-(4-chlorophenyl)imino-5-[[3,5-dibromo-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one 6-[[2,6-difluoro-4-(2-phenylethynyl)phenoxy]methyl]pyridine-3-carboxylate 5-(2,4-dimethylphenoxy)-3H-pyrido[3,4-d]pyrimidin-4-one 2-[[4,5-bis(ethenyl)imidazol-1-yl]methoxy]benzaldehyde;1-pyrrolidin-3-ylpiperidine N-[(Z)-1-amino-3-ethenyliminoprop-1-en-2-yl]-3-cyclopentyloxy-5-methanimidoylbenzamide N-[4-(2,6-dimethoxyphenyl)sulfinamoylnaphthalen-1-yl]-3-pyridin-2-ylpropanamide 2-(2-chlorophenyl)-3-[(1R,2S)-1-methyl-4-[[(6S)-5,7,8-trifluoro-5-oxooctyl]carbamoyl]cyclohexanecarbonyl]oxypropanoic acid (2E)-4-[6-methyl-7-oxo-3-propanoyl-5-(pyridine-3-carbonyl)oxycarbonylpyrazolo[1,5-a]pyrimidin-2-ylidene]butanenitrile 1-[1-(3,5-dimethoxyphenyl)cyclopropyl]pyrrolidine 3-(4-fluorophenyl)-N'-(5,6,7,8-tetrahydronaphthalen-1-ylmethyl)propanehydrazide;hydrochloride 3-[1-(4-methylphenyl)pyrazol-3-yl]propanamide 4-[(2,6-dimethylphenyl)-[(2Z)-3-oxobuta-1,3-dien-2-yl]phosphoryl]-N-(2-ethylphenyl)pentanamide 2-(3,4-dimethoxyanilino)quinazoline-7-carbohydrazide N-[4-(3,5-dimethyl-1H-pyrrol-2-yl)phenyl]-2-methoxyacetamide N-(3,5-difluorophenyl)-4-[2-fluoroethyl(propylsulfonylamino)methylidene]piperidine-1-carboxamide 2-(3,4-dichlorophenyl)-5-[[4-methoxy-3-(3-methylbutyl)phenyl]methylidene]-1,3-thiazolidine 4-[(E)-2-cyanoethenyl]-5-fluoro-N,3-dimethylpyridine-2-carboxamide (Z)-3-amino-N'-[amino(methyl)amino]prop-2-enimidamide;ethane;4-[[5-[2-fluoro-4-(trifluoromethoxy)phenyl]-1,6-dihydropyridazin-2-yl]methyl]-1H-pyrrole-2-carboxylic acid 5-(2,3-dihydrothiophen-4-yl)-1-(2,6-dimethylphenyl)sulfonyl-7H-pyrazolo[3,4-b]pyridin-6-one 1-[(3R)-5,6-dichloro-2,3-dihydroindol-1-yl]propan-1-one 5-(2,4-dihydroxy-6-methylphenyl)-N'-(2-sulfanylphenyl)furan-2-carboximidamide 1-(9,9-dimethylfluoren-2-yl)-3H-[1]benzofuro[3,2-c]pyridine 7-methyl-5-[1-(2,4,6-trichlorophenyl)pyrazole-3-carbonyl]-5a,10a-dihydro-4H-pyrrolo[1,2-b]isoquinoline-3-carbonitrile (3R,5S)-2-[6-amino-4-[(1R,2R)-2-(methoxymethyl)cyclopropyl]pyridin-2-yl]oxy-7-azaspiro[4.5]decane-7-carboxylic acid N-[4-[1,5-bis(4-chlorophenyl)pyrazol-3-yl]butanoyl]-2-[3-fluoro-5-(trifluoromethoxy)phenyl]acetamide 1-(2,6-dimethylpyridine-4-carbonyl)-3H-indole-2-carboxamide 1-(4-ethylcyclohexyl)-5-[2-fluoro-4-(trifluoromethoxy)phenyl]pyrazolidin-3-one 2-azidooxy-6-methylsulfonylpyridine N-[1-(7-fluoro-5-methyl-4,6-dioxobenzo[g]pteridin-2-yl)piperidin-3-yl]-1H-indazole-4-carboxamide N-[2-(methylamino)ethyl]-7-oxoheptanamide;6-phenyldibenzothiophen-4-ol 3-(2,4-dichlorophenyl)-N-[(E)-1H-indol-3-ylmethylideneamino]-5-oxopyrrolidine-3-carboxamide N-[1-(cyclohexylmethoxy)-5,6-dihydrobenzo[f]quinoxalin-3-ium-2-yl]-4-chlorobenzenesulfonamide 3-[(4,5-dimethylthiophen-2-yl)methyl]piperidine;ethane (1-benzoylpiperidin-3-yl)carbamic acid 4-(azidooxymethyl)-1,2-dipropylbenzene 3-(4-chloro-5-methylthiophen-2-yl)-N-(3,5-ditert-butylphenyl)pyridine-2-carboxamide N-[3-[3-(1,2-dihydrotriazol-5-ylmethoxy)phenoxy]phenyl]-N'-propan-2-ylmethanediamine 6-[4-[(2,4-dimethylphenyl)methoxy]piperidin-1-yl]pyrazine 5-(4-aminobutyl)thiophene-3-carboxylic acid;hydrochloride 2-[4-methoxy-N-(1,3-thiazol-5-yl)anilino]acetonitrile 4-bromo-2-[(E)-2-(1,3,5-trimethylpyrazol-4-yl)ethenyl]phenol 6-(4-methylpiperidine-1-carbonyl)oxynaphthalene-2-carboxylic acid 3-(azidomethyl)-2,5-dibromopyridine 2-[1-(5,6,7,8-tetrahydro-3H-imidazo[4,5-c]azepin-4-ylmethyl)cyclopentyl]ethanol 2,5-diphenylbenzo[h]chromene N-[1-[(3S,5R)-5-aminooxepane-3-carbonyl]piperidin-4-yl]benzamide;hydrochloride 1-[(2R,5R)-4-azido-2-ethyl-5-methylpiperazin-1-yl]-3-phenylpropan-1-one 4-[(1S)-1-aminoethyl]-6-[3,5-dichloro-2-fluoro-4-[(2R)-pentan-2-yl]oxyphenyl]pyridine-3-carboxylic acid 3-bromo-7-methyl-6H-furo[2,3-e]indole [4-(6-chloro-3,7-dimethylimidazo[4,5-b]pyridin-2-yl)phenyl]-morpholin-4-ylmethanone;ethane 1-[5,6-bis(4-fluorophenyl)pyrazin-2-yl]-N-tert-butyl-N-methylpyrrolidin-3-amine 1-N,4-N-bis[(3R)-oxolan-3-yl]benzene-1,4-dicarboxamide 3-[7-[5-(ethylaminomethyl)pyridin-2-yl]imidazo[1,2-a]pyridin-3-yl]benzaldehyde (6S,11bR)-10-acetyl-3-methoxy-6-propanoyl-2-pyridin-4-yl-5,6,7,8,9,11b-hexahydrobenzo[a]quinolizin-11-ol 2-[3,5-dimethyl-1-(4-phenoxyphenyl)pyrazol-4-yl]oxyacetamide 1-[3,5-bis(trifluoromethyl)benzoyl]piperazine-2-carboxamide 2-chloro-6-[(2S)-1-methoxypropan-2-yl]oxycarbonylbenzoic acid 4-(8,9-difluoropyrido[3,2-b]indol-6-yl)-3-methoxybenzonitrile 2-(4-chlorophenyl)-N-[3-methoxy-5-[1-[[5-(2,2,2-trifluoroethylsulfanylmethyl)pyridine-2-carbonyl]amino]cyclopropyl]pyridin-2-yl]acetamide 4-chloro-5-iodo-1H-pyrimidin-6-one 1-[3-methyl-4-(2-pyrimidin-5-ylethynyl)phenyl]-N-propan-2-ylpiperidine-4-carboxamide 3-benzyl-6-(4-methoxyphenyl)-2,5-dihydropyrazolo[3,4-d]pyrimidin-4-one N-(5,6-dihydropyrrolo[1,2-b]pyrazol-3-ylidene)-4-fluorobenzenesulfonamide N-(1H-indazol-5-yl)-2-methyl-6,7-dihydro-4H-thieno[3,2-c]pyran-4-carboxamide (4S)-1,1,3,7-tetramethyl-3-[2-oxo-5-phenyl-3-[3-(trifluoromethoxy)phenyl]imidazole-1-carbonyl]-1,4-thiazepane-2,5-dione 7-(cyclopropylmethoxy)-6-fluoro-2,3-dihydrochromen-4-one 2-(4,6-dimethylpyrimidin-1-ium-5-yl)propanoic acid;chloride (2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3,3-difluoro-2-hydroxybutanamide 1-azidooxy-2-methyl-3,4-dihydroisoquinoline N-(5-fluoropyridin-2-yl)-1-(1,3-thiazol-4-ylmethyl)benzimidazol-2-amine (2R)-N'-[6-(4-chlorophenyl)pyrimidin-4-yl]-N,N'-dipropylbutane-1,3-diamine (1S,3R)-N-[8-amino-6-(4-methylpyridin-3-yl)isoquinolin-3-yl]-2,2-difluorocyclopropane-1-carboxamide 2,2-diamino-6-[3-(1H-imidazol-5-yl)phenyl]hexanoic acid 1-(4-chlorophenyl)-3,5-bis[(Z)-(2,4-dihydroxyphenyl)methylideneamino]urea 4-[2-[5-[(3,3-difluoropyrrolidin-1-yl)methyl]pyridin-3-yl]-9H-imidazo[4,5-b]fluoren-7-yl]-N-(furan-2-ylmethyl)pyrimidin-2-amine 4-[(1R)-3-(2-chloropyridin-4-yl)-1,1,3,3-tetrafluoropropoxy]benzenecarboximidamide 4-(dimethylamino)-N-[1,3,5-trimethyl-7-[[2-oxo-2-(5,6,7,8-tetrahydronaphthalen-2-ylamino)ethyl]amino]pyrazolo[4,3-d]pyrimidin-6-yl]benzenesulfonamide 1-[2,6-difluoro-4-(trifluoromethyl)phenyl]pyrrolidine (2R)-6-hydroxy-1'-[(4-methoxyphenyl)methyl]spiro[3H-indene-2,4'-piperidine]-2'-one 1-[4-hydroxy-3,5-bis(methoxycarbonyl)phenyl]ethenesulfonate N-[2,4-difluoro-3-(5-pyridin-2-ylimidazo[1,5-a]pyrazin-8-yl)phenyl]methanesulfonamide 4-bromo-2,6-dimethylbenzenesulfonate 2,5-dinitro-N,N-bis(3-nitrophenyl)aniline 2-[1-[2-(oxan-4-yl)ethoxy]isoquinolin-3-yl]acetamide 3-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-6-[4-[2-ethoxyethyl(methyl)amino]piperidine-1-carbonyl]-8-phenyl-1H-quinolin-2-one N-(3-methylcyclobutyl)-4-[1-[(E)-2-phenylethenyl]pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-2-amine N'-[(2,4-dimethylphenyl)iminomethyl]-N-[2-(oxiran-2-ylidenemethyl)phenyl]methanimidamide;ethane 1-[(3-chlorophenyl)methyl]-6-hydroxy-5-oxo-N-piperidin-4-ylpyridine-2-carboxamide (1S,3R)-3-[[2-amino-6-chloro-5-(4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]cyclohexane-1-carboxylic acid ethane;N-[(4Z)-3,6,8-trimethylideneundeca-2,4,9-trien-5-yl]oxybenzamide (7S)-7-[3-chloro-4-[(4-methylphenyl)methoxy]anilino]-1,1-dioxothiepane-2-carboxylic acid 3,5-dimethoxy-4-[(2E)-4-nitrohexa-2,5-dien-2-yl]phenol N-[3-(5,6-dihydronaphthalen-1-yl)phenyl]benzamide N-[(2S)-5-azido-1,3-dioxo-6-phenylhexan-2-yl]-4-fluorobenzamide 3-[4-(1,3-benzodioxol-5-ylmethylamino)cyclohexyl]-2-N-phenylquinoline-2,8-diamine N-[(4-chlorophenyl)methyl]-2,5-difluorobenzenesulfonamide 1-[2,4-dichloro-3-[(6-ethyl-2-methoxy-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-yl)oxy]phenyl]ethanone 1-[5-(2,2-dimethylpropyl)pyridin-3-yl]-4-[[5-[methyl-[2-(oxan-2-yloxy)ethyl]amino]pyridine-2-carbonyl]amino]cyclohexa-2,4-diene-1-carboxylic acid [1-(6-bromopyridin-2-yl)piperidin-4-yl]carbamic acid 5-fluoro-6-[(1R)-2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl]pyridine-3-carbonitrile 1-[5,7-difluoro-2-(4-methylphenyl)-1H-indol-3-yl]butan-1-one 1-(2,4,6-trichlorophenyl)-1H-indene 4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazol-5-yl]benzenesulfonamide 2-[3,5-bis(trifluoromethyl)phenyl]-1-[4-[(7-bromoimidazo[4,5-c][1,8]naphthyridin-1-yl)-ethoxymethyl]piperidin-1-yl]-2-cyclopropylideneethanone 4-hydroxy-N-[(3R)-1-[5-methyl-2-(methylideneamino)benzoyl]pyrrolidin-3-yl]benzamide 1-[(3R)-3-[6-(4,5-dimethylimidazol-1-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]oxypyrrolidine-1-carbonyl]-N,N-dimethylcyclopropane-1-carboxamide [1-(4-fluorophenyl)cyclopropyl]-(3-methoxyazetidin-1-yl)methanone 5-[3-(2,2-difluoroethyl)phenyl]-5H-pyrazolo[1,5-a]pyridine 2-[6-(difluoromethyl)pyridin-3-yl]-5-(2,6-dimethoxyphenyl)-N-methyl-4H-1,3-thiazole-2-carboxamide;ethane 5-[3-(3,4-dihydro-2H-chromen-6-yl)imidazol-1-ium-1-yl]pentanoic acid 2-[4-(3,5-dimethylpyrazole-1-carbonyl)phenoxy]acetic acid 5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]furan-3-carboxylic acid N-azido-4,6-bis(methylsulfanyl)pyrimidine-5-carboxamide 1-[5-methyl-2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)phenyl]ethanone 3,6-bis(4-chloroanilino)benzene-1,2-dicarbonitrile 5-ethyl-3,4-dimethoxy-N-[(Z)-[1-methyl-6-methylidenecyclohexa-2,4-dien-1-yl]methylideneamino]aniline 3-[3-(2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl]butanoic acid 5-chloro-N-[(2,4-dimethoxyphenyl)methyl]pyrimidine-2-carboxamide 4-methoxy-N,1-bis(phenylmethoxy)butan-2-imine 6-[(3R)-1-[[7-chloro-5-(difluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methyl]pyrrolidin-3-yl]oxypyridine-2-carbonitrile 2-methyl-5-[3-(1,3-oxazol-4-yl)-5,8-dioxoimidazo[1,5-a]pyrazin-6-ylidene]pentanoic acid 4-[6-(1,2-benzoxazol-3-yl)pyridin-3-yl]sulfonyl-N,N'-dimethylpiperazine-1-carboximidamide 2-[2,4-dichloro-6-[(E)-1-(2H-tetrazol-5-ylamino)prop-1-en-2-yl]phenoxy]acetic acid N-cyclohexa-1,3-dien-1-yl-2-[4-(7H-purin-6-yl)piperazin-1-yl]acetamide 2-[4-fluoro-2,6-di(propan-2-yl)phenyl]acetonitrile 3-(3-azidooxy-5-chlorophenoxy)pyridine 3-(4,6-dichloro-2-oxochromen-3-yl)benzenesulfonic acid 1-[2-azido-5,5-dichloro-4-(5-methylfuran-3-yl)pentyl]piperazine (6S)-2-benzylsulfanyl-6-methyl-7,8-dihydro-6H-pyrido[1,2-a]pyrazine-3,5-dione N-(3,5-dichlorophenyl)sulfanyl-5,7-difluoro-4H-imidazo[1,2-a]quinoline 5-[(4-butoxyphenyl)methyl]-3-[3-[4-(morpholine-4-carbonyl)cyclohexa-1,3-dien-1-yl]propanoylamino]thiophene-2-carboxylic acid (2S)-1,3-diethyl-4-methoxyimino-2H-pyridine-2-carboxylic acid 2-[4-(1,5-dimethylpyrazol-3-yl)piperazin-1-yl]-N-(3-fluorophenyl)acetamide N-[2-(3,5-difluorophenyl)ethyl]piperidine-1-sulfonamide (3R,5S)-7-[(2-chlorophenyl)methyl]-4-hydroxy-N,N-dimethyl-1-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide;hydrochloride (NZ)-N-[[4-amino-2-fluoro-6-[methyl(3-sulfanylpropyl)amino]phenyl]methylidene]hydroxylamine N-methyl-1'-(pyridine-4-carbonyl)spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 1-[(3E,5Z)-hepta-3,5-dien-4-yl]-N-methoxy-1H-indene-2-carboxamide 4-hydroxy-5,8-dihydrobenzo[f]quinazoline (3-fluorophenyl)-[4-(1H-pyrrolo[2,3-b]pyridin-4-ylmethyl)piperazin-1-yl]methanone ethane;(E,2Z)-6-hydroxy-N,4-dimethyl-N-[2-[[5-methylidene-3-oxo-1-[4-[(2-phenylacetyl)amino]phenyl]hexan-2-yl]amino]ethyl]hept-2-enamide 2-[(5Z)-1-(4-chlorophenyl)-5-(2-oxopropylidene)imidazolidin-2-yl]acetic acid 5-cyclopropyl-2-[(4,4-difluoropiperidin-1-yl)methyl]pyridine;ethane 1-[4-methoxy-3-(4-phenylbutanoyl)-2H-naphthalen-1-ylidene]-2,6-dihydropyridine-4-carboxylic acid 2-ethylbutanoic acid;5,7,8-trimethoxy-6-[(4-propan-2-ylphenyl)methyl]-1H-quinazoline-2,4-dione 2,4-difluoro-3-hydroxybenzenesulfonic acid 1-methyl-N-[(1R)-2,3,4,5-tetrahydro-1H-naphthalen-1-yl]piperidine-4-carboxamide N-[(2-chloropyridin-4-yl)methyl]-1-[(3R,5S)-1-[(5,6-dimethylpyrimidin-4-yl)amino]-5-methylpiperidin-3-yl]triazole-4-carboxamide 1-bromo-4-ethenylnaphthalen-2-ol 6-ethoxy-2-(2-oxopropyl)benzoic acid 4-[2,3-dichloro-5-(4-hydroxyphenyl)phenyl]phenol 4-[[(2S)-2-azidooxybutyl]amino]benzenesulfonamide 5-chloro-2-(difluoromethyl)-N-[4-[4-oxo-4-(triazolo[1,5-a]pyridin-7-ylamino)butanoyl]phenyl]benzamide N'-hydroxy-3,5,6-trimethylbenzenecarboximidamide 3-[(4-chlorophenyl)methyl]-2H-chromen-7-ol 5-[[(3S)-2,7-dimethyloct-6-en-2-yl]sulfamoyl]thiophene-2-carboxylic acid 6-[(E)-3-methoxybut-2-enyl]-1,10-dihydrophenanthrene 6-N-azido-7H-purine-2,6-diamine 2-[4-bromobutan-2-yl(methoxycarbonyl)amino]benzenesulfonic acid (5-azido-6-benzyl-2,3,4,9-tetrahydrocarbazol-1-ylidene)-phenylmethanolate (E)-3-[4-[5-methyl-2-(2,2,2-trifluoroethoxy)phenyl]piperidin-1-yl]prop-2-enal (5E)-5-[(4-ethylphenyl)methylidene]-2-(3-methoxypropylimino)-1,3-thiazolidin-4-one 1-(3,4-dihydroxyphenyl)-5-methylcyclohexa-2,4-dien-1-ol 5-(1H-indol-2-yl)-3,4-dimethoxybenzenethiol (3-fluoroazetidin-1-yl)-[5-(5-fluoro-2H-indazole-4-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]methanone (3-bromophenyl)methyl-diethoxyphosphane 3-(8,9a-dihydro-1H-fluoren-9-ylmethoxy)-4-fluoroaniline 5-[2-[3,4-dimethoxy-6-[(E)-prop-1-enyl]pyridin-2-yl]ethenyl]-N,2-dimethylaniline 1-[(3R)-3-[6-(methylamino)purin-9-yl]piperidin-1-yl]propan-2-one 5-[3-(difluoromethyl)-4,7-dihydropyrazolo[4,3-d]pyrimidine-1-carbonyl]-2-methyl-N-propan-2-ylbenzenesulfonamide 4-azido-1-benzyl-3-methoxypiperidine 4-chloro-5-[(2S)-5-oxopyrrolidine-2-carbonyl]oxypyridine-3-carboxylic acid (1Z,3E)-2-[4-[8-[(5-methoxy-2,3-dihydroindole-1-carbonyl)amino]imidazo[1,2-a]pyridin-2-yl]phenoxy]hexa-1,3,5-triene-1-sulfonate (4-cyclopropyloxyphenyl)methanediol 2-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-N-[[4-[3-(oxetan-2-yloxy)propyl]phenyl]methyl]acetamide 3-[[(Z)-2-(4-methoxyphenyl)ethenyl]sulfonylamino]benzoic acid 4-N,5-N-diethyl-2-N-(4-fluorophenyl)-[1,3]thiazolo[4,5-d]pyrimidine-2,4,5-triamine (5-chloro-3,6-dihydro-2H-pyridin-1-yl)-[1-(4-methoxyphenyl)cyclobutyl]methanone [4-(4-hydroxybutan-2-yl)phenoxy]-methylidene-[4-[4-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]benzoyl]azanium 2-[(3R)-3-methylpyrrolidin-1-yl]-N-(4-pyrazol-1-ylphenyl)quinoline-4-carboxamide 2-(4,5-dimethoxy-1H-indole-2-carbonyl)iminopentanoic acid (1S,2R)-3-[(4-fluorophenyl)methyl]-2-hydroxycyclopentan-1-ol 2-methoxy-4-[[3-(1-prop-1-en-2-ylazetidin-3-yl)oxycyclobutyl]amino]pyrimidine-5-carboxamide (2-methoxy-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-3-yl)-pyrrolidin-1-ylmethanone;2,2,2-trifluoroacetic acid 2,4-ditert-butylbenzene-1,3,5-tricarboxylic acid 4-[(2R,3S)-1-acetyl-5-(3,4-dichlorophenyl)iminopyrrolidine-3-carbonyl]benzonitrile 4-N,2-bis(ethenyl)-1-N,8a-diphenylnaphthalene-1,4-diamine;9H-carbazole 1-(2,6-dimethylphenyl)-3-[[4-[(2-methoxyphenyl)methyl]morpholin-2-yl]methylsulfonyl]urea N-[(3S)-3,4-dihydro-2H-chromen-3-yl]-2,2,3,3-tetramethylcyclopentane-1-carboxamide (4S)-2-methyl-3,4-diphenylbicyclo[5.1.0]octa-2,6-diene N-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide N-(4-aminophenyl)-2,4,6-trimethylpyridine-3-carboxamide 3-(N-cyclopropylanilino)-5,6-dimethoxyisoquinoline-7-carboxylic acid 2-[N-(furan-2-ylmethyl)-4-(pyrimidin-2-ylsulfamoyl)anilino]acetic acid 5-[3-(3,4-dichlorophenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-6-methoxyimidazo[2,1-b][1,3]thiazole 4-[(2S)-1-[2-chloro-3-[(5-cyclopropyl-6-oxopyridin-1-yl)methyl]benzoyl]pyrrolidin-2-yl]oxybenzonitrile (Z)-[1-amino-2-[4-(N'-hydroxycarbamimidoyl)phenyl]propylidene]carbamic acid 1-[2-(benzenecarboximidoylamino)ethoxy]-4-chloro-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-b]pyridin-2-one 1-[4-(2,6-dichlorophenyl)-5-methyl-1H-pyrazole-3-carbonyl]-N'-ethylpiperidine-4-carboximidamide;formic acid 6-(4-hydroxyphenyl)sulfonyl-3,5-dihydro-2H-pyrrolo[3,4-f]quinoline-1,7-dicarboximidamide N-(1H-indazol-4-yl)-2,5-dimethoxybenzenesulfonamide 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-pyridin-3-ylethyl)morpholine-4-carboxamide 1-N'-[4-methyl-3-(trifluoromethyl)phenyl]-2,6-dioxo-1H-pyrimidine-4,5-dicarboximidamide N-[1-(5-chloropyridin-2-yl)pyrazol-4-yl]cyclopropanecarboxamide 6-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-(4-hydroxybutyl)amino]naphthalene-2-sulfonic acid (E)-N-[(3Z,5Z)-1H-1,5-diazonin-2-yl]-3-methoxy-4-thiophen-2-ylbut-3-enamide 2-[[(1R)-1-[3-chloro-5-fluoro-2-hydroxy-4-(trifluoromethyl)phenyl]ethoxy]carbonylamino]acetic acid N-[(2R,3S)-1-methyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]cyclohexanesulfonamide 1-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)azetidine-2-carboxylic acid [5-(furan-3-yl)-1H-pyrazol-4-yl]-[2-(thiophen-2-ylmethylamino)pyrimidin-5-yl]methanone 2-[3,5-bis(trifluoromethyl)phenyl]-N-[1-(2-hydroxyethoxymethylamino)isoquinolin-6-yl]-N',2-dimethylpropanediamide 2-(4-butoxyphenyl)-6-fluoroquinoline-5,8-dione 3-cyclopropylsulfonyl-6,7-difluoro-N-[2-[(1R)-5,5,5-trifluoro-1-methoxypentyl]pyridin-4-yl]quinoline-4-carboxamide (2S)-N-[5-cyclopropyl-3-[2-fluoro-4-(trifluoromethoxy)phenyl]pyrazol-1-yl]-2-hydroxybutanamide 5-hydroxy-2,2,4-trimethyl-6-oxochromene-3-carboxamide 6-methoxy-3-N-[(E)-3-piperazin-1-ylpropylideneamino]quinoline-2,4-diamine 2-[(4-chlorophenyl)-diphenylmethoxy]-3,3-difluoro-5-hydroxypentanoic acid 2-(4,5-dichlorothiophen-3-yl)-1-[4-(2H-pyridin-1-ylmethoxymethyl)phenyl]ethanone [5-tert-butyl-2-(4-fluorophenyl)pyrazol-3-yl]urea;formonitrile 2-methylpropane;5-(1,3-oxazol-5-yl)-3H-indene-1-carboxamide (2S)-N'-hydroxy-2,4-diphenylbutanediamide (7R)-2,7-bis[[4-(methylsulfanylmethoxy)phenyl]methylideneamino]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 4-methyl-3,4,5a,6,7,8,9-octahydrophenanthrene-2,7-diol N-benzylsulfonyl-N',1-dimethylcyclopentane-1-carbohydrazide 5-[[1-(6-tert-butylpyridine-2-carbonyl)azetidin-3-ylidene]methylsulfonyl]thiophene-3-carboxamide N-[2-fluoro-5-[(6-methylpyridine-3-carbonyl)amino]phenyl]-1,5-dimethylpyrazole-4-carboxamide 4-(azidomethyl)-3,5-diethoxyphenol N-[(3R)-1-(2,5-dihydroxybenzoyl)pyrrolidin-3-yl]-4-fluorobenzamide 4-(2,2-dimethylbutyl)anthracene 1-[(E)-[(3R,4S,5R)-2,2-dimethyl-3-propan-2-ylidene-7-oxa-11-azatricyclo[6.4.0.02,6]dodeca-1(12),8,10-trien-4-yl]diazenyl]naphthalene-2-carboxamide 4-[(3S,5R)-4-[[3,6-dimethoxy-2-[[1-(methylamino)cyclopentyl]methyl]phenyl]methyl]-3,5-bis(hydroxymethyl)piperazin-1-yl]benzonitrile (1-methylcyclopropyl)-[3-(4-methylpiperazin-1-yl)azetidin-1-yl]methanone;2,2,2-trifluoroacetic acid 4-N,5-diethyl-2-N-[2-methoxy-4-(4-morpholin-4-ylpiperidin-1-yl)phenyl]-7H-pyrrolo[3,4-d]pyrimidine-2,4-diamine N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-5-[5-(morpholine-4-carbonyl)-3-piperidin-4-ylphenyl]benzamide 2-(3,4-dihydroquinolin-6-yloxy)-N-[(E)-1H-indol-3-ylmethylideneamino]acetamide 2-[3-(2,6-dioxopiperidin-3-yl)-4-methyl-2H-1,2,4-triazin-5-ylidene]-2-isocyanoacetonitrile N-[2-[N'-(6-bromopyridin-3-yl)carbamimidoyl]-5H-pyrrolo[3,2-d]pyrimidin-6-yl]acetamide [(4S,5R)-3-(2,4-difluorophenyl)-4-(oxan-4-yloxymethyl)-6-(2H-triazol-4-yl)-1,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]-piperidin-1-ylmethanone (5R,6S)-4-[[4-(2-ethyl-1H-imidazol-5-yl)-3,6-dihydro-2H-pyridin-1-yl]methyl]-2-methoxy-9-oxa-3,14-diazatricyclo[8.4.0.02,7]tetradeca-1(10),11,13-triene 4-(9H-fluoren-9-ylmethoxycarbonylamino)-5-(hydroxymethyl)pentanoic acid 3-ethenyl-N,2-dimethylidenechromene-7-sulfonamide [4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]phenyl]urea 7-[[3-(methoxymethyl)piperidin-1-yl]methyl]-2,4-dimethylpyrrolo[2,3-d]pyrimidine 1,3-ditert-butylbenzimidazole 2-methyl-N-[[3-(trifluoromethoxy)phenyl]methyl]propanamide (Z)-2,3-diamino-N'-[1-[4-[4-[(E)-hept-4-enoxy]phenyl]phenyl]ethyl]prop-2-enimidamide (1S,3R)-N-[4-(cyclopenten-1-ylmethoxymethyl)phenyl]-2-cyclopropylidene-3-methyl-1-propan-2-ylsulfonyl-6,7-dihydro-5H-pyrrolizine-1-carboxamide 1-[4,6-di(propan-2-yl)pyrimidin-5-yl]-N'-methoxyethane-1,2-diamine 4-ethyl-N-[2-(1-methylpyrazol-4-yl)ethyl]-3,5-dihydro-2H-pyrazine-6-carboxamide 2-methoxy-6,7-dihydro-5H-indolo[3,2-d][1]benzazepine 4-[2,3-bis(ethenyl)phenyl]pyrimidine [2-chloro-4-(3,5-ditert-butylphenyl)sulfanylcyclopenta-1,3-dien-1-yl]methanol N-(3,5-dichlorophenyl)-2-methyl-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]propanamide 3-(4,5-dimethyl-2-phenyldiazenyl-N-prop-2-enylanilino)butanoic acid N-[4-chloro-2-(6,7-dimethoxyquinolin-4-yl)phenyl]carbamate 1-[2,6-di(propan-2-yl)phenyl]pyrrole-3-carboxylic acid 1-(2,3-difluorophenyl)-N-[[2-methoxy-4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]cyclopropane-1-carboxamide (2R,5S)-3-amino-5-benzylsulfanyl-6-[(2-bromoacetyl)oxymethyl]oxane-2-carboxylic acid 3-[[7-chloro-5-(2,4-dimethoxyphenyl)-1H-2-benzazepin-8-yl]oxy]-N,N-dimethylpropan-1-amine 1-[1-(cyclohexylmethyl)cyclobutyl]-5,6-difluorobenzimidazole 4-(2,3,5,6-tetrafluorophenyl)-1H-indole 7-(2,4-dichlorophenyl)-8-methyl-3H-pyrido[3,2-d]pyrimidin-4-one 5-methyl-N,N'-bis(thiophen-2-ylsulfanyl)pyrimidine-2-carbohydrazide 2-[3-[[(2S)-5,7-dioxooxepan-2-yl]methoxy]phenyl]propanal 7-[2,3-dihydroxypropyl(methoxy)amino]-1H-quinoxaline-2,6-dione 2,4-ditert-butyl-6-[[(3R)-3-phenylmorpholin-4-yl]methyl]phenol 5-(3,4-dichlorophenyl)-2-[1-(1H-indole-3-carbonylamino)ethyl]pentanoic acid 3-[(4R)-5,6-dimethoxy-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepine-8-carbonyl]benzoic acid N-[5-[3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]cyclohexanecarboxamide N-(5-amino-2,3-dimethylphenyl)carbamate 4-cyclohexylsulfonyl-N-[2-(diethylamino)ethoxy]aniline 7-(methanesulfonamido)-4-oxo-1H-quinoline-3-carboxylic acid 1-[(E)-3-(2,4-dihydroxyphenyl)prop-2-enoyl]pyrrolidine-2,5-dione 3-[6-ethylsulfanyl-2-[5-(trifluoromethyl)pyridin-3-yl]pyridin-4-yl]propanenitrile 2-(3-cyclohexa-1,5-dien-1-yloxyphenyl)acetaldehyde 2-[3-(6,7-dichloroquinoxalin-5-yl)oxypropyl]isoindole-1,3-dione 1-(1-azidoethyl)-3-tert-butylbenzene [(3S,5R)-1-(cyclopropylmethoxycarbonyl)-7-fluoropiperidin-3-yl]-methylidyneazanium (Z)-2-[1-(2,6-diphenylpyridin-4-yl)ethylideneamino]ethenol 2-(5-aminopyridin-3-yl)-1H-benzimidazole-4-carboxamide 2-[5-carbamoyl-9-[(3,4-difluorophenyl)methyl]-2-(hydroxymethoxy)carbazol-4-yl]peroxyacetic acid 1-[(2R)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyanthracene-9,10-dione N-(5,6-dimethoxypyridin-3-yl)-1H-benzimidazole-2-carboxamide 1-[4-(2-azidoethyl)phenoxy]-3,5-ditert-butylbenzene N-[6-(2,6-dimethylphenyl)imidazo[1,2-a]pyridin-3-yl]formamide 2-(2,6-dichloroanilino)benzoic acid N-[5-(trifluoromethyl)pyridin-2-yl]pyridine-3-carboxamide N-[(3S)-5,8-dimethyl-4-oxo-2,3-dihydropyrido[1,2-a]pyrimidin-3-yl]-1-(2,6-dimethylphenyl)cyclopropane-1-carboxamide 2-(2,3-difluorophenyl)-N-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]acetamide (Z)-1-(4-methylphenyl)-2-methylidenepent-3-en-1-amine 2-(2,3-dihydroindole-1-carbonylamino)benzoic acid 3,5-dimethyl-2H-pyrano[3,2-g]quinoline 6-methoxy-1,3-dimethylbenzimidazol-2-one;propane 2-[[4,5-bis(4-methoxyphenyl)-1,3-thiazol-2-yl]sulfanyl]-N-[(Z)-(4-hydroxyphenyl)methylideneamino]acetamide N-[5-bromo-4-methyl-6-(2,3,3-trifluoropropanoylamino)pyridin-3-yl]-2,2-dimethylpropanenitrilium 1-(3,4-dihydro-2H-pyrano[3,2-b]pyridin-6-yl)-N-ethyl-N-methyl-5-(4-propan-2-ylphenyl)pyrazole-3-carboxamide (2-benzylpyrrolidin-1-yl)-[4-methoxy-5-methyl-2-[(E)-2-nitroethenyl]phenyl]methanone 5-[4-[6-(trifluoromethyl)pyrimidin-4-yl]oxypiperidin-1-yl]pyridine-2-carbonitrile (6S,8aR)-N-[2-(4-chlorophenyl)ethyl]-6-hydroxy-1,2,3,5,7,8-hexahydroindolizine-8a-carboxamide 2-cyclohexyl-N-[5-(2,3-difluorophenyl)sulfonyl-1H-indazol-3-yl]acetamide N-(3,4-dichloro-5-methylphenyl)-2-hydroxybutanamide N-(4-aminobutyl)-3,7-dioxo-2,6,8,12-tetrazatricyclo[7.5.0.02,6]tetradeca-1(9),10,11-triene-12-carboxamide 2-[(3R)-1-[2,5-difluoro-4-[4-[4-(trifluoromethyl)phenyl]cyclohexa-1,3-dien-1-yl]phenyl]sulfonylpyrrolidin-3-yl]oxyacetic acid 2-cyclopropyloxy-6-(3-oxobutyl)benzoic acid [3-(hydroxymethyl)phenyl]-propan-2-ylsulfamic acid (E)-3-(2,5-dimethylfuran-3-carbonyl)oxy-4-oxobut-2-enoic acid 4-hydroxy-2,3,6-trimethoxybenzoic acid N-[1-[4-[3-chloro-4-(pyridine-2-carbonylamino)phenoxy]phenyl]ethyl]oxane-4-carboxamide (3R,5S)-1-[4-(chloromethyl)benzoyl]-N-[(E)-(4-hydroxyphenyl)methylideneamino]-2-oxopiperidine-3-carboxamide N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-propan-2-ylidene-7,8-didehydroquinoline-6-carboxamide N-[4,5-diamino-2-(methylamino)phenyl]-2,2-difluoroacetamide 3-[2-(1,1-dioxothiolan-3-yl)-5-phenyl-1H-imidazol-4-yl]pyridine 2-[(1S,3R)-3-aminocyclopentyl]oxy-N-(5-fluoropyridin-3-yl)pyrimidine-4-carboxamide;dihydrochloride N-[3-chloro-4-(pyridine-2-carbonyl)phenyl]benzamide 3-[1,4-dihydroxy-7-(2,6,6-trimethylcyclohexen-1-yl)naphthalen-2-yl]oxypropanoic acid 4-(3-chloropropoxy)-1-benzothiophene 6-(2,4-dichlorophenyl)-N'-diazenylpyrazine-2-carboximidamide 5-[(1,2-diethyl-4,6-dimethylpyrrolo[2,3-b]pyridin-4-ium-5-yl)methoxy]-N-[3-fluoro-4-(trifluoromethylsulfanyl)phenyl]pyrimidin-2-amine 2-[4-ethylsulfonyl-1-[(4-fluoro-3,5-dimethylphenyl)methyl]piperidin-4-yl]-5,7-dihydrofuro[3,4-d]pyrimidine 4-[2,3-difluoro-4-(5-pentylpyrimidin-2-yl)phenyl]benzonitrile 2-[5-fluoro-6-(4-fluorophenyl)pyrimidin-4-yl]oxyethanol 2-[4-chloro-3-fluoro-6-(methylamino)pyridin-2-yl]sulfanyl-4-propyl-1H-pyrimidin-6-one (2R)-3-[1H-pyrrolo[2,3-b]pyridin-6-yl(5,6,7,8-tetrahydroquinolin-4-yl)amino]propane-1,2-diol 2-[N-(4-ethoxyphenyl)sulfonyl-3,5-dimethyl-1H-pyrazol-4-yl]acetic acid 2-[N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-hydroxyanilino]acetamide 4-[(3aR,6aS)-5-ethylsulfonyl-1,2,3,3a,4,6a-hexahydrocyclopenta[b]pyrrole-2-carbonyl]-N-methylpyridine-2-carboxamide 5-[(3R)-1-benzylpyrrolidine-3-carbonyl]-2,4-dimethyl-1H-pyrimidin-6-one 2-[4-(3-aminopropoxy)phenyl]-1-ethylbenzimidazole-5-carboxamide 7,12-dibromo-14-methyl-1,3,8,10,11,12-hexazatetracyclo[7.6.0.02,6.011,15]pentadeca-2(6),4,7,9,12,14-hexaene [6-(2,3-dihydro-1H-inden-5-yloxymethyl)pyrimidin-4-yl]-[4-(4-methylpyridine-2-carbonyl)piperazin-1-yl]methanone 1-(2,5-dimethylhexan-3-yl)triazole 1-[(2R,4S)-2-methyl-4-[[5-(3-methylpyrazole-1-carbonyl)pyridin-2-yl]methoxy]pyrrolidin-1-yl]ethanone N-(4-azidocyclohexyl)aniline 2,5-dinitrobenzenethiol;methanol 6-tert-butyl-4,4a,5,7,8,8a-hexahydropyrano[3,2-c]pyridine-2,3-dione 2,6-difluoro-4-[5-fluoro-3-(trifluoromethyl)pyrazol-1-yl]benzaldehyde 1-[(Z)-but-2-enyl]sulfanyl-3,4-dimethoxy-5-phenylpentan-3-amine N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]-4-methylbenzenesulfonamide 4-[2,3-dibromopropyl(1,3-thiazol-5-yl)amino]butan-1-ol 3,4-difluoro-2-(3-fluoropyridin-4-yl)phenol 1-[(4,6-dimethoxypyrimidin-2-yl)carbamothioylamino]cyclobutane-1-carboxylic acid 1-[5-azido-2,4-dichloro-3-[(4-methoxyphenyl)sulfonylamino]phenyl]-3-cyclohexylurea 2-[3,5-bis(trifluoromethyl)phenyl]-N'-hydroxy-6-[3-[4-(2-hydroxyethoxy)phenyl]phenyl]-1H-benzimidazole-4-carboximidamide 4-N,4-N-dimethyl-2-N-[(3S)-1-pyrrolidine-1-carbonylpyrrolidin-3-yl]pyrimidine-2,4-dicarboxamide (Z)-3,7-diethyl-6-hydroxynon-5-en-4-one;iridium;2-methanidyl-8H-isoquinolin-6-ide 6-(4,5-dimethylpyridin-2-yl)oxy-1H-pyrrolo[3,2-b]pyridine (2Z)-2-[(2E,4Z)-2-methylhepta-2,4,6-trienylidene]quinoline 4-N,4-N-bis[2,6-di(propan-2-yl)phenyl]-1H-1,3,5-triazine-2,4-diimine 2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-[[3-(trifluoromethyl)phenyl]methyl]acetamide (2E)-5,7-difluoro-2-[2-methylidene-1-[3-(pyrrolidine-1-carbonyloxy)propyl]pyrimidin-4-ylidene]-3H-inden-1-one 2-(1H-benzimidazol-2-yl)-7,8-dihydroquinoline 1-cyclopropylsulfonyl-N,3-dimethylindole-7-carboxamide 6-[2,4-bis(sulfanyl)phenyl]-1,3-dimethyl-5H-pyrazolo[3,4-d]pyrimidin-4-one 1-[3,5-bis(trifluoromethyl)phenyl]-2-(1H-indol-6-yloxy)ethanone (Z)-2,3-dimethylhex-4-ene;ethane;1-[(E)-3-[2-ethoxy-4-[(E)-pent-2-en-2-yl]phenyl]but-2-enyl]pyrrolidine 5-amino-6,7-diethoxy-4-methylchromen-2-one;1-[(6-chloropyridin-3-yl)methoxy]-9-(methyliminomethyl)anthracene (4R)-5,7-dichloro-3,4-bis(methoxyimino)-1-(2-oxoethylamino)quinoline-2-thione 2-[3,4-bis(ethenyl)phenyl]-N-phenylaniline 3-[(5E)-5-ethylidene-4-methyl-6-methylidenepyridin-2-yl]sulfanylpropanamide N-(1H-imidazol-5-ylmethylideneamino)thiadiazole-4-carboxamide 5-[4-(diethylamino)phenyl]-2-[[6-(methylaminomethoxy)pyridin-3-yl]methylsulfanyl]-1H-imidazole-4-carbonitrile;methane N-[4-[(3,5-dimethyl-1H-pyrazole-4-carbonyl)amino]phenyl]cyclopropanecarboxamide (1S)-N-[4-[2-(benzylamino)ethoxy]phenyl]-4,6-dioxocyclohexane-1-carboxamide 1-azido-4,7-diphenylpyrrolo[2,3-b]pyridine 1-(2-nitro-4-propylphenoxy)ethanamine 2-(2-methyl-4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxylic acid (4R)-N,2-dimethyl-1'-[5-(trifluoromethyl)pyridine-3-carbonyl]spiro[5,6-dihydrocyclopenta[d]pyrimidine-7,4'-piperidine]-4-carboxamide N'-[4,6-diamino-2-(3-chlorophenyl)pyrimidine-5-carboximidoyl]piperidine-1-carboximidamide 2,4-difluoro-1-(3-pentylphenyl)benzene 2,6-bis(ethylcarbamoyl)benzamide 5-[8-(4,6-dimethyl-1H-benzimidazol-2-yl)quinolin-5-yl]-3-iodobenzene-1,2-disulfonic acid 1-azido-2,4,5-trimethoxybenzene 2-(4,6-dimethylpyrimidin-5-yl)-7-[1-(oxolan-3-yl)piperidin-4-yl]-5H-pyrido[3,2-b]indole N-[3-(4-chlorophenyl)phenyl]formamide;2-methylpropane 7-azido-5,8-dimethylnaphthalene-2-carboxylic acid 1-[(2R)-2-azidopyrrolidin-3-yl]benzotriazole 2-[(E)-3-(aminomethyl)hex-1-enyl]-7,9-dihydropurin-8-one N-(2,2-dimethoxyethyl)-N-hexyl-6-(4-propan-2-ylphenyl)pyridazin-3-amine 1-[5-bromo-6-(4,4-difluoropiperidine-1-carbonyl)pyridin-3-yl]-2-ethylpentan-3-one N-(4-cyanophenyl)sulfonyl-3,4-diethyl-2-[2-oxo-2-(1H-pyrrolo[2,3-b]pyridin-3-ylamino)ethoxy]benzamide N-[5-(3,4,6,7,8,9-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-8a-ylmethyl)pyridin-2-yl]acetamide 2-[3-(dimethylamino)phenyl]-N-(3,5-dimethyl-1H-pyrazol-4-yl)morpholine-4-carboxamide [1-(2-hydroxyethyl)cyclobutyl]-[4-[2-(4-iodophenyl)ethynyl]piperidin-1-yl]methanone 1-chloro-3,5-difluorobenzene;4-(2-formyl-7-methoxy-6-methylindol-1-yl)butanenitrile 6-(3,4-dimethylphenyl)-5-(4-fluorophenyl)-N-hydroxy-1,2,4-triazine-3-carboxamide N'-[(3R)-1,1-dioxothiolan-3-yl]-4-[4-fluoro-6-(trifluoromethoxy)cyclohepta-1,3,5-trien-1-yl]benzenecarboximidamide N-[4-(1-aminocyclopropyl)pyridin-2-yl]-5-bromo-4-methoxypyrimidin-2-amine 5-amino-N,2-dimethylbenzenesulfonamide;ethane;uranium(2+) 2-[3-amino-4,5-dimethyl-6-(trifluoromethyl)pyridin-2-yl]sulfanyl-4-propyl-1H-pyrimidin-6-one 2-[4-chloro-3-(methanesulfonamido)phenyl]-6-(1,3-dimethylpyrazole-4-carbonyl)-5,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide (2S,4R)-N-[(Z)-(5-chloro-3-ethoxy-2-hydroxyphenyl)methylideneamino]-1,9-diazatricyclo[6.3.0.02,4]undeca-10.1(11),12-diene-7-carboxamide 6,8-dimethyl-2-phenylmethoxyimidazo[1,5-a]pyridine 3-[[4,5,6-trideuterio-2-(oxan-2-yloxy)pyridin-3-yl]amino]cyclobutan-1-ol N-[(5-bromopyridin-3-yl)methyl]-N-butylformamide 4-bromo-1,3,5-trimethylpyrrole-2-carboxylate 3-(1H-indazol-5-yl)-1H-pyrrolo[2,3-b]pyridine [4-(2,6-difluorophenyl)piperazin-1-yl]-(5-methoxy-3-methylidene-4H-isoquinolin-8-yl)methanone;ethane 1-[4,6-bis(methylamino)pyridine-2-carbonyl]-5-hydroxyazepan-3-one [3-(6,7-dimethoxy-4-oxochromene-2-carbonyl)phenyl]-ethylphosphinic acid 6-methyl-4-oxo-3,7-dihydropyrazolo[5,1-c][1,2,4]triazine-2-carboxamide 2-bromo-1-(4,6-dimethoxypyrimidin-5-yl)ethanone 5-chloro-4-(oxolan-3-ylamino)pyrimidine-2-carboxylic acid N-[5-(1,3-benzothiazol-2-yl)-6-methylpyridin-3-yl]-4-[4-[[ethyl(propan-2-yl)amino]methyl]phenyl]-1,2,4-triazol-3-amine 4-[(2R)-2,5-diaminopentanoyl]-N'-hydroxybenzenecarboximidamide (2E)-4-cyclohepta-1,3-dien-5-yn-1-ylidene-2-[2-(3-methylphenyl)cyclohexa-1,3-dien-1-yl]-6H-pyrido[2,3-d]pyrimidine 2-[2,3-dihydroxypropyl(hexyl)amino]benzoic acid 4-[(Z)-3-cyano-2-(2H-tetrazol-5-yl)prop-2-enimidoyl]-N-[3-hydroxy-1-methoxy-1-oxo-2-(4-pyridin-4-ylphenyl)propan-2-yl]benzamide 1-(3,4-dichlorobenzoyl)-2-[4-hydroxy-2-oxo-5-(trifluoromethoxy)-4H-benzo[g]chromen-8-yl]pyrrolidine-3-carboxylic acid (1S)-5,6-difluoro-4-oxo-2-pyridin-3-ylcyclohexane-1-carboxylic acid 6-[(2S,4R)-4-[5-(cyclopropylmethoxy)pyridin-3-yl]oxy-1-(1H-pyrazol-4-ylmethyl)pyrrolidin-2-yl]pyridine-3-sulfonamide (2R)-1,3-dimethyl-4-[[3-[5-(trifluoromethoxy)pyridine-2-carbonyl]imidazolidine-1-carbothioyl]amino]piperazine-2-carboxamide (5Z)-2-(3-chlorophenyl)imino-5-[[4-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidin-4-one (Z)-3,7-diethyl-6-hydroxynon-5-en-4-one;[6-(2,6-difluorophenyl)-9H-fluoren-9-id-2-yl]carbamic acid;platinum(2+) (1S)-1-[4-chloro-3-(6-methylpyridin-3-yl)phenyl]ethanethiol 6-azidooxy-N,N'-dimethylnaphthalene-1-carbohydrazide (6S)-5-amino-N-(2,3-dihydro-1H-inden-2-yl)-6-propan-2-ylidene-4-(2,4,6-trifluorophenyl)-1,4-diazepane-1-carboxamide N-[2-(cyclopropylmethylamino)-1,3-benzoxazol-5-yl]-4-[(3R,5S)-3,5-dimethylpiperazin-1-yl]benzamide 7,8-dimethoxy-2-(2-pyridin-4-ylphenyl)quinoline 2-hydroxy-N,N'-bis[(Z)-1H-indol-3-ylmethylideneamino]-4-methoxybenzenecarboximidamide (7-cyclohexylthieno[3,2-b]pyridin-5-yl)-phenylmethanone;ethane 4-chloro-6,7,8-trimethylquinazoline;ethane 1-(4-bromophenyl)-2-(5-methylpyrazol-1-id-3-yl)ethanone;uranium 4-[1-(3,5-dimethylphenyl)ethenyl]benzenesulfonic acid 4-azidosulfonylbenzenesulfonic acid 4-benzyl-6-chloro-3,9a-dihydrocarbazole 1-[2-(6-fluoroquinolin-4-yl)ethenyl]cyclohexan-1-amine 5-[5-chloro-2,4-difluoro-3-(triazol-1-ylmethyl)phenyl]pyridine-2-carboxamide 3-[(Z)-but-1-enyl]-4-methoxy-6-(2-phenylethynyl)pyran-2-one;ethane N-[5-(benzenesulfonyl)-4-chloropyridin-2-yl]nitramide 4-(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)piperazin-2-one N-[(1S)-2-[[4-[(3R,5R)-4-acetamido-3,5-dihydroxypiperidin-1-yl]pyridin-3-yl]amino]-2-oxo-1-phenylethyl]-3-methoxybenzamide 2-(3-azidophenyl)sulfanyl-5,7-dichlorocyclohepta-1,4,6-trien-1-ol 4-chloro-5,6,7-trideuterio-2-methoxyquinoline 6-[2,4-bis(4-methoxyphenyl)thiophen-3-yl]-5H-[1,2]oxazolo[5,4-d]pyrimidin-7-one [4-(5,7-difluoroquinolin-2-yl)morpholin-2-yl]methanol 1-(4-chlorophenyl)-N,2-dimethyl-5-[2-oxo-3-[4-(trifluoromethoxy)phenoxy]propanoyl]pyrrole-3-carboxamide 2-[(3S,7R,8aS)-7-azido-2-oxo-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]-N-benzylacetamide 5-methyl-N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]naphthalene-2-carboxamide 1-[2,6-dimethyl-4-[3-(1H-pyrazol-5-yl)phenoxy]phenyl]ethanone 2-[3,5-bis(trifluoromethyl)phenyl]-N-[5-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]acetamide 4-methyl-N'-(2,3,5,6-tetrafluorobenzoyl)benzohydrazide 2-methyl-1-[4-(1,3,5-trimethylpyrazole-4-carbonyl)piperazin-1-yl]propan-1-one 2-(3-hydroxysulfanylphenoxy)terephthalic acid 2-tert-butyl-6-[(1E,3Z)-hexa-1,3,5-trienyl]-7-hydroxypyrido[2,3-d]pyrimidine-4-carboxylic acid 2-bromo-1-(4,5-dimethyl-1,3-thiazol-2-yl)ethanone (5-cyanopyrazine-2-carbonyl)-[3-fluoro-4-(2H-tetrazol-5-ylmethoxyiminomethyl)phenyl]azanium 3-[4-(methoxymethyl)phenyl]sulfonylpyridine 2-[6-(7-chloro-1H-indole-4-carbonyl)oxan-3-yl]acetamide 3-[(Z)-1,2-diphenylbut-1-enyl]iminopropanamide 2-[5-(4-fluorophenyl)-1H-pyrazol-3-yl]-3-[2-methoxyethyl(methyl)amino]quinoxaline-6-carboxylic acid 5-hydroxy-1-methyl-N',4-diphenylpyrazole-3-carbohydrazide 2-[1,4-bis(cyclopropylmethoxy)cyclohexa-2,4-dien-1-yl]-N,N-dimethylpyridin-3-amine 4-(4,6-diphenylpyrimidin-2-yl)-3-methoxybenzonitrile (4S)-1,4-bis[(6-chloropyridin-3-yl)methoxy]-5,5-difluoropentan-2-one (3R)-N-cyclopropyl-1-ethenylpyrrolidin-3-amine;methanol;2,4,5-trifluoro-N-[1-oxo-7-[3-(trifluoromethoxy)phenyl]isoquinolin-2-yl]benzamide 2,3-dibromo-5-(4-chlorophenyl)sulfanyl-1H-pyrrole N'-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enoyl]pyridine-2-carbohydrazide (2Z)-N',3-dimethyl-5-(1H-pyrazol-4-yl)penta-2,4-dienimidamide 3-[1-(4-oxochromene-2-carbonyl)pyrrolidin-2-yl]propanenitrile (E)-2,4-dimethylpent-3-enoic acid;ethane;formaldehyde;N'-(1,4,5-trimethylimidazol-2-yl)prop-2-yne-1,3-diamine 2-[(4E)-4-[(3Z,5Z)-3-ethenylocta-3,5,7-trienylidene]-5H-1,3-oxazol-2-yl]ethane-1,1-dithiol 2-(1H-indol-3-yl)-2,5-diphenylpentanoic acid (5S)-2,3-dimethoxybicyclo[9.4.0]pentadeca-1(15),11,13-triene 2-tert-butyl-4-[(7-cyclopropyliminopyrazolo[1,5-a]pyrimidin-3-ylidene)methyl]-6-iodophenol 4-[6-amino-5-[1-(2,3-difluorophenyl)propan-2-yl]pyridazin-3-yl]-N-(2,3-dihydro-1H-isoindol-5-yl)pyrimidin-2-amine (2R)-2-[[4-methoxy-6-(methylamino)pyrimidine-5-carbonyl]amino]pentanedioic acid 2,6-diethyl-4-[(3S)-pyrrolidin-3-yl]pyridine;dihydrochloride 5-amino-6-[4,5-dibromo-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-N-phenylsulfanylpyridine-2-carboxamide N-[2-(4,5-diethyl-6-oxo-1H-pyrimidin-2-yl)-5-(furan-2-ylmethylsulfamoyl)pyrazol-3-yl]cyclopentanecarboxamide 2-hydroxypropanedioate;1-(4-methoxyphenyl)-3,5-bis[3-(trifluoromethyl)phenyl]pyrazole 1-(1,2-dichlorocyclohexyl)-3-phenylthiourea 2-[(5S)-5-azido-3,6-dimethyloctyl]furan 2-(7-fluoro-3,4-dihydro-1H-isoquinoline-2-carbonyl)benzamide N-[4-chloro-2-(ethylamino)phenyl]-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxamide;dihydrochloride N'-hydroxy-5,6-dimethyl-3-[(1S)-1-phenylethoxy]pyridazine-4-carboximidamide 3-[(2R)-1,4-dimethylpiperazin-2-yl]aniline 1-(disulfanylmethoxy)-2,6-dinitronaphthalene 3-cyclohexa-1,5-dien-3-yn-1-yl-6-fluorophenanthridine N-(2,6-dichlorophenyl)prop-1-ene-2-sulfonamide 4-[3-(aminomethyl)phenyl]-N,6-dimethoxypyrimidin-2-amine 1-[4,6-dimethoxy-2-(3-phenyl-2H-triazolo[4,5-b]pyridin-5-yl)pyrimidin-5-yl]ethanone N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-[2-chloro-6-fluoro-4-(methylamino)phenyl]-4-methylcyclohexa-2,4-diene-1-carboxamide N-[2-(3-chlorophenyl)ethyl]-4,5-dimethylpyrimidin-2-amine 2-(5,6-difluorobenzimidazol-1-yl)-N'-hydroxyethanimidamide N-butan-2-yl-5,7-dimethoxy-3H-indole-4-carboxamide N-(2,6-dichloro-4-nitrophenyl)-2,4,6-trimethyl-N-propylbenzenesulfonamide N-[(E)-1H-indol-3-ylmethylideneamino]-2-oxo-1,3,4,5-tetrahydrochromeno[4,3-b]pyridine-10-carboxamide 7-methoxy-3-[3-(1,2,3,4-tetrahydroisoquinolin-8-yl)propanoyl]chromen-2-one 6-[(4,5-dichlorothiophene-2-carbonyl)amino]hexanoic acid 1-amino-5,7-dichlorophthalazine-4-carboxylic acid (5S)-3,4-dimethyl-7-oxo-6-[(Z)-pent-2-en-3-yl]-1-azabicyclo[3.2.0]heptane-2-carboxylic acid 1-(4-fluorophenyl)-2-methoxy-7,8,9-trihydrocyclohepta[d]pyrimidine-4-thione 2-[4-(azepan-1-ylsulfonyl)-N-hexanoylanilino]acetic acid 5-[(3-chlorophenyl)methylimino]-4-(6-fluoroquinolin-2-yl)pyrazolidine-1,4-dicarbonitrile N-[3,5-dichloro-4-(6-oxo-1H-pyridine-2-carbonyl)phenyl]propanamide 7-[(4E)-5-iminohepta-1,4-dien-3-yl]oxy-N-(2-methoxyethyl)-2,3-dihydrothieno[3,4-b][1,4]dioxine-6-carboxamide (1S)-2-[2,4-bis(phenylmethoxycarbonyl)phenyl]cyclopropane-1-carboxylic acid 2-bromo-1-(5,6,7,8-tetrahydronaphthalen-1-yl)ethanone 3-(4,6-dihydropyrrolo[3,4-c]pyrazole-1-carbonyl)piperidine-2,6-dione 2-[4-[1,3-benzoxazol-2-yl-(2,5-dimethoxyphenyl)sulfonylamino]naphthalen-1-yl]oxyacetamide 5-[(3,4-dimethoxyphenyl)diazenyl]-1H-imidazole-2-carboxamide (2-azido-1,3-thiazol-4-yl)-morpholin-4-ylmethanone N-[2,4-difluoro-3-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)phenyl]-2,5-dimethylpyrazole-3-sulfonamide (4S)-4-azido-1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidin-2-one 6,7-bis(3-chlorophenyl)-10H-phenoxazine;ethane N-[4-(cycloheptanecarbonylamino)phenyl]benzamide 4-[(6E)-5,7-dimethylideneocta-6,8-dienoxy]-2-phenylbenzaldehyde N-ethyl-6-methoxy-2-phenylpyrimidine-4-carboxamide 3-(2,4-difluorophenyl)propyl-(7H-purin-6-yl)azanide 7-[(4-bromophenyl)sulfonylamino]-N'-hydroxyimidazo[1,2-a]pyridine-2-carboximidamide 3-(5,7-dimethyl-4,6-dihydropyrazolo[1,5-a]pyrazine-2-carbonyl)-1H-pyridin-2-one 2-[5,6-dibromo-3-(4-chlorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]propan-2-ol;ethane N-benzyl-1-(3,4-dihydroxybenzoyl)piperidine-4-carboxamide 1-(4-chlorophenyl)-5,6-difluoro-2-oxopyridine-3-carboxylate 2-cyclopropyl-1-(4,7-difluoro-6-methoxyquinolin-3-yl)ethanone 5-fluoro-3,4,7-trimethylchromen-2-one 2-(1-azidonaphthalen-2-yl)oxypyridine N-[(3,4-dichlorophenyl)methyl]-9-hydroxy-1,8-dioxo-2-propan-2-ylpyrido[1,2-a]pyrazine-7-carboxamide N-[3-methylbut-2-enyl(propyl)amino]benzamide 4-[2-amino-4-(trifluoromethyl)phenyl]aniline;dihydrochloride N-[3-(2,4-difluorophenyl)prop-1-en-2-yl]-5-[5-methyl-6-[(4-pyridin-3-ylpyrimidin-2-yl)amino]pyridin-3-yl]-1H-pyrrole-2-carboxamide 1-[2,6-di(propan-2-yl)phenyl]-3-[4-[3-(methoxymethyl)-2H-pyridin-5-ylidene]piperidine-1-carbonyl]urea 1-(2,5-dimethylphenyl)-4-[[5-(3-fluorophenoxy)-4H-1,2,3-benzotriazin-3-yl]amino]piperidin-2-one 3-[N-(1,3-thiazol-5-yl)anilino]butanoic acid 7-azidosulfanyl-3,4-dimethoxyquinoline 2-N,7a-dimethyl-2,4,8,9,10-pentazatetracyclo[11.4.0.03,8.015,20]henicosa-1(21),3(8),4,6,16,18-hexaene-2,11-diamine 4-[(3S,4R)-1-(2-ethylpyrazole-3-carbonyl)-4-methoxypyrrolidin-3-yl]-1H-pyrimidin-6-one 5-[4-amino-3-(6-phenoxypyridine-2-carboximidoyl)phenyl]-N,N-dimethylpyridin-3-amine 2-(2,4-dimethylanilino)-N'-hydroxypyrimidine-5-carboximidamide 2-hydroxy-3-(methylamino)naphthalene-1,4-disulfonic acid;hydrochloride 3-[4-(2,6-difluoro-4-heptoxyphenyl)cyclohexyl]-1,2,8-trifluoro-7-propylnaphthalene 5-[4-(diethoxymethyl)phenoxy]-1H-pyrazole N-[(5Z)-5-(furan-2-ylmethylidene)-4,8-dioxo-6,7-dihydro-5H-1,3,6-benzotriazepin-3-yl]furan-2-carboxamide (3R,4S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]-4-[4-fluoro-2-(trifluoromethoxy)phenyl]pyrrolidine-3-carboxylic acid 2-amino-5-[4-(difluoromethyl)pyridin-3-yl]-N-(5-hydroxypentan-2-ylidene)benzamide (7S)-5-methyl-2-[4-(trifluoromethoxy)phenyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine 1-methylsulfonyl-3-[(2,4,5-trichlorophenyl)methyl]urea 2-tert-butyl-5-chloro-N'-[(1S)-1-cyclohexylethyl]-3-methoxybenzenecarboximidamide 4-azido-N,2-diphenylaniline N-[(E)-butylideneamino]-4-[(1Z)-1-methylsulfanylbuta-1,3-dienyl]benzamide (2S,3R)-2-amino-3-[4-[[1-cyclohexyl-5-[difluoro(iodo)methyl]pyrazole-3-carbonyl]-[[4-(2-phenylethynyl)pyridin-3-yl]methyl]amino]phenyl]butanoic acid 2-[4-(6-methoxypyridin-3-yl)-2,5-dioxoimidazolidin-1-yl]acetic acid 1-[4,5-bis(ethenyl)-6-methylpyridin-3-yl]propan-2-one N-[(3S)-1-(cyclopropanecarbonyl)pyrrolidin-3-yl]-7-fluoro-2-[6-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-3H-benzimidazole-5-carboxamide (5S)-2-[(3R,5R)-3,4,5-trihydroxyhexyl]isoindole-1,3-dione N-[5-(dimethylamino)pentyl]formamide;1-ethoxy-2-[2-(4-fluorophenyl)propan-2-ylamino]-3-nitrobenzene 2-(4,5-dimethyl-1H-pyrazole-3-carbonyl)oxyethanesulfonate 2-(azetidin-1-yl)-3,5,6-trifluoro-4-[3-hydroxy-2-oxo-4-[6-(1H-pyrazol-5-yl)pyridine-2-carboximidoyl]pentoxy]benzonitrile 3-(2,6-dimethylpyridin-4-yl)-7-[1-(4-methoxyphenyl)sulfanylpiperidin-3-yl]-5H-pyrrolo[3,2-f]purine 3-[3-oxobutyl(prop-2-enylamino)amino]benzoic acid 5-bromo-4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-N-[3-methoxy-4-(4-methylpiperazin-1-yl)phenyl]pyrimidine-2,4-diamine (2R,4S)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-3,3,4-trihydroxy-2-(methoxymethyl)pyrrolidine-1-carboxamide [2-(azidomethyl)pyrrolidin-1-yl]-(4,6-difluorocyclohexa-1,3-dien-1-yl)methanone 6-(diethylaminomethyl)-7,8-dihydroimidazo[1,2-a]pyrimidin-5-one (2S)-4-methyl-N-[3-(trifluoromethoxy)phenyl]piperidine-2-carboxamide 4-[6-(1,3-benzodioxol-5-yl)pyridin-2-yl]oxybutanoic acid 2-[3-(4-aminophenyl)imidazo[1,2-b]pyridazin-7-yl]oxyacetic acid 2-(4-acetyl-N-prop-2-enoylanilino)-5-methoxybenzoic acid N-[4-(5-aminopentyl)phenyl]-2,3-dichlorobenzenesulfonamide 5-chloro-3-[(4R)-1-ethyl-6-oxo-4-phenylazepane-2-carbonyl]-7,8-dihydro-6H-cyclopenta[b]naphthalen-2-one N-methyl-2,6-di(pyrazol-1-yl)pyridine-4-carbothioamide N-azido-1-(cyclopropylmethoxy)-N-phenylcyclohexane-1-carboxamide 2-amino-6-borono-4-[3,4-dimethoxy-5-(methoxymethyl)phenyl]-4H-pyran-3-carboxylic acid 2-methyl-5-[5-(trifluoromethyl)pyridin-3-yl]pyrazole-3-carboxylic acid 2-(9H-fluoren-1-yl)-4,5-dihydrobenzo[e]azulene (3R,4S)-3-amino-1-[6-fluoro-2-(1,1,2,2,2-pentadeuterioethoxy)quinolin-4-yl]piperidine-4-carboxylic acid 2-[3,4-bis(3,5-ditert-butylphenyl)phenyl]-4-methyl-6-methylidene-1H-pyrimidine ethane;2-[1-(8H-pyrido[3,4-b]pyrazin-7-yl)pyrrolidin-2-yl]acetonitrile 3-(6-aminopyridin-1-ium-3-yl)-2,4-difluorobenzenesulfonamide 3-amino-4-cyano-5-(2,3-dichlorophenyl)-1H-pyrrole-2-carboxamide ethane;methanol;1-methoxy-2,4-dinitrobenzene;6-(piperidine-1-carbonyl)-3H-quinazolin-4-one ethane;2-N-[1-(4-methylpiperazin-1-yl)ethylideneamino]-4-N,5-diphenylpyrimidine-2,4-diamine [5-amino-1,3-bis(2,6-dichlorophenyl)pyrazol-4-yl]-(5-chloro-1H-indol-2-yl)methanone 1-[4-[3,5-bis(trifluoromethyl)phenyl]cyclohexa-2,4-dien-1-ylidene]butane-2-thione 6-[3,4-bis(phenylmethoxy)phenyl]-2-hydroxy-9H-fluorene-1,7-dicarbonitrile 6-[(3S)-1-[3-chloro-4-(4-fluorophenyl)butanoyl]piperidin-3-yl]oxypyridine-3-carbonitrile 2-chloro-4-(3,5-dimethoxyphenyl)quinazoline N-[1-[2-(dimethylamino)-2-oxoethyl]piperidin-4-yl]-5,6-dimethoxypyridine-3-carboxamide 2-(3,5-difluoro-4-hydroxyphenyl)-N'-[[(1S)-2-methyl-1-(1H-pyrazol-4-yl)propyl]amino]ethanimidamide N-[(3,5-dichloropyridin-2-yl)methylidene]hydroxylamine 2-[5-(3,5-ditert-butylphenyl)tetrazol-1-yl]-6-nitrophenol N-(1-butanoylpiperidin-4-yl)-5-methoxy-2-propan-2-ylidene-3H-indene-1-carboxamide 2,5-bis(3-chloropropoxy)-1H-indole N-ethyl-3,5-difluoro-4-[6-fluoro-2-methoxy-7-(trifluoromethoxy)benzimidazol-1-yl]pyridine-2-carboxamide 4-[(3-methylphenyl)sulfonylamino]-N-pyridin-2-ylbenzamide 3-(3,4-dihydro-2H-chromen-6-yl)-1-[(1S)-8-fluoro-7-methoxy-5-methyl-3,4-dihydro-1H-isoquinolin-2-yl]propan-1-one 4-[4-(2,3-dihydropyridin-6-yl)phenyl]piperidine N-[5-bromo-2-oxo-3-[2-(trifluoromethoxy)phenyl]pentyl]acetamide 1-[(2S)-6-[[5-chloro-4-(methylamino)pyrimidin-2-yl]amino]-2,3,4a,9b-tetrahydroindeno[2,1-b][1,4]dioxin-8-yl]ethanone N-(2,3,4,5,6,7-hexahydroazepin-1-ylmethyl)-1-methyl-4-pyridin-2-yloxypiperidine-4-carboxamide 3-[3-(3,4-dimethoxyphenyl)propyl]benzoic acid N-(4-cyanophenyl)-3,5-dimethylpiperidine-1-sulfonamide 3-(2,4-dichlorophenyl)sulfanylpropan-1-amine N-ethyl-4,8-dimethoxy-1H-quinoline-2-carboxamide (5S)-1-[4-[(4-azidophenyl)methyl]piperazin-1-yl]-5-(3,4-dihydro-2H-quinolin-1-yl)-3-(propylamino)hexan-1-one 2-(2-methylphenyl)-6,7-dihydrothieno[3,2-b]pyridine 2-[4-[2-(oxolane-3-carbonylamino)ethylcarbamoyl]phenoxy]acetic acid 1-[(4,5-diphenylfuran-2-yl)methylideneamino]-3-(1H-indol-7-yloxymethyl)naphthalene-2-carboxylic acid 2-[(4R,5S)-1-methyl-3-pyridin-3-yl-6,7-dihydro-4H-pyrano[4,3-c]pyrazol-4-yl]phenol 7-[(2,6-difluorophenyl)methoxy]-1H-quinolin-2-one 3-[2-chloro-4-(4-oxo-7,8-dihydro-6H-pyrido[1,2-a]pyrimidine-2-carbonyl)phenyl]propanamide 2-[3-(5,6-difluoro-1H-benzimidazol-2-yl)phenyl]-N'-hydroxy-6-nitrobenzenecarboximidamide 4-cyclopropylsulfonyl-6-[4-(3,5-dimethylphenyl)piperazine-1-carbonyl]pyridine-2-carboxamide 6-(3,4-dichlorophenyl)hexanoic acid;hydrochloride (3R,4S)-5-[1-amino-2-(3,5-difluorophenyl)ethyl]-N'-[3,3-bis(trifluoromethyl)cyclobutyl]-3-hydroxy-4-methoxypentanehydrazide 2-methyl-4-[(2S)-1-[4-(3-oxobutanoylamino)benzoyl]piperidin-2-yl]-N-phenylpyridine-3-carboxamide N-[2-methoxy-4-(trifluoromethyl)phenyl]pyridine-3-carboxamide 7-[2-chloro-4-(1-hydroxycyclopropyl)phenyl]-8a-ethyl-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-1,3-dione 2-ethyl-4-[3-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazine-1-carbonyl]-2H-isoquinolin-1-one 3-butyl-N-ethenoxy-2,4,6-trimethylaniline N-(4-chloro-2-methoxyphenyl)pyrimidine-5-carboxamide 2-[[1-(furan-3-ylmethyl)piperidin-4-ylidene]amino]oxy-N,N-dimethylethanamine 6-(2-aminophenyl)sulfanyl-N',3-dihydroxy-2H-indazole-4-carboximidamide (2S,3R)-N-[3-chloro-4-[4-[1-methyl-6-oxo-5-[[[2-(oxetan-3-ylamino)ethylamino]methyl]pyridine-3-carbonyl]pyridazin-3-yl]butyl]phenyl]-2-fluoro-3-hydroxyhexanamide [3-(dimethylamino)azetidin-1-yl]-[6-methoxy-2-methyl-4-(1H-pyrazol-5-yl)phenyl]methanone 2-(6-chloroimidazo[1,5-a]pyridin-3-yl)-N-methyl-7H-purin-6-amine 4-[2,6-dimethyl-3-(5-propanoyloxy-1H-indole-2-carbonyl)phenyl]benzoic acid [3-[(4-chlorophenyl)methyl]thiophen-2-yl]boronic acid 3-[6,7-dimethoxy-4-(2-morpholin-4-ylethyl)-1-oxoisoquinolin-2-yl]piperidine-2,6-dione 4-[6-(1,3-benzothiazol-5-yl)imidazo[1,2-a]pyrazin-8-yl]phenol 2-(4-aminocyclohexyl)-3-[ethoxy(propan-2-yloxy)methyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one N-butyl-2-chloro-5-fluoropyrimidine-4-carboxamide 2-(3,5-dichlorophenyl)sulfanyl-1-[(4S,6R)-6-methyl-6-[4-[4-(trifluoromethoxy)phenoxy]phenyl]-3-azabicyclo[3.1.0]hexan-3-yl]ethanone 5-[6-(2-ethoxypyridin-3-yl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-yl]-N-propan-2-yl-1H-pyrazole-4-carboxamide 2-tert-butyl-6,7,8,9-tetrahydropyrido[2,3-b]azepine 2-[(2Z,5S)-4-oxo-2-[(E)-(3,4,5-trimethoxyphenyl)methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid N-methyl-1,3-diphenylbutane-1,4-diamine 5-[(2-cyclopropylacetyl)amino]-3-methyl-4-[1,3,3-trimethyl-6-(oxan-2-yloxy)indol-2-ylidene]pentanoic acid 3-[(E)-1-naphthalen-2-ylpent-1-enoxy]-4-(trifluoromethylsulfanylamino)benzoic acid N-cyclopentyl-2-[5-(4-methoxyphenyl)spiro[1,3-dihydroindene-2,3'-piperidine]-1'-yl]acetamide;ethane 4-[4,7-dimethoxy-6-[3-[(4-methylphenyl)sulfonylamino]naphthalen-1-yl]naphthalen-2-yl]butanoic acid 3-bromo-N'-[(2Z,4E)-7-ethyl-2-methylhepta-2,4-dienyl]benzenecarboximidamide 2-[(2S)-5-(3-chlorophenyl)-1,4-dioxan-2-yl]-N,N-dimethylethanamine;hydrochloride 2-(3-azidopropyl)-1,4,7,8-tetramethoxynaphthalene 3-(4-acetamidophenoxy)-N-[2-[(5R)-7-chloro-10-fluoro-1,4-diazatricyclo[6.4.0.02,6]dodeca-2(6),8,11-trien-12-yl]ethyl]propanamide 2-(2,3-dihydro-1H-inden-5-yloxy)-N-[4-[2-[[6-oxo-3-(trifluoromethyl)pyridazin-1-yl]methyl]cyclobuten-1-yl]phenyl]acetamide N'-methyl-4-(pyridine-3-carbonylamino)benzohydrazide 3-[4-(1H-indol-2-yl)-2-methoxyphenyl]cyclobutan-1-ol 2-amino-6-[1-(4-aminobenzoyl)piperidin-3-yl]oxypyridine-4-carbonitrile 2-[3,5-bis(trifluoromethyl)phenyl]sulfanyl-N-(2-chloroethyl)aniline 3-[1-azido-3-(4-methylphenyl)but-2-enyl]cyclopentan-1-ol [(3Z)-3-(methylideneamino)-5,6-dihydro-2H-1,4-benzothiazocin-8-yl]-morpholin-4-ylmethanone 1-butylanthracene 1-(4-bromophenyl)cyclohexa-2,4-dien-1-amine (6S)-7-acetyl-3-ethylsulfanyl-6-pyridin-1-ium-4-yl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 2-[4,6-bis(methylamino)pyrimidin-5-yl]propanamide 1-[4-(6-azidopyrimidin-4-yl)piperazin-1-yl]ethanone N-[(6S)-8-oxo-5,6-dihydroimidazo[2,1-b][1,3]thiazine-6-yl]acetamide [3-amino-4-(2-methylpyridin-4-yl)pyrrolidin-1-yl]-[2-(1H-pyrazol-5-yl)phenyl]methanone 2-[(1-methyltetrazol-5-yl)amino]ethanesulfonic acid 2-[(1S)-2-methylcyclohexanecarbonyl]oxybenzoic acid 7-[5-methyl-3,6-bis(2-propan-2-yloxyethoxy)pyridine-2-carbonyl]furo[3,2-c]pyridine-4-carboxamide N'-hydroxy-3-pyridin-2-ylsulfanylpyridine-4-carboximidamide [(1S)-3-hydroxycyclopentyl]-(4-piperazin-1-ylpiperidin-1-yl)methanone N-(4,6-dimethylpyrimidin-2-yl)-4-[(2-phenylpyrazol-3-yl)sulfamoyl]benzamide 3-cyclopentyl-5-[(1R,2R)-2-methoxycyclohexyl]-8-pentan-3-ylsulfanylpyrimido[4,5-b][1,4]thiazine-6,7-dione (5Z)-5-[[2-[4-(ethylaminomethoxy)-3-fluorophenyl]sulfanylphenyl]methylidene]imidazolidine-2,4-dione 2-(6-tert-butylpyridin-3-yl)-N-[1-(2,4-difluorophenyl)ethyl]acetamide 2-[5-carbamoyl-9-[(3,4-dimethoxyphenyl)methyl]-2-propan-2-ylcarbazol-4-yl]peroxyacetic acid 1-(4-butoxybenzoyl)-6,7-dihydro-5H-indolizine-3-carbonitrile 2-(4,4-dimethylcyclohexen-1-yl)oxy-N'-hydroxypyridine-4-carboximidamide 4-[(2,5-dimethyl-1H-imidazol-4-yl)sulfonyl]-7-methoxy-8a-methyl-1,3,4a,6,7,8-hexahydroquinoxaline-2,5-dione (4-propylcyclohexa-1,5-dien-1-yl)oxybenzene 4-[3-chloro-5-[(2S)-1,1,1-trifluoropropan-2-yl]oxyphenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 4-[(4-cyclopropylpyridine-2-carbonyl)amino]butanoic acid 6,7-dimethoxy-1-[2-methylsulfanyl-4-(trifluoromethyl)phenyl]phthalazine 6-[(2E)-1,1-bis(4-methoxyphenyl)penta-2,4-dienyl]-7H-purine 2-[(1S)-2-methylcyclopropyl]-4H-3,1-benzoxazine N-(1,3-benzodioxol-5-ylmethyl)-2-[(6S)-5-hydroxy-4,8-dioxo-6-phenylpyrano[3,4-f]chromen-9-yl]acetamide (2Z,4E)-2-[5-chloro-2-ethoxy-4-(3-methylsulfonylpropoxy)phenyl]-6-methylidene-N-(4-pyridin-4-ylpiperazin-1-yl)octa-2,4,7-trienamide 2-[4-[2-fluoro-6-(trifluoromethyl)phenyl]phenyl]acetamide (1E,4E)-1-chloro-5-(3-methoxyphenyl)penta-1,4-dien-3-one (2S)-2-[9H-fluoren-1-ylmethoxycarbonyl(trifluoromethyl)amino]propanoic acid 4-bromo-2-fluoro-1,5-dimethyl-3-propan-2-ylbenzene 2-bromo-3,4-bis(phenylmethoxy)phenol 6-bromo-N-methylnaphthalene-2-carboxamide;1,2,3-trifluorobenzene N-(2,3-dihydro-1H-pyrrolo[1,2-a]indol-4-yl)benzenesulfonamide 1-(azidomethyl)-4-(4-phenoxyphenyl)piperazine 4-(diethylamino)-2-[7-ethyl-1'-[[3-fluoro-2-(trifluoromethoxy)phenyl]methyl]spiro[2H-indole-3,2'-pyrrolidine]-5-yl]benzamide;hydrochloride N-[4-[(3R,5S)-3-amino-5-methylpiperidin-1-yl]pyridin-2-yl]-8-(difluoromethyl)quinoline-4-carboxamide 1-(2-ethoxyethyl)-3-[6-(5-fluoropyridin-3-yl)-4-(3H-imidazo[4,5-c]pyridin-2-yl)pyridin-2-yl]imidazolidin-2-one 2-[(E)-2-phenylethenyl]-1,3,4,5-tetrahydropyrido[4,3-b]indole 4-(5,7-dioxopyrano[3,2-c]chromen-2-yl)benzaldehyde 4-[2,6-di(propan-2-yl)anilino]isoindole-1,3-dione 3-(4,6-dimethylquinolin-2-yl)phenol 5-[(2-ethoxyphenyl)diazenyl]-3H-1,3,4-oxadiazol-2-one N-[6-(N-amino-2,3-dimethylanilino)pyrimidin-4-yl]-2-piperazin-1-ylacetamide (3-iodo-2,4,5-trimethylphenyl)boronic acid N-cyclopropylsulfonyl-4-[(2Z,5E)-3-methylideneocta-1,6-dien-2-yl]oxybenzamide (2S,3R)-5-[4-(1-benzofuran-2-yl)piperidin-1-yl]-N'-hydroxy-2-propan-2-yl-2-pyridin-2-ylpentanediamide 3-[4-(3,4-dihydropyridin-2-yl)-1H-benzimidazol-2-yl]-5-(5-methylthiophen-2-yl)-1H-pyrazolo[3,4-c]pyridine 4-(2-chlorophenyl)-N-[2-methyl-1-[3-[methyl(piperidine-4-carbonyl)amino]propyl]indol-5-yl]piperazine-1-carboxamide 2-(3,4-dichlorophenyl)cyclohexa-1,5-dien-1-ol 2-(6-butyl-3,4-difluoro-5-phenylmethoxypyridine-2-carbonyl)cyclohexane-1,3-dione 3-(4-butan-2-yloxybutoxy)carbonylbenzoate 2-methyl-N-[4-[1-(methylamino)ethenyl]phenyl]butanamide 3-[2,6-dichloro-4-nitro-N-(1,3-thiazol-5-yl)anilino]butanoic acid N-(6-bromo-2,3-dihydroimidazo[1,2-b]pyrazol-1-yl)benzamide 4-azidooxy-6,8-dichloro-3,7-dimethylquinazoline 2-[(5R,10bS)-9-chloro-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 4-[5-[[(3R,6R)-2,6-dimethylmorpholine-4-carbonyl]amino]pyridin-2-yl]piperazine-1-carboxylic acid 1-(4-chlorophenyl)sulfonyl-4,5,7,8-tetrahydrooxepino[4,5-d]imidazole;hydrochloride 2-methyl-N,5-diphenyltriazolo[4,5-d]pyrimidine-3-carboxamide N'-tert-butyl-4-(9H-fluoren-9-ylmethoxycarbonylamino)-1,2,5-oxadiazole-3-carboximidamide 1-(1,2,3,4-tetrahydroquinolin-5-ylmethyl)piperidine-3,4-diol 3-[4-chloro-5-(2,6-difluorophenyl)pyrimidin-2-yl]-N'-iodobenzenecarboximidamide 5-chloro-N'-hydroxy-3-[2-methoxyethyl(4,4,4-trifluorobutanoyl)amino]pyridine-2-carboximidamide 4-[4-(2,6-diphenylpyridine-4-carbonyl)piperazin-1-yl]benzaldehyde 2-[5-fluoro-3-(2-methoxyquinolin-6-yl)pyridin-4-yl]acetaldehyde 1-[(2S)-4,5-bis(phenylmethoxy)pentan-2-yl]piperidine (2R)-3-azido-5,7-difluoro-N,2-dimethyl-2H-1,4-benzothiazin-6-amine 2-(3,4-dimethoxyphenyl)-1-[5-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]ethanone (Z)-1,3-bis[5-tert-butyl-2-(3-chloro-4-fluorophenyl)pyrazol-3-yl]prop-2-en-1-one 2-azido-4,5,6-trimethylindazole [4-hydroxy-3,5-di(propan-2-yl)phenyl]phosphonic acid 1-(4-fluorophenoxy)butane-2-thiol 2-azidosulfanylquinoline 6-[2,5-dichloro-4-(ethylamino)phenyl]imino-1H-pyrrolo[3,4-c]pyrrol-7-one (E)-2,3-bis[(4-butyl-3-hydroxyphenoxy)methoxy]prop-1-en-1-olate;nickel(2+) 2-[1,1,1,2,3,3,4,4,5,6,7,8,9,9,10,11-heptadecafluoro-2-(trifluoromethyl)nonoxy]benzenesulfonic acid N'-[amino(methyl)amino]-3-[2,4-difluoro-5-(6-propan-2-ylpyrimidin-4-yl)phenyl]benzenecarboximidamide 4-(3,5-dibromo-2,6-dihydroxyphenyl)-8-methyl-1-methylidenequinolin-2-one N-[(2R)-4-hydroxy-4-methylhexan-2-yl]pyridine-3-carboxamide 7-chloro-5-[5-fluoro-2-(oxolan-3-yl)phenyl]spiro[1H-indole-3,4'-piperidine]-2-one 2-(2,3-dihydrobenzo[g][1]benzofuran-7-yl)acetamide 5-butyl-2-phenyl-1,3,4-oxadiazole 4-(4,6-diphenyl-1,3,5-triazin-2-yl)-11H-benzo[a]carbazole N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-ylmethyl)azepane-1-carboxamide 3-[2-(2,6-dichloro-3,5-dimethoxyphenyl)ethyl]-1-[1-(methylamino)piperidin-4-yl]-2H-pyrazolo[4,3-d]pyrimidin-8-amine 1-(3,5-dimethylphenyl)sulfonylpyrrole 1-N,3-N-dimethyl-4-(8-methyl-2H-quinoline-1-carbonyl)benzene-1,3-dicarboxamide;ethane 4-N-(4,5-dimethylpyrimidin-2-yl)benzene-1,4-disulfonamide 4-[(2R)-4-(1,3-benzothiazol-6-ylamino)-5-(methanesulfonamidomethoxy)-5-oxopentan-2-yl]oxybenzenecarboximidamide 2-amino-6-[(3S,5R)-1-(cyclohexylmethoxy)-5-pyridin-4-ylpyrrolidin-3-yl]-3H-pteridin-4-one 3-cyclobutyl-5,6-dimethyl-7H-purine-2,8-dione 1-[[4-[[3-(2,6-dichlorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]methoxy]cyclohexa-1,3-dien-1-yl]carbamoyl]piperidine-4-carboxylic acid 6-(8,10-dioxo-2,3,4a,5,6,7,11b-octahydrobenzo[a]quinolizine-1-carbonyl)pyridine-3-carbonitrile (2S)-6-[[1-(4-aminobenzoyl)pyrrolidin-3-ylidene]amino]-5-oxohexane-2-sulfonic acid 3-[2-(1H-indol-3-yl)ethenyl]-5-phenyl-1H-pyrazole-4-carbonitrile 3-[1-(4-chlorophenyl)sulfonylpiperidin-2-yl]pyridine 4-methyl-N-[3-(1,2,4-triazol-1-yl)propyl]pyridine-3-carboxamide 2-N-[4-(1,4-dioxan-2-ylmethoxy)phenyl]-5-ethylpyrimidine-2,4-diamine 3-[(1S)-1-(4-acetamidophenyl)ethyl]-5-(4-fluorophenyl)imidazole-2,4-dicarboxamide 2-(N-ethylsulfonyl-4,5-dimethyl-2-phenyldiazenylanilino)acetamide N-[4-(4-cyanophenyl)phenyl]-6,7-diethoxyquinazoline-4-carboxamide 4-(4-azidophenyl)-N,N-dimethylaniline (1Z,3E)-4-[4-amino-2-methyl-5-(trifluoromethyl)pyrazol-3-yl]buta-1,3-diene-1,4-diamine 2-[4-[(3,4-dimethoxyphenyl)methylamino]-6-propan-2-yl-1H-benzimidazol-5-yl]acetamide (7S)-2-[4-chloro-3-(trifluoromethyl)phenyl]-N-[3-(1,1-difluoropropyl)phenyl]-5-oxo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide N-[4-(1H-benzimidazol-2-yl)phenyl]-5-ethoxy-1,3-diphenylpyrazole-4-carboxamide 1-[4-(2,3-dihydropyrrol-1-yl)phenyl]-4-methylideneheptan-4-ol 2-[4,5-dimethyl-3-(oxan-3-yl)imidazol-1-ium-1-yl]ethanethiol 2,4-ditert-butylbenzoic acid 4-[1-[(3,5-dichlorophenyl)carbamoyl]cyclopropanecarbonyl]piperazine-1-carboxylic acid 6-[2-[4-[2-(5,6-difluoronaphthalen-2-yl)ethynyl]phenyl]ethyl]-1-fluoro-2-methoxynaphthalene 4-[(8S)-10-[[2,5-difluoro-4-(2-methoxyethylamino)benzoyl]amino]-8-[2-hydroxyethyl(methyl)amino]-1-oxo-6,7-dihydropyrazino[1,2-a]indole-3-carbonyl]piperazine-1-carboxylic acid 5-(6,8-difluoroquinoline-2-carbonyl)-N'-[3-methylbutanoyl(propyl)amino]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-3-carbohydrazide 3-[[2-[4-[[4-(1,5-dimethylpyrazole-3-carbonyl)piperazin-1-yl]methyl]phenyl]acetyl]amino]propanoic acid 3-methyl-2,6-bis(pyridine-4-carbonyl)benzenesulfinic acid 4-[6-(3,5-dichloroanilino)pyrimidin-4-yl]sulfanyl-2-methoxyphenol 6-(4-tert-butylcyclohexen-1-yl)oxychromen-2-one N-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl]butanamide 1-[(2R,6S)-4-hydroxy-3-(trifluoromethylsulfanyl)-5-thia-1-azabicyclo[4.2.0]oct-2-en-2-yl]-3-phenylurea 2-(6-fluoro-4-propan-2-ylcyclohexa-1,5-dien-1-yl)-N'-hydroxypyridine-3-carboximidamide [4-hydroxy-3-(trifluoromethoxy)phenyl]-[2-(quinoline-6-carbonylamino)phenyl]sulfanium 1-[4-(2,3-dimethylcyclopenta-2,4-dien-1-yl)naphthalen-1-yl]ethenol 3-(4-ethenylphenyl)-1,2-oxazole;5-methylheptane 1-[4-[3-(azidomethyl)phenyl]butyl]pyrrolidine 4-[4-methyl-6-(morpholine-3-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]benzamide 4-[(3Z)-3-ethylideneoxolan-2-yl]-1,8-naphthyridine 1-[3-(4,5-difluorocyclohexa-1,5-dien-1-yl)butanoyl]-N-hydroxybenzimidazole-2-carboxamide 6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonylamino)hexanoic acid 6-methyl-1'-(pyridine-4-carbonyl)spiro[5,7-dihydropyrazolo[3,4-d]pyrimidine-4,4'-piperidine]-2-one 3-[N-(2,4-dichloropyrimidin-5-yl)-4-(quinoxalin-2-ylsulfamoyl)anilino]propanoic acid 2-[5-azido-4-(1H-benzimidazol-2-yl)pentoxy]acetic acid N-(5,6-dimethylimidazo[2,1-b][1,3]thiazol-3-yl)-3-oxocyclobutane-1-carboxamide 6-[[1,4-dimethyl-2-(3-nitrophenyl)sulfanyl-5-propoxycarbonylpyrrole-3-carbonyl]amino]pyridine-3-carboxylic acid 2-amino-6-(3-bromoquinolin-7-yl)oxy-N'-propan-2-ylpyridine-4-carboximidamide 2-amino-3-[4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]propanoic acid;hydrochloride N-[4-(3,5-dimethyl-1,2-oxazol-4-yl)phenyl]-2-(4-ethylsulfonylphenoxy)acetamide 4-[3,5-bis(trifluoromethyl)phenyl]-N-[(E)-(2-hydroxynaphthalen-1-yl)methylideneamino]benzamide 5-[3,3-bis(4-fluorophenyl)propyl]-2-propan-2-yloxy-1H-pyrrole 1-[4-(2,6-diethylphenyl)butyl]-3,5-dimethylbenzene 3-[(Z)-N'-[amino-[6-amino-4-chloro-1-methyl-2-oxo-8-[(Z)-prop-2-enylideneamino]quinoline-3-carbonyl]amino]carbamimidoyl]pyrrolidine-1-carboxylic acid N-[1-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)piperidin-3-yl]-2-phenoxyacetamide 2-(N-(2,4-dichloropyrimidin-5-yl)-3-hydroxyanilino)-1-phenylethanone 1-[[5-(3,4-difluorophenyl)-2H-triazolo[4,5-b]pyrazin-7-yl]methylamino]-3-methoxypropan-2-ol (2R)-1-[3,3-dimethylbutanoyl(propyl)amino]-N-[2-hydroxy-4-[5-(4-phenoxyphenyl)pyrimidin-2-yl]oxyheptyl]pyrrolidine-2-carboxamide 2-N,6-dimethyl-4-N-(3-methylhexyl)pyridine-2,4-dicarboxamide 1,1-dimethoxy-2H-naphthalene N-[1-(2,6-dioxopiperidin-3-yl)-3-ethylsulfonylpiperidin-4-yl]-7H-purine-6-carboxamide (5S,7R)-N-(3-chlorophenyl)-7-[2-[(4-methylphenyl)methoxy]phenyl]-5-phenyl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 2-[5,5-dimethyl-3-(1-methylazetidine-2-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]pyridine-4-carboxylic acid (E)-3,4-dichloro-N-[5-(4-fluorophenoxy)pyridin-2-yl]sulfanyl-1,6,7,8-tetrahydroisoquinoline-6-carboxamide;propane N-[5,6-difluoro-3-(4-propylphenyl)-1H-inden-2-yl]pyridine-3-sulfonamide 1-[4-[2-(3-bromopropoxy)ethyl]phenyl]ethanol N-[3-methoxy-4-(7H-purin-6-ylamino)phenyl]-2-phenylacetamide (Z)-3,5-diamino-4-[2-methoxy-5-(trifluoromethyl)phenyl]pent-3-enal 1-phenylsulfanyl-2,3,4,5-tetrahydro-[1]benzothiepino[5,4-c]pyrrole 1-(2,4-dimethoxyphenyl)-5-oxo-N,7-diphenylheptanamide (6-fluoropyridin-3-yl)-[3-methoxy-4-(5H-pyrrolo[2,3-b]pyrazin-2-yl)phenyl]azanide 1-methyl-3-[4-(2,4,6-trichlorophenyl)pyridin-2-yl]indole 4-[(3R)-1-(2,3-dimethylbutanoyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one 3-bromo-1-(1,2-dihydronaphthalen-1-yl)naphthalene N-[1-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]dioxin-8-ylsulfonyl)piperidin-4-yl]benzenesulfonamide N-[[4-(4-chlorophenoxy)cyclohexyl]methylidene]hydroxylamine 4-[(2R)-2-[5-chloro-2-(methylamino)pyrimidin-4-yl]oxolan-3-yl]phenol 5-[1-(4,6-dimethoxypyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-4-carboxylic acid 4-tert-butyl-2-[(5-methoxybenzotriazol-1-yl)imino]-6-methylpyran-3-carbonitrile 4-[(3S)-1,5-dimethylpiperidin-3-yl]-N'-hydroxypyridine-2-carboximidamide (6S)-4-hydroxy-5-phenylmethoxycyclohexa-2,4-dien-1-one [5-bromo-2-(4,5-dimethylpyridine-3-carbonyl)phenyl]iodanium ethane;[3-hydroxy-2-(4-methoxyphenyl)propyl]-trimethylazanium N-(2,6-dimethylphenyl)-1-pyridin-3-yloxycarbonylazetidine-3-carboxamide 2-[3-[4-[(6Z)-7,8-dichloroocta-1,6,8-trienyl]piperazine-1-carbonyl]-5-[4-(ethoxymethyl)piperidin-1-yl]phenoxy]acetaldehyde;2,2,2-trifluoro-N-propan-2-ylacetamide 1-[(5R,10bR)-5-thiophen-2-ylsulfonyl-4,10b-dihydro-3H-[1,2]oxazolo[3,4-b]isoindol-1-yl]propan-1-one N-[3-(dimethylamino)phenyl]-4,5-bis(ethenyl)-1H-imidazole-2-carboxamide N-[(3S)-1-(2,5-difluorophenyl)pyrrolidin-3-yl]-3-methanimidoyl-4-(prop-2-enylideneamino)benzamide;ethane 2-[3-(methoxyamino)phenyl]benzenecarboximidamide 3-[6-methyl-4-(2H-tetrazol-5-yl)cyclohexa-1,3-dien-1-yl]propanamide 2-(4,6-difluorocyclohexa-1,5-dien-3-yn-1-yl)-5-[5-ethoxy-2-methyl-4-(trifluoromethyl)phenyl]-N-(5-hydroxypentan-2-yl)thiophene-3-carboxamide 2-[(4aS)-6-methyl-3,4,4a,5,7,8,8a-octahydro-1H-isoquinoline-2-carbonyl]benzoic acid 3,3-dimethyl-1-(2-methyl-1H-indol-5-yl)pentan-1-one 1,4-dichlorobutane;N-[(3E)-5-phenylhexa-3,5-dienyl]acetamide 2-bromo-N-cyclohexyl-4,6-dimethoxyaniline 5-[2-fluoro-4-(3-methoxypropoxy)phenyl]pyrimidine 2-[1-(1,3-benzoxazol-2-yl)pyrrolidin-3-yl]oxyacetamide N-(2-oxopropyl)benzenesulfonamide 7-fluoro-2,4-dimethylquinoline;5-[(3Z)-hexa-1,3,5-trien-2-yl]oxy-6-hydroxyspiro[1H-indole-3,3'-piperidine]-2-one N-[4,7-bis(3-aminophenyl)-1H-inden-2-yl]cyclohexa-1,5-dien-1-amine 4-[1-[(2S)-2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxybutanoyl]piperidine-4-carbonyl]benzonitrile 2-(4,5-dimethyl-1H-pyrazole-3-carbonyl)cyclopentan-1-one 2-methyl-1-[[3-(pyridin-4-yloxymethyl)oxetan-3-yl]carbamoylamino]cyclohexane-1-carboxamide 2-[4-hydroxybutyl(pyridin-3-yl)amino]-1-phenylethanone 2-[(1R)-1-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]-7-(oxan-4-yl)-3H-imidazo[5,1-f][1,2,4]triazin-4-one 1-(azidomethyl)-2,5-dichloro-3-propan-2-yloxybenzene 2-fluoro-3-methyl-4-nitro-1H-indole 3-(2,6-dibromopyridin-4-yl)oxy-1H-carbazole 2-(1-benzylcyclobutyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine N-[4-(4-azidophenoxy)phenyl]-2,5-dimethoxybenzamide 3-[(3Z)-5-fluorohexa-1,3,5-trien-2-yl]oxy-N'-hydroxypyridazine-4-carboximidamide 3-[6-(2,7-dimethylquinazolin-4-yl)oxynaphthalen-1-yl]-5-(trifluoromethyl)pyridine-2-carbonitrile [5-cyclobutyloxy-2-(trifluoromethyl)-1,3-thiazol-4-yl]methanamine;hydrochloride 3-[1-(4,6-diamino-1,3,5-triazin-2-yl)-2-methoxyindol-3-yl]propanoic acid 2-methyl-4-[4-(5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-3-carbonyl)morpholin-3-yl]-1H-pyrimidin-6-one 1-[(2E,4Z)-hexa-2,4-dien-3-yl]oxycarbonylnaphthalene-2-carboxylic acid 5-[(2Z,4E)-hepta-2,4-dien-4-yl]-3-(4-pyridin-4-yl-1H-indole-2-carboximidoyl)pyridin-2-amine 2-[4-[[4-(1,3,7,8-tetrahydroimidazo[4,5-g]quinazolin-2-ylidene)piperidin-1-yl]methyl]phenoxy]acetonitrile 4-[2-[2,6-dichloro-N-(4-hydroxybutyl)-4-nitroanilino]ethyl]-2-methylbenzenesulfonic acid 4-(5-chloro-1,3-thiazol-2-yl)cyclohexan-1-one 2-(1H-pyrazol-4-yl)-4,5-dihydropyrrolo[3,4-d][1,3]thiazole 2-(4-chloroanilino)-N-[3-(2,6-dioxopiperidin-1-yl)phenyl]acetamide ethane;6-(4-ethylphenoxy)-N,1-dimethylpyridin-2-imine 4-(3-cyclobutylimidazolidin-1-yl)quinoline 3-[4-chlorobutyl(1,2,4-triazol-4-yl)amino]propane-1,2-diol 4-N,6-N-bis[(2-fluorophenyl)methylideneamino]pyrimidine-4,6-diamine 4-(4-amino-3,5-dimethylphenyl)-2,6-dimethylaniline 6-[(3,4-dimethoxyphenyl)methyl]-2-thiophen-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (2S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-1-[2-fluoro-6-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-ylamino)pyrimidin-4-yl]pyrrolidine-2-carboxamide 3-(1,3-benzodioxol-5-yl)-6-chloro-2H-pyrazolo[3,4-c]isoquinoline 3-(4-azidophenyl)-5,6-bis(ethenyl)cyclohexa-2,4-diene-1,1,3-tricarbonitrile 2-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]quinoline-6-carbonitrile 1-[[5-(difluoromethoxy)pyridin-2-yl]methyl]-3,4-dihydro-2H-quinoline N-[1-[2,4-dichloro-3-(difluoromethoxy)phenyl]ethyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide 2-N,5-N-bis(1H-indazol-6-yl)pyridine-2,5-dicarboxamide [2-[(3,5-dimethylpyrazole-1-carbonyl)amino]imidazo[1,2-b]pyridazin-6-yl]boronic acid [2-methylsulfonyl-4-(propanoyloxymethylamino)phenyl]sulfanium 3-[1-(2,6-difluorophenyl)ethoxy]azetidine;hydrochloride 1-[4-(9H-fluoren-9-ylmethoxy)phenyl]-2,2-dimethoxyethanol 7-bromo-6,7a-dihydro-1H-benzo[h]quinazoline N-(6,7-dihydro-4H-furo[3,2-c]pyran-6-yl)-2-hydroxyethanesulfonamide 3-[(1R)-3-methylcyclohexyl]-2-(1H-pyrrolo[3,2-c]pyridin-3-yl)-1,5-naphthyridine 2,6-dichloro-N-[3-(methylamino)phenyl]benzamide;ethane 4-(4-bromophenyl)-2,6-dichlorobenzenethiol 2,3-dimethyl-5,6-bis(1H-pyrazol-4-yl)pyrazine;ethane (5S)-1-[2-(2,4-dichlorophenyl)ethyl]-2,5-dimethoxypiperazine N-(4-bromobutan-2-yl)-3-methoxyaniline 2,4-dichloro-N-methyl-N-[(3S)-piperidin-3-yl]benzamide;hydrochloride 4-[2-(dimethylamino)ethyl]-3,7,8-trihydroxypyrano[2,3-c]quinolin-9-one (3aR,6aS)-5-[4-[2-(2-methoxyphenyl)ethynyl]cyclohexa-1,5-dien-1-yl]-2-(oxan-4-yl)-3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrole 1-(4-hydroxybutyl)-5-phenylcyclohexa-2,4-dien-1-ol N-[3,6-bis(ethenyl)-2H-pyridin-1-yl]-5-chlorothiophen-2-amine [5-chloro-2-(4,6-dimethoxypyrimidin-2-yl)sulfanylphenyl]urea N-[4-(2,3-difluorophenoxy)-3-(4-methylsulfonylphenoxy)phenyl]ethanimine N-[2-methylsulfanyl-1-(5H-pyrrolo[3,2-d]pyrimidin-4-yl)ethylidene]hydroxylamine 6-azidooxy-2,3-difluoro-5-phenylpyridine 2-[3-[(4-cyanophenyl)methyl]imidazol-4-yl]-N-[1-cyclopentyl-3-[(E,2S)-6-oxohex-4-en-2-yl]sulfonylpropan-2-yl]acetamide 1-[2,3,5-trifluoro-4-(2H-tetrazol-5-yl)phenyl]ethanone 4-[(2E,4Z)-5-(but-3-enoxymethyl)hepta-2,4,6-trien-3-yl]aniline;formaldehyde 2-ethyl-N-[1-(1,3-oxazol-4-yl)cyclopropyl]-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide 1-[2,6-di(propan-2-yl)phenyl]sulfanylimidazolidine;gold(1+);triphenylphosphane 2-bromo-6-chloro-N-[(3S)-oxolan-3-yl]pyridine-4-carboxamide 5-hydroxypentanoic acid;2-(3-methylphenyl)-6,7-dihydroquinoline 6-azidooxy-2,3-dihydrothiochromen-4-one N-[6-(2,3-dihydrofuran-4-yl)-3H-inden-1-yl]quinoline-7-carboxamide (5S)-3,8-diethyl-2,2-bis(4-fluorophenyl)-7-(trifluoromethyl)pyrano[3,2-g]chromene (5-fluoropyridin-2-yl)methyl-[6-hydroxy-3-(thiophen-2-ylmethoxycarbonylamino)cyclohexa-1,5-dien-1-yl]-diphenylphosphanium [1-(4-methylcyclohexanecarbonyl)piperidin-3-yl]-phenylmethanone N-butyl-6-hydroxy-N',4-dimethylpyridazine-3-carboximidamide N-[4-[6-[[1-amino-2-(ethylideneamino)-3-oxoprop-2-enyl]amino]imidazo[1,2-a]pyrazin-3-yl]phenyl]methanesulfonamide 2-(2,4,5-trifluorophenyl)-N-[3-(2H-tetrazol-5-yl)phenyl]cyclopropane-1-carboxamide (4S)-2,8-dimethyl-4-[5-(pyridine-3-carbonyl)thiophen-2-yl]-6-sulfanylidene-1,4-dihydro-[1,3]thiazino[3,2-a]benzimidazol-3-one 5-hydroxy-3-[(4-methylphenyl)iminomethyl]-6,7,8,9-tetrahydropyrido[1,2-a]benzimidazole-10-carbonitrile 2-(4,6-dimethoxypyrimidin-2-yl)sulfanyl-5-iodo-3H-thieno[3,2-d]pyrimidin-4-one (E)-2,3,4-trifluoro-N-[4-[[4-[(2-hydroxy-5-nitrophenyl)diazenyl]pyridin-1-ium-1-yl]methoxy]-2,6-dimethylphenyl]but-2-enethioamide (E)-N,2-dimethyl-3-[2-methylidene-5-oxo-7-[4-phenylmethoxy-3-(trifluoromethyl)anilino]heptylidene]hex-5-enamide;ethane N-[(3S)-4-amino-1,1-dioxothiolan-3-yl]-2-[5-(2,6-dichlorophenyl)pyridin-3-yl]butanamide;ethane 4-[N'-(2,5-dimethylphenyl)carbamimidoyl]cyclohepta-1,3,6-triene-1-carboxylic acid 1-[7,8-difluoro-6-(4-propylphenyl)naphthalen-2-yl]ethanone 3-[5-(1,4-dioxaspiro[4.6]undecan-8-yl)tetrazol-2-yl]-N,N-diethylpropan-1-amine;hydrochloride (3R)-7-methylsulfanyl-N,1',1'-trioxospiro[2H-indene-3,4'-piperidine]-5-carboxamide 1-(2-bromophenyl)-N-methyl-3,4-dihydro-1H-isoquinoline-2-sulfonamide 3-benzyl-2,5-dimethylbenzohydrazide 5-[6-[4-(4,4-difluoropiperidine-1-carbonyl)anilino]imidazo[1,2-b]pyridazin-3-yl]pyridine-3-carbonitrile 2-chloro-4,5-diethylthiophene-3-carboxylic acid 3-azido-1-(diethoxyphosphorylmethyl)pyrazole 1-[2-(difluoromethyl)-6-phenylpyridine-3-carbonyl]-4-hydroxypiperidine-4-carboxylic acid (5E)-2-imino-5-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one 2-azido-4,5-dichloro-1H-benzimidazole 2-N,4-N-bis[(2S)-3-chlorobutan-2-yl]-1-N,4-N-dimethylbenzene-1,2,4-triamine 4-[(7R)-5-methyl-2,3-diphenyl-4H-pyrazolo[1,5-a]pyrimidin-7-yl]phenol N-[(1R,3R)-3-hydroxycyclopentyl]-2-(6-methoxyquinolin-4-yl)oxyacetamide 4-[2-chloro-6-methyl-4-(trifluoromethyl)anilino]sulfanylbenzoic acid 3-ethenyl-N-(4-formylphenyl)benzenesulfonamide 3,6-dihydroxy-4-(3-methylpyridine-2-carbonyl)cyclohexa-2,5-dien-1-one 1-butan-2-yl-N-[4-(cyclopropylmethoxy)phenyl]pyrazole-3-carboxamide 1-[4-[2-[2-[(4S)-6-chloro-3,4-dihydro-1H-isoquinoline-2-carbonyl]imidazo[1,2-a]pyridin-5-yl]oxyethyl]piperidin-1-yl]-2,2,2-trifluoroethanone 6-(2,4-dimethylanilino)-1H-pyrimidine-2,5-dione 5-N,7-dimethyl-1-(2-phenyl-1H-indol-3-yl)-3H-imidazo[4,5-c]pyridine-2,5-diamine N-[5-cyano-2-(trifluoromethyl)phenyl]-6-(3,4-dichlorocyclohexa-1,3-dien-1-yl)-7-oxo-8H-imidazo[1,2-b]pyridazine-3-carboxamide 1-[6,7-bis(ethenyl)thieno[3,2-d]pyrimidin-4-yl]piperidine-2-carboxamide N-[2,6-di(propan-2-yl)phenyl]-1-methylpyrrole-2-carboxamide;rhenium N-(2,4-difluorophenyl)sulfonyl-1-hydroxypyridin-1-ium-3-carboxamide [1-[6,7-dimethyl-2-(oxolan-3-yl)quinolin-4-yl]azetidin-3-ylidene]methanamine 3-(2,6-dichloro-N-hexylanilino)propane-1,2-diol [4-[2,6-difluoro-N-(1,3-thiazol-5-yl)anilino]phenyl]sulfonylurea 4-[[(1S)-1,5-dimethyl-3-phenyl-2H-imidazo[4,5-b]pyridin-7-yl]amino]piperidine-1-carboxylic acid (1S,3R)-2,2-dichloro-N-[4-fluoro-5-[6-(1H-indole-3-carbonyl)-1H-benzimidazol-2-yl]pyridin-2-yl]cyclopropane-1-carboxamide 4-(2-azidoethenyl)-2-nitroaniline N-[(5R)-6,7-dihydro-5H-cyclopenta[b]pyridin-5-yl]-2-(4-methoxycyclohexa-1,3-dien-1-yl)acetamide [1-(2,4-dichlorophenyl)cyclopentyl]carbamic acid 1-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2-[3-[4-[ethoxyphosphanyl(pyridine-3-carbonyl)amino]piperidin-1-yl]propyl]cyclopropane-1-carboxylic acid;ethane 1-[3,5-bis(trifluoromethyl)phenyl]-N,2-diethoxypropan-1-imine;hydrochloride 4-(2,3,5,6-tetramethylpyrazin-1-ium-1-yl)benzoate;3,3,4-tripropoxybuta-1,3-dien-2-olate 3-benzylsulfanyl-4-phenylbut-1-enylsulfonic acid 2-(1H-imidazol-5-yl)-N-[4-[3-oxo-3-(1,1,6-trimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)propyl]phenyl]acetamide 3-[(2,4-dioxo-1H-pyrimidine-6-carbonyl)amino]propanoic acid 2-fluoro-N-[3-[[4-oxo-5-(thian-4-ylmethylidene)-1,3-thiazolidin-2-ylidene]amino]phenyl]benzamide 4-cyclopropyl-6-fluoro-3,3a-diphenyl-2H-pyrazolo[3,4-b][1,5]benzodiazepine 3-[2,4-bis(phenylmethoxy)-5-propanoylphenyl]cyclohexane-1-carboxylic acid 5-chloro-2-[(3R)-1-(cyclopropanecarbonyl)pyrrolidin-3-yl]oxypyridine-4-carbonitrile N-[1-[6-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)pyridin-3-yl]ethyl]acetamide (2R,4S)-N-[(6R)-1-amino-4,5,6,7-tetrahydroindazol-6-yl]-2-hydroxy-2,3-dimethyl-3a,4,5,6,7,8-hexahydrocyclopenta[b]naphthalene-1-carboxamide 2-cyclohepta-1,3,6-trien-1-yl-5-ethenyl-4-methoxythiophene 5-[(1S)-1-cyclopropylethoxy]-4-iodopyridine N-methyl-2,3,4,5-tetrahydro-1H-[1,4]diazepino[6,7-b]indole-8-carboxamide 2-[3-(3-hydroxyphenyl)propyl]-4-(phenoxymethyl)piperidine-1-carboxylic acid (3R)-N'-[2-methyl-4-(3-methylphenyl)phenyl]-5-oxopyrrolidine-3-carbohydrazide N-[4-(2-oxopropanoyl)phenyl]prop-2-enamide 2-N,5-ditert-butylbenzene-1,2-dicarboxamide 3-azido-2-methyl-N,N-diphenylpropanamide 5-(1,3-benzodioxol-4-yl)-N-[4-[4-chlorobutyl(methylsulfonyl)amino]phenyl]furan-2-carboxamide N-[[2,6-di(propan-2-yl)phenyl]-[4-(trifluoromethoxy)phenyl]methylidene]hydroxylamine 1-methyl-3-[6-(2,4,5-trifluorophenyl)pyridin-3-yl]-2H-quinazoline 3-[4-[[(5E)-6,7-dimethylocta-1,5,7-trien-2-yl]oxymethyl]phenyl]-5-methoxybenzoic acid;ethane 3-[(4-aminocyclohexyl)methylamino]-6-N,1-diethyl-5H-pyrazolo[3,4-d]pyrimidine-2,6-diamine;hydrochloride 2-[2-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-6-yl]oxypropanoic acid (2S)-1-[4-(cyclopropylmethoxy)phenyl]sulfonyl-N-hydroxypiperidine-2-carboxamide 1-[2,2-difluoro-3-(4-propylphenyl)cyclopropyl]-N-ethoxymethanamine N-[4-methyl-2-[(E)-2-nitroethenyl]phenyl]prop-2-enamide 2-[3,4-dichloro-5-(trifluoromethyl)pyridin-2-yl]-1H-indole N-(furan-2-ylmethyl)-1-[3-hydroxy-4-[3-(2H-tetrazol-5-yl)phenyl]sulfanylnaphthalene-2-carbonyl]piperidine-2-carboxamide 2,6-ditert-butyl-4-(2,3-dimethylphenyl)sulfonylphenol 2-[2,6-dichloro-4-nitro-N-(1,3-thiazol-5-yl)anilino]acetonitrile (4E,5Z)-4-butylsulfanylimino-5-[3-methoxy-1-oxo-2-(2,4,6-trifluorophenyl)isoquinolin-8-yl]-N'-(methylideneamino)hexa-2,5-dienimidamide 2-[4-(ethylsulfonylamino)piperidin-1-yl]pyridine-3-carboxamide (E)-1-chlorobut-2-ene;ethane;2-[4-(methylaminosulfanyl)phenyl]acetaldehyde;1,3-xylene 1-[(3S,4R)-3-methoxy-4-(2H-triazol-4-yl)pyrrolidin-1-yl]-3-phenylpropan-1-one 1-[(6,7-dimethoxyquinolin-4-yl)methyl]piperidine-4-carboxamide 3-[(Z)-1-[[(2S,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)oxolan-2-yl]methoxy]prop-1-enyl]-5-chloro-N-ethylpyridin-2-amine 1-[6-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)pyridin-2-yl]piperidine-3-carboxamide 4-(2,3-dimethylphenyl)-5-iodo-1H-pyrimidin-6-one 1-(4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl)-3-[4-(trifluoromethoxy)phenyl]urea 4-[[4-[(4-carboxybenzoyl)amino]phenyl]methylidenecarbamoyl]-3,5-dihydroxybenzoic acid 4-bromo-N'-[(Z)-(3,5-dichloro-2-hydroxyphenyl)methylideneamino]benzenecarboximidamide 4-cyclohexylsulfanyl-N',N'-dimethylbenzohydrazide 3-(1H-indazol-4-yl)-6,7-dihydro-1H-indole (2S)-4-fluoro-N,6,8-trimethyl-1,2,3,5,5a,11b-hexahydroisochromeno[3,4-c]pyridine-2-carboxamide 2-[4-(1H-pyrazol-5-yl)phenyl]propanoic acid 5-(2-azidopropan-2-yl)-1,3-benzodioxole 2-[6-(diethylamino)-1-phenylpyrazolo[3,4-b]pyridin-3-yl]phenol N-[(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-3-iodobenzamide ethane;4-fluoronaphthalene-2,3-dicarboxylic acid 2-amino-4,5-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide;5-(4-ethoxy-3-methylphenyl)-3-methyl-2H-triazolo[4,5-b]pyridine (4aR,7aS)-4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-6-isocyano-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine 5-amino-4-[(2-bromonaphthalen-1-yl)diazenyl]-3-methoxy-1H-pyrazole-2-carbonitrile 3-azido-6,7-difluoro-2H-indazole 2-[2-(benzenesulfonyl)-5-chloro-1H-pyridin-3-yl]ethanol 5-(1-methylpiperidine-4-carbonyl)oxypyridine-2-carboxamide (3R)-4-[2-azido-5-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-methoxybutan-1-ol [2-(cyclohexylmethoxy)phenyl]urea [(1R)-3,4-dihydro-1H-isochromene-1-carbonyl]-[2-hydroxy-5-[(3-methylphenyl)carbamoylamino]phenyl]carbamic acid 2-[(6,7-dimethoxyquinazolin-4-yl)amino]acetate 1-(3,4-difluorophenyl)sulfanyl-3-[3-[3-(2-pyridin-3-ylethoxymethoxy)phenoxy]propyl]urea [3-(2,6-dichlorophenyl)-5-(ethylamino)-4-hydroxypyrazol-1-yl]-phenylmethanone 2-[[4-methoxy-6-(1,5-naphthyridin-3-yl)pyrimidin-2-yl]amino]-N-propan-2-ylacetamide 2-[3,5-dibromo-4-hydroxy-N-(3-methylbutanoyl)anilino]octanoic acid 2-[4-(dimethylamino)phenyl]imino-3,5-dihydro-1H-imidazo[2,1-b]quinazolin-8-one 7-azidooxy-4H-1,4-benzoxazine 2-methoxy-3-(oxiran-2-ylmethyl)naphthalene (2S,4R)-1-[(4-aminophenyl)methyl]-N'-hydroxy-4-methoxypyrrolidine-2-carboximidamide;dihydrochloride 7-amino-5,6-dimethyl-N'-(1H-pyrrolo[2,3-b]pyridine-4-carboximidoyl)spiro[3.5]nonane-8-carboximidamide (5R,6S)-1-cyclopropylsulfonyl-N-[(2,3-dimethoxyphenyl)methyl]-4,7-dioxo-6-[(2,4,6-trifluorobenzoyl)amino]-5,8-dihydro-2H-pyrido[2,3-d]pyrimidine-3-carboxamide 4-[(4E)-2,5-dimethylhepta-1,4,6-trien-3-yl]benzoic acid 1-(4-methylpiperidin-2-yl)-2,3,5,6-tetrahydro-1,4-benzodioxocine 1-(4,5-dihydro-2H-benzo[g]indazol-3-yl)ethanone 4-(1,5-dimethylpyrazol-3-yl)benzene-1,2-diol;ethane 6-ethenyl-5,6,7,8-tetrahydronaphthalene-1-carboxylic acid 2-[4-[(E)-2-aminoethenyl]piperidine-1-carbonyl]oxy-N-azidobenzamide 2-[5-carbamoyl-9-[(4-fluorophenyl)methyl]-2-propan-2-ylcarbazol-4-yl]peroxyacetic acid N-[(3S,4R)-1-benzylpiperidin-3-yl]-6-methoxypyrazolo[1,5-a]pyridine-3-carboxamide 1-[2-amino-5-bromo-3-(cyclohexylmethoxy)benzoyl]pyrrolidine-2-carboxylic acid 7-bromospiro[3H-furo[2,3-c]pyridine-1,4'-oxane] (3Z)-5,6-dimethylhepta-1,3,5-triene;N-ethyl-6-hydroxy-9H-fluorene-4-carboxamide N-[2,6-difluoro-4-(2H-triazol-4-yl)phenyl]-1-ethylpyrrolidine-3-carboxamide (3-azidooxyphenoxy)methanediol 1-[4-(trifluoromethyl)phenyl]butan-2-ol 2-[4-hydroxy-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)anilino]acetic acid 3-[(3S)-1-[2-chloro-4-(2-fluorophenoxy)benzoyl]piperidin-3-yl]-1,6-dimethylimidazo[4,5-c]pyridin-2-one 4-amino-6-[(3-cyanopyridin-2-yl)methoxy]pyrimidine-5-carbonitrile 2-[4-(4-fluorophenyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinoline;methanol N-[5-methyl-6-(trifluoromethyl)pyrimidin-4-yl]nitramide 3-[(5Z)-5-[2-imino-3-(4-phenylmethoxyphenoxy)propylidene]cyclopenten-1-yl]oxybutanal 2-bromo-3-chloro-5,6-dimethylpyridine;ethane 1-cyclohexyl-5-(2,6-dimethoxyphenyl)-N-pyridin-4-ylpyrazole-3-carboxamide 3-azidooxy-1,4-dichloronaphthalene (2S)-N'-[(4R,5Z)-1-ethyl-4,5-diphenylimidazolidin-2-ylidene]piperidine-1-carboximidamide 3-methylsulfanyl-6-[(Z)-prop-1-enyl]phenanthridine 2-[1-(dimethylamino)ethenyl]-N-methylaniline N-benzylsulfonyl-1-[(4-methoxyphenyl)methyl]piperidine-2-carboxamide 7-(2,6-dichlorophenyl)-12-[5-[4-(2-fluoropropan-2-ylsulfonylamino)piperidin-1-yl]pyridin-3-yl]-2,5,11,13-tetrazatricyclo[7.4.0.02,6]trideca-1(13),3,5,9,11-pentaen-8-one 2-[3-methoxy-4-(2H-pyridin-1-yl)phenoxy]ethanamine 5-[(4-cyclopentyl-2,3,6-trimethoxyphenyl)sulfonylamino]benzene-1,3-dicarboxylic acid 4-[1,3-bis(4-methylphenyl)propan-2-ylideneamino]-N'-pyrimidin-2-ylbenzenecarboximidamide 4-[2-(4-hydroxypiperidin-1-yl)ethoxy]benzoic acid 5-azido-3-[3,4-bis(trifluoromethyl)phenyl]-1H-pyrazole 4-[(3,5-difluorophenyl)methyl]cyclohexan-1-amine;2-(1H-indol-6-yloxy)-N-propan-2-ylpyridine-3-carboxamide 2-(1,1-dioxo-3H-2-benzofuran-5-yl)-1,4-benzothiazin-7-amine 4-(3-ethyl-7H-benzo[c]fluoren-8-yl)phenol (2S,3R)-N-cyclopropyl-4-methyl-5-oxo-3-phenylpyrrolidine-2-carboxamide N-[2,2-diethoxy-1-[6-(trifluoromethyl)pyridin-3-yl]propylidene]hydroxylamine 5-[[1-(2,6-dimethylphenyl)triazol-4-yl]methoxy]benzene-1,3-dicarbonitrile N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]naphthalene-1-carboxamide 4-[2-(2,3,4-trifluorophenoxy)phenyl]sulfonyloxypiperazine-1-carboxylic acid 2-[2-(3,5-dimethylphenoxy)ethoxy]-1H-pyridine-4-thione 3-[(5-chloroquinolin-8-yl)sulfonylamino]-N,N,2-trimethylbenzenesulfonamide 6-hydroxy-3-[[4-(4-methylphenyl)piperazin-1-yl]methyl]chromen-2-one 5-chloro-N-methyl-2-(1H-pyrrole-3-carbonyl)thieno[3,2-b]thiophene-3-carboxamide [2-methyl-5-(oxan-4-ylamino)phenyl]methanol 6,6-dichloro-1-(4-methoxyphenyl)hexan-2-one;N-ethylbut-3-enamide 3-fluoro-2-(4-octylphenyl)pyridine (5R,6S)-5-[4-(benzylcarbamoyl)piperidine-1-carbonyl]-6-methoxy-4,7,8-trioxo-N-propan-2-yloctanamide 2-N,3-N-dibutylbenzene-1,2-disulfonamide 2-[3-fluoro-5-(trifluoromethyl)phenyl]-N,1-bis[(4-methoxyphenyl)methyl]-4-prop-1-ynylpyrrole-3-carboxamide 5-azidosulfanyl-3H-1,4-benzodiazepine (1S)-N,2-dimethyl-N-[4-[(3R)-3-methylpyrrolidin-1-yl]phenyl]cyclopentane-1-carboxamide 4-chloro-3-(difluoromethyl)-1-ethylpyrazole 4-azidosulfanyl-N'-benzamidobutanimidamide 3-aminosulfanyl-5-(4-methoxyphenyl)-N-(2-thiophen-2-ylethyl)thiophene-2-carboxamide 4-[4-(diethylamino)anilino]-2-methylphenol 1-(2,3-dimethylphenyl)-6,7-dihydro-4H-triazolo[4,5-c]pyridine 4-[4-bromobutan-2-yl(cyclohexyl)amino]-N-quinoxalin-2-ylbenzenesulfonamide (6R,9S)-6-methyl-2-phenylsulfanyl-8-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-9-one 2-[4,5-di(propan-2-yl)-1H-pyrazol-3-yl]-N,N-diethylaniline 2-[3,5-dichloro-N-(2-oxopropyl)anilino]decanoic acid 3-[2-hydroxy-4-(7,11,12,13-tetrazapentacyclo[10.8.0.02,10.03,8.014,19]icosa-1(20),2(10),3,5,8,14,16,18-octaen-17-yloxymethyl)phenyl]propanoic acid (4S)-3-[2-[[1-(3,5-difluorophenyl)pyrrolidin-3-yl]amino]pyrimidin-4-yl]-1,3-oxazolidine-4-carboxylic acid 2-amino-6-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-hydroxypyridine-3-carboximidamide 2-[1-(6-chloroquinoline-4-carbonyl)piperidin-3-yl]oxyethyloxidanium 2-[(1Z,3E)-1-(methylideneamino)penta-1,3-dienyl]-5-phenylaniline 3-amino-4-cyano-5-[2-methoxy-6-(trifluoromethyl)phenyl]-1H-pyrrole-2-carboxamide 1-[6-(3,4-dichlorophenyl)-5-methylpyridine-2-carbonyl]-N'-(2H-triazol-4-yl)piperidine-4-carbohydrazide [1-[2-[2,6-dimethyl-4-(1,1,2,2,3,3,3-heptafluoropropyl)phenyl]ethynyl]cyclopentyl]methanesulfonate (E)-4-[3-[2-(5-bromoindol-1-yl)ethyl]cyclohexa-1,3-dien-1-yl]but-3-en-2-one 4-chloro-2,7-di(butanoyl)fluoren-9-one N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1,3-benzothiazol-2-amine 3-cyclopropyl-1,2,4-thiadiazine;N'-(5-fluoropyridin-3-yl)butane-1,4-disulfonamide N-[(2,3-dichlorophenyl)methyl]-N'-ethoxymethanimidamide 3-[5-amino-6,8-dideuterio-2-(trideuteriomethyl)-4-oxoquinazolin-3-yl]-1,1-dimethylurea 4-[3-fluoro-5-(methylamino)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile 2-[(3R)-3-aminopyrrolidin-1-yl]-N',4,6-trimethylpyridine-3-carboximidamide 2-amino-4,5-dimethoxybenzoic acid;2-methylpropane 1-[3-methoxy-5-[4-(trifluoromethyl)phenyl]sulfonylthiophen-2-yl]propan-2-one 2-[5-chloro-4-[3-methyl-6-(trifluoromethyl)imidazo[4,5-b]pyridin-2-yl]-1H-pyrazol-3-yl]benzenethiol 4-[5-(1H-indole-2-carbonyl)pyridin-3-yl]piperazine-1-carboxylic acid 4-methylpentanoic acid;3,5,8,11-tetrahydro-2H-[1]benzoxepino[3,4-e]indole (1R)-2,2,2-trifluoro-1-[6-methyl-3-(4-pyridin-2-yloxypiperidine-1-carbonyl)-3H-inden-5-yl]ethanol (4-ethylthiadiazol-5-yl)methanesulfonic acid [3-[(4R)-1,4a-dimethyl-7-oxo-5,6-dihydrocyclopenta[c]pyridin-4-yl]phenyl]methanesulfonate 6-(4-bromo-2-cyclohexylpyrazol-3-yl)oxynaphthalene-1,4-dione 1-[2-hydroxy-3,4-bis(phenylmethoxy)butyl]piperidin-4-ol 5-chloro-N,2-dimethylbenzamide;1-(1H-indol-4-yl)-3-pyridin-4-yl-4,5,7,8-tetrahydrooxepino[4,5-c]pyrazole 2-[(5-chloropyridin-3-yl)methylamino]-7,8-dihydro-3H-pyrimido[4,5-d]pyrimidine-4,6-dione 1-(oxolan-3-yl)-4-phenyl-N-[1-[4-(trifluoromethoxy)phenyl]ethyl]pyrrole-2-carboxamide 1-cyclohexyl-4-[(E)-3,7-diphenylhept-2-enoxy]benzene N-[5-chloro-2-(3,4-dimethylpiperazine-1-carbonyl)phenyl]-6-oxo-1H-pyridine-3-carboxamide 3-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-6-methylsulfonylpyrazolo[1,5-a]pyrimidin-7-one 2-[4-methoxycarbonyl-N-(1,3-thiazol-5-yl)anilino]acetic acid 2-hydroxy-4-[2-methylpropyl(phenacyl)amino]benzoic acid 3-[2-chloro-6-fluoro-5-(4,4,5,5-tetramethyloxaborolan-2-yl)phenyl]butanoic acid (3S,4S)-1-[4-cyano-3-(trifluoromethyl)phenyl]-4-[1-(cyclopropanecarbonyl)piperidin-4-yl]pyrrolidine-3-carboxamide (2S)-2-amino-N-[1-[2-(3,4-dimethoxyphenyl)ethyl]pyrrolidin-3-yl]butanediamide (2E,4Z)-5-[4-chloro-3-[[cyclopropyl(methyl)amino]methyl]phenyl]-2-ethenylhepta-2,4,6-trienenitrile 2-[[1,3-bis(4-methylphenyl)-5-oxopyrazolidin-4-ylidene]methylsulfonyl]acetic acid 6-(3,4-dimethoxyphenyl)-2-ethylsulfinyl-3-[6-methoxy-5-[(1Z,3E)-penta-1,3-dienyl]pyridin-2-yl]pyrazolo[1,5-a]pyrimidine N-[4,5-bis(ethenyl)cyclopenta-1,3-dien-1-yl]-N'-ethyl-2-methylidenepentanediamide;1,2,7-trifluoro-3-propan-2-ylnaphthalene 1-(azidomethyl)-2,3-dibutoxybenzene 2-[4-bromobutan-2-yl(3,5-dimethylphenyl)sulfonylamino]benzenesulfonic acid N-(2,4-dimethylphenyl)-2-[4-ethoxy-3-[(4-oxo-1,5,6,7-tetrahydropyrazolo[3,4-d]pyrimidin-6-yl)methyl]phenoxy]acetamide 2-(3,4-dichlorophenyl)acetamide;ethane 2-methyl-1'-[(2S)-1,4-oxazepan-2-yl]spiro[5H-furo[3,4-d]pyrimidine-7,3'-piperidine];dihydrochloride 3-[(Z)-1,2-diphenylprop-1-enyl]pyrazine-2-carboxamide 3-(4-chlorobenzoyl)-6-(4-methylphenyl)cyclohex-2-en-1-one 5-chloro-N'-hydroxy-3-[2-(hydroxymethyl)pyrrolidin-1-yl]sulfonylpyridine-2-carboximidamide 2-chloro-N-[2,4-difluoro-3-[5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl]phenyl]-5-(trifluoromethylsulfanyloxy)benzenesulfonamide (2Z,4E)-5-[8-(dimethylamino)quinolin-3-yl]penta-2,4-dienoic acid 3,5-difluoro-N-[[(2S)-4-methylmorpholin-2-yl]methyl]benzenesulfonamide 2-(3,4-dimethoxyphenyl)sulfonyl-N-(2-phenylethyl)benzenecarboximidate N-(4-fluorophenyl)sulfanyl-3-methoxy-6-nitro-1,2,4-triazin-5-amine N-[(3R)-1-[4-methoxy-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperidin-3-yl]cyclopropanecarboxamide N-[3-chloro-4-(2,3-dihydropyrrole-1-carbonyl)phenyl]-3-methylpyridine-2-carboxamide 4-azido-6-methyl-5-phenylpyrimidine (3,5-ditert-butylphenoxy)-nitrophosphinic acid 2-[5-ethenyl-3-(1-iodoethoxy)thiophen-2-yl]pyrimidine N-[1-(3-methoxypropyl)pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-6-carboxamide (3-azido-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-yl)-pyrrolidin-1-ylmethanone 2-chloro-4-[(2R)-2,5,7,11b-tetramethyl-1,3,6,8-tetrahydropyrido[2,1-a]isoindol-9-ium-2-yl]aniline 5-[[[(1S)-2,3-dihydro-1H-indene-1-carbonyl]amino]methyl]thiophene-3-carboxylic acid 2-[1-[2-(dimethylamino)phenyl]propylamino]ethanol;ethane 1,7-di(pyrimidin-5-yl)pyrido[2,3-b]pyrazine 1-[5-(2,3-dimethylpentan-3-yl)thiophen-2-yl]-N-propan-2-ylethanimine N-[(4R)-7-bromo-4-methyl-3,4-dihydro-2H-thiochromen-6-yl]acetamide 2-(4-fluorophenyl)-1-[2-(2H-tetrazol-5-yl)pyrrolidin-1-yl]ethanone 3-(4-methylpiperazin-1-yl)-6-[2-(2H-triazolo[4,5-b]pyridin-5-yl)ethynyl]quinoline 1,2-bis(4-methoxyphenyl)ethane-1,2-diol 2-amino-4,5-bis[2-(3-chlorophenyl)ethyl]-1H-pyrimidin-6-one 4-[[3-[(2,6-dichlorobenzoyl)amino]-2,4-dimethylphenyl]carbamoyl]piperazine-1-carboxylic acid 5-[3-(4-fluorophenyl)pyrazin-2-yl]sulfanylpentanoic acid (3-chlorophenyl)-[2-[4-[[[4-(dimethylamino)quinazolin-6-yl]amino]methyl]triazol-1-yl]phenyl]methanone N-(3,5-dimethylphenyl)-6-hydroxy-N'-[4-[(1-methoxycyclopropanecarbonyl)amino]benzoyl]spiro[2H-1-benzofuran-3,3'-piperidine]-1'-carboximidamide 2-(3,5-difluorophenyl)-N-[(1R,2R)-2-methylcyclohexyl]imidazo[1,2-a]pyrimidin-7-amine (5Z)-2-sulfanylidene-5-[[3-[4-(trifluoromethyl)phenyl]sulfonylphenyl]methylidene]imidazolidin-4-one N-[5-[3-(4-pyridin-2-yl-1H-imidazo[4,5-c]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclopentanecarboxamide 3-azidooxy-1-(benzenesulfonyl)pyrrole N-(3,5-dimethoxyphenyl)sulfanylquinolin-6-amine 1-(2,2-dimethoxyethyl)-3-[[1-(2-fluorophenyl)cyclopropyl]methylamino]thiourea 3-methylsulfonyl-4-[(2R,6S)-2-propan-2-yl-6-propan-2-ylmorpholine-4-carbonyl]benzonitrile 2-[3,5-bis(trifluoromethyl)phenyl]-4,6-diethoxypyrimidine 6-[2-[3,5-difluoro-4-(trifluoromethyl)phenyl]ethynyl]-1-fluoronaphthalene-2-carbonitrile 2-(1,3-benzodioxol-5-ylmethyl)-N'-[4-(carbamoylamino)cyclohexa-2,4-dien-1-ylidene]-3H-furan-5-carboximidamide 2-[4-(cyclohexen-1-yl)phenyl]-3-phenylquinoxaline 3-[2,6-dichloro-N-(4-chlorobutyl)-4-nitroanilino]propane-1,2-diol 3-[2-(dimethylamino)ethyl]indole-1,5-dicarboxylic acid;hydrate 4-azidooxy-6,7-dimethylquinazoline (3S,4R)-1-azido-N-methyl-4-phenylpiperidin-3-amine 2-[4,5-difluoro-3-(trifluoromethyl)pyrazol-1-yl]pyridine 2-(4-ethoxyphenoxy)-N'-hydroxypyrimidine-4-carboximidamide N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-piperidin-1-ylsulfanylpropanamide;oxolane 1-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-7-yl)-6-fluoro-3H-indol-2-one 6-bromospiro[3,4-dihydro-1H-quinazoline-2,3'-piperidine] (1-methoxy-2,3-dihydroinden-5-yl)-[4-[2-(triazol-1-yl)ethyl]piperazin-1-yl]methanone (5Z)-2-imino-5-[[1-(4-phenoxyphenyl)cyclopropyl]methylidene]-1,3-thiazolidin-4-one N'-[(Z)-(3,5-dichloro-4-hydroxyphenyl)methylideneamino]-N-pentanoyloxamide [5-(1,3-thiazol-2-ylmethyl)pyrimidin-2-yl]hydrazine N-(1-benzofuran-6-ylmethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide;dihydrochloride [[4-(2,3-dimethylanilino)-1H-pyrazole-5-carbonyl]amino]carbamodithioic acid (Z)-3-[5-chloro-2-ethoxy-3-methyl-4-(trifluoromethyl)phenyl]-2-cyanoprop-2-enamide 4-[N-(4-bromobutan-2-yl)-2,6-difluoroanilino]-1,5-dimethyl-2-phenylpyrazol-3-one 2-bromo-N'-hydroxyquinoline-4-carboximidamide (2S)-1-[3-fluoro-5-(trifluoromethylsulfanyl)phenyl]sulfonylpyrrolidine-2-carboxamide 5-(5,6-dihydropyrido[2,3-b]pyrazin-7-yl)pyridine-3-carboxylic acid 1-[5-(4,5-diphenyl-2H-triazol-1-ium-1-yl)-3,4-dihydroxyfuran-2-yl]pyrrolidin-2-one N-[(3R,5S)-1-cyclopropyl-7-fluoro-5-methyl-2-oxopiperidin-3-yl]-4-[2-(4-hydroxyphenyl)ethynyl]benzamide 4-(1H-indazol-5-yl)benzenesulfinic acid N-[1,3-benzodioxol-5-yl-(2-bromophenyl)methyl]-4-methoxyaniline N-[1,5-bis(2,4-dimethoxyphenyl)pyrazol-3-yl]methanesulfonamide (5Z)-5-[[3-bromo-5-ethoxy-4-[(2R)-butan-2-yl]oxyphenyl]methylidene]-2-cyclopentylimino-1,3-thiazolidin-4-one N-[6-(2,3-dihydrothiophen-5-yl)pyridin-2-yl]-8-ethoxyquinazolin-4-amine 3-[6-methyl-5-[(Z)-pent-1-enyl]-2,4-dioxo-3H-pyrimidin-1-yl]-N-propan-2-ylpropanamide 7-[4-(5-chloro-6-fluoropyrimidin-2-yl)piperazin-1-yl]-1,3-dimethylimidazo[4,5-b]pyridin-2-one;ethane 7-chloro-1-(2,6-difluorophenyl)-6-nitroquinolin-4-one 2-amino-4-[4-(cyclopentylmethoxy)phenyl]-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carbonitrile 2-[3,4-bis(difluoromethyl)phenyl]-5-methyl-4H-1,2,4-triazol-3-one (1R,3S)-3-[4-aminobutyl(methyl)carbamoyl]-N'-cyclohexa-2,4-dien-1-ylsulfonyl-N-hydroxybenzenecarboximidamide 2-[(5,8-dimethoxynaphthalen-1-yl)iminomethyl]phenol N-[(4S,5R)-3-(2,6-dichlorophenyl)-7-bicyclo[3.2.0]heptanyl]formamide;2-methoxypropane 2-methyl-1,3-di(propan-2-yl)naphthalene 6-chloro-4-N,5-N-bis(2-propan-2-ylsulfonylethyl)pyridine-3,4,5-triamine 1-[4-[7,9-dimethyl-2-(propan-2-ylamino)purin-6-yl]piperazin-1-yl]ethanone 4-[8-(2,6-difluorophenyl)-7-oxopyrido[2,3-d]pyrimidin-2-yl]-N-methylpiperazine-1-carboxamide 3-fluoro-N,4-dimethylbenzamide;1-[(2Z,4E)-6-(methylideneamino)hexa-2,4-dien-3-yl]piperidine-4-carboxamide 1-[5-(2,4-dichlorophenyl)-3,6,12-triazatricyclo[8.4.0.02,6]tetradeca-1(10),11,13-trien-13-yl]ethanone 2-(1H-benzimidazol-2-ylsulfonyl)-N,N-dimethylethanamine;propane 1-(3,5-dimethylphenyl)-2-hydroxy-2-iodoethanone 3-[3-[(4,5-dimethylpyrimidin-2-yl)amino]cyclohexyl]-N-methylimidazo[1,2-a]pyridine-6-carboxamide N-[2,4-difluoro-3-[2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-7-yl)ethynyl]phenyl]pentane-1-sulfonamide 3-azido-1-[4,5-dichloro-2-(4-chlorophenoxy)phenyl]sulfonylindole 2-[azidooxy(naphthalen-1-ylsulfonyl)amino]acetic acid N-(2,3-dihydro-1H-inden-5-yl)-2-methoxybenzamide N-(3,4-dichlorophenyl)-2-[6-(6-methylpyridine-3-carbonyl)-7,8-dihydro-5H-1,6-naphthyridin-3-yl]acetamide 5-(dimethylcarbamoyl)pyridine-3-sulfonic acid [3-[(4-hydroxyphenoxy)methyl]-2,6-diazabicyclo[3.2.0]heptan-6-yl]-naphthalen-1-ylmethanone (5R)-1-[[4-chloro-2,6-difluoro-3-(2-methylpropoxy)phenyl]methyl]-N-[[4-[(4S)-2-oxoimidazolidin-1-yl]cyclohexyl]methyl]-3,5-bis(trifluoromethyl)pyrrolidine-3-carboxamide 1-(2-methylphenyl)-3-[N'-methylidene-N-(4-propanoylpyridin-2-yl)carbamimidoyl]urea 1,5-diamino-2-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl)anthracene-9,10-dione N-benzyl-5,7,8-trimethoxy-1H-indole-2-carboxamide 2-amino-1-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)piperazin-1-yl]ethanone 2-hydroxy-5,6-bis(2,4,4-trimethylpentan-2-yl)benzotriazol-1-ium 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[1-(5-propan-2-ylthiophen-2-yl)sulfonylpiperidin-4-ylidene]urea 3-[3,5-bis(trifluoromethyl)phenyl]sulfanylbutanenitrile 1-[2,5-diethyl-4-(2-phenylhydrazinyl)phenyl]ethenol N-methyl-1'-(2,4,5-trifluorophenyl)spiro[3H-chromene-2,4'-piperidine]-4-amine (2-hydroxycyclohexyl)-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)piperidin-1-yl]methanone N-(2,6-difluorophenyl)-N-[2-[1-(2-methylpropyl)piperidin-4-ylidene]ethanimidoyl]benzamide 3,8-difluoro-6-(2-fluoro-4-pentylphenyl)-7-fluoronaphthalene-2-carbonitrile 2-(6,7-difluoronaphthalene-2-carbonyl)butanedioate 4-[4-[[2-methylpropyl(pyridin-3-yl)amino]methyl]phenyl]-N-pyrimidin-2-yl-1,3-thiazol-2-amine 1-[3,5-bis(trifluoromethyl)phenyl]-N-methylpiperidine-4-carboxamide 1-ethyl-3-[7-fluoro-2,2-dimethyl-4-(1H-pyrazol-5-yl)-3H-1,4-benzoxazin-6-yl]urea [4-(methylcarbamoylamino)phenyl]sulfanium N-cyclohexylformamide;2-(methylamino)pyridine-4-carbonitrile N-(5,6-dimethyl-[1,2]thiazolo[3,4-b]pyridin-3-yl)-3-fluorobenzamide N-(1,4-dihydropyridin-2-ylmethyl)-3-[[7-hydroxy-5-[4-(3-hydroxypropylsulfonylamino)phenyl]-6H-pyrrolo[3,4-d]pyrimidin-4-yl]oxy]cyclobutane-1-carboxamide 5-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]benzene-1,3-diol N-[1-(3,5-difluorophenyl)-4-methoxybutyl]-6-nitropyridine-2-carboxamide N-[6-(hydroxyamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]acetamide 1-[(3Z,5E)-7-amino-5-methylhepta-3,5-dien-2-yl]-N-benzyl-6-methoxy-4-oxoquinoline-3-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-3-hydroxybenzamide 1-[3-(3,4,5-trimethoxyphenyl)propyl]pyrrolidine-2-carboxamide 5-fluoro-4-(2-hydroxyethylamino)-1H-pyrimidin-6-one 1-[5-methylsulfonyl-6-(2,3,4,9-tetrahydro-1H-carbazol-3-yl)pyrimidine-4-carbonyl]piperidine-4-carboxylic acid N'-hydroxy-3,5-dimethylbenzenecarboximidamide 2,6-difluoro-N-(3-fluorophenyl)pyridine-4-carboxamide N-[1-(2,3-dichlorophenyl)butan-2-yl]carbamate N-[3,5-difluoro-4-(quinolin-8-ylsulfonylamino)phenyl]-4-methoxybenzamide 1-[3,4-difluoro-2-(triazol-2-yl)phenyl]-N,5-bis(oxan-2-yloxy)pyrazole-4-carboxamide 2-(3-chloro-5-methylphenyl)-4-[(2R,4S)-2,4-dihydroxycyclopentyl]butanoic acid 2-[4-(1,3-benzothiazol-6-yl)-5H-chromeno[4,3-c]pyridin-8-yl]ethanamine 1,1-dimethyl-3-[4-(methylamino)phenyl]thiourea 5-chloro-N-(7,8-difluoroquinolin-3-yl)-2-hydroxybenzamide (2R)-1-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluoroanilino]-2-methylpropan-2-ol 2-bromo-5-[(E)-2-methylbut-1-enyl]benzenesulfonic acid 2-chloro-4-[2,3-dihydro-1,4-benzodioxin-5-yl(pyridin-3-yl)amino]benzamide 4-[(6E,10Z)-16,18-dihydroxyoctadeca-9,11,14-trienyl]benzene-1,3-disulfonic acid;ethane 2,4-diaminopyrimidine-5-carbonitrile;3-ethyl-8-[2-(1-methylpyrazol-4-yl)ethynyl]-2-phenylisoquinolin-1-one 1-ethenyl-4-[(Z)-2-iodoethenyl]benzene 7-[[3-cyclopropyloxy-5-(2,2,4,6,7-pentamethyl-3H-1-benzofuran-5-yl)pyridin-2-yl]methylsulfonyl]-2H-triazolo[4,5-b]pyridine 4-(3-bromophenyl)-6-chlorohexanoic acid 2-(4-fluorophenyl)-6,8-dimethoxy-N-[(3S)-pyrrolidin-3-yl]quinazolin-4-amine 1-azidosulfanyl-4-fluorobenzene 4-benzyl-N-(2,6-dibromophenyl)-3-hydroxy-1-oxo-2H-pyrrolo[1,2-a]pyrazine-8-carboxamide 4-[1-(4-hydroxyphenyl)ethyl]-2,6-dimethoxyphenol 1-(2,4-dichlorophenyl)-4-pyridin-3-yl-5H-tetrazole 2-[4-[(Z)-(3,5-dichlorophenyl)methylideneamino]-1-(morpholine-4-carbonyl)pyrazol-3-yl]sulfanyl-N-ethylacetamide 6-(1,3-benzothiazol-2-yl)quinoline-5,8-dione 4-N-(3-nitrophenyl)benzene-1,4-diamine N-[(3-methoxyphenyl)methyl]spiro[1,4-dihydroquinoxaline-3,1'-cycloheptane]-2-imine 1-ethyl-2-[6-(1,3,4-oxadiazol-2-yl)naphthalene-2-carbonyl]azetidine-2-carboxylic acid [4-(4,6-dimethoxypyrimidin-2-yl)piperazin-1-yl]-(4-fluorophenyl)methanone N'-[6-(4-fluorophenyl)-1,2-dimethylpyrazolo[3,4-d]pyrimidin-4-yl]propane-1,3-diamine;hydrochloride 1-[2,4-bis(trifluoromethyl)phenyl]ethanone;ethane 3-methoxy-6-(2,2,6,6-tetramethylpiperidin-4-yl)triazin-4-one 5-[2-methylpropyl(pyridin-3-yl)amino]naphthalene-2-sulfonic acid [3-(aminomethyl)phenyl]sulfonyl-[(4E,5Z)-5-ethylidenehepta-1,4,6-trien-2-yl]azanium 1-[4,6-bis(diethylamino)pyridin-2-yl]-3-dodecylthiourea [2-(cyclohexylmethylamino)thieno[3,2-d]pyrimidine-4-carbonyl]azanium 5-methoxycarbonyloxyfuran-2-carboxylic acid 3-[[6-(1,2,4-thiadiazol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino]methyl]phenol 1-[(3aR,8aS)-2,3a-dimethyl-3,4,5,7,8,8a-hexahydro-1H-pyrrolo[3,4-d]azepine-6-carbonyl]pyrazole-4-carbonitrile 2-methoxy-N,N-dimethyl-5-[[6-(4-methylimidazol-1-yl)pyridine-3-carbonyl]amino]benzamide [2-azidooxy-1-(3,4-dichlorophenyl)-3-ethylhexan-3-yl]benzene (4R)-2-methylspiro[4,6-dihydro-1H-cyclopenta[d]pyridazine-7,3'-piperidine]-4-ol 5-[(2-methylphenyl)diazenyl]benzene-1,3-diol 4-[[(1R,2S)-2-methylcyclohexanecarbonyl]amino]-N-[5-(3-pyridin-3-yloxyphenyl)-2H-triazol-4-yl]benzamide 1-[2,4-dimethyl-6-(trifluoromethyl)phenyl]sulfonylpiperazine [3-[[6-(3-methoxyphenyl)pyridin-2-yl]amino]pyrrolidin-1-yl]-(4-piperidin-4-yloxycyclohexyl)methanone;dihydrochloride 2-methyl-5,6-diphenylpyridine;rhenium (1R)-5-[[4-[2,6-difluoro-3-(phenylsulfanylamino)benzoyl]piperazin-1-yl]methyl]-N-hydroxycyclohepta-2,4-diene-1-carboxamide 6-[(2,3-dichlorophenyl)methylsulfanyl]-1,3,5-triazine-2,4-diamine 5-(4-chlorophenyl)-2-fluoro-N-[(3S,4R)-3-hydroxyoxan-4-yl]benzamide;methane 4-(3,5-difluoropyridin-2-yl)-N,1-dimethylpiperazine-2-carboxamide 3-[3,5-dichloro-4-(6-oxo-1H-pyridazin-3-yl)phenyl]sulfonylazetidine-1-carboxylic acid 2-fluoro-3,6-diiodobenzenesulfonate 2-hydroxy-1,3-bis(4-methoxyphenyl)propane-1,3-dione (4E)-4-[(3,5-dimethoxyphenyl)methylidene]-2-pyridin-1-ium-1-yl-1H-imidazol-5-one (2R)-2-amino-N-[(1S,3R)-3-hydroxycyclopentyl]-2-phenylacetamide 1-(3,5-diethylphenyl)-2-phenyldibenzothiophene 2-(3,4-dibromophenyl)imidazo[1,2-b]pyridazine 3-(1-ethoxybutyl)-2,5-dihydropyrazolo[3,4-d]pyrimidine 4-amino-5,6,7,8-tetradeuterionaphthalene-2,3-dicarboxylic acid 3-[(2E)-penta-2,4-dien-2-yl]-1H-carbazole (1-amino-2H-azepin-5-yl)-[3-(4-methoxyphenyl)propyl]-oxoazanium N-(1,3-benzodioxol-5-yl)-2-[6-methoxy-7-[(3-morpholin-4-ylpropanoylamino)methyl]quinolin-4-yl]oxyacetamide 1,3-diphenylhexane-2,5-dione 2-[[(3R)-1-azabicyclo[2.2.2]octan-3-yl]methylamino]pyridine-4-carbonitrile 1,2-dibenzyl-3-(4-chlorophenyl)sulfonyl-5-methoxyindole 1-(2,3-dihydroxypropyl)-2,4,5-trimethoxyanthracene-9,10-dione N-(5-fluoro-1,3-thiazol-2-yl)propane-1-sulfonamide N-[4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl)phenyl]propanamide (3-methylphenyl)-[4,5,6-tris(4-methylphenyl)pyrimidin-2-yl]phosphane 1-[4,6-bis(ethoxycarbonyl)-5-fluoropyridin-2-yl]piperidine-3-carboxylate 1-(3-butanoyl-4,5-dimethoxyphenyl)ethyl-[[4-(trifluoromethoxy)phenyl]carbamothioyl]azanium (1R,3S)-6-chloro-N-[4-[2-hydroxyethyl(methylsulfonyl)amino]phenyl]-3-methoxy-1-(5-methoxypyridin-3-yl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxamide 7-[4-(difluoromethoxy)phenyl]-1,3-benzodioxol-5-amine;1-methylpyrrolidine (1Z,3E)-2-[4-[4-ethyl-5-(trifluoromethyl)thiophen-3-yl]phenyl]-4-phenylbuta-1,3-dien-1-amine;2-ethylbutane N-[(3,5-dibromophenyl)methyl]spiro[1,4-dihydroquinoxaline-3,4'-thiane]-2-imine 3-[6-[2,3-difluoro-4-(2-methoxyethylamino)phenyl]pyrazolo[1,5-a]pyridin-3-yl]-N-propan-2-ylcyclobutane-1-carboxamide 4-[3-(2,6-dichlorophenyl)sulfanylcyclobutyl]pyridine 6-ethyl-4,5-dihydrobenzo[g]indole (2R,3S)-1,1-bis(4-chlorophenyl)-2-[5-(2-methoxyphenyl)thiophen-2-yl]sulfonylpiperazine 4-[3,4-difluoro-2-(hydroxymethyl)phenyl]-N-hydrazinylidene-3,5-dinitrobenzenecarboximidamide 1-[5-(4-fluorophenyl)-2,3,5a,6,7,8,9,9a-octahydropyrimido[4,5-b]quinolin-4-yl]butan-1-one 3-(2-fluoro-4-nitrophenoxy)propanal 5-ethyl-2,3,4-trimethoxybenzaldehyde 5-(N-tert-butylanilino)naphthalene-2-sulfonic acid N-[1-(2,3-dihydro-1H-inden-5-yl)pyrazol-4-yl]spiro[2.3]hexane-5-carboxamide 2-[2-(4-cyanophenyl)ethyl]-6-methoxypyrimidine-4-carboxylic acid 1-[4,5-di(propan-2-yl)-3H-1-benzothiophen-3-id-2-ylidene]-2,2,6,6-tetradeuterio-1,3-bis(phenylmethoxy)piperidine (2S)-1,2-diamino-3-hydroxy-4-[4-methoxy-3-(trifluoromethyl)phenyl]butan-1-one 5-[2-(5,6-diethyl-1H-benzimidazol-3-ium-2-yl)phenoxy]-N-pentanoylnaphthalene-2-carboxamide;bromide 4-azidosulfanyl-3,5-dimethoxyaniline 1-[2,2-diethoxyethyl(hexyl)amino]-4a,9a-dihydroanthracene-9,10-dione 2-methyl-1-[3-(pyridin-2-ylsulfanylamino)piperidin-1-yl]propan-1-one 1-[4-methylsulfonyl-2-(trifluoromethoxy)phenyl]pyrrolidine (5-methylfuran-2-yl)-[8-methyl-3-(trifluoromethyl)quinoxalin-6-yl]methanone 4-chloro-2-[[3-(trifluoromethyl)pyridin-2-yl]amino]benzonitrile 4-fluoro-3,5-diiodothiophene 1-methyl-6-phenyl-3,4-dihydroquinoxaline-2,7-disulfonic acid 2-[4-(1H-pyrrol-3-yl)phenyl]ethanol 5-benzyl-6,7,8,9-tetrahydropyrimido[4,5-d]azepine 2-[5-[4-(1-formyloxycyclopropanecarbonyl)phenyl]pentyl]propanedioic acid (2R,4S)-N-[3,5-difluoro-4-[6-(trifluoromethyl)pyridin-3-yl]phenyl]-1-(2,6-difluorobenzoyl)-4-hydroxypyrrolidine-2-carboxamide 6-chloro-5-(4,8-dimethylnonan-3-yl)oxypyridine-3-carbonitrile 2-[6-(4,4-difluorocyclohexyl)oxynaphthalene-2-carbonyl]cyclobutane-1,3-dione 2-azido-5,8-dimethylpyrido[3,4-d]pyrimidine 3-[2,6-dimethyl-4-(pyrrolidine-1-carbonyl)phenyl]propanamide 1-(7-bromopyrazolo[4,3-d]pyrimidin-2-yl)-N'-methyl-N'-(5,6,7,8-tetrahydronaphthalen-1-yl)ethane-1,2-diamine 1-cyclohexyloxycarbonyl-3,4-dihydronaphthalene-2-carboxylic acid 5-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)benzene-6-id-1-yl]benzo[b]carbazole;platinum(2+) 4-(5-fluoropyridin-2-yl)pyrimidine 6-[4-[(2R)-2-aminopropoxy]phenyl]-N',2-dimethylpyrimidine-4-carboximidamide (6-methoxypyridin-3-yl)-[3-[[methyl(propan-2-yl)amino]methyl]spiro[4,7-dihydrotriazolo[5,1-c][1,4]oxazepine-6,4'-piperidine]-1'-yl]methanone;2,2,2-trifluoroacetic acid 4-[(E)-2-phenylethenyl]benzenesulfonate 2-[(E)-4,6-dimethylhept-3-en-3-yl]pyridine 1-(3,4-dichlorophenyl)sulfinylpyrrolidine;2-[3-methoxy-5-(6H-pyrido[2,3-b]azepin-9-yl)phenoxy]ethanol 2,7-dichloroquinoline-8-carboxylic acid (5S)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2,3-dimethoxyphenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide [4-(1,5,6,7-tetrahydropyrazolo[4,3-b]pyridine-4-carbonyl)piperazin-2-yl]cyanamide 2-azido-5-(4,6-diphenyl-1,3,5-triazin-2-yl)benzonitrile 1-benzyl-2,3,4,5-tetramethoxy-6-(4-methoxyphenoxy)benzene (1R)-N'-[4-(1,2-dimethyl-3H-pyrazol-4-yl)phenyl]-2,2,2-trifluoroethane-1,4-diamine 5-[(6S)-1,2-dimethyl-3,4-dihydroisoquinoline-6-carbonyl]-1H-quinolin-2-one 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5-ethanimidoyl-1H-pyridazin-6-one 2-(3-fluoro-4-iodoanilino)pyrimidine-5-carboxylic acid (2Z,4E)-5-[3,5-dimethyl-1-[2-oxo-2-(propan-2-ylideneamino)ethyl]pyridin-2-ylidene]-N'-ethyl-2-hydroxypenta-2,4-dienimidamide 1-(4-ethenylphenyl)sulfonylbutane-2,3-dione (4-methoxyphenyl)-[3-[[[3-methyl-2-(trifluoromethylsulfanyl)quinoline-6-carbonyl]amino]methyl]pyrrolidin-1-yl]methanesulfinic acid 1-(2,6-dimethylphenyl)-3,5-bis[4-(trifluoromethyl)phenyl]imidazolidine 4-chloro-N-[1-(4-chlorobutanoyl)cyclopentyl]benzenesulfonamide 3-[2-[4-[2-(5-chloro-1H-indol-2-yl)ethoxy]phenyl]-5,6-difluorobenzimidazol-1-yl]propanoate 3-benzylsulfonylpropanenitrile (4-chlorophenyl)-[1-ethylsulfonyl-3,5-dimethoxy-2-(3-morpholin-4-ylpropyl)indol-7-yl]-diphenylsulfanium 1-azido-3,4-dichlorophenanthrene 4-[(2E,5S)-4-oxo-2-[(Z)-(1-phenylindol-3-yl)methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]benzoic acid 2-[1-[(6,7-dimethoxyquinazolin-4-yl)amino]ethylideneamino]benzenesulfonamide 3-fluoro-4,5-dimethoxy-2-propylbenzaldehyde 3-azido-N,4-dimethyl-2-phenylaniline ethane;methanamine;3-[4-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylcarbamoylsulfamoyl)phenoxy]propanoic acid 4-ethenylimino-3,6-bis(2,3,4,5,6-pentamethylphenyl)cyclohexa-1,5-diene-1-carbonitrile N-[4-(1-azido-2,2,6,6-tetramethylpiperidin-4-yl)oxyphenyl]-3-(4-ethylsulfonylanilino)quinoxaline-5-carboxamide 3-(2,4-difluorophenyl)pyridine-2-carboxamide N-[(4-chlorophenyl)methyl]-2-[[2-[3-ethoxy-1-(6-ethoxypyrimidin-4-yl)cyclobutyl]acetyl]amino]acetamide 5-bromo-2,3-dimethylpyrrolo[1,2-b]pyridazine (5-benzylsulfanylpyridine-3-carbonyl)hydrazine 2-[(5Z)-5-[[3,5-dibromo-4-[(4-chlorophenyl)methoxy]phenyl]methylidene]-4-oxo-2-sulfanyl-1,3-thiazolidin-3-yl]acetic acid 2-N,4-N-dimethyl-1-N-[[(5S)-3-[4-(4-phenoxybenzoyl)phenyl]-2-azabicyclo[3.1.0]hexan-2-yl]sulfonyl]pentane-1,2,4-tricarboxamide N-[1-(4-phenylcyclohexyl)ethenyl]aniline 6-[2,5-difluoro-4-[3-(5-methylsulfonylpyridin-2-yl)propyl]phenyl]pyridine-3-carbonitrile 3-fluoro-2-methoxy-5-[2-(1,3-thiazol-2-yl)propanoylamino]benzoic acid 2-(N-(2,6-dichloro-4-nitrophenyl)-4-propylanilino)octanoic acid 1-[2-(4,5-dichlorothiophen-3-yl)ethynyl]cyclohexan-1-ol 4-[(Z)-2-(5,7-dimethyl-2H-1,4-benzothiazin-3-ylidene)hydrazinyl]phenol 1-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]-3-[2-[2-(trifluoromethylsulfanylamino)phenyl]ethenyl]thiourea 4-[2-[4-(7,8-dimethyl-6,7-dihydroquinolin-5-yl)but-1-ynyl]anilino]benzonitrile 5-(2,6-difluorophenyl)-3-[4-hydroxy-3-[(2R)-2-methylmorpholine-4-carbonyl]anilino]thiophene-2-carboxamide (2-nitrophenyl)sulfonylmethanethiol 1-(3,3-difluoro-4H-1-benzothiophen-2-yl)ethanimine 4-(6,7-dimethoxyquinazolin-2-yl)phenol 4-[3-fluoro-5-(trifluoromethyl)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 2-(4-fluorophenyl)-6,7-dihydro-5H-cyclopenta[b]pyridine 6-(1,3-benzothiazol-2-ylamino)-N-propylpyridine-3-carboxamide 3-(2,4-dichlorophenoxy)-1-[[3-(2,6-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]amino]propan-1-ol 1-[2-(4-ethoxycyclohexyl)ethynyl]-4-[2-[3-fluoro-5-methyl-4-[4-(trifluoromethyl)phenyl]phenyl]ethynyl]benzene [(2S)-1-[6-amino-5-[4-(3,3-difluoropyrrolidine-1-carbonyl)cyclohexa-1,5-dien-1-yl]pyridazin-3-yl]azetidin-2-yl]methanol 3-[[2,6-difluoro-4-(2-propylphenyl)phenyl]methoxy]-1-fluoro-1-methylsulfanyl-1-sulfidourea [3-hydroxy-5-(6-iodohexyl)phenyl]-methoxycarbonylazanium N-[1-[(5-bromo-2,3-dihydro-1H-inden-2-yl)carbamoyl]cyclohexyl]-4-(trifluoromethoxy)benzamide 4-[(2,6-diethylanilino)methyl]benzoic acid 4-(6,7-dichloro-3-oxo-2,5-dihydro-1H-[1,3]thiazolo[3,2-a]quinolin-4-yl)-N-(3-methylphenyl)piperidine-1-carboxamide (2-azidooxyethylamino)oxybenzene N-[4-(2,6-dimethylpyrimidin-4-yl)phenyl]-5,5-dimethylhexanehydrazide 2-aminoacetaldehyde;3,5-dimethylpyridine;1-methyl-6-(1-pyridin-4-ylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyrazine 4-amino-5,7-dichloro-2-methylisoquinolin-1-one (5E)-2-[1-chloroethenyl(methyl)amino]-4-propan-2-ylidenehepta-5,7-dienoic acid;6-cyclopentyloxy-N-[[4-(trifluoromethyl)phenyl]methyl]hexanamide 6-[4-chlorobutyl(2,2-diethoxyethyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 4-[(1R,3S)-5-bromo-2-methylidenecyclohexyl]oxyquinoline (6S)-4-chloro-3,5,8-trihydroxyanthracene-1-carboxylic acid 5-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)pyrazolo[1,5-a]pyridine 5-chloro-4-N-[3-ethenyl-1-(3-methoxypropoxy)pentan-2-yl]pyridine-2,4-dicarboxamide N-[2-hydroxy-4-methyl-3-(1,6-naphthyridin-8-ium-4-carbonylamino)pentoxy]-N'-propanoyl-2H-pyran-5-carbohydrazide N-(6-methylpyrazolo[1,5-a]pyrimidin-3-yl)-4-(5-methylpyridin-2-yl)piperazine-1-carboxamide;hydrochloride N-[6-(difluoromethoxy)pyridin-2-yl]cyclopropanecarboxamide N-[2-[3,5-bis(trifluoromethyl)phenyl]ethynyl]-1-cyanocyclopropane-1-carboxamide 1-ethenyl-N-(3-methoxyphenyl)pyrrolidine-2-carboxamide 1-[4-(3-azidopropyl)phenyl]cyclohexan-2-ol 1-[[(3R,4S)-3-[1-(difluoromethyl)pyrazol-4-yl]oxy-4-hydroxypyrrolidine-1-carbonyl]amino]cyclopentane-1-carboxylic acid;2,2,2-trifluoroacetic acid 4-(3-chlorophenyl)benzene-1,2,3,5-tetrol (4aR,10aS)-9-methoxy-2-[(1R)-1-naphthalen-1-ylethyl]-5,6,7,8a,9,10-hexahydrophenanthrene 5-[1-(4-chlorophenyl)ethenyl]-N,3,6-trimethylpyrazin-2-amine 5-azido-2-[4-(dimethylamino)phenyl]phenol (4aR,8aS)-6-[3-(2,2-dimethylpropoxy)azetidine-1-carbonyl]-4a-methyl-4H-pyrido[3,4-d][1,3]oxazin-7-one 4-azido-3,6-dimethyl-2-[4-(trifluoromethyl)pyridin-2-yl]pyridine 2-ethyl-6,7-dimethoxy-3H-quinazolin-4-one N-(2-bromophenyl)-3,5-bis(difluoromethyl)pyrazole-1-carboxamide 5-bromo-4-N-[(2S,3R)-6-[(dimethylamino)methyl]-2-propan-2-yloxy-1,2,3,4-tetrahydronaphthalen-1-yl]pyrimidine-2,4-diamine 1-(2,4-difluorophenyl)sulfonylpiperidine;2-[(E)-prop-1-enyl]cyclobutan-1-ol 1-[4-(5,6,7,8-tetrahydronaphthalen-2-yloxy)piperidin-1-yl]but-3-en-1-one 3-azidooxy-1,2-bis(phenylmethoxy)propane-2-thiol N-[(1R,3S)-4-(6,7-dimethoxyquinolin-4-yl)oxy-2,3-dihydro-1H-inden-1-yl]carbamate 2-[4-methyl-3-(1-pyrrolidin-1-ylbutan-2-ylsulfamoyl)phenyl]acetic acid 6-(5,7-difluoroquinolin-4-yl)-3H-indole-2-carboxylic acid ethane;1-(4-methoxyphenyl)sulfinyl-6-propan-2-ylindazole (5Z)-5-[[6-methoxy-2,3-bis(4-propan-2-ylphenyl)phenyl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione 4-chloro-N,3-dimethyl-2-oxopyridine-1-sulfonamide 2-methyl-4-[(2-oxo-2-propoxyethyl)-phenacylamino]benzenesulfonic acid 5-[3-(4-carboxyphenyl)phenyl]furan-2,3-dicarboxylic acid N-[3-(3-azidoanilino)propyl]acetamide 6-amino-1,3-dimethylbenzo[g]indole-2-carboxylate N-[3-(5-chloropyridin-2-yl)-1,7-diethyl-4-methoxy-6H-pyrazolo[4,3-d]pyrimidin-5-yl]-2-(1,4-diazepan-1-yl)acetamide (2S)-3-[4-[6-[(2,4-difluorophenyl)methoxy]pyridin-2-yl]phenyl]-2-(propanoylamino)propanoic acid N-[2-(1,3-benzothiazol-2-yl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]formamide N-[2-chloro-3,5-bis(4-methoxyphenyl)phenyl]-1,6-dimethyl-3,4-dihydropyrido[4,3-d]pyrimidin-7-amine 3-(4-aminophenyl)-6,7-dimethylquinoxalin-2-amine N-[5-chloro-4-(6,7-dimethoxyquinolin-4-yl)oxy-2-fluorophenyl]formamide N-[4-(2,3-dimethoxyphenyl)-1,3-thiazol-2-yl]-2,5-dimethylfuran-3-carboxamide (E)-5,7-dihydroxy-6-[3-hydroxy-4-(naphthalen-1-ylmethoxymethyl)phenyl]hept-6-enoic acid 1-methylsulfinyl-5,6-dihydro-4H-pyrazolo[3,4-e]indazole 3-(4-bromophenyl)imino-2,2-dimethylcyclohexan-1-one 3-[(2-bromophenyl)methoxy]-1,7-dihydropurine-2,6-dione N'-(1,3-benzodioxol-5-yl)-2,4-dihydroxybenzenecarboximidamide 3-[4-(1,2,4-triazol-1-ylmethyl)phenyl]oxirane-2,2-dicarbonitrile 1-butoxy-4-[(Z)-3-methylidenepent-1-enyl]benzene;ethane 4-[2-azido-6-(4-chlorophenyl)phenyl]morpholine (Z)-1,3-dichloropent-2-ene;ethane;5-(4-formylpiperazine-1-carbonyl)-2-methylpyridine-4-carboxylic acid 2-azido-3,4-dimethylaniline [3-amino-2-(methoxycarbonylamino)-3-oxoprop-1-enylidene]azanium 2-[4-(3,5-dimethylanilino)phenyl]cyclopentan-1-one 2-[N-(2,6-difluorophenyl)-4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]anilino]ethanol N-(2,3-dihydroindol-1-yl)-1,5-dimethylpyrazole-4-sulfonamide ethane;2-(4-methoxyphenyl)sulfanyl-4,6,7,8-tetrahydroisoquinoline-1,3-dione N-[(1R,2S)-3-fluoro-1-methoxy-4-methylpentan-2-yl]pyridine-2-carboxamide 7-fluoro-5,11-dimethoxy-2H-indeno[1,2-g]quinoline 4-[(2R)-1-hydroxybutan-2-yl]-3,5-dimethylbenzamide 5-(5,6-dihydro-4H-cyclopenta[d][1,3]thiazol-2-yl)-2-iodophenol 3-[3-(4-chlorophenyl)-2,5,6-trifluorocyclohexyl]pyridine 2-(2,4-difluorophenyl)-1H-imidazole N-[4-(benzenesulfonyl)phenyl]-6,7-dichloro-1-phenylmethoxyquinazolin-4-imine 2-(azidomethyl)-N-benzylaniline [4-fluoro-2,5-dimethyl-3-(1H-pyrazol-4-yl)phenyl]phosphane 5-[2-(3,4-dichloroanilino)-1,2-bis(4-hydroxyphenyl)ethenyl]benzene-1,3-diol 4-[(E)-3-[3,5-bis(trifluoromethyl)phenyl]prop-2-enoyl]thiomorpholine-3-carboxylic acid 2-[(4S)-3,4-dihydronaphthalen-1-yl]-5,6-dimethoxynaphthalene 7-[3-(aminomethyl)pyrrolidine-1-carbonyl]-8,9,10,11-tetrahydronaphtho[2,1-b][1]benzofuran-6,12-dione N-[3-(1,2-benzoxazol-3-yl)propyl]-4-oxo-3H-quinazoline-7-carboxamide 4-(4-iodophenyl)phenol (E)-4-fluoro-1,2-bis[3-fluoro-5-(trifluoromethyl)phenyl]pent-2-en-1-one 5-[(2R)-2,3-dimethylcyclopropen-1-yl]-3-ethoxy-N-[(4-imidazol-1-ylphenyl)methyl]-4-methylpyridine-2-carboxamide (2-fluorophenyl)-[(4R,5S)-4,5-dimethyl-1-pyrimidin-2-yl-6,7-dihydro-4H-triazolo[4,5-c]pyridin-5-yl]methanone 6-bromo-4-[1,2,2-trifluoro-2-(2,3,5-trimethylphenyl)ethoxy]naphthalen-2-ol 1-(2,5-difluorobenzenecarboximidoyl)piperidin-4-amine;hydrochloride 3-[1,4,8-trimethyl-2-(2-phenylethyl)-5-propan-2-ylidenecycloocta-1,6-dien-1-yl]propanenitrile 1-(2-methoxyphenyl)-N'-[4-(5-oxopyrrolidin-3-yl)phenyl]cyclopropane-1-carboximidamide 2-[3,4-dimethoxy-5-(trifluoromethyl)phenyl]-4H-imidazole 1-(5-ethyl-4-methylidenehexyl)-3,6-dimethoxynaphthalene 4-[(Z,3E)-1-amino-3-ethylidenehex-4-en-2-yl]oxybenzamide;5-(7H-purin-6-yl)pyrimidine-4,6-diamine 3-ethyl-1,5-dimethoxy-2,4-bis(3-phenylpropoxy)benzene 1-[4-[2-fluoro-6-methyl-4-(oxan-3-yl)phenoxy]piperidin-1-yl]ethanone 1-[2,4-dichloro-3-[2-(methylamino)butanoyl]phenyl]ethanesulfonamide 4-[2-[(1-methylpyrazole-3-carbonyl)amino]ethyl]piperidine-1-carboxylic acid (2R)-1,6-dimethoxy-N-phenylheptan-4-amine 5-bromo-4-tert-butyl-2-(6-methoxypyridin-3-yl)-1H-pyrimidin-6-one 4-(4,5-dimethylfuran-2-carbonyl)-3,5-dihydro-1H-pyrido[4,3-b]indole-2-carboxylate 4-[5-chloro-2-(tetrazol-1-yl)phenyl]sulfonylmorpholine ethane;methoxymethane;3-[6-(2-morpholin-4-ylethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl]propanal [4-(2,3-dihydrofuro[3,2-b]pyridin-7-yloxy)phenyl]-[4-hydroxy-4-(piperidine-1-carbonyl)piperidin-1-yl]methanone (1R,2S)-2-[5-[2-(3-chlorophenyl)pyrrolidine-1-carbonyl]pyrazolo[3,4-b]pyridin-1-yl]cyclohexan-1-ol 5-[3-methyl-6-(methylamino)indazol-1-yl]-2-propan-2-yloxybenzonitrile 1-[4-[[5-chloro-2-(trifluoromethoxy)phenyl]methylamino]-3-(trifluoromethoxy)phenyl]pyrrolidine-3-carboxylic acid 5-[(1S)-6,7-dimethoxy-1-propyl-3,4-dihydro-2H-isoquinolin-1-yl]-3-methyl-2-nitroaniline 4-[2,3-dihydroxypropyl(ethyl)amino]-N-(2,6-dimethoxypyrimidin-4-yl)benzenesulfonamide 1-(2,5-dimethoxyphenyl)heptane-1,7-diol ethane;1-[3-[6-(methylamino)quinazolin-8-yl]oxypiperidin-1-yl]prop-2-en-1-one (5Z,6E)-5,6-bis[(3,4-dimethoxyphenyl)methylidene]-1-propan-2-yl-1,3-diazinane-2,4-dione 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-[4-fluoro-7-(trifluoromethoxy)-2,3-dihydroindol-1-yl]ethyl]acetamide N-[4-methylsulfonyl-3-(2H-tetrazol-5-yl)phenyl]-1-(trifluoromethoxy)methanesulfinamide [4-(2-hydroxy-2,3-dihydrochromene-6-carbonyl)piperazin-1-yl]-(6-methylpyridin-3-yl)methanone 2-(N-pyridin-3-ylanilino)propanoic acid N-[(1R)-1-phenylethyl]quinazoline-8-carboxamide 2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzo[de]isoquinoline-1,3-dione 1-benzyl-N,6-dimethylpyrazolo[3,4-b]pyridine-5-carboxamide N-[(1S)-1-phenyl-2-piperidin-4-ylethyl]propanamide (E)-3-[4,5-dimethyl-2-[5-methyl-1-(oxan-2-yloxy)cyclohexa-2,4-dien-1-yl]pyrazol-3-yl]prop-2-enenitrile 3-chloro-5-(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanyl-N'-hydroxythiophene-2-carboximidamide 2,5-dichloro-N-[[3-[(4-methoxybenzoyl)amino]phenyl]carbamothioyl]-4-nitrobenzamide 1-[4-(4,5-diphenyltriazol-2-yl)phenyl]cyclopropan-1-amine 5-[(5R)-4,8,9-trimethyldecan-5-yl]pyrimidine 1-[4-(4-chlorobenzoyl)piperidin-1-yl]-2-[[3-fluoro-6-methoxy-5-(trifluoromethyl)pyridin-2-yl]methoxy]ethanone N-(2,5-dimethylphenyl)-3-methoxypropanamide;ethane (3S,4R)-4-(1-benzofuran-2-ylmethylamino)-3-fluoropiperidine-1-carboxylic acid N-(4-methoxyphenyl)sulfanyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide 2-[[3-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yloxy)piperidin-1-yl]methyl]benzonitrile 4-[2-(8,9-dihydro-7H-fluoren-9-ylmethoxycarbonylamino)ethyl]benzamide N-[4-[3-[2-(1,3-benzodioxol-5-yloxy)pyrimidin-5-yl]imidazolidin-1-ium-1-ylidene]butyl]acetamide 1-[5-fluoro-2-(oxan-4-yloxy)phenyl]ethanone 4-[[5-chloro-2,3-dideuterio-6-(furan-2-yl)phenyl]methoxy]piperidine 2-[3-cyano-5,7-dimethyl-1-(oxan-4-yl)-6,8-dihydro-5H-naphthalen-2-yl]acetic acid 5-hydroxy-3-methoxy-6-[(E)-2-[(Z)-3,4,4-trifluoro-1-iminobut-2-en-2-yl]prop-1-enyl]pyran-2-one 1-(6-tert-butylpyridazin-3-yl)-2,3-dihydroindole 4-methoxy-3,5-dinitrobenzoic acid 3-fluoro-2-[3-[(E)-3-methoxybut-1-enyl]phenyl]benzaldehyde (3S)-5-methyl-1-[5-(5-methyl-4,5-dihydro-1H-imidazol-2-yl)pyrazin-2-yl]pyrrolidin-3-ol N-[5-(1H-benzimidazol-2-yl)-1H-pyrazol-4-yl]-3,5-dimethoxybenzamide N-[2,6-bis(hydroxymethyl)phenyl]propanamide 2-(7,8-dihydronaphthalen-1-ylmethyl)pyridine 1-(4,4-dimethylcyclohexen-1-yl)-5-ethynylnaphthalene 2-chloro-4,6-bis[(Z)-pyridin-2-ylmethylideneamino]thieno[3,2-d]pyrimidine N-azido-6,7-dimethoxy-1,3-benzothiazol-2-amine N-[2-methoxy-5-(3-pyridin-2-ylpyrrolidine-1-carbonyl)phenyl]ethenesulfonamide 3-bromo-1,6-bis(4-chlorophenyl)-2-hydroxy-8H-quinoline-2-carboxylic acid N-[(2,4-difluorophenyl)methyl]-3-(4-pyrimidin-5-ylphenyl)propanamide;ethane (3-amino-5-methylbenzenecarbothioyl)carbamic acid 5-[2,6-difluoro-3-(propylaminomethyl)phenyl]-1,3-oxazole-4-carboxylic acid 2-[7-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]acetic acid 2-cyclopropylsulfonyl-6-[4-(2,3-dihydroindole-1-carbonyl)phenyl]pyridazin-3-one 4-(3-azidopropyl)quinoline 3-methoxy-4,4,5-trimethyl-N'-[(E)-1-[4-(1-phenylethylideneamino)-2,5-dihydropyrrol-1-yl]prop-1-enyl]pentanimidamide 6-azido-3,4-dihydroquinoline-2-carboxylic acid (2R)-4-[7-chloro-6-[4-(2-fluoroethylsulfonyl)piperazin-1-yl]pyrazolo[1,5-a]pyridine-3-carbonyl]-N-cyclopropylmorpholine-2-carboxamide 2-(4,4a,10b-tetrahydrophenothiazin-1-yl)ethanol 1-[(4R)-3,4-bis(2,5-dimethylfuran-3-carbonyl)piperidine-1-carbonyl]pyrazole-3-carboxylic acid 7-[4-(aminomethyl)-3-fluorophenyl]-5-pyridin-2-ylimidazo[1,2-c]pyrimidine-8-carbonitrile;dihydrochloride 2-[7-(4-methyl-1,3-oxazol-5-yl)quinazolin-2-yl]benzamide 4-[(2,5-dimethyl-1H-pyrrole-3-carbonyl)amino]-N-propan-2-ylcyclohexane-1-carboxamide 1-[4-(3,5-dimethylpyridin-2-yl)oxypiperidin-1-yl]ethanone 1-[(6-chloropyridin-3-yl)methoxy]-2H-pyrimidine [2-amino-5-(1H-pyrrolo[2,3-b]pyridine-6-carbonyl)phenyl]methylideneazanium 3-benzyl-5-(3-fluoropyridin-4-yl)iminopyrazolidine-1-carboximidamide [2-methyl-3-[(3-methylcyclohex-2-en-1-yl)oxyamino]propanoyl]-phenylazanium 1-cyclohexyl-5,6,7,8-tetrahydro-4H-pyrazolo[3,4-b][1,4]diazepine 2-amino-6-hydroxybenzoic acid;1,5-bis(methoxymethyl)cyclohexa-1,3-diene (3R,4S)-1-(cyclopropylmethylsulfonyl)-4-(fluoromethoxy)pyrrolidine-3-carboxylic acid;hydrochloride N-[5,8-bis(3-chloro-4-cyanophenyl)quinoxalin-2-yl]-2-phenylacetamide 2-ethoxy-3-phenyl-1H-indole (4Z,6E)-6-amino-2-methyl-N-(5-propan-2-ylpyridin-3-yl)hepta-1,4,6-triene-3-sulfinamide N-(1,3-benzodioxol-5-ylmethyl)-5-(2-ethyl-7-methoxyimidazo[1,2-a]pyridin-3-yl)pyrimidin-4-amine 6-fluoro-3-[3-(2-methylbutan-2-yloxycarbonyl)-4,5,6,7-tetrahydroindazole-1-carbonyl]indole-1-carboxylic acid N-(2,6-difluorophenyl)-4-[3-methoxy-7-(piperidine-1-carbonyl)quinoxalin-2-yl]piperazine-1-carbothioamide N-[(3,4-dichlorophenyl)methyl]-3-[5-[2-(2-oxopyrrolidin-1-yl)ethoxy]pyridin-3-yl]-2H-pyrazolo[3,4-b]pyridine-5-carboxamide 1-(2,3,5,6-tetradeuteriopyridin-4-yl)oxy-4H-pyrazolo[3,4-d]pyrimidine 5-[2,3-difluoro-4-(trifluoromethoxy)phenoxy]-6-phenylpyridine-2-carbonitrile 2-[3-azido-2,4,6-tri(propan-2-yloxy)phenyl]ethanol (E)-1-(4-chlorophenyl)-3-[2-(trifluoromethyl)phenyl]prop-2-en-1-one 2-N-[4-[(dimethylamino)methyl]-5-(trifluoromethoxy)cyclohexa-1,3-dien-1-yl]-6-(1H-pyrazol-4-yl)-8-pyridin-3-ylquinazoline-2,4-diamine 6-amino-4-(3,5-dibromo-2-hydroxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 4-[(E)-4-chlorobut-1-enyl]-3-(2,3-dihydrobenzotriazol-5-ylidenemethyl)-2-hydroxybenzenesulfonic acid 1-(5-cyclohexylthiophene-2-carbonyl)pyrrolidine-3-carboxylic acid 4-(2,3,4,6-tetrabromophenyl)aniline 1-[6-(5,6-dimethyl-4H-pyridine-3-carbonyl)cyclohexa-1,5-dien-1-yl]ethanone 6-amino-4-[4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl]-3-propyl-4H-pyrano[2,3-b]pyridine-2-carbonitrile N-[4-cyano-2-fluoro-5-(trifluoromethyl)phenyl]benzenesulfonamide 2-azido-5-ethoxy-3,4-dimethylpyridine 2-[4-[(3R)-3,5-dimethylpiperazine-1-carbonyl]anilino]-8-[2-methyl-5-(trifluoromethoxy)phenyl]imidazo[1,2-b]pyridazin-6-one;ethane 2-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-yl)-N-(furan-2-ylmethyl)morpholine-4-carboxamide 1-(5-bromopyrimidin-2-yl)-4,7-dihydro-3H-thieno[3,4-c]pyridine 4-(2-methoxyphenyl)-5-methyl-1H-pyrimidin-6-one (2R)-4,4-dimethyl-2-[3-(1H-pyrrol-2-ylmethylideneamino)propanoyl]pentanamide 1-bromo-4-(6,7-dihydro-2H-cyclohepta[b]pyridin-4-yl)phthalazine 6-chloro-4,5-dihydrothieno[3,2-d][1]benzoxepine (3S)-3-methyl-4,7-diphenoxy-2,3-bis(trifluoromethyl)heptanoic acid N-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-imidazol-1-yl-1-methylcyclobutan-1-amine 2-(2,5-dimethylphenyl)-4-propyl-1H-pyrazole-3-thione 3-[2-aminoethyl(pyridine-4-carbonyl)carbamoyl]butanoic acid 3-benzyl-2-[(2E,4Z)-hepta-2,4,6-trien-2-yl]-1H-indole 5-bromo-2-tert-butyl-4-propan-2-yl-1H-pyrimidin-6-one N-[4-[(Z)-2-aminoethenyl]phenyl]sulfanylcyclohexanamine 6,8-difluoro-2-(1H-pyrazol-5-yl)-4,5-dihydrothieno[3,2-d][1]benzazepine 2-ethoxy-6,7-dihydroindolo[1,2-a]quinoxaline N-[[5-chloro-2-(3-methylpyridin-2-yl)pyrazol-3-yl]methylideneamino]aniline 5-[1-[2,3-dichloro-4-(6-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)phenyl]ethenylamino]-3-iodo-N'-methylpyridine-2-carboximidamide N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-methyl-1-[[1-[1-[3-[2-[methyl(propyl)amino]ethoxy]benzoyl]piperidine-4-carbonyl]-2,3-dihydroindol-5-yl]methyl]-6-methylidenepyrimidine-4-carboxamide 3-[3,5-bis(trifluoromethyl)phenyl]butanal 2-[[3,5-dimethoxy-4-(4-methylcyclohexa-1,3-dien-5-yn-1-yl)phenyl]carbamoylamino]-N-methylbenzamide 2-[2-(4,5-dihydropyrimidin-1-ium-2-yl)phenoxy]ethanol 3-(5,7-dichloro-2,4-dioxo-1H-quinazolin-3-yl)-N-[2-(6-methoxypyridin-3-yl)ethyl]propanamide (E)-N'-[1-[2-(difluoromethyl)phenyl]ethylideneamino]-3,4-bis[4-(2-methoxyethoxy)phenyl]-N-propan-2-ylbut-3-enimidamide (7S)-2-[(3,4-dichlorophenyl)methylsulfanyl]-5-methyl-N-pyridin-3-yl-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 2-(6-azido-5,7-dimethoxyquinolin-4-yl)oxyethanol N-(3-fluorophenyl)-2-propanoylpentanediamide 4-azido-2-methylsulfanyl-5,6,7,8-tetrahydroquinazoline 4-[2,5-dimethyl-4-(4-propanoylpiperidin-1-yl)phenyl]-7-N-propan-2-yl-3H-pyrrolo[2,3-d]pyrimidine-2,7-diamine 3-cyclopropyl-3-[3-[4-(5,6,7,8-tetrahydropyrido[2,3-b]azepin-9-yl)pyrazol-1-yl]phenyl]propanoic acid 1-[2,5-dichloro-3-(trifluoromethyl)phenyl]-4-ethynoxy-5,8-dioxo-9H-carbazole-4-carboxylic acid 6-tert-butyl-3,5,6-trimethoxycyclohexa-1,3-diene;1-(2,4,6-trimethoxyphenyl)propan-1-one 2-(6-methylpyridin-3-yl)oxy-N-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)cyclohexylidene]propanamide N-[[1-cyclohexyl-4-(4-hydroxyphenyl)piperidin-4-yl]methyl]naphthalene-2-carboxamide [4-[1-(2,3-dihydroindol-1-yl)ethenyl]-2,6-bis(trichloromethyl)phenyl]phosphane;ethene 2-[4-[[6-[2,5-dimethyl-4-(2-methylsulfonylethyl)phenyl]pyridin-3-yl]methoxy]-1-benzothiophen-2-yl]acetic acid 2-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]aniline [4-(4-amino-3-methylpiperidine-1,4-dicarbonyl)-2,6-dichlorophenyl]azanium 3-[[7-(6,7-dimethoxyquinolin-4-yl)oxy-1H-indol-3-yl]oxy]-N-(pyridin-2-ylmethyl)benzamide 7-[2,3-dihydroxypropyl(octyl)amino]-5-hydroxynaphthalene-2-sulfonic acid 4-[4-hydroxybutyl(2-methylpropanoyl)amino]benzoic acid N-[2-[3-(dimethylamino)propyl]phenyl]-5-methyl-6H-indolo[1,2-c]quinazoline-12-carboxamide 4-(4,6-dimethoxypyrimidine-2-carbonyl)thiomorpholine-3-carboxylic acid 2-[2,6-bis(2-methylbutan-2-yl)-4-phenylphenyl]ethoxy-chlorophosphinite 1-[3,5-bis(trifluoromethyl)phenyl]-2-chloro-N'-(4-iodophenyl)sulfonylethane-1,2-diamine 4-[[2,6-bis(trifluoromethyl)phenyl]iminomethyl]-3-hydroxy-1H-imidazol-2-one [4-[6-(aminomethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]-cyclobutylmethanone 2-[4,5-dimethyl-N-(2-phenylethyl)-2-phenyldiazenylanilino]acetamide N-[(3S)-1-acetylpiperidin-3-yl]-7-methoxy-4-oxo-1H-quinoline-3-carboxamide (2-azidophenyl)-cyclopentylmethanone [(1R,2S)-1-methoxy-3-naphthalen-2-yl-1-oxopropan-2-yl]sulfanium 7-bromo-1-cyclopropyl-8-(methoxymethyl)imidazo[4,5-c]quinoline 3-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-7-(2-ethylhexoxy)isoquinoline 6-[1-(cyclopropanecarbonyl)piperidin-3-yl]oxypyridine-2-carboxylic acid 2-[[4-[3-(dimethylamino)pyrrolidine-1-carbonyl]phenyl]iminomethyl]-6,7-dimethoxynaphthalen-1-ol 2-(3,4-dihydroxyphenyl)-5-[4-(trifluoromethyl)phenyl]sulfonylbenzenesulfonic acid 4-(2,3-dihydro-1H-indene-5-carbonylamino)butanoic acid;ethane 3-(4-fluorophenyl)sulfinylpropanenitrile 3-methyl-4,5-dihydroimidazo[1,2-a]quinoline-2-carboxylic acid 2-[(3,5-dibromopyridin-4-yl)methoxy]quinoline 1-(3,5-difluorophenyl)-N-[(2S,3R)-2-hydroxyoxolan-3-yl]pyrazole-4-carboxamide (5Z)-5-[(4,5-dimethylfuran-2-yl)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione 2-[4-azido-3,5-dimethyl-2-(2,3,6,7-tetrahydrooxepino[3,2-b]pyridin-4-yl)phenyl]ethanamine 3-(N-butanoyl-4-methoxyanilino)propanoic acid (3S)-6-[[4,7-dichloro-2-(4-ethylcyclohexyl)pyrrolo[1,2-a][1,5]benzodiazepine-10-carbonyl]amino]-3-hydroxyhexanoic acid 2-[6-oxo-5-(4-pyrrolidin-1-ylphenyl)-3,4-dihydropyridin-1-yl]acetic acid N-[[(2S)-1-[4-[5,7-dichloro-2-(fluoromethyl)benzimidazol-1-yl]butanoyl]pyrrolidin-2-yl]methyl]ethanesulfonamide 2-(4-ethoxyphenyl)-5-methyl-3-phenylmethoxy-1,3-dihydropyrazole 3-(4,6-dihydroxy-1-benzofuran-2-yl)-1H-indole-7-carboxamide 5-(2,4-difluorophenyl)-1,3-bis(2-methylsulfonylethyl)benzimidazol-1-ium 4-[2,6-di(propan-2-yl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile N-(2,6-dichlorophenyl)sulfonyl-4-fluoro-1H-indazole-3-carboxamide N-(4-bromobutan-2-yl)-N-tert-butyl-5-chloropyridin-2-amine 5-[3,4-bis(ethenyl)phenyl]-2-methoxy-N,N-dipropylaniline 2-[(5-azido-1,3,4-oxadiazol-2-yl)methoxy]ethanol 6-[2-(oxan-4-yl)ethynyl]quinoxaline 4-methyl-N-(oxolan-2-ylmethyl)-N-(1,3-thiazol-5-yl)benzenesulfonamide 4-methyl-1-(2-phenylpyridine-3-carbonyl)piperidin-4-ol 2-[4-(4,5-dihydro-1H-imidazol-2-yl)-3-hydroxyphenyl]-N-[2-(furan-2-yl)ethoxy]acetamide 2-bromo-5,7-dimethoxy-3H-pyrido[3,4-d]pyrimidin-4-one N-[2,4-difluoro-3-[1-[[6-(trifluoromethyl)pyridin-3-yl]amino]ethylideneamino]phenyl]-1-methylcyclopropane-1-carboxamide 1-(benzenesulfonyl)-5-methoxy-4-methyltriazole N-[3-(2,4-dihydroxyphenyl)pyrazolo[1,5-a]pyridin-7-yl]benzamide 2-[4-chlorobutyl(pyridin-3-yl)amino]benzenesulfonic acid 2-[5-carbamoyl-9-[(4,6-dichlorocyclohepta-1,3,6-trien-1-yl)methyl]-2-thiophen-2-ylcarbazol-4-yl]peroxyacetic acid 2-(4-nitrophenyl)-4H-1,3-benzodioxine 5-(furan-3-yl)-4-[7-propanoyl-6-(trifluoromethoxy)spiro[2,1-benzodiazepine-3,4'-piperidine]-1'-carbonyl]pyridazine-3-carbonitrile 5-(4,6-dichloro-2H-chromen-3-yl)-N-phenyl-1,3,4-oxadiazol-2-amine 3-[(4,7-dioxo-1,4a,5,6,8a-hexahydropyrazolo[3,4-d]azepin-2-yl)methyl]-N-ethylbenzamide 4-(1-amino-2,6-dihydro-1H-pyrido[3,4-d]pyrimidin-7-yl)-N-(2-methoxypyridin-4-yl)benzamide (5Z)-3-(4-bromophenyl)-N-[4-(morpholin-4-ylmethyl)phenyl]-5-(pyridin-2-ylhydrazinylidene)-4H-1,3-thiazol-2-imine (Z)-3-amino-4,4,5,5-tetramethyl-1-phenylhept-2-en-1-one N-[(2-ethylnaphthalen-1-yl)methyl]pyrimidine-4-carboxamide N-[4-(1,3-dioxolan-2-yl)butan-2-ylidene]-5-phenylsulfanyloxypyrimidine-2-carboxamide 1-[2,4,6-trimethyl-3-(3-oxopentanoyl)phenyl]ethanesulfonic acid 2-amino-6,8-dimethyl-1-propan-2-yl-N-[4-(trifluoromethoxy)phenyl]imidazo[1,5-a]pyrazine-3-carboxamide 5-(2,6-dimethoxyphenyl)-3-iodo-1H-pyrrolo[2,3-b]pyridine 1,2-dichloro-5-ethoxybenzene;ethane 4-[4-[[2-[(6-chloropyridin-3-yl)methyl]-5,7-dihydroxy-3-methoxy-4H-pyrazolo[4,3-d]pyrimidin-6-yl]sulfanyl]phenyl]-2-methylbut-1-ene-2-thiol 2-(4-bromophenyl)-5,6,7,8-tetrahydro-3H-pyrido[4,3-d]pyrimidin-4-one (5-tert-butyl-2-methoxy-4-methylsulfonylphenyl)boronic acid N-(2,4-dibromophenyl)-2,3-dihydroxybenzamide 4-[[7-(2,6-difluorophenyl)-8-oxo-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-N'-ethyl-3-methoxybenzenecarboximidamide 2-amino-N-[4-(azidomethyl)-3,5-bis(trifluoromethyl)phenyl]pentanamide N'-hydroxy-5-[methyl(1H-pyrazol-4-yl)amino]pyrazine-2-carboximidamide 7-[5-azido-6-(3-chloropropyl)pyridin-2-yl]quinoxaline N-[5-(3,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-2-(oxan-4-ylamino)benzamide 2-azido-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine 2-[7-(azidomethoxy)-6-(difluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]ethanamine 1-[(2R)-3,4-dihydroxy-4-methylpentan-2-yl]-3-methylpyridin-2-one 5-[6-(4-methoxyphenyl)-2,3-dihydropyrrolo[2,3-b]pyridine-1-carbonyl]-N-propan-2-yl-1H-indole-7-carboxamide 5-[1-[4,6-di(propan-2-yl)pyrimidin-2-yl]imidazol-2-yl]-2H-triazole 2-[4-(2,3,5,6,7,8,9,10-octahydroanthracen-1-yl)phenoxy]acetic acid 1-[2,4-dimethyl-5-(1-methylpyrrolidin-3-yl)oxyphenyl]-N-methylethenamine N-[2,4-difluoro-3-(5H-pyrrolo[2,3-b]pyrazine-7-carbonyl)phenyl]propane-1-sulfonamide N-benzyl-7,8-dichloro-2-(methoxymethyl)-1H-imidazo[4,5-c]quinolin-4-amine 7-[(E)-1,2-diaminoethenyl]-6-[4-(trifluoromethoxy)phenyl]quinazoline-4,8-diamine 3-(4-fluoro-3-methylphenyl)propanoyl-[2-(4,5,6,7-tetrahydrobenzimidazol-1-id-2-ylamino)ethyl]carbamic acid (E)-3-[4,5-dimethyl-1-[2-(4-methylphenyl)ethoxy]cyclohexa-2,4-dien-1-yl]-N-[4-(1-formylazetidin-3-yl)oxyphenyl]prop-2-enamide 1-(azidomethyl)-3,5-bis(ethenoxymethyl)benzene 2-[4-[[(3Z)-2,6-difluorohexa-1,3,5-trien-3-yl]methoxy]phenyl]-N-hydroxypyrimidine-5-carboxamide 6-amino-5-methyl-1-(naphthalen-2-yloxymethyl)pyrimidine-2,4-dione N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-8-methylimidazo[1,5-a]pyridine-3-carboxamide;2,2,2-trifluoroacetic acid N-[2,4-difluoro-5-(methanesulfonamido)phenyl]pyrrolidine-1-carboxamide (5E)-2-(2,4-dimethylphenyl)imino-5-[[4-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl]methylidene]-1,3-thiazolidin-4-one 3-methyl-2-[4-(1,3-thiazol-5-yl)phenyl]butanoic acid 4-[4-[(1S)-6-chloro-2-(tetrazol-1-yl)-3,4-dihydro-1H-isoquinoline-1-carbonyl]piperazin-1-yl]quinazoline-8-carbonitrile (Z)-3,5,5-trimethyl-1-[2-(4-phenylbutoxy)ethoxy]hex-1-en-1-ol N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-N-(5-hydroxypentyl)cyclobutanecarboxamide N-(8-bromoquinoxalin-5-yl)-2,4,6-trimethyl-N-(4-propylphenyl)benzenesulfonamide 4-(2,6-difluorophenyl)-1H-indole 7-chloro-5,6,8-trimethoxynaphthalene-1,2-diamine N-[(3S)-2,2-dimethylpyrrolidin-1-yl]-4-[1-[4-(4-fluorophenyl)piperazine-1-carbonyl]cyclopropanecarboximidoyl]benzamide 6-ethyl-2,3-dihydrothieno[3,4-b][1,4]oxazine-4-carboxylic acid 2-(1-ethoxy-2,3-dihydronaphthalene-2-carbonyl)-4-phenylbutanenitrile 7-azido-1,3-dicyclopropyl-5H-imidazo[1,2-a]quinoxaline 5-amino-2,4-diiodobenzenesulfonic acid 6-[3-(1-phenylcyclopropyl)oxyphenoxy]hexanoic acid N-[(5Z)-5-[(3,4-dihydroxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]benzamide (2S,4R)-1-[2-oxo-3-phenyl-3-[1-[5-(trifluoromethyl)pyridin-3-yl]pyrazol-4-yl]propyl]piperidine-2,4-dicarboxylic acid N-(2,6-dimethoxypyrimidin-4-yl)-4-[2-nitro-N-(1-phenylpropyl)anilino]benzenesulfonamide 2-[4-methyl-N-(3-methylbutyl)anilino]acetic acid 3-[(2R)-5,6-dichloro-4-ethylsulfonyl-1H-inden-2-yl]benzonitrile 7-azidooxy-4,5-dichloroisoquinoline N-[1-cyclohexyl-2,4-dimethyl-6-(trifluoromethyl)-3H-quinolin-2-yl]furan-2-carboxamide N-(3,5-dichlorophenyl)sulfonyl-6-[2-hydroxyethyl(methylsulfanyl)amino]-1-benzofuran-2-carboxamide 7-fluoro-6-[3-hydroxy-4-(2H-indol-6-ylmethylidene)piperidine-1-carbonyl]-4H-chromen-3-one 3-(4-bromophenyl)benzenethiol;ethane 2-[(1S,2R)-1,4-dimethylcyclohexa-2,4-dien-1-yl]benzoic acid ethane;5-(4-fluorophenyl)sulfonyl-3,6-dihydro-2H-pyran 5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-2-chlorobenzenesulfonamide N-[2-(3-methylimidazol-4-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]propane-2-sulfonamide 2-azido-3,7-dichloronaphthalene 6-(2-chloro-3-fluorophenyl)hexanamide (3E)-4-amino-3-[(5-chloro-2-hydroxyphenyl)methylidene]azete-2-thione 4-hydroxy-2-[[3-(methylsulfonylmethoxy)benzoyl]-propan-2-ylamino]butanoic acid N-[1-(2-cyclohexylethoxymethyl)indol-3-yl]acetamide 3-(4-ethoxycarbonylphenyl)-6,7,8,9-tetrahydroimidazo[1,2-a]azepine-3-carboxylic acid 4-azido-5-methylsulfanyl-1H-indole (4Z)-2-methyl-4-[(3,5-dimethoxyphenyl)methylidene]-1,3-oxazol-5-one 2-[(3R)-1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl]oxypyridine (2Z,6E)-7-[4-amino-3-(cyclopropylmethoxy)phenyl]-5-methylideneocta-2,6-dienenitrile [5-chloro-4-(cyclobutylamino)-1H-pyrrolo[2,3-b]pyridin-2-yl]-methoxymethanol 4-[1-(benzylamino)ethenyl]-2,6-dichloroaniline 4-N,4-N-dimethyl-2-(methylideneamino)-5-[(Z)-prop-1-enyl]benzene-1,4-disulfonamide N-[4-(4,5-dimethyltriazol-1-yl)pyridin-2-yl]-3-methoxyazetidine-1-carboxamide 4-[(4R,5S)-2,6-bis(hydroxymethyl)-4,5-dihydro-1H-indol-4-yl]phenol 1-(4,6-dimethylpyrimidin-2-yl)-5-(oxolan-3-yl)spiro[2H-indole-3,3'-azetidine] 7-(1H-indole-2-carbonyl)-1',4-dimethylspiro[6,8-dihydropyrazolo[3,4-b][1,4]oxazepine-5,3'-piperidine]-3-one 2-methyl-N,5-dipyridin-3-ylthiophene-3-carboxamide 1-butylsulfanyl-4,5-dichloro-2-methoxybenzene N-[(2,4-dimethoxyphenyl)-difluoromethyl]piperidine-4-carboxamide 1-[4-chloro-6-(2,3-dimethoxyphenyl)pyrimidin-5-yl]-7,8-dihydro-6H-furo[3,2-e]indole 4-[(2R)-3-amino-4-methylpentan-2-yl]oxy-1H-benzimidazole-2-carboxamide;formic acid N-[2,6-difluoro-4-[2-(3H-isoindol-1-yl)acetyl]phenyl]-5-nitrothiophene-2-carboxamide 1-(2-methylphenyl)-4-[5-(trifluoromethoxy)-1,3-benzodioxol-4-yl]butan-2-one (E)-5-hydroxy-2,6-dimethylhept-4-enal;methoxyethane;N,3,5-trimethyl-1,4-oxazepin-7-amine 1-(2,3,3a,4-tetrahydro-1H-indole-3-carbonyl)-3,4-dihydroquinolin-2-one [3-(4,5-dimethyl-1H-imidazole-2-carbonyl)phenyl]boronic acid 4-methylsulfonyl-2,3,5,6-tetrahydro-1H-pyrrolo[2,1-c][1,4]oxazepine 4-azido-6,8-dichloro-7-hydroxychromen-2-one 5-methylsulfanylpyrimidine;4,5,7-trihydroxychromen-2-one 4-[(6R)-5,6-dihydroimidazo[2,1-b][1,3]thiazol-6-yl]benzoic acid 3-[[4,6-diamino-5-(benzenesulfonylmethyl)pyrimidin-2-yl]-methylamino]propanal 7-[(3,5-dimethylphenyl)sulfonylamino]heptanoic acid 4-[5-(1,3-dihydroxypropan-2-yloxy)pyridine-2-carbonyl]piperazine-1-carboxylic acid N-[(5R)-5-(hydroxymethyl)-2-oxo-1,3-oxazolidin-3-yl]-4-(trifluoromethylsulfanyl)benzenesulfonamide N-(6-aminopyridin-3-yl)sulfonyl-2-[7-fluoro-4-[(4,5,6-trimethoxy-1H-indol-2-yl)methyl]naphthalen-2-yl]acetamide 2-methyl-7-[(E)-3-phenylprop-2-enyl]-1,4-dihydroazepino[6,5-b]indole N-(4,6-dimethylpyrimidin-2-yl)-5-[(E)-(2-methoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide N-(5-bromopyridin-2-yl)-N-(2,4,6-trimethylphenyl)sulfonylbutanamide 6-[4-(2,5-dimethoxyphenyl)piperazine-1-carbonyl]cyclohexa-2,4-diene-1-carboxamide 4-(5-methyl-1,3-oxazol-2-yl)-N'-[1-oxo-4-phenyl-6-(pyrrolidine-1-carbonyl)phthalazin-2-yl]benzohydrazide 6-(methoxyiminomethyl)chromene-2,4-dione (2Z,5R)-2-[(Z)-1-(furan-3-yl)ethylidenehydrazinylidene]-5-methyl-1,3-thiazolidin-4-one N-[2-methyl-4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)phenyl]cyclopropanecarboxamide 1-(6-bromohexoxy)quinolin-4-one N-[(E)-(3,4-dichlorophenyl)methylideneamino]-5-(2-ethyltetrazol-5-yl)thiophene-2-carboxamide 6-bromo-N,7-dimethyl-N-(1-oxopropan-2-yl)-3,4-dihydro-1H-isoquinoline-2-carboxamide (7S)-7-[4-chloro-3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidin-5-one 4-[1,3-bis(5,6,7,8-tetrahydronaphthalen-2-yl)propan-2-yl]benzoic acid 3-(1,4-dimethyl-2-oxoquinolin-6-yl)propanoic acid (E)-3-[4-[6-(4-chlorophenoxy)pyridin-2-yl]oxyphenyl]-1-(1H-imidazol-2-yl)prop-2-en-1-one;2,2,2-trifluoroacetic acid 2-(3,5-difluorophenyl)-1,1,1,3,3,3-hexafluoropropan-2-ol 3-methyl-1,3,4,5-tetrahydrochromeno[2,3-c]pyridine 4-(2,5-difluorophenoxy)-3-phenylpyrazolo[1,5-a]pyridine 3-[3-azido-5-(4-methylpyrazol-1-yl)phenyl]cyclopentan-1-ol (2-ethylphenyl)-(4-hydroxy-3,5-diiodophenyl)methanethione N-(3-bromophenyl)sulfanyl-1,1,1,2,3,3,3-heptafluoropropan-2-amine;ethane 1-N,3-N-dimethylbenzene-1,2,3,4-tetracarboxamide 1-[2-(trifluoromethyl)pyridin-4-yl]benzimidazole 3-ethenyl-N'-(2,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-1-yl)benzenecarboximidamide 6,8-bis[4-(1,3-benzodioxol-5-ylmethylideneamino)butoxy]-3H-quinazolin-4-one 2-(3-aminocyclobutyl)-4,5-dichlorophenol (4E)-4-[(3,5-dimethoxyphenyl)methylidene]-2-ethylsulfanyl-1H-imidazol-5-one N-(1,4-dichloroisoquinolin-6-yl)sulfonylbicyclo[2.2.1]heptane-1-carboxamide 6-bromo-N-(2,4-dichloropyrimidin-5-yl)-N-(1H-indol-5-ylmethyl)pyridin-3-amine (5Z)-5-[[4,6-dioxo-1-phenyl-2-sulfanylidene-5-[(Z)-3-pyrrolidin-1-ylprop-1-enyl]thieno[3,4-d]pyrimidin-3-yl]methylidene]-1,3-thiazolidine-2,4-dione 1-[4-[2-(6,7-dimethoxyquinolin-4-yl)ethynyl]cyclohexa-1,5-dien-1-yl]-3-(4-fluorophenyl)urea (E)-1-[9,10-difluoro-2-(piperidine-1-carbonylamino)-4,6,8,11-tetrazatricyclo[7.4.0.03,7]trideca-1(13),3,5,7,9,11-hexaen-5-yl]-N-methoxyethanimine 7-tert-butyl-3,5-dihydropyrrolo[2,3-f]benzimidazol-6-one;4-fluorobenzaldehyde (Z)-3-(4-chlorophenyl)-2-cyanoprop-2-enamide 1-methylsulfanylimidazo[4,5-c]quinoline 1-azidooxy-5-(3,4-dichlorophenyl)pentan-2-ol 2-[(2S)-1-[2-fluoro-4-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethoxy)phenyl]propan-2-yl]-3-methylpyridine-4-carboxamide 1-[3,4,6-tris(ethenyl)naphthalen-2-yl]ethanone 1-[[3,5-dimethyl-2-(trifluoromethoxy)phenyl]methylideneamino]-4,4-dimethylpiperidine-4-carboxylic acid 2-[2-(benzylamino)pyrimidin-4-yl]-N-(3,4-difluorophenyl)-1H-indole-6-carboxamide 4-(1-azidopropan-2-yl)-5-chloropyridine 2-[(4-methoxybenzoyl)amino]-3-[4-(trifluoromethyl)phenyl]propanoic acid 2-[2,6-dichloro-4-nitro-N-(1,3-thiazol-5-yl)anilino]octanoic acid 6-bromo-2-(cyclobutylamino)-4-[(1-hydroxypyridin-1-ium-3-yl)methoxy]pyridazin-3-one 3-(2,6-difluorophenyl)-2-methylbenzaldehyde (4-bromophenyl)methanamine;2,2,3,5-tetramethyl-1H-indole 1-(2-tert-butyl-4,6-dimethoxypyrimidin-5-yl)ethanimine 4-[(2E,4Z)-5-methylhepta-2,4,6-trien-3-yl]oxyaniline 1,4-dihydroxy-3-[2-(4-methylbenzoyl)oxypropanoyl]naphthalene-2-carboxylic acid 4-[(1S)-2-[(3R,4S,5R)-3,4-dihydroxy-5-methyloxolan-2-yl]-6-fluoro-2-(trifluoromethoxycarbonylamino)-3,4-dihydrochromen-8-yl]benzoic acid (2R)-2,4-diamino-2-[1-(4-chloro-2,3,5,6-tetradeuteriophenyl)ethyl]butanal 6-[4-(1,1-difluoroethyl)phenyl]-3H-1-benzothiophen-2-one 4-azido-2,6-dichloro-3-cyclohexylpyridine 2-[(6-hydroxy-1H-benzimidazol-2-yl)-pyridin-2-ylamino]acetamide 1-[4-(hydroxymethyl)piperidin-1-yl]-2-methoxy-2-phenylethanone 4-[(5R)-3,5-difluoro-1-phenyloctyl]benzamide 2-(3,4,5-trimethoxyphenyl)-[1]benzofuro[3,2-d]pyrimidine 4-benzamido-2,6-difluorobenzoic acid 4-[2-(5,7-dihydroxy-1,3-benzothiazol-6-yl)ethoxy]butanehydrazide N-[(Z)-1H-indol-3-ylmethylideneamino]-6,7,8,9-tetrahydro-5H-carbazole-3-carboxamide 7-chloro-6-(3,4-dihydroquinolin-8-yl)isoquinolin-1-amine 3-[(4S)-5,7-dioxo-2-propylsulfanyl-3,4-dihydropyrimido[4,5-d]pyrimidin-4-yl]-N,1,6-trimethylindole-4-carboxamide 6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-iodo-3-[1-(2-methoxyacetyl)azetidin-3-yl]-5-nitro-1H-quinolin-2-one N-[4-bromo-2-(butylcarbamoyl)-6-chlorophenyl]-5-(4-fluorophenyl)-2-methoxypyridine-3-carboxamide 4-(4,6-dicyclohexyl-1,3,5-triazin-2-yl)-N,N-diethylaniline 2-[1,3-benzodioxol-5-ylsulfonyl-[(6R)-6-phenylnonan-4-yl]amino]acetic acid 4-(5-methylsulfonylpyrazin-2-yl)oxybutanal 2-[[4-(2,3,5-trifluorophenyl)pyridin-3-yl]methoxy]propanoic acid 4-[1-carboxyethyl(2,3-dihydroxypropyl)amino]benzoic acid 1-(2,6-difluorophenyl)-4-[4-methoxy-3-(sulfinatoamino)benzoyl]piperazine 1-methyl-N-[(1S)-1-pyridin-2-ylethyl]indole-3-carboxamide 1-[7-(4-ethylcyclohexyl)-2,3-difluoropyrazolo[1,5-a]pyrimidin-6-yl]ethenol 6-fluoro-7-[4-(1,3-oxazol-2-yl)piperazine-1-carbonyl]-2H-isoquinolin-1-one 3-[2,6-bis(2-methylpropoxy)phenyl]-N-(1H-indazol-5-yl)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-2-carboxamide 7-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-N-ethylimidazo[1,2-c]pyrimidine-3-carboxamide 5-[(Z)-1-amino-3-methyliminoprop-1-en-2-yl]-N-cyclopentyl-4-methanimidoylpyridine-2-carboxamide 3-azidosulfanyl-N,2,4-trimethoxybenzamide 3-(1H-indazol-5-yl)propanoic acid;4-methoxy-2,6-dimethylbenzenethiol (5E)-2-[(Z)-2-[4-[(2,4-dichlorophenyl)methoxy]-3-ethoxyphenyl]ethenyl]-6-imino-1,3-thiazinan-4-one 5-[[4-(3,4-dimethoxyphenyl)sulfonylpiperazin-1-yl]methyl]-4-pyridin-2-ylpyrimidine;hydrochloride 3-[(3aR,6aR)-2-cyclobutyl-5-oxo-1,3,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-4-carbonyl]benzoic acid 2-[3-methoxy-4-(propylamino)phenyl]acetic acid 5-(2-azidoethyl)-3,4-dihydroisochromene-1,6-dione 3-bromo-N'-(1,5-dichlorohexyl)-4-fluorobenzenecarboximidamide (1S,2R)-3-[5-chloro-6-[3-fluoro-4-(triazol-1-yl)anilino]pyrazolo[1,5-a]pyrimidin-2-yl]cyclohexane-1,2-diamine (Z)-2,6-dimethylidene-N'-[1-[4-(trifluoromethylsulfonyl)phenyl]ethyl]oct-3-enimidamide 5-[4-(1-azidohexan-3-yl)phenyl]-2H-tetrazole N-(2,6-difluorophenyl)-N-[1-methyl-3-(pyrrolidin-1-ylmethyl)pyrazole-4-carbonyl]-2H-pyridine-1-carboxamide 5-[(4-bromothiophen-3-yl)methylamino]imidazo[1,2-c]pyrimidine-8-carbonitrile 5-bromo-3-butylsulfonyl-1H-pyridin-2-one 1-[[4-(dimethylamino)phenyl]methyl]-3-[2,2,6,6-tetradeuterio-5-fluoro-4-[3-(trideuteriomethoxy)-5-(trifluoromethyl)pyridin-2-yl]phenyl]urea (2S)-2-azido-1,3,4-trimethyl-5-phenylpyrrole (1Z)-3-benzyl-2,4-dimethyl-1-sulfanylidenepenta-1,3-dien-3-olate (5E)-5-[[4-[3,5-bis(trifluoromethyl)phenyl]furan-2-yl]methylidene]-2-(4-ethoxyphenyl)imino-1,3-thiazolidin-4-one 3-(2,2-dimethylpentanoyl)benzenesulfonic acid 3-azido-5,7-dimethylimidazo[1,2-a]pyrimidine 2-cyclopropyl-4-methoxy-1-[6-(3,3,3-trifluoropropoxy)pyridin-3-yl]indole 1-(4-bromopyridin-2-yl)-3-cyclopentylurea 1-(3,5-difluorophenyl)-2-[(7R)-4-hydroxy-6,11-dioxo-8-oxa-12-azatetracyclo[7.7.0.02,7.010,15]hexadeca-2,4,9,13,15-pentaen-3-yl]guanidine 2-(1,5-dimethylimidazol-4-yl)sulfonyl-N-hydroxyacetamide (3R,5S)-1,3-bis[2-[(1S)-2-[(E,4Z,6E)-8-chloro-4-ethylidenedeca-6,9-dienyl]cyclopentyl]oxycarbonyl]-7-imino-4-oxoheptane-2-sulfonic acid N-[(4R)-2-oxo-1,3-oxazolidin-4-yl]-7H-purine-6-carboxamide 2-[(5-aminopentylamino)methyl]-3H-quinazolin-4-one 2-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-6-(5-ethoxypyrimidin-4-yl)quinoxaline 3-[(6,8-dimethoxyquinazolin-4-yl)amino]oxolane-2,5-dione 5-[(E)-(5-hydroxy-2,3-dihydroinden-1-ylidene)methyl]-N,4-diphenyl-1H-pyrrole-3-carboxamide 5-azido-6-(methoxymethyl)-1,3-benzodioxole 2,3-difluoro-1-[4-(4-propoxyphenyl)cyclohexyl]-4-(trifluoromethyl)benzene N-[6-amino-2,4-bis(ethenyl)pyridin-3-yl]-2-chlorobenzamide (4E)-2,2-dimethyl-4-[[6-nitro-5-[2-(trifluoromethoxy)phenyl]-1H-benzimidazol-2-yl]methylidene]oxan-3-one (5S)-N-(3,4-dimethylphenyl)-2-[(2Z)-2-[(Z)-(3-nitrophenyl)methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetamide 3-methylsulfanyl-4,6-diphenylbenzene-1,2-disulfonic acid 2-amino-4-[5-(3,5-dichlorophenyl)furan-2-yl]-6H-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-dithione 3-(difluoromethoxy)-2,6-bis[(4-ethenylphenoxy)methyl]pyridine 3-(6-methyl-1H-benzimidazol-2-yl)cyclopropane-1,1,2-triol 4-[2,3-dichloro-6-(hydroxymethyl)phenoxy]benzonitrile (5S,7R)-2-methylsulfanyl-N-phenyl-5-thiophen-2-yl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide N-[(3,5-dimethylphenyl)methyl]-4-(1H-indazole-3-carbonyl)morpholine-2-carboxamide 5-(5,6-dimethyl-1H-benzimidazole-2-carbonyl)-N,7,8,9-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-10-carboxamide 4-[(2E,4Z)-5-fluorohepta-2,4,6-trienyl]sulfanyl-N-(3-imidazol-1-ylpropyl)benzamide 2,4-dichloro-N-(2-fluorophenyl)-5-[3-iodo-1-(methylsulfanylamino)propyl]aniline (6S,9R)-6-(furan-2-ylmethyl)-1,4-dimethyl-5,7,8,9-tetrahydropyrazolo[3,4-b]quinoline 2-methyl-3-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carbonyl)azetidin-3-yl]oxybenzonitrile 5-chloro-N'-[1-(2,3-dihydro-1H-inden-2-yl)-4-hydroxybutan-2-yl]pyridine-3-carboximidamide 6-(3,5-dichloropyridin-4-yl)oxy-1',1'-dimethylspiro[3H-chromene-2,4'-piperidine] 1-[(3R,4S)-2-hydroxy-5-[(3R)-3-phenylpyrrolidine-1-carbonyl]-4-thiophen-3-ylpiperidin-3-yl]ethanone;hydrochloride (2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-1-ethanimidoyl-4,4,4-trifluoro-N'-(4-fluorophenyl)butanediamide 2-(3-chlorophenyl)sulfanyl-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-5-ylmethyl)acetamide 4-[(3S,5S)-3,5-dimethyl-2-oxoheptan-3-yl]benzonitrile N-(3,4-dihydro-2H-pyrano[3,2-b]pyridin-4-ylmethyl)-2,2-difluoroacetamide (4R,5S)-1-(cyclopentylmethyl)-2-oxo-3,4,5,6-tetraphenylcyclohexane-1-carbonitrile 7-[(E)-2-[4-[bis[(3-fluorophenyl)methyl]amino]phenyl]ethenyl]-N,N'-diethylquinoxaline-6-carboximidamide (4S)-4-[6-[3,5-dimethyl-4-[(2-methylpyridin-3-yl)oxymethyl]pyrazol-1-yl]pyrimidin-4-yl]-1-methylpyrrolidin-2-one 5-[3-(2-ethylphenyl)propanoyl]-N,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide 5-[2-(benzylamino)phenyl]pyrimidine-2,4-diamine (4R)-N-[(2,4-difluorophenyl)methyl]-8-(3,4-dihydroxyphenyl)-2-ethynyl-7-hydroxy-1,6-naphthyridine-5-carboxamide 4-azidosulfonylbenzoic acid 1-N,3-dimethyl-6-nitronaphthalene-1,2-disulfonamide 4-[[2-methoxyethyl(methyl)amino]methyl]benzoic acid;5,7,8,10-tetrahydropyrimido[4,5-b]quinoline 5-(4-fluorophenyl)-N-[2-methyl-1-oxo-1-[4-(3,4,5-trimethoxyanilino)quinazolin-6-yl]propan-2-yl]pentanamide 1-[2,6-dibromo-4-(6-methyl-5-oxopyrido[3,4-d]pyrimidin-4-yl)oxyphenyl]-N-ethyl-1-methylpiperidine-2-carboxamide 3-[(1,2-dimethylindol-4-yl)amino]cyclohexane-1-carboxylic acid N-(4-azidophenyl)-6,7-dimethoxyquinazolin-2-amine 3-(2-aminoethyl)-5,6-dichloro-1H-pyrimidine-2,4-dione 2-(4-chlorophenyl)-N-[3-methylsulfanyl-1-oxo-1-[4-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-ylamino)piperidin-1-yl]propan-2-yl]acetamide 5-butyl-1,3-benzodioxole 4-amino-1-benzylsulfonylazepan-3-one N-[(2S)-1-amino-4-methylsulfanylbutan-2-yl]-5-chlorothiophene-3-carboxamide N-[1-(2,4,6-trimethylphenyl)ethenyl]ethanimine (E)-1-N',2-N'-bis[(4R)-8-chloro-2-methyl-3,4-dihydrochromen-4-yl]but-1-ene-1,1,2,2-tetraamine 1-(2-azidoethyl)-4-phenoxybenzene [3-amino-2-(aminomethyl)phenoxy]boronic acid 3-(diethylaminomethyl)-6-[5-[4-(trifluoromethoxy)phenyl]furan-2-carbonyl]-1,4,5,7-tetrahydropyrazolo[3,4-c]pyridine-4a-carboxylic acid 2-[(4R)-7-bromo-3,4-dihydro-2H-chromen-4-yl]acetic acid 2-[(4R)-4-(6,7-dimethoxyquinazolin-4-yl)oxypyrrolidine-1-carbonyl]benzoic acid N-(2,6-dimethoxypyrimidin-4-yl)-4-[(5-oxo-6-phenyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]benzamide 5-chloro-N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-(6-fluoroquinolin-4-yl)oxybenzenesulfonamide (4S)-2-N,4-N-diethyl-3-phenylpentane-1,2-diamine 2-[4-(benzoylsulfamoyl)-N-phenacylanilino]propanoic acid 3,4-bis(ethenyl)-2-(5-methoxypyridin-3-yl)thiophen-1-ium N-[4-(1,2-dihydroazet-3-yl)phenyl]piperidine-4-carboxamide [1-(3,5-difluorophenyl)pyrazol-4-yl]-[4-(dimethylamino)azepan-1-yl]methanone 1-[(4,5-dichlorothiophene-2-carbonyl)amino]-3-(2-phenylethyl)urea 3-cyclopentyloxypyridine-4-carboxylic acid 2-(4,5-diethylthiophen-3-yl)oxyacetamide 4-[(2-methoxy-5-nitrophenyl)diazenyl]-3,6-bis(sulfanylidene)cyclohexa-1,4-diene-1-carbonitrile N-(1H-benzimidazol-2-yl)-6-chloropyrazolo[1,5-a]pyrimidine-3-carboxamide 3-[4-(azidomethyl)-2,6-difluorophenyl]prop-1-en-2-ol 3-(1H-benzimidazol-2-yl)-7,8-dichlorochromen-4-one 5-azido-4-(2-chlorophenyl)sulfanyl-3,6-dimethoxy-1H-indole 5-[3,4-dimethyl-2-(trifluoromethoxy)phenyl]imidazolidine-2,4-dione 2,3-dichloro-4-methylsulfonylaniline N'-[5-[4-(2-aminopropanoyl)piperazine-1-carbonyl]-4-chlorocyclohexa-1,3-dien-1-yl]thiophene-2-carboximidamide;ethane N-[1-[4-chloro-3-(trifluoromethyl)phenyl]piperidin-2-ylidene]nitramide N-[(E)-1H-indol-3-ylmethylideneamino]benzamide 5-[2,3-difluoro-4-(trifluoromethyl)phenoxy]-1H-indazole 7-methylsulfonyl-2-[1-(pyridine-4-carbonyl)piperidin-3-yl]-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 2-[4-chlorobutyl(4,5-dimethyl-2-phenyldiazenylphenyl)amino]decanoic acid N-[1-(methoxymethyl)-4,5-dihydroimidazol-2-yl]-3-propan-2-yl-1H-pyrrolo[3,4-c]pyridine-6-carboxamide 3-ethylsulfonyl-N,4-dimethylpyridine-2-carboxamide 1-[(4R)-7,8-dimethoxy-2-oxospiro[3H-chromene-4,1'-cyclohexane]-1-yl]pyrrole-2,5-dione N-azido-2,5-dichloro-1-[4-(furan-2-yl)benzoyl]indole-3-carboxamide (1R,2R)-2-N-[3-fluoro-4-methyl-5-(trifluoromethyl)phenyl]cyclohexane-1,2-diamine;hydrochloride N-benzyl-6-chloro-N,2,3,4-tetramethylaniline (3R)-5,10-dioxo-N,4-bis(phenylmethoxy)-1,2,6,8-tetrahydrobenzo[c]chromene-3-carboxamide 3-azido-N-[2-(3,4-dimethoxyphenyl)ethyl]aniline 2-[4-[3-amino-5-(cyclopropylcarbamoyl)pyridin-2-yl]phenyl]-N-[[2-(difluoromethoxy)-6-(tetrazol-1-yl)phenyl]methyl]acetamide 1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-[3-fluoro-5-(methanesulfonamido)phenyl]-4-methoxycyclohexa-2,4-diene-1-carboxamide [3-methyl-3-(methylamino)pyrrolidin-1-yl]-(6-pyridin-2-ylpyridin-2-yl)methanone N-ethyl-4,6-dimethyl-7-[[2-(trifluoromethoxy)phenyl]methylsulfanylamino]heptanamide N-(2,3-dihydro-1H-indol-5-ylmethyl)-4-[5-fluoro-6-[2-methoxyethyl(methylsulfonyl)amino]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide 3,4-difluoro-2-(trifluoromethyl)phenol 2-[N-(benzenesulfonyl)-4-bromoanilino]acetamide 1,4-diamino-2-(trifluoromethyl)anthracene-9,10-dione 2-[4,6-di(propan-2-yl)pyrimidin-5-yl]sulfanyl-N,N-bis(4-fluorophenyl)acetamide 2-(4,6-dimethoxypyrimidin-2-yl)iminoacetic acid 5-N-(3,3-dimethylpiperidin-1-yl)-2-ethanimidoylbenzene-1,4-diamine (1R,5S)-7-benzyl-2-chloro-2-azabicyclo[3.2.0]heptane 5-[4-(6-chloroquinolin-7-yl)phenyl]hexanal;N-methylmethanamine (4R)-4-[6-(cyclopentylmethoxy)pyridin-3-yl]-1,3-dimethyl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one (3E)-4,6-dimethyl-2-methylidene-N-[(3R)-piperidin-3-yl]-5-oxo-7H-1-benzofuran-3-carboxamide (2S,3R)-4,5-dimethoxy-2,3-bis[(1S,2S)-2-methylcyclopropyl]-1-phenylpentan-1-one 3-[(E)-2-(5,5-dimethyloxolan-3-yl)ethenyl]pyridine N-[[4-(trifluoromethyl)phenyl]methyl]-2,3,4,5-tetrahydropyrrolo[3,2-f]benzimidazole-1-carboxamide 3-[2,4-bis(trifluoromethyl)phenyl]-5-[1-(4-chloroanilino)ethenyl]oxolan-2-one 1-but-3-enyl-4-[(Z)-3,7-dimethoxyoct-2-en-2-yl]benzene N-[4-(dimethylamino)phenyl]-2-nitro-N-octylbenzamide N-(3,5-dichlorophenyl)-4-nitro-N-prop-2-enylbenzamide (3,5-difluorophenyl)-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]piperidin-1-yl]methanone (3E)-3-[[4-(aminomethyl)phenyl]sulfonyl-methylhydrazinylidene]-5,5,8,8-tetramethyl-6,7-dihydronaphthalene-2-carboxylate 2-N,6-N-bis(1H-benzimidazol-2-ylmethylideneamino)pyridine-2,6-diamine;ruthenium(2+);chloride 4-[2,3-difluoro-4-(methoxymethyl)phenyl]aniline 5-methyl-4-[(2Z,3E)-2-propylidenehexa-3,5-dienoxy]-1H-pyrazole 4-(4-pyridin-2-ylpiperazine-1-carbonyl)cyclohexane-1-carboxylate 4-amino-3,5,6-trichloro-N-(4-chloropyridin-2-yl)pyrazine-2-carboxamide 2-[2,6-difluoro-4-(trifluoromethyl)phenyl]-5-heptan-3-ylpyridine 6-[(2R)-butan-2-yl]-3-ethoxy-8-methylidene-4,5,7,9,10-hexahydrobenzo[g]indazole 4-cyclohexa-1,5-dien-3-yn-1-yl-2-(6-methoxypyridin-2-yl)-1H-pyrimidin-6-one N-(2-methylphenyl)-1,3-dioxopyrrolo[2,3-c]pyridine-2-carboxamide (5S)-2-(3,4-dihydro-1H-isoquinolin-2-ylmethylimino)-5-[(4-iodophenyl)methoxy]-1,3-thiazolidin-4-one (4R)-3-methyl-1-(2-phenylethyl)piperidin-4-ol 3-[2-[[5-(3,4-dimethoxyphenyl)tetrazol-1-yl]methyl]pentanoylamino]propaneoic acid ethane;4-(4-oxopiperidin-1-yl)benzaldehyde 5-[(2-methoxynaphthalen-1-yl)diazenyl]-3H-1,3,4-thiadiazol-2-one 5-azidooxy-2-(3,4-dimethylphenoxy)pyridine 3-(azidomethyl)-1,6-dibenzylpiperidine (E)-3-[1-[4-(5,6-diethoxy-7,8-dimethylnaphthalen-2-yl)cyclopenta-1,3-dien-1-yl]ethenylsulfanyl]-N,N-bis(prop-2-ynyl)but-2-en-1-amine 2-chloro-7-(1-cyclopropylpyrazol-3-yl)-6,8-dihydropyrimido[5,4-d]pyrimidine 7-(9H-fluoren-9-ylmethoxycarbonylamino)-3,5-dimethylideneheptanoic acid 3-[[2-(3,4-dichlorophenyl)acetyl]amino]-N-[2-(1,3-dioxoisoindol-2-yl)ethoxy]-1H-pyrazole-5-carboxamide 1,5-bis(3-chloropyridin-2-yl)-4-hydroxypentan-3-one 3-[(4-methylpiperazin-1-yl)methyl]-N-phenyl-2H-indazole-6-carboxamide 7-(3,4-dimethylphenyl)-2,5-dimethylheptanoic acid (7S)-N-(2,4-dimethoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 2-(6,7-dimethyl-3H-quinazolin-4-ylidene)guanidine N-[3,5-dichloro-4-(6,7-dimethoxyquinazolin-2-yl)oxyphenyl]-1-(4-fluorophenyl)-3-oxo-2-phenylpyrazole-5-carboxamide (2Z)-3-[3,5-bis(trifluoromethyl)phenyl]-2-[(Z)-prop-1-enyl]penta-2,4-dienenitrile 1-(4-azidooxyphenoxy)-2,3-dimethylbenzene 4-[2-(4-hydroxyphenyl)ethyl]benzaldehyde;4-[[5-[4-(oxiran-2-ylmethoxy)phenyl]thiophen-2-yl]methyl]phenol 7-bromo-2,5-dimethyl-N-[4-(trifluoromethoxy)phenyl]-[1,3]oxazolo[4,5-b]pyridine-6-carboxamide;cyclobutanamine (5E)-2-(4-ethoxyphenyl)imino-5-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one 7-chloro-4-(methylamino)chromen-2-one;ethane 7-[3-[4-(1-ethoxypropan-2-yl)piperazin-1-ium-1-ylidene]piperidin-1-yl]-5,6-dimethylpyrazolo[1,5-a]pyrimidine N-(3-nitrophenyl)-N-(3-nitrophenyl)-4-phenoxyaniline 1-(cyclohexa-2,4-dien-1-ylmethoxy)-3-[4-(1H-imidazole-5-carbonylamino)phenoxy]propane-2-carboxylic acid 1,2-dichlorobenzene;N-[4-(3-methylimidazole-4-carbonyl)phenyl]propanamide N-[5-(2,3-dihydrothiophen-5-yl)pyridin-3-yl]-6-fluoro-4-oxo-1H-pyridazine-3-carboxamide N-[(Z)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-2-[(1S)-3-oxocyclohexyl]acetamide 1-(3,5-difluorophenyl)-5-iminopyrrolidine-2,4-dione 2-[4-[(1S)-3,3a,4,5,6,7,7a-octahydro-1H-indene-1-carbonyl]piperazin-1-yl]pyridine-3-carboxylic acid 6-[(4-aminophenyl)diazenyl]-2,3-bis(hydroxymethyl)phenol [(3-chlorophenyl)methyl-propylamino]oxy-hydroxy-oxophosphanium 2-[(4R)-4,8,12-trimethyltridecyl]benzenesulfonic acid N-[(E)-but-2-enyl]-5,6-diethoxypyridine-3-carboxamide 1-ethylsulfonyl-3-[6-(2H-tetrazol-5-yl)-7,8-dihydroimidazo[1,2-a]pyrimidin-2-yl]urea 2-[3-[(5,6-diethoxypyridin-2-yl)-methylsulfonylamino]phenyl]acetamide 3-(2,6-dimethylphenoxy)-4-methoxyaniline 1-(cyclohexa-2,4-dien-1-ylmethoxy)naphthalene 2-chloro-4-ethyl-6,7,8,9-tetrahydropyrimido[4,5-d]azepine 4-[(3,5-diamino-6-chloropyridine-2-carbonyl)amino]pentanedioic acid 5-[5-(1,3-benzodioxol-4-yl)-7H-cyclopenta[b]pyridin-2-yl]-3-methyl-2H-pyrazolo[3,4-b]pyridine 5-[3-(2-acetamidoethylcarbamoyl)phenyl]-1-[4-(cyclohexa-1,5-dien-1-ylamino)benzoyl]pyrrolidine-2-carboxylic acid 5-amino-N,1-diethylpyrrolo[3,2-b]pyridine-7-carboxamide 3-(dimethylamino)-1-(2,4-dinitrophenyl)propane-1,3-dione ethane;3-methyliodanuidylbenzenethiol 4-ethoxy-5,6-dimethyl-N-(2-phenylpropan-2-yl)pyrimidine-2-carboxamide N-[2-(2,4,6-trimethylphenyl)sulfanylethyl]butane-1-sulfonamide 1-[(2S,3R)-4-methylsulfanyloxolan-3-yl]-N-(5-phenylpyridin-2-yl)benzimidazole-2-carboxamide 3-methoxy-4-(4,7-dihydroxynaphthalen-1-yl)sulfonyloxybenzenesulfonate N-[3-cyano-6-[4-(trifluoromethyl)phenyl]pyridin-2-yl]-3-fluoroazetidine-1-carboxamide N-[(6R)-3,5,12-trimethyl-9-oxo-2-thia-8,11-diazatetracyclo[8.4.0.02,6.07,10]tetradeca-1(10),3,11,13-tetraen-14-yl]acetamide 5-[2-(4,5-dimethyltriazol-1-yl)ethoxy]-4-phenyl-3-piperidin-1-ylpyridazine N-[4-[(7aS)-8-oxo-3-phenyl-5,6,7,7a-tetrahydroimidazo[1,2-a]pyrazine-1-carbonyl]phenyl]propane-1-sulfonamide 3-methyl-1,2-dihydrobenzo[e]indole-7,6-disulfonic acid N-(3-bromobutyl)-N-cyclohexyl-5-nitro-1,3-thiazol-2-amine 3,4-bis(ethenyl)fluorene-1,2-disulfonic acid 2-[(4Z,6E)-8,9-dichloronona-3,6,9-trienyl]-3,5-dimethylimidazo[1,5-a]pyridine-7-carbonitrile N-[4-(2,3,5,6,7,8-hexahydro-1H-pyrrolizine-1-carbonyl)phenyl]-2-[(2R)-1-(naphthalen-2-ylsulfonylamino)propan-2-yl]butanediamide 5-methoxy-2,3,4-trimethyl-6-phenylphenol N-methoxy-2-[[4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl]amino]propanamide 5-[3,4-difluoro-2-(trifluoromethyl)phenyl]imidazolidine-2,4-dione 3-hydroxy-1,4-dioxoisoquinoline-6,8-disulfonic acid;hydrate N-azido-N',2-dimethylbenzo[e]azulene-1-carboximidamide 5-(2,3-dihydro-1H-inden-4-yl)-N-[2-(4-methoxyphenyl)ethyl]-6-methylpyrazin-2-amine N-(1,3-benzodioxol-5-yl)-2-(3-bromophenyl)-5-methylidene-7,8-dihydropyrimido[4,5-d]pyrimidin-6-amine (7R)-2,4-dioxo-N-[3-[4-(trifluoromethyl)phenyl]propyl]spiro[1H-quinoline-3,3'-pyrrolidine]-6-carboxamide (2R,3S)-2-[4-chloro-5-ethyl-1-methyl-6-(4-piperidin-1-ylphenyl)benzimidazol-2-yl]thiolan-3-ol 4-[4-[2,3-dihydroxypropyl(phenacyl)amino]phenyl]-N-(oxolan-2-ylmethyl)-1,3-thiazol-2-amine 2-(3,5-dimethylbenzene-6-id-1-yl)quinoline;(Z)-6-hydroxy-2,8-dimethylnon-5-en-4-one;iridium 2-[(3,4-dimethylphenyl)methylamino]-5,6,7,8-tetrahydro-1H-pyrido[3,4-d]pyrimidine-4-thione N-[(4-methoxyphenyl)methyl]-1-phenylcyclohexan-1-amine 5-[(3R)-1-(2-fluoroethyl)piperidin-3-yl]oxy-4,6-dimethylpyrimidine N-[3-(2,4-difluorophenyl)pyrrolidin-1-yl]benzenesulfonamide 2-[5-amino-4-cyano-1-(2,6-dichlorophenyl)-3H-pyrazole-2-carbonyl]pyrrolidine-1-carboxamide 2-[7-(trifluoromethyl)-3H-benzimidazole-5-carbonyl]pentanoic acid 4-[2-(3,5-difluorophenyl)morpholine-4-carbonyl]benzaldehyde 2-(4,6-dichloropyrimidine-5-carbonyl)-3,4-dihydro-1H-isoquinoline-7-sulfonamide 1-cyclopentyl-3,4-difluoro-2-(trifluoromethoxy)benzene 2-N,4-N-bis(4-tert-butylphenyl)-1,3,5-triazine-2,4-diamine 4-(2,3-dichlorophenyl)sulfanyl-7H-pyrrolo[2,3-d]pyrimidine N-[3-(2,5-dihydroxypyrrol-1-yl)phenyl]acetamide 6-[6,7-dimethyl-8-(3-piperidin-1-ylpropoxy)-4H-chromeno[4,3-c]pyrazol-2-yl]-9-methylidenexanthene-1,2-disulfonic acid 4-[(2S)-1-methylpiperidin-2-yl]sulfonylbenzamide 2-[[5,6-di(propan-2-yl)pyridine-3-carbonyl]amino]-2-(1H-indol-4-yloxy)acetic acid 2-methyl-1,6-di(propan-2-yl)isoquinoline 2-[6,9-dihydroxy-2-(4-hydroxyphenyl)-5a,10-dihydrothieno[3,2-c]quinoline-8-carbonyl]benzaldehyde 2-[2,5-di(cyclobutyl)phenyl]pyridine 2-(3,4-difluorophenoxy)-N-[(Z)-(3-ethoxy-4-hydroxyphenyl)methylideneamino]acetamide N-[(4-chlorophenyl)methyl]-2-methoxyspiro[6,8-dihydropyrrolo[1,2-a]pyrazine-7,4'-piperidine]-5-carboxamide;hydrochloride 3-(2,5-dimethyl-1H-pyrrole-3-carbonyl)piperazine-1-carboxamide N-[4,5-difluoro-2-(1H-indol-3-yl)phenyl]-1-ethylcyclopropane-1-carboxamide 3-[6-(4,5-dimethylimidazol-1-yl)pyrimidin-4-yl]-N'-methanimidoyl-2-propan-2-ylideneimidazolidine-4-carboximidamide 6-chloro-3-(1,3-dimethylbenzimidazol-2-ylidene)-7-fluoro-4H-isoquinolin-1-one 4-(4-azido-2-fluorophenoxy)pyridine 3-[4-(2,6-diphenyl-1H-pyridazin-3-yl)phenyl]pyridine 1-[4-(2,5-difluorophenoxy)piperidin-1-yl]propan-2-ol 2,5-difluoro-N-[(2S)-1-hydroxypropan-2-yl]benzamide;2,6-difluoro-4-pyrrolidin-3-yloxypyridine N-[5-(3-aminopropanoyl)-4,6-dimethylpyrimidin-2-yl]-1-(3-pyridin-4-ylphenyl)cyclobutane-1-carboxamide [1-(2,6-dimethylpyrimidine-4-carbonyl)pyrrolidin-3-yl]-[(3S,5R)-3,5-dimethylpiperazin-1-yl]methanone 1-(2,4-dimethylthiophene-3-carbonyl)piperidine-4-carboxamide 2-(1H-imidazol-5-ylmethyl)-7,10-dihydrophenazine N-(2,4-dichloropyrimidin-5-yl)-N-[3-(trifluoromethyl)phenyl]methanesulfonamide 2-(N-tert-butyl-4-chloroanilino)acetamide 4-(3,5-difluorophenyl)imino-5-[(E)-1-(2,4-dihydroxyphenyl)ethylideneamino]-1,3-thiazolidin-2-one 5-(2,3-dihydrothiophen-4-yl)-N-[2-fluoro-6-methoxy-4-[4-[1-(methylcarbamoylamino)propan-2-yl]piperidin-1-yl]phenyl]-1-methylimidazole-2-carboxamide 5-bromo-6-chloro-N'-hydroxypyridine-2-carboximidamide 1-(4-phenylsulfanylphenyl)sulfonylpyrrolidine 1-(3,5-difluoropyridin-4-yl)-N'-methanimidoyl-2-methoxy-6-propan-2-ylindole-3-carboximidamide 2-(2,6-diphenylpyridin-4-yl)-8-[4-(trifluoromethyl)phenyl]pyrimido[1,2-a]benzimidazole (3,4-dichlorophenyl)-dimethyl-[2-(1H-indazol-6-ylamino)pyrimidin-5-yl]sulfanium [2-amino-4-oxo-6,8-di(propan-2-yl)pteridin-7-ylidene]methylideneazanium 1-(2,3-dimethylphenyl)-6-hydroxy-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]pyrimidine-2,4-dione 4-(azidomethyl)-3,5-dichlorobenzenesulfonamide 5-[4,6-bis(2-hydroxyphenyl)-1,3,5-triazin-2-yl]-2-propoxyphenol 4-(1,2-oxazol-3-yl)-3H-quinolin-2-one 4-N-(1-cyclopropylpiperidin-3-yl)-5-methoxypyrimidine-2,4-diamine 3-[3-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]propanoic acid N-(2,5-dichlorophenyl)-2,4,6-trimethyl-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]benzenesulfonamide (3E)-1-[3,5-dimethoxy-4-[4-(2-phenylethylamino)butanoyl]phenyl]penta-1,3-dien-3-ol 3-(2,6-dichlorophenyl)-7-[4-[methyl-(1R)-1-piperidin-4-ylethoxy]anilino]-2H-pyrimido[5,4-e][1,3]thiazin-4-one 2-[3-(4,4a-dihydrocarbazol-9-yl)phenyl]benzonitrile 4-[[5-methoxy-2-(2-phenylethenyl)pyridin-3-yl]amino]-1H-indole-7-carboxamide 2-(4,7-dimethylindol-1-id-3-yl)acetic acid;2-(dimethylamino)ethyl-(3,5-dimethylcyclohexa-2,4-dien-1-ylidene)azanium 1-ethyl-2,7-dimethoxypyrene (Z)-3-[4,5-dimethyl-2-(propylamino)phenyl]-2-fluoroprop-1-en-1-amine;ethane 5-(4,4,5,5-tetramethyloxaborolan-2-yl)furo[3,2-b]pyridine 6-[(4-aminophenyl)methyl]-2-N,7-N-dibenzyl-5H-pyrrolo[3,2-d]pyrimidine-2,7-diamine N-(2,5-difluorophenyl)sulfonyl-1-phenyl-6-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide N-[(2R)-3,3,3-trifluoro-1-(4-iodophenyl)propyl]benzamide (3S)-3-(4,6-dimethylpyrimidin-2-yl)oxypiperidine-1-carboxylic acid N-cyclopropyl-1,4-dimethyl-7-(5,6,7,8-tetrahydronaphthalene-2-carbonylamino)-3,6-dihydro-2H-pyridine-5-carboxamide (6R)-3-[2-[5,7-difluoro-1-methyl-6-(5-nitrothiophen-2-yl)benzimidazol-2-yl]-3H-benzimidazol-5-yl]-N,2,2-trimethyl-4-oxo-1,3,6,7,8,9-hexahydropyrido[1,2-a]pyrazine-6-carboxamide 4-[3,5-dimethyl-1-(2-phenylethyl)pyrazol-4-yl]-N,N-diethylaniline 1-[5-(4-chlorophenyl)-2,3-dihydrothiophen-4-yl]-3-[(3R)-4,6-dihydroxyoxan-3-yl]urea 3-[1-(2,6-difluorophenyl)ethyl]-4H-1,2,4-oxadiazol-5-one 2-[4-(4-ethylphenyl)-3,5-dimethoxyphenyl]propan-1-ol 2-[(4,6-dihydroxy-5-methylcyclohexa-1,3-dien-1-yl)-(4-ethoxyphenyl)methyl]-5-hydroxypyran-4-one 2-[1,3-benzodioxol-5-yl(3H-pyrrol-4-yl)methylidene]propanedinitrile 1-[5-[[4-(3,7a-dimethyl-1H-benzimidazol-2-ylidene)piperidine-1-carbonyl]amino]pyridin-3-yl]piperidine-4-carboxylic acid (3S)-3-(4-methoxyphenyl)-2,2-dimethylpentanal N-[2,4-bis(trifluoromethyl)phenyl]-3-ethoxy-6-[(E)-2-(1H-pyrazol-5-yl)ethenyl]pyridazin-4-amine N-(3,4-dimethylphenyl)-2-[2-[(4R)-4-methoxy-5-methylhexanoyl]phenoxy]propanamide 5-chloro-1-[(2,4-difluorophenyl)methyl]spiro[indole-3,7'-6H-furo[2,3-f][1,3]benzodioxole] 2-[3,5-dichloro-4-[4-(cyclobutylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenyl]-1-methyl-5-(trifluoromethyl)benzimidazole-4-carboxamide;hydrochloride 3-chloro-N-[(5R)-3-methyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b]azepin-5-yl]-5-phenylbenzamide 2-(2-ethylbenzimidazol-1-yl)-N'-hydroxypyridine-4-carboximidamide N-[3-(4-acetylpiperazine-1-carbonyl)phenyl]-2,5-dimethoxybenzenesulfinamide 3-[(2Z)-5-benzylidene-4-oxo-1,3-thiazolidin-2-yl]benzoic acid N-(2-hydroxyethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-sulfonamide 5-[1-(ethylideneamino)ethenyl]-N-methylpyridin-2-amine N-[1,6-dimethyl-2-(4-methylphenyl)-3-oxopyridazin-4-ylidene]-4-nitrobenzamide 5-azidooxy-6,7-difluoroquinoline 2-[4-(carbamoylsulfamoyl)-N-methylsulfonylanilino]octanoic acid 4-[(Z)-3-amino-1,1,1-trifluoropent-2-en-2-yl]-N-benzylaniline 2,3-diphenylpropanethioate 3-(2,2,6,6-tetramethylmorpholine-4-carbonyl)-1H-quinoxalin-2-one 2-[7-(3,5-difluorophenyl)-4-[2-methoxyethyl(methyl)amino]quinoline-3-carbonyl]cyclohexane-1,4-dione N-(1-tert-butylpiperidin-4-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide 7-cyclopropyl-2,3-dimethylpyrimido[1,2-b]pyridazin-4-one 2-[3-hydroxy-1-(2,4,6-trichlorobenzoyl)pyrrolidin-3-yl]-N-methylacetamide 3-chloro-5-[2-(4,5-dihydro-1H-imidazol-2-yl)ethyl]-7-(thiophen-2-ylmethylamino)pyrazolo[1,5-a]pyrimidine-6-carboxamide 2-(ethoxymethyl)-7,8-dihydro-6H-imidazo[1,5-a]pyrazine-5-carboxylic acid 2-cyclopentyl-4-(difluoromethoxy)benzaldehyde 4-chloro-2-fluoro-N-[2-(4-methoxyphenyl)ethyl]benzamide (Z)-4-[3,5-bis(trifluoromethyl)phenyl]imino-1-(2-hydroxyphenyl)but-2-en-1-one 4-[5-(2,3-dimethylmorpholin-4-yl)pyrazin-2-yl]benzoic acid 3-[4,5-dihydroxy-2-(oxan-2-ylmethyl)phenyl]propanoic acid 5-chloro-1,2,3-trifluoro-6-(2-methylsulfanylethoxy)-4-[4-(sulfinatoamino)cyclohexyl]benzene ethane;N-[3-(3,4,5-trifluorophenyl)butanoyl]propanamide 2-chloro-3-[6,6-dimethyl-1-(2-morpholin-4-ylethyl)azepan-5-ium-1-yl]phenol N-[(4-fluorophenyl)methyl]-3-hydroxypyridine-2-carboxamide (3Z)-3-[(5Z,8E,11Z,14E)-icosa-5,8,11,14,17-pentaenylidene]-6H-benzimidazolo[2,1-a]isoquinolin-7-ium 7-[(4-azidooxyphenyl)methyl]naphthalene-2-carbonitrile N-[(Z)-1H-indol-3-ylmethylideneamino]-2-pyrrolidin-1-ylacetamide N-azido-1-(4,5,6,7-tetrahydroindazole-3-carbonyl)pyrrolidine-2-carboxamide (3S)-5,7-difluoro-N-[[2-fluoro-4-[6-(trifluoromethyl)pyridin-3-yl]phenyl]methoxyiminomethyl]-1-(oxetan-3-yl)-2,3,4,9-tetrahydro-1H-carbazole-3-carboxamide 5-[(Z)-1-amino-3-methyliminoprop-1-en-2-yl]-7-(1,4-dioxan-2-ylmethoxy)-3H-quinazolin-4-one [4-amino-1-(2-phenylethyl)cyclohexyl]azanium (3,4-dimethylphenyl)-[[(2S)-6-fluoro-1H-indol-2-yl]methylamino]methanol 3-(dimethylamino)-5,6-bis[2-hydroxyethyl(sulfino)amino]-1H-indazole (5R)-1,4-bis[3,5-dimethoxy-N-methyl-2-(trifluoromethyl)anilino]-5,6-dihydrocyclopenta[c]pyrazole-3-carboxylic acid N-(2,6-dioxopiperidin-3-yl)-5-[4-fluoro-3-(trifluoromethoxy)phenyl]-1-(2,2,2-trifluoroethyl)pyrazole-3-carboxamide 5-[6-[3-(3,4-dichlorophenyl)propylamino]pyrimidin-4-yl]pyridine-2-carbonitrile;ethane N-[2-(dimethylamino)ethyl]-3-[7-methoxy-4-[[5-(trifluoromethyl)pyridin-2-yl]amino]quinazolin-6-yl]-1,2,4-oxadiazole-5-carboxamide 1,2-dimethyl-6-[[4-(prop-2-enoxymethyl)phenyl]methyl]-5,7-dihydropyrrolo[3,4-d]pyrimidine 4-[1,2-dideuterio-2-(1H-pyridin-2-yl)ethenyl]-N-phenylaniline (Z,6E)-3-[5-amino-1-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]pyrazol-3-yl]oct-4-enoic acid 1-(azidomethyl)-5,7-dichloroquinolin-2-one 3-[4-(1,3-dioxoisoindol-2-yl)butyl]-1H-benzo[f]indole-7-carboximidate 2-(1H-indol-3-yl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine [(3R)-3-[4-[(2S,5S)-6,15-dichloro-16-methyl-4,8-diazatricyclo[7.5.0.02,7]tetradeca-1(9),10,12-trien-4-yl]butoxycarbonylamino]piperidin-1-yl]-oxidoazanium N-(2,3-difluorophenyl)sulfanyl-7,8-bis[(4-methoxyphenyl)methyl]-6-methyl-5,6,9,10-tetrahydropyrimido[4,5-b]quinolin-2-amine;formaldehyde 3-[4-(1H-benzimidazole-2-carbonyl)piperazin-1-yl]oxolane-3-carboxylic acid 6-chloro-3-(trifluoromethyl)imidazo[1,2-a]pyridine 5-chloro-4-[(3S)-1,2,3,6-tetrahydrofuro[3,2-d]imidazol-3-ium-3-yl]benzene-1,2-diol 4-methyl-2,3-diphenylbutanal 4-(3-chloro-2-fluoroanilino)-7-methoxyquinoline-6-carbonitrile 4-[6,7-dimethoxy-2-(methylamino)quinazolin-4-yl]piperazine-1-carboxylic acid 2-(4-bromophenyl)imino-5-[(3-methoxy-1,6-naphthyridin-8-yl)methylidene]-1,3-thiazolidin-4-one 2-methyl-4-[1,3]thiazolo[5,4-f][1,3]benzoxazol-6-amine 4-[6-(methylamino)hexanoyl]benzoic acid 2-[1-[5-[(6,7-dimethoxy-1,3-benzothiazol-2-yl)amino]pyridine-2-carbonyl]piperidin-4-ylidene]acetic acid 3-(5-methylindol-1-yl)cyclohexa-2,4-diene-1-carboxamide 2-[3,5-dichloro-4-(6-oxo-1H-pyridine-2-carbonyl)phenyl]sulfanylacetic acid 4-(2,2-difluoro-1,3-benzodioxol-5-yl)-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 1-(2,3-difluorophenyl)ethanone;4-[[5-[2-(4-hydroxy-2-oxopyrrolidin-1-yl)pyridin-4-yl]-1H-pyrrolo[2,3-b]pyridin-3-yl]methylideneamino]benzenecarboximidamide 2-(2,4-dichlorophenyl)-5-methylsulfonylbenzenesulfonic acid N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-2-[3-(4-propylphenoxy)propoxy]acetamide 4-[4-(3,5-dimethylcyclohexyl)phenoxy]phenol 2-(3,5-dichlorophenoxy)-N'-hydroxypyrimidine-4-carboximidamide 1-N,3-N-bis(4-cyanophenyl)benzene-1,3-dicarboxamide 2,6-ditert-butyl-3-(2-ethoxy-6-phenyldiazenylpyrimidin-4-yl)phenol (3R)-4-methyl-3-[4-methyl-2,5-dioxo-1-(4-phenylphenyl)imidazolidin-4-yl]sulfanylbutanenitrile ethane;N-(2-phenylsulfanylphenyl)pyridine-3-carboxamide 6-(2,3-difluorophenyl)-4-[6-methoxy-5-[2-(oxan-2-yl)pyrazol-3-yl]pyridin-3-yl]oxypyrido[3,2-d]pyrimidine (4S)-2,3,9-trimethyl-4-(2,4,6-trimethoxyphenyl)non-1-en-4-ol 3-[4-(9H-fluoren-1-yl)phenyl]propanoate N-[2-[5-(6-methoxyquinolin-4-yl)oxypyridin-3-yl]-1,3-benzoxazol-5-yl]-4-methylidenepiperidine-1-carboxamide (7S)-7-(6-bromo-2,4-dioxoquinazolin-3-yl)-1-[1-(trifluoromethylsulfonyl)piperidin-4-yl]oxydecane-3,5-dione 3-chloro-N,2-dimethyl-4-[1-(3-pyridin-2-ylphenyl)ethylamino]sulfanylaniline 2-[(3,5-dimethylphenyl)iminomethyl]-6-ethoxyphenol 5-ethyl-2-(3,4,5-trifluorophenyl)pyrimidine 2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyridine 1-(7H-purin-6-yl)indazole [(3S,4R)-1-azido-2-oxopiperidin-3-yl]-(1H-imidazol-2-ylmethyl)carbamic acid N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-fluoro-3-morpholin-4-ylsulfonylbenzamide 2-(4-nitrophenyl)-1,3-dioxo-N-[2-[(E)-pent-3-enyl]cyclopropyl]isoindole-5-carboxamide 1-[4-(4-amino-3,5-dimethylphenoxy)pyridin-2-yl]ethanol 4-azidooxysulfonylbenzoic acid 4-[2,6-bis(prop-1-en-2-yl)phenyl]-3H-1,3-oxazole-2,2-diamine 2-amino-6-methylsulfanyl-4-(2,3,5-trifluorophenyl)pyridine-3,5-dicarbonitrile 4-azido-1H-quinazoline-2,4-dione N-[(1S,3S)-3-(4-methoxyphenoxy)cyclohexyl]pyrimidine-5-carboxamide 1-benzyl-2,3,4,5-tetrabutylpiperazine 6-[(E)-1-(5-azidothiophen-2-yl)prop-1-en-2-yl]-3,4-dihydro-2H-chromene N-[4-(2,6-dimethoxyphenyl)-5-(6-methylpyridin-3-yl)-1,2,4-triazol-3-yl]-4,5,7,8-tetrahydro-1H-pyrazolo[3,4-d]azepine-6-carboxamide (4S)-5-[2-(2,3-dihydro-1H-inden-2-yloxy)acetyl]-11-hydroxy-4-methyl-3,4-dihydro-1H-pyrido[1,2-b]phthalazine-8-carboxylic acid 3-(3,5-dimethylbenzene-6-id-1-yl)benzonitrile;propan-2-one;uranium(2+) (E)-3-[5-bromo-2-hydroxy-4-methoxy-6-(trifluoromethyl)phenyl]-1-(4,5-dimethyl-1H-pyrrol-2-yl)prop-2-en-1-one [7-(1H-indazol-4-yl)indolizin-3-yl]methanol 5-methoxycarbonyl-2,6-dimethyl-4-[3-(trifluoromethyl)phenyl]-1,4-dihydropyridine-3-carboxylic acid 6-(cyclohexen-1-yl)-3-[5-hydroxy-4,4-dimethylpentyl(methyl)amino]pyrazine-2-carboxylic acid (4E)-N-[(3-chlorophenyl)methyl]-5,6-dihydro-2H-1,5-benzothiazocine-8-carboxamide 4-[5-(2-methylpropoxy)pyridin-3-yl]cyclohexa-1,3-diene-1-sulfonamide 2,4-ditert-butyl-6-[(3,5-dimethyl-4-propan-2-yloxyphenyl)iminomethyl]phenol N-[3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methanesulfonamide N-(4-methoxyphenyl)sulfanyl-2,5-dimethylaniline 3-(4-chlorophenyl)-N-[[2,4-difluoro-6-(1H-pyrazol-5-yl)phenyl]methylideneamino]propanamide 2-[4-[(6-chloronaphthalen-2-yl)methoxy]phenyl]-N-[(1R)-5-cyano-6-fluorocyclohexa-2,4-dien-1-yl]sulfonylacetamide 1-azidooxy-2,3,4,5,6,7-hexamethylnaphthalene 2-[3-(aziridine-1-carbonyl)anilino]-9-[2-(dimethylamino)ethoxy]-6,7-dihydrobenzo[d][1]benzoxepin-5-one (2R)-2-azido-3-cyclobutyl-1,2-diphenylpropan-1-one N-[5-(2,3-dimethylimidazol-4-yl)-1H-pyrazol-3-yl]-2-[6-(hydroxymethyl)-7,8-dihydronaphthalen-2-yl]acetamide (2S)-2,6,8-trimethyl-3,4-dihydro-2H-naphthalen-1-one (3S)-4-benzyl-1,2,3-trimethylpiperidine 4-chloro-3-[[3-(4-ethoxyphenyl)-1H-indazol-6-yl]methylideneamino]-N,N-dipropylbenzenesulfonamide N-[3-cyano-4-(furan-2-yl)thiophen-2-yl]benzenesulfonamide 2-[2,6-difluoro-4-(3-methyl-1H-pyrazolo[3,4-b]pyridin-5-yl)phenoxy]-N-(oxan-4-yl)acetamide (1R)-2-ethyl-7-(trifluoromethoxy)-3,4-dihydro-1H-isoquinoline 2-(4,6-dimethylpyrimidin-5-yl)oxy-3-[(E)-1-[(2S)-4-[4-(trifluoromethyl)phenyl]pyrrolidin-2-yl]prop-1-en-2-yl]pyridine (3-fluoro-5-methoxyphenyl)iodanium;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide [(2R)-1-hydroxy-3-methylbutan-2-yl]-triphenylphosphanium 2,4-dichloro-5-[4,6-bis(trifluoromethyl)pyrimidin-2-yl]sulfanylaniline 4-[2-[4,5-bis(ethenyl)-1H-imidazol-2-yl]-5-chloropyridin-3-yl]-N-(2-methoxy-6-propan-2-ylphenyl)-1,3,5-triazin-2-amine 5-(4,8-dimethylnonan-3-yl)-2-(6-ethoxypyridin-3-yl)-1H-benzimidazole [1-(7-propylnaphthalen-2-yl)propylideneamino]urea (1-azido-2,3,4,5-tetrabromo-9H-fluoren-4-yl)carbamic acid 2-[(2R)-1-phenylpyrrolidin-2-yl]-2-[3-(trifluoromethyl)phenyl]ethanimidamide N-(2,3-dihydro-1H-inden-5-yl)-2-ethoxy-2-oxoacetamide;ethane (5R)-2,9-dimethyl-3,4,4a,5,6,10b-hexahydro-1H-pyrido[4,3-g]isoquinoline 4-(methylamino)-N-[3-[5-[5-[[1-(trifluoromethyl)cyclopropyl]methoxy]pyridin-2-yl]-1,3,4-oxadiazol-2-yl]phenyl]benzenesulfonamide 4-fluoro-3-[3-(2-pyrrolidin-1-ylethoxy)phenyl]pentan-3-amine (Z)-3,4-bis[2-(methylamino)phenyl]hept-3-en-2-one N-[2,4-dichloro-3-(6-fluoroquinolin-4-yl)sulfanylphenyl]-1,5-naphthyridine-3-carboxamide 2-(4-butylphenyl)sulfanyl-N-[1-(4-fluoro-3,5-dimethoxyphenyl)ethyl]acetamide 2-[3,5-bis(trifluoromethyl)phenyl]-N'-hydrazinylidene-5-oxo-1H-pyrazole-4-carboximidamide 4-[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-N-propan-2-ylthiophene-2-sulfonamide N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-[(6R)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]acetamide 5-bromo-3,4-diphenyl-2H-thieno[3,4-c]pyrazole 3-[1,1-bis(ethenyl)-4-methyl-2H-inden-5-ylidene]-4H-naphthalene-1,2-dione N-cyclohexyl-2-[1,3-dioxo-4-(pyridin-3-ylmethoxy)isoindol-2-yl]acetamide 2-[5-[4-(3,4-difluoro-1H-indole-2-carbonyl)piperazine-1-carbonyl]pyridin-3-yl]-N'-hydroxypyrimidine-5-carboximidamide 4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-N,3,7-trimethyl-2,3,4a,5,6,7,8,8a-octahydroquinoxaline-1-carboxamide 3-[[2-(5-chloropyrimidin-4-yl)oxy-6,7-dihydronaphthalen-1-yl]amino]benzoic acid 2,6-dichloro-N-[4-chloro-3-(2-methylsulfanylbenzoyl)phenyl]benzamide 5-[3,4-bis(methoxycarbonyl)naphthalene-1-carbonyl]oxy-2,3,4-trichlorobenzoic acid 2-methyl-N-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3-bis[(Z)-prop-1-enyl]phenyl]propanamide 1-(3,5-dimethoxyphenyl)-2-[(4-ethyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]propanoic acid (2S)-2-[[(2R,3aR)-4-phenyl-1,2,3,3a,4,5,6,7,7a-octahydroisoindole-2-carbonyl]amino]-8-oxooctanoic acid 3-[3-(2-phenylpropan-2-yl)phenyl]cyclohexane-1,2-dione 3-methyl-N-[(2S)-4-oxo-4-[2-(1H-pyrrolo[2,3-b]pyridin-6-ylsulfonylamino)ethoxy]butan-2-yl]butanamide 2-N,4-N-dimethylquinazoline-2,4-diamine;3-(5-ethynylpyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-imine 1-[5,5-bis(4-fluorophenyl)pyrazolidin-3-yl]pyrazole;chloromethane 5-[1-(2-methylpropylamino)ethenyl]pyrimidine-4,6-diamine 2,5-diphenyl-1H-imidazole;ethane 2-fluoro-3,4,5-triphenyl-1H-pyrrole (6S)-5,6-bis(4-chlorophenyl)-1,3-dihydroxy-2-[(2S)-2-methylpiperidine-1-carbonyl]cyclohexa-2,4-diene-1-carboxylic acid 6-chloro-N-(4-methoxyphenyl)-3,5-dimethylcyclohexa-1,5-dien-1-amine 1-[3-[5-(4-chlorophenyl)-4-methyl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-2-yl]piperidin-1-yl]-2-pyrazol-1-ylethanone 3-(8-fluoroquinolin-6-yl)-2-phenyl-5H-pyrido[4,3-b]indole (E)-1-[6-(2,4-dimethoxyphenyl)-3-methyl-[1]benzothiolo[3,2-b]pyrrol-8-yl]pent-2-en-1-one 2-[1-[[(4S)-4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)cyclohexen-1-yl]methoxy]propan-2-ylideneamino]oxyacetonitrile 2-(4-chlorophenoxy)-N-[2-(methylsulfonylamino)phenyl]acetamide 2-(3,6-dihydro-2H-pyran-4-yl)-1'-ethylspiro[6,7-dihydropyrrolo[2,1-c][1,2,4]triazole-8,4'-piperidine] 4-(2,6-difluoro-3,5-dimethoxyphenyl)-6-[2-hydroxyethyl(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile 2-[1-hydroxy-3-methylsulfanyl-4,6-bis(trifluoromethyl)naphthalen-2-yl]-1-methoxybutan-1-ol 4-[(2R,3S)-1-azido-5-(3,5-dichloropyridin-4-yl)-4-oxopentan-3-yl]piperazine-1-carboxylic acid 2-(1H-imidazol-5-yl)-N-[2-(methoxymethyl)phenyl]thieno[3,2-d]pyrimidin-4-amine 3-[1-[(Z)-5-aminopent-2-enyl]azepane-4-carbonyl]benzaldehyde (3S,4R)-N-[(4-methylphenyl)methyl]-1-propanoylpiperidine-3-carboxamide 3-[2-(4-bromophenyl)ethyl]benzamide 7-[2-(hydroxymethyl)pyrrolidine-1-carbonyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylic acid;2,2,2-trifluoroacetic acid N-azido-2-[5-(benzenesulfonyl)pentyl]isoindol-4-amine 5-tert-butyl-N,4-dimethyl-1H-imidazole-2-carboxamide 2,3-dimethyl-1-[(3-phenylpyrrolidin-1-yl)methyl]pyrrole;oxalic acid 4-N,6-dimethyl-2-[5-methyl-1-(4-phenylpyridin-3-yl)pyrrolidin-3-yl]pyrimidine-4,5-diamine 2-ethyl-1-[4-(3-methoxyphenyl)piperazin-1-yl]pentan-1-one 4-[N-(2,3-dihydroxypropyl)-2,5-dimethylanilino]benzenesulfonic acid 4-(azidomethyl)-N'-(2,3-dihydro-1H-inden-1-yl)benzenecarboximidamide (5R)-3-(azidomethyl)-2,8-diethoxybicyclo[4.2.0]octa-1(6),7-diene N-[[2-(2,4-dichlorophenyl)phenyl]methyl]acetamide 5-chloro-2-fluoro-4-[1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-3-yl]benzoic acid 1-[5-chloro-4-(3,5-difluorophenyl)sulfanyl-6-methoxypyridin-2-yl]ethanone 6-(3,4-dihydropyridin-5-yl)-2H-[1]benzofuro[3,2-b]pyridine [5-(4,4-difluorocyclohexyl)-2-methoxy-3-propan-2-ylphenyl]azanide N-(4-hydroxycyclohexyl)-6-[(3R)-1-(oxolane-2-carbonyl)piperidin-3-yl]oxypyridine-2-carboxamide 3-(2-bromophenyl)-4,6-dichloro-2H-1,3,5-oxatriazine N-[4-chloro-3-(trifluoromethyl)phenyl]-2,3-dihydroxypropanamide 3-(1-azidooxy-4-pyridin-3-ylbutan-2-yl)pyridine 2-(5-ethylfuran-2-yl)-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidine (2S,3aS,7aR)-N-cyclopropyl-6-[(5-methylfuran-2-yl)methyl]-3,3a,4,5,7,7a-hexahydro-2H-furo[2,3-c]pyridine-2-carboxamide;2,2,2-trifluoroacetic acid N-(5,6,7,8-tetrahydroquinazolin-4-yl)imidazo[1,2-a]pyridine-3-carboxamide 2-(2,3-dimethylphenyl)-1H-indole N-[4-(1H-benzimidazol-2-yl)butanoyl]-N-ethyloxolane-3-carboxamide 3-[[2-(4-methylsulfanylphenyl)acetyl]amino]cyclobutane-1-carboxylic acid 1-(1H-indole-2-carbonyl)pyrrolidine-3-carbonitrile 4-[[2,6-difluoro-4-(5-methylsulfanylpyrimidin-1-ium-2-yl)phenyl]carbamoyl]cyclohexane-1-carboxylic acid 2-[4-(1,3-dioxolan-2-ylmethoxy)-2-fluorophenyl]acetaldehyde 7-(2,4-dichlorophenyl)sulfonyl-9-methylsulfinyl-5,6,8,10-tetrahydro-3H-pyrimido[4,5-b]quinoline-4,6-dione 5-[1-(4-tert-butylanilino)ethenyl]-N,6,11-trimethylindolo[3,2-b]carbazole-10-carboxamide 5-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]-2-cyanobenzenesulfonic acid 5-(4-hydroxyphenyl)-3,7-dihydropyrrolo[2,3-d]pyrimidine-4,6-dione 2-[1-carboxypropan-2-yl(phenacyl)amino]octanoic acid N-(diaminomethylidene)-2-[3,5-bis(trifluoromethyl)phenyl]acetamide 3,4-dichloro-N-(2,6-difluorophenyl)benzenesulfonamide (2R)-4,6-dichloro-2-phenyl-2-(trifluoromethyl)morpholine 4-azido-5-(2,6-difluorophenyl)-3H-1,2,4-oxadiazole 2-(6,7,8,9-tetrahydrodibenzofuran-2-yl)-4H-cyclohepta[b]thiophene 2-[3-[[4,5-bis(ethenyl)imidazol-1-yl]methoxy]phenyl]-N'-pyridin-4-yl-3H-benzimidazole-5-carboximidamide 5-[4-bromobutan-2-yl(ethenylsulfonyl)amino]naphthalene-2-sulfonic acid 2-(7,8-dimethoxyquinolin-3-yl)-5-iodo-1H-indole-6-carbonitrile 3-N-[2-chloro-5-(trifluoromethyl)phenyl]-1H-1,2,4-triazole-3,5-diamine 2-[1,3-dimethyl-5-(methylideneamino)-6H-pyrazolo[4,3-d]pyrimidin-7-yl]phenol 5-chloro-2-(cyclopropylamino)benzamide 1-[(3R,4S)-1-benzyl-2-hydroxypiperidin-4-yl]-6-methylsulfonylbenzimidazole [(3-chlorophenyl)methyl-(2-ethoxypyrimidin-5-yl)amino]-oxidocarbamic acid 4-(4-ethoxycyclohexa-2,4-dien-1-yl)aniline N-[1-(2,5-dichlorophenyl)ethyl]-4-[1-[[3-methoxy-5-(trifluoromethyl)phenyl]carbamoylamino]ethenyl]benzamide;ethane 2-chloro-N-[5-(1,4-dimethylpiperidin-4-yl)oxypyrazin-2-yl]benzamide 2-[1-(6,7,8a,9-tetrahydro-5H-pyrrolo[1,2-a]azepin-3-yl)benzimidazol-2-yl]phenol 2-[(4,5-dichloro-3-fluorothiophene-2-carbonyl)amino]-1,1a,6,7,9,10b-hexahydrocyclopropa[a]naphthalene-1-carboxylic acid 3-benzyl-1-[(4-methoxyphenyl)methyl]-2H-pyridine N-(2,4,6-trimethylphenyl)butanamide 2-[4-[2,6-di(propan-2-yl)phenoxy]piperidine-1-carbonyl]butanedioic acid 3-fluoro-2,4,6-trihydroxybenzenesulfonate (6S)-7,8-dimethyl-9-[4-(1H-pyrazol-5-yloxy)phenyl]-2-thiophen-3-yl-5,6-dihydropurine (4-amino-2,5-difluorophenyl)-(methylamino)azanium 1-[2-(4-methylphenyl)pyrimidin-5-yl]ethenol 1-N,1-N',4-N,4-N,2,5-pentamethylcyclopentane-1,4-diamine;nickel(2+);nickel(3+);tetrabromide 4-[(1S)-3-[(2,5-dioxopyrrolidin-1-yl)methoxycarbonylamino]cyclohexyl]benzoic acid 3-[(1R)-1-(6,7-dimethoxy-4-oxochromen-2-yl)ethyl]-5-methoxycarbonyltriazole-4-carboxylate 3-azido-2-(difluoromethyl)acridine (3R,4S)-1-ethyl-N'-[(6-methoxypyridin-2-yl)methyl]-5-oxo-3-phenylpyrrolidine-3-carbohydrazide 5-azido-3-chloro-6,8-difluoro-2-methylquinoline N-[(1S)-2,3-dihydro-1H-inden-1-yl]-N',N'-dimethyl-4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidine-2-carbohydrazide 2-N,7a-dimethyl-1H-oxireno[2,3-c]isochromene (2R,6R)-1-[[3,5-bis(trifluoromethyl)phenyl]methylsulfonylmethyl]-4-(4-bromophenyl)sulfonyl-6-ethylpiperidine-2-carboxylic acid 2-(methylsulfonylmethyl)benzenesulfonic acid 4-(4,7-dichloro-6-phenylpteridin-2-yl)benzonitrile 6-(3,4-dihydro-2H-chromen-7-yl)-5-(4-phenoxyphenyl)-1,2,4-triazine-3,8-diamine N'-(cyclopropylmethoxy)-4,6-dimethylpyridine-2-carboximidamide ethane;5-methoxy-3,4-dihydro-1H-naphthalene-2,6-disulfonic acid 7-benzyl-8-methoxy-N,N,3,5-tetraphenyl-2,4-dihydropyrazolo[1,5-a][1,3]benzodiazepine-6-carboxamide 2-(N-butyl-3,5-dichloroanilino)propanoic acid 4-[5,7-diamino-2-(6-ethenylpyrimidin-4-yl)furo[3,2-b]pyridin-3-yl]-N-(1-methoxypropan-2-yl)benzamide 3-ethenyl-5-methoxycarbonylthiophene-2-carboxylic acid 4-hydroxy-2,6-dimethyl-N-(oxan-3-yl)benzenesulfonamide 3-chloro-N-[1-(4-fluorophenyl)ethyl]-6,8,11-trimethyl-5,6-dihydroindolo[2,3-b]quinoline-2-carboxamide;propane 1-[2,4-dimethyl-5-(pyrrolidine-1-carbonyl)thiophen-3-yl]ethanone 2-[4-fluoro-6-(4-fluorophenyl)-7,8-dihydroimidazo[1,5-a]pyrimidin-3-yl]ethanamine N-methyl-1,2-diphenyl-4a,5,6,7,8,9,10,11,12,12a-decahydropyrazolo[3,4-a]acridine-8-carboxamide 1-[2-methoxy-5-(trifluoromethyl)phenyl]pentane-1,4-dione N-(3-aminophenyl)-4,5-difluoropyrimidine-2-carboxamide 2-(4-chlorophenyl)-N-(2,2-dimethoxyethyl)butanamide 2-[4-(2-bromophenyl)piperazin-1-yl]ethanamine;hydrochloride (E)-3-[4-[(Z,2R,5S)-6,6-dimethylnon-5-enoxy]phenyl]-N-propan-2-ylbut-1-ene-1,3-diamine;ethane N-[2-[[2-(4-chlorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl]amino]ethyl]pyridine-4-carboxamide;2,2,2-trifluoroacetic acid N-(2,3-dihydro-1H-inden-2-yl)-5-(methoxymethyl)-4-phenylpyrrolidine-3-carboxamide N-[2,6-bis(trifluoromethyl)phenyl]propanamide;1-(8H-carbazol-4-ylsulfanyloxy)piperidine 3-[(2R)-5-hydroxy-2,6-dimethyloxan-4-yl]oxybenzonitrile 1,2-diamino-4-[3-bromo-5-methoxy-4-[(3-nitrophenyl)methoxy]phenyl]-6-oxopyridine-3,5-dicarbonitrile 5-amino-3-[4-(4-cyanophenyl)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile 2-(3,5-difluorophenyl)-1-hydroxy-6,6a,7,8,10,10a-hexahydrobenzo[b]quinolizine 2-(3,5-dichlorophenyl)-N-[[(4S)-3-[3-fluoro-4-[1-[2-(oxan-4-yloxymethyl)phenyl]ethylamino]phenyl]-2-oxo-1,3-oxazolidin-4-yl]methyl]acetamide 3-[3,5-difluoro-N'-(7H-purin-2-yl)anilino]benzonitrile 5-methoxy-2-methylsulfanylquinoline (E)-N',N'-dimethyl-1-[4-[3-[2-(methylideneamino)phenyl]propoxy]cyclohexa-2,5-dien-1-yl]-1-phenylethene-1,2-diamine;heptane 2-[(1R,5S)-3-benzylsulfonyl-3-azabicyclo[4.1.0]heptan-6-yl]pyrimidine 5-(4,5,6,7-tetrahydro-1H-benzimidazol-2-ylmethylidene)-4H-thieno[3,2-c]pyridine (E)-4-[3-bromo-6,7-difluoro-1-(2-hydroxypropan-2-yl)indol-5-yl]-N'-methanimidoyl-3-methoxybut-3-enimidamide 1,3-difluoro-5-phenylcyclohexa-2,4-diene-1-sulfonic acid 1-(4-aminophenyl)sulfanyl-N',3-dimethylpyrazole-4-carboximidamide 4-(3,3-dimethylpentan-2-ylamino)-1H-pyrimidin-6-one (2S,4R)-2-tert-butyl-1-[3-(trifluoromethoxy)phenyl]sulfonylpiperidine-4-carboxylic acid 4-azidooxy-3,6-dichlorophthalic acid 5-[4,6-bis(9H-fluoren-1-yl)pyrimidin-2-yl]pyrimidine (Z)-3-[4-chloro-1-methyl-5-(2,4,6-trifluorophenyl)pyrazol-3-yl]prop-2-enoic acid (3S)-1-[1-amino-4,6-difluoro-8-methoxy-7-(2-morpholin-4-ylethoxy)-3H-isoquinoline-1-carbonyl]piperidine-3-carboxylic acid [3-(2,6-diphenyl-1H-1,3,5-triazin-4-yl)cyclohexa-2,4-dien-1-ylidene]methanamine N-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-4,6-dimethylcyclohexa-1,3-diene-1-sulfonamide 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethanol 1-[2,4-bis(methylsulfanyl)phenyl]imidazolidine [5-(3,3,3-trifluoropropyl)pyridin-2-yl]hydrazine 3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-ethylsulfanyl-6-thiophen-2-ylpyrimidin-4-one 2-(4-bromophenyl)-1H-indole N-azido-2,3,4-tris(hydroxymethyl)benzenesulfonamide [5-[(3,4-difluorophenyl)methyl]-2-phenylmethoxyphenyl]boronic acid 4-(7,8-difluoroquinolin-3-yl)-N-(2,6-dimethoxypyridin-3-yl)piperazine-1-carboxamide;ethane N-(2,3-dihydroimidazo[1,2-a]benzimidazol-5-ylmethyl)-6-hydroxy-N-phenylcyclohexa-2,4-diene-1-carboxamide 2-[4-[3-(methoxymethyl)-5-methylphenyl]quinolin-6-yl]propan-2-amine 6-[2,3-difluoro-4-(trifluoromethoxy)phenyl]-5-fluoropyridin-2-amine 4-[4,4,4-trifluoro-1-methoxy-3-(2,4,5-trichlorophenyl)butyl]benzenesulfonic acid 2-[5,7-dimethyl-6-(4-pyridin-3-yloxyphenyl)pyrrolo[3,2-d]pyrimidin-4-yl]oxy-N-propan-2-ylbenzamide 2-(2,2-dimethylpropoxy)-N'-hydroxypyrimidine-4-carboximidamide 2-[4-(hydroxymethyl)phenyl]benzene-1,3-dicarboxylic acid N-(2,3-dihydropyridin-4-yl)-N'-phenylmethanediamine 7,8-difluoroquinoline;1-(methylamino)cyclopropane-1-carboxylic acid 3-[1,3-bis(1H-indol-2-yl)propan-2-ylideneamino]propanenitrile [4-(azidomethyl)-3,5-dimethoxyphenyl]methanamine 4-(2,3,5-tribromophenyl)oxane (4R)-3-[2-chloro-6-hydroxy-5-(1H-pyrrol-2-yl)pyrimidin-4-yl]-4-propan-2-yl-1,3-oxazolidin-2-one 1-[3,5-difluoro-2-(hydroxymethyl)phenyl]-3-(2-methoxyethylamino)urea N-[1-(3,5-dimethoxyanilino)-2H-pyrimidin-4-yl]piperidine-3-carboxamide (E)-1-[2-tert-butyl-3-(5,6-dimethoxypyridine-3-carbonyl)indolizin-7-yl]-3-hydroxyprop-2-en-1-one (4-aminopiperidin-1-yl)-[3-[[6-fluoro-8-(methoxymethyl)imidazo[1,2-a]pyridin-2-yl]carbamoyl]phenyl]carbamic acid 1-[5-chloro-2-(trifluoromethyl)phenyl]sulfonyl-4-[[3,4-dichloro-6-[5-(1H-pyrazol-5-yl)pyridin-2-yl]oxypyridin-2-yl]methyl]piperazine 4-[5-chloro-2-hydroxy-3-(1H-pyrrolo[2,3-b]pyridin-2-yl)indol-1-yl]-N-(oxolan-2-ylmethyl)benzamide 2-[4-(cyclohexylcarbamoyl)anilino]propanoic acid 2-[(1S)-4,5-dimethoxy-3-oxo-7-propanoyl-1H-isoindol-2-yl]-N-[(2R)-2-hydroxypropyl]acetamide 1-[2-(cyclopropylmethylamino)pyridin-4-yl]-3-[3-fluoro-4-[5-(trifluoromethyl)pyridin-3-yl]phenyl]urea 1-azido-4-(4,5-diphenylpentyl)benzene (E)-3-[4-fluoro-2-methoxy-6-[5-(1,3-thiazol-4-yl)-1H-imidazol-2-yl]phenyl]prop-2-enamide [3-amino-1-(2-methylpropanoyl)cyclobutyl]-pyridin-4-ylmethanone 2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propanal 4-[(3R)-1-[(2E,6E)-7-ethyl-9-methylideneundeca-2,6-dienoyl]piperidin-3-yl]oxybenzonitrile 4-[1-hydroxy-3-(2H-triazolo[4,5-b]pyridin-6-yl)piperidine-3-carbonyl]morpholin-3-one 5-(trifluoromethyl)-3H-furo[2,3-c]pyridine N-(3,4-dichlorophenyl)sulfanyl-2,5-dimethoxyaniline 1-(2,4-difluorophenyl)sulfonyl-4-[[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)naphthalen-2-yl]methoxy]piperidine N'-(4-azidophenyl)piperidine-1-carboximidamide 4-[(5-methoxy-2-propylsulfonylpyrimidin-4-yl)amino]cyclohexan-1-ol 3-[(1R)-2,3-dimethylcyclohexyl]-N-ethylaniline 6-(azidomethoxy)naphthalene-2,3-dithiol (E)-4-[4-[2,3-difluoro-4-methyl-5-[3-methylbutyl(methyl)amino]phenyl]anilino]-N'-[(2-hydroxy-1H-indol-3-yl)imino]but-2-enimidamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-7-pentylphenanthrene 3-hydroxy-4-[1-(2,2,6,6-tetramethylpiperidin-4-yl)imidazol-2-yl]-9H-carbazole (2-hydroxypyridin-4-yl)-[5-methoxy-1-[3-[[3-propan-2-yl-5-(trifluoromethyl)phenyl]sulfamoyl]benzoyl]piperidin-2-yl]iodanium 4-amino-6-(3-chloro-5-fluoro-2,4-dihydroxyphenyl)-1H-1,3,5-triazin-2-one 4-ethyl-5-(6-fluoroquinolin-4-yl)-3,8-dihydropyrimido[4,5-d]pyrimidine-2,7-dione (5E)-2-(2-hydroxyphenyl)imino-3-[(1R,2S)-2-[4-[(E)-2-pyridin-3-ylethenyl]phenoxy]cyclohexyl]-5-[(4Z)-2,3,5-trimethoxyhepta-2,4-dienylidene]-1,3-thiazolidin-4-one N-[(2S)-3-(5,6-dihydro-4H-cyclopenta[d][1,3]thiazol-2-yl)-1-[3-oxo-4-[[4-[[5-(trifluoromethyl)pyrimidin-2-yl]amino]cyclohexyl]oxymethyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]formamide;fluorobenzene 5-(4-fluorobenzoyl)-N-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 4-[4-(2-hydroxyethyl)-3,5-dimethoxyphenyl]butanoic acid 1-[4-(5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-1-yl]pentan-1-one 2-methoxy-5-[3-(3-phenylpropyl)morpholine-4-carbonyl]benzonitrile 2-[(Z)-2-amino-2-fluoroethenyl]-5,6,7,8-tetrahydroquinoline-4-carboxylic acid N-[(2S)-1-amino-1,4-dioxopentan-2-yl]-3-chloro-1H-indole-6-carboxamide (6S)-2-amino-4,5,6-trimethyl-1'-[(3,4,5-trifluorophenyl)methyl]spiro[5H-pyrimidine-6,3'-indole]-2'-one 3-(hydroxymethyl)-2,5,7,8-tetramethylchromen-4-one ethane;(E)-N-methyl-3-[2-[4-(6-methylpyridin-3-yl)anilino]pyrimidin-4-yl]sulfanylprop-1-en-1-amine 6-(4,5-dichloropyridine-3-carbonyl)-3,7-dihydropyrrolo[2,3-d]pyrimidin-4-one [(2S,4R)-1-azido-4-methoxy-5-phenylpentan-2-yl]benzene 4-[4-(2-azido-1,3-thiazol-5-yl)phenyl]aniline 2-[4-(3,6-dihydroxycyclohexa-1,3-dien-1-yl)pyridin-1-ium-1-yl]acetic acid 1-butyl-3-[4-(2,5-difluorophenoxy)piperidine-1-carbonyl]pyrrolidin-2-one (2R,3S)-1-cyclopentyl-N-[(5-fluoropyridin-2-yl)methyl]-2-pyridin-4-ylpyrrolidine-3-carboxamide 2-[5-(diethylamino)pentyl]isoindole-1,3-dione (4-ethylpiperazin-1-yl)-[3-(2-methoxyphenyl)furan-2-yl]methanone 2-[3-amino-5-(trifluoromethyl)phenyl]phenol 2-methoxy-N,5-dimethylpyridine-3-sulfonamide 4-[(2S,3R)-1-tert-butylpyrrolidine-2-carbonyl]-N-propan-2-ylbenzamide 2-[4-(3,4-dimethoxyphenyl)piperazin-1-yl]-8,9-dihydropurine N-[(1Z)-3,4,5-trimethylhepta-1,6-dienyl]aniline 2,5-dimethyl-7-[(1R)-1-[3-methyl-4-(pyridin-2-ylcarbamoyl)phenyl]ethyl]pyrrolo[2,3-d]pyrimidine-6-carboxylic acid 2-N-(4-bromophenyl)-4-N-methyl-4-N-(4-propan-2-yloxyphenyl)-5-(trifluoromethyl)pyrimidine-2,4-diamine 3-[4,6-di(propan-2-yl)-1,3,5-triazin-2-yl]-9H-pyrido[2,3-b]indole 1-(2,3,3a,4,5,6a-hexahydro-1H-pentalen-2-yl)-2-methoxy-N-(1-phenylethyl)ethanamine 6-[(2S)-5-ethylpyrrolidin-2-yl]-1H-benzimidazole 2-azido-1-[4-(2,6-difluorophenyl)piperazin-1-yl]propan-1-one 4-fluorobenzenesulfinate;2-(pyridin-4-yldiazenyl)naphthalen-1-ol (2E)-1-N-[3-[1-(2,6-dioxopiperidin-3-yl)-5-fluoro-3-methylbenzimidazol-1-ium-2-yl]propyl]-2-N-(pyridin-4-ylmethyl)penta-2,4-diene-1,2-diamine N-[(1S)-2-amino-2-oxo-1-pyridin-3-ylethyl]-6-[[4-(trifluoromethoxy)benzoyl]amino]imidazo[1,5-a]pyrimidine-7-carboxamide N-[[2-hydroxy-3-(4-methylphenoxy)phenyl]methylideneamino]-2-(pyridin-2-ylsulfanylmethoxy)acetamide 1-[4-(1,2-dihydropyridine-5-carbonylamino)phenyl]piperidine-3-carboxylic acid 2-[(5-chloropyridin-2-yl)methoxy]-3-oxo-3-[6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)pyridin-3-yl]propanenitrile N-[3-(1H-imidazol-5-yl)propyl]-4-phenylbut-2-ynamide 1-[(2S,4R)-2-methoxyoxan-4-yl]-N-[6-(trifluoromethoxy)pyridin-3-yl]indazole-5-carboxamide N-[1-(8-bromoquinoxaline-5-carbonyl)pyrrolidin-3-yl]methanesulfonamide 3-azido-1,2-difluoro-4,5-bis(prop-1-enoxy)benzene 2-(4-bromo-5-methylfuran-3-yl)-1,3-oxazole N-(4,6-dimethylpyrimidin-2-yl)-4-[ethylsulfonyl(propyl)amino]benzenesulfonamide N-[1-(4-fluorophenyl)ethyl]-2,3,5,6-tetrahydro-1H-pyrrolizin-8-amine 4-[2-(3,5-dibromophenyl)phenyl]pyridine 2-[5-(4,7,8,12b-tetrahydrodibenzothiophen-3-yl)pyridin-2-yl]-[1]benzofuro[2,3-b]pyridine 4-(4-methoxyphenyl)-2,3-dihydrothiophen-5-amine N-[4-fluoro-3-(trifluoromethyl)phenyl]imidazo[1,2-a]pyrazine-8-carboxamide (E)-3-[4-bromo-2-(methoxymethyl)phenyl]-1-cyclopropylidenepropan-2-one (E)-3-[2,6-difluoro-4-(trifluoromethylsulfanylamino)phenyl]prop-2-enenitrile 1-(4,4a,6,7,8,9,10,11,12b-octahydro-3H-benzo[c]phenanthridin-1-yl)-2,2-dimethylpropan-1-one 4-[2,3-dimethyl-5-(pyrrolidine-1-carbonyl)phenyl]sulfanylbenzenethiol 1-(2,4-dimethoxyphenyl)-3-[5-methyl-6-oxo-1-[4-(trifluoromethylsulfanyl)phenyl]pyridazin-4-yl]urea 4-chloro-N',1,3-trimethylindole-2-carbohydrazide 4-[2-chloro-4-(hydroxymethyl)phenyl]-5,7-difluoro-1H-indole-2-carboxylic acid 2-[4-(2,3-dihydro-1H-inden-5-yl)piperazin-1-yl]ethanol;hydrochloride (2Z,4E)-1,5-dichloro-3-ethenyl-6-methylidenecyclohexa-1,4-diene;ethane 7-(difluoromethyl)imidazo[1,2-c]pyrimidine-5-carboxylic acid 5-ethyl-6-methoxy-3,4-dihydro-2H-chromene 1-[5-chloro-2,4-bis(phenylmethoxy)phenyl]-3-methylsulfonylthiourea [(3R,4S)-4-[4-amino-5-(7-methoxy-1H-indazol-6-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-3-fluoropiperidin-1-yl]-(4-propan-2-ylpyridin-2-yl)methanone;hydrochloride 4-[2-(3,5-dichloropyridin-4-yl)-1-oxophthalazin-6-yl]-N'-methylpiperazine-1-carboximidamide 3-methylsulfonyl-4H-furo[2,3-c]chromene N-[3,5-bis(methylamino)phenyl]ethanesulfonamide 3-[(1-benzylpyrazole-4-carbonyl)amino]-5-(4-cyclopropylphenyl)thiophene-2-carboxylic acid 3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazole-5-carbonyl]-2-fluorobenzoic acid 2-[(3R,6S)-6-methoxycarbonyl-4-[2-[1-(thiophen-2-ylmethyl)piperidin-4-yl]ethyl]-2,8-diazaspiro[4.5]decan-2-yl]acetic acid 2-chloro-5-[2-chloro-4,6-di(propan-2-yl)phenyl]thiophene 1-[4-chloro-2,6-di(propan-2-yl)phenyl]-3-[[5-cyano-2-fluoro-4-[[(1R)-4-methyl-2,3-dihydro-1H-inden-1-yl]amino]phenyl]sulfamoyl]urea 6-(4,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8,11-pentaen-3-yl)pyridine-2,3-diamine 1-methyl-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)thiourea N-[1-(1H-benzimidazol-2-ylmethyl)piperidin-4-yl]-N-ethyl-3,7-dihydro-2H-oxepine-5-carboxamide 2-[(3S)-5-ethylpyrrolidin-3-yl]-4,6-dimethylpyrimidine N-[(Z)-(3-chloro-2-hydroxyphenyl)methylideneamino]-4-(pyridin-1-ium-1-ylmethyl)benzamide 4-[(4,6-dimethylpyrimidin-2-yl)methoxy]piperidine-1-carboxylate (5Z)-2-(3,4-dimethylphenyl)imino-5-[[4-[(3-nitrophenoxy)methoxy]naphthalen-1-yl]methylidene]-1,3-thiazolidin-4-one 1-[4-(3,5-dimethyl-1H-pyrazol-4-yl)phenyl]ethanone 1-(2,3-dibromophenyl)-N-[[4-[5-(trifluoromethyl)pyridin-2-yl]oxycyclohexyl]carbamothioyl]methanesulfonamide (E)-N,3-bis(4-chlorophenyl)-2-(4,5-dihydro-1H-imidazol-2-ylmethoxyimino)pent-3-enamide N-azido-3-chloro-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-sulfonamide 4-[1-(2,3-difluorophenyl)ethylamino]quinazoline-8-carboxylic acid (Z)-3-[5-[2,6-difluoro-4-(methylaminomethyl)phenyl]pyridin-3-yl]prop-2-enal;N-(cyclobutylmethyl)formamide (6S)-2-amino-8,9-dimethyl-4-[3-(oxan-3-yloxy)propyl]-5-thia-1,7,10,11-tetrazatricyclo[6.4.0.02,6]dodeca-2(6),3,7,10-tetraen-12-one 5-[(3R)-2-acetyl-3-(2-fluorophenyl)-3,4-dihydropyrazol-5-yl]-6-hydroxy-1,3-dimethylpyrimidine-2,4-dione N-[3,4-dihydroxy-2-(hydroxymethyl)butyl]-5-[4-methoxy-6-(5-propan-2-ylsulfonylpyridin-3-yl)pyrazolo[1,5-a]pyrazin-2-yl]pyridine-3-carboxamide 3-(2,4-dimethylphenyl)-5-[1-[2-(dimethylamino)ethoxy]propan-2-yl]-1H-imidazole-2-thione (3-aminophenyl)-[4-[1-(2,6-dimethylpyridin-4-yl)ethyl]piperazin-1-yl]methanone 3-(4-fluorophenyl)-N,2-dimethylimidazo[1,2-a]pyrazine-6-carboxamide 1-[4-(4,5-dicyclopropyl-1H-imidazole-2-carbonyl)piperazin-1-yl]-2-(tetrazol-1-yl)ethanone N-[5-bromo-2-methyl-3-(trifluoromethyl)phenyl]ethanesulfonamide 1-[(2,3-dimethylcyclohexen-1-yl)methoxy]-4-ethylbenzene N-(3-bromopropyl)-2-methoxy-N,4-dinitroaniline [3-[(3,4-dichlorophenyl)carbamoylamino]phenyl]methylazanium (4aS,12aR)-9a-[3-(2,2-difluoroethyl)benzimidazol-5-ylidene]-1,3,4,5,11,12-hexahydropyrido[3,4-b]acridin-12a-ol 2-[4-[1,3-benzothiazol-2-yl(1H-inden-1-yl)amino]phenyl]sulfonylethanol N-[4-chloro-2-(7H-purin-6-yl)phenyl]oxazinane-3-carboxamide 3-[(2S,4R)-1-cyclopropylsulfonyl-4-fluoropyrrolidin-2-yl]-5-propan-2-yl-1H-pyrazole 6-butyl-1,2,3,4-tetrahydropyrido[1,2-a]benzimidazole 7-methyl-2-(4-methylidenepiperidine-1-carbonyl)chromen-4-one 2-(4-methyl-1H-pyrrol-3-yl)-5,6,7,8-tetrahydroquinoline 2,4-diphenyl-6H-cyclohepta[b]thiophene 4-fluoro-1,3-bis(phenylmethoxy)cyclohexa-2,4-dien-1-amine 4-hydroxy-5,6-dimethyl-3-[[4-(3-phenylmethoxypropyl)piperazin-1-yl]methyl]pyran-2-one N-[[4-(6,7-dimethoxyquinazolin-4-yl)phenyl]methyl]propan-1-amine 2,5-diamino-3-[(2R)-2-hydroxyhexyl]-8-methoxyquinazolin-4-one 2-[(3R,4S)-4-(6-methylpyridin-2-yl)piperidin-3-yl]oxypyrazine 2-(3,4-dimethoxyphenyl)-N-[5-(3,4-dihydropyrazol-2-yl)pent-4-yn-1-yl]-N-methylacetamide 6-benzylsulfanyl-5,7-dihydropyrrolo[3,4-d]pyrimidine 1-(4-azidooxyphenyl)-3-chloropropane-2,1-diol (5Z)-5-[(7-bromonaphthalen-2-yl)methylidene]-2-(4-chlorophenyl)imino-1,3-thiazolidin-4-one 2-amino-6,8-dimethyl-7H-purine-1,3-diium-5-thione 3-(2-ethoxyphenyl)-1,1-dimethylurea N-[4-(7,8-dihydronaphthalen-1-yl)phenyl]-6-propoxycyclohexa-2,4-dien-1-imine N-(3-cyanopyrazin-2-yl)-6,7-dihydroquinoline-5-carboxamide 1-azido-3,5-dichloronaphthalene 5-[3-amino-4-(2-methylpyrazol-3-yl)phenyl]pyrimidine-2,4-diamine;ethane 3-[(1S)-2,3,4-trifluorocyclohexyl]benzaldehyde 1-(4-ethoxyphenyl)sulfonyl-6,7-dimethylindolizine-3-carboxylic acid 2-[3,5-bis(trifluoromethyl)phenyl]-3H-pyrrole [3-(4-hydroxyphenyl)morpholin-4-yl]-[3-(2H-tetrazol-5-ylsulfanyl)phenyl]methanone 2-[(2Z)-4-oxo-2-[(Z)-propan-2-ylidenehydrazinylidene]-1,3-thiazolidin-5-yl]-N-phenylacetamide 2-N,7-diethylpyrene-1,2-disulfonamide (3S,4R)-1-[5-cyclopropyl-2-[2-methoxyethyl(methyl)amino]pyridine-3-carbonyl]-N-cyclobutyl-3-fluoropiperidine-4-carboxamide N-(2-fluorophenyl)-3,6-dimethylthieno[2,3-b]pyridine-2-carboxamide 2-(3,5-difluorophenyl)-4-[4-[1-ethyl-6-oxo-4-(trifluoromethyl)pyridin-3-yl]phenoxy]-N'-hydrazinylthieno[3,2-c]pyrazole-5-carboximidamide N'-hydroxy-3-(4-methylsulfonylpiperazine-1-carbonyl)pyridine-2-carboximidamide (2Z)-N,4-dimethylpenta-2,4-dienamide;ethane;2-[6-(5-oxospiro[6H-naphthalene-7,1'-cyclopentane]-3-yl)oxyhexyl]guanidine 1-[5-bromo-4-chloro-2-(difluoromethyl)phenyl]ethanone 5-azidooxy-2,3-dihydrobenzo[g]indazole N-cyclohexyl-6,7-dihydroquinazoline-5-carboxamide 1-(4,5-dimethylcyclohexen-1-yl)-3,5-diphenylbenzene 7-bromo-5,6-dimethylnaphthalene-1-carbonitrile (E)-3-[4-[4-(dimethylamino)phenyl]sulfonyloxynaphthalen-1-yl]prop-2-enoic acid (Z)-2,4-diamino-4-methoxy-N'-[1-[[2-methyl-5-[(2R)-5-oxopyrrolidine-2-carbonyl]phenyl]methyl]piperidin-3-yl]but-2-enimidamide 4-[2-(oxan-2-yl)benzimidazol-1-yl]piperidine-1-carboxamide 3-[5,7-bis(4-chlorophenyl)-1-methyl-2-oxo-3H-imidazo[1,2-b]pyrazol-3-yl]benzoic acid 4-[2,3-bis(4-aminophenyl)benzoyl]-1H-pyrrole-2-carboxamide 2-[2-(4-fluorophenyl)-5-[1-[4-[[(2S)-oxiran-2-yl]methoxycarbonylamino]cyclohexyl]piperidin-4-yl]anilino]acetic acid 3-(4-azidophenyl)-5-(3,7-difluoroheptanoylamino)thiophene-2-carboxylic acid 2-[4-(4-ethoxy-3,5-difluorophenyl)-3,5-difluorophenyl]-1,3-difluoro-6-propylnaphthalene 2-azido-5-bromo-4,6-dimethylbenzene-1,3-dicarbonitrile 2-[4-ethyl-6,7-difluoro-1-[[4-(trifluoromethoxy)phenyl]methoxy]naphthalene-2-carbonyl]oxypropanoic acid 6-[(5Z)-4-methylhepta-1,3,5-trien-3-yl]-2,8-dihydro-1H-quinazoline 4-[6-bromo-2-chloro-3-(trifluoromethyl)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile [1-(4-ethylphenyl)sulfonylpyrrolidin-2-yl]-morpholin-4-ylmethanone 2-(3,4,5-trimethylphenyl)iminopyrido[2,1-a]isoindole-1,3-dione 5-ethyl-1,3-bis(methoxymethyl)-6-nitrobenzimidazol-2-one 7-(2,6-difluorophenyl)-12-[2-fluoro-4-(1H-pyrazol-5-yloxy)phenyl]-3-methyl-2,3,11,13-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene 7-benzyl-6,10-dihydroxy-3-(4-methoxyphenyl)imino-1-azatricyclo[7.3.1.05,13]trideca-9,11-bis(13),12-triene-2,4-dione 4-[2,3,6-trichloro-5-(1H-indole-4-carbonyloxymethyl)phenyl]butanoic acid (2S)-3,4,5-trihydroxy-6-(oxolan-2-ylmethoxycarbonylamino)-7-phenylmethoxyheptanoic acid 1-(2,6-dimethyl-4-nitrophenyl)piperazine 3-amino-5-[2-(difluoromethyl)pyridin-4-yl]-6-(3-ethoxyphenyl)pyrazine-2-carboxamide N-[4-fluoro-3-(trifluoromethyl)phenyl]formamide;4-hydroxy-5-methoxy-2,8-dipropyl-3H-2,7-naphthyridine 2-[[4,5-dimethyl-3-(2-methylphenyl)pyrazol-1-yl]methyl]-N-methylbenzamide 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]oxirane-2,2-dicarbonitrile 1-(4,6-dimethoxypyrimidin-2-yl)-3-[5-[2-(dimethylamino)ethylsulfanyl]-6-oxo-11H-benzo[c][1]benzazepin-8-yl]urea 4-(8,14-dioxapentacyclo[11.7.0.03,11.04,9.015,20]icosa-1(13),2,4(9),5,7,11,16,18-octaen-7-yl)pyrimidine 5-[3-(4,4-difluorocyclohexyl)oxypyrrolidine-1-carbonyl]furan-2-carbonitrile 2-[3-(5-bromopyrimidin-4-yl)oxypyrrolidin-1-yl]pyrazine 4-(9H-fluoren-1-yloxy)-6-[4-(1H-imidazol-5-ylmethylcarbamoylamino)phenyl]pyrimidine-2,4-dicarboxamide 5-methyl-6-(4,4,5,5-tetrafluoropentoxy)pyridine-3-carboxylic acid 2-(dimethylamino)-1,3-dihydroindazole-5-carboxylic acid 4-azidooxy-2,6-difluoro-3-(trifluoromethyl)benzonitrile 5-chloro-4-[methyl(oxan-3-yl)amino]-1H-pyrimidin-6-one 4-[(Z)-(3,5-dimethoxyphenyl)methylideneamino]-3-(oxolan-2-ylmethylsulfanyl)-1H-1,2,4-triazol-5-one 2-amino-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxylic acid;6-chloro-2-ethyl-3,4-dihydroisoquinolin-1-one 1-[(2,6-difluorophenyl)methyl]-3-(ethoxymethylamino)thiourea 6-[2,5-bis(trifluoromethyl)phenyl]imino-3,4-dihydro-2H-benzo[b][1]benzoxepine-1-carboxylic acid;ethane 2-(6,7-dihydronaphthalene-1-carbonylamino)-N-[2-(4-ethylphenyl)ethyl]pyridine-3-carboxamide [4-[5-bromo-3-(2,6-dichlorophenyl)pyrazol-1-yl]phenoxy]boronic acid N'-(2,5-dimethylphenyl)sulfanyl-3,4-dihydropyridine-6-carboximidamide N-[1,3-bis(4-hydroxyphenyl)propan-2-yl]-N',5-dimethylfuran-2-carbohydrazide 4-[4-(1-azidoethyl)phenyl]benzene-1,3-diol 3-[5-(2,4-difluorophenyl)-1H-imidazol-2-yl]pyrazine;ethane N-benzyl-3-(6,7-dimethoxyquinolin-4-yl)oxyaniline 1-[(6R)-2-(5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carbonyl)-6,11-dihydroxy-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-6-yl]propan-2-one 4-(3,5-dichloroanilino)-6-methylpyrimidine-2-carbonitrile 2-[(3Z,5E)-6-aminohepta-1,3,5-trien-4-yl]-7-chloroquinolin-8-ol;1-cyclohexa-1,5-dien-1-ylazetidine-3-carboxylic acid N-[[1-(2,5-dihydroxyphenyl)isoquinolin-6-yl]methylideneamino]pyridine-3-carboxamide 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5-ethylpyrazole N-[1-(4-methylthiadiazole-5-carbonyl)piperidin-3-yl]acetamide (5E)-2-imino-3-methyl-5-[[4-(N-phenylanilino)phenyl]methylidene]-1,3-thiazolidin-4-one 5-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-2-yl]imidazolidine-2,4-dione 6-(2,3-difluorophenyl)-1-[2-[[4-methyl-5-(1H-pyrazol-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one 3-(2,6-dichlorophenyl)-4-hydroxy-5-(1H-imidazol-5-ylmethylidene)-1-[2-(4-nitrophenoxy)ethyl]pyrrolidine-2-thione ethane;[2-(trifluoromethyl)phenyl]urea 2-[3-(aminomethyl)phenoxy]-N-[1-hydroxy-5-[3-(4-methoxyphenoxy)propoxy]pyridin-1-ium-3-yl]acetamide;bromide 3-chloro-N'-hydroxy-2-(trifluoromethyl)pyridine-4-carboximidamide N-[(E)-3-bromopropylideneamino]methanamine;2,4-ditert-butyl-6-ethynylphenol 4-[2,3-bis(ethenyl)cyclobutyl]benzoic acid N-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl]-3-methyloxetane-2-carboxamide 1-(cyclopropanecarbonyl)-N'-[(3S,4R)-3-hydroxyoxan-4-yl]pyrazole-4-carboximidamide;dihydrochloride 3-ethyl-2,6-dimethoxyquinazolin-4-one 1-(2,3,6-trifluoro-5-pyridin-4-ylphenyl)propan-2-one N-(2,5-dimethylphenyl)-4-methylpyridine-3-carboxamide (3R)-1,4-dibenzyl-N'-hydrazinylpiperazine-2-carboximidamide (7R)-2-[(4-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 4-[5,5-bis(4-hydroxyphenyl)-2H-tetrazol-1-ium-1-yl]benzenesulfonamide 2-(N-methylanilino)-5,6,7,8-tetrahydroquinoline-3-carbonitrile 6-[(4S)-2,8-dimethyl-3,5,7,9-tetrahydropyrido[4,3-b]azepin-4-yl]-1H-indole 3-[2,6-dimethyl-4-(6-methylpyridine-3-carbonyl)piperazin-1-yl]oxolane-3-carbonitrile 2-hydroxy-1,3-diphenylbutane-1,4-dione 2-[5-(carbamoylamino)-6-(4-chloroanilino)pyridine-3-carbonyl]oxyacetic acid 3-(5-aminotetrazol-1-yl)-N-cyclopropyl-4-methoxybenzamide (1S,3R)-1-N'-[5-fluoro-4-[6-methoxy-7-[(2-methyl-1,3-benzothiazol-6-yl)oxy]quinolin-4-yl]oxyphenyl]-1-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide 2-azidooxy-1,3-difluoro-5-(4-fluorophenyl)benzene 3-[5-azidooxy-2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-4-ylmethoxy)phenyl]-4-phenyl-1H-pyrrole-2-carboxylic acid 4-[(2,3-dibromo-6-hydroxyphenyl)methylideneamino]-1H-pyrazole-5-carboxylic acid 5-cyclohepta-1,4,6-trien-1-yloxy-4-methyl-3,6-dihydro-2H-pyridine;ethane 6-(1,3-benzodioxol-5-yl)imidazo[2,1-b][1,3]thiazole 2-[(2,6-dimethoxyphenyl)methyl]-7-morpholin-4-yl-5-pyrimidin-5-ylsulfanylthieno[3,2-b]pyridine 2-(azidomethyl)-1,3-difluorobenzene 2-hydroxyimino-1,4-dipyridin-3-yl-6,7-dihydro-5H-indole-3-carboxamide 3-(5-azidopyridin-2-yl)-2H-pyrazolo[3,4-b]pyridine 3-chloro-2,5-difluoro-N-(4-methylphenyl)aniline N-[6-(2,3-dihydroindol-1-ylmethyl)imidazo[1,2-a]pyridin-2-yl]benzamide 3-[4-[2-(1,3-benzothiazol-6-ylamino)-5-methoxypyrimidin-4-yl]pyrazol-1-yl]-N-ethoxypropanamide 4-(5-azido-2,3-dichlorophenyl)-N-methylaniline 2-azido-5,6-dibenzylpyrimidine [2-(cyclopropylmethoxy)phenyl]-[4-(pyridin-3-ylmethyl)piperidin-1-yl]methanone 5-methyl-7-[3,4,6-trichloro-2-(deuteriosulfanyl)phenyl]-1H-indole 2-tert-butyl-4-[1-(disulfanyl)ethyl]phenol N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethoxy)-2-[[4-(trifluoromethyl)phenyl]sulfonylamino]benzamide (2R)-N-[2-chloro-5-[[(1S,3R)-3-[4-(trifluoromethyl)phenyl]cyclohexanecarbonyl]amino]benzoyl]piperidine-2-carboxamide 4-[[1-(2,5-dimethylphenyl)-6-hydroxy-3-propanoyl-7,8-dihydronaphthalen-2-yl]amino]benzoic acid 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidin-4-imine N-[3,5-bis(trifluoromethyl)phenyl]-2-(4-chlorophenyl)-1H-imidazo[4,5-b]pyridin-7-amine N-[2-[(3S)-3-aminopyrrolidin-1-yl]-4-methoxyphenyl]thieno[2,3-c]pyridine-2-carboxamide 2-[(3,4-dimethylphenyl)iminomethyl]-6-iodophenol 2-[4-ethenyl-5-methoxy-3-(methylideneamino)-1H-pyrazol-2-ium-2-yl]-N-(5-fluoropyridin-2-yl)acetamide N-cyclopentyl-6-hydroxy-4,5-dimethylpyrimidine-2-carboxamide 2-azido-1,3,5,6-tetrachlorobenzene N-[1-(2,4-dichlorophenyl)ethenyl]-5-ethenylpyrazin-2-amine 4-amino-N-[3-(4-methylpiperazin-1-yl)propyl]benzamide (6Z)-3-[5-ethyl-1-methylidene-3-oxo-2-[4-(trifluoromethyl)phenyl]isoindol-4-yl]-6-hydrazinylidenehexanoic acid N-[2-(3,5-dimethylphenyl)pyrazol-3-yl]butanamide [4-(3,3-dichloroprop-2-enoxy)phenyl]methanol 4-methyl-N-[1-(pyridine-3-carbonyl)piperidin-3-yl]quinazoline-8-sulfonamide [4-(4-amino-3,5-dimethylphenyl)sulfanyl-2-methoxy-3-(1H-pyrrole-2-carbonylamino)butanoyl]oxidanium 4-methoxy-6-[5-[3-[2,2,2-trifluoro-1-[3-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]ethoxy]-1H-pyrazole-5-carbonyl]pyridin-2-yl]pyridine-3-carboxylic acid 3-[5-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]-1H-pyridazine-6,7-dione 2-(3,4-dihydropyridin-6-yl)indole 1,2-diamino-4-[2-chloro-3-(trifluoromethoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile (4-ethenylphenyl)-[(E)-2-[[(Z,1S,3E)-1-(methylideneamino)penta-1,3-dien-3-yl]amino]ethenyl]azanium 1-[5-(3,3-dichloropropoxy)-4,6-dimethylpyrimidin-2-yl]pyrrolidine-3,4-diol 6-[4-bromobutan-2-yl(hexadecanoyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 6-[(2E)-2-butan-2-ylidenehydrazinyl]pyrimidine-4-carboxamide 4-[2-methyl-3-(piperidine-1-carbonyl)indol-1-yl]cyclohexan-1-one 3-chloro-4-(trifluoromethyl)-1,3-dihydroquinoxaline-2,6-dione (1Z)-1-[3-bromo-4-[(2,6-difluorophenyl)methoxy]-6H-benzo[c][1]benzoxepin-8-ylidene]guanidine N-[6-[3-(2,4-dioxo-1H-pyrimidin-5-yl)propanoyl]pyridin-2-yl]benzamide 5-N-[(3,4-difluorophenyl)methyl]-2-N-(2-propan-2-ylidenehydrazinyl)thiophene-2,5-dicarboxamide 2-(3,4-dimethoxyphenyl)-6-[[5-[3-(trifluoromethyl)phenyl]furan-2-carbonyl]amino]chromene-4-carboxylic acid 1-[[4,5-bis(ethenyl)furan-2-yl]methylamino]hexan-3-one;cyclopropane 2-methyl-5-(N-prop-2-enoylanilino)benzenesulfonic acid 1-[2-azidooxy-6,8-dimethyl-3-(methylideneamino)naphthalen-1-yl]ethanone N-[(3R)-3-[[4-amino-3,5-difluoro-2-(trifluoromethoxy)phenyl]sulfonylamino]-1-bicyclo[1.1.0]butanyl]-3-fluoropropane-1-sulfonamide N-[5-(furan-3-yl)-2-(6-oxo-4-propan-2-yl-1H-pyrimidin-2-yl)pyrazol-3-yl]-3,5-dimethoxybenzamide 4-[(4,5-diphenyl-1,3-oxazol-2-yl)methoxyimino]azepine-2-carboxylic acid N'-[(1R,2S)-1-methoxy-1-phenylpropan-2-yl]butanediamide 4-bromo-2,5-dimethyl-N-(3-oxo-3-piperazin-1-ylpropyl)-N-phenylbenzenesulfonamide;2,2,2-trifluoroacetic acid 4-(2-azidopropyl)benzamide N-[(3R,4S)-1-benzyl-3-methoxypiperidin-4-yl]acetamide;hydrochloride (E)-3-[4-chloro-3,5-bis[(2-fluorophenyl)methoxy]phenyl]-N-[4-(difluoromethylsulfonyl)phenyl]prop-2-enamide 3-[2-hydroxyethyl(methylsulfonyl)amino]-N-[6-(1,2,4,5-tetrazin-3-yl)pyridin-2-yl]-2,3-dihydrothiophene-5-carboxamide N-[(2R)-1,1-bis(4-chlorophenyl)propan-2-yl]-3-fluoroaniline (5R,7S)-N-[(3R)-1-[(2,4-difluorophenyl)methyl]piperidin-3-yl]-5,7-dimethyl-1,4,5,7-tetrahydropyrano[3,4-c]pyrazole-3-carboxamide 2-[(Z)-2-hydroxy-3-phenylprop-1-enyl]oxiran-2-ol 3-bromo-1-(3,5-dichloropyridin-4-yl)-2H-pyridine 6,7-dimethoxy-3H-quinazolin-4-one 4-tert-butyl-2,6-difluoro-N'-(3-propan-2-ylidenecyclohexyl)benzenecarboximidamide 3-[(1R,2S)-2-methylcyclopentanecarbonyl]-N-phenylbenzenesulfonamide 1-(3,4-dihydro-2H-chromen-6-yl)propan-2-one 2-(9H-fluoren-1-yl)-3,4,6-trimethylquinoline N-[(6S)-6-benzylsulfanyl-4,5-dihydro-1,3-oxazin-2-yl]pyridine-3-carboxamide 4-(4,4,5,5-tetramethyloxaborolan-2-yl)thieno[3,2-d]pyrimidine 6-bromo-4-[(3R)-3-methoxypyrrolidin-1-yl]-2-phenylsulfanylquinazoline 5-[(E)-2-[3,5-bis(trifluoromethyl)phenyl]ethenyl]-1,3-benzodioxole;ethane 2-[[(Z)-(3-ethoxyphenyl)methylideneamino]carbamothioyl]benzoic acid 2-[7-(aminomethyl)-4,9-dihydropyrazolo[3,4-f]quinolin-3-yl]benzenesulfonamide;ethane 6-[4-(1,3-benzodioxol-5-yl)phenyl]-N-(3-chlorophenyl)pyrazin-2-amine N-(4,6-dimethylpyrimidin-2-yl)-4-[ethylsulfonyl(pyridin-3-yl)amino]benzenesulfonamide 3-(4-bromophenyl)-4-nitrocyclohexa-1,5-diene-1,2-dicarboxamide 6-amino-1,3-dimethylpyrazolo[3,4-d]pyrimidine-7-carboxylic acid 2-cyclohexyl-3,6,7-trimethoxychromene-4,5-dione 3-(2,6-difluorophenyl)-4-[(2,5-dimethylphenyl)sulfonylamino]benzoic acid;2,2,2-trifluoroacetic acid 1-[(2S,4R)-2-amino-5-ethoxycarbonylpiperidin-4-yl]-3-ethoxypyrazole-4-carboxylic acid 4-(2,4-dichlorophenyl)sulfanyl-7-propoxybicyclo[3.1.0]hexane 2-methyl-N-[4-(tetrazolo[1,5-a]quinoxalin-8-ylamino)phenyl]propanamide N-[(3S,4R)-1-methyl-4-propan-2-ylpyrrolidin-3-yl]-4-[(E)-[(6-nitroquinazolin-4-yl)hydrazinylidene]methyl]benzamide (1R,2S)-3-[5-amino-6-[2,4-difluoro-5-[[2-methylpropyl-(2-morpholin-4-ylethylcarbamoyl)amino]methyl]phenyl]pyrazine-2-carbonyl]cyclopentane-1-carboxylic acid 2-(3,4,6,7-tetrahydro-1H-pyrrolo[3,4-c]pyridine-5-carbonyl)-1-benzofuran-3-carboxamide N-[2-(2,3-dihydroindol-1-yl)ethyl]-2-[5-(4-methoxyphenyl)pentanoylamino]acetamide [(2R,5S)-4-hydroxy-5-methoxy-2-methyl-3,4-dihydro-1H-naphthalene-2-carbonyl]azanium 1-(2,4-dimethylphenyl)-3-[5-(furan-2-carbonylamino)naphthalen-1-yl]urea 2-[(6R)-4-(5-chloro-1H-indazole-7-carbonyl)-2,6-dimethylpiperazin-1-yl]acetaldehyde 4-bromo-2,6-dichloro-N-diazobenzenesulfonamide 5-(4-bromo-2,6-difluorophenyl)-3H-1,3,4-oxadiazol-2-one 1-[(3E)-6,7-dimethylocta-1,3,5,8-tetraen-4-yl]oxyethenamine;ethane 2-[(4,6-dimethyl-1,3,5-triazin-2-yl)amino]-1-(3-fluorophenyl)ethanol 4-[2-(furan-2-yl)ethynyl]-5-methoxy-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaene 6-bromo-2-[1-(4-fluorophenyl)-3H-pyrazol-2-yl]quinazoline N-(4-methylphenyl)sulfanyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide 4-(4-fluorophenyl)-6,8-dihydro-5H-pyrido[3,2-d]pyrimidine 1-[2,6-di(propan-2-yl)phenyl]sulfanyl-4-methoxyazetidine ethane;methanamine;4-[(2E,3Z)-penta-2,3-dienyl]-N-(1-phenylethenyl)aniline [3-[(4,6-dimethylpyrimidin-2-yl)amino]pyrrolidin-1-yl]-(4-propan-2-yloxyphenyl)methanone 3-(4-bromophenyl)-7,7a-dihydroisoindole 3-(1,3-benzodioxol-5-yl)-2H-[1]benzofuro[2,3-d]pyrimidin-8-ol N-[[4-chloro-3,5-bis(difluoromethyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-8-yl]methanimine N-[2-(3,5-dichloropyridin-4-yl)ethylidene]hydroxylamine N-[2-(2,4-dimethylphenyl)ethyl]-7H-purin-6-amine [2-[(5R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-5-yl]morpholin-4-yl]-thiophen-3-ylmethanone;dihydrochloride ethane;3-[(4Z)-2,6,6-trimethylhepta-1,4,5-trien-3-yl]pyrido[1,2-a]pyrimidin-4-one 1-[4-(1,3-benzothiazol-2-yl)-7-methoxyindol-1-yl]ethanone 4-chloro-5-methyl-2-propan-2-ylidene-3H-1,3-benzoxazole 5-(1,3-benzodioxol-4-ylmethyl)-2-[[hydroxy-[5-[(E)-pent-1-enyl]thiophen-2-yl]methoxy]methylidene]cyclohexane-1,3-dione 2-(5,6-diphenylpyrimidin-4-yl)propanamide 2-(3,5-diphenyl-1,2-oxazol-4-yl)acetic acid 1-[3-(2,4-dichlorophenoxy)propyl]azetidine 2-(3-chlorophenyl)-N-[4-(5,6,7,8-tetrahydroquinolin-4-ylamino)butyl]acetamide N-[(1R)-1-naphthalen-2-ylethyl]acetamide 2-methoxy-4-[3-(oxolan-3-yl)pyridine-4-carboximidoyl]aniline N-[3-(6,7-dihydropyrrolo[2,1-c][1,4]benzoxazepin-8-yl)-4-hydroxyphenyl]-2-fluoroacetamide 2-[5-(4-amino-3,5-dichlorophenyl)-1H-imidazol-2-yl]pyridin-3-ol (Z)-3,7-diethyl-6-hydroxynon-5-enoic acid;1-phenylisoquinoline (4E)-2-[4-(4-bromophenyl)sulfonylpiperazine-1-carbonyl]-3,4-dihydro-1H-quinoline-6-carbonitrile N-[5-(2,6-dimethoxyphenyl)-1,3-thiazol-2-yl]-4-[3-hydroxypropyl(methyl)amino]benzamide 2-(4-benzoylanilino)-N,N-dibutylacetamide (3-fluorophenyl)-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-6-yl)methanone 6-[2-hydroxyethyl(propan-2-yl)amino]-5,6,7,8-tetrahydronaphthalene-1,3-diol 1-[3-(3,4-dimethoxyphenyl)propyl]azetidine 4-[3-[4-[4-(1,2,6-trimethylindole-3-carbonyl)piperazin-1-yl]piperidine-1-carbonyl]-7,8-dihydropyrido[3,4-b]pyrazin-5-yl]benzonitrile (1S)-3-[(3R)-3-methylpyrrolidin-1-ium-1-ylidene]-1,2-dihydronaphthalene 1-ethylsulfanyl-2,3-dimethoxyanthracene 2-[4-[5-chloro-3-(trifluoromethyl)pyrazole-1-carbonyl]piperazin-1-yl]ethanesulfonamide N-[5-cyano-6-(1,3-thiazol-2-yl)pyridin-3-yl]acetamide;4-[3-methyl-4-(methylamino)phenyl]morpholine 6-N-[3-fluoro-4-(trifluoromethoxy)phenyl]-2-(5,8,11-triazatricyclo[7.4.0.02,7]trideca-1(9),10,12-trien-13-yl)-1H-pyrimidine-2,6-diamine N-[(Z)-[2,4-bis(ethenyl)phenyl]methylideneamino]-3-hydroxy-5-sulfanylpyridine-2-carboxamide 1-[(2S)-4-[7,8-difluoro-6-(2-fluoro-5-methoxyphenyl)quinazolin-4-yl]-2-ethylpiperazin-1-yl]prop-2-en-1-one N-[2-(4,5-dihydroimidazol-1-yl)ethyl]-6-piperidin-4-yloxyquinazolin-4-amine;hydrochloride 1-[2,6-di(propan-2-yl)phenyl]-3-(2-methoxyethylsulfanyl)thiourea 3-[3,5-dimethyl-4-(2-pyrrolidin-1-ylethoxy)phenyl]-N-piperidin-1-ylbenzamide 2-tert-butyl-1'-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazole-1-carbonyl)spiro[7H-furo[3,4-b]pyridine-5,3'-azetidine]-8-one N-[4-(2,3-dichlorophenyl)-1,3-thiazol-2-yl]carbamate 2-[(2Z)-2-ethenylpenta-2,4-dienyl]benzoic acid 2,6-difluoro-N-[(3S)-1-[4-(trifluoromethylsulfanylamino)benzoyl]pyrrolidin-3-yl]cyclohexa-1,5-diene-1-carboxamide 5-methyl-3,4,7-tris(phenylsulfanyl)quinoline 4-[2-(1H-imidazol-5-yl)ethynyl]-N-(oxolan-3-ylmethoxy)benzamide N-[3-(4,5-dihydro-1H-imidazol-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]formamide 3-azidooxy-6,11-dihydrobenzo[c][1]benzoxepine N-(2,6-difluorophenyl)-N'-[5-methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]propanediamide 2-amino-4-(3-cyanophenyl)benzenecarboximidamide N-[(1S)-2-(3,4-dimethylphenyl)-1-[5-methoxy-6-oxo-2-(trifluoromethyl)pyrimidin-1-yl]ethyl]formamide N-[4-(benzylcarbamoylamino)butyl]-2-ethoxy-2-phenylacetamide 4-bromo-6-chloro-2,3-difluorobenzaldehyde 6-ethyl-4-methoxycarbonyl-2,3-dihydrobenzoic acid 4-[5-(cyclohexylmethylamino)pyridin-2-yl]-N',1,5-trimethylpyrrole-3-carbohydrazide ethane;N-[2-(4-fluorophenyl)-1,3-benzodioxol-5-yl]-N'-methanimidoylbenzenecarboximidamide N-(4-bromobutan-2-yl)-N-(1,3-thiazol-5-yl)ethenesulfonamide N-ethyl-2-methoxy-N,4-diphenylaniline 4-[6-(3-aminoanilino)-9H-carbazol-3-yl]-N,N-dimethylbenzamide 2-[(2-ethoxyphenyl)methyl]-N'-hydroxypyrimidine-4-carboximidamide N-(4-hydroxyphenyl)-N'-[(Z)-(2-oxo-1H-quinolin-3-yl)methylideneamino]oxamide 2-[4-(dimethylamino)piperidine-1-carboximidoyl]pyridine-3,5-diamine 2-(3,4-difluorophenyl)-7-heptoxy-9-hydroxypyrano[2,3-c]quinolin-6-one 3-(6-bromoheptyl)-2-methoxy-1,5-diphenylpyrrole 4-[2-(trifluoromethyl)phenyl]sulfanylidenepiperidine 2-(4-bromophenoxy)-3-(methylamino)propanal 2-[3,5-dichloro-4-(3,6-dihydro-2H-pyran-4-yl)anilino]propanoic acid (2S)-1,2-diphenyloctane-2,4-diol 6-[(3-chlorophenyl)methylsulfonylamino]-1,2-benzoxazole-4-carboxylic acid 1-ethylsulfonyl-4-(2-phenylethynyl)benzene 3-(hydroxymethyl)-5-[[2-methoxy-6-(trifluoromethyl)pyrimidin-4-yl]amino]benzonitrile 4-(4-bromophenoxy)phenol 2-[[6-(3,4-difluorophenyl)pyridin-3-yl]methyl]isoindole-1,3-dione 3-(4,5,6,7-tetrahydro-1-benzothiophen-2-ylsulfonyl)butanenitrile N-[3-[4-(4-methoxyphenyl)sulfonylpiperazin-1-yl]propyl]benzamide 1-N,3-N-dimethylbenzene-1,3-dicarboxamide;ethane [(2R,3S)-3-azido-2-methylpiperidin-1-yl]-(4-pyridin-3-ylphenyl)methanone (6S,7R)-3-[4-(1-fluorocyclopropanecarbonyl)piperazine-1-carbonyl]-7-methoxy-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid N-(4-anilinophenyl)-N-butylethenesulfonamide 2-[4-cyano-3,5-di(propanoyl)phenyl]sulfanyl-6-methylbenzenesulfonate 3-[4-chloro-3-(trifluoromethyl)phenyl]-5,5-dimethyl-1-(2-methylpropyl)imidazolidine-2,4-dione 5-[[(Z)-1,2-diaminoethylideneamino]carbamoyl]-N'-[3-(trifluoromethyl)phenyl]thiadiazole-4-carboximidamide 4-[5-(3,4-difluorophenyl)-2-hydroxypentoxy]benzoic acid [(2-amino-3,5-difluorophenyl)methyl-[1-[3-carbamoyl-4-[(E)-2-[2-[ethyl(methyl)amino]ethenylsulfanyl]ethenyl]anilino]-1-oxopropan-2-ylidene]azanium 1,4-difluoro-6-[2-fluoro-4-[(E)-pent-3-enyl]phenyl]naphthalene-2-carbonitrile 2-(methylamino)-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one N-[(2R)-3-hydroxy-1-[4-(5-methylsulfanylpyrimidin-2-yl)phenyl]propan-2-yl]formamide N-[(1R,2S)-2-methylcyclohexyl]spiro[4H-quinoxaline-3,1'-cyclopentane]-2-imine 2-[(4-acetamidophenoxy)methyl]piperidine-1-carboxylic acid 3-(7,8-dimethoxyquinazolin-4-yl)-2-fluorobenzamide N-butyl-5-(1H-indol-2-ylamino)pentanamide 4-[(6R)-7-acetyl-3-pentanoylsulfanyl-1,2,4-triazin-5-yl]-3-methoxybenzoic acid N-[(2S)-5-[(3,4-dichlorophenyl)methylsulfanyl]-1-(8-ethynoxyoctylamino)-1-oxopentan-2-yl]cyclohexanecarboxamide 5-[1-(4,6-dichlorocyclohexa-2,4-dien-1-yl)sulfonylpiperidin-3-yl]-3H-pyrido[3,4-d]pyrimidine-4,7-dione [3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methanesulfonate 1-[4-(dimethylamino)-N-(4-hydroxybutyl)anilino]propan-2-one 1-[(4R)-2,4-bis(hydroxymethyl)pyrrolidine-1-carbonyl]-3-cyclopentylpyrazole-4-carboxylic acid 1-(2-ethoxyethyl)-7,8-dimethyl-6-(4-methylpiperazine-1-carbonyl)-5,9-dihydropyrazolo[3,4-h]quinazolin-4-one [2-(4,6-diaminopyrimidin-5-yl)-6-fluoro-7H-pyrrolo[2,3-d]pyrimidin-4-yl]carbamic acid 4-N-(1-aminoethyl)-5-chloro-2-N-[2-methoxy-4-morpholin-4-yl-5-nitro-3-(trifluoromethyl)phenyl]pyrimidine-2,4-diamine;ethane 1-[[3-(2,6-difluoro-4-methoxyphenyl)triazolo[4,5-d]pyrimidin-5-yl]amino]propan-2-one;hydrochloride 2-methylpropane;4,5,6,7,8,9-hexahydrocycloocta[b]pyridine-3,7-dicarboxylic acid (2R)-1-[(3-fluoropyridine-4-carbonyl)amino]piperidine-2-carboxylic acid N-[(2R,3S)-1-(2,4-difluorophenyl)-4-(ethylamino)-2-hydroxy-5-oxopentan-3-yl]-2-[6-fluoro-2-methoxy-4-(3-pyrrolidin-1-ylprop-1-ynyl)cyclohexa-1,3-dien-1-yl]acetamide N-[2-[[4-(benzylamino)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-2-yl]amino]-5-chlorophenyl]propanamide 1-(3,5-diethoxyphenyl)heptan-2-one 1-butyl-2,3,5-trimethoxybenzene 6-[1-(4-ethylphenyl)sulfinylpiperidin-3-yl]-1,5,7,10-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaene 5-(4,6-dimethylpyrimidin-2-yl)sulfanyl-1,3,8a-trimethyl-9H-[1]benzofuro[2,3-b]pyridine 2-(5-amino-3-fluoropyridin-1-ium-2-yl)sulfanyl-4-propyl-1H-pyrimidin-6-one 5-methoxy-1,3-dimethyl-2-(trifluoromethyl)indole 2,5-difluoro-4-(3-methylbutoxy)benzaldehyde [1-methyl-3-(2H-tetrazol-5-yl)indol-4-yl]boronic acid 1-[(5R)-2,7-diazaspiro[4.5]decan-2-yl]-2-(3-ethoxyphenyl)sulfanylprop-2-en-1-one (4R)-1-benzyl-N,2-dimethylpiperidin-3-amine 6-[(2R,4S)-2-methylpiperidin-1-yl]pyridazine-3-carboxamide 3-[5,6-dimethyl-2-(1H-pyrrolo[2,3-c]pyridin-2-yl)-9H-pyrido[3,4-b]indol-8-yl]benzonitrile 4-(1,3-dimethylpyrrolidin-2-yl)sulfanylbenzaldehyde 1-(2,4-dichlorophenyl)-5-methyl-N-[3-[4-[2-oxo-2-[2-oxo-6-(trifluoromethoxy)spiro[1H-indene-3,4'-piperidine]-1'-yl]ethyl]piperazine-1-carbonyl]phenyl]-4-(trifluoromethyl)pyrazole-3-carboxamide 5-[7-(trifluoromethyl)dibenzofuran-3-yl]-2H-tetrazole 6-amino-1-(1,3-dioxoisoindol-2-yl)-4-ethynylhexan-2-one 4-(3,5-dimethoxyphenyl)-1,1-bis[2-(dimethylamino)ethyl]piperidine-3,6-diol N-[4-[5-[3-chloro-4-(3,3-dimethylbutyl)phenyl]triazol-1-yl]but-2-ynyl]benzamide 4-[[5-chloro-2,3-dihydropyridin-6-yl-(3-methoxyphenyl)carbamoyl]amino]benzamide 3-(1H-imidazole-5-carbonylamino)-4-[4-(3-methylphenyl)piperazin-1-yl]benzoic acid;2,2,2-trifluoroacetic acid 6-(4-aminocyclohexyl)-N-ethylpyrimidin-4-amine;dihydrochloride N-[2-(4-bromophenyl)-5,6,7,8-tetrahydrothieno[3,2-b]azepin-3-yl]-4-methoxypyridine-2-carboxamide 2-ethyl-3,4-dimethoxybenzoic acid N-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]imidazo[1,2-a]pyridine-6-carboxamide [2-(dimethylamino)-5-fluorophenyl]urea 1-[(2,4-dichlorophenyl)methylamino]-3-[(3-fluorophenyl)methyl]urea [(1S)-3,4-dihydro-2H-chromen-1-yl]carbamic acid 1-(4,5-dichlorocyclohexa-2,4-dien-1-yl)sulfonyl-3-[7-[(4-methoxyphenyl)-(methylamino)methylidene]-6H-furo[2,3-b]pyrrol-4-yl]urea 4-[(2,6-dichlorobenzoyl)amino]naphthalene-1-sulfonic acid [1-(2,6-diphenylpyrimidine-4-carbonyl)pyrrolidin-3-yl]carbamic acid 1-cyclohexa-2,4-dien-1-yl-N-[(E)-N'-[4-(7-methoxyquinolin-4-yl)oxyphenyl]carbamimidoyl]-5-methylidenepyrrolidine-3-carboxamide 2-(4-methoxyphenoxy)-N-[(5R,7S)-5,7,9,10-tetrahydronaphtho[2,1-g][1]benzofuran-6-yl]acetamide 1-benzyl-2-(4-bromobutoxy)pyrazin-1-ium [(1R)-3,4-dimethylcyclopent-2-en-1-yl]sulfonylbenzene [(Z)-[6-iminocyclohexa-2,4-dien-1-ylidene]methyl]sulfonyl-triphenylphosphanium (E)-2-benzylsulfanyl-3-[[4-[5-chloro-1-methyl-6-oxo-2-[[(Z)-prop-1-enyl]amino]pyrimidin-4-yl]oxyphenyl]methylideneamino]but-2-enoic acid;ethane 5-[2-(difluoromethoxy)phenyl]-1H-pyrazole [5-(diethylamino)-2-[[3-methyl-1-oxo-4-(naphthalen-2-ylsulfonylamino)butan-2-ylidene]carbamoyl]phenyl]boronic acid 2-[N-(4-bromobutan-2-yl)-3-methylsulfanylanilino]benzenesulfonic acid [4-(2,6-dimethylphenyl)-2-phenylpyridin-3-yl]-trimethylsilane;iridium;8-methyl-5-pyridin-2-yl-7H-[1]benzofuro[2,3-b]pyridin-7-ide 1-(8H-cyclohepta[b]pyridin-2-ylamino)-4-methylpentan-3-one 3-(2-methyl-1,3-benzothiazol-6-yl)cyclopropane-1,1,2,2-tetracarbonitrile 4-bromo-N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]benzamide 4-N-(4-tert-butylphenyl)-6-N-phenylpyridine-2,3,6-triamine 2-(benzenesulfonyl)-4,5-dimethylthiophene 5-[1-cyclopentyl-6-(difluoromethoxy)benzimidazol-2-yl]-1,3-diethylbenzimidazol-2-one 2,2-dimethylbutane;3,5-dimethyl-2-[[1-[(1S)-2,2,2-trifluoro-1-phenylethyl]piperidine-4-carbonyl]amino]hexanoic acid 3-amino-4-cyano-5-[1-[2-(2,6-difluorophenoxy)ethyl]piperidin-4-yl]-1H-pyrrole-2-carboxamide 4-(1,5-dimethylpyrazol-3-yl)-N-[2-(2-ethoxy-1-hydroxycyclopentyl)ethynyl]benzamide 4-N-[5-(3,5-difluorophenyl)-1H-pyrazol-3-yl]-6-methoxypyrimidine-2,4-diamine [4-(1-methoxyethyl)triazol-1-yl]-(4-propan-2-ylphenyl)methanone 7,8-dimethoxy-1-(3-nitrosopropyl)cinnoline 3-azidosulfanylnaphthalene-2,7-dicarbonitrile 5-[3-(4-bromophenyl)thiophen-2-yl]thiophene-2-carboxylic acid N-azido-2,3-dihydroxynaphthalene-1-carboxamide 5-[(1S)-2,3-dihydro-1H-inden-1-yl]cyclohexa-1,5-dien-1-amine 3-[[2-(3-hydroxy-4,6-dimethylnaphthalen-1-yl)-5-methoxybenzimidazol-1-yl]methyl]benzamide 3-(7-propan-2-yl-1H-indol-4-yl)cyclobutane-1,2-dione 1-[4-[5-[(2,6-dioxopiperidin-3-yl)amino]pentanoyl]phenyl]-N,N-dimethylpyrrolidine-3-carboxamide N-[(Z)-1H-indol-3-ylmethylideneamino]-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide 2-[4-(hydroxymethyl)-5-nitropyridin-3-yl]-2,4-diazaspiro[4.5]decan-1-one 7-hydroxy-5,9-dimethyl-2-[(1E)-4-phenylbuta-1,3-dienyl]xanthen-3-one 1-[4-(7-aminoquinoxalin-5-yl)oxycyclohexyl]-3-pyrrolidin-3-ylurea N-[2,3-difluoro-4-[(3R)-3-[4-methyl-5-[[(3S)-pyrrolidin-3-yl]methoxy]pyridin-2-yl]pyrrolidine-1-carbonyl]phenyl]propane-2-sulfonamide 4-N-[5-(3,3a,4,8b-tetrahydro-1H-pyrrolo[2,3-c]quinolin-2-yl)pentan-2-yl]benzene-1,4-diamine 2-chloro-N-[(3-methoxypyrazin-2-yl)methyl]acetamide N-(4-bromobutan-2-yl)-N-(3,5-dimethoxyphenyl)naphthalen-2-amine 5-(2,3,4,5-tetrahydropyrido[4,3-b]indole-1-carbonyl)piperidin-2-one 3-(1H-indol-6-yl)-5-[4-methoxy-3-(trifluoromethyl)phenyl]imidazolidine-2,4-dione N-[4-(2,3-dihydrofuro[3,2-c]pyridin-5-ium-1-yl)phenyl]benzamide N-(3,4-dichlorophenyl)-5,6-dihydroquinazoline-2-carboxamide 2-(5,6,7,8-tetrahydronaphthalen-1-yl)benzoic acid 2-[3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-4-carbonyl)azetidin-1-yl]benzonitrile N-[4-amino-3-(1,2-dihydropyridine-5-carboximidoyl)phenyl]-4,4,4-trifluorobutanethioamide 4-[4-(N,2-dimethylanilino)butyl]cyclohexan-1-amine (4Z)-3,6-dimethylhepta-1,4,6-triene;ethane;2-hydroxyacetaldehyde;(Z)-1-phenyl-N-prop-2-enylbutan-1-imine N-methylsulfonyl-1,3,4,5,7,8,9,10-octahydrocyclohepta[b]indole-2-carboxamide 1-methoxy-3,7-diphenylheptacyclo[d]imidazole N-[(Z)-3-(methylideneamino)pent-2-en-4-ynyl]-2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-6-ylsulfanylamino)acetamide [[2-chloro-4-(propylcarbamoyl)phenyl]-hydroxymethylidene]azanium 4-[5-(2,3-difluorophenyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]cyclohexane-1-carboxylic acid (7R)-3-[(4-chlorophenyl)carbamoyl]-5-oxo-N-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide 6-cyclopropyl-1'-[(4-methoxyphenyl)methyl]spiro[5,7-dihydropyrazolo[3,4-b]pyridine-4,3'-azetidine] 2-[5-amino-6-[5-(methylamino)-1,3,4-thiadiazol-2-yl]pyrazin-2-yl]oxyethanol N-[5-(1,2-dihydroxyethyl)-3-fluoropyridin-2-yl]sulfonyl-1H-pyrrole-3-carboxamide (1-amino-2,2,6,6-tetramethylpiperidin-4-yl)oxycarbonyl-[[5-[4-[4-(dimethylcarbamoylamino)phenoxy]phenyl]-3-propan-2-ylpyrazol-1-yl]methyl]azanium 2-[(7S)-7-amino-8-oxodecanoyl]benzoic acid 1-[2,6-di(propan-2-yl)phenyl]-3-(oxolan-2-ylmethylsulfonyl)urea (2R)-1-[5-chloro-6-methyl-8-(3,4,5-trifluorophenyl)imidazo[1,2-a]pyridine-7-carbonyl]pyrrolidine-2-carboxamide 3-[4-(2,6-diphenylpyrimidin-4-yl)phenyl]-5-(trifluoromethyl)benzonitrile 2-(dichloromethyl)-6-(3,5-difluorophenyl)imidazo[2,1-b][1,3]thiazole N-[3-[3,5-bis(trifluoromethyl)phenyl]sulfonylpyridin-4-yl]acetamide N-[2-(diethylamino)pyridin-3-yl]-4-methoxypyrrolidine-2-carboxamide;hydrochloride (5Z)-5-[1-ethyl-4,5-dimethoxy-3-(trifluoromethyl)pyrazol-2-ium]iminopentanal 5-[4-(4-ethylphenyl)cyclohexyl]pentanoic acid N-(4-chlorophenyl)-5-methyl-2-[2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl]pyrazole-3-carboxamide 3-[2,6-dimethyl-4-(trifluoromethyl)phenyl]-7-[4-fluoro-2-(propoxymethyl)pyrrolidine-1-carbonyl]-9H-fluorene-2-carboxamide 3-[[(5Z)-5-benzylidene-4-oxo-2-phenyliminoimidazolidin-1-yl]methyl]benzoic acid N-benzyl-2-[(3R,4S)-1-[[4-[(3-cyanophenyl)methoxy]phenyl]methyl]-4-methylpyrrolidin-3-yl]acetamide N-[3,5-dimethyl-1-[2-(3-oxocyclohexa-1,4-dien-1-yl)ethyl]pyrazol-4-yl]formamide;N-ethyl-4-fluoro-6-[4-(4-methylpiperazine-1-carbonyl)phenyl]pyrazolo[1,5-a]pyridine-3-carboxamide N-methyl-3-(2,6,11-trithia-1-azabicyclo[12.4.0]octadeca-2,7,9,14,16-pentaen-15-ylsulfanyl)propan-1-amine N-ethenyl-2,5-diphenylaniline 3-azido-1-propyl-2-(trifluoromethyl)-9H-fluorene 5-azido-3,4-difluorothiophene-2-carbonitrile 5-methoxy-4-(2,3,5-triethylimidazol-4-yl)pyrimidine 2-[2,3-bis(trifluoromethyl)phenyl]-1-benzofuran 2-(1,3-dioxoisoindol-4-yl)-N-[2-(4-fluorophenyl)-6-methoxyindazol-5-yl]acetamide 2-(aminomethyl)-4,6-dichlorophenol;1-[3-(cyclohexen-1-yloxy)propyl]-3-methylbenzene N-(1,3-benzodioxol-5-yl)-2-[4-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl)-5,6-difluoro-2-methoxyindol-1-yl]acetamide 1-[6-(4-propylcyclohexyl)oxynaphthalen-2-yl]ethanone [4-chloro-1-(oxetan-3-yl)pyrrolo[2,3-b]pyridin-5-yl]-(furan-3-yl)methanone N-azido-1H-indole-5-sulfonamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-methylidenepyrrolidine-2-carboxamide (6E)-5-amino-6-[(3,4-difluorophenyl)methylidene]cyclohexa-2,4-dien-1-one 2-[4-(3-methyl-1H-pyrrolo[2,3-b]pyridine-5-carbonyl)piperidin-1-yl]acetic acid 3-[5-(5-cyclohexyloxypyridin-3-yl)-1H-indazol-3-yl]-N,N-dimethylaniline (2R)-N'-[(4-chlorophenyl)methyl]-3-(4-fluoro-1H-indol-3-yl)butanehydrazide N-[3-[6-[2,4-bis(trifluoromethyl)phenyl]-5-(trifluoromethyl)pyridin-2-yl]oxypropyl]butanamide 5-(5,8-dimethylimidazo[1,2-a]pyridine-6-carbonyl)-3-nitrobenzenesulfonamide 1-[5-amino-2-(6-aminohexan-3-yl)-6-methoxy-4,5-dihydropyrimidin-4-yl]indole-2-carbonitrile 1-[6-(1H-pyrazol-5-ylmethoxy)hexan-2-ylideneamino]piperidine-3,4-diamine 2-[[1-(hydroxymethyl)cyclopropyl]methoxy]benzonitrile (7R)-4,5,6,9-tetrahydroxy-10-(2-nitrophenyl)sulfanyloxy-8a,12a-dihydroindeno[1,2-b]fluorene-7,11-diol 3-fluoro-2,5-dimethyl-4-N-(2-methylpropyl)benzene-1,4-diamine 2-[5-[(4S)-3,3-difluoropiperidine-4-carbonyl]pyridin-2-yl]-N'-methanimidoylpyrrolo[1,2-a]pyrazine-1-carboximidamide (2-bromoacetyl)oxymethylbenzene;ethane 4-amino-2-chloro-5,6-dimethylpyridine-3-carboxylic acid N'-[5-[2,4-bis(trifluoromethyl)phenoxy]pyridin-3-yl]-1H-imidazo[4,5-b]pyridine-7-carboximidamide (2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-4-(2-ethoxyacetyl)-1-methylpyrrolidine-2-carboxamide 3-[(2R,4S)-2-methylpiperidin-4-yl]-5H-pyrrolo[2,1-f][1,2,4]triazin-4-one 1-(2,3-dichlorophenyl)sulfonylpiperidine-4-carboxylic acid 2-(3,4-dimethoxyphenyl)-5,6-dimethyl-3H-quinazolin-4-one [4-[(4-carboxy-3,5-dimethylpyrazol-1-yl)methyl]phenyl]-[4-hydroxy-4-(methoxymethyl)piperidine-1-carbonyl]azanium 3-(1,2,4-triazol-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine 4-amino-1,2-dihydroanthracene-9,10-diol (5R,7S)-N-[3-(1H-imidazol-2-yl)phenyl]-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide (3Z)-5-cyclopropyl-2,4,6-trimethylidenehepta-3,5-dienal;ethane;methanol;5-[1-(2-oxo-2-phenylmethoxyethyl)piperidine-4-carbonyl]pyrrolidin-2-one 2,4-dibromo-N-[(Z)-1-[5-chloro-2-hydroxy-3-methoxy-6-(2-nitroethoxy)phenyl]ethylideneamino]benzamide 3-fluoro-5-[2-[(4-fluoro-1,3-benzothiazol-2-yl)amino]pyrimidin-5-yl]benzamide 4-[2,3-dihydroxypropyl(1,3-thiazol-5-yl)amino]-N-pyridin-2-ylbenzenesulfonamide [3-(5-azidooxypyridin-2-yl)phenyl]methanamine 4-(aminomethyl)-6-(trifluoromethyl)quinazoline-7-carboxamide 3-ethylsulfanyl-6-methyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 5-[3-methylbutanoyl(prop-2-enyl)amino]naphthalene-2-sulfonic acid 4-[(1R)-6-fluoro-2,3-dihydro-1H-inden-1-yl]benzenesulfonamide 1-ethyl-2-[4-(oxan-4-ylamino)pyrimidin-5-yl]indole-6-carbonitrile 7-cyclopentyl-2-(cyclopropylamino)spiro[5H-pyrrolo[3,4-d]pyrimidine-6,3'-pyrrolidine]-2'-one 4-(1,3,3a,4,5,6,7,7a-octahydroisoindole-2-carbonyl)benzenesulfonamide 2-[4,6-bis(3,4-dihydroxyphenyl)pyridin-1-ium-2-yl]-N-diazoethanesulfonamide 2,5-dibromo-N-[[3-(difluoromethyl)-1H-1,2,4-triazol-5-yl]methyl]pyrimidine-4-carboxamide [(1R,3S)-1,2,3,4-tetrahydronaphthalen-1-yl]phosphonic acid 5-(1,4-diazepan-1-yl)-2-[[2-(3,4-difluorophenyl)imidazo[1,2-a]pyridin-7-yl]oxymethyl]-4-ethylaniline 2-[4,6-bis(4-chlorophenyl)-5-phenylpyrimidin-2-yl]phenol 2-[4-(2-azidopyrimidin-5-yl)phenyl]-N,N-dimethylethanamine 2-(4,4-difluoropiperidine-1-carbonyl)-3H-benzimidazole-5-carboxamide;hydrochloride 5-[2-(4-chlorophenyl)ethynyl]-3-methoxy-2H-isoquinolin-1-one 2-(4-bromophenyl)-5-chlorothiophene 4-[3,5-dimethyl-1-(2-methylpropoxycarbonyl)pyrrol-2-yl]benzoic acid 5-(4-oxo-3H-quinazoline-7-carbonyl)-1,4-dihydroquinoxaline-2,3-dione 6-amino-2-[(3,5-difluorophenyl)methylsulfanyl]-3H-quinazolin-4-one 2-[(5R)-7,10-dibromo-5-phenyl-1,4,7,9-tetrahydropyrazolo[3,4-b]acridin-6-yl]-4-methoxyphenol 2-hydroxy-5-methyl-N-[1-(3-methylphenyl)butan-2-yl]benzamide 4-benzylsulfanyl-3-methoxybenzoic acid 4-azido-3,6-dichloropyridine-2-carbonitrile 2-[3-(4-butylphenyl)-5-[5-[[4-cyclohexyloxycarbonyloxy-1-[methyl(propanoyl)amino]cyclopentanecarbonyl]amino]pyridin-2-yl]-6-fluoro-9H-carbazol-4-yl]acetic acid [7-benzylsulfonyl-5-(1,3-thiazol-2-ylmethyl)pyrrolo[2,3-d]pyrimidin-4-yl]hydrazine N-[(3S,4R)-1-cyclopentyl-4-(pyridine-2-carbonylamino)pyrrolidin-3-yl]oxane-4-carboxamide;hydrochloride [(4-chlorophenyl)-diethoxyphosphorylmethyl]phosphane (2S)-4-[3-[(3,5-dichloropyridin-2-yl)sulfanylmethoxy]phenyl]sulfonyl-N-hydroxyoxane-2-carboxamide N-[6-[3-(4-ethylpiperidine-1-carbonyl)phenyl]imidazo[1,2-a]pyridin-2-yl]cyclopropanecarboxamide;2,2,2-trifluoroacetic acid 5-[(2,3-difluorophenyl)methyl]-N-[1-[(2S)-1-ethoxypropan-2-yl]pyrrolo[2,3-b]pyridin-4-yl]-6-oxo-1H-pyrimidine-4-carboxamide (1S)-2,3,4,5-tetrafluoro-1H-indene 5-[(3E)-2,6-dimethylhepta-1,3,5-trien-4-yl]pyrimidine 1-(2,4,6-trimethylphenyl)sulfonylpyrrole 2-amino-1-[4-(3-phenylpropanoyl)piperazin-1-yl]ethanone 2-[4-chlorobutyl(hexyl)amino]benzoic acid N-cyclohexyl-3,4-difluoro-5-nitrobenzamide 2-(3,4-difluorophenyl)-3-methyl-6,7-bis[2-(pyridin-2-ylamino)ethoxy]quinazolin-4-one 4-azido-6,7-dihydro-5H-cyclopenta[b]pyridine-2-carboxylate N-[[1-(2,6-dioxopiperidin-3-yl)-5-methoxy-3-methylidene-2H-isoindol-4-yl]iminomethyl]-2-fluorobenzenecarboximidate [1-(2,4-dichlorophenyl)sulfonylpyrrolidine-3-carbonyl]azanide 3-[(2R)-1-aminopropan-2-yl]-N,5-dimethylaniline 2-[3-fluoro-4-[(2R)-2,3,5,6-tetrahydroindole-1-carbonyl]phenyl]-8H-pyrido[2,3-d]pyrimidin-7-one 2-[1,2-difluoro-2-(4-methylcyclohexen-1-yl)ethenoxy]-7-fluoroquinoline (2E)-6,11b-dihydrobenzimidazolo[1,2-c]quinazoline [4-[[(5,6,7-trimethoxyquinazolin-4-yl)amino]methyl]phenyl]cyanamide 3-(2,5-dimethylphenyl)-N-methyl-1-[4-(4-methylpiperazine-1-carbonyl)-1H-benzimidazol-2-yl]piperidine-4-carboxamide N-[(4S)-2,3,4-trimethylheptan-5-yl]pyrido[2,3-b]pyrazin-6-amine (3S)-1,2,3-trimethyl-6-[(E)-prop-1-enyl]-3a,4-dihydrothieno[3,2-b]pyrrole (4-benzylpiperidin-1-yl)-[4-[(Z,1Z)-1-aminopenta-1,3-dienyl]phenyl]methanone 5-[4-(aminomethyl)phenyl]-2-hydroxybenzene-1,3-dicarboxamide 4-(benzenesulfonyl)-6-hydroxycyclohexa-1,3-diene-1-carboxylic acid 1-(5-bromothiophen-2-yl)sulfonyl-3,4-dihydro-2H-quinoline 1-[4-(5-fluoropyridin-2-yl)piperazin-1-yl]prop-2-en-1-one (3R)-N'-[4,5-bis(ethenyl)pyridin-2-yl]-N-ethyl-1-[2-methoxy-5-(2-oxobutylsulfanyl)phenyl]pyrrolidine-3-carboximidamide 2-(4-cyanophenyl)-N,6-dimethylpyridine-3-carboxamide 6-[1-(2,3-dichlorophenyl)ethyl]-5H-pyrrolo[3,4-b]pyridin-7-one;propane 4-chloro-N-[(2R)-3-[4-[1-(ethylaminomethyl)cyclopropanecarbonyl]piperidin-1-yl]-1-oxo-1-phenylbutan-2-yl]benzamide 5-(3,4-difluorophenyl)-2-[1-[3-fluoro-4-(trifluoromethoxy)phenyl]pyrrolidin-2-yl]-N'-hydroxy-1H-imidazole-4-carboximidamide 2-[3,5-dichloro-4-(1-methylsulfonylpiperidine-4-carbonyl)phenyl]-6-(4-ethoxycyclohexyl)oxyphthalazin-1-one 2-ethyl-N-(4-methoxyphenyl)-6,7-dimethylthieno[3,2-d]pyrimidin-4-amine 2,3-dichloro-4H-1,8-naphthyridine (Z)-2-cyano-3-[4-[(1,2-dichlorocyclohexa-2,4-dien-1-yl)methoxy]phenyl]prop-2-enamide 4-amino-6-[(3,5-ditert-butyl-2-hydroxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-(3,5-dimethoxyphenyl)sulfonyl-1-[2-fluoro-4-(trifluoromethylsulfanyl)phenyl]piperazine ethane;2-[(4-methylphenyl)sulfonylamino]-N,3-diphenylbutanamide 1-[7-(3,5-dimethyl-4-propanoylpiperazin-1-yl)-3-phenylimidazo[1,2-a]pyridin-2-yl]ethanone N-cyclopentyl-6-(1,2,4-triazol-1-yl)pyrimidine-4-carboxamide N-(3,5-dichlorophenyl)-4-ethoxy-6-methylpyrimidine-2-carboxamide 1,4-diethyl-2-(isocyanatomethyl)benzene 2-(methylamino)-1,3-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-9-one 2-[5-(4,6-diphenylpyrimidin-2-yl)pyridin-3-yl]pyrido[1,2-a]benzimidazole 2-[4-bromo-N-(3,5-dichlorophenyl)-2,5-dimethylanilino]acetic acid 1-[2,3-difluoro-4-(2-methylbutanoyl)phenyl]-N-propylethanesulfonamide 3-(4-chlorophenyl)-2-methyliminospiro[5,6-dihydrocyclopenta[d]pyrimidine-7,4'-piperidine]-1'-carboxylic acid 3-fluoro-4-[(3-oxopiperidine-1-carbonyl)amino]benzoic acid [4-(2,3-dihydropyrrolo[1,2-a]pyridin-7-ylamino)sulfanylphenyl]methanol 6-[(6-aminopyridine-3-carbonyl)amino]hexyl-trimethylazanium N-[4-amino-3-(2,5-difluorobenzenecarboximidoyl)phenyl]-1-methylpyrazole-4-carboxamide;formaldehyde 3-(4,7-dihydroxy-2-oxochromene-6-carbonyl)benzenesulfonamide (3Z)-4-[(2R,5S)-5-[1-(benzenesulfonyl)ethenyl]oxolan-2-yl]buta-1,3-dien-2-amine 4-[5-chloro-6-(2,6-difluorophenyl)pyridin-3-yl]butanal 2-(4-cyclopropylphenyl)-N,5-dimethyl-6H-1,3,4-thiadiazin-3-ium-2-amine N-(6-methylpyridin-2-yl)spiro[5,7-dihydropyrrolo[1,2-a]imidazole-6,4'-piperidine]-1'-carboxamide ethane;2-(3-methoxypropylsulfanylamino)-4-phenylbenzonitrile 2-(1H-indazol-5-yl)-N-methylethanamine;7-[4-(2-morpholin-4-ylethoxy)phenyl]-2,3-dihydrothieno[3,4-b][1,4]oxazepine 4-(3,5-dimethylanilino)quinazoline-2-carboxylic acid 4-[2,3-bis(ethenyl)cyclopenta-1,4-dien-1-yl]-2-(4,5-dihydrobenzo[e]indol-1-id-2-yl)pyridine;cobalt(2+) 3-[7,8-dimethoxy-2-oxo-3-(oxolan-3-yl)chromen-5-yl]oxypropanenitrile N-(3,4,5-trimethyl-1H-pyrrol-2-yl)dodecanamide (2Z)-1,3-diamino-N-[2-(4-cyanophenyl)ethyl]-2-hydroxyiminopentanamide N-[(1R)-1-(3,4-dichlorophenyl)propyl]azetidine-2-carboxamide 5-[[2,6-difluoro-4-(trifluoromethyl)phenyl]carbamoylamino]pyridine-3-carboxylic acid 4-[(1Z)-buta-1,3-dienyl]sulfanyl-N-(5,6-dihydroisoquinolin-7-yl)benzamide 2-(4-chlorophenyl)-N-[4-fluoro-3-(pyrrolidine-1-carbonyl)phenyl]acetamide N-(1,5-dimethylpyrazol-3-yl)sulfanyl-2-[2-(trifluoromethyl)phenyl]quinazolin-4-amine 2-ethylsulfonyl-6-methylquinoxaline 4-[[[2-(2-aminoethyl)phenyl]-hydroxymethyl]amino]butanoic acid (7R)-7,8-dimethyl-5,11-dihydrochromeno[2,3-c]chromene 2,5-dichloro-4-[[(2S)-3-hydroxy-1-oxo-2-phenyl-1-benzothiophen-6-yl]methylideneamino]benzenesulfonamide N-(3,4-dichloro-2-methylphenyl)-5-piperidin-1-ylsulfonylpyrimidine-2-carboxamide 4-[5-chloro-3-methyl-2-(naphthalene-1-carbonylamino)phenyl]-7-hydroxy-3-methylquinoline-6-carboxylic acid 1-[5-(2-hydroxyethyl)-4,6,12b-trimethoxy-9-methyl-2,3,4a,10b-tetrahydro-1H-benzo[h][7]naphthyridin-8-yl]ethanone 1-(2,3-dimethylphenyl)-5H-pyrazolo[4,3-c]quinolin-8-one (2-azidophenyl)-(4-cyclohexylpiperazin-1-yl)methanone (2R)-N-[4-amino-3,4-dioxo-1-phenylbutan-2-yl]-4-(1H-pyrazol-5-ylmethylidene)pyrrolidine-2-carboxamide 2-[2-(1H-indol-6-yl)ethynyl]benzoic acid (5S)-2-[(Z)-1,3-benzothiazol-6-ylmethylidenehydrazinylidene]-5-ethyl-N,N-dipropyl-1,3-thiazinane-4-carboxamide 3-[2-(1H-benzimidazol-2-yl)acetyl]-N,N-bis[(4-methoxyphenyl)methyl]pyrrolidine-1-carboxamide N-[[5-(2,4-dihydroxyphenyl)-1H-pyrazol-4-yl]methylideneamino]benzamide 2-[(3-methylphenyl)sulfanylmethyl]azetidine 1-[(4-aminophenyl)methyl]naphthalene-2,7-diamine;N-[4-(2,3,5-trihydroxyphenyl)pyridin-2-yl]formamide 4-(2,3-dihydropyrrolo[2,3-c]pyridin-1-ylmethyl)-2-phenyl-1,3-thiazole;2-[3-ethoxy-5-(2-methylpropyl)pyridin-2-yl]-N-methylbutanamide 4-[6,8-bis(3-bromophenyl)-7H-purin-2-yl]morpholine 5-chloro-N-[2-(4-cyclopentyloxyanilino)pyrimidin-5-yl]thiophene-2-sulfinamide 2-[(5S)-3-chloro-4,7-dioxo-1,2,3,6,8,9-hexahydropyridazino[1,2-a]diazepin-10-yl]-N-[1-(4-fluorophenyl)cyclopropyl]acetamide 1-[6,7-dimethyl-2-(trifluoromethyl)-2H-chromen-3-yl]ethanimine 5-[[(5,6-dimethyl-2-oxopyridine-3-carbonyl)amino]carbamoyl]thiophene-2-carboxylic acid 2-[4-(5-cyano-6-oxo-1H-pyrimidin-4-yl)piperazin-1-yl]butanoic acid (E)-3-[2,4-dihydroxy-6-(hydroxymethyl)phenyl]prop-2-enal 5-[2-(6,7-dimethoxyquinolin-4-yl)ethynyl]-N,N-dimethylpyridine-3-carboxamide 2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-N'-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)butanehydrazide (2R)-1,5-bis(4-fluorophenyl)pentan-3-one 4-[2-[3,5-dichloro-4-(hydroxymethyl)phenyl]ethylsulfonyl]benzonitrile N-[3-(5,6-diethylthieno[2,3-d]pyrimidine-4-carbonyl)phenyl]propanamide [4-(5-methoxypyridin-3-yl)piperazin-1-yl]-(2,3,6-trimethoxyphenyl)methanone 1-[(2S)-6-fluoro-3,4-dihydro-2H-chromen-2-yl]propan-2-one [3-[(1Z)-buta-1,3-dienyl]iminopentan-2-ylideneamino]sulfanium;2,2,2-trifluoroacetate (3-fluoroazetidin-1-yl)-[2-[6-methoxy-5-(4-propan-2-ylimidazol-1-yl)pyridin-2-yl]quinolin-7-yl]methanone 2,3-dimethyl-8,9,10,11-tetrahydro-6H-pyrazolo[4,3-a]phenanthridine 2-[4-(1,4-dioxan-2-yl)phenyl]-5,6-difluoro-1H-benzimidazole;methanol 1-(4-azido-2,3-dimethylphenyl)piperidine 3-(2-chlorophenyl)-5-(4-cyclopropylpiperazin-1-yl)imidazo[1,2-a]pyridine;ethane (2R)-1,4-dibenzyl-5,7-diazatricyclo[6.3.0.02,6]undeca-8,10-diene (3R,4R)-1-cyclohexyl-N-[2-hydroxy-2-(1H-indol-3-yl)ethyl]-4-(trifluoromethyl)pyrrolidine-3-carboxamide 3-(azidomethyl)-2,6-dichloroquinoline 4-bromo-2,5-dimethyl-N-[3-(trifluoromethoxy)phenyl]pyrazole-3-carboxamide [1-(7,8-dihydronaphthalene-2-carbonyl)pyrrolidin-3-yl]azanide 1-(1H-indol-2-yl)-3,7-dimethylnonan-5-one 4-[[[5-cyclopropyl-2-(3-fluorophenyl)pyrazole-3-carbonyl]amino]methyl]benzoic acid 1-amino-2-azido-3H-fluorene 5-(4-aminophenyl)benzene-1,3-diamine 3-[(Z)-1-methoxyprop-1-enyl]-N'-(6-morpholin-4-ylpyridin-2-yl)benzenecarboximidamide 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;8-chloro-3-ethyl-2-phenylisoquinolin-1-one 2,7-dihydroxy-5-[(E)-2-phenylethenyl]-4H-pyrido[3,2-b]indole-1,3-dione;hydrochloride 6-(1,3-benzothiazol-2-ylamino)pyridine-3-carboxylic acid [3-[1-(benzenesulfonyl)indol-5-yl]-2,3-dihydroimidazo[4,5-c]pyridin-6-ium-5-ylidene]-(3-chlorophenyl)methanol 2-[3-(1-ethylpiperidin-4-yl)propanoyl]-N,N-dimethylpyridine-4-carboxamide 3-amino-5-[2-methoxy-4-(oxan-4-ylmethoxy)phenyl]pent-1-en-2-ol 4-(2-methylpropoxy)-N-[(Z)-1H-pyrazol-5-ylmethylideneamino]benzamide 4-[5-(1,3-benzoxazol-2-yl)pyridin-2-yl]piperidine-4-carboxylic acid N-[4-methyl-1-[3-(2H-pyridine-1-carboximidoyl)phenyl]pentylidene]hydroxylamine 2-(5,7-dihydro-4H-thieno[3,2-c]pyridin-6-yl)cyclopropan-1-amine 2-chloro-N-[6-(4-methoxybutoxy)pyridazin-3-yl]acetamide 5-chloro-2,4-dideuterio-N-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]benzamide ethane;N-(1,3-thiazol-2-yl)benzamide 1-[2,6-di(propan-2-yl)phenyl]sulfonyl-5-methoxyindazole 6-(3,5-dimethylphenyl)-2H-[1,3]thiazolo[4,5-b]pyridine 2-(6-chlorohexyl)naphthalene 4-[(2R)-1-[3-(1H-imidazol-5-yl)propanoyl]pyrrolidin-2-yl]-2-methyl-1H-pyrimidin-6-one (2R)-N'-hydroxy-2-[4-methyl-1-(pyridine-4-carbonyl)piperazin-2-yl]pyrrolidine-1-carboximidamide N-[(2E,4Z)-5-aminopenta-2,4-dienyl]quinoline-8-carboxamide N-azido-5-chloro-6,7-difluoro-2H-indazole-3-carboxamide N'-[4-(cyclohexylamino)sulfanylphenyl]-2,5-dimethoxybenzenecarboximidamide 3-(2,4-dichlorophenyl)-5-[[2-(3-methoxypropylsulfanylamino)-1,3-benzothiazol-6-yl]oxymethyl]-1-[(4-methoxyphenyl)methyl]pyrazole-4-carbonitrile 6-(cyclopentylmethylamino)-N'-hydroxypyrazine-2-carboximidamide 4-(4-fluorophenyl)-2,3-dimethyl-1-phenylpyrrolo[2,3-b]pyridine (3S)-1'-benzyl-7-methylspiro[1H-indole-3,4'-5,7-dihydropyrazolo[3,4-b]pyridine]-2,6'-dione N-(3,5-dimethylphenyl)sulfanyl-1-[(6-fluoropyridin-2-yl)-hydroxymethoxy]propan-2-amine 1-cyclohexyl-3,4-dimethoxybenzene;N-(5,6,7,8-tetrahydronaphthalen-2-yl)formamide 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;5-(4-oxocyclohexen-1-yl)-N-propan-2-yl-3H-isoindole-1-carboxamide 4-[3-(4-chlorophenoxy)phenyl]-6,7-dimethoxyquinazoline 5-cyclopropyloxypyridine-3-carboxamide 2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N'-hydrazinyl-6-propan-2-yloxybenzenecarboximidamide N-(1,3-benzothiazol-2-yl)-4-[[3-(5-chloropyridin-2-yl)-4-hydroxyphenyl]methylideneamino]benzamide N-[4-[2-amino-3-methyl-5-(1,2,3,6-tetrahydropyridin-4-yl)phenyl]-4-oxobutyl]-5-(3-fluorophenyl)furan-2-carboxamide 3-[4-(furan-2-yl)cyclohexa-1,5-dien-1-yl]oxy-N,N-dimethylpropan-1-amine N-[2-(4-azidophenyl)ethyl]-3,3-dimethoxycyclobutan-1-amine N-[(3S)-9-[2-cyclopropyl-6-(trifluoromethoxy)benzoyl]-1,9-diazaspiro[4.5]decan-3-yl]pyridine-3-carboxamide (6E)-5-hydroxy-4,8-dihydro-3H-oxocino[3,2-b]pyridine-9-carboxamide (1S)-2,2,2-trichloro-N-[3-[5-(difluoromethyl)furan-2-yl]propyl]cyclohexan-1-amine 2-[1,3-dihydroxy-5,6-di(propan-2-yl)inden-2-yl]acetic acid 2-[3,5-bis(trifluoromethyl)phenyl]-1,3-dioxolane-4-carboxylic acid 5-[(4S,9aR)-8-(2-methylbutan-2-yl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine-2-carbonyl]thiophene-2-carbonitrile;formic acid 3-[[4-[2-(1,3-thiazol-2-ylamino)pyrimidin-5-yl]benzoyl]amino]propanoic acid N-(1H-imidazol-5-ylmethyl)-3-methoxy-2,2-dimethylpropanamide 3-[4-methoxycarbonyl-2,6-di(propan-2-yl)phenyl]oxirane-2,2-dicarbonitrile 6-ethyl-5-[2-[3-(1H-imidazol-5-yl)propoxy]phenyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine [3-[5-(6-methylpyrazin-2-yl)pyridin-2-yl]oxyphenyl]urea 3,4-dimethyl-1,2-benzothiazole;2,2-dimethoxypropane 2-[4-cyano-3,5-di(propan-2-yl)phenyl]acetamide 6-[2-(difluoromethoxy)phenyl]-3-[1-[4-(triazol-2-yl)phenyl]ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one 3-[(2E)-5-chlorohepta-2,4,6-trienyl]sulfanylprop-1-en-2-ol;N-[6-methylidene-7-phenyl-1-(4-pentylcyclohexyl)oct-1-yn-3-yl]cyclohexanecarboxamide 2-[(3-chlorophenoxy)methyl]-7-(cyclobutanecarbonyl)-N,N-diethyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-4-carboxamide 3-[4-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]phenyl]-N,N-dihydroxybenzamide 7-ethyl-5,6-dimethoxynaphthalene-2,3-dione 2-[4-bromobutan-2-yl(1,3-thiazol-5-yl)amino]benzenesulfonic acid 7-chloro-5-(2,4-difluorophenyl)-1H-indazole (3S,5R)-1-[6-cyano-4-(dimethylamino)pyridine-2-carbonyl]-5-(hydroxymethyl)pyrrolidine-3-carboxylic acid 4-[2-(3,5-dibromopyridin-2-yl)ethenyl]-N-ethenylaniline 7-butyl-4H-1,2-benzoxazole 2-[4-[2-[8-(5-chlorothiophene-3-carbonyl)-1,8a-dihydroisoquinolin-3-yl]ethynyl]phenyl]-2-methylpropanenitrile;methanamine (E)-N,2-diamino-3-[4-[cyclopropyl(methylsulfonyl)amino]phenyl]prop-2-enamide 2-chloro-6-(1,3-dimethylpyrazol-4-yl)-7H-pyrrolo[3,4-d]pyrimidine 1-(4-azidophenoxy)-3,5-dichlorobenzene 5-[2-(3,4-dichlorophenoxy)phenyl]imidazolidine-2,4-dione 6-fluoro-N-[(E)-(5-methylpyridin-2-yl)methylideneamino]-1,3-benzothiazol-2-amine 3-[4-(2-methoxyethyl)piperazin-1-yl]quinoline 1-[4-(4-chlorophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylsulfonylethanone (3S)-1-(2,4-difluorophenyl)sulfonyl-N-[[3-(1H-indol-3-ylmethyl)oxolan-3-yl]methyl]pyrrolidin-3-amine 5-(4-cyclopropylphenyl)-1-methylpyridin-2-one 4-[2-(1-ethoxy-3,3,5,5-tetramethylhexan-2-yl)phenyl]phenol 4-bromo-3-(1,1-difluoroethoxy)benzaldehyde N'-[1,2,5-tris(ethenyl)imidazol-4-yl]ethanimidamide (3S)-N'-[(4-chlorophenyl)methyl]-2,5-dioxooxolane-3-carbohydrazide 3-[2,6-dichloro-4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]-2-oxoimidazolidine-1-carboxylic acid 1-[5-(1,3-benzodioxol-5-yl)pyridin-2-yl]ethanamine;dihydrochloride N'-[4-(3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-N-iodoethane-1,2-diamine N-[5-[2-(4-fluorophenyl)ethyl]pyridin-2-yl]-6,7-dihydro-4H-imidazo[1,5-a]pyrazine-5-carboxamide 5-amino-4-[3-(cyanomethoxy)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 1-[[4-(2,6-difluorophenyl)sulfonylcyclohexyl]methoxy]cyclobutane-1-carboxylic acid 4-[5-(hydroxymethyl)furan-2-yl]sulfanylcyclohexa-2,5-diene-1-carboxamide N-[(1S,2R)-2-hydroxy-4-(imidazol-1-ylmethyl)cyclopentyl]-3-methoxypyridine-2-carboxamide 2-(azetidin-1-ylmethyl)-5,8-dimethylpyrido[3,4-b]pyrazine 7-chloro-6-[3,4-dihydro-2H-chromen-7-yl(methoxy)methylidene]-1,3-diphenyl-5H-pyrazolo[3,4-d]pyrimidine-4-thione (4R)-4-[2,6-difluoro-4-(trifluoromethoxy)phenyl]-1-(oxetan-3-ylsulfonyl)piperidine N-[5-(2,3-difluoro-4-methoxyphenyl)pyridin-3-yl]acetamide 3-[6-(4-methylphenyl)-1,2,4,5-tetrazin-3-yl]phenol (5R)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[[3,5-dibromo-4-[(2S)-butan-2-yl]oxyphenyl]methylidene]-1,3-thiazolidin-4-one 5-bromo-N-[2-(1,3-dioxolan-2-yl)ethyl]furan-2-carboxamide [2-fluoro-4-(trifluoromethyl)phenyl]-[3-methoxyimino-5-[[5-(2,4,6-trichlorophenoxy)pyrimidin-1-ium-2-yl]amino]pentanoyl]azanide N-[(Z)-1H-indol-3-ylmethylideneamino]-2,6-dimethoxybenzamide (5S)-7-azido-4-[3,4-bis(phenylmethoxy)phenyl]-5-hydroxyheptanoic acid 1-[4-chloro-2-(methylamino)phenyl]pyrrolidine-3-sulfonamide (1-azidocyclopropyl)-[4-[2-[(3S,5R)-5-ethynylpyrrolidin-3-yl]oxyethoxy]-6-methoxypyridin-3-yl]methanone 1-methoxyiodanuidyl-2,3-dihydroindole N-[(3R)-piperidin-3-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide N-benzyl-2,5-dichloropyridine-3-carboxamide N-[2-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl]-2-pyrrolidin-1-ylacetamide 2-[3-(4,6-diphenylpyrimidin-1-ium-2-yl)phenyl]-5-methylpyrimidine (2S)-2-[4-chloro-3-methyl-5-(6H-benzo[b][1,4]benzoxazepine-5-carbonylamino)pyrazol-1-yl]butanoic acid 3-[3-amino-4-[amino(methyl)carbamoyl]phenyl]propanoic acid (5Z)-3-[2-(6-ethylpiperidin-1-ium-3-yl)oxyphenyl]-5-[[4-[(E)-2-hydroxy-2-iodoethenyl]phenyl]methylidene]-1,3-thiazolidine 1-[6-methyl-4-(2,3,3-trimethylpentan-2-yl)cyclohexa-1,5-dien-1-yl]naphthalene 2-(4-ethyl-2,3,5,6-tetrafluorophenyl)sulfanylacetaldehyde (6-chloro-1H-imidazo[4,5-b]pyridin-2-yl)-hydroxymethanesulfonic acid 2-bromo-N,3-dimethyl-4H-quinoline-7-carboxamide 1-ethyl-N-[2-(5-methoxy-1,3-benzothiazol-2-yl)ethyl]piperidine-4-carboxamide;2,2,2-trifluoroacetic acid 5-[4-(1,1,2-trimethoxyethyl)dodecan-3-yl]naphthalene-2-carboxylic acid 5-[2,4-diamino-6-[(3-fluoropyridin-2-yl)methoxy]pyrimidin-5-yl]-2-fluorobenzaldehyde [3-(4-methylphenyl)pyrazolo[1,5-a]pyrimidin-7-yl]thiourea 2-(4-chlorophenyl)imino-3-propyl-N-pyrimidin-5-ylhexanamide (5S)-N-[[6-(3,4-difluorophenyl)pyridin-2-yl]methyl]-1,8-dioxa-7-azaspiro[4.4]nonane-7-carboxamide 2-(4-chloro-3,5-dimethylphenoxy)-N-[(2S)-1,3-dihydroxypropan-2-yl]acetamide 2-[(1R)-2,2-dimethylcyclopentyl]oxycarbonylbenzoate 4-[(3R)-1-[2-[5-(4-tert-butylphenyl)thiophen-2-yl]acetyl]pyrrolidin-3-yl]-2H-triazole (5R,6S)-3-[1-cyclopentyl-2-hydroxy-5-[4-(oxetan-3-ylsulfonyl)phenyl]indol-3-yl]-6-methoxycarbonyl-3-azabicyclo[3.1.0]hexane-2-carboxylic acid (2R)-N-[5-bromo-3-fluoro-6-(triazol-2-yl)pyridin-2-yl]-3,3,3-trifluoro-2-hydroxy-2-methylpropanamide (1S)-2,4-ditert-butyl-3-oxo-5-phenylcyclohexane-1-carboxylic acid (4R)-N-[(1S,2R)-3,3-difluorocyclopentyl]-3-methoxy-1-oxo-2-phenyl-6,7,8,9-tetrahydroquinolizine-4-carboxamide 5-[(4,4-difluoropiperidin-1-yl)methyl]pyridine-2-carboxylic acid (2S)-2,3-diamino-N'-[1-[(4-methoxyphenyl)methyl]-6-oxopyrimidin-5-yl]propanimidamide (1E,4Z,6E)-8-[4-[5-(2-carboxypropylamino)naphthalen-2-yl]oxyphenyl]-7-hydroxyundeca-1,4,6,9-tetraen-3-one (2R)-N'-hydroxy-3-methyl-4,5-diphenylpyrrolidine-2-carboximidamide (2R)-N'-(3,4-dichlorophenyl)sulfanyl-2-hydroxy-3-[[methyl-[3-(trifluoromethyl)cyclohexyl]amino]methyl]butanediamide 3,4-dichloro-N-[2-(2-methylphenyl)ethyl]-1H-indole-6-sulfonamide (E)-2,3-diamino-3-[5-fluoro-6-methyl-4-oxo-1-(2,4,5-trifluorophenyl)pyridin-3-yl]sulfanylprop-2-enamide N-[4-amino-6,7-dimethyl-2-oxo-1-(1,3-thiazol-5-yl)quinoline-3-carboximidoyl]benzamide 5-[(4R)-4-amino-3,3,3-trifluoropyrrolidine-1-carbonyl]-2-methylbenzonitrile 2-[3,5-bis(trifluoromethyl)phenyl]-N-(3,4-dihydroxybutoxy)acetamide (2E,5Z)-2-[(3,4-difluorophenyl)methylidene]-5-[(4-methylphenyl)methylidene]oxolane 4-[4-(trifluoromethyl)phenyl]imino-2,3,5,6-tetrahydrobenzo[h]quinolin-1-one 4-[4-(hydroxymethyl)piperidine-1-carbonyl]benzoate [2-bromo-4,5-di(propan-2-yl)cyclohexa-1,3-dien-1-yl]-bis(3,5-dimethoxyphenyl)sulfanium 2-cyclopropyl-6-[(3,5-difluoropyridin-4-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-[[5,6-bis(ethenyl)pyridin-2-yl]amino]propan-1-ol (7R)-N-(4-chlorophenyl)-2-(2,6-dimethylpyridin-3-yl)-5-oxo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide 6,7-dimethoxy-4-[2-(3-nitrophenyl)ethylamino]quinoline-3-carbonitrile 3-[4-[2,6-di(propan-2-yl)phenyl]-1,2,4-triazol-3-yl]-5H-benzimidazol-5-ide;iridium 5-[4,5-bis(ethenyl)-6-methoxypyridin-2-yl]-1-N,3-N-dibutylbenzene-1,3-diamine;(Z)-3,3-dihydroxy-N'-propan-2-ylidenepent-4-enehydrazide N-[3-(dimethylamino)propyl]-5,6-bis(ethenyl)-2-phenylpyrimidine-4-carboxamide 2-(3,4-dichlorophenyl)-5-[[6-fluoro-1-(4-propan-2-yloxyphenyl)-2H-quinazolin-4-yl]amino]pentanenitrile (7S)-7-[4-ethoxy-3-(pyrazol-1-ylmethyl)phenyl]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one N-(5-fluoropyridin-3-yl)-2-[6-fluoro-4-oxo-1'-[(1S,3R)-3-phenylcyclohexanecarbonyl]spiro[3H-chromene-2,4'-piperidine]-7-yl]benzamide 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-naphthalen-2-ylamino]decanoic acid 2,4-diaminopyrimidine-5-carbonitrile;3-ethyl-8-(1-methoxyethyl)-2-phenylisoquinolin-1-one 5-tert-butyl-2,3,4-trifluoro-1H-pyrrole 1-[[3-(dimethylamino)phenyl]methyl]-4-(2,6-dimethylpyridin-4-yl)piperazine-2-carboxylic acid (7S)-N-(2,4-dimethoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 6-amino-7-[(2R)-3,4-dihydroxybutan-2-yl]oxy-3H-quinazolin-4-one 1-[5-(2,3-dihydro-1H-inden-4-yl)-6-hydroxy-1H-indazole-3-carbonyl]azetidine-3-carboxylic acid N-benzyl-6,7-dichlorospiro[1,4-dihydroquinoline-3,1'-cyclohexane]-2-imine 1-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]-3-quinolin-5-ylurea 1-(4-chlorophenyl)-2,3,5-trimethylbenzene;ethane (3Z)-3-[[5-chloro-2-[4-(trifluoromethylsulfonyloxy)anilino]pyridine-3-carbonyl]hydrazinylidene]azetane-1-carboxylic acid 2,4-dimethyl-N-(1-pyridin-3-ylpropan-2-yl)benzenesulfonamide 1-(2,4-dimethylpentanoyl)-N'-[1-[2-fluoro-6-(trifluoromethyl)phenyl]ethyl]spiro[5,6-dihydroimidazo[2,1-c][1,4]oxazine-8,3'-pyrrolidine]-2'-carbohydrazide 3-[[4-(benzenesulfinyl)phenyl]methyl]-5-phenylimidazolidine-2,4-dione N-[(Z)-3-amino-1,4,4,4-tetrafluorobut-2-enylidene]-1-methyl-5-[6-(trifluoromethoxy)-1H-benzimidazol-2-yl]pyrazole-4-carboxamide (2S)-4,7-dichloro-1-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-N-methyl-6-nitroheptan-2-amine 3-methyl-2,4,6-trioxo-N'-[(Z)-(3-phenyl-1H-indol-5-yl)methylideneamino]-1H-pyrimidine-5-carboximidamide N-(5,6,7,8-tetrahydronaphthalen-1-yl)pyrazine-2-carboxamide 1-[(3,5-difluorophenyl)methyl]-5-(2-phenylethynyl)cyclohexa-2,4-diene-1-carbonitrile 1-[2,6-dimethyl-4-(pyrrolidine-1-carbonyl)phenyl]sulfonylpiperazin-3-one N-[(2R,3S)-2-(1H-pyrazol-5-yl)oxan-3-yl]imidazo[1,2-b]pyridazine-6-carboxamide N-(3,5-dimethyl-1H-pyrazol-4-yl)-7H-purin-6-amine 2-[3-chloro-1,2-dihydropyridin-6-ylmethyl(methyl)amino]benzoic acid 4-[(7R)-5-methyl-7,8-dihydro-6H-pyrido[2,3-d]pyrimidin-7-yl]benzoic acid (2E)-N-[2-methyl-4-oxo-3-(6-pyrrolidin-1-ylpyridine-3-carboximidoyl)-1,5-dihydropyrido[2,3-e][1,4]diazepin-7-ylidene]butane-2-sulfonamide 5-(1,3-benzodioxol-5-yl)hexan-2-one 6-amino-2-methylsulfanylpyrimidine-4,5-dicarbonitrile (5S)-1-methyl-2-oxo-N'-[4-(trifluoromethylsulfanylamino)phenyl]pyrrolidine-3-carboximidamide 2-(5-ethoxybenzotriazol-2-yl)benzenesulfonic acid 5-(2-methylpropanoylamino)-4-oxo-3H-isoquinoline-1-carboxamide N-[3,4-bis(phenylmethoxy)phenyl]-4-(1-fluoroethenyl)-2-propanoylbenzamide N-[(2S)-3-methyl-1-oxo-1-(4-pyrimidin-5-ylphenyl)butan-2-yl]prop-2-enamide [2-chloro-4-(trifluoromethyl)phenyl]methanamine;hydrochloride 1-azido-3-(4,7-difluoro-2-methyl-1H-indol-5-yl)-N-methylpropan-2-amine 2,3-difluoro-4-[(E)-4,6,7,8-tetrafluorooct-5-enyl]phenol 7-(2,3-dihydropyridine-6-carbonyl)-N-ethyl-5,9,10,11-tetrahydroindolizino[1,2-h]quinoline-8-carboxamide 2-(2,6-dimethylphenyl)-7-[4-fluoro-3-[6-(hydroxymethyl)pyridin-2-yl]anilino]imidazo[1,2-a]pyridine-8-carboxamide (3R,5S)-7-benzoyl-N-[6-[[2-methoxyethyl(methylsulfonyl)amino]methyl]pyridin-2-yl]-1,4-oxazepane-3-carboxamide 2-azido-1,3-diethylanthracene 2-[[3,4-bis(cyclohexylamino)phenyl]methyl]benzamide (1-methylpiperidin-3-ylidene)-[2-phenylmethoxy-4-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]benzoyl]azanium 3-[2-(methylamino)ethyl]-2-methylsulfanylpyrazolo[1,5-a]pyridine-6-carbonitrile 1-benzyl-3,4-dimethoxypyrrole 2-[3-cyclopropyl-4-(methanesulfonamido)phenyl]propanamide N-[1-(4-fluorophenyl)ethenyl]-2,3-dihydro-1H-inden-5-amine;methane 2-[5-(2,4-dichlorophenyl)pyrimidin-2-yl]pyridine 2-[3-bromo-5-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-2-fluorophenyl]acetamide 3-methylsulfonyl-1-(6-phenylpyridin-2-yl)butan-2-one 1-methylsulfonyl-2-phenyl-3,4-dihydro-1H-isoquinoline 2-(4-tert-butylcyclohexyl)oxyphenol 1-(3,4-dihydro-2H-quinolin-1-yl)-2-imidazol-1-ylpropan-1-one 3-(5-chloropyridin-2-yl)-7-(7,7-difluoro-6H-1,4-oxazepin-5-yl)imidazo[1,2-a]pyrazin-8-one 5-[[4-(methylamino)benzoyl]amino]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 2-(4,6-dichloropyrimidin-5-yl)pyridine 2-(9H-fluoren-1-yl)-N,5-dimethoxyaniline 1-(4-azidophenyl)-2,3-dimethoxybenzene 4-[(6-methylpyridine-3-carbonyl)amino]piperidine-1,2-dicarboxylic acid (Z)-3-amino-1-[3-[2-[2,6-dichloro-4-(trifluoromethoxy)phenoxy]ethoxy]phenyl]prop-2-en-1-one 4-amino-5-hydroxy-1,6-bis(sulfanyl)naphthalene-2-carboxylic acid N-cyclopropyl-1-[4-(4-fluorobenzoyl)piperazin-1-yl]-2,3-dihydro-1H-indene-5-carboxamide 3-(4,5-dimethylpyrazol-1-yl)pyridine;ethane 2-amino-4,4-dimethoxy-6-(3-propoxyphenyl)-3-azabicyclo[3.1.0]hex-2-ene-1,5-dicarbonitrile 4-amino-6-[(3,5-dichlorophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-[azido(phenyl)methyl]benzenethiol 4-azido-1-(furan-2-yl)piperidine 3-[4-(1H-indol-5-yl)but-2-enyl]phenol 2-chloro-4-hydroxybenzo[e]benzimidazole-1-sulfonic acid 3-cyclohexyl-1H-indole 1,4-diphenylanthracene;ethane 2-amino-5-[3-(4-methoxyphenyl)propyl]-7-methylsulfinylpyrazolo[1,5-a]pyrimidine-3-carbonitrile 4-(1H-indole-2-carbonyl)-N-[2-(3,4,5-trimethoxyphenyl)ethyl]piperazine-1-carboxamide 4-azido-2-[6,8-bis(2-methoxyethyl)purin-9-yl]benzonitrile 1-bromo-2,3,4-trimethoxybenzene;ethane 2-(2-hydroxy-4-oxopyrido[1,2-a]pyrimidin-3-yl)-N-methylacetamide 5-azido-1,3-dichloroacridine 4-[(2E,3Z)-1,1,1,5,5,5-hexafluoro-2-(2,3,5-tribromophenyl)penta-2,3-dien-2-yl]phenol 6-[(4,5-difluoropyridin-2-yl)methoxy]-1-[2-(1H-pyrazol-5-yl)ethyl]-3,4-dihydroquinolin-2-one 2-(4,5-dichlorothiophene-2-carbonyl)-3,6-dihydro-2H-pyran-5-carboxylic acid 2-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-thiophen-2-yl-1,5-dihydropyrrolo[3,2-b]azepine 4-(2,2-dimethoxyethyl)-3-propan-2-ylidene-N-[(2S)-1,1,1-trifluoro-6-hydroxyhexan-2-yl]quinoxaline-2-carboxamide 2-fluoro-4-(3,7,11-trithia-8-azatricyclo[6.3.0.02,6]undeca-1(8),2(6),4,9-tetraen-10-yl)aniline (NZ)-N'-[1-[2,3-dihydro-1H-inden-5-yl-[4-(3,4-dimethoxyphenyl)butanoylamino]methylidene]-2-methylsulfonylpiperidin-4-ylidene]oxamide 2-(1,3,5-triazinan-2-ylidene)-6-(3H-thiophen-2-ylidene)-4,7-dihydro-3aH-imidazo[4,5-c]pyridine 1-[2-(3,5-difluorophenyl)ethylamino]-3-(4-nitrophenoxy)propan-2-ol;2,2,2-trifluoroacetic acid 5-[2,3-difluoro-4-(3-methylphenyl)phenyl]sulfanyl-N-propan-2-ylpyridine-3-carboxamide 2-[1-(4,7-difluoro-2-methylindazol-5-yl)sulfonylpiperidin-3-yl]-4-morpholin-4-yl-1H-pyrimidin-6-one 4-ethenyl-N-phenyl-1-[2-[(E)-3,3,3-trifluoroprop-1-enoxy]pyridin-4-yl]sulfonylpiperidine-4-carboxamide 4-(2,3-difluorophenyl)-1H-pyrazole;N-[3-(ethylaminomethyl)pentan-2-ylidene]-5-propan-2-ylthiophen-3-amine (2-azidoimidazo[1,2-a]pyridin-6-yl)-spiro[2H-indole-3,4'-piperidine]-1'-ylmethanone 4-[[[2,3-difluoro-4-[4-(4-methylcyclohexyl)phenyl]phenyl]-hydroxymethoxy]methylamino]phenol 2-(aminomethyl)-1-[4-[8-(6,8-difluoro-1-prop-2-enoyl-3,4-dihydro-2H-quinolin-7-yl)imidazo[1,2-a]pyridin-3-yl]phenyl]guanidine 6-[4-[3,5-dimethyl-1-(4-oxocyclohexanecarbonyl)piperidine-2-carbonyl]piperazin-1-yl]pyridine-3-carbonitrile 5-[2-(4-hydroxyphenyl)ethylamino]-3,7-dimethyl-1H-pyrido[2,3-d]pyrimidine-2,4-dione 3-[[6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]amino]piperidine-1-carboxamide N-(2,6-dioxopiperidin-3-yl)-1,3-thiazole-4-carboxamide (4S)-4-(2,5-dimethylpyrazole-3-carbonyl)-1-[(6-imidazol-1-ylpyridin-3-yl)methyl]pyrrolidin-2-one N-azido-1-[4-methoxy-3-(5,6,7,8-tetrahydronaphthalen-2-yl)phenyl]methanamine [3-(1H-indol-2-yl)phenyl]methanol 3-methylsulfonyl-N-[(1R,2S)-2-phenylcyclopropyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-6-carboxamide (2S)-1-[(3R,4S)-4-azidopiperidine-3-carbonyl]-N-cyclopropyl-4-hydroxy-3,5-dihydro-2H-1,4-benzodiazepine-8-sulfonamide 4-[2,3-dichloropropyl-(4-ethoxycarbonylphenyl)sulfonylamino]benzoic acid 4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)benzaldehyde N-[3,5-dichloro-4-(2-methylpyrazol-3-yl)phenyl]sulfonylformamide (1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)urea 4-ethoxy-2-N,5-di(propan-2-yl)benzene-1,2-diamine 3-[(3R)-6-chlorohexan-3-yl]-4-methoxybenzenesulfonic acid N-[4-(1,3,2-dioxaborolane-2-carbonyl)phenyl]acetamide N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-methoxy-6-methyl-N-octyl-1,3,5-triazin-2-amine N-[(3R)-8-fluoro-7-(hydroxymethyl)-4,5-dihydro-3H-2,6-benzodioxocin-10-yl]benzenesulfonamide 2-azido-4,5-dichloropyridine-3-carbonitrile N'-[(2S)-1-oxo-4-phenylbutan-2-yl]-2,3-dihydrofuran-5-carbohydrazide 2-[4-ethyl-5-oxo-2-phenylmethoxy-3,6-di(propan-2-yl)pyridin-1-ium-1-yl]-N-phenylacetamide;bromide 6-[2-(aminomethyl)-3-chlorophenoxy]-5-(cyclohexen-1-yl)-N-(2,4-difluorophenyl)pyridine-3-carboxamide N-[(2R)-1-hydroxy-3,4-dihydro-2H-naphthalen-2-yl]-3-pyridin-2-ylsulfanylpropanamide 3-[4-(4-aminopiperidine-1-carbonyl)anilino]-5-(quinolin-6-ylmethyl)imidazole-2,4-dione 4-methoxy-N-[2-(4-methylpiperidin-1-yl)ethyl]benzamide 7-[2,3-bis(4-fluorophenyl)quinoxalin-6-yl]-2,5,8-triazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-1(21),4,6,8,10,12,14,16,18-nonaene N-[2-[(2,4-dimethylphenyl)methyl]-5,6,7,8-tetrahydroquinolin-8-yl]-3-(trifluoromethoxy)benzamide 6-benzyl-5-[2,3-bis(ethenyl)phenyl]pyridin-2-amine N-[(3-chlorophenyl)methyl]-5,6-dioxo-4H-1,2,4-triazin-3-amine 4-[[5-tert-butyl-3-(3-pyridin-2-ylpropoxy)pyridin-2-yl]methylideneamino]pyridine-2,6-diamine 5-methyl-2,4-diphenyl-7H-pyrrolo[3,4-d]pyrimidine 6-[(1R)-1-aminoethyl]-5H-imidazo[1,2-a]pyridine-7-carboxylic acid N-[(Z)-1-amino-3-hydroxyprop-2-enylidene]-4-(azetidine-1-carbonyl)benzamide (3S)-6-azido-2-methyl-5-phenylmethoxycarbonylhexanoic acid N-[1-amino-3-(2,6-dichlorophenyl)propan-2-yl]-4-methoxybenzamide 2-(cyclopropylmethyl)-4-iodo-1H-pyrimidin-6-one N-(cyclohexylmethyl)-2-[[1-hydroxy-7-(3-hydroxyphenyl)heptan-2-yl]amino]acetamide 1-[4-(azidomethoxy)phenyl]sulfonylpiperidine 2-[6-(4,5-dihydro-1H-imidazol-2-yl)spiro[3.4]octan-7-yl]oxypyridine 4-[(E)-[7-cyclopropylimino-5-(3,4,5-trimethoxyanilino)pyrazolo[1,5-a]pyrimidin-3-ylidene]methyl]-5-hydroxy-1,2-dihydropyrazol-3-one 3-ethyl-5-[(4-phenylpyrazol-1-yl)methyl]-6,7-dihydro-4H-imidazo[2,1-c][1,4]oxazine 1-[2,3-difluoro-4-(4-propylcyclohexen-1-yl)phenyl]-6-ethoxy-7-fluoro-1,2,3,4-tetrahydronaphthalene 2-methyl-N'-(4-nitrobenzenecarbothioyl)propanehydrazide N-azido-3,4,5-trifluoro-2-hydroxybenzamide (3S)-4-[2-chloro-4-[[6-(cyclobutylcarbamoylamino)-8-fluoro-7-methoxyquinazolin-4-yl]amino]phenoxy]pyrrolidine-3-carboxamide 5-methoxy-2-[(1E,3E)-4-phenylbuta-1,3-dienyl]-3H-isoindol-1-one 2-[1-(4-bromophenyl)ethyl]-3-methoxy-6,7-dihydro-5H-pyrido[4,3-b]azepine (2S,5R)-4-hydroxy-7-(4-methoxyphenyl)-3-methyl-8-[3-(trifluoromethoxy)benzoyl]-2,4-dihydropyrrolo[1,2-a]pyrimidine-5-carboxylic acid 1-[(3S)-1-(4-chlorophenyl)pyrrolidin-3-yl]-3,5-dimethylimidazolidine-2,4-dione 2-[N-(4-hydroxybutyl)-3,5-dinitroanilino]ethanol N-[(3S)-9-chloro-2,3,5,6-tetrahydro-1H-1,4-benzodiazocin-3-yl]formamide 6-(2,3-dihydropyridine-4-carboximidoyl)-N,5-dimethylpyrimidin-4-amine 1-[(2R)-3,3-dimethylpentan-2-yl]-4-fluoro-5-(3-methoxypropoxy)isoquinoline 2-ethoxy-N-[5-(4-oxo-3H-quinazolin-2-yl)-1,3,4-thiadiazol-2-yl]acetamide 1-(2,3-dimethylimidazo[4,5-b]pyridin-7-yl)-3-ethanimidoylthiourea (4E)-4-ethenyl-1-ethylidene-6-methoxy-2,3-dihydrophenalene [1-(2-bromophenyl)cyclopropyl]methanol;ethane 5-(3,4-dimethoxyphenyl)-2-ethyl-1H-imidazole 4-[(Z)-6-ethylhept-5-en-2-yl]benzoic acid 2-amino-4-(1H-indol-3-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine-6-carbonitrile 2,4-dichloro-N-[2-(1H-indol-3-yl)ethyl]-N-pyridin-2-ylpyrimidin-5-amine N-[5-[(Z)-1-amino-3,3,4,4,4-pentafluorobut-1-enyl]-2-hydroxyphenyl]pyridine-2-carboxamide 2-(hydroxymethyl)-7,9-dihydropurine-8-carboxylic acid (E)-3-[4-[6-chloro-5-(trifluoromethyl)pyridine-2-carbonyl]oxyphenyl]prop-2-enoic acid 2-bromo-4-[4-chloro-3-(2,6-dioxopiperidin-3-yl)phenyl]butanoic acid N-[4-[3,5-bis(2,6-difluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl]cyclopropanesulfonamide 2-[1-azido-1,4-bis(2-methoxyethyl)piperazin-2-yl]acetonitrile 3-amino-2-[(2R,5S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-6-methyl-5H-pyrazolo[3,4-d]pyrimidin-4-one N-methyl-3-(2-methylanilino)sulfanyl-5,6,7,8-tetrahydronaphthalene-1-carboxamide 6-azido-N,1,4-trimethylindole-2-carboxamide N-methyl-1,8,9,10-tetrahydroanthracene-2-sulfonamide 3-[(2S)-1-azidopyrrolidin-2-yl]benzonitrile N-[2,4-dimethyl-3-(1-morpholin-4-ylethenyl)phenyl]-4-methoxynaphthalene-2-sulfonamide (E)-3-[4-[7-(ethylamino)heptylsulfonyl]phenyl]prop-2-enamide 3-ethenylsulfanyl-4-(2,4,6-trimethoxyphenyl)-1H-pyridazin-6-one (6Z)-6-[[3,5-dimethyl-4-[[(2S)-1-sulfanylpropan-2-yl]carbamoyloxymethyl]-1H-pyrrol-2-yl]methylidene]-N'-hydroxy-3-imino-2-oxopiperidine-4-carboximidamide 2-[[2-[2-methylpropanoyl-(2,4,6-trichlorophenyl)sulfonylamino]benzoyl]amino]acetic acid 2-[3,6-bis(4-methylphenyl)carbazol-9-yl]-5-isocyanobenzonitrile 7-chloro-4-[(5-methylpyrimidin-2-yl)amino]-3-propan-2-yl-1H-benzimidazol-2-one 1-[4-fluoro-2-(trifluoromethyl)phenyl]-N,N-dimethylbutan-1-amine 3-[[(1R,2S)-2-aminocyclohexyl]iminomethyl]benzene-1,2-diol 1-(3,5-dimethoxyphenyl)-4-[[2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenoxy]methyl]-7-propanoyloxyisoquinoline-6-carboxamide 3-bromo-N'-[(4,6-difluorocyclohexa-1,5-dien-1-yl)methylidene]-2-methoxybenzohydrazide 3-(2-tert-butyl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)benzaldehyde 4-(5-bromopyrimidin-2-yl)oxypiperidine-1-carboxylic acid 7-[(2R)-butan-2-yl]oxy-1,3-benzothiazol-6-amine N-[1-(4,5-dihydro-1H-imidazol-2-yl)butan-2-yl]-3,6-dimethylpyridazine-4-carboxamide 3-[4-chloro-2-fluoro-5-(3,4,5-trimethylpyrazol-1-yl)phenyl]imino-2-[1-[methoxy(propyl)amino]propan-2-ylideneamino]butan-2-ol N-(3-chlorophenyl)-2-[4-methyl-6-oxo-2-(1-phenylethylsulfanyl)-1H-pyrimidin-5-yl]acetamide 1-(2,4-difluorophenyl)sulfonyl-N-[(3S)-2,6-dioxopiperidin-3-yl]indole-5-carboxamide 4-[(3R)-3-(dimethylamino)pyrrolidine-1-carbonyl]benzonitrile;2,2,2-trifluoroacetic acid N-[1,6-bis(4-aminophenyl)hexyl]acetamide 5-methyl-4-(3,4,5-trifluorophenyl)oxane-2,6-dione 4-(2,4-dichlorophenyl)-N'-[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]thiadiazole-5-carboximidamide [3,5-bis(trifluoromethyl)phenyl]-[(2R,4S,7S)-4-hydroxy-3-oxatetracyclo[9.3.0.02,7.013,17]octadeca-1(11),12,14,16-pentaen-15-yl]methanone N-(5-bromopyridin-2-yl)-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]acetamide 2-(4,6-dichloro-3,5-dicyanopyridin-2-yl)sulfanyl-N-[2-fluoro-5-(trifluoromethoxy)phenyl]acetamide 4-[3-(3,5-dichlorophenoxy)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 4-(2-aminoethyl)-2,6-bis[3-(trifluoromethyl)phenyl]aniline [2-(azidomethyl)phenyl]-thiomorpholin-4-ylmethanone (E)-3-[2-cyclohexyl-4,6-dimethoxy-5-(2-pyridin-2-ylethynyl)phenyl]prop-2-enoic acid 2-amino-7-(4-methylsulfanyloxybutanoyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one (2Z,4E)-6-[5-fluoro-3-[2-(trifluoromethyl)phenyl]sulfinylpyridin-2-yl]oxy-2-[hydroxy(piperidin-1-yl)methylidene]-8-methylidenenona-4,7-dienoic acid 4-[4-(3,5-dichlorophenyl)-2-oxopyrrolidin-1-yl]piperidine-1-carboxylate 2-(5-bromo-4-methoxythiophene-3-carbonyl)cyclohexane-1,3-dione 2-[(1Z)-buta-1,3-dienyl]-N,6-dimethylpyridine-4-carboxamide;ethane 1-[4-(2-azidoethyl)phenyl]-3-benzylurea 3-[(2Z,4E)-1-aminohepta-2,4-dien-4-yl]oxypropan-1-ol;5-[4-(morpholine-4-carbonyl)phenyl]imidazolidine-2,4-dione 4-[2-(6,7-difluoroquinoxalin-5-yl)ethynyl]cyclohexan-1-amine N-[3-chloro-4-(1,2,4-triazol-1-yl)phenyl]-2-cyanopyridine-3-carboxamide 3-methyl-6,11-dihydrobenzo[b][1]benzazepine N-[(4R)-1-methyl-2-oxo-3,4-dihydroquinolin-6-yl]ethanesulfinamide 1-methyl-N-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carbonyl)phenyl]pyrazole-4-carboxamide [3-methoxy-4-(trifluoromethyl)phenyl]phosphane 4-(2,3-dihydro-1H-inden-5-yl)-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 1-[2,3-bis(2-methoxyethyl)phenyl]-N-methylethenamine N-[(2S)-3,3-dimethyl-1-oxobutan-2-yl]-1H-indazole-3-carboxamide 4-[[2-hydroxy-2,3-dihydro-1H-indene-5-carbonyl-[(1S)-1-phenylethyl]amino]methyl]benzoic acid [4-[3-aminopropyl(2,3-dihydropyrrolo[1,2-a]indole-1-carbonyl)amino]phenyl]sulfamic acid 2-amino-9-[(3R)-1-[4,5-bis(ethenyl)-3,6-dioxopiperazin-2-yl]piperidin-3-yl]-8H-purin-6-amine 4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-6-phenylpyridine-2-carboxylic acid 2-[5,6-bis(trichloromethyl)pyrazolo[3,4-d]pyrimidin-1-yl]ethanol N'-hydroxy-5,6-dimethyl-3H-indene-1-carboximidamide N-[(4-hydroxyphenyl)methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 1-[5-[6-chloro-7-(4-methylpiperazin-1-yl)quinazolin-2-yl]pyridin-2-yl]pyrrolidine-3,4-diol N-(6,7,8a,9-tetrahydro-6H-imidazo[4,5-a]indolizin-1-yl)formamide 2-(6,7-dimethylcyclohepta[b]pyrrol-1-yl)benzaldehyde 2-[(6S,7R)-4-azido-3-benzyl-8-oxo-5-thia-1,8-diazatricyclo[9.4.0.02,7]pentadeca-2(7),10,12,14-tetraen-12-yl]-N-(oxan-4-ylmethoxy)acetamide (2S)-2-[9H-fluoren-1-yl(phenylmethoxycarbonyl)amino]-3,6-dihydropyrrolo[2,3-h]quinoline-7-carboxylic acid 4-[(3S)-3-azidopyrrolidine-1-carbonyl]benzonitrile 1-[5-(4,4-difluoropiperidin-1-yl)-2H-triazolo[4,5-b]pyridin-3-yl]ethanone 7-[(1E,3Z)-2-[4-(1-cyclopentylpiperidine-4-carbonyl)piperazine-1-carbonyl]penta-1,3-dienyl]imidazo[1,2-a]pyridine-3-carboxylic acid N-(8-bromoquinoxalin-5-yl)-N-cyclohexa-1,3-dien-1-yl-4-nitrobenzamide (4R)-1'-[2,3-bis(methoxycarbonyl)benzoyl]spiro[6H-pyrrolo[3,4-b]pyrrole-5,4'-piperidine]-7-carboxylic acid 4-benzamido-2,6-dimethoxybenzoic acid 4-(2,5-dichlorophenyl)-1H-pyrimidine-6-thione 5-fluoro-N'-hydroxy-2-[methyl(oxan-4-yl)amino]pyridine-4-carboximidamide 1-azido-3,4-dihydro-2H-quinoline-7-carboxylic acid N-[1-[6-(cyclohexylmethoxy)pyridin-3-yl]ethylidene]hydroxylamine N-[4,5-difluoro-2-(3-phenylmethoxyphenyl)phenyl]formamide 2,3-dihydroxy-5-[2-(2-hydroxyphenyl)ethenyl]cyclohexa-2,4-dien-1-one 2-[4-[(Z)-2-cyano-2-[3,5-dichloro-4-[(6-methoxynaphthalen-2-yl)methoxy]phenyl]ethenyl]benzoyl]cyclopropane-1-carboxylic acid N-[2-(1,4-dimethylpiperidin-3-yl)ethyl]-4-(trifluoromethoxy)benzamide (3S,5R)-1-[6-(dimethylamino)pyrimidin-4-yl]-5-ethylpiperidine-3,4-diol 2-[4-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]phenyl]-3H-benzimidazole-5-carboximidamide 5-(4-aminophenyl)-N,2-dimethoxypyridine-3-carboxamide;ethane 4-azidooxy-6,7-dimethylnaphthalen-1-ol N-[(3R)-1,2,3,4-tetrahydroisoquinolin-3-yl]spiro[1H-2-benzofuran-3,3'-pyrrolidine]-1'-carboxamide N-[3-(4-methylpiperazin-1-yl)propyl]benzamide (2-aminophenyl)methyl-phenylazanide;N'-[4,5-ditert-butyl-3-(oxocarbamoyl)furan-2-yl]benzenecarboximidamide (Z)-3-amino-2-methylbut-1-en-1-ol;1,4-dimethoxybutane;ethene;1-ethyl-3-[1-(4-ethenylphenyl)ethyl]benzene (E)-2,5-diamino-N'-[2-chloro-4-fluoro-3-(2-hydroxyethylsulfanylmethyl)phenyl]hex-2-enimidamide 2-ethyliodanuidyl-N'-hydroxypyridine-4-carboximidamide 2-[4-(4-methoxyphenyl)-3,4-dihydropyridin-5-yl]-1H-indole 3-[3,5-bis(trifluoromethyl)phenyl]-1H-indazole 1-[4-(benzimidazol-1-yl)piperidine-1-carbonyl]cyclopropane-1-carbonitrile (2E)-N-[4-chloro-3-(trifluoromethyl)phenyl]-3,5-dinitrohepta-2,6-dienamide [(1Z,3E)-2-[1-[6-methoxy-5-(4-methylimidazol-1-yl)pyridin-2-yl]ethenylsulfanyl]penta-1,3-dienyl]carbamic acid 2-methylsulfinylethylphosphane;palladium(2+);triphenylphosphane;tetrafluoroborate N-[4,5-dimethyl-2-([1,3]thiazolo[5,4-c]pyridin-6-yloxy)phenyl]carbamate (5E)-2-(3-chlorophenyl)imino-5-[(4,7-dimethoxynaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one N-[(1,5-dimethyl-4-propan-2-ylpyrazol-3-yl)methyl]-6-morpholin-4-ylpyrimidin-4-amine N-[5-[3-(4-thiophen-2-yl-1H-imidazo[4,5-c]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]cyclopropanecarboxamide 2-(2-chlorophenyl)-4,6-dimethylpyrimidine 3-cyclobutyl-1-[4-[2-(trifluoromethoxy)phenyl]quinolin-7-yl]propan-1-one;ethane 4-tert-butyl-3,5-dichloro-N-(1,5-dimethylpyrazol-3-yl)benzamide 1-methyl-2,3-bis(phenylmethoxy)-4-propan-2-ylbenzene 6-[3,5-dimethyl-1-(2-pyrrolidin-1-ylethyl)pyrazol-4-yl]imino-5H-quinoline-2-carbonitrile N-azido-2,4,6-trichlorobenzohydrazide 2-[7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)naphthalen-2-yl]-4-[4-(10,12,20-triazapentacyclo[11.7.0.02,10.03,8.014,19]icosa-1(13),2(10),3(8),4,6,11,14(19),15,17-nonaen-13-yl)phenyl]quinazoline 4-[5-(difluoromethoxy)pyrimidine-2-carbonyl]-N,N'-bis[2-hydroxyethyl(methylsulfonyl)amino]piperazine-1-carboximidamide 1-(2,3-dihydro-1H-inden-5-yl)-N-[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyridin-2-yl]cyclobutane-1-carboxamide 5-(5-aminocyclohepta-1,4,6-trien-1-yl)sulfanyl-N-[(3E)-penta-1,3-dien-3-yl]thiophene-2-carboxamide N'-[(2E,4Z)-6-bromohepta-2,4,6-trien-3-yl]-2-propanimidoylbenzenecarboximidamide;ethane 2-(4-iodoanilino)-1-phenylethanone ethane;N-[3-[4-methoxy-7-(oxan-2-yloxy)quinolin-6-yl]prop-1-en-2-yl]-2-pyridin-2-ylacetamide 3-cyclopentyl-4-[(1-methylpiperidin-4-yl)amino]cyclobut-3-ene-1,2-dione N-[3,5-bis(trifluoromethyl)phenyl]-2-oxochromene-3-carboxamide 5-(2,4-dinitrophenoxy)carbonylbenzene-1,3-dicarboxylic acid [2-(7,8-dioxabicyclo[4.1.0]hepta-1(6),2,4-trien-3-ylmethylsulfanylamino)pyrimidin-5-yl]-[4-fluoro-3-(hydroxymethyl)phenyl]methanone 5-methyl-3-[[(E)-2-methylpent-1-enyl]sulfanyl-prop-1-en-2-ylamino]-N-[4-(trifluoromethyl)pyridin-2-yl]-1,2-thiazole-4-carboxamide 7-(5,6,7,8-tetrahydronaphthalene-1-carbonyl)-3H-quinazolin-4-one 2-[(3E)-6-bromohepta-1,3,5-trien-4-yl]-3H-benzimidazole 1-(4-fluorophenyl)-3-hydroxyimino-2-[3-(trifluoromethyl)phenyl]propan-1-one 3-[[1-(3,4-dichlorophenyl)cyclobutyl]amino]propanoic acid 2-[3-[2-(1,3-dihydroisoindole-2-carbonyl)phenyl]sulfanylprop-1-ynyl]benzonitrile 2-[6-[(3S)-3,4-dimethylpiperazin-1-yl]pyridazin-3-yl]acetonitrile N-cyclopropylsulfonyl-1,3-benzothiazole-6-carboxamide 2,6-dimethoxy-4-[(E)-[3-(5-nitrofuran-2-yl)propylidenehydrazinylidene]methyl]phenol 4-(3-aminopropyl)-2-bromophenol;dihydrochloride 1,4-bis(furan-2-ylmethylideneamino)guanidine 1-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butan-2-one 6-(2,4,4-trimethylpentan-2-yl)quinoline 5-amino-6-[(2R)-2,3-dihydroxypropoxy]-N-[(1R,2S)-2-methylcyclopentyl]pyridine-3-carboxamide (E)-3-[1,2-diamino-6-(3,4-dichlorophenyl)-7H-purin-8-yl]prop-2-enoic acid 3-[(3S,4R)-1-[2-methyl-6-(trifluoromethoxy)pyridine-4-carbonyl]piperidin-4-yl]-5-phenylimidazol-4-ol 1-(2,4-dimethylphenyl)-2-fluoro-3,5-bis[(Z)-prop-1-enoxy]benzene 3-[4-(pyridine-2-carbonyl)piperazin-1-yl]propanamide N-[(3R)-1-[4-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]phenyl]pyrrolidin-3-yl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 7-(2,4-dichlorophenyl)-12-methyl-3-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]imidazo[1,5-f]phenanthridine 1-methylsulfanyl-2-(3,3,4,5,5-pentafluoro-1-benzothiophen-2-ylidene)hydrazine [1-(2,4-dichlorophenyl)sulfonylcyclopentyl]methanol 4-[3-fluoro-2-(2H-tetrazol-5-yl)phenoxy]aniline 3-fluoro-4-(5-methylsulfanyl-2,4-dioxoimidazolidin-1-yl)benzenecarboximidamide 4-(1,2,3,5,6,7-hexahydropyrrolizin-8-yloxy)butanoic acid 2-[3,4-bis(phenylmethoxy)phenyl]acetamide (5E)-5-[(2,5-dimethoxyphenyl)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione (E)-4-(dimethylamino)-N-[2-(4-ethylphenyl)-5-fluoropyrimidin-4-yl]but-2-enamide [6-(5,8,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-11-ylmethoxycarbonylamino)hexan-2-ylideneamino]carbamic acid 1-(5-methyl-3-phenyl-4,6,12-triazatetracyclo[7.7.0.02,6.010,15]hexadeca-1,4,8,10(15),11,13-hexaen-12-yl)butan-2-one 2,7-diethyl-4,5-bis(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine 2-amino-5,6-dibromobenzaldehyde 5-chloro-3-fluoro-2-methoxy-6-[1-(pyrrolidin-3-ylamino)ethyl]aniline (1-naphthalen-2-ylsulfanylpyrrolidin-2-yl)methanol;hydrochloride 5-[(2,6-dichlorophenyl)methylsulfanyl]pyridine-2-carboxylic acid 3-[2-chloro-5-methyl-4-(trifluoromethyl)phenyl]sulfanyl-4,6-dihydro-1H-pyrrolo[2,3-c]pyrazole 2-(4-phenylcyclohexa-1,5-dien-1-yl)propanoic acid 2-[4-methoxycarbonyl-N-(4-nitrobenzoyl)anilino]decanoic acid 4-(2,6-dimethylphenyl)-1-[(E)-3-(oxan-4-yl)but-2-enylidene]pyrrolidine-3-carboxamide 2-[4-chloro-3-(trifluoromethyl)phenyl]-1-[4-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]piperidin-1-yl]ethanone N-[6-(3,5-difluorophenyl)-2-(methylaminomethyl)thieno[2,3-d]pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline-7-sulfinamide [2-(hydroxymethyl)pyrrolidin-1-yl]-[6-(4-methoxyphenyl)pyridin-3-yl]methanone N-[4-(2,3-dihydroxypropylcarbamoyl)phenyl]-6-oxocyclohexa-1,3-diene-1-carboxamide (6R,9S)-2-amino-4-benzylsulfanyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-3-carbonitrile 1-[3,5-difluoro-4-[6-methyl-7-(2-piperazin-1-ylethoxy)quinolin-4-yl]oxyphenyl]-3-[2-methyl-4-(5-methylpyrazol-1-yl)phenyl]urea 6-(4-azidobutyl)-7-phenylmethoxyquinoline [2-hydroxy-1-(4-naphthalen-1-ylphenyl)-5-oxopentan-3-yl]azanide 1-[5-(2,3-dihydro-1H-indene-4-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]piperidine-4-carboxylic acid 2-[2,4-di(propan-2-yloxy)phenyl]-N-methylpropanamide 2-cyclobutyloxy-6-[4-(furan-3-yl)-1H-pyrazol-5-yl]pyridine 4-chloro-5-[2-(difluoromethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridine;oxane 6-[3,5-bis(trifluoromethyl)phenyl]-N-methyl-N-[(2R)-1-phenylpropan-2-yl]benzo[b][1,4]benzoxazepine-3-carboxamide N-(3-butanoylphenyl)formamide;ethane 3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-5,7-difluoro-1H-quinolin-4-one 3-hydroxy-4-[2-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)ethoxyiminomethyl]pyrrolidine-2,5-dione (2S)-N-[4-(1H-benzimidazol-2-yl)phenyl]pyrrolidine-2-carboxamide 5-(8-chloronaphthalen-1-yl)imidazolidine-2,4-dione N-[2,5-bis(phenylmethoxy)-3-propan-2-ylphenyl]acetamide (2Z)-2-[6-(4-chlorophenyl)-2-[(4S)-3,3-difluoropyrrolidine-1-carbonyl]cyclohexa-2,4-dien-1-ylidene]acetamide 2-(N-acetylanilino)ethanimidate N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]acetamide N-[2-hydroxy-3-(4-thiophen-2-ylpiperazin-1-yl)propoxy]formamide (2S)-1,2,3,5,6-pentahydroxyanthracene-9,10-dione 2-amino-N,6-diethyl-5-methoxypyridine-3-carboxamide 5-[4-(5,7-dimethoxy-1H-indole-2-carbonyl)piperazin-1-yl]pyrimidine-2-carboxylic acid (2R)-1-(3,4,5-trimethylphenyl)sulfonylpyrrolidine-2-carboxylic acid 1-(2,5-dimethylphenyl)sulfonyl-4-[(3-fluoro-2-propoxyphenyl)-(oxan-4-yl)methyl]piperazine 3-[(4-hydroxyphenyl)methyl]thiophene-2,5-dicarboxylic acid 4-N-cyclopropyl-2,3-dihydro-1H-benzimidazole-4,6-disulfonamide;hydrochloride N-[1-[(2R,4S)-6-methyloxan-2-yl]ethylideneamino]naphthalene-2-carboxamide 4-[(5-but-2-enoxy-6-propylpyridin-3-yl)amino]piperidine-1-carboxylic acid 4-[1-(2,5-difluoro-3-methylphenyl)-2,2,2-trifluoroethoxy]-1H-pyrazole 1-[(E)-3,5-difluoro-2-[(E)-prop-1-enyl]hex-3-enoxy]-4-methylbenzene 5-amino-3-[4-(2,2,2-trifluoroethoxy)phenyl]-1,2-oxazole-4-carbonitrile 2,4-diphenyl-6-[4-(2,4,5-trimethylphenoxy)pyridin-2-yl]oxypyrimidine 1-(4-chlorophenyl)sulfonyl-2-[(Z)-1-phenylprop-1-enyl]piperazine 1-[3,5-bis(trifluoromethyl)phenyl]-N-diazoethanesulfinamide 3-(5-tert-butyl-2-hydroxyphenyl)-N'-methylprop-2-enimidamide 2-azidooxynaphthalene 1-[1,3-bis(2,4,6-trimethylphenyl)imidazolidin-2-ylidene]ethanol 2-(N-ethylsulfonyl-4,5-dimethyl-2-phenyldiazenylanilino)-1-phenylethanone 4-[2,5-dimethyl-1-(oxan-3-yl)pyrrole-3-carbonyl]piperazin-2-one 2-[(3S,4S)-3-fluoropiperidine-4-carbonyl]benzaldehyde [1-methylsulfonyl-3-(phenylcarbamoyl)azetidin-2-yl]boronic acid N-[(4,6-dimethylpyridin-2-yl)methylideneamino]-3-hydroxypyridine-4-carboxamide 2-[3-amino-4-(methyliminomethyl)pyridin-2-yl]sulfanyl-4-propyl-1H-pyrimidin-6-one 3-(2,4-dichlorophenyl)-2-[(Z)-2-iodoethenyl]quinazolin-4-one 2-[6-[(2,4-difluorophenyl)methoxy]pyridin-3-yl]acetamide N-[1-[(3S)-oxolane-3-carbonyl]azetidin-2-yl]-4,5-dihydro-1H-imidazolo[1,2-d][1,4]benzoxazepine-2-carboxamide [3-(1H-indol-5-yl)phenyl]urea 1-[3,5-bis(trifluoromethyl)phenyl]-N-chloro-2,2,4,4-tetramethyl-3H-quinoline-6-carboxamide 5-[2-(7,8-dihydronaphthalen-1-yl)ethyl]pyrimidine 5-ethyl-3-[1-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione 1-[6-[[5-(2,3-dimethylpyridin-4-yl)-8-fluoroquinazolin-4-yl]amino]-2H-pyrazin-1-yl]-N',N'-diethylpropane-1,3-diamine 5-[4-(1H-imidazol-5-ylmethylamino)-2,3-dihydro-1H-inden-5-yl]-N-piperidin-4-yloxypyridine-3-carboxamide 4-amino-N-(5,6-dihydroisoquinolin-8-yl)piperidine-1-carboxamide 4-[[4-(4-acetylanilino)quinazolin-6-yl]amino]benzaldehyde;propan-2-amine 2-(4-methoxyphenyl)sulfinyl-N-[3-(4-propan-2-ylphenoxy)pyridin-4-yl]acetamide 1-[4-(3,5-dimethylphenyl)cyclohexa-2,4-dien-1-ylidene]propan-2-one N-[4-(6,8-dimethoxy-4-oxoquinazolin-3-yl)phenyl]-4-hydroxybutanamide 3-(3-ethoxy-4-phenylmethoxyphenyl)propanoic acid (2R)-N-[4-[7-fluoro-1-methyl-3-oxo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindol-2-yl]cyclohexyl]-2-hydroxypropanamide N-[2-(diethylamino)ethyl]-4-methoxybenzamide 3-[4,5-bis(ethenyl)furan-2-yl]sulfonylbenzenesulfonamide 4-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2H-phthalazin-1-one 2-[1,3-bis(4-methylphenyl)-2H-benzimidazol-2-yl]acetamide 3-(2,4-dihydroxyphenyl)hexanehydrazide N-[2,6-dimethyl-3-(oxan-4-yl)cyclohexa-1,5-dien-1-yl]-3,5-difluoroaniline 2-[N-(4-nitrobenzoyl)-3,5-dioxo-1-[2-(4-sulfobutoxy)phenyl]sulfonylpiperidine-4-carbonyl]-1H-imidazole-5-carboxylate 2,4-ditert-butylpyrimidine;ethane;1,3,5-trifluorobenzene (5S)-6-amino-5-[3-methoxy-4-(2,2,2-trifluoroethoxy)phenyl]hexanoic acid 4-[6-(6-chloropyridin-2-yl)-5-methoxypyrimidin-4-yl]morpholine 6-(2,4-dimethoxybenzoyl)-2-(6-ethoxypyridin-3-yl)-3-oxopyridazine-4-carboxylic acid (3-ethyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-[4-(2-pyridin-3-ylethynyl)phenyl]methanone [7-(dimethylamino)-3,4-dihydronaphthalene-1-carbonyl]carbamic acid (2E,4Z)-5-ethylimino-6-(2-nitrophenyl)hepta-2,4-dienoic acid 3-[5-(4-chlorophenyl)thiophen-2-yl]-1-phenylpropan-1-one 1-[4-(methylamino)-2,7-dioxo-3H-purin-8-yl]pyrazole-4-carboxamide 1,3-bis[(2-fluorophenyl)methyl]thiourea N-butyl-7,9-dimethoxy-4,6-bis(prop-2-ynoxy)benzo[b][1]benzoxepine-3-carboxamide 5-tert-butyl-1-ethyl-3-[[4-(hydroxymethyl)cyclohexanecarbonyl]amino]pyrazole-4-carboxylic acid (E)-3-[4-[[4,6-di(propan-2-yloxy)pyrimidin-5-yl]carbamoylamino]phenyl]-N-[(1R)-1-naphthalen-1-ylethyl]prop-2-enamide 5-[[4-(diethylamino)phenyl]methylidene]-1,3-thiazolidine-2-thione N-[1-(4-aminophenyl)propan-2-yl]-5-chloro-3,6,7,8-tetrahydroimidazo[1,5-a]pyridine-1-carboxamide 6-[(4aS,7S)-3,4a,5,6,7,7a-hexahydro-2H-cyclopenta[b][1,4]oxazin-4-yl]-N-[3-(1H-pyrazol-4-yl)phenyl]pyrimidine-4-carboxamide 3,5-diethoxy-N-[(2E,4Z)-6-[2-[2-[(2S)-1-hydroxypropan-2-yl]oxy-6-pyrrolidin-1-ylpyridine-4-carbonyl]-5-methoxy-1H-indol-3-yl]hexa-2,4-dienyl]benzamide (2S)-N-[1-(2-cyanopyrimidin-4-yl)cyclohexa-2,4-dien-1-yl]pyrrolidine-2-carboxamide 4-[3,5-bis(2-methylpropyl)phenyl]-N-[(1R)-1-(2-iodo-4,6-dimethoxyphenyl)ethyl]-1,3-thiazol-2-amine 1-azido-2,4-bis(3-chlorophenyl)benzene 5-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-[6-(3,5-dimethoxyanilino)pyrimidine-4-carboximidoyl]-N-methylthiophene-2-carboxamide (2S)-4-[3,5-bis(trifluoromethyl)phenyl]-1,2-dibutoxy-4-oxobutane-1-sulfonate N-benzyl-2,4,5-trimethyl-N-(6-nitro-1,3-benzothiazol-2-yl)aniline 3-[2-methoxy-4-(trifluoromethyl)anilino]-5-nitrobenzonitrile 2-[3,5-dimethyl-1-(2-phenylethyl)pyrazol-4-yl]-6-[5-(hydroxymethyl)-1H-pyrazol-3-yl]-3H-thieno[3,2-d]pyrimidin-4-one 7-[4-(5-methylheptan-2-ylidene)cyclohexa-1,5-dien-1-yl]-4H-quinolizine 1-[2-azido-6-(2,2-difluoroethoxy)phenyl]-4-methylpiperazine N-butyl-3,4,5-trifluoro-2-hydroxybenzamide 4-[5-[(2Z)-2,3-dimethylpenta-2,4-dienyl]-1H-pyrrol-3-yl]pyridine 1-[6-(cyclopropanecarbonyl)pyridin-3-yl]-2,4,4a,5-tetrahydro-1H-pyrazino[2,1-c][1,4]benzoxazin-3-one N-ethyl-2,4-dimethoxy-3-[(2S)-3-[2-phenylpropan-2-ylsulfanyl-[(Z)-1-pyridin-2-ylbutylideneamino]amino]butan-2-yl]aniline N-azido-2,4,6-trichlorobenzenesulfonamide 3-azidooxy-1,2,4,5-tetrafluorobenzene 4-[(2S)-butan-2-yl]oxy-N'-hydroxypyridine-2-carboximidamide 2-[(3S)-6,8-difluoro-7,7-dimethyl-3-phenyl-3H-imidazo[1,5-a]pyridin-1-yl]acetic acid 3-bromo-5-cyclopropylpyrazine-2-carboxamide [3-[(2E,4Z)-1,1-dimethyl-5-phenylpenta-2,4-dien-2-yl]oxy-6-methylsulfonylpyridin-2-yl]carbamic acid 1-[(3S)-5,6-diethyl-4-(pyridin-2-ylmethyl)morpholin-3-yl]-N-(1H-imidazol-2-ylmethyl)ethenamine 1-[(4S)-3,4-diphenylcyclopenten-1-yl]cyclopropan-1-amine N-[(1R)-1-(2,3-dihydro-1H-benzotriazol-5-yl)propyl]-6-oxo-2-pyrimidin-2-yl-1H-pyrimidine-4-carboxamide 4-[1-(3-azido-4,6-dihydrocyclopenta[d][1]benzoxepine-2-carbonyl)piperidin-4-yl]benzonitrile 4-[5-(2,6-difluorophenyl)-3-(2H-tetrazol-5-yl)pyrazole-1-carbonyl]benzonitrile 4-(5-azidopyridin-2-yl)piperazine-1,3-dione (Z)-3-(4,5-dimethoxy-2-nitrophenyl)prop-2-enenitrile N-[1,3-dimethyl-5-(2-oxa-8-azatricyclo[7.3.1.05,13]trideca-1(13),5,7,9,11-pentaen-10-ylmethylideneamino)pyrazol-4-yl]ethanimine 4-chloro-6-(3-methoxyphenyl)imino-N'-pyridin-2-ylcyclohexa-1,3-diene-1-carboximidamide 2-cyclohexyl-1-[(1S,5R)-3,8-diazabicyclo[3.2.0]heptan-3-yl]ethanone;6-methoxy-7-methyl-2H-isoquinolin-1-one 5-(3,4-dichlorophenyl)-2H-1,2,6-thiadiazin-3-amine;3-nitropropan-1-ol (6Z)-1'-[5-(1H-imidazol-2-ylmethylsulfanylmethyl)furan-2-carbonyl]spiro[3,9-dihydrofluorene-10,4'-piperidine]-2'-one N-[5-(difluoromethyl)-2-methoxyphenyl]sulfonylcyclohexanecarboxamide 1-(2-ethenyl-3,4,6-trimethylphenyl)piperidine (3R)-1-[3,5-difluoro-4-[1-[5-[(2-methylpropan-2-yl)oxycarbonyl]pyridine-2-carbonyl]piperidin-4-yl]oxyphenyl]pyrrolidine-3-carboxylic acid 3-azidosulfanyl-2,4,6-trichloropyridine 1-methyl-5-[2-methylidene-4-(trifluoromethoxy)-3,4-dihydronaphthalen-1-yl]pyridin-1-ium 2-[(3-amino-5-nitropyridin-4-yl)amino]ethanol 3-[2,6-dichloro-4-nitro-N-(2-phenylethyl)anilino]propane-1,2-diol 4-(3,5-dimethylphenyl)-N-[5-(2,2-dimethylpropanoylamino)pentyl]-1-phenylimidazole-2-carboxamide 1-cyclopropylsulfonyl-3-[6-(1,5-dimethylpyrazol-4-yl)isoquinolin-3-yl]azetidin-3-ol 1-(3,5-dichlorophenyl)sulfonyl-3-[4-fluoro-6-methoxy-7-(piperidine-1-carbonyl)-2,3-dihydroindol-1-yl]propan-1-one 5-(2,3,4,6-tetrahydroxyphenyl)benzene-1,3,4-triol N-[(2S)-1-hydroxybutan-2-yl]-4,7-dimethylpyrrolo[3,2-d]pyrimidine-5-carboxamide 3-[2-(cyclopropylsulfonylamino)pyrimidin-4-yl]-N-[5-methoxy-1,7-naphthyridin-8-yl]piperidine-1-carboxamide 1-[2-[3-chloro-4-[(5-methylpyrazin-2-yl)amino]phenyl]ethynyl]cyclopropane-1-carbonitrile [2-methoxy-4-(5,6,7,8-tetrahydronaphthalen-2-yl)pyridin-3-yl]urea 5-(1,3-benzothiazol-2-yl)-6-[3-methoxy-4-(trifluoromethoxy)phenyl]imino-5-oxohexanoate 4-[5-(cyclopentylmethylamino)pentanoyl]benzenesulfonamide 5-amino-2-(4-nitrophenyl)-1,3-thiazole-4-carboxamide 4-N,4-N-dimethyl-2-(1H-pyrazol-5-yl)benzene-1,4-diamine N-[3,5-bis(trifluoromethyl)phenyl]-4-fluoropiperidine-1-carboxamide 2,3-diamino-N-[4-(N'-butylcarbamimidoyl)phenyl]propanamide;5,6,7,8-tetrahydroquinoline 1-[4-[2-(5-ethylpyridin-3-yl)-4H-thieno[3,2-b]pyrrole-5-carbonyl]piperazin-1-yl]ethanone 1-bromo-6-(4-methylphenoxy)imidazo[4,5-c]pyridine N-[(E)-1H-indol-3-ylmethylideneamino]-1-phenylethanimine;2,3,4-trinitrobenzenesulfonic acid 1-[4-chlorobutyl-(2,6-dibromopyridin-4-yl)amino]propan-2-one 2-(3,5-dimethoxyphenyl)-4,4,5,5-tetramethyl-1H-pyrazol-3-one 2-[[2-chloro-1-[(5R)-4,7-dioxo-5-phenylheptanoyl]indolizine-3-carbonyl]amino]propanoic acid 1-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]cyclohexane-1-carbonitrile 1-(cyclohepten-1-yl)-3-diazo-1-[[4-[5-(trifluoromethyl)pyridin-2-yl]oxyphenyl]methyl]urea 4-amino-6-[(2,3-dibromophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one (5E)-2-cyclohexylimino-5-[[3,4-dimethoxy-5-[(4-nitrophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one 4-methylsulfanyl-2-(trichloromethyl)benzamide 2-(4-amino-3-iodobenzoyl)oxyacetic acid 4-chloro-N-[4-[(Z)-N'-hydroxycarbamimidoyl]phenyl]butanamide [3-(4,5,6,7,8,9-hexahydrocycloocta[d][1,2]oxazol-3-yl)pyrrolidin-1-yl]-(4-methoxypyrazolo[1,5-a]pyridin-3-yl)methanone 7,8-difluoro-3-[2-(4-pentylphenyl)ethynyl]-1H-isochromene 3,4-difluoro-5-[(2R)-oxepan-2-yl]phenol [4-(2,3-diphenylquinoxalin-6-yl)cyclohexa-1,5-dien-1-yl]azanide ethane;5-[3-(4-hydroxyphenoxy)propyl]imidazolidine-2,4-dione 1-(2,3-dihydroindole-1-carbonyl)-4-(1H-pyrazol-5-ylmethyl)pyrrolidin-2-one 2-(3,5-dimethoxyanilino)pyridine-4-carboxamide 1-[4-(2,4-dichlorophenyl)-5-methyl-2,3-dihydropyrrol-1-yl]-2-pyridin-2-ylethanone 3-chloro-4-[4-(difluoromethoxy)phenyl]-1H-pyridazin-6-one N-methyl-6-[4-(trifluoromethoxy)phenyl]pyridin-2-amine 1-[(2R,3S)-2-hydroxyoxolan-3-yl]imidazo[4,5-c]pyridine-2-carbonitrile 3-(hydroxymethyl)-1-(oxan-4-yloxy)isoquinoline-8-carboxamide 4-[2-[1-(4-tert-butylphenyl)sulfonylpiperidin-3-yl]ethoxymethyl]-5-cyclopropyl-3-methyl-1,2-oxazole 2-(6,8-difluoronaphthalen-2-yl)-5,7-dimethoxychromen-4-one (4-chlorophenyl)methylcarbamoyl-[3-[4-ethynyl-2,6-dioxo-5-(phenylsulfanyloxyamino)pyrimidin-1-yl]cyclobutyl]azanium 3-(dimethylamino)propyl-[(5-ethynylfuran-2-yl)methyl]azanide;uranium(2+) 3-[2,4-bis(trifluoromethyl)phenyl]-1-[6-[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]pyridazine-3-carbonyl]azetidin-3-ol 2,4-dichloro-6-[(Z)-[[4-(trifluoromethoxy)phenyl]hydrazinylidene]methyl]phenol (7S)-8-N-benzyl-5-N,6,8-trimethylspiro[2.4]heptane-5,7-dicarboxamide 4-(1H-indol-5-yl)pyridine-2,6-diamine 6-[4-(3-methyl-2-piperidin-1-ylbutoxy)phenyl]naphthalene-2,7-dicarbonitrile N-[(4Z)-5,6-dimethylhepta-1,4,6-trien-3-ylidene]benzenesulfonamide 1-(4-bromophenyl)butan-2-one (E)-3-[5-chloro-2-hydroxy-3-methoxy-6-(3-methylbut-2-enylamino)phenyl]-2-sulfanylprop-2-enoic acid 2-methylpropanamide;N',2,3,4-tetrahydrochromene-8-carboximidamide 1-[2,6-di(propan-2-yl)phenyl]butylidenehydrazine 4-[5-bromo-2,3-difluoro-6-(2H-tetrazol-1-ium-5-yl)phenyl]-7-phenylquinoline N-methyl-1-[4-(2-piperidin-3-ylethynyl)benzoyl]pyrrolidine-3-carboxamide 3-[6-chloro-1-(2,3-dihydro-1H-inden-4-yl)pyrido[2,3-b]indol-9-yl]cyclobutan-1-ol 2-(dimethylamino)-1-(2,4-dimethylphenyl)sulfinyl-3-(trifluoromethyl)guanidine;methanol 5-chloro-4-N,4-dimethyl-2-N-[3-(1H-pyrazol-5-yl)phenyl]pyrimidine-2,4-diamine;ethane N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[[5-ethyl-7-hydroxy-8-[(1R,3S,5S)-3-hydroxy-5-nitrocyclohexyl]quinazolin-4-yl]amino]acetamide 1-[2-(4-ethylphenyl)ethynyl]-3,6-dimethylpyrimidine-2,4-dione 2-(3,4-dichlorophenyl)-N-[[1-[2-[3-(trifluoromethoxy)phenoxy]acetyl]piperidin-3-yl]methyl]acetamide (2S)-2-[5,7-difluoro-6-(4-isocyanophenyl)naphthalen-2-yl]-1,1,1-trifluoropropan-2-ol 7-fluoro-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole 7-[2-(azetidin-1-ylmethyl)morpholine-4-carbonyl]-3H-quinazolin-4-one 2-[[(5S)-3,7-diethyl-4,8-dioxo-6,7-dihydro-5H-pyrimido[5,4-b]pyrrolizine-5-carbonyl]amino]benzoic acid 3-N-[4,6-dichloro-1-[(2R)-2-methyloxiran-2-yl]-5,6-dihydroindol-4-yl]isoquinoline-1,3-diamine (E)-1-(2,3,4,5-tetramethylphenyl)prop-1-en-1-ol N-[4-(3,5-dichlorophenyl)sulfonylphenyl]quinoline-2-carboxamide 6,7-bis(4-methoxyphenyl)pyrrolo[2,3-b]pyridine 2-(3,4-dichlorophenyl)-2-oxoethanesulfonic acid 6-[4-(2,3-dihydroindol-1-yl)butanoyl]-N'-methylpyridine-2-carboximidamide (E)-3-[4-[5,5-dimethyl-7-oxo-6-(4-phenoxyphenyl)-2H-pyrazolo[1,5-a]pyrimidin-4-yl]phenyl]prop-2-enamide 1-phenyl-N-[2-(trifluoromethoxy)ethyl]imidazo[4,5-c]pyridin-6-amine 2-N,5-dipyridin-2-yl-2-N-(2-pyridin-4-ylethoxy)pyrimidine-2,4-diamine N'-(2,6-difluorophenyl)-3-oxobutanimidamide 3-[4-(2,4-dimethylimidazol-1-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-5-(4-methylpyridin-3-yl)-1H-pyrazolo[4,3-b]pyridine 2-[4-[[5-(dimethylamino)thiophene-3-carbonyl]amino]pyrazol-1-yl]acetic acid 4-(2,3-dihydro-1H-inden-5-yl)-N'-(methylideneamino)-1,3-thiazol-2-amine 4-(2,6-dimethylphenyl)-5H-pyrrolo[3,4-b]pyridine;3-fluoropyridine (5R)-2-[(3R,4S)-3-hydroxypiperidin-4-yl]-2-phenyl-1,3-dioxane-4,6-dione 2,6-ditert-butyl-4-(5-methoxy-3-methylsulfanyl-1H-pyrazol-4-yl)phenol N-[1-(4,5-difluoropyrimidin-2-yl)piperidin-4-yl]-2-methoxyacetamide N-[1-(4,5-dimethylfuran-2-carbonyl)piperidin-3-yl]benzenesulfonamide (2S)-1-[3-[[4,7-dimethyl-6-(oxan-4-yloxymethyl)quinolin-2-yl]amino]cyclobutyl]piperidine-2-carboxylic acid (1S,2R)-N-[5-ethyl-6-fluoro-2-hydroxy-3-(4-methoxybenzoyl)phenyl]-2-methylcyclopropane-1-carboxamide 7-[(2R,3S)-3,4-dihydroxybutan-2-yl]oxyquinoline-6-carbonitrile 2-[[4-(1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yloxymethyl)phenyl]methyl]isoindole-1,3-dione;methanol ethane;1-[2-(3-methylcyclopenten-1-yl)ethynyl]-4-nitrobenzene N-(1,2-diamino-2-oxoethyl)-3-[4-[4-(1,3-benzothiazol-5-yl)-6-morpholin-4-ylpyrimidin-2-yl]phenyl]propanamide 1-benzylsulfanyl-4,5-bis(ethenyl)pyrazole 4-N,8,8-trimethyl-1H-pyrano[3,2-f]quinoline-2,5-diamine 3-(6,7-dihydropyrazolo[1,5-a]pyrazin-4-yl)-2H-pyrazolo[3,4-c]isoquinoline (4-bromocyclohexyl)oxymethylbenzene 7-[(Z)-1-amino-3-iminoprop-1-en-2-yl]-N,6-dimethylquinazolin-4-amine;ethane N-(cyclohexylmethyl)-3-[4-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylsulfanylmethyl)-1H-benzimidazol-2-yl]aniline 2-methoxycarbonyl-4,5-dimethylbenzoate 2-[2,3-dimethyl-1-(6-propan-2-yloxypyridazine-4-carbonyl)indol-7-yl]acetic acid 1-[(3R)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-3-yl]-4-hydroxypiperidin-3-one 4-[1-[2-fluoro-5-methyl-3-(trifluoromethyl)phenyl]ethylideneamino]piperidine-1-carboxamide 2-[2,4-dioxo-6-(2-phenylethyl)-1H-quinazolin-3-yl]acetamide N-cyclohexyl-2,5-dimethoxybenzenesulfonamide [3-amino-4-(5,7-dihydropyrrolo[3,4-b]pyridin-6-yl)-2-methanimidoylphenyl]methylideneazanium 4-methyl-N'-(1H-pyrazol-5-yl)benzenecarboximidamide 1,2-bis(3-chlorophenyl)-4-methylbenzene N-(5,7-dimethylcyclohepta-1,3-dien-1-yl)-4-[2-(2-hydroxyethoxy)phenyl]benzamide 2-(1-methylindol-3-yl)oxy-1-[4-[2-(oxolan-3-ylamino)ethyl]piperidin-1-yl]ethanone 3-[5-[[(2S,4R)-4-fluoropiperidin-2-yl]methoxy]-2,3-dihydroindole-1-carbonyl]benzonitrile 5-butyl-2-fluoro-3-phenylphenol 4-(9H-fluoren-1-yl)phenol 1-[4-(2,3-dihydroxypropyl)phenyl]ethanone;ethane (Z)-N-methyl-2-[4-(1-phenylethylamino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]ethenamine 4-N,6-N-bis(2-chloroacetyl)naphthalene-1,4,6-tricarboxamide 1-ethenyl-4-[(2Z,4E)-5-methoxyhepta-2,4,6-trien-3-yl]benzene;formic acid 4-[(1,2-dimethylpiperidine-3-carbonyl)amino]pyridine-2-carboxamide (6R)-N-[(4-methoxyphenyl)methyl]-2,7-diazaspiro[5.5]undecan-8-imine N-(2,3-dihydro-1H-inden-1-yl)-N',N'-diethylbutanediamide 2-(1,3-benzodioxol-5-yl)-6-[(2S,5R)-2,5-dimethylcyclopenten-1-yl]pyridine 2-amino-3-(2,6-dimethoxyphenyl)butanal;4,5-dimethylcyclohexa-1,5-dien-1-ol 2-[[5-(ethoxymethyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-4-methyl-1H-pyrimidin-6-one (4-fluorophenyl)methyl-[2-[2-[2-[2-[formyl-[3-hydroxy-1-(hydroxyamino)-1,5-dioxopentan-2-ylidene]azaniumyl]ethoxy]ethoxy]ethoxy]ethyl]azanide 2-(ethoxymethyl)-N-[[1-[2-[4-[6-[(Z,3S)-3-hydroxypyrrolidin-1-yl]-2-methylpyrimidin-4-yl]phenyl]acetyl]cyclopropyl]methyl]pyridine-4-carboxamide N-[1-[5-amino-3-(1-hydroxyethyl)-6-methoxypyrazin-2-yl]pyrrolidin-3-yl]acetamide 3-[4-[(E)-6-(cyclohexen-1-yl)hept-2-enoxy]-3-methoxyphenyl]propanoic acid 2-methyl-4-(2-piperidin-3-ylpyrazol-3-yl)pyridine 1-[(2Z,5E)-6-aminohepta-2,5-dienyl]-N'-hydroxyimidazole-2-carboximidamide;ethane 7-(4,5-dimethyl-1H-pyrazol-3-yl)-6,8,9,10-tetrahydro-[1]benzothiolo[2,3-b]quinoline (E)-1-(2,4-dihydroxyphenyl)-3-thiophen-2-ylprop-2-en-1-one [3-(ethylsulfanylamino)phenyl]-methoxymethanol 5-[(1E,4Z)-3,5-dichlorohepta-1,4-dienyl]-1H-indole 2-(4-tert-butylphenoxy)-N-[(3R,5S)-1-(oxan-4-ylmethyl)-5-propylpyrrolidin-3-yl]acetamide 5-[(1R)-1-[[6,7-bis(2-methoxyethylimino)-1,3-diazinan-5-ylidene]amino]-2-hydroxyethyl]thiophene-2-carboxamide 3-[1-(4,5-dichloro-2-propylphenyl)ethoxy]pyridine 1-ethenyl-3-[(4-iodophenyl)methoxy]benzene (6E)-7-[2,5-bis(phenylmethoxy)phenyl]-6-[(3-iodophenyl)methylidene]heptanoic acid 5-[(E)-3,4-dihydroxybut-2-enyl]-7-ethyl-1H-indazole-6-carboxylic acid 3-chloro-5-[(2R,6S)-4,4,6-trifluoro-1-methylpyrrolidine-2-carbonyl]benzonitrile 3-(4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-ylmethylidene)piperidine-2,6-dione N-[4-(4-amino-2-butylimidazo[4,5-c]quinolin-1-yl)butyl]-3-methoxypropane-1-sulfonamide [(3S,4R)-2,6-dihydroxypiperidin-3-yl]-[1'-(thiophen-2-ylmethyl)spiro[1H-isoquinoline-4,3'-azetidine]-7-yl]methanone;dihydrochloride 2-(3,5-difluorophenyl)benzenethiol;hydrochloride [(2E,4Z)-hepta-2,4,6-trien-3-yl]sulfonylbenzene 1-amino-3,5-bis(2,6-dimethoxyphenyl)-4H-quinazolin-2-one 1,2-diamino-4-[5-chloro-3-fluoro-2-(trifluoromethoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile (E)-3-[4-[5-[6-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)pyridin-3-yl]sulfonylpyridin-2-yl]phenyl]-N'-methylbut-2-enimidamide (2R)-2-[3,5-difluoro-4-[7-(furan-3-yl)-1H-imidazo[4,5-b]pyridin-2-yl]phenoxy]propanoic acid (3Z)-4-[(E)-but-2-enoxy]hexa-1,3,5-triene;N,4-dimethylcycloheptanamine;ethane;6-[4-fluoro-2-(prop-1-ynylamino)phenyl]quinazolin-4-amine N-[2-azido-1-(3-chlorophenyl)ethyl]-2,5-dimethoxyaniline 5-amino-1-[(2S,3R)-4-hydroxy-3-methylbutan-2-yl]pyrazolo[3,4-d]pyrimidine-3-carboxylic acid (3R)-4-[3-(4-hydroxyphenyl)prop-2-ynoyl]-N,N-dimethylmorpholine-3-carboxamide 3-(4-azido-2,5-dimethoxyphenyl)propanoic acid N-[5,6-dimethyl-2-(4-propan-2-ylcyclohexyl)oxypyridin-3-yl]formamide N-(2,2-dimethoxyethyl)-N-(4-nitrophenyl)butanamide (2E)-N,N'-bis[(3,4-dichlorophenyl)methyl]penta-2,4-dienimidamide 1-(2-azidooxyethyl)-3-(4-chlorophenyl)pyrazolo[3,4-c]pyridine 3-[2-(6-amino-1,3-dioxobenzo[de]isoquinolin-2-yl)ethoxy]-N-propylpropanethioamide 6-[5-(dimethylamino)-2-(ethoxymethyl)imidazo[1,2-c]pyrimidin-7-yl]pyridine-3-carbonitrile 3-[5-aminosulfanyl-6-(methylamino)pyridin-2-yl]oxy-4,7-difluorobenzaldehyde;ethane 2-chloro-N-[2,4-dioxo-6-(trifluoromethyl)-1H-pyrimidin-5-yl]acetamide 2-[(1E)-2,4-dimethylpenta-1,3-dienoxy]-6-[2-(4-fluorophenyl)pyrazol-3-yl]benzonitrile 2-(5,6,7-trimethylnaphthalen-1-yl)propanamide 6-[(1S)-4,5-dimethylcyclohexa-2,4-dien-1-yl]oxypyridazine-3-carboxamide 3-bromo-5-[(2S)-4-(2-chloro-6-methylphenyl)sulfonylmorpholin-2-yl]-N,N-diethylpyrazolo[1,5-a]pyrimidin-7-amine 4-(4-ethoxyphenyl)-1,3,5-triphenylpyrazole 5-[2-methylpropyl(pyridin-3-yl)amino]-3H-1,3,4-thiadiazole-2-thione 2-methyl-6-[3-[(4-methylpyrazol-1-yl)methyl]azetidine-1-carbonyl]pyridazin-3-one 5-fluoro-3-[2-(1,1,4-triazol-1-yl)ethoxy]quinoline 1-(4-aminobutanoyl)-N,N'-diethyl-2-[[3-(hydroxymethyl)phenyl]methyl]piperidine-2-carbohydrazide 3-[2,6-dibromo-4-(1,1,2,2-tetrafluoroethoxy)phenoxy]-3-phenylpropanal (4S)-N,N-diethyl-1-[5-(5-methylpyridin-3-yl)-1H-imidazol-2-yl]-6-phenylpiperidin-4-amine 3-[4-chlorobutyl(2H-tetrazol-5-yl)amino]propanoic acid 1-[4-(4-azidophenoxy)piperidin-2-yl]-N,N-dimethylmethanamine 4-methoxycarbonyl-3,5-bis(phenylmethoxy)benzoic acid 2-[(4E)-5,7-dimethylocta-1,4-dien-3-yl]-5,6-dihydroquinoline 1-[(2S,3aR)-5-(2-methylpropoxy)-2,3,3a,4,9,10,11a-octahydro-1H-benzo[g]quinolizin-2-yl]-3-hydroxyimidazolidine-2,4-dione N-(2,6-dichlorophenyl)-4-oxo-3H-quinazoline-8-carboxamide 1-[(4-ethylphenyl)methoxy]carbonylpiperidine-3-carboxylic acid 4-(3,3-difluorocyclobutyl)oxy-1-[2-methyl-6-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenoxy]butan-2-ol 6-[6-fluoro-1,4-dioxo-7-(trifluoromethyl)phthalazin-2-yl]-N-[(3S)-oxolan-3-yl]pyridine-3-carboxamide 1-(2,6-dichlorophenyl)-5-[(3R)-3-methyl-4-morpholin-4-ylpiperidin-1-yl]pentan-1-one 3-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]-N-ethanimidoyl-6-(4-fluorophenyl)pyridine-2-carboxamide 5-methyl-3-[4-(pyridin-2-ylamino)piperidin-1-yl]pyrazine-2-carbonitrile N-(2,6-difluorophenyl)-N-ethylsulfonylbenzenesulfonamide 4-[[3,5-dimethyl-1-(2-methylpropanoyl)pyrazol-4-yl]methyl]-6-oxopiperazine-2-carbonitrile 1-[5-(2,3,4-trimethoxyphenyl)sulfanylthiophen-2-yl]ethanone N-[5-(furan-2-yl)-1H-pyrazol-3-yl]-2-hydroxy-4-nitrobenzamide 5-fluoro-2-[4-[(Z)-1,3,3-trifluoroprop-1-enyl]phenyl]-N-[[3-(trifluoromethoxy)phenyl]methyl]pyrimidine-4-carboxamide 5-[2,6-difluoro-4-(trifluoromethyl)phenoxy]-N,N-dimethyl-4-oxopentanamide (5Z)-2-(3,4-dichlorophenyl)imino-5-[[5-(1,2-dihydropyridin-6-ylmethoxy)furan-2-yl]methylidene]-1,3-thiazolidin-4-one 3-[2-(2,6-dioxopiperidin-3-yl)-1,3-thiazol-4-yl]-N-methylsulfonylpropanamide 2,4-dimethyl-6-propanoyloxybenzoate (5Z)-2-sulfanylidene-5-[(3,4,6-trimethylcyclohexa-1,3-dien-1-yl)methylidene]imidazolidin-4-one 1-[4-fluoro-3-(trifluoromethyl)phenyl]-3H-pyrazole-2-carbonitrile 2-(benzenesulfonyl)-1-(4-methoxybutyl)guanidine 4-[4,5-bis(phenylmethoxy)pentyl]benzoic acid 3-[(2-chlorophenyl)methoxy]-5,6-dihydroimidazo[1,2-b]pyrazole-7-carboxylic acid (4R)-2,2-dimethyl-1'-[6-(trifluoromethoxy)pyridin-3-yl]spiro[5H-1-benzofuran-3,4'-piperidine] 3-bromo-4-methyl-5-[2-(trifluoromethoxy)phenyl]pyridine 3-N,4-N-di(propanoyl)benzene-1,2,3-tricarboxamide;hydrate (2S)-N'-hydroxy-1-[4-(3-methoxyphenyl)thiophen-2-yl]sulfonylpiperidine-2-carboximidamide;hydrochloride (E)-1-[4-amino-5-cyclopropyl-3-(hydroxymethyl)pyrazol-1-yl]prop-1-en-2-ol 3-fluoro-4-[(2R)-1,1,1-trihydroxypropan-2-yl]oxybenzamide 2-[3-(6,7-dimethylquinazolin-4-yl)-5-propan-2-yloxyphenoxy]ethanol 2-(4,5-dihydroimidazo[1,2-a]quinolin-3-yl)-N,N-dimethylethanamine;ethane 4-[(2Z)-3-fluoro-3,7-dimethylocta-2,6-dienoxy]-2,5-dihydroxybenzoic acid 7-fluoro-4,5,9a,10-tetrahydrophenanthrene (5E)-4,6-dihydroxy-3-(1-naphthalen-2-ylethylideneamino)hexa-5,7-dienoic acid (Z)-2-cyano-3-(3-ethoxyphenyl)prop-2-enamide N-(3-chloropropyl)-3,4,5-trimethoxybenzamide 6-[4-(N'-hydroxycarbamimidoyl)pyrazol-1-yl]hexanoic acid 2-azidooxyacridine 2-(4-methylcyclohexa-1,3-dien-5-yn-1-yl)sulfanyl-1H-indole N-methylspiro[1,4-dihydroisoquinoline-3,1'-cyclopropane]-2-imine N-[4-[6-amino-5-(azetidine-1-carboximidoyl)pyridin-2-yl]oxycyclohexylidene]hydroxylamine (Z)-2,3-bis[2,6-di(propan-2-yl)phenyl]but-2-enedioate 2-chloro-4-[[4-(trifluoromethyl)-1,3-thiazol-5-yl]methoxy]benzaldehyde N-[2-(3,4-dimethoxyphenyl)ethyl]-5-hydroxy-1-methyl-6-oxo-7H-pyrazolo[3,4-b]pyridine-4-carboxamide 1-[(2S,3R)-3-aminooxan-4-yl]-N-methoxypyrazolo[3,4-d]pyrimidine-3-carboxamide 5-[(E)-3-fluoro-2-methylprop-1-enoxy]-4-phenyloxolan-2-one N-[5-(2-chlorophenyl)-1,3,4-thiadiazol-2-yl]-6,7-dihydro-5H-cyclopenta[c]pyridine-6-carboxamide 2,6-bis[(4-chlorophenyl)methyl]-3-pentoxyaniline N-[3,5-bis(trifluoromethyl)phenyl]-4-[1-(diaminomethylideneamino)ethenyl]benzamide 2-methyl-N-(3-nitrophenyl)-6-(trifluoromethyl)pyridine-4-carboxamide 4-amino-N'-(1,3-benzodioxol-5-yl)-2-methyl-6-[[4-(trifluoromethoxy)benzoyl]amino]pyrimidine-5-carboximidamide 3-(4-acetylphenyl)-2,5-dimethoxybenzaldehyde 1-[4-(3,5-dimethylthiophen-2-yl)-6-methoxy-7-methylquinazolin-2-yl]ethanamine [(3Z,5E)-1-cyclohexylhepta-3,5-dien-2-ylidene]-dimethylazanium 2-[3-(1H-pyrazol-4-yl)phenyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine 5-(3,4-dichlorophenyl)-7H-pyrrolo[2,3-d]pyrimidine 2-(4-bromophenyl)-1,6-dioxobenzo[b][1,8]naphthyridine-5,11-dione 4-(3,5-dimethylphenyl)benzoic acid;ethane 2-benzyl-N-[4-(propanoylsulfamoyl)phenyl]furan-3-carboxamide 2-[6,7-dichloro-4-(difluoromethyl)-5-iodoisoquinolin-1-yl]ethanesulfinate 1-(2-aminoethyl)-6-(4,4-dimethoxybut-2-enyl)-3H-imidazo[4,5-c]pyridine-2-thione;hydrochloride 4-[(6R)-7-(3,5-dichloro-2-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]benzonitrile 4-(2,6-difluoro-3,5-dimethoxyphenyl)-N-[4-[[4-(trifluoromethylsulfonyl)piperazine-1-carbonyl]amino]cyclohexa-1,3-dien-5-yn-1-yl]pyridine-2-carboxamide 6-[1-(4,4-dimethylcyclohexen-1-yl)-3-(trifluoromethyl)pyrazol-4-yl]pyridazine-3-carbonitrile 1-azido-6,8-dibutoxyanthracene N-(2,4-dichlorophenyl)-2-[1-(3-methylbenzoyl)piperidin-4-yl]acetamide;4-methoxy-6-propan-2-yloxypyrimidine 7-fluoro-2,4-dimethyl-3H-isoindol-1-one;3-[4-(2-propanoyloxyethoxy)butoxy]propanoic acid N-[(4,5-dichlorocyclohexa-1,3-dien-1-yl)methyl]-N-[6-[ethyl-[2-(1H-imidazol-5-yl)ethylcarbamoyl]amino]pyrimidin-4-yl]formamide N-[[(2S,4R)-1-acetyl-5-cyclohexyl-3,4-dihydro-2H-quinolin-7-yl]methyl]acetamide 2-(2,6-dibromoanilino)acetate 3-(2-azidooxyethyl)-1H-quinolin-4-one 1-[(Z,2S)-4-amino-3,3,5-trimethylhex-4-en-2-yl]pyridin-2-one 4-chloro-3-(4,5-dihydro-1H-imidazol-2-yl)benzamide (5R)-3-[4-[1-cyclohexyl-2-[6-methoxy-5-[(4S)-4-methyloxolan-3-yl]pyridin-3-yl]ethynyl]phenyl]-5-ethynyl-1,3-oxazolidine 4-cyclohexyl-N-(2,3-dimethoxyphenyl)butanamide (3S)-N-[1-(2,6-difluorophenyl)cyclopropyl]-1-methylpyrrolidine-3-carboxamide (2S)-3,3,4-trimethyl-2-[[5-phenylpentanoyl-(pyridin-3-ylmethyl)amino]carbamoyl]azetidine-1-carboxylic acid 1-[2,4-dimethyl-5-(2-methylphenyl)-3-phenyl-5H-1,2-oxazol-2-ium-4-yl]ethanone;ethane 3-bromo-N'-(1-hydroxyethyl)benzenecarboximidamide 5-tert-butyl-N,3-dimethylthiophene-2-carboxamide (4-aminophenyl)sulfonyl-propylazanide (5Z)-2-imino-5-[(4-propoxyphenyl)methylidene]imidazolidin-4-one 2-amino-4-[5-bromo-3-(4-iodopyrazol-1-yl)furan-2-yl]-6-methylbenzene-1,3-dicarbonitrile 2-(6,7-difluoro-1H-indol-3-yl)-6-[4-ethoxy-3-(trifluoromethyl)phenyl]pyrido[3,4-d]pyrimidine 6-[(3R)-5-amino-2,3-dihydro-1H-isoindole-3-carbonyl]-N'-cyano-4-oxo-7,8-dihydro-5H-pyrazolo[1,5-d][1,4]oxazepine-2-carboxamide (5Z)-2-cyclohexylimino-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 1-chloro-5,7-dihydropyrrolo[2,3-f]benzimidazole 1-[5,7-dimethyl-6-(2-phenylethynyl)cycloocta-1,3,7-trien-1-yl]propan-1-one 2-[[4-methyl-3-(phenylcarbamoyl)pyridine-2-carbonyl]amino]acetic acid 1-azidooxy-2,3-dichloro-4-nitrobenzene 3,4-difluoro-N-[6-(1H-imidazol-5-yl)hexyl]benzamide 2-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-N'-[3-fluoro-5-methoxy-4-[4-(trifluoromethylsulfanyl)piperazin-1-yl]phenyl]propanediamide 2-[6-amino-5-(4-chlorophenyl)pyridazin-3-yl]phenol 3-(9H-fluoren-9-ylmethoxycarbonylamino)-2-propan-2-ylbutanoic acid 5-[(1-benzylpiperidin-4-yl)carbamoylamino]-2,3-dihydroindole-1-carboxamide N-[(2S)-1-[[3-azido-6-(4-chlorophenyl)hexyl]amino]propan-2-yl]acetamide 2-tert-butyl-6-[(3E,5Z)-hepta-1,3,5-trien-4-yl]naphthalene 3-azidooxy-1H-indazole-6-carboxamide (1R)-2-[4,4-bis[3,5-ditert-butyl-4-hydroxy-N-methylanilino)anilino]butanoylamino]cyclohexane-1-carboxylic acid 2-[4-(dimethylamino)phenyl]-N-methyl-1H-imidazole-5-carboxamide 3-[5-chloro-2-(methoxymethoxy)phenyl]-1,8a-dihydroquinoline 3-[[(2S)-1-[4-[2,4-bis(aminomethyl)phenoxy]butanoyl]pyrrolidine-2-carbonyl]amino]propanoic acid (2S)-2-amino-3,3-dimethyl-N-[4-[3-[methyl(sulfanyl)amino]propoxy]phenyl]butanamide 6-(1,3-benzodioxol-5-ylmethyl)-7H-pyrrolo[2,3-c]azepine 3-ethenyl-6-methylidene-4,5,7-triphenyl-1H-cyclopenta[c]pyrazole;1-methyl-2-(4-methylphenyl)benzene 2-chloro-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxylic acid [(2S,4R)-1-(cyclohexanecarbonyl)-2-methyl-3-oxopiperidin-4-yl]-[3-(5-fluoropyridin-3-yl)propanoyl]azanium 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]-6-ethenyl-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 2,3-dihydro-1H-indol-6-yl(pyridin-4-yl)methanol 7-(aminomethyl)-4-ethynyl-2-iodo-1,4-benzoxazin-3-one 3-[(2Z,4E)-6,7-difluorohepta-2,4,6-trien-3-yl]-5-[2-[5-(1-methylpyrazol-4-yl)-1H-pyrazolo[3,4-c]pyridin-3-yl]-1H-imidazo[4,5-b]pyridin-7-yl]phenol 3-methoxyimino-2,5-dimethyl-4-[(1S)-1-naphthalen-1-ylethyl]piperazine-1-carboxylic acid 5-(2-phenylethenyl)bicyclo[2.1.1]hexane N-ethyl-6-[(1S)-4,5,7-trifluoro-2,3-dihydro-1H-inden-1-yl]naphthalene-2-carboxamide N-[2,4,6-trichloro-3-(6-ethylhexyl)phenyl]methanimine 1-(3,4-dichlorophenyl)-5H-pyrrolo[2,3-d]pyridazin-7-one (1S,2R)-1,5-dichloro-2-[3-chloro-6-(methoxymethyl)-2-phenylphenoxy]cyclohexa-3,5-diene-1,3-dicarboxylic acid 5-[4-(cyclopropylmethoxy)phenyl]-3,4-dimethylthiophene-2-carboxylic acid 2-amino-6-(4-oxospiro[3H-chromene-2,1'-cyclopentane]-7-yl)benzenesulfonamide 4-(1,2,3,6-tetrahydropyridine-5-carbonyl)-8-[3-[(2S,4R)-4-phenylpyrrolidin-2-yl]propanoyl]-1-oxa-4,8-diazaspiro[5.5]undecan-3-one 3-chloro-2,4-dinitrobenzoic acid;methanol (1E,3Z)-2-[amino(naphthalen-1-ylmethyl)amino]penta-1,3-diene-1-thiol;ethane 7-chloro-2-ethyl-N,1-dimethylimidazo[4,5-c]pyridine-6-carboxamide (6S)-2-(1,3-benzothiazol-4-ylmethoxymethylamino)-4,8-dioxo-N-propan-2-yl-6-[3-[2-(trifluoromethyl)pyrimidin-5-yl]phenyl]-6,7-dihydro-5H-pteridine-9-carboxamide (2R,3S)-2-azido-1-N-[4-[(4-methoxyphenyl)sulfonylmethyl]cyclohexa-1,5-dien-1-yl]-4-oxo-4-N-[(4-propan-2-ylphenyl)methyl]butane-1,3-dicarboxamide 2,3-dihydroxy-7-[4-(trifluoromethoxy)phenyl]-1H-pyrrolo[2,3-b]pyridine N-cyclopentylformamide;ethane;1,4,5,8-tetrafluoronaphthalene 5-(2,3-dihydro-1H-inden-4-yl)-N'-ethoxy-N-hydrazinylidenepyridine-2-carboximidamide [3-(7-amino-2-azido-1H-imidazol-5-yl)phenyl]methanol 2-[4-chloro-5-(methylamino)pyrazol-1-yl]propanoic acid 2-[(3R)-6-(4,4-dimethylpiperidine-1-carbonyl)-3-propan-2-yl-3,4-dihydro-2H-chromen-2-yl]-N'-[3-fluoro-4-(trifluoromethoxy)phenyl]acetohydrazide 6-[(3,4-difluorophenyl)methyl]-2-pyridin-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-[(E)-3-phenylprop-2-enoxy]benzenesulfonamide 1-(2-azidoethylsulfanyl)-4-fluorobenzene 2-(3-methylsulfanylpiperidin-1-yl)-4,7-dioxo-5-[2-[3-(trifluoromethoxy)phenyl]phenyl]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile 2-[(3Z)-6-fluorohepta-1,3-dien-4-yl]-1H-benzimidazole (3S)-5,7-dichloro-N-(2,6-difluorophenyl)-1'-methylspiro[1H-indole-3,4'-5,7-dihydropyrazolo[3,4-b]pyridine]-2-imine 7-cyclopentyl-6-hydroxy-3,5-dimethoxythieno[3,4-d]pyrimidin-4-one (1R,2S)-N-[8-amino-6-(4-methylpyridin-3-yl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 4-[2-(4,6-diaminopyridin-3-yl)ethynyl]benzoic acid 1-azidooxy-2-(1,2,3,4-tetrahydronaphthalen-1-yl)naphthalene 5-methoxy-2-[[6-(1,3-oxazol-5-yl)pyridine-2-carbonyl]amino]-4-phenylthiophene-3-carboxylic acid 3-[(Z)-1H-indol-5-ylmethylideneamino]-2-pentan-3-ylquinazolin-4-one 2-[[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxospiro[3H-isoindole-4,2'-cyclopropane]-5-yl]-7,8-dihydronaphthalene-2-carbonyl]amino]acetic acid (3R)-7-[4,5-bis(ethenyl)imidazol-1-id-2-yl]-9-methyl-3-pyridin-2-yl-2H-carbazole;1-prop-1-en-2-yl-3,6-dihydro-2H-pyridine;ruthenium(2+) 1-[1-(4-fluorophenyl)ethyl]-3,5-dimethylbenzimidazol-2-one 2-(3,5-dimethyl-1H-pyrazole-4-carbonyl)benzaldehyde (5R)-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one;1-ethyl-4-methoxycyclohexane 1-azido-2-(dimethylamino)-3,4,6-triethyl-5-phenylcyclohexa-2,4-diene-1-carbonitrile 2-[(3R)-1-cyclobutylpiperidin-3-yl]oxy-5-pyrimidin-5-ylbenzoic acid (2R)-1-[6-cyano-5-methyl-3-[4-(trifluoromethoxy)phenyl]pyrazine-2-carbonyl]piperidine-2-carboxamide 1-(2,4-difluorophenyl)sulfonylpiperazine 2-[4-[2,6-dimethyl-3-(methylcarbamoyl)-1-benzofuran-5-carbonyl]-2,5-bis[[4-(trifluoromethoxy)phenyl]methoxy]phenoxy]-2-methylpropanoic acid (Z)-1,2-diamino-3-[2-amino-5-(4-hydroxypiperidine-1-carbonyl)phenyl]prop-2-en-1-one 4-(2,6-difluorophenyl)-3-[2-methyl-4-(2-methylpropoxy)anilino]sulfanylbenzoic acid 4-N-(2,3-dihydro-1H-isoindol-5-yl)-6-pyridin-3-ylpyrimidine-2,4-diamine 5-(4-phenylmethoxybutyl)pyrazine N-[1-(2,3-dimethylphenyl)-5-hydroxy-4-oxopyridazin-3-yl]thiophene-2-sulfonamide 4-azido-2-phenoxyquinazoline N-(4-chlorophenyl)-3-propyloctanamide 4-[5-(methylamino)pyrazin-2-yl]phenol 5-(4-chlorophenyl)-2-methyl-3-propanoylfuran [4-[3,5-difluoro-4-(2-isothiocyanatoethoxy)phenyl]phenyl]boronic acid 1-[4-[2-(dimethylamino)ethoxy]-6-propan-2-ylpyrimidin-5-yl]-3-[[7-fluoro-2-(trifluoromethyl)quinolin-4-yl]amino]cyclobutane-1-carboxamide 1-(2-methoxyethyl)-4-[(3-phenylimidazol-4-yl)methyl]piperazine;2,2,2-trifluoroacetic acid 2-chloro-N-(4-methylphenyl)-N-pyridin-3-ylacetamide;methanamine 4-methyl-3,6-diphenylpyridine;pentane N'-[amino(methyl)amino]-4-[4-[[8-[[(2R)-pentan-2-yl]amino]pyrido[3,4-d]pyrimidin-2-yl]amino]phenyl]piperazine-1-carboximidamide N-(3,5-dichloropyridin-4-yl)-2-[8-methoxy-1-(pyridine-3-carbonyl)-6H-pyrrolo[3,2-e]indol-3-yl]acetamide 4-(6-fluoro-2H-pyran-3-yl)pyridine 2-[7-methyl-2-(trifluoromethyl)pyrazolo[1,5-a]pyridine-3-carbonyl]cyclohexane-1-carboxylic acid 6-[3-chloro-4-(trifluoromethyl)phenyl]-2-methylidene-1,5-dihydropyrido[3,4-b]azepine N-(4-aminocyclohexyl)-N,5-dimethylnaphthalene-2-carboxamide 4-[[(3S)-3,4-dimethylpiperazin-1-yl]methyl]-N'-hydroxypyridine-2-carboximidamide N-(cyclopropylmethyl)-1,3-dimethoxy-2-phenylbutan-2-amine 2-[4-[(6E)-7,9-dimethylundeca-1,6,8,10-tetraen-3-yl]-5-ethenylthiophen-2-yl]-1H-benzimidazole 2-[(3,4-diethylphenyl)methylidene]propanedinitrile 1-(1H-benzimidazol-2-yl)-6,7-dimethoxy-3-[4-[2-oxo-2-[[5-(trifluoromethyl)pyrimidin-2-yl]amino]ethoxy]butanoyl]quinolin-4-one 1-[4-fluoro-3,5-bis(trifluoromethyl)phenyl]-3-pyrrolidin-2-ylpropan-1-one N-[4-(trifluoromethoxy)phenyl]pyridine-3-carboxamide 3-azidooxy-2,6-dimethyl-4-(trifluoromethylsulfanyl)pyridine 1-(3,4,5-trimethoxyphenyl)ethanol 4-[5,6-dimethyl-2-(1H-pyrazol-5-yl)thieno[2,3-d]pyrimidin-4-yl]-N'-propan-2-ylpiperazine-1-carbohydrazide 2-(4-ethyl-3,5-difluorophenyl)pyridine 5-methoxy-2-[(4E,6Z)-3-(6-propan-2-ylpyridin-3-yl)nona-1,4,6,8-tetraen-2-yl]phenol 4-methyl-3,5-disulfobenzenediazonium 2-chloro-4-(2,6-difluorophenyl)-5-[(Z)-hydroxyiminomethyl]-1H-pyrimidin-6-one 3-(4-bromothiophen-2-yl)-4H-1,2,4-oxadiazol-5-one 4-[(E)-4-[1-(3,4-difluorophenyl)ethylsulfanyl]but-2-enimidoyl]phenol;1,3-dimethoxypropane 2,6-dichloro-3,5-dimethoxybenzenecarbothioamide 3-[(4-methoxyphenyl)methyl]-5,6,7,8,9,10-hexahydrocycloocta[d]pyridazine 2-[6-(ethylamino)pyridine-3-carbonyl]hexanamide 1-methyl-3-[4-(trifluoromethyl)phenyl]indole 1-(4-chlorophenyl)-3,5,6,7,8,9-hexahydropyrazolo[4,3-c]quinoline-4-carbonitrile 1-[4-(2,6-difluorophenyl)-3-methylpiperazine-1-carbonyl]-7H-pyrrolo[3,2-c]pyridin-4-one (2S)-N-[1,3-bis(2-methoxyphenyl)propan-2-yl]-2-propoxybutanamide 7-bromo-1,2,3,4-tetrahydronaphthalene-2-carboxamide 7-bromo-5,6,8,9-tetrahydrocyclohepta[b]pyridine;ethane 6-(4,5-dihydrobenzo[g][1]benzothiol-2-yl)-4-phenoxycyclohexa-1,3-diene-1-carboxylic acid 4-amino-N'-(cyclopropylmethyl)benzenecarboximidamide 2-(4-azidophenyl)ethanesulfonic acid N-[2-(4-phenylpiperazine-1-carbonyl)thieno[3,2-b]pyridin-7-yl]naphthalene-1-sulfonamide [4-(6-fluorospiro[2H-pyrrolo[1,2-a]pyrimidine-3,4'-piperidine]-1'-yl)phenyl]-methoxyazanide N-[4-(carbamoylsulfamoyl)phenyl]-2,4,6-trimethyl-N-phenacylbenzenesulfonamide 2-(1H-indazol-3-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 2-(5-azidoindol-1-yl)quinoline [4-[4-(5-chloro-2H-pyridine-1-carbonyl)phenyl]piperazin-1-yl]-[4,7-difluoro-5-(hydroxymethyl)-3-nitro-6,8-dihydro-5H-1,7-naphthyridin-7-yl]methanone;4-ethoxy-N-methylaniline 2-amino-N-(cyclohexa-1,3-dien-5-yn-1-ylmethyl)-4-[(5E,7Z)-2-ethenylnona-1,5,7-trien-3-yl]-5H-pyrrolo[2,3-d]pyrimidine-6-carboxamide 2-[3-(1,5-dimethylpyrazol-4-yl)pyrrolidin-1-yl]-N-(2-methoxyethyl)ethanamine N-[5-[[(Z)-1,4-diaminobut-2-enylidene]amino]pentyl]-5-[ethyl(propan-2-yl)amino]pyrazine-2-carboxamide 4-[[1-(4-chlorophenyl)cyclohexyl]methoxy]-1H-triazole-5-carboxylic acid 1-[6,8-difluoro-3-[2-hydroxyethyl(methyl)amino]quinolin-4-yl]-4-(4-hydroxyphenyl)piperidine-4-carbonitrile 2-[(5R,10bR)-7-methoxy-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-6-bromophenol 2-[4-(3,6-dihydro-2H-pyran-5-yl)-1H-pyrazole-5-carbonyl]-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-1-carboxylic acid N-[2-[(4,6-diamino-1,3,5-triazin-2-yl)oxy]ethoxy]-4-ethenoxybutanamide 4-[3,5-difluoro-2-(2H-tetrazol-5-yl)phenyl]-1H-indole N-methyl-1-(4-propan-2-yloxyphenyl)pentan-3-amine [6-hydroxy-3-(piperidine-1-carbonyl)-2H-indazol-5-yl]-(5-methoxy-1,3-dihydroisoindol-2-yl)methanone N-(3,5-dimethylphenyl)-2-[4-fluoro-2-(methoxymethyl)pyrrolidin-1-yl]acetamide N-[4-(4-oxo-4aH-phthalazine-1-carbonyl)phenyl]pentanamide 2-(3-methylbutanoyl)-7-[(4-phenyl-1,3-thiazol-2-yl)carbamoyl]-5,6-dihydropyrrolizine-1-carboxylic acid 2-(azidomethyl)-3,4,5-trichloropyridine N-[(3,5-dimethoxyphenyl)methyl]-1H-pyrazolo[4,3-d]pyrimidin-7-amine 5-[2-(4-fluorophenyl)hydrazinyl]pyrimidine-2,4-diamine [7-bromo-2-[3-(2-methylphenoxy)phenyl]pyrazolo[1,5-a]pyrimidin-5-yl]methanol [3-[2-(8-hydroxyquinolin-7-yl)imidazol-1-yl]propanoylamino]urea 2-amino-1,3-dihydroindene-2-carboxamide;ethane 1-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[2-[(4R)-4,6-diaminopyrimidine-5-carboximidoyl]hydrazinyl]naphthalen-1-yl]urea 4-ethyl-N,2-dimethoxy-5-phenylaniline 1-(4-methoxyphenyl)-2-[3-(5,7,8,10-tetrazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,9,11-hexaen-13-ylsulfanylmethyl)phenyl]ethanethiol N-(1H-benzimidazol-2-ylmethyl)-3,7-dimethyl-4-oxophthalazine-6-carboxamide (5Z)-2-(4-bromophenyl)imino-5-[[3,6-dibromo-1-(naphthalen-1-ylmethyl)indol-2-yl]methylidene]-1,3-thiazolidin-4-one 1-(6-hydroxy-3,4a,5,7,8,9b-hexahydro-2H-pyrido[4,3-b]indole-4-carbonyl)pyrazole-3-carboxylic acid 2,4-dichloro-3,5,6-trideuterio-N-[dideuterio-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(methyl)amino]methyl]benzamide 2-ethoxy-7,8-dimethylanthracene 2-[(E)-[4,5-dichloro-3-(4-hydroxyphenyl)iminospiro[1H-indole-2,4'-piperidine]-6-ylidene]methyl]benzoic acid 4-[(3R)-1-[2-(dimethylamino)pyrimidine-5-carbonyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one 3-methyl-N'-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-ylmethoxy)phenyl]butanimidamide (E)-4-[2-[[3-[(Z,1S)-1-aminobut-2-enyl]cyclopentylidene]methoxy]-5-bromophenyl]-N-[3-chloro-2-fluoro-6-methyl-5-(trifluoromethoxy)phenyl]-2-hydroxyiminobut-3-enamide N-[3-(2,4-diaminopyrimidin-5-yl)phenyl]methanesulfonamide N-azido-4,5,6-triphenyl-1H-benzimidazol-2-amine 4-amino-6,8a-dimethyl-3,5,6,7-tetrahydro-1H-quinazoline-2-thione 4-(2-chlorophenyl)-5-methylhexane-1,3-diamine 1-(3,5-difluorophenyl)-N-[4-methyl-3-(methylamino)phenyl]sulfonylcyclopropane-1-carboxamide [(2R)-4-(2,4-dichlorophenyl)sulfonyl-2-(3-ethoxy-5-propanoylphenyl)piperazin-1-yl]-(6-imidazol-1-ylpyridin-3-yl)methanone N-(diaminomethylidene)-5,6,7,8-tetrahydro-1H-isoquinoline-4-carboxamide 3-[2,5-dimethyl-1'-(pyridine-3-carbonyl)spiro[indole-3,4'-piperidine]-6-yl]propanoic acid;2,2,2-trifluoroacetic acid 2-azidooxy-5-bromo-N,3-dimethylaniline [[2-[4-chloro-3,5-dimethyl-N-(4-sulfobutyl)anilino]acetyl]amino]carbamodithioic acid 3-chloro-6,8,9-trifluoro-7-(4-methylphenyl)dibenzothiophene N-[(3,5-dimethylphenyl)methyl]-2-oxo-3H-1,3-benzoxazole-7-carboxamide 2-[3-(1,3-benzodioxol-5-yl)propanoyl]-N-hydroxy-4-methylcyclohexa-2,5-diene-1-carboxamide (3S,4R)-1-benzyl-4-(2,6-difluorophenyl)pyrrolidine-3-carboxylic acid 2-[4,6-dichloro-1-(3-methoxyphenyl)benzimidazol-2-yl]-7,9-difluoro-3,5-dihydro-2H-[1,3]oxazolo[3,2-a]quinazoline 4-(3,6-dihydro-2H-pyran-5-yl)-1H-pyrrolo[2,3-b]pyridine [2,3-bis(4-fluorophenyl)quinoline-6-carbonyl]oxidanium 2-[4-(1H-indole-3-carbonyl)piperazin-1-yl]-N,N-dimethylacetamide 6-methoxy-3H-[1]benzothiolo[2,3-b]pyrazine 4-[3-(difluoromethyl)phenoxy]-N-[(2S,3R,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]benzamide N-[4-(2,6-difluorophenyl)pyridin-3-yl]-1H-benzimidazole-2-carboxamide 4-(5-aminopentan-2-yl)-N'-[3-chloro-4-(methanesulfonamido)phenyl]-1,2,5-oxadiazole-3-carboximidamide;hydrochloride 1-(5,6-dimethyl-2H-thiopyran-3-carbonyl)pyrrolidine-3-carboxylic acid 2-[3-[(4-chlorobenzoyl)amino]-1-methoxycarbonylindole-5-carbonyl]propanedioic acid 4-[2,3-difluoro-4-(4-methoxyphenyl)phenyl]-1H-triazole-5-carboxylic acid 1-(1,3-benzodioxol-5-yl)-N-[[2-chloro-4-(trifluoromethoxy)phenyl]carbamoylamino]formamide (1-methylindazol-4-yl)-[5-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]oxyspiro[3,4-dihydrochromene-2,4'-piperidine]-1'-yl]methanone 3-[1-(4-ethylphenyl)-4,5-dimethoxyindole-2-carbonyl]-3a,7a-dihydro-3H-indol-2-one [4-(dimethylamino)phenyl]sulfanium;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide 2-[1-(5-chloro-6-oxo-4-phenylpyrimidin-1-yl)propan-2-ylamino]benzonitrile N-[(3-fluorophenyl)methyl]-3-hydroxybutanamide (5Z)-3-[2,6-dichloro-4-(trifluoromethylsulfonyloxy)phenyl]-5-[(1,5-diphenylpyrazol-3-yl)hydrazinylidene]-2H-1,2,4-triazin-6-amine 4-azidooxysulfanyl-3,5-dimethyl-1H-pyrazole 3,4-bis[(2-methylpropan-2-yl)oxycarbonylamino]benzenesulfonic acid 2-(4-nitrophenyl)sulfonyloxyacetic acid 4-azido-2,6-ditert-butylphenol 1-(3-aminopyrrolidin-1-yl)-2-[6-(4-methoxyphenyl)imidazo[1,5-a]pyridin-8-yl]ethanone 5-(4,6-diphenyl-1,3,5-triazin-2-yl)-N-[3-methoxy-4-(2-pyridin-2-ylethoxy)phenyl]furan-2-carboxamide 2-[1'-(thiophene-3-carbonyl)spiro[4,7-dihydropyrano[4,3-c]pyrazole-6,4'-piperidine]-3-yl]acetamide 2-[2,4-dichloro-5-(trifluoromethyl)phenyl]cyclopropane-1-carboxamide 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]-6-[(E)-pent-3-enoxy]-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 2,3-bis(ethoxycarbonyl)naphthalene-1-carboxylate 2-[5-(3-chlorophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-N-methoxyacetamide 5-[4-fluoro-3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-amine 3-[4,6-bis(trichloromethyl)-1H-benzimidazol-2-yl]-7-chlorochromen-2-one (5Z)-5-[[4-(3,6-dihydro-2H-pyran-4-ylmethoxy)phenyl]methylidene]imidazolidine-2,4-dione (2S)-1,4-dibenzylpiperazine-2-carboxylic acid N-(2,4-dimethylpent-1-en-3-yl)-5-[1-(pyridin-3-ylmethylamino)ethenoxy]pyrazine-2-carboxamide 5-methoxy-4-(1,3-oxazol-2-yl)cyclohexa-3,5-diene-1,3-dicarboxylic acid N-[2-[5,6-dimethoxy-1-(methylamino)hexan-3-yl]indazol-5-yl]-2-(4-fluorophenyl)acetamide 4-[(2E,3Z)-5-ethenyl-2-propylidene-1H-pyrrole-3-carbonyl]morpholin-3-one 7-(methylamino)-5-pyridin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxylic acid N-[2,4-dinitro-6-(2-phenylethylamino)phenyl]formamide 3-[(3S,4R)-1-benzylpyrrolidin-3-yl]oxypyridine N-(2,3-dihydropyridin-6-ylmethyl)-1-[5-(2-hydroxyethoxy)-2,3-dihydro-1H-inden-4-yl]methanesulfonamide ethane;1-methylpyrene;prop-1-ene 4-[(3S)-1-(3-chlorobenzoyl)piperidin-3-yl]-2-[1-(thiophene-2-carbonyl)pyrrolidin-3-yl]-1H-pyrimidin-6-one 2-(1,4-dioxan-2-yl)-6-methoxyaniline 6-[1-(benzylamino)ethyl]-2,3,4a,5-tetrahydropyrano[3,2-b]chromene-4,8-dione [4-(3,3a,4,5,6,7a-hexahydro-1H-cyclopenta[c]pyridin-2-yl)cyclohexanecarbonyl]-(4-aminophenyl)azanium 4-[(Z)-3,3-dimethylbutylideneamino]-2-[[2-[(3E)-hexa-1,3,5-trien-3-yl]-5-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazole-3-carbonyl]amino]benzoic acid 5-chloro-N-[6-(5,7-dimethylpyrrolo[2,3-b]pyrazin-1-yl)pyridin-3-yl]-4-fluoro-2-(oxan-4-ylsulfanylamino)benzamide 2-(3,4-dimethoxyphenyl)ethanamine;1-fluoro-3,5-bis(trifluoromethyl)benzene 1-(benzenesulfonyl)-4,5-dihydroimidazole N-[4-(methoxyiminomethyl)phenyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 4-[(2,3-dichlorophenyl)methyl]-5H-1,2,4-oxadiazole 2-[(6R)-2,6-dimethylmorpholine;(1R,4S)-3-fluoro-9-oxo-2-oxatricyclo[8.5.0.03,7]pentadeca-3(7),4,10-trien-5-carbonyl]-2,3,4,6,7,8,9,10,11,12-octahydro-1H-phenanthrene-17-carboxamide 2-[(3R)-6-chloro-3-methyl-2,4-dihydrochromen-3-yl]acetic acid 3-(2,2-dimethylpropanoyl)-4-hydroxy-6-(7-hydroxynaphthalen-1-yl)pyran-2-one 6-[3-(difluoromethoxy)azetidine-1-carbonyl]spiro[2H-indole-3,4'-piperidine]-1-one 6-(2,3-dihydro-1H-pyrrolo[1,2-a]benzimidazol-7-yl)hexan-1-amine 5-[(3,5-dioxo-1,2,4-triazolidin-1-yl)methyl]-N-methylthiophene-3-sulfonamide 2-[(6-bromonaphthalen-2-yl)methylidene]propanedinitrile 2-chloro-4-[(5-methyl-3,4-dihydropyrazol-2-yl)methyl]pyridine 1-azido-3,5-dimethylindole-2,4-dione 2-(3-azidophenyl)sulfonyl-1,4-dimethoxybenzene 7-(1,4-dithiepan-2-yl)-3-ethyl-1H-quinazoline-2,4-dione 3-(N-(4-bromo-2,5-dimethylphenyl)-4-hydroxyanilino)propane-1,2-diol 1-[2,5-difluoro-4-(2-methylphenyl)phenyl]piperidine 1-(4-benzylphenyl)-5-(4-bromobutyl)-4-methoxypyrazole (6S,11aS)-3-methylsulfanyl-8-oxo-7,9-dihydro-6aH-pyrrolo[2,1-c][1,4]benzodiazepine-11-carbonitrile (4R)-4-[3-(1,2,4-triazol-1-ylmethyl)phenyl]oxan-2-one N-[3,5-bis(trifluoromethyl)phenyl]-4-methoxyaniline (2R)-5,10,11-trihydroxy-9,12-dioxo-N-propyltricyclo[8.4.0.03,7]tetradeca-1(14),6,10,12-tetraene-15-carboxamide [3-[(3S,5R)-2,2-dimethyl-4,4-bis(phenylmethoxycarbonylamino)cyclobutyl]-1H-indol-7-yl]methanesulfonate 1,2-dibromo-4-(3-chloroethoxy)benzene;ethane 3-(1-azidoethyl)-5,6-difluoro-2H-indazole 6-N-[1-(4-fluorophenyl)ethyl]-4-N-(3-nitropyridin-2-yl)pyrimidine-4,6-diamine [6-(2,3-dimethylcyclopropyl)pyrazin-2-yl]carbamic acid N-[4-fluoro-2,6-di(propan-2-yl)phenyl]-2-methoxy-3H-1-benzofuran-6-sulfonamide 5-[2-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]pyrimidine 4-[(E)-2-[5-[[3,6-bis(4-methylpiperazin-1-yl)-4H-pyridine-3-carbonyl]amino]pyrazin-2-yl]ethenyl]benzoic acid 4-[5-fluoro-7-hydroxy-6-(2,2,2-trichloroethoxy)quinolin-8-yl]sulfanylphenol (3R)-4,4-difluoro-1-[6-(1H-pyrazol-5-ylamino)pyrimidin-4-yl]piperidine-3-carboxylic acid 4-(8,9-dichloro-5-hydroxy-6-oxobenzo[c]phenanthridin-12-yl)benzaldehyde 4-bromo-2,5-dimethyl-N-(2-methylphenyl)-N-[4-(thiophen-2-ylsulfamoyl)phenyl]benzamide 4-(9H-fluoren-1-yl)-2,6-dimethylpyridine 3-[(4E)-2,4-dimethylhexa-1,4-dien-6-yn-3-yl]-5-fluoro-N-[1-[4-[4-[hydroxy(phenyl)methylidene]piperidine-1-carbonyl]phenyl]ethenyl]benzamide 3-(4-chloro-2,5-dimethylpyrazol-3-yl)-5-[5-(trifluoromethyl)pyridin-2-yl]oxybenzoic acid (2E,4Z)-N-(5-chloropyridin-2-yl)hepta-2,4-dien-7-ynamide N-[3-(4-cyanophenyl)propyl]-2,6-difluoroaniline;cyclopentanamine 2-[(1R,5S)-3-[(4,6-dioxo-1H-1,3,5-triazin-2-yl)amino]-9-azabicyclo[3.3.1]nonan-9-yl]-N-methyl-N-phenylacetamide N-(3,4-difluorophenyl)-1H-indole-2-carboxamide 2-[4-(4,4-dimethylpiperidin-1-yl)-5-[5-[2-(4-fluoro-2-methoxyphenyl)ethoxy]pyridin-3-yl]-2-methylpyridin-3-yl]acetaldehyde;2-methoxyethanol 5-chloro-2-fluoro-4-[(3S,4R)-1,1,3-trimethylpiperidin-4-yl]oxyaniline (2R)-N'-(4,6-dichloro-1H-indazole-3-carbonyl)-3-fluorospiro[2.5]octane-2-carbohydrazide [6-carboxy-5-(trifluoromethyl)pyridin-3-yl]azanium 2-(4,4-diethoxycyclohexa-1,5-dien-1-yl)sulfanylphenol 3-[1-azido-2-(4-methoxyphenyl)ethyl]pyridine 1-(3,6-dibromocarbazol-9-yl)-5H-pyrazolo[3,4-d]pyrimidin-4-one 3-amino-2-hydroxybenzenesulfonic acid N-[(2E,4Z)-hexa-2,4-dien-3-yl]benzamide N-(4,5-dihydropyrimidin-2-yl)-3H-benzimidazole-5-carboxamide 1-[4-(aminomethyl)cyclohexyl]-2,2,2-trifluoroethanone;5-chloro-6-N-(3-methoxypropyl)-2H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 6-[4-(difluoromethoxy)phenyl]-N-[3-fluoro-5-[2-(methylamino)ethylcarbamoyl]thiophen-2-yl]pyridine-3-carboxamide 6-bromo-N-[5-(2,4-dimethylphenyl)sulfanyl-1H-indazol-3-yl]-1-methoxyindole-2-carboxamide 1-[4-(cyclohexylmethoxy)phenyl]-2,4-difluorobenzene N-(3,4-difluorophenyl)-1-methyl-2-[3-(trifluoromethoxy)pyridin-2-yl]cyclopropane-1-carboxamide 5-[6-(1H-pyrazol-4-yl)-2-[3-(trifluoromethoxy)phenyl]pyrimidin-4-yl]-2,3-dihydrothiophene-3-carboxamide 3-[2,4-dihydroxy-6-(oxan-4-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile (3S)-6-bromo-2,3-dimethyl-4-oxo-3H-pyrido[3,2-d]pyrimidine-5-carboxylic acid 4-[3-[5-[(2,6-difluorophenyl)methoxy]pyridin-3-yl]-1,7-thia-6-azaspiro[3.5]nonan-6-yl]but-2-ynoic acid N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2,3-dihydroindole-1-carboxamide 4-(2-butoxyethyl)-6-ethynylpyridine-3-carboxylic acid (2R)-1-(4-methoxyphenyl)sulfonylpyrrolidine-2-carboxamide 3-(3,4-dimethoxyphenyl)sulfanylpropylphosphane 1-[(Z)-1-ethylsulfanylprop-1-en-2-yl]-3,5-bis(trifluoromethoxy)benzene 2-[4-(2,6-dichlorophenyl)sulfanylpiperazin-1-yl]-3H-pyrido[3,4-d]pyrimidin-4-one 4-[2-[4-(4-aminophenyl)piperazin-1-yl]ethyl]oxan-4-ol [2-(2-chloro-4,5-difluoroanilino)pyrimidin-4-yl]-[3-hydroxy-3-(trifluoromethoxy)pyrrolidin-1-yl]methanone (3,4-dichlorophenyl)-[5-fluoro-2,6-bis(trifluoromethyl)pyrimidin-4-yl]methanone 2-(diethylamino)-N',N'-bis[(1S,3R)-3-methylcyclohexyl]benzohydrazide 1-[2,3-dimethyl-4-(trifluoromethoxy)phenyl]piperazine 4-bromobenzene-1,2,3-tricarbonitrile;4-ethyl-2H-benzotriazole [(2S)-2-fluoro-2-(4-phenylmethoxyphenyl)ethyl]carbamic acid 6-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]spiro[3.4]octane-8-sulfonamide N-[1-[5-(cyclohexylmethylamino)pentanoyl]piperidin-4-yl]-2,4-difluorobenzamide N-[5-methoxy-4,6-di(propan-2-yl)pyrimidin-2-yl]-2H-pyrimidin-1-amine 3-[1,2-bis(4-fluorophenyl)ethyl]-5-chloro-2-(2-methoxy-6-propan-2-ylpyridin-3-yl)pyrimidin-4-one 1-azidosulfanyl-3-phenylpropane-2,2-dithiol 2-(1H-indazole-3-carbonylamino)thiophene-3-carboxylic acid 7-[(4,5-dimethyl-1H-pyrazol-3-yl)diazenyl]naphthalene-2-sulfonic acid N-[2-(3,5-dimethyl-1,2-oxazol-4-yl)propan-2-yl]-N'-[(4R)-6,8,9,10-tetrahydro-5H-imidazo[1,5-d][1,4]benzoxazepin-4-yl]oxamide;2,2,2-trifluoroacetic acid 1-[2-(4,5,6,7-tetrahydro-3H-benzimidazol-5-yl)pyridin-3-yl]ethanone 2-methylsulfonyl-7,8-dihydropyrido[4,3-d]pyrimidine 4-[[1-[2-(2,6-dichlorophenyl)acetyl]azetidine-3-carbonyl]amino]benzenesulfinic acid 2-azidooxy-6-chloro-3,4-bis(phenylmethoxy)benzenesulfonic acid N-[[4-(furan-2-yl)thiophen-3-yl]methyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-5-carboxamide (6E)-6-[aminomethylidene-[2-[4-(diethylamino)phenyl]sulfanylquinolin-8-yl]hydrazinylidene]-N'-[1,3]benzothiazolo[5,6-b]indole-4-carboximidamide 5-amino-4-[4-(methylsulfanylamino)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 4-ethoxy-2,5-dimethyl-1H-imidazole;3-ethyl-5-(6-fluoro-2-methylbenzimidazol-1-yl)-N,N-bis(methylideneamino)aniline 2-[(5-oxopyrrolidin-2-ylidene)amino]benzenesulfonic acid N-[3-(4-bromophenyl)propyl]-2,7-diazaspiro[3.5]nonane-7-carboxamide;hydrochloride (2S)-2,5-diamino-3-[4-[2-oxoethyl(phenylmethoxycarbonyl)amino]benzoyl]sulfanylpentanoic acid 1-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-3-[4-fluoro-3-(trifluoromethyl)phenyl]urea 3-[[2-(4,5-difluoro-2-propan-2-yloxyphenyl)imidazol-1-yl]methyl]piperidine;dihydrochloride 2-[(5-chloroquinoline-8-carbonyl)amino]acetic acid (2S)-5-methoxy-1,2,3,4-tetrahydronaphthalene-2,7-disulfonic acid 1-ethylsulfonyl-6-(trifluoromethoxy)indole (E)-1,3-bis(2,4-dichlorophenyl)prop-2-en-1-one N-[3-hydroxy-1,5-bis(trifluoromethyl)pyrazol-4-yl]acetamide 2-[5-chloro-6-(4-fluoro-3-methylphenyl)pyrimidin-4-yl]oxy-N-ethylethanamine 1-cyclopropyl-4-methylidene-7,8-dihydroquinoline 4-[2-(5,8-difluoroquinolin-6-yl)ethyl]benzonitrile (1E,4Z)-3,5,8-trifluoro-2-(trifluoromethylsulfonyl)cyclonona-1,4,7-triene 3-(4-chlorophenoxy)-N-[[(6S)-2,5-dioxo-6-phenylpiperidin-3-yl]methyl]propane-1-sulfonamide 3-(5-azido-1H-pyrrol-2-yl)benzonitrile 6-[4-(4-fluorophenyl)piperazine-1-carbonyl]-4H-1,2,4-triazin-3-one (E)-3-[4-bromo-2-fluoro-5-(trifluoromethyl)phenyl]-2-sulfanylprop-2-enoic acid N-[(1R,5S)-6-oxobicyclo[3.2.0]heptanyl]-1-phenyltetrazole-5-carboxamide 2-[[4-(5-chlorocyclohexa-1,3-dien-1-yl)sulfonylmorpholine-2-carbonyl]amino]-1,3-thiazole-5-carboxamide 2-[4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxyphenoxy]-N-[(Z,3S)-6-hydroxy-7-oxohept-1-en-3-yl]acetamide N-[2-(3,4-dimethoxyphenyl)ethyl]-1-ethyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide 5-chloro-3-[4-[1-(2,6-difluorophenyl)ethenyl]piperazin-1-yl]-1,2-benzothiazole N-[4-(2,6-dimethylmorpholin-4-yl)phenyl]quinazoline-8-carboxamide 5-chloro-4-[1-(2,3-dihydro-1H-inden-5-yl)ethylamino]-1H-pyrimidin-6-one (Z)-3-[4-(5-oxo-1,4-dihydropyrazol-3-yl)phenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile 1-(2-azidooxyethyl)-3,7-dimethylpurine-2,6-dione 4-[3-(2,6-dimethylphenyl)phenyl]benzenethiol 1-(2,2-difluoroethyl)-N-[[3,4-difluoro-2-(2-fluoro-4-methylanilino)phenyl]-hydroxymethoxy]-3-(triazol-1-ylmethyl)cyclobutane-1-carboxamide 4-fluoro-N-[(3R)-6-nitro-2,3,4,9-tetrahydrocarbazol-1-ylidene]benzenesulfonamide 1-[2-(4-cyclobutylphenoxy)ethoxy]-3,5-difluorobenzene 2-(3-methylcyclopenten-1-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine (2E)-N,3-bis[4-[2-cyanoethyl(methylsulfonyl)amino]phenyl]-2-hydrazinylidenepentanamide 4-[5,6-bis(ethenyl)pyridin-3-yl]-2,3,5-trifluoroaniline N-[3-(5-chlorothiophen-2-yl)-4H-chromen-7-ylidene]hydroxylamine 1-(4-iodophenyl)ethanone;2,3,6-trimethyl-1H-indole [(2R)-2-benzylpyrrolidin-1-yl]-[5-(4-methoxypyrimidin-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]methanone [4-(6,7-dimethoxyquinoline-4-carbonyl)piperazin-1-yl]-[1-(hydroxymethyl)cyclopropyl]methanone N-[(2S,3R)-4-[[1-(azetidin-3-ylmethoxy)-7-fluoroisoquinoline-5-carbonyl]amino]-3-hydroxybutan-2-yl]carbamate (2R,4R)-1-acetyl-N-[3-fluoro-5-[2-(2-methoxypyrimidin-5-yl)pyridin-4-yl]oxyphenyl]-2-methylpiperidine-4-carboxamide N-[2-(3,4-dimethoxyphenyl)ethyl]-1H-benzimidazole-2-carboxamide;hydrochloride 2,4-dichloro-6-[(E)-2-nitroethenyl]phenol 2-[4-(2-fluoroethyl)cyclohexyl]oxy-3,5-dimethoxybenzonitrile 1-phenyl-4-[3,3,3-trifluoro-2-methoxy-2-(trifluoromethyl)propoxy]benzene 4-(2-bromo-N-pyridin-3-ylanilino)benzoic acid N-(2,4-dimethylphenyl)-N'-[(Z)-1H-indol-3-ylmethylideneamino]oxamide 3-[2-(3,4-dihydro-1H-isoquinolin-2-yl)pyrimidin-5-yl]-N'-hydroxybenzenecarboximidamide 2-[(4-fluorophenyl)methoxy]-5,8-dioxo-6,7-dihydronaphthalene-1-carboxylic acid N-[(2S)-3,3-dimethylbutan-2-yl]-4-[[4-(trifluoromethoxy)phenyl]carbamoylamino]benzamide N-[3-[2-(4-chloro-3-fluorophenoxy)ethylamino]propyl]-2,2-dimethylcyclohexane-1-carboxamide 2-(2,6-difluorophenyl)-4-(1H-pyrrolo[2,3-b]pyridin-6-yloxy)-2,3-dihydropyran-7-one 1-[3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethanesulfinate 7-[3-(2-benzylhydrazinyl)cyclobutyl]pyrrolo[2,1-f][1,2,4]triazin-4-amine (2R,3S)-1-(3H-benzimidazol-5-ylmethyl)-N'-[2-fluoro-6-(trifluoromethoxy)benzoyl]-2-methylpyrrolidine-3-carbohydrazide 1-[2-azido-6-(2,2-difluoropropoxy)phenyl]-N-methylmethanamine 2-[3-(4-fluorophenyl)sulfanylcyclohexa-1,5-dien-1-yl]propan-2-amine 3-[6-(1H-benzimidazol-2-yl)-9-methoxyxanthen-3-yl]-4-benzylphenol (Z)-3-amino-2-aminosulfanyl-N',N'-bis(2-methoxyethyl)but-2-enediamide;5-bromo-7H-pyrrolo[2,3-d]pyrimidine 2-(2,3-dimethyl-5-nitroimidazol-4-ylidene)acetic acid 3-[2-[4-(8-chloro-7-fluoroisoquinolin-4-yl)phenyl]ethynyl]cyclobutane-1,1-dicarboxylic acid 3-[(2Z)-4-oxo-4-[4-[4-(1,3-thiazolidin-4-ylmethoxy)phenyl]-1,3-thiazol-2-yl]buta-2,5-dienyl]benzamide N-(2,4-dimethylpentan-3-yl)-N,1-dimethyl-5-[1-methyl-5-[(Z)-prop-1-enyl]pyrazol-4-yl]imidazole-4-carboxamide N-[2-methyl-4-(trifluoromethoxy)phenyl]spiro[1,5,6,7-tetrahydropyrrolo[3,2-c]pyridine-4,1'-cyclopentane]-3-carboxamide 5-[3-methyl-4-(1H-pyrazol-5-yl)phenyl]-1,2,3,6-tetrahydropyridine (5E)-5-[[3,4-bis(ethenyl)phenyl]methylidene]-2-imino-1,3-thiazolidin-4-one 2-[3-(3-fluorophenyl)propanoyl]-4H-1,2,4-triazol-3-one 2-(7,8-dihydronaphthalen-1-ylmethoxy)benzoic acid 1-[2-hydroxy-3,4-bis(methylsulfanyl)-5-nitrophenyl]propane-1,2,3-trione 5-[1-(3,5-dimethyl-2H-pyridine-2-carbonyl)pyrrolidin-2-yl]-N-hydroxythiophene-2-carboxamide 3-methyl-1-[(3R)-6-pyridin-2-ylspiro[2H-indole-3,4'-oxane]-1-carbonyl]pyrrolidine-2-carboxylic acid (2R,4S)-4-hydroxy-N-[5-(2-methoxyphenyl)-3-methylpentanoyl]pyrrolidine-2-carboxamide N-[(3S,5R)-1-(8-chloroquinolin-6-yl)-5-methylpiperidin-3-yl]-2-ethoxypyridine-4-carboxamide N-(4-chlorobutyl)-N-cyclohexyl-1,2,3,5,6,7-hexahydropyrrolizin-8-amine [3-methyl-2,6-di(propan-2-yl)phenyl]-trioxidophosphanium 5-[3,6-difluoro-4-(2-phenylethoxy)-1H-indole-2-carbonyl]cyclohexa-1,5-diene-1-carbonitrile 2-(3,5-dihydro-2H-1,4-benzothiazepin-4-yl)acetaldehyde 4-[2-aminoethyl(methyl)amino]-5,6-dihydroquinazoline-8-carboxylic acid 2-[2,6-difluoro-N-(3-methylbut-2-enyl)anilino]acetic acid 4-[2,3-difluoro-4-(trifluoromethoxy)phenoxy]-2,6-difluorophenol (6R,9S)-2-amino-6-methyl-7,8-dihydro-5H-[1,4]thiazolo[3,2-a]pyrimidine-5-carboxylic acid;hydrochloride 1-(azidomethyl)-3-(trifluoromethoxy)benzene N-(4,6-dimethylpyrimidin-2-yl)-5-fluoro-3-hydroxy-1H-indole-2-carboxamide N'-hydroxy-2-[methyl(pyridin-3-ylmethyl)amino]pyrimidine-4-carboximidamide 3-[(6E)-6-chloro-2,7-dihydrotriazolo[4,5-d]pyrimidin-5-yl]benzoic acid 2-(4,6-diamino-1,3,5-triazin-2-yl)benzenesulfonic acid (5E)-2-(4,7-dihydrotriazolo[1,5-a]pyrimidin-6-yl)imino-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidin-4-one 2-(4-hydroxyphenyl)-N-[[1-methyl-5-(trifluoromethoxy)pyrazol-3-yl]methyl]acetamide 1-azidooxy-2,3-dichloro-4-(4-propan-2-ylphenyl)benzene 2-methyl-4-[5-(6-phenoxypyridine-3-carbonyl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]-1H-pyrimidin-6-one ethane;5-[(4-ethylphenyl)sulfanylamino]-2,4-difluoro-N-methylidenebenzamide 1-[(6R)-7-chloro-2,4,5,6,11,12-hexahydro-3H-cyclopenta[c][1]benzazocin-10-yl]ethanone 4-amino-6-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-isocyanopyridine-3-carboxylic acid (5Z)-5-[[1-(2,4-dimethylphenyl)pyrrol-2-yl]methylidene]-3-(3-phenoxypropyl)-1,3-thiazolidine 2,4-bis(3-chlorophenyl)pyrrole-1,3-dicarboxylic acid (2Z)-N'-[1,3-bis(4-ethoxyphenyl)-5-methylsulfonylpyrazol-4-yl]-2-hydroxyiminopropanimidamide 2-[(6Z)-6-[3,4-difluoro-5-[3-methyl-2,6-dioxo-1-(triazin-4-yl)pyrimidin-4-yl]oxyphenyl]iminohexanoylamino]ethylcarbamic acid 1,2-dichloroethane;N'-[(E)-[4-(dimethylamino)phenyl]methylideneamino]-N-(pyridin-4-ylmethyl)oxamide 3-[4-(cyclopropylmethoxy)anilino]-N-[(2R,5S)-1-ethyl-5-(hydroxycarbamoyl)piperidin-2-yl]pyrazine-2-carboxamide 1-aminosulfanyl-4-[4-ethenyl-2,5-dimethyl-3-[(Z)-prop-1-enyl]pyrrol-1-yl]butane-2,3-dione 3-[(2E)-2-[[4-chloro-5-methoxy-2-(2H-tetrazol-5-yl)phenyl]methylidene]hydrazinyl]benzenesulfonamide 2-[4-(3,3-difluoroazetidine-1-carbonyl)phenoxy]-5H-pyrrolo[3,4-b]pyridin-7-one;ethane N-benzyl-3,4-difluoro-2-(methanesulfonamido)benzamide 6-[4-(6-methylpyrimidin-4-yl)piperazine-1-carbonyl]-5H-pyrazolo[1,5-a]pyrimidin-4-one 2-(5-ethyl-3,4-dihydro-2H-chromen-6-yl)-7H-purine N-[5-[4-fluoro-3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]cyclobutanecarboxamide 4-(7-chloroquinolin-4-yl)piperazine-1-carboxylate 2-(3,4-dihydropyridin-6-yl)-2-phenylmethoxyacetonitrile 5-cyclopentyl-N'-[(2,3-dichlorophenyl)methyl]-4-ethynylimidazole-1-carboximidamide 4-[5-chloro-2-[(E)-6,7-dimethyloct-1-enoxy]phenyl]benzenesulfonamide 1-[6,9-dimethyl-3-(4-propanoylphenyl)-2H-furo[2,3-h][3]benzazepin-7-yl]-3-hydrazinylurea 1-[2,6-di(propan-2-yl)phenyl]-4H-pyrazole 1-cyclopropyl-2-[3-(hydroxymethyl)phenyl]sulfonylethanone (2S,3R)-2-N-[4-cyclobutyloxy-6-(trifluoromethyl)pyridin-3-yl]pyrrolidine-1,2-dicarboxamide N-[2,2-dimethyl-3-(4-oxohexanoylamino)propyl]naphthalene-1-carboxamide 2-[4-amino-6-oxo-1-(4-phenoxyphenyl)pyrimidin-5-yl]oxy-N-azidoacetamide 2-(1H-indol-3-yl)-N-[5-methoxy-2-methyl-4-oxo-7-(2,4,6-trifluorophenoxy)pyrido[2,3-d]pyrimidin-3-yl]acetamide N-[(E)-4-azidobut-3-enyl]-2,3-dihydropyrido[3,2-b][1,4]oxazine-6-carboxamide 4-[7-[(E)-2-aminoethenyl]quinazolin-2-yl]benzene-1,3-diamine 2-[2,4,6-trimethyl-N-[(3-nitrophenyl)methyl]anilino]acetamide 1-[(4aS,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]oxazin-1-yl]-3-(2,6-diethoxyphenyl)propan-1-one 1-cyclopentyl-4-(6,7-dichloropyrido[2,3-d]pyrimidine-2-carbonyl)piperazin-2-one [4-(1,3-benzothiazol-2-yl)-7-amino-3H-benzimidazol-5-yl]-morpholin-4-ylmethanone N-ethyl-3,5-dimethoxy-N'-[(Z)-4-(4-methylphenyl)pent-2-en-2-yl]sulfanylbenzenecarboximidamide 2-[4-methylsulfanyl-6-oxo-2-(2-phenylethylsulfanyl)-1H-pyrimidin-5-yl]-N-(2,2,2-trifluoroethyl)acetamide N-cyclohexyl-3-(trifluoromethoxy)benzenesulfonamide 2-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxylic acid N-[2,4-difluoro-3-(morpholine-4-carbonyl)phenyl]-1H-pyrrolo[2,3-b]pyridine-5-sulfonamide (1S,2S)-2-[5-methyl-4-(piperidine-4-carbonylamino)pyrazol-1-yl]cyclopentane-1-carboxylic acid 4-azido-3,5-bis(2H-tetrazol-5-yl)benzenesulfonic acid 4-[3-(4-bromophenyl)-2H-pyrazolo[3,4-b]pyridin-5-yl]-N-methylaniline N'-[2-[7-bromo-3-[3,4-dichloro-1-(2-methylpropoxy)butan-2-yl]iminobuta-1,4-dien-2-yl]pyrimidin-5-yl]-N-ethylethane-1,2-diamine 2-methoxyimino-2-[3,5,6-trichloro-4-[(4-phenoxyphenyl)diazenyl]pyridin-2-yl]acetamide 5-[3-(methoxymethyl)phenyl]pyrimidine N-[6-(2,4,5-trifluorophenyl)imidazo[1,2-a]pyridin-3-yl]benzamide 3-chloro-2-methylsulfonyl-4,7-dihydropyrazolo[1,5-a]pyrimidine 1-cyclopropyl-2-ethyl-6-(3-methoxyphenyl)indole 1,3-dimethyl-N-(5-methylpyridin-2-yl)-4-[6-(4-methylpyridin-2-yl)pyridin-2-yl]imidazol-2-imine 1-[(2-phenylimidazo[1,2-a]pyridin-3-yl)methyl]pyrrolidine-2-carboxamide 3-[2-(4-methylphenyl)propanoyl]-2,3a,7a-tetrahydroindole-1,6-dione 2,5-dichloro-N-[(1-methylindazol-3-yl)amino]benzamide 1-[3-ethylsulfonyl-5-(trifluoromethyl)pyridin-2-yl]-6,8,13-triazatricyclo[7.4.0.02,7]trideca-2,4,6-trien-12-one 4-methyl-5-(1H-pyrazol-3-yl)pyrrolo[3,2-d]pyrimidine 1-[(3Z)-4,5-difluorohexa-1,3,5-trien-2-yl]-3-methoxy-5-propan-2-ylbenzene 2-(3-cyclopentyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-8,3'-pyrrolidine]-1'-yl)-N,N-dimethylacetamide;2,2,2-trifluoroacetic acid 6-[1-(2,3-dimethylcyclohexyl)piperidine-4-carbonyl]pyridine-3-carbonitrile 5-phenyl-7H-furo[3,4-c]pyridine-6-carbonitrile N-(4-chlorobutyl)-2,4,6-trimethyl-N-phenylbenzenesulfonamide (3R,4S)-1-ethyl-N'-[3-methoxy-2-(methylideneamino)phenyl]sulfonyl-4-methylpyrrolidine-3-carbohydrazide 1-benzylsulfanyl-3-N,3-N,4-trimethylnaphthalene-2,3-diamine ethane;N-methyl-2-methylidenebutanamide;(E)-1-[3-(propylideneamino)-4,5-dihydro-1H-indol-7-yl]but-1-en-1-amine (1S)-1-[4-(4,5-dihydropyrimidin-2-yloxy)phenyl]ethanamine 3-[6-amino-5-(azepane-1-carbonyl)-4-hydroxycyclohexa-2,4-dien-1-yl]sulfanylbenzoic acid (E)-2-[4,5-dihydroxy-3-[4-[3-[4-[methyl(2-oxoethyl)amino]phenyl]propoxy]butoxy]oxolan-2-yl]oxy-N,N-dimethylacetamide 1-N',3-N-bis(4-chlorophenyl)benzene-1,3-dicarboximidamide [7-bromo-5-(4-chlorophenyl)thieno[3,2-b]pyridin-3-yl]methanol [4-[[(1S)-5-cyano-2,3-dihydro-1H-inden-1-yl]carbamoylamino]cyclohexylidene]azanium 4-(2,4-dihydroxyphenyl)-7-[6-(dimethylamino)pyridine-3-carbonyl]-8a-benzoyl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-2-one [7-(3,4-dimethylphenyl)naphthalen-2-yl]-(4-pyridin-4-ylpiperidin-1-yl)methanone (4-tert-butylphenyl)methanesulfonamide;2-phenylbenzenesulfonamide 5-cyclopropyl-4-(2,6-difluorophenyl)-1H-pyridazin-6-one 4-cyclopropyl-5-[2-hydroxyethyl(methyl)amino]-1H-pyrimidin-6-one 4-[(2R)-1,4-dioxaspiro[4.5]decan-8-yl]benzonitrile (4-azidooxypyridin-2-yl)-[3-[(E,4Z)-4-hydroxyimino-2-phenylbut-2-en-2-yl]pyrrolidin-1-yl]methanone 6,13-dibromophenanthro[9,10-d]pyrimidine;ethane 3-[(4-bromo-1,2,5-thiadiazol-3-yl)oxy]propane-1-sulfonic acid 4-(1,3-benzodioxol-5-yl)-2-[3-methoxy-5-[(2S,3R,5S,6R)-3,4,5,6-tetrahydroxyoxan-2-yl]phenyl]-5H-1,2,4-oxadiazol-3-one [2-(3,5-dimethylpyridin-4-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl]-piperidin-1-ylmethanone (E)-3,7,7-trifluoro-6-hydroxy-2-[5-oxo-1-[4-(2,3,5,6-tetrachlorophenoxy)butyl]pyrrolidin-2-yl]non-2-enoic acid 3-(4-chlorophenyl)-N'-hydroxybenzenecarboximidamide 5-ethenyl-2-methoxypyridine;N'-(2,4,6-trifluorophenyl)-1H-pyrazole-5-carbohydrazide 2-methyl-7-(naphthalen-1-ylmethylamino)quinoline-5,8-dione [5-(benzylcarbamoyl)-1H-pyrrol-2-yl]methyl-oxoazanium 2-[4-(1H-imidazol-5-ylmethyl)piperidine-1-carbonyl]-3,4-dihydro-1H-isoquinoline-6-carbonitrile;dihydrochloride 4-(8,13,14,15-tetrazatetracyclo[7.6.0.02,7.010,14]pentadeca-1(9),2,4,6,10,12-hexaen-16-yl)benzaldehyde 1-[5-[2-(6-methylimidazo[1,2-a]pyridin-3-yl)ethynyl]pyridin-2-yl]piperidine-4-carboxylic acid (6-cyclopentyloxypyridine-2-carbonyl)azanium 2-[[3-azidooxy-1-(pyridin-4-ylmethylamino)propan-2-yl]oxymethyl]phenol 2-[(Z)-[3-amino-4-oxo-5-(trifluoromethylsulfonyloxy)-1H-pyrrolo[3,2-d]pyrimidin-2-ylidene]methyl]benzenesulfonic acid 1-[5,6-bis(methylamino)pyridin-3-yl]sulfanylethanol (3,4-dimethylpiperazin-1-yl)-[5-iodo-7-methoxy-2-(oxan-4-yl)indazol-6-yl]methanone 2-[4-[(E)-1-amino-3-oxoprop-1-enyl]-6-fluoroquinolin-2-yl]oxyacetamide 4-chloro-2-(1,3-dihydroisoindole-2-carbonyl)phenolate (2E,5Z)-5-[[1-[[3-chloro-4-[(2-fluorophenyl)methoxy]phenyl]methyl]indole-7-carbonyl]hydrazinylidene]-N-hydroxyocta-2,6-dienamide (4R)-1'-benzyl-3-phenylspiro[5,7-dihydropyrazolo[3,4-b]pyridine-4,3'-indole]-2',6-dione 2-ethyl-5,7-dimethyl-3H-thieno[3,4-d]pyrimidine-4,6-dione N-[(4S)-1-methyl-6-oxo-7,8-dihydro-5H-naphthalen-2-yl]acetamide (E)-N,4,8-trimethyl-1-pyridin-2-yloct-6-en-5-imine 1,5-dimethyl-2-[[6-(phenylmethoxyiminomethyl)pyridin-2-yl]methylidene]-3H-pyridin-3-id-4-one;yttrium 3-[(2,6-dichlorophenyl)sulfanylamino]-4-methylbenzoic acid 5-bromo-2-[(4-methylphenyl)sulfanylmethoxy]benzoic acid 3-(5-tert-butylpyridin-2-yl)-4H-1,2,4-oxadiazol-5-one 7-[4-(3,5-dimethoxyphenyl)butyl]-2H-triazolo[4,5-b]pyridine 3-[5,6-bis(4-chlorophenyl)pyrazin-2-yl]benzenethiol (Z,3R)-4-azidooxy-N-ethyl-5,6-difluoro-2-methylidenehex-4-enamide N-[4-[(4S)-3-(cyclobutylamino)piperidine-1-carbonyl]phenyl]prop-2-enamide 1-(2-aminophenyl)sulfanyl-4,5-dibutoxyheptan-1-one (3R,5R)-2-[6-chloro-4-methyl-8-(trifluoromethylsulfonyloxy)quinolin-7-yl]-3,5-dimethylpiperazine-1-carboxylate 4-[[4,5-bis(ethenyl)imidazol-2-ylidene]amino]oxyaniline 3-amino-N'-(4-fluorophenyl)-2-oxo-6,7-dihydroquinoline-1-carboximidamide ethane;6-N-[2-(4-methoxyphenyl)ethyl]-5H-benzo[h]quinazoline-2,3,8-triamine N-(1,3-benzothiazol-5-yl)-3-[2,4-difluoro-6-[4-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]phenyl]oxetane-3-carboxamide 5-[3,5-dimethoxy-4-(trifluoromethyl)phenyl]-2-(1H-inden-1-yl)pyrazole-3-carboxylic acid 4-[5-(2,3-dihydro-1H-inden-2-yloxy)-6-propanoylpyrimidin-4-yl]piperazine-1-carboxylic acid (Z)-1,3-bis[2-hydroxy-5-(trifluoromethoxy)phenyl]prop-2-en-1-one [3-(2,6-difluorophenyl)-1,4,5,7-tetrahydropyrazolo[3,4-c]pyridin-6-yl]-(7H-purin-6-yl)methanone N-cyclohexyl-7-[2,4-dihydroxy-5-(3-methoxypropanoylamino)phenyl]-8-oxoimidazo[1,2-a]pyrazine-6-carboxamide 4-[2-(cyclohexylamino)ethoxy]benzamide 4-cyclopropyloxy-3-[5-(difluoromethyl)-1H-pyrazol-4-yl]-6-[4-(trifluoromethylsulfonyl)phenyl]pyridazine 2,3-diamino-N'-[(4-chlorophenyl)methyl]-1H-indole-5-carboximidamide;2-phenylacetaldehyde 1-(cyclopentylmethoxy)-4-ethynylbenzene;3-(3,5-difluorophenoxy)propanal 5-[(2R,3S)-3-hydroxybutan-2-yl]pyrazolo[1,5-a]pyridine-7-carbonitrile N-[4,7-dioxo-2-(3,4,5-trimethoxyphenyl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]naphthalene-1-carboxamide 1-[6-methoxy-3,3-bis(methylsulfanyl)cyclohexa-2,4-dien-1-ylidene]propane-2-thione 4-(2,3-dihydro-1H-inden-5-yl)-N-methylidenebenzamide;heptane;2-methoxyethanol 2-(2,6-dioxopiperidin-3-yl)-4-[[4-(trifluoromethoxy)phenyl]methylamino]isoindole-1,3-dione 4-(2,5-dimethoxyphenyl)benzaldehyde 4-(2-methoxyphenyl)sulfanyl-N-[3-(trifluoromethylsulfonylamino)propyl]benzamide N-(3,4-difluorophenyl)-1H-indazole-7-carboxamide (3R)-4,7-dioxo-5-(trifluoromethyl)-N'-[4-(trifluoromethyl)phenyl]spiro[1H-indole-3,4'-thiane]-2-carboximidamide 1,3-dicyclohexylpropan-2-ylbenzene;1,2,5-trimethyl-4-[(Z)-pent-2-en-2-yl]benzene 1-cyclobutyl-N,N-dimethyltriazolo[4,5-c]pyridine-7-carboxamide [3-(7-ethoxynaphthalen-1-yl)oxycyclohexa-2,4-dien-1-ylidene]phosphane 3-[4,5-bis(2-methoxyethyl)imidazol-1-yl]phenol [3-(1,2,4-triazol-1-yl)piperidin-1-yl]-(5H-pyrrolo[2,3-b]pyrazin-7-yl)methanone 2-[4-(4-fluorobenzoyl)piperidin-1-yl]acetaldehyde;3-hydroxyoxolane-4,5-dione 1-azido-4,6-diethylnaphthalene 5-(1,3-benzothiazol-2-ylsulfanylmethyl)-4-chloro-N-[2-[5-(trifluoromethoxy)cyclohepta-1,4,6-trien-1-yl]ethyl]-1,2-oxazole-3-carboxamide 4-[(6,7-dimethoxyquinazolin-2-yl)amino]phenol 4-[(Z)-(2,3-diethoxy-6-hydroxyphenyl)methylideneamino]piperazine-1-carboxylic acid 4-ethyl-N-[3-(3,4,5-trimethoxyphenyl)-1,2-oxazol-5-yl]thiadiazole-5-carboxamide 6-chloro-4-[2-methoxy-5-(1,3-oxazol-5-yl)phenyl]-2-sulfanylidene-1H-pyrimidine-5-carbonitrile (E)-N-[(2R)-butan-2-yl]-3-ethoxy-2-fluoro-3-pyridin-4-ylprop-2-enamide 2-[2,4-bis(phenylmethoxy)phenyl]-1-benzofuran 3-[5-(methylideneamino)-4,7-dioxo-1,6-naphthyridin-2-yl]benzamide 4-[4-[1,3-benzodioxol-5-ylsulfonyl(2H-tetrazol-5-yl)amino]phenyl]benzoic acid 1,3-dichloro-5-(2,4-difluorophenyl)benzene 3-ethyl-2,4-dimethoxyacridine N-(3-bromophenyl)sulfonyl-N,6-dimethylpyridine-2-carboxamide 1-ethyl-5-methoxycarbonylpyridine-3,4-dicarboxylic acid N-[(2E,4Z)-2,3-dimethylhepta-2,4,6-trienoxy]benzenesulfonamide;ethane N-(4-chlorophenyl)-5,7-dihydroxy-6-methyl-2-phenylchromene-4-thione N-[4-(8-chloro-2,6-dioxo-1H-purin-7-yl)phenyl]-1-[(3S)-pyrrolidine-3-carbonyl]piperidine-3-carboxamide [4-[3-chloro-5-(trifluoromethoxy)phenyl]piperazin-1-yl]methanimine 2-[(4-ethylpiperazin-1-yl)methyl]pyridine-4,7-dicarboxylic acid 5-(1H-indol-3-ylmethyl)-N-[4-[5-[2-[2-(methanesulfonamidomethyl)phenoxy]ethoxy]-2,3-dihydro-1H-inden-1-yl]phenyl]pyrimidine-2-carboxamide 5-hydroxy-1,4-dimethyl-3-[5-[(2S)-2-(4-nitrophenyl)propyl]thiophen-2-yl]pyridin-2-one 2-[4,6-bis(carboxymethoxy)naphthalen-1-yl]acetic acid 4-(2,6-dimethylphenyl)-5-iodo-1H-pyrimidin-6-one 3-methyl-2-[3-methyl-5-(trifluoromethyl)phenyl]butanamide 3-[4-hydroxy-2,6-dimethyl-N-(4-methylphenyl)sulfonylanilino]propanoic acid 5-(3,4-dihydroxyphenyl)-N-[1-(5-methylhexanoylamino)pentan-2-yl]-1H-imidazole-2-carboxamide 4-(7,8,9a,10a-tetrahydrophenothiazin-2-yl)aniline 4-[2-(8-methoxy-4-oxo-3H-quinazolin-2-yl)ethynyl]benzoic acid N-[1-(2,2-difluoroethyl)piperidin-4-yl]-3,4-dihydro-1H-quinolin-2-imine 6-chloro-3-[(Z)-2-(4-methoxyphenyl)propylideneamino]quinazolin-4-one 5-methoxy-N,2-diphenylaniline [3-(4-chlorophenyl)pyrrolidin-1-yl]-[5-methoxy-6-methyl-2-(methylideneamino)pyrimidin-4-yl]methanone 3-[(6,7-dimethoxyquinazolin-4-yl)amino]benzamide 3-(benzylsulfonylamino)-1,2,4-thiadiazol-5-amine 1-(2,5-dimethylphenyl)sulfonyl-3-[(4S)-4-(trifluoromethoxy)cyclohepta-1,6-dien-1-yl]pyrrolidine 4-N-[2-(3,5-dimethoxyphenyl)ethyl]-6-(4-nitropyrazol-1-yl)pyrimidine-2,4-diamine N-methyl-2-[(3S)-2-methylidenepyrrolidin-3-yl]imidazo[1,2-a]pyridin-6-amine (6R,7S)-3-[2-hydroxy-3-(4-propanoylanilino)propyl]-8-oxo-7-[(2-phenoxyacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid [[2-(2,3-dichlorophenyl)-5-methylpyrazole-3-carbonyl]amino]thiourea 1-(4-aminophenyl)-2,3-dicyclohexylguanidine N-[5-chloro-2,4-difluoro-3-[2-oxo-2-(3,4,5-trimethoxyphenyl)ethyl]benzoyl]propane-1-sulfinamide 2-(4-aminopiperidin-1-yl)-5,6,7,8-tetrahydronaphthalene-1,3-diol 2-(7,8-difluoro-1H-isoquinolin-4-yl)propan-1-ol [4-(2-methylbenzimidazol-1-yl)phenyl]urea 5-(2,4-dimethylphenyl)pentanethioamide 1-N,4-N-bis(2-pyridin-3-ylethyl)benzene-1,4-disulfonamide;methanol [2-(2-bromobenzoyl)phenyl]-(2,3,4-trichlorophenyl)methanone (6R,9S)-9-[4-bromo-2-(trifluoromethyl)phenyl]-1,3,8-triazaspiro[5.5]undecan-2-one 1-[4-hydroxy-3,5-di(propan-2-yl)phenyl]ethanone (3E)-5-ethyl-3,4-bis[hydroxy(phenyl)methylidene]oxolane-2,6-dione 5-[4-[2-(azetidine-1-carbonyl)morpholin-4-yl]phenyl]thiophen-3-amine 1-(4-chlorophenyl)sulfonylpiperidine;ethane 2-[2-(4-chlorophenyl)-7,8-dihydro-6H-pyrido[3,4-b]pyrrolizin-5-yl]acetic acid 2-chloro-5,6-dimethyl-4-pentan-3-ylpyrimidine 5-bromo-4-(2,6-dimethylmorpholin-4-yl)-1H-pyrimidin-6-one 4-cyclobutyloxy-2-ethenylpyrimidine 6-[5-fluoro-3-methyl-2-(1,1,2,2-tetradeuteriopropoxy)phenyl]imidazo[2,1-b][1,3,4]thiadiazole 2-(3-benzoylphenyl)-7,12b-dihydrobenzo[c]xanthen-12a-one 2-ethyl-4-(4-fluorophenyl)-1,3-thiazole 2-cyclohexylimino-5-[(4,6-diethoxy-1,3,5-triazin-2-yl)methylidene]-1,3-thiazolidin-4-one 2-[2-(2,4-dimethylphenyl)iminoethylidene]propanedioic acid 2-(2-azidophenyl)-N,N-diethylaniline [6-(4,5-dihydroimidazol-1-yl)naphthalen-2-yl]-(4-pyridin-3-ylphenyl)methanimine 4-(1-benzofuran-5-yl)-2-pyridin-4-yl-6-(5-pyridin-4-ylthiophen-3-yl)pyrimidine 1-[(Z)-5,6-diamino-2-ethyliminohex-3-enoyl]-N'-methyl-4-phenylpiperidine-4-carbohydrazide 4-chloro-1,6-diphenylpyrimidine 1-[4,5-dihydroxy-7-methoxy-2,6-bis(prop-1-ynyl)anthracen-1-yl]oxyperoxypropan-2-one 1-(3-methoxypropylamino)-4,8-dihydropyrazolo[4,3-e][2]benzazepine-7-carboxylic acid 4-azido-1-N,3-N-diethylbenzene-1,3-disulfonamide N-[1-(3,4-dichlorophenyl)ethyl]-6-fluoro-5-methanimidoylpyridine-2-carboxamide;3,3,4,4-tetramethylpentane 2,6-dichloro-N-(2-fluorophenyl)pyrimidine-4-carboxamide N-(4-chlorophenyl)sulfanyl-3-methoxyaniline 6-[4-(2,5-dimethylphenoxy)phenyl]-7-oxo-4H-thieno[3,2-b]pyridine-5-carboxylic acid N-(1-azidobutyl)-2-phenylethanimidate 3-[2,5-bis(trifluoromethyl)anilino]propanoic acid (4-bromophenyl)-[3,5-dibromo-2-methoxy-6-[[(E)-[(Z)-1-[2-[3-nitro-5-(trifluoromethyl)anilino]ethylideneamino]pent-2-en-4-ynylidene]amino]iminomethyl]phenoxy]methanol;ethane 3-methoxy-5-(2-morpholin-4-ylethylsulfamoyl)benzamide (5S)-2-(4-bromoanilino)-N-(3,4-dichlorophenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-(3,5-dichloropyridine-2-carbonyl)-1,4-benzoxazin-3-one (2-cyclopentylsulfanylcyclohexa-1,5-dien-3-yn-1-yl)benzene 6-chloro-3-[(4R)-2-oxo-4-propan-2-yl-1,3-oxazolidin-3-yl]-5-(trifluoromethoxy)pyridine-2-carbonitrile 4-tert-butyl-N,N-diphenylaniline N-(3,4-dimethylphenyl)-2-[[6-[(2-hydroxynaphthalen-1-yl)iminomethyl]pyridin-2-yl]methoxy]benzamide (Z)-4-N-[2-[difluoro(iodo)methyl]phenyl]-1-N-ethenylbut-3-ene-1,2,4-triamine N-(3-hydroxypropyl)-4-methoxy-6,7-dihydronaphthalene-1-carboxamide (2S,4R)-N'-[3-fluoro-4-[2-(5-methyl-1H-imidazol-4-yl)ethynyl]phenyl]-2-(4-fluorophenyl)-3,3,6-trimethylpiperidine-1-carboximidamide 1-[2-[(3E)-3,5-difluorohexa-1,3,5-trien-2-yl]phenyl]piperidine 2-(1,3-dioxoisoindol-2-yl)oxypropanedioate 3-[1-methylsulfonyl-5-(trifluoromethoxy)indol-2-yl]cyclopropane-1,1,2,2-tetracarbonitrile 1-[3-[2,3-bis(chloromethyl)phenyl]propylsulfonyl]-4-fluorobenzene (2Z,6S)-N-benzyl-7,8-dimethoxy-4-oxo-2-[(Z)-thiophen-3-ylmethylidenehydrazinylidene]-1,3-thiazinane-6-carboxamide 5-[2-(4-bromo-3,5-dimethylphenyl)acetyl]imidazolidine-2,4-dione (2R,6S)-5-(4-chlorophenyl)-2-(1H-indol-7-yloxymethyl)-1,3,6,7,8,9-hexahydropyrazolo[3,4-h]isoquinoline N-(3-fluorophenyl)-4,4a-dihydro-1H-quinazolin-2-imine 1-[4-[[6-(2,3-difluorophenyl)pyridine-3-carbonyl]amino]cyclohexyl]piperidine-3-carboxylic acid 4-(6,7-dihydro-1H-indole-2-carbonyl)-3,5-dihydro-2H-1,4-benzoxazepine-8-carbothioamide 5-[(1Z,3E)-2-phenylhexa-1,3,5-trienyl]pyridine-2,4-dicarbonitrile 1-[2-(4,4-difluoropiperidin-1-yl)phenyl]-3-methylidenecyclobutane-1-carbonitrile N-[3-(4-cyclopropyl-1,2,4-triazol-3-yl)phenyl]-5,6-dihydroquinoline-7-carboxamide 4-[4-(2-ethenoxyethylsulfanylamino)phenyl]-1H-pyrrole-3-carbonitrile 5-cyclohexyloxy-4,6-diphenylbenzene-1,2,3-tricarbonitrile 5-bromo-2,6-dichloro-N-(4-chlorophenyl)pyrimidin-4-amine 3-[6-[4-(6,7-dihydrodibenzofuran-4-yl)phenyl]pyridin-2-yl]benzonitrile 5-(furan-3-yl)-N',N'-dimethoxy-2-[6-(trifluoromethyl)pyridazin-4-yl]benzenecarboximidamide 7-bromo-6-(4-chlorophenyl)pyrazolo[1,5-a]pyrimidine (1S)-N,5-bis[2-[3-chloro-4-(trifluoromethoxy)phenyl]ethylamino]-4-methylsulfonyl-6,7-dihydro-2H-[1,3]thiazolo[5,4-c]pyridine-2-carboxamide 5-ethyl-4-[1-(5-fluoro-2-methoxyphenyl)propan-2-ylamino]-1H-pyrimidin-6-one 4-[(1R,2S)-5-benzylsulfanyl-2-ethylcyclohexyl]oxy-6-methylpyridine-3-carbonitrile (2S)-5,6-diamino-2-[[1-carboxy-3-phenylpropan-2-yl]carbamoyl]hexanoic acid 2-[(4S)-1-cyclopropylsulfonyl-3,4-dihydro-2H-quinolin-4-yl]acetic acid (4R)-1-[5-chloro-2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-4-(4-fluorocyclohexa-1,3-dien-1-yl)sulfonylpyrrolidin-2-one 5-[(3E)-hexa-1,3,5-trien-3-yl]sulfonyl-1-piperidin-4-yltriazole-4-carboxylic acid 2-azido-N,N-bis(2-fluorophenyl)benzamide 6-amino-3-(2-cyclopropylethynyl)pyrazine-2-carboxylic acid N-[(4-chlorophenyl)methyl]-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carboxamide (Z)-2,3-bis(ethenyl)-N'-[4-[2-(4-methoxyphenoxy)ethyl]phenyl]hex-5-enediamide 5-(4-aminophenyl)-3-N-[4-(methylcarbamoyl)cyclohexa-1,5-dien-1-yl]pyrazine-2,3-dicarboxamide (2-aminophenyl)-dimethoxyphosphanium 7-(3,4-dihydroxybutyl)-2-[[(1R,2S)-2-hydroxycyclohexyl]amino]-5H-pyrrolo[3,2-d]pyrimidine-6-carboxamide [(5R,7S)-1-methyl-3-phenyl-5,7-dihydro-4H-pyrazolo[3,4-c]pyridin-6-ylidene]-(4-pyrrolidin-1-ylphenoxy)methanol 1-(4-methylsulfanylphenyl)cycloheptane N-[3-(difluoromethoxy)phenyl]-2,4,6-trimethyl-N-prop-2-enylbenzenesulfonamide 2-methylsulfinyl-4-[(3R)-3-[[2-[2,2,2-trifluoro-1-hydroxyethyl(pyridin-2-ylmethyl)amino]acetyl]amino]pyrrolidin-1-yl]benzoic acid 7-(4-propylcyclohexyl)oxy-1,2-dihydronaphthalene 1-(5,6-diaminopyridin-2-yl)-3-[2-fluoro-4-[1-(trifluoromethyl)cyclopropyl]phenyl]urea 5-bromo-4-(1H-indol-3-yl)-N,2,5-trimethylhexanamide 5-methoxy-2,4,6,10b-tetrahydro-1H-isoindolo[2,3-a][2,8]naphthyridine 6-azidooxy-1H-phenanthro[9,10-c]pyridine 4-[3-(8,10-diazatetracyclo[7.6.0.02,7.011,15]pentadeca-1(9),2,4,6,11(15),12-hexaen-13-ylmethoxy)phenyl]butanoic acid 4-amino-6-[(Z)-N'-(1,3-dimethylimidazol-1-ium-2-yl)carbamimidoyl]pyridine-3-carboxylic acid N'-[(E)-1-(2,4-dihydroxy-6-methoxyphenyl)ethylideneamino]-N-octyloxamide 1-[5-bromo-2-(propylamino)phenyl]ethanone 2-[3-(dimethylamino)propoxy]-5-ethyl-7,8-dihydro-6H-naphthalene-1,6-diol 2-[5-ethylsulfonyl-6-[3-methyl-7-(trifluoromethyl)imidazo[4,5-c]pyridazin-2-yl]pyridin-3-yl]acetic acid [4-(1-ethoxy-2,3-dihydroindole-6-carbonyl)morpholin-3-yl]methanesulfonamide N-[6-(1H-pyrazol-5-yl)-1,3-benzothiazol-2-yl]formamide 2-[[4,4-difluoro-3-hydroxy-1-methyl-5-(methylideneamino)pentan-2-yl]sulfamoyl]benzoic acid 2-[6,8-dihydroxy-2-(4-methoxyphenyl)quinoxaline-5-carbonyl]oxyethanesulfonate 6,7-difluoro-2-methyl-3,5-dihydroimidazo[4,5-f]benzimidazole 4-amino-6-[(1E,3Z)-2-methylpenta-1,3-dienoxy]-N-propan-2-ylpyridine-3-carboxamide;chlorobenzene 2-(3,5-dimethylphenyl)-7-methoxy-9H-carbazole;ethane 4-methylsulfanyl-3-(2,3,5-trichlorophenyl)-1H-pyrazolo[3,4-d]pyrimidine 1-[4-(3,5-dimethylphenyl)piperazin-2-ylidene]-3-(4-methoxyphenyl)urea 5-azido-N,N-dimethyl-6-(2H-tetrazol-5-yl)naphthalene-1-sulfonamide 2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-2-yl)pyridine-3-carboxamide 2-(1,3-benzothiazol-6-yloxy)benzamide;methanamine 5-(3,6-dichlorocarbazol-9-yl)-5H-isothiochromeno[4,3-d]pyrimidine 2-(4-tert-butylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine N'-[(4E,6Z)-7-(1H-indol-3-ylmethylideneamino)hepta-2,4,6-trienoyl]propanehydrazide 5-[(1R)-2-amino-1-hydroxyethyl]sulfonylbenzene-1,3-diol 1-[(2S)-butan-2-yl]-3,5-dimethyl-6-pentoxybenzimidazol-2-one 4-(3,5-dimethyl-1H-pyrazole-4-carbonyl)-N-[4-(4-methoxyphenyl)-5-oxotetrazol-1-yl]piperazine-1-carboxamide N-(3,3-dimethylcyclohexyl)-2-(4-phenylpyrazol-1-yl)acetamide (2S)-1,4-diamino-5-(2-diazohydrazinyl)-6-oxo-3-phenylmethoxyhexan-2-olate N-[(3S,4R)-3-hydroxyoxan-4-yl]-6-pyrazol-1-ylpyridine-2-carboxamide 4-amino-5-(N-methylanilino)sulfanylbenzene-1,3-diamine 2,4-dichloro-1-(3-methylbutanoyloxy)benzene N-[1,3-benzothiazol-2-yl(phenylmethoxy)phosphoryl]methanamine 2-(N-(1,3-diethoxy-1,3-dioxopropan-2-yl)-4-methoxyanilino)octanoic acid 1-benzyl-4-[3-(2,6-dimethoxyphenyl)propyl]piperazine 6-[3-(2-cyanopropan-2-yl)cyclobutyl]-N-methoxypyridine-2-carboxamide N-[4-(1,5-dimethylpyrrole-2-carbonyl)pyridin-3-yl]-2,6-difluorobenzamide (4R,5S)-1-cyclopropyl-7-(3,4-dimethoxyphenyl)-6-oxo-4,5-dihydropyrazolo[3,4-c]pyridine-4-carbonitrile 2-[3,6-dimethyl-1-(4-nitrophenyl)sulfonyl-2H-indol-3-yl]acetic acid 4-[2-[[6-[1-(4,5-dimethylfuran-3-carbonyl)piperidin-4-yl]pyridin-3-yl]amino]pyrimidin-5-yl]benzonitrile 1-[6-(4,5-dimethyl-1H-imidazol-2-yl)naphthalen-2-yl]-N'-methylpropane-1,3-diamine 5-[(1S)-2,3-dimethylcyclohexyl]pentanoic acid;(E)-3-[4-(methylamino)phenyl]prop-2-enal 2-(2,4-dichlorophenyl)-7H-[1,2]oxazolo[5,4-f]quinoline 2-[(3,5-dimethoxyphenyl)iminomethyl]benzenesulfonic acid 2,3-dichloropyrido[2,1-b]quinazolin-11-one 6-chloro-2-ethyl-N-[(4-methoxyphenyl)methyl]imidazo[1,2-a]pyridine-3-carboxamide 6-(4,5-dihydropyridazin-3-yl)-2-(trifluoromethyl)-1H-indole N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-ethoxy-2-methyl-8-(2-morpholin-4-ylethylamino)-3-phenylimidazo[1,5-a]pyrazine-7-carboxamide 1-[4-[4-(2,5-dioxopyrrolidin-3-yl)butoxy]phenyl]cyclopropane-1-carboxylic acid N'-[4-(3,5-dimethylphenyl)pentanoyl]-2-phenylacetohydrazide;hydrate 3-bromo-5-chloro-N-(3,4-dimethylphenyl)benzenesulfinamide;cyclopropane 4-amino-6-[(2,5-dimethoxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 1-[2-amino-4-(3-hydroxyphenyl)sulfanylphenyl]ethanethiol (1Z)-1-butan-2-ylidene-3,4-dichloronaphthalene N-[(E)-(5-bromo-2,3-dihydroxyphenyl)methylideneamino]-4-chlorobenzamide (1E,3Z)-2-methyl-N-(3,3,5,5-tetramethylcyclohexen-1-yl)oxy-4-[2-(trifluoromethyl)phenoxy]penta-1,3-dien-1-amine 4-[(2S,3aS,6aS)-5-[(1R,2R)-2-hydroxycyclohexanecarbonyl]-1,3,3a,4,6,6a-hexahydropentalen-2-yl]benzamide 6-bromo-4-hydroxy-2,8b-dihydro-1H-cyclobuta[c]chromene-9-carboxylic acid 5-bromo-N,4-dimethyl-1H-benzimidazole-2-carboxamide 4-fluoro-1,3,5-trimethylindazole 2-[4-chlorobutyl(cyanomethyl)amino]benzenesulfonic acid 4-(cyclopropylmethoxy)-N-[1-[3-(4,5-dihydropyrimidin-2-ylamino)phenyl]ethyl]benzamide 3-(2-hydroxyphenyl)-2-[4-phenyl-1,3-di(propanoyloxy)butyl]propanoic acid N-[(3S,4R)-1-[2-(oxan-4-ylamino)pyrimidine-5-carbonyl]-4-phenylpyrrolidin-3-yl]cyclopropanecarboxamide N-(1,2-benzoxazol-5-yl)benzenesulfonamide 2-chloro-N-(4,5-dimethyl-1H-pyrazol-3-yl)butanamide 1-[(3R,4R)-3-[(2S,6R)-6-tert-butylmorpholine-2-carbonyl]-3,8-dimethyl-1,5,9-triazacyclododec-9-yl]-3-(2-chlorophenyl)propan-1-one;hydrochloride (Z)-N-[1-(4-chlorophenyl)ethenyl]-2,6-dimethylhept-3-enethioamide 3-[4-(dipropylamino)-2H-1,3-thiazol-5-ylidene]benzaldehyde 1-[2,4-bis(2-methylbutan-2-yl)phenyl]ethoxy-(2-tert-butylphenoxy)phosphinic acid N-[2-(N-acetyl-4-hydroxy-3,5-dimethoxyanilino)ethyl]formamide 2-[3,4-bis(ethenyl)phenoxy]aniline 3-[[5-(4,6-dimethylcyclohexa-2,4-dien-1-yl)tetrazolo[1,5-a]quinolin-8-yl]oxymethyl]aniline 5-bromo-4,6-dimethoxypyrimidine-2-carboxylic acid 5-fluoro-3-[4-(furan-2-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-1H-pyrazolo[4,3-b]pyridine 1-[[4-(5-bromo-2,3-difluorophenyl)-1H-pyrazole-5-carbonyl]amino]-5-(difluoromethyl)indazole-6-carboxylic acid 2-(dimethylamino)-6-[3-(5,7-dimethyl-1H-indol-4-yl)phenyl]-9-(oxan-2-yl)purine-8-carboxamide 2-[(E)-2-phenylethenyl]quinoline 2-(1-azidoindol-3-yl)ethanol 4-[1-[2-(2,3-dichlorophenyl)acetyl]piperidine-4-carbonyl]benzoic acid 1-(4,7,9-trimethyl-5,6-dihydro-[1]benzoxepino[5,4-d]pyrimidin-2-yl)pyrrolidine-3-carboxylic acid 4-(2,5-diaminopentyl)-3-methoxybenzenethiol 4-[[5,7-dichloro-1-(ethoxymethyl)indole-2-carbonyl]amino]cyclohexane-1-carboxylic acid 6-[2-[(4E,5Z)-5-ethylidene-4-prop-2-enylidenepyrrol-3-yl]phenyl]-9-phenylxanthene-3,7-dione 1-(3,5-dichlorophenyl)-3-[2-(6-oxo-4-propan-2-yl-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]urea 2-[(1S)-4-oxo-5-phenylmethoxycarbonyl-3,6-dihydro-2H-pyridine-1-carbonyl]pentanoic acid 2-fluoro-4-methyl-3-[1-(1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carbonyl)piperidin-4-yl]oxybenzamide 5-(4-fluorophenyl)sulfanyl-N,4-dimethyl-6-propan-2-ylidenepyrimidine-2-carboxamide 7-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)-5,10,12-triazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,8,11-hexaene 4-N-(3,5-difluoropyridin-2-yl)-7-methoxyquinoline-3,4-diamine;ethane 4-[1-(2,6-dichlorocyclohexa-1,3-dien-1-yl)pyrazol-3-yl]pyridine 1-(3,4,5-trifluorophenyl)benzimidazole 4-methyl-2-(3-phenylpropoxyimino)pentanoic acid 1-[2,6-bis(4-chlorophenyl)pyridin-3-yl]-N-methylsulfonylmethanesulfonamide 4-bromo-5,6-dimethyl-N'-(2,2,2-trifluoroacetyl)-1-benzofuran-7-carbohydrazide;ethane 3,6-difluoro-5-methoxybenzene-1,2-disulfonate 2-N,4-N-dihexyl-1,3,5-triazine-2,4,6-triamine;hydrate N-[(1R)-2-cyano-1-phenylethyl]-4,5,6,7-tetrahydro-3H-benzimidazole-5-carboxamide N-[4-(3-fluorophenyl)cyclohexyl]benzenecarbothioamide 3-cyclopropyl-2-[6-[5-methoxycarbonyl-1,4-di(propan-2-yl)pyrrol-2-yl]pyridin-3-yl]imidazole-4-carboxylic acid 3-(difluoromethyl)-2,4,6-trifluoro-N-[2-[(2R)-1-hydroxypropan-2-yl]oxypyridin-4-yl]benzamide 2-(4-bromo-3,5-dimethoxyphenyl)-1H-indole 4-[2,3-difluoro-5-(phenylmethoxycarbonylamino)benzoyl]piperazine-1-carboxylic acid 1-methylcyclopentane;2,4,6-trifluoro-3-hydroxy-5-propan-2-yloxybenzonitrile 4-(2,1,3-benzothiadiazol-5-yl)-N-methylbenzamide N-benzyl-2-[(4R,5S)-1-benzyl-3-oxo-1-sulfanylidene-6-(trifluoromethyl)-2H-imidazo[1,2-a]benzimidazol-2-yl]acetamide N-[3-[4-(1,5-dimethyl-6-oxopyridin-3-yl)phenyl]pentan-3-yl]acetamide 4-bromo-5,6-diethylnaphthalene-2,7-disulfonate 1-[3,5-bis(trifluoromethyl)phenyl]-2H-pyrazine 5-cyclopropyl-4-[7-(cyclohexylamino)imidazo[1,2-b]pyridazin-3-yl]-N-ethyl-2-methoxybenzamide 6-[4-(aminomethyl)-3,5-dichlorophenyl]-1H-triazin-2-amine 3-[3-(4-methoxyphenyl)pyridin-2-yl]benzoic acid N-[(E)-2-[methyl-[6-(4-methylpiperazin-1-yl)-1,3-benzothiazol-2-yl]amino]ethenyl]formamide 2-[1-(2,4,5,6-tetramethylcyclohexa-1,3-dien-1-yl)propan-2-yloxycarbonyl]benzoate 5-[8-(2,6-dimethylpyridin-4-yl)-7-oxo-6-propan-2-ylpyrazino[2,3-c]pyridazin-3-yl]pyridine-2-carbonitrile (3-chloro-4,5-dimethylphenyl)sulfonylthiourea 1-cyclopropyl-2,3-difluoro-4-[(E)-pent-3-enyl]benzene 6-[4-[(3S)-3-aminopiperidine-1-carbonyl]pyridin-2-yl]-7,8-dihydropyrido[4,3-d]pyrimidin-5-one N-(4-methoxyphenyl)-N',N',2-trimethyl-N-[4-[2-[(4Z)-3-methylidene-1-[5-[3-(trifluoromethyl)phenyl]furan-2-yl]hexa-4,6-dien-2-ylidene]hydrazinyl]phenyl]propane-1,3-diamine 3-(2,4-dimethylphenyl)-7,8,9,10-tetrahydrobenzo[a]azulene (2R)-1-[4-(6-tert-butylpyridazin-3-yl)piperazin-1-yl]-2,3-dihydroxypropan-1-one 4-N,6-dimethyl-2-N-[3-(trifluoromethoxy)phenyl]-1H-quinoline-2,4-diamine 2-[(E)-2-[4-hydroxy-3,5-bis(methylsulfanyl)phenyl]ethenyl]quinolin-8-ol 3-(5,6-dimethoxypyridin-3-yl)-1H-indole N-[(1S,3R)-2,2-dimethyl-3-phenylcyclopropyl]pyridine-4-carboxamide 2-[(2S)-1-[3-cyano-5-(trifluoromethyl)pyridin-2-yl]sulfanylpropan-2-yl]-N,N-diethylbenzenesulfonamide 5-chloro-2-(2,6-dimethylphenyl)benzene-1,3-disulfonamide N-[(1R)-4,6-dichloro-2,3-dihydro-1H-inden-1-yl]carbamate 4-[4,6-bis(trichloromethyl)-1H-1,3,5-triazin-2-ylidene]-1-methylpyrazolidine 3-[(2Z,4Z)-hexa-2,4-dienyl]-6-pyridin-2-ylpyridazine;platinum 1-[3-(3,4-dihydropyridin-5-yl)phenyl]-9H-carbazole 3-[(2,4-dichloropyrimidin-5-yl)-ethylamino]phenol 1-azidooxy-5,6-dichloronaphthalene 3-[4-(2,6-diethylphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-1-one 3-[4-[[6-(oxan-2-yloxy)pyridine-3-carbonyl]amino]cyclohexyl]propanoic acid 5-methoxy-4-[4-(methoxymethyl)phenyl]sulfonylmorpholine 6-[4-fluoro-2-(3,4,5-trifluorophenyl)phenoxy]-2-N,1-N-dimethylhexane-1,2-diamine 2-[3-(2-methylphenyl)prop-2-enoylamino]-4,6-di(pyrazin-2-yl)benzenesulfonic acid 2-[[(4-chlorophenyl)methylamino]methyl]benzoic acid 1-[3-(oxolan-2-yl)azetidin-1-yl]-2,7-naphthyridine (E)-N-[3,4-dimethyl-1-oxo-1-(4-pyridin-2-yloxyanilino)pentan-2-yl]-4-pyridin-4-ylbut-3-enamide;ethane 3-[[4-hydroxy-1-(6-piperidin-1-ylpyridine-2-carbonyl)piperidin-4-yl]methyl]-7-methoxyquinazolin-4-one 2-benzyl-4-iodo-5,6-dimethoxy-1H-isoindole 1-[3,5-dimethyl-4-(2-piperidin-4-ylethoxy)phenyl]propan-2-one (3-bromophenyl)methylcyclopentane;3,3-diethylpentane 5-(2-diazohydrazinyl)-2,3-dihydro-1H-indene-4-carbonitrile 4-[2,6-di(propan-2-yl)phenyl]imino-2-[(2,5-dimethylpyrrol-1-id-3-yl)methyl]isoindole-1,3-dione;platinum(2+) 6-[(4-fluorophenyl)methyl]-3,9-dihydropyrrolo[3,2-f][1,7]naphthyridine 4-[1-(cyclobutanecarbonyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one 1-(4-methylphenyl)sulfonyl-3-pent-2-enoylpyrrolidine-3-carbonitrile (3R,4S)-3-[4-[(3-propanoylphenyl)methoxy]benzoyl]piperidine-4-carboxylic acid 1-[4-(4,5-dimethylpyridin-2-yl)piperazin-1-yl]ethanone 4-[(6-chloropyridin-3-yl)methyl]-N',N'-dimethylpiperazine-1-carboximidamide 7-hydroxy-2-methyl-3,4-dihydro-1H-acridine-9,10-dione 2-[4-(difluoromethoxy)phenyl]-3-ethyl-5,7-dihydro-1H-pyrrolo[2,3-f]benzimidazole-6,8-dione (6Z)-1,4,7-trimethyl-5-methylidene-2H-3-benzazocine (3Z)-2,4-dimethylpenta-1,3-diene;ethane;(E)-4-[6-[4-(4-ethenylphenyl)phenyl]naphthalen-2-yl]hex-4-enal 2,3-difluorobenzaldehyde;1-(2-methylpentan-2-yl)-5-[1-[4-[(4Z)-4-(4-propoxyphenyl)hexa-2,4-dienoxy]phenyl]ethyl]triazole N-[5-(1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene-2-carbonyl)pyridin-2-yl]benzamide 6-(difluoromethoxy)-3-ethenylisoquinoline 2-[1,3-dioxo-2-(3-propanoyloxypropyl)isoindol-4-yl]acetic acid [2-(benzenesulfonylmethyl)phenyl]boronic acid 2-methyl-4-[4-(5,6,7,8-tetrahydronaphthalen-1-yloxy)piperidin-1-yl]-10H-thieno[2,3-b][1,5]benzodiazepine 7-ethoxy-4-fluoro-2-propylisoquinolin-1-one [2-fluoro-3-(trifluoromethyl)phenyl]-[2-methyl-2,4-di(propan-2-yloxy)butyl]azanide N-ethenylsulfonyl-2,4,6-trimethyl-N-[(1-phenylpyrazol-3-yl)methoxy]benzenesulfonamide 5-[2-[1-(3,4-dichlorophenyl)-4-methylimidazol-2-yl]phenyl]pyridine (7R)-N,8-dimethyl-7-propan-2-ylidene-6-sulfanylidene-5H-naphthalene-2-sulfonamide 5-methyl-4-(oxolan-3-ylamino)-1H-pyrimidin-6-one 4-(2-azidoethyl)benzo[g][1,3]benzodioxole 1-(4-methylphenyl)sulfonylindazole N-(cyclopropylmethyl)-1-[(E)-2-[4-[3,5-dichloro-4-(piperidine-4-carbonylamino)phenyl]phenyl]-1-phenylbut-1-enyl]-4-hydroxypyrrolidine-2-carboxamide 2-[[5-amino-4-(cyclopentanecarbonyl)imidazol-1-yl]methyl]-7-cyclopentyloxy-3H-quinazolin-4-one (3E)-4,5-diethoxycarbonyl-6-methylimino-N-phenylpyridine-2-carboxamide (4S)-1,2,3,4,5-pentadeuterio-6-[3-oxo-7-[[2,3,5-trideuterio-6-fluoro-4-(morpholin-4-ylmethyl)phenyl]methoxy]-1H-isoindol-2-yl]piperidine-3-carboxylic acid 2-[4-(4,6-dimethylpyrimidin-5-yl)phenyl]-N-[5-(2H-tetrazol-5-yl)pyridin-3-yl]propanamide N-[(2R)-4,4-difluoro-3-hydroxy-1-phenylbutan-2-yl]formamide 4-N,4-N-bis(2-chloroethyl)-6-methylpyrimidine-2,4-diamine 4-[5-methoxy-2-(methylamino)phenyl]-N,6-dimethyl-1,3,5-triazin-2-amine N-(2,6-dichlorophenyl)sulfonyl-1-methylindazole-7-carboxamide N-[(3R)-piperidin-3-yl]-2-[[4-(trifluoromethoxy)phenyl]sulfonylamino]benzamide;2,2,2-trifluoroacetic acid 3-[[(2R)-4-methyloxan-2-yl]amino]propanenitrile;1,4-xylene 2-[3-(2-hydroxyethoxy)propyliminomethyl]phenol 2-[3-methylbut-2-enyl(1,3-thiazol-5-yl)amino]decanoic acid 5-[(Z)-(5-hydroxyindol-3-ylidene)methyl]-2-imino-1,3-dimethylimidazol-4-ol 1-[5-(4-cyanopyridin-2-yl)pyridin-3-yl]-N,N-dimethylpyrrolidine-3-carboxamide 6-chloro-3,4-dimethoxypyridazine-1-carboxylic acid (7-aminophenanthren-2-yl)boronic acid 2-azido-5-methoxy-N,4-diphenylaniline 2-methyl-5,6-dinitrobenzene-1,3-diol 3,4-dichloro-2-[(2S)-2-ethoxycarbonyl-5-methylpiperazin-1-yl]sulfonylbenzoic acid 7-(2-nitrophenoxy)pyrrolo[1,2-c]pyrimidine 5-(3,4-dihydro-2H-chromene-6-carbonylamino)-1H-indazole-7-carboxylic acid 1-(5,6-diaminopyridin-2-yl)ethanol 2-[(1R,5S)-3,8,9-trimethyl-6-phenyl-7H-benzo[a]quinolizin-4-ium-10-yl]quinoline 2-aminooxy-5,6,7-trihydroxynaphthalene-1,4-dione 1-[2-[5-[(E)-2-[3,4-difluoro-2-(trifluoromethyl)phenyl]ethenyl]pyrimidin-2-yl]oxyethylsulfonyl]pyrrolidin-3-ol 4-bromo-N'-hydroxy-3-(trifluoromethyl)benzohydrazide N-[(4,5-dimethoxycyclohexa-1,3-dien-1-yl)methylidene]hydroxylamine;ethane N-[(2R)-3,3-difluoro-1-hydroxypropan-2-yl]-3-(6-methoxypyridin-3-yl)sulfonylbenzamide (Z)-5-hydroxy-2,2,6,6-tetramethylhept-4-en-3-one;iridium(3+);2-phenylquinoline (1S,5R)-3-[4-[6-methoxycarbonyl-7-(pyrrolidine-1-carbonyl)quinolin-4-yl]oxyphenyl]-7-oxa-3,10-diazabicyclo[3.2.0]heptane-9-carboxylic acid 3-methyl-2-oxo-6-pyridin-4-ylhexanedioic acid N-(1H-indol-6-yl)-3,5-dimethoxybenzamide N-[2-(1,3-benzodioxol-5-ylmethoxy)ethyl]-6-bromopyridine-3-carboxamide 6-chloro-5-[3,4-difluoro-2-(methoxymethyl)phenyl]-1H-pyrrolo[2,3-b]pyridine 3-(2,4-dichlorophenoxy)-N-[4-(4,6-dimethoxypyrimidin-5-yl)cyclohexa-1,3-dien-1-yl]aniline N-[1-(2-cyanopropanoyl)piperidin-4-yl]-5,7-dimethoxyisoquinoline-8-carboxamide 2-[4-(methylamino)-3-nitrophenyl]acetic acid (1R)-2,3-bis[2-(3-methoxy-4-methylphenyl)ethyl]cyclohexan-1-amine 3-(3,4,5-trichlorophenyl)oxirane-2,2-dicarbonitrile 4-(3,5-difluoroanilino)-1H-pyrazole-5-carboxamide [(4aR,7aS)-1,2,3,4,5,6,7a-octahydrocyclopenta[c]pyridin-4a-yl]-(3-chlorothiophen-2-yl)methanone 4-(2,6-dichloro-3,5-dimethoxyphenyl)quinoline 1-amino-3-[(4-chlorobenzoyl)amino]thiourea 1-methyl-6-pyridin-2-ylpyrrolo[2,3-b]pyridine 2-N-[(3E,5Z)-4-(8-aminoquinolin-7-yl)hepta-1,3,5-trien-2-yl]-5-methanimidoylpyrimidine-2,4-diamine 2-[4-[1-[4-(3-phenylpropanoylamino)benzoyl]piperidin-4-yl]butoxy]benzoic acid 6-(4-chlorophenyl)-N,4-dimethyl-5,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-2-imine 6-amino-4-(3-bromo-4-ethoxy-5-iodophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 2-(1,3-benzoxazol-6-ylsulfanyl)propanedioic acid 3-N,4-diethyl-5-fluoro-2-nitrobenzene-1,3-diamine [1-(2,6-dichlorobenzoyl)pyrrolidine-3-carbonyl]azanide N-[3-cyano-4-(2-hydroxyethylamino)phenyl]propanamide;3,3-dimethyl-2H-1-benzofuran N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-5-fluoro-2-methoxypyridine-4-carboxamide 3-[3,6-bis(ethenyl)carbazol-9-yl]-7-(5-pyridin-4-ylthiophen-2-yl)dibenzofuran-4-carbonitrile N-[(4,5-dichlorothiophen-3-yl)methyl]-3-[methyl-[1-[4-(trifluoromethyl)pyrimidin-2-yl]azetidin-3-yl]amino]cyclobutane-1-carboxamide 2-(6-chloropyridazin-3-yl)sulfanylpyridine 1-methyl-3-[5-(6-piperidin-4-yloxypyridin-2-yl)-2,3-dihydro-1H-inden-4-yl]urea;hydrochloride (2S)-N-ethylsulfonyl-1,4-dioxane-2-carboxamide;1-[4-fluoro-2-[3-(trifluoromethyl)phenyl]-6-propan-2-ylphenyl]ethanone (6S,8aS)-N-benzhydryl-2-amino-5,6,7,8-tetrahydroquinazoline-6-carboxamide 1-(3,5-dichlorophenyl)-N-[3-fluoro-4-[2-[6-hydroxyhexyl(propanoyl)amino]pyridin-4-yl]oxyphenyl]cyclopropane-1-carboxamide;hydrate 3-(difluoromethyl)-N-[2-[1-(5,6-dihydronaphthalen-1-yl)cyclopropyl]ethyl]pyridine-4-carboxamide 5-[(3,4-difluorophenyl)methyl]-2,3,6-trimethylpyrimidine-4-thione 2-[5-[3-chloro-4-(trifluoromethyl)phenoxy]naphthalen-1-yl]oxyacetic acid 5-(7-azido-3-methylimidazo[1,2-a]pyridin-6-yl)-2-N-butan-2-ylpyrimidine-2,4-diamine N-[(1R,2S)-2-hydroxycyclohexyl]pyrazolo[1,5-a]pyridine-3-carboxamide 5-[4,6-difluoro-2-[(E)-oct-1-enyl]phenyl]-2-hydroxybenzoic acid 3-(2-cyclopentylethynyl)aniline 2-[3-(cyclopropanecarbonylamino)pyrazol-1-yl]-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazole-6-carboxylic acid 3-ethyl-7-(4-fluoro-2-propan-2-ylphenyl)isoquinoline;methane 2-[1,4-dichlorobutyl(ethyl)amino]phenol N-methoxy-1,2-dimethylpyrazole-3-carboxamide 2-(2,6-dichlorophenyl)iminopropanoic acid 3-[2,4-bis(phenylmethoxy)-5-propan-2-ylphenyl]-5-cyclohexyl-1H-pyrrole-2-carboxylic acid 4-N,6-bis(3,5-dimethylphenyl)pyrimidine-2,4-diamine 1-(3,4-dichlorophenyl)-6,8-dimethoxy-N-[4-(2-oxopiperidin-1-yl)sulfonylphenyl]-7-propan-2-yloxyisoquinoline-3-carboxamide 2-[[1-(4,6-dichloro-3-methylquinoline-2-carbonyl)piperidin-4-yl]amino]acetic acid;ethane N-[4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]phenyl]quinoline-8-sulfonamide 3-(6,7-dichloro-1H-indazol-4-yl)benzamide 3,4-dichloro-N-(2-chloro-5-methylphenyl)-1H-pyrrole-2-carboxamide 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-2-[4-(4-hydroxybut-3-enylsulfanyl)phenoxy]-2H-ethanone 2-[4-(3-chlorophenoxy)piperidin-1-yl]-7H-purine 6-[[4-(3,5-dichlorophenyl)sulfonylpiperazin-1-yl]methyl]pyrazine-2-carboxamide ethane;3-methyl-2,6,7,8-tetrahydrocyclohepta[d]pyrimidin-4-one 2-[5,10-dimethoxy-3-(4-methoxyphenyl)-6H-benzo[c]chromen-8-yl]pyridine 2-(4-methoxycarbonylanilino)-6-oxohexanoic acid ethane;ethene;formaldehyde;1-[3-(5-methylcyclohepta-1,4,6-trien-1-yl)-2-phenylpropyl]piperidine 3-(2,6-dioxopiperidin-3-yl)-4-[3-(oxan-4-yl)prop-1-ynyl]benzenesulfonamide 6-(3-chlorophenyl)spiro[2H-1-benzofuran-3,4'-piperidine] 4-(methyliminomethyl)benzenecarboximidamide 2-[(6-chloropyridin-3-yl)-ethoxyamino]acetonitrile 4-[[4-(hydroxymethyl)phenyl]diazenyl]-5-methoxy-1,2-dihydropyrazol-3-one N-(3-methylbutyl)-N',N'-dipropylethane-1,2-diamine;naphthalene-2,6-disulfonic acid N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]prop-2-enamide N-[4-[2,3-dihydroxypropyl(2H-tetrazol-5-yl)amino]phenyl]sulfonylbenzamide 2-[(E)-5-methyliminopent-3-enoxy]benzoate 7-hydroxy-2,3-bis(2-methoxyethyl)-5H-pyrimido[4,5-b][1]benzazepine (3S)-4,5-dihydroxy-3-[(E)-(2-oxo-1H-indol-3-ylidene)methyl]pentanoic acid 4-[1-carboxyheptyl(hexadecanoyl)amino]benzoic acid 3-(dimethylamino)-4-[methyl-[(3S,6R)-1-(pyridine-2-carbonyl)-6-(trifluoromethoxy)piperidin-3-yl]amino]benzonitrile [(1R,2S)-2-[4-(3-morpholin-4-ylpropylcarbamoyl)phenoxy]cyclohexyl]azanium 3-bromo-N-[3-(2,4-difluorophenyl)-1H-indazol-5-yl]-1-methylpyrazole-4-carboxamide N-(4-fluorophenyl)-1,2,3,5-tetramethylcyclohexa-2,4-dien-1-amine 4-[6-chloro-2-[2-(4,5-dihydro-1H-imidazol-3-ium-3-yl)ethoxy]quinazolin-4-yl]morpholine (4-carboxyphenyl)methyl-[4-[6-(2,2-dimethylpropanoyloxy)hexoxy]benzoyl]azanium 1-[[(2R,4S)-4-fluoropyrrolidine-2-carbonyl]amino]pyrazole-4-carboxylic acid 4-azido-6-methoxy-N-(oxetan-3-yl)pyridin-2-amine 2-azidooxy-5,6-dihydro-4H-thieno[2,3-c]pyrrole 4-N,8-N-bis(2-bromophenyl)pyrimido[5,4-d]pyrimidine-4,8-diamine N-[(2S)-1,5-dihydroxypentan-2-yl]-4-phenylbutanamide N'-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-2,5-bis(trifluoromethyl)pyrazole-3-carboximidamide N-(2,6-dimethylphenyl)-3-[3-[1-[(5R)-7-fluoro-5-methyl-5H-[1]benzoxepino[3,4-c]pyridin-9-yl]ethyl]pyrazol-1-yl]propanamide (1R,2R)-N-[8-amino-6-(4-methylpyridin-3-yl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide;2,2,2-trifluoroacetic acid 4-[2-hydroxy-5-(1,3,5-trimethylpyrazol-4-yl)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 5-ethyl-4,6-dimethyl-2-(4-nitrophenyl)sulfanylpyridine-3-carboxylate 2-[4-fluoro-3-(trifluoromethyl)phenyl]benzoic acid 2-methyl-N,N'-bis[(2R)-1-oxo-3-phenylpropan-2-yl]butanediamide (3S,5R)-4-benzoyl-3-hydroxy-1-(2-thiophen-2-ylsulfanylethyl)-3,5-dihydro-2H-pyrido[3,2-e][1,4]oxazepine-7-carbonitrile 2-[3,5-dibromo-4-(3-chloro-4-hydroxyphenyl)sulfonylsulfanylphenyl]acetonitrile 2,4-dichloro-N-[2-(dimethylamino)ethyl]-5-nitrobenzamide;3-(2,3,6,7-tetrahydrooxepin-8-yloxy)propanal N'-[[6-[(E)-2-[4-amino-3-(methyliminomethyl)phenyl]ethenyl]pyridin-2-yl]methyl]-N,N'-diethylbutane-1,4-diamine (2-fluoro-5-methoxyphenyl)-[3-hydroxy-3-(methoxymethyl)pyrrolidin-1-yl]methanone ethane;5-fluoro-3-[2-(furan-2-yl)propan-2-yl]pyridine 5-[8,9-dihydroxy-2-[(3R)-piperidin-3-yl]-4H-chromeno[4,3-c]pyrazol-3-yl]pyridine-2-carbonitrile ethane;2-(3-hydroxypropoxy)-5-[4-(1,1,6-trioxo-1,2,5-thiadiazocan-5-yl)phenyl]benzonitrile 4-methyl-2,6-bis[(E)-1-phenylpropylideneamino]phenol 2-[1-azido-3-(4-fluorophenyl)propan-2-yl]-1H-indole 2,6-difluoro-3-methylbenzoic acid;ethane 3-[1,2-bis(4-methoxyphenyl)ethyl]-6-bromochromene-2,4-dione 3-(2,4-dimethyl-1,3-oxazol-5-yl)-N-[2-methyl-6-(trifluoromethyl)pyridin-4-yl]pyrrolidine-1-carboxamide N-[4,5-dichloro-2-hydroxy-3-(trifluoromethyl)phenyl]acetamide 5-[2-(difluoromethyl)phenyl]-1,3-thiazolidine N-methyl-N-[2-(4-propan-2-ylphenyl)ethyl]butanethioamide 2-[(1S)-5,6-dimethoxy-3,4-dihydro-2H-naphthalen-1-ylidene]propanedinitrile 3-aminosulfanyl-N'-ethenyl-2-fluorobenzohydrazide 1-[4-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethanone 2-bromo-N-(2,4-dichloropyrimidin-5-yl)-N-(1,3-thiazol-2-yl)benzamide N-ethyl-3-methylsulfonylbenzamide;1,2,4-trimethoxybenzene [(2S)-1-methyl-6-phenylmethoxy-5,7-dihydro-4H-pyrazolo[3,4-c]pyridin-3-yl]-phenylmethanone 3-[4-(3,5-dichlorophenyl)triazol-1-yl]-6-phenylmethoxycyclohexa-2,4-dien-1-amine (1S)-2,3-dihydro-1H-benzo[f]chromene-1-carboxamide 2-(4,5-diphenyl-3H-1,2-oxazol-2-yl)aniline 1-[2,3-dimethyl-6-(1H-pyrrolo[2,3-b]pyridin-4-yl)-5,7-dihydro-4H-pyrazolo[3,4-c]pyridin-3-yl]butan-2-one ethane;3-[2-methylpropoxy(phenyl)methyl]oxiran-2-ol 5-[(5-fluoropyridin-2-yl)methoxy]pentanoate N-[2-(1,3-benzothiazol-5-yl)-6-methoxypyridin-4-yl]-2-hydroxybenzamide (Z)-1-[2,5-dimethyl-4-[(E)-1-(2-methylanilino)but-1-enyl]phenyl]-3-ethylpent-3-ene-2,4-dione 3-(1-azidopyrrolidin-2-yl)pyridine (2E,5Z)-2-ethenyl-1-(3-methylsulfanylphenyl)hepta-2,5-diene-4,6-dione N-[2-(5-cyanopyridin-3-yl)-1,6-naphthyridin-7-yl]-N'-cyclohexa-1,5-dien-1-ylethanimidamide;ethane N-[(2R,3S)-1-(azetidine-1-carbonyl)-2-(1-methylpyrazol-4-yl)pyrrolidin-3-yl]-5-fluoropyrimidine-2-carboxamide 1-[2,6-di(propan-2-yl)phenyl]-5,7-dihydroindolo[3,2-c]carbazole 3-[[(5Z)-5-[[2,4-bis(2-chloroethoxy)phenyl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzonitrile N-[3-(dimethylamino)propyl]-1,7-bis(trifluoromethoxy)naphthalene-2-carboxamide 4-azidooxy-2,3,5,6-tetrachlorobenzenesulfonic acid 3-[(2R,3S)-3-(3-fluorophenyl)pyrrolidin-2-yl]propane-1,2-diol 1-[4-chloro-3-(1,2,4-triazol-1-ylmethyl)phenyl]pyrazole 4-(2,3,4,5-tetrafluorophenyl)cyclohexane-1,3-diol 2-[1-(3-aminopyridin-4-yl)piperidin-4-yl]sulfanyl-4-methyl-1H-pyrimidin-6-one 6-chloro-N-[3-(2,4-difluorophenyl)phenyl]-1H-indole-2-carboxamide 4-(2,3,6-trifluorophenyl)quinoline (7R)-2-amino-6,10-dimethyl-7-[(2-nitrophenyl)methoxy]-6,7-dihydro-5H-imidazo[1,2-d][1,4]benzodiazepin-3-one 4-ethylbenzoic acid;2-[5-(3-methoxyphenoxy)pentanoyl]-2,6-diazaspiro[3.3]heptane-7-sulfonamide [7-(2,4-dimethylanilino)pyrazolo[1,5-a]pyrimidine-3-carbonyl]iminothiourea N-[2-(6-fluoropyridin-3-yl)oxyethyl]butanamide [2-azido-1-(4-chlorophenyl)-1,3-thiazolidin-5-ylidene]cyanamide N-[2-(3,4-dichlorophenyl)ethyl]-7H-purine-6-carboxamide 2-[(1R,2S)-3,3-dimethylcyclohex-4-en-1-yl]-5-ethoxycarbonylbenzoate (E)-2-[[3,5-dimethyl-4-(phenylsulfanylamino)thiophene-2-carbonyl]amino]pent-2-enoic acid 2-tert-butylsulfanyl-1H-pyrimidine-2,4-diamine 1-[4-(aminomethyl)phenyl]sulfonylpropan-2-ol 1-[4-[2,5-dimethyl-4-(3,4,5-trifluorophenyl)pyrazol-3-yl]oxypiperidin-1-yl]-2-[methyl(pyrrolidin-3-yl)amino]ethanone;hydrochloride N-[[4-amino-3,5-difluoro-2-(methyliminomethyl)phenyl]methoxycarbonylamino]carbamate N-[2-(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]benzamide 4-[(2Z,3E)-1-cyclohexa-1,5-dien-1-yl-2-ethylidenehexa-3,5-dienyl]pyridine 4-[2-[5-cyclopropyl-6-(2,2-difluoroethoxy)pyridin-3-yl]pyrimidin-4-yl]-3-methylmorpholine (E)-N-[2,4-dimethyl-3-[7-[4-[1-(trifluoromethyl)cyclopropyl]phenyl]imidazo[1,2-a]pyridin-3-yl]butan-2-yl]ethanesulfonamide 2-[4-[3-[2,6-dimethyl-5-(methylamino)pyrimidin-4-yl]oxy-5-fluorophenyl]-1H-imidazol-2-yl]-2-(hydroxymethylidene)butanenitrile (2E)-N-[2-(4-chloro-3-fluoroanilino)-5-methylpyrimidin-4-yl]-2-ethoxyiminopropanamide 2-(3,5-ditert-butylphenyl)-4-ethylquinoline 7-methoxy-1,2-dimethyl-4-(2H-pyridin-3-ylidene)quinazoline N-[(4-nitrophenyl)methyl]-N-pyridin-2-yl-1,3-thiazol-5-amine 2-(4-bromo-N-hexylanilino)acetic acid N-[2,6-di(propan-2-yl)phenyl]-1-pyridin-3-ylbut-3-en-2-imine;nickel(2+) 7-azido-2,6-dimethylthieno[3,2-f]chromene 1-[4-methyl-5-(2-phenoxyethoxy)cyclohexa-1,3-dien-1-yl]propan-2-one 1-(5-cyclobutylthiadiazol-4-yl)-3-[2,6-dichloro-4-(trifluoromethoxy)phenyl]urea 7-benzyl-2-[(3E)-penta-1,3-dien-3-yl]-5-propan-2-ylpyrazolo[1,5-a]pyrimidine [(5Z)-3,4-diaminoocta-1,5,7-trienyl]azanide;2-(3,4-dimethoxyphenyl)pyridine;manganese(2+);oxygen(2-) N-[5-fluoro-2,4-di(propan-2-yl)phenyl]-1-methylpyrazole-3-carboxamide [3-(3-chlorophenyl)pyrrolidin-1-yl]-pyridin-4-ylmethanone (2-methylfuran-3-carbonyl)-[4-oxo-5,7-diphenyl-1-(1H-pyrazol-4-ylmethyl)-1,8-naphthyridin-3-yl]azanium 3-(2-fluoro-4-propoxyphenyl)oxirane-2,2-dicarbonitrile 7-(2,6-dichlorophenyl)-N-[4-[3-[ethyl(2-hydroxybutanoyl)amino]piperidine-1-carbonyl]phenyl]-5-methylimidazo[1,2-a]pyrimidine-2-carboxamide;ethane 5-chloro-N,3-dimethyl-4-(triazolo[4,5-b]pyridin-1-yl)benzimidazole-7-carboxamide 2,4-dihydroxy-N,N'-bis(2-methylbutanoyl)benzohydrazide 1-[3-fluoro-2-methoxy-5-(trifluoromethyl)phenyl]-4-[4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]piperidin-1-yl]butan-1-one 1-(2,4-difluorophenyl)-4-[5-methylsulfonyl-4-[1-(trideuteriomethoxy)pyrrolo[2,3-b]pyridin-4-yl]-1,3-thiazol-2-yl]piperazine-2,6-dione 2-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]benzene-1,4-diol (2E)-N,3-bis[4-(diethylamino)phenyl]-2-hydrazinylidenepropanamide 2-[5-(1,3-benzodioxol-4-yl)-7-(pyridin-3-ylmethoxymethyl)-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-3-yl]-N-methylacetamide;2,2,2-trifluoroacetic acid 2-[6-(2-chloroanilino)-4,5-dihydrothieno[3,2-d][1]benzazepine-11-carbonyl]-N'-(4-fluorophenyl)-3H-pyrrole-4-carbohydrazide 2-[(5S,10bR)-7-methoxy-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-methylphenol 1-[2-[4-(trifluoromethoxy)phenyl]propanoylamino]piperidine-4-carboxylic acid (1Z)-N',2-dimethyl-N-[2-(4-phenylmethoxyphenyl)prop-2-enylidene]buta-1,3-diene-1,4-diamine 3-[4,5-dihydro-1H-imidazol-2-yl(hydroxy)methylidene]-6-methoxy-1H-indol-2-one 2-(2,4-dimethylphenyl)-N'-[3-fluoro-4-[6-methoxy-7-(piperidin-1-ylmethyl)quinolin-4-yl]oxyphenyl]propanediamide 1-butyl-5,5-difluoro-3-(2-methoxyethyl)-3H-2-benzofuran-6-carboxylic acid 4-[4-(2,4-dimethylphenoxy)anilino]-6-nitroquinoline-3-carbonitrile;ethane 2-[[7,8-difluoro-6-(5-methylsulfanylpyridin-3-yl)isoquinolin-3-yl]amino]-N-(oxolan-3-ylmethyl)acetamide 2-[4,6-bis(hydroxymethyl)pyrimidin-2-yl]oxy-N-[3-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfanylphenyl]acetamide (Z)-[4,5-bis(ethenyl)-3,6-dihydro-2H-pyran-8-ylidene]hydrazine (5E)-5-[(3,6-dichloro-2-hydroxyphenyl)methylidene]-1-(4-phenoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione [6-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydroxynaphthalen-2-yl]methanesulfonic acid (5Z)-3,7-dimethyl-2-[1-(2-piperidin-1-ylethoxy)naphthalen-2-yl]-4-(2-pyridin-3-ylethynyl)undeca-5,8,10-trienoic acid 1-[4-chloro-6-[(3S)-3,4-dimethylpiperazin-1-yl]pyrimidin-2-yl]-N-ethoxysulfanylpiperidine-3-carboxamide 4-(2,6-difluorophenyl)benzenesulfonamide 2-[(2R)-4-methoxyimino-1-(4-methylphenyl)sulfonylpyrrolidin-2-yl]pyridine-4-carboxylic acid 3-(4-fluorophenyl)-2,6-dimethylpyrazolo[1,5-a]pyrimidine 1,3-difluoro-5-[4-[(2E)-4-propoxypenta-2,4-dienyl]phenyl]benzene 4-[(1-acetylpiperidin-3-ylidene)amino]sulfanyl-N,N-dimethylbenzenecarboximidamide (E)-4-[(2S,6R)-6-methylpiperidin-2-yl]oxy-3-phenylbut-3-enal N-[(2-oxo-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl)methyl]methanesulfonamide 5-chloro-2,3-dihydrothieno[3,4-c]pyrrole-4-carboxamide 3-[3-[2-[2-(dimethylamino)ethoxy]anilino]quinoxalin-6-yl]benzenesulfinic acid 5-[2-(2,4,6-trihydroxyphenyl)sulfonylphenyl]imidazolidine-2,4-dione N-[3,5-dimethyl-4-[[2-(trifluoromethoxy)phenyl]methoxy]phenyl]-2-oxopyrrolidine-1-carboxamide 2-[(4S,9aR)-8-(3-chlorophenyl)sulfonyl-1-methyl-4,6,7,9a-tetrahydro-3H-pyrazino[2,1-c][1,4]oxazin-4-yl]-N,N-dimethylacetamide;2,2,2-trifluoroacetic acid 2,7-dimethyl-N'-(5-phenyl-1,3,4-thiadiazol-2-yl)naphthalene-1-carboximidamide;hydrochloride 1-(azidomethyl)-4-[3,5-bis(trifluoromethoxy)phenyl]benzene (7S)-2-(4-chlorophenyl)-3-[(1R,3S)-3-methylcyclohexyl]-6,7,8,9-tetrahydroimidazo[4,5-c]quinoline 1-[2-(4-fluorophenyl)ethyl]pyrrolidine-3,4-dicarboxamide 4-[3-[(2Z,4E)-5-[(2-chlorophenyl)methylamino]hepta-2,4-dien-6-yn-3-yl]phenyl]phenol 6-[4-[6,7-dimethoxy-2-(4-morpholin-4-ylphenyl)quinazolin-4-yl]piperazine-1-carbonyl]pyridine-3-carboxamide [(2S,3S)-5-amino-1-(benzenesulfonyl)-4,4-difluoropyrrolidine-3-carbonyl]carbamic acid 7-(3,5-dimethyltriazolo[4,5-b]pyridine-6-carbonyl)-1,3-benzoxazole-2-carbonitrile (6E)-1-methyl-6-[[(3R,4S)-3-phenyloxolan-3-yl]methylidene]-5H-triazolo[1,5-a]pyrazine 1-(2,6-difluorobenzoyl)-2-(methoxymethyl)piperidine-3-carboxylic acid 5-hydroxy-6-[(1S)-2,2,3,3-tetrafluoro-1H-inden-1-yl]cyclohepta-1,4,6-trien-1-ol 1-(4,6-dimethoxypyrimidin-2-yl)pentane-3-sulfonamide 2-[2-ethoxy-5-(4-methylpiperazin-1-yl)sulfonylphenyl]-7-methyl-8H-imidazo[1,2-a]pyrimidin-5-one 4-[(E)-1-fluorobut-2-enyl]sulfonylphenol 2,6-dimethoxy-N'-methylbenzenecarboximidamide N-[5-chloro-3-(1H-pyrrolo[2,3-b]pyridine-2-carbonylamino)cyclohexa-1,4-dien-6-yn-1-yl]thiophene-2-carboxamide N-cyclobutyl-6,7-difluoro-1H-indazole-3-carboxamide 3-(6-aminopyridin-2-yl)-N,5-dimethoxyaniline 1-(2,6-difluorophenyl)-3-[2-[[4-[2-[(E)-pent-2-en-2-yl]pyridin-4-yl]oxynaphthalen-1-yl]amino]ethyl]urea 4-[(3R)-3-amino-1,1,2-trifluoropentyl]benzenesulfonic acid 5-phenyl-2,3,4,6,7,8-hexahydropyrimido[1,2-a]pyrimidine 5-(4-bromophenyl)-2,3-bis(9H-fluoren-1-yloxycarbonylamino)pentanoate 1-[(2,3-difluorophenyl)methyl]-3-[5-(2-hydroxyethoxy)-3-imino-4-oxohexan-2-ylidene]urea [7-(3,4-dimethoxyphenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carbonyl]carbamic acid 4-(2,3-dihydroindol-1-ylmethyl)-N'-hydroxypyridine-2-carboximidamide 1-[4-[8-amino-3-(3-ethoxyphenyl)imidazo[1,5-a]pyrazin-1-yl]cyclohexyl]propan-2-one 1-(4-chlorophenyl)-3-[4-[(5-cyanothiophen-2-yl)methoxy]naphthalen-1-yl]urea (4S)-2-[2-methyl-7-[5-methyl-1-[4-(trifluoromethoxy)phenyl]pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-5-yl]-4-phenylpiperidine N-(2,3-dihydro-1H-isoindol-5-yl)-6,8-difluoroquinoxalin-2-amine 5-methyl-2-[3-(oxan-4-yloxy)propyl]pyrimidine 6-[1-(cyclopropanecarbonyl)piperidin-3-yl]-2-methylsulfanyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-4-carboxylic acid 2-[1-(4,5-dimethylpyrimidin-2-yl)azetidin-3-yl]-7H-purine 1-butanoyl-2,5-dimethylindole-3-carboxylic acid 7-(4-butylcyclohexyl)-3,4-difluorodibenzofuran N-[1-[6,7-difluoro-2-(4-fluorophenyl)-3a,4-dihydro-1H-indole-5-carbonyl]piperidin-4-yl]carbamate 3-[(5-ethylthiophen-2-yl)methylamino]piperidine-1-carboxylate 6-butanoyl-2-[1-(4-chlorobenzoyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (5E)-3-(2-methylpyridin-3-yl)-5-[(2Z,4E)-4-morpholin-4-ylhepta-2,4-dienylidene]-1,3-oxazolidine 2-(azepan-1-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine 2-(azidomethyl)phenanthrene 3-[4-(2,5-dimethylfuran-3-carbonyl)piperazin-1-yl]cyclopentane-1-carboxylic acid 2-(2-methylpropoxy)ethoxybenzene;3-[4-[1-[2-(3,4,5-trifluorophenyl)acetyl]piperidin-4-yl]oxyphenyl]hex-4-ynoic acid 2-[4-ethyl-3-(2-methylbutan-2-yl)phenyl]propane-1,3-diol N-[3-(dimethylamino)propyl]-4,5-bis(4-ethoxyphenyl)imidazolidine-1-carboxamide 3-[1,2-difluoro-2-(4-methylphenyl)ethenyl]benzonitrile 6-[(E)-2-[4-[5-chloro-1-(2,4-difluorophenyl)indole-3-carbonyl]piperazin-1-yl]prop-1-enoxy]pyridine-3-carbonitrile 3-[2-[[4-[(1R)-1-aminoethyl]benzoyl]amino]phenyl]propanoic acid 1-[4-(2,6-dichloro-3,5-dimethoxyphenyl)-3-[5-(2-hydroxyethylamino)pyridine-2-carbonyl]piperazin-1-yl]-4-(propan-2-ylamino)butan-1-one 2-(3,5-dichlorophenyl)sulfanyl-N'-[1-[3-(trifluoromethoxy)phenyl]ethyl]acetohydrazide 2-(4-fluorophenoxy)-N,N-dipropylethanamine 2-(3,4-dichlorophenyl)-N-[[5-fluoro-6-(trifluoromethyl)pyridin-3-yl]carbamoyl]acetamide 4-hydroxy-3,5,7-trimethyl-1H-1,6-benzodiazonin-2-one 3-(1,2,4-triazol-1-yl)benzoic acid 5-(3,5-dichlorophenoxy)-2H-triazole-4-carboxylic acid N-[3-(4,5-difluoro-1H-benzimidazol-2-yl)cycloheptyl]formamide 2-[3-(1H-benzimidazol-4-yl)propyl]benzoic acid 5-[1-(3,4-dichlorophenyl)ethoxy]-6-methyl-2-thiophen-3-yl-[1,3]thiazolo[4,5-c]pyridine N'-[2,3-di(propan-2-yloxy)phenyl]ethane-1,2-diimine N-[4-fluoro-3-(2-morpholin-4-ylpyridine-3-carbonyl)phenyl]-6-oxo-5H-benzo[b][1,4]benzoxazepine-11-carboxamide (NZ)-4-methyl-N-[[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonylamino)phenyl]methylidene]benzenesulfonamide 5-(1,2-benzothiazol-3-yl)-N-[1-[(2R,4S,5R)-4,5-dihydroxyoxan-2-yl]-2H-pyridin-6-yl]pentanamide 4-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]-N-(2-pyridin-4-ylethyl)benzamide N-[(1R)-5-cyano-6-methyl-3,4-dihydro-2H-1,8-naphthyridin-1-yl]-1-phenylcyclopropane-1-carboxamide 3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)quinoline;ethane 3-[(2Z)-4-methylhepta-2,5-dienoxy]quinoline (4R)-3,5,13-trimethyl-2-oxa-8-azabicyclo[12.4.0]octadeca-1(18),14,16-trien-17-one (4E)-2,5-bis[4-[(Z)-1-aminoprop-1-enyl]phenyl]hexa-2,4-dienenitrile 2-[(2,4-dichloropyrimidin-5-yl)-hexylamino]-1-phenylethanone 4-N,4-N-bis(ethenyl)-1-(2-methoxyphenyl)hexane-1,4-diamine 1-[(3S)-3-(2,5-difluorophenyl)pyrrolidine-1-carbonyl]cyclopentane-1-carbonitrile 2-(5,7-dichloro-1H-indol-3-yl)-N-[2-methoxy-4-[1-[5-methyl-6-(trifluoromethyl)pyridin-3-yl]pyrazol-4-yl]phenyl]acetamide 5-(3-bromoimidazo[1,2-a]pyridin-7-yl)oxy-4H-pyran-2-carbonitrile N-(3,4-dihydronaphthalen-2-ylmethyl)propan-1-amine;5,6-difluoro-1-benzothiophene 3-(2-ethyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl)thiophene-2-carboxamide (3S)-1,3,4,5-tetrahydro-[1]benzofuro[5,4-c]pyridine 2-cyclohexylimino-5-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)methylidene]-1,3-thiazolidin-4-one 2-N,3-bis(4-fluorophenyl)sulfanylcyclohexa-1,5-diene-1,2,6-tricarboxamide 5-[4-(diethylamino)phenyl]-6,7-dimethoxy-3H-quinazolin-4-one N-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]ethenesulfonamide 2-chloro-N-(4-methoxyphenyl)-1,3,5,6-tetrahydroazepino[4,3-b]indole-9-carboxamide 2,3-dichloro-N-[1-(5-methoxypyridin-3-yl)ethyl]benzamide (2S)-3-[4-(1H-benzimidazol-2-ylamino)phenyl]-2-[(5-oxopyrrolidine-2-carbonyl)amino]propanoic acid (4-aminopiperidin-1-yl)-[2,3-dimethoxy-5-(3-methylbutyl)phenyl]methanone N-[2-chloro-5-methyl-4-(trifluoromethyl)phenyl]-1-[2,6-dimethoxy-4-(pyridin-3-ylsulfamoylamino)phenyl]cyclopropane-1-carboxamide 5-[1-(4-chlorocyclohexa-2,4-dien-1-yl)ethenyl]-N-(3-methoxypropyl)-6H-thieno[2,3-c]pyrrole-4-carboxamide N-(1-azidocyclohexyl)aniline N-[5-bromo-4-(trifluoromethyl)pyridin-2-yl]piperidine-3-carboxamide 2-cyclopentyl-4-methoxypyrimidine;3,3,5,5-tetradeuterio-1-[7-(3,5-difluorophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidine N-(4-nitrophenyl)-1H-indole-2-carboxamide 6-amino-3-(2,4-dihydroxyphenyl)-1H-pyrazole-5-carbonitrile 1-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)ethyl]pyrrolidin-2-one;hydrochloride 5-[1,4-bis(ethenyl)cyclohexa-2,4-dien-1-yl]-4-phenyl-N-[4-(trifluoromethoxy)phenyl]-3,4-dihydropyrazole-2-carbothioamide [(7R,8aS)-2-[4-cyano-3-(trifluoromethyl)phenyl]-1-oxo-5,6,7,8,8a-pentahydroimidazo[1,5-a]pyridin-7-yl]carbamic acid 2-methyl-6-[1-methylidene-3-(4-methylphenyl)-2H-isoindol-5-yl]benzonitrile 4-(1H-benzimidazol-2-ylmethoxy)-N',3-dichlorobenzenecarboximidamide (5Z)-2-cyclopentylimino-5-[(3,4-dimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 4-(3,5-difluorophenyl)-2-[(2S,4R)-4-[2-(6-methoxyquinolin-8-yl)ethynyl]pyrrolidin-2-yl]butanoic acid;ethane 2-(1-ethylpyrrolidin-3-yl)oxy-N-[4-[4-[4-(hydroxymethoxy)phenyl]piperidine-1-carbonyl]pyridin-2-yl]-5-methanimidoylbenzamide [2-[1-(2,3-dimethylphenyl)-5-oxopyrrolidine-3-carbonyl]pyridin-4-yl]carbamic acid N-[(3S,4R)-1-(4-fluorophenyl)sulfonylpyrrolidin-3-yl]-5-methyl-2-phenylpyrazole-3-carboxamide N-butyl-2,3,5-trifluoro-6-methoxyaniline;ethane 2,4-dibromo-6-[3-(3,4,5-trifluorophenyl)propanoyl]benzenesulfonic acid 1-[2-methoxyethyl(propan-2-yl)amino]-3-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]propan-2-ol N-[3-(2,5-dimethylpyrazol-3-yl)-1,7-naphthyridin-6-yl]-4-methoxy-2-methylpentanamide 1,4-bis(3-methylbutoxy)-7-propanoyloxynaphthalene-2-carboxylic acid 2-[(4-ethoxynaphthalen-1-yl)-hydroxymethylidene]propanedinitrile 4-azidooxy-2,6-ditert-butylphenol (4-azidooxypiperidin-1-yl)-[3-methyl-4-[6-(trifluoromethyl)quinazolin-2-yl]phenyl]methanone (Z)-4-[5-[2-(diethylamino)ethyl]-4,6,7,8-tetrahydrothieno[3,2-c]azepine-2-carbonyl]hept-4-enoic acid 1-[3-(hydroxymethyl)piperidin-1-yl]-2,2,2-trifluoroethanone;4-[[3-(4-phenoxyphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]-N-(1,3-thiazol-2-yl)benzamide 3,5-dimethyl-4-[(1S)-1-phenylethyl]-N-(3-pyridin-2-ylpropyl)aniline 1-(1H-indole-4,6-diyl)-5-N-(2-phenoxyphenyl)pyrazole-3,5-diamine (4aR,6S)-N-[2-(1H-indol-3-yl)ethyl]-6-morpholin-4-yl-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine-4-carboxamide 6-bromo-3-(4-fluorophenyl)imidazo[1,2-a]pyrazin-8-amine 4-[5-(4-butylphenyl)thiophen-2-yl]sulfinylmorpholine 1-[(2-azidocyclopentyl)methoxy]-4-chlorobenzene 2-[1-(furan-3-ylmethylamino)ethenyl]phenol 4-(2-fluorophenyl)-1,3-thiazol-5-amine N-[4-methylsulfonyl-2-(trifluoromethoxy)phenyl]acetamide 3-[1-(4-iodophenyl)ethoxy]azetidine 3-[7-chloro-6-(cyclopropylmethoxy)pyridin-3-yl]pyrrolidine-1-carboxylic acid 2-[N-benzyl-4-(carbamoylsulfamoyl)anilino]octanoic acid 2,5-bis[(E)-2-pyridin-1-ium-4-ylethenyl]thiophen-3-ol;bromide 4-azidooxy-1H-quinazoline-2-thione 7-[(6R)-1,1-difluoro-2-hydroxycyclohexyl]-2-[(5-methoxypyridin-3-yl)amino]pyrrolo[1,2-b]pyridazine-3-carboxamide N-[(2R,3S)-1-ethyl-3-methylpiperidin-4-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]acetamide 2-[1-(2,4-difluorophenyl)sulfonylpiperidin-3-yl]oxypyridine 1-(2,3-dihydroxypropyl)-5,6-bis[(3R)-piperidin-3-yl]imidazo[4,5-b]pyridine-7-carbonitrile;hydrochloride 3-(4-chlorophenyl)-2,5-dimethyl-1,3-thiazolidine N-[3,5-dichloro-4-(7H-pyrrolo[2,3-d]pyrimidin-6-yl)phenyl]ethanesulfonamide 3-amino-5-methyl-N,N-bis[(4-methylphenyl)methyl]-2-[6-(oxolan-2-yl)-2-pyridin-2-ylpyrimidine-4-carbonyl]imidazole-4-carboxamide 4-[6-(cyclopropylamino)pyrimidin-4-yl]oxypiperidine-1-carboxylic acid 5-[2,4,7-tris(sulfanylidene)-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidin-5-yl]benzene-1,3-dicarbonitrile (2E)-3-[1-[4-[(5Z,8Z)-7,10-dihydroxyimino-4H-cyclohepta[b]pyran-9-yl]phenyl]ethylideneamino]buta-2,4-dienal 5-(4-fluoro-3-hydroxyphenyl)-2,3-dihydro-1H-pyrido[2,3-e][1,4]diazepine-7,8-dione [3-amino-2-[(4-fluorophenyl)carbamoyl]prop-2-enylidene]azanium 2-(4,5-dimethylpyridin-3-yl)-1H-indole ethane;(3E)-1,2-dimethyl-4-[(Z)-pent-2-en-3-yl]-3-propylidenenaphthalene [3-(1-methyltetrazol-5-yl)phenyl]-[2-[4-(trifluoromethyl)pyridin-2-yl]piperidin-1-yl]methanone N'-[(2S)-1,1,1-trifluoropropan-2-yl]benzohydrazide N-[(4,6-dimethylpyrimidin-2-yl)methyl]-N-propylaniline;hydroiodide 2-benzylsulfanyl-6-(4-chlorophenoxy)-1,3-benzothiazole 2-[3-[[(Z)-aminodiazenyl]carbamoyl]-5-cyclopropylideneoxycarbonylphenyl]acetic acid 1-[3-[(6S)-3,6-dimethyl-1,4-diazepan-1-yl]-5-(1H-pyrazol-4-yl)phenyl]pyrrolidine-2,5-dione 1-methyl-3-[(E)-4-phenylbut-2-en-2-yl]pyrazolo[5,1-d][1,2,3,5]tetrazin-4-one 2-[1,5-dimethyl-4-(oxan-4-yl)pyrazol-3-yl]propanenitrile 6-[[4-(2,5-difluorophenyl)phenyl]sulfonylmethyl]pyridine-3-carboxamide N-[(2-hydroxynaphthalen-1-yl)methylideneamino]-6,7-dihydro-4H-1-benzofuran-5-carboxamide 1-(4,5-dihydro-1H-imidazol-2-yl)naphthalene-2,7-disulfonic acid;hydrochloride (5R,7S)-5,7-dimethyl-N-[3-morpholin-4-yl-1-oxo-1-(2-phenylethylamino)propan-2-yl]-1,4,5,7-tetrahydropyrano[3,4-c]pyrazole-3-carboxamide 2-[(7-chloro-3,4-dihydroisoquinoline-1-carbonyl)amino]-5-(trifluoromethyl)benzamide;ethane 4-[5,6-dimethoxy-2-[[4-(trifluoromethyl)phenyl]sulfonylamino]benzimidazol-1-yl]butanethioic acid 7-fluoro-6,11-dihydrobenzo[c][1]benzoxepine (2S)-1-methyl-4-[[3-(naphthalen-2-yloxymethyl)phenyl]methylideneamino]piperazine-2-carboxylic acid 3-[(4-butylphenyl)diazenyl]-4,5-dihydroxynaphthalene-2-sulfonic acid 2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)naphthalene-1,4-dione (2S)-5,6-diamino-N'-[(1R)-3-oxocyclopentyl]-2-(4-phenylmethoxyanilino)hexanimidamide 3-[4-[(2E,6E)-7-chlorodeca-2,6-dienoxy]phenyl]-1,3-oxazolidine 3-(4-phenylmethoxyphenyl)sulfonylbicyclo[1.1.1]pentane 1-phenyl-3,4-bis(prop-2-enyl)pyrrole-2,5-dione 1-[1-(benzenesulfinyl)indol-2-yl]-3,4-dihydro-2H-quinoline 1-(2,6-difluorophenyl)-7,8-dimethoxy-4-methyl-4H-3,1-benzoxazin-2-one (5R,6S)-3,9-diazatricyclo[8.4.0.02,7]tetradeca-1(10),11,13-triene;hydrochloride 2-methylsulfonyl-4H-pyrido[3,2-b][1,4]oxazin-6-one 3-(3,5-dimethoxyphenyl)-N-[(1S,2R)-2-hydroxycyclopentyl]propanamide 1,7-dihydroxy-3-propylnaphthalene-2-carboxylic acid 2,4-dihydroxy-N-(2-methoxyphenyl)-5-propan-2-ylbenzamide N-(2,6-dimethylphenyl)-5-[[1-[(4-fluorophenyl)methyl]-2,3-dihydropyrrol-3-yl]sulfanyl]-1,3-thiazol-2-amine 3-(4-methylcyclohexa-2,4-dien-1-yl)naphthalen-1-ol N-(3,5-difluorophenyl)-2-[6-methyl-7-[(Z)-prop-1-enyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]cyclohexane-1-carboxamide 4-azido-2-(6-methylpyridazin-3-yl)oxypyridine 1-(3-methylphenyl)-4-propanoylpiperidine-2,6-dione 2-[2,4-bis(trifluoromethyl)phenyl]-N-butan-2-ylacetamide 2-(4,5-diphenyl-1H-imidazol-2-yl)phenol 6-(3,5-ditert-butylphenyl)thieno[3,2-c]pyridine 4-(5,6-dimethoxypyridin-2-yl)-N-[3-fluoro-4-(morpholine-4-carbonyl)phenyl]-1,3-thiazole-2-carboxamide 4-(3,5-dichlorophenyl)sulfanylbutanehydrazide 2-[(4R)-4-tert-butyl-3,5-dimethylcyclohexa-1,3-dien-1-yl]-6-hexan-3-ylquinoline 3-(5-bromofuran-2-yl)-7,7-dimethyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine 4-[(1E,3Z)-1-(2H-pyran-6-yloxy)penta-1,3-dienyl]quinoline 5-[2-(3-azidopyridin-4-yl)oxyethyl]-6,7-dihydro-4H-thieno[3,2-c]pyran 5-ethyl-6,7-dihydroxy-2-pyridin-4-ylchromen-4-one (3R)-4-methoxy-N-[3-methyl-5-[2,2,2-trifluoro-1-hydroxy-1-[6-(morpholin-4-ylmethyl)pyridin-3-yl]ethyl]phenyl]piperidine-3-carboxamide 2-tert-butyl-1-[1-(4-chlorophenyl)-3,3-dimethylbutan-2-ylidene]guanidine 7-benzyl-8-[5-(4,4-dimethylcyclohexa-1,5-dien-1-yl)-2-fluorophenyl]-2H-purine 4-[[4-(4-cyclobutylpiperazin-1-yl)phenyl]carbamoylamino]-2-methylsulfanylthiophene-3-carboxylic acid;ethane 1-[4-chloro-2,6-di(propan-2-yl)phenyl]pyrazole;platinum(2+);4,5,6,7-tetrafluorobenzimidazol-1-ide N-[[1-(3,5-dichloro-2-methoxyphenyl)sulfonylpyrrolidin-3-yl]methyl]ethenesulfonamide 3-[(Z)-but-1-enyl]sulfonylbenzenethiol 1-[(3E)-penta-1,3-dien-3-yl]-2,4-bis[(Z)-prop-1-enyl]benzene [2-(dimethylamino)pyrimidin-5-yl]-[3-(oxan-4-yl)piperidin-1-yl]methanone N-[5-[(3,4-dichlorophenyl)methyl]pyridin-2-yl]-6-fluoro-1H-indole-3-sulfonamide 2-amino-N,3-dimethyl-5-[6-(trifluoromethoxy)pyridin-3-yl]benzamide N-[6-(4-chlorophenyl)pyridazin-3-yl]-2,4,6-trimethyl-N-phenacylbenzenesulfonamide [4-[3-(fluoromethoxy)phenyl]piperidine-1-carbonyl]azanide 5-[3,5-dimethyl-4-(2H-tetrazol-5-yl)phenyl]-N,N-diethyl-2-[1-(6-methylpyridin-2-yl)piperidin-4-yl]oxyaniline 4-azido-1,3-dimethylpyrrolo[2,3-b]pyridine 6-[4-[2-(difluoromethyl)benzimidazol-1-yl]piperidine-1-carbonyl]-3,4-dihydro-2H-pyrazino[1,2-a]pyrimidine-1,8-dione N-benzyl-6,9-dihydro-5H-[1]benzoxepino[4,3-d]pyrimidin-2-amine 1-(4,4-dichlorobutyl)-7,9-bis[3-(trifluoromethoxy)phenyl]carbazole 5-bromo-6-ethyl-N',4-dimethylthieno[2,3-d]pyrimidine-2-carboximidamide 1-(8,9,11-trimethoxy-3-methylsulfanyl-6,7-dihydro-5H-benzo[a]heptalen-2-yl)piperidine 5-[1-(2,4-dimethoxyphenyl)-3-methylpyrazol-4-yl]-3H-1,3,4-oxadiazol-2-one 4-[3-amino-5-(trifluoromethoxy)phenoxy]-N-(2-hydroxyethyl)cyclohexane-1-carboxamide (4R)-4-fluoro-5-methylidene-1,3,6-triazatetracyclo[7.7.0.02,6.010,15]hexadeca-9,11,13,15-tetraen-8-one N-[(2R,3S)-4-amino-2-(hydroxymethyl)-1-phenylbutan-3-yl]-5-[(3Z,5E)-8-chloro-6-fluoro-2-methylideneocta-3,5-dienoxy]pyrazine-2-carboxamide (2Z)-3-[4-(aminomethyl)phenyl]sulfanyl-2-[6-ethoxy-5-[4-[2-fluoroethyl(propyl)amino]phenyl]pyridin-2-yl]iminobutanenitrile 2-(3,4-dimethoxyphenyl)-6-(1,3,4-oxadiazol-2-yl)-N-[1-(2-phenylsulfanylphenyl)ethylideneamino]pyridazin-3-imine 6-bromo-3,5-dimethyl-4H-quinazoline 3-azido-5,6-dimethoxyquinoline 1-azidooxy-3,4-dinitronaphthalene 2-[(6-oxo-4-propyl-1H-pyrimidin-2-yl)sulfanyl]acetic acid 3-amino-1,6-dimethylpyridine;N-cyclohexyl-4-phenylbenzamide 4-[1-(5-chloropyridin-2-yl)pyrrolidin-3-yl]oxy-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine N-[(2-fluoropyridin-4-yl)methyl]-1-propanoylpyrrolidine-3-carboxamide 4-bromo-2,3-dimethylcyclopenta-1,3-diene;4-ethoxycarbonylcyclohexa-2,5-dien-1-olate;oxolan-2-ylmethylidenesilane;zirconium(2+) 5-[2,4-difluoro-3-(trifluoromethyl)phenyl]-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide (2S,4R)-N,7-dimethyl-6-oxo-1-[(2R)-2-phenylpropanoyl]-N-[(1R)-1-phenylethyl]azepane-2-carboxamide [5-azidooxy-1,2-dimethyl-4-(4-propan-2-ylphenyl)hex-3-enyl]benzene 4-(3,5-dimethylphenyl)-6-oxo-2-pyridin-4-yl-1H-pyrimidine-5-carbonitrile (3S,4R)-1-[2-cyclopropyl-6-(trifluoromethoxy)benzoyl]-4-methylpyrrolidine-3-carboxylic acid 4-[(6-chloro-2,3-dimethoxyphenyl)methyl]piperazine-1,3-dicarboxamide N-methyl-3-[5-methylidene-4-(6-methyl-2,3-dihydropyrrolo[1,2-a]imidazole-1-carbonyl)-3H-2,6-naphthyridin-7-yl]benzamide 4-[3-[(1R)-2-(difluoromethoxy)cyclohexyl]phenyl]benzaldehyde;4,6-dimethylpyridine-3-carbonitrile 2-methylsulfanyl-6,8-dioxo-5H-pyrido[3,4-d]pyrimidine-7-carboxylic acid 1-(5,6-dimethylpyrazin-2-yl)-4-[3-(trifluoromethoxy)phenyl]-N'-[2-(trifluoromethyl)pyridine-3-carboximidoyl]imidazole-2-carboximidamide N-[1-(2,3-dihydro-1H-inden-5-yl)imidazol-4-yl]pyridine-4-carboxamide N-[(E)-1-[2-hydroxy-4-methoxy-6-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-3-yl)phenyl]ethylideneamino]acetamide 2-azido-3,4-dimethylnaphthalen-1-ol 1-methyl-5-(2-phenylethenyl)pyridin-2-one [4-hydroxy-5,8-dimethyl-2-(4-phenoxyphenyl)imidazo[1,2-a]pyrazin-6-yl]azanide 6-[4-(2,3-dimethylphenyl)-5-oxotetrazol-1-yl]hexanoic acid N-[5-(4,4-dimethylpiperazin-4-ium-1-carbonyl)-2-fluorophenyl]-6-fluoroquinoline-8-sulfonamide [1-[4-(2,3-dihydro-[1]benzofuro[5,4-c]pyridine-1-carbonyl)-2-methylphenyl]piperidin-4-yl]phosphonous acid 4-amino-6-[(4-chlorophenyl)methyl]-5-fluoro-3-[6-(hydroxymethyl)-1H-benzimidazole-2-carboximidoyl]-1,2-dihydropyridin-2-ol 7-azido-1,3-dibenzyl-5-hydroxy-8-methoxy-4H-imidazo[4,5-c]quinolin-2-one 2-[(4Z)-6-ethoxy-7-methylhepta-1,4,6-trien-3-ylidene]indene 3,5-difluoro-N-[1-(4-methylphenyl)ethenyl]aniline 2,5-di(propan-2-yl)-N-[(E)-(6-pyridin-4-ylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-1H-pyrrole-3-carboxamide [4-(3-butan-2-ylphenyl)cyclohexyl]methanediol N-[4-(1,3-dimethoxybutan-2-yl)phenyl]acetamide 2,3-dihydroxy-4-(7H-purin-6-yl)cyclobutane-1-carboxylic acid 3-(1,2,4-triazol-1-ylmethoxy)-2,6-bis(trifluoromethyl)pyridine 4-[2-(3,5-dimethoxyphenyl)ethylamino]-7H-pyrrolo[2,3-d]pyrimidine-2-carbonitrile (Z)-2-bromo-N-methylidene-N',3-diphenylprop-2-enethioamide;(5E)-5-[(3S)-3-formylpyrrolidin-1-yl]iminopentanal 3-(2-methoxyethyl)-5H-pyrimido[4,5-b]indol-4-one 4-(2,6-difluorophenyl)-5-methyl-1H-imidazole 2-chloro-3,4-diphenyl-5,6-bis(2,4,4-trimethylpentan-2-yl)benzenethiol N-[(E)-2,2-dimethyl-3-nitropropylideneamino]-1H-imidazo[4,5-b]pyridine-7-carboxamide 2-[6-(3,3-difluoropyrrolidin-1-yl)pyridin-3-yl]-4-[(4-methoxyphenyl)methylsulfanyl]-5-propan-2-ylimidazole-1-carboxylate N-[2-(1,3-benzothiazol-6-ylamino)sulfanylphenyl]-4-prop-1-en-2-ylamino]benzamide 3-(2,6-dimethoxyphenyl)-7-[4-[[(2S)-1-hydroxypropan-2-yl]amino]pyrimidin-5-yl]-8H-1,8-naphthyridin-4-one N-[1-(4-methoxybenzoyl)piperidin-3-yl]-5,6-dimethylpyridazine-3-carboxamide 5-[2-cyclopropyl-4-(methylamino)pyrimidin-5-yl]-6-methoxypyridine-3-carbonitrile [5-(4,7-dimethoxynaphthalene-1-carbonyl)thiophen-2-yl]methylideneazanium 4-[5-(1,3-benzothiazol-2-yl)furan-2-carbonyl]-N-(cyclopropylmethoxy)piperazine-1-carboxamide 2-[5-(aminomethyl)-1,3,4-thiadiazol-2-yl]cyclohexan-1-amine;dihydrochloride 3-amino-N,N'-dimethylbenzenecarboximidamide;8-cyclopenta-1,4-dien-1-yl-6-(1,3-oxazol-5-yl)-2H-[1]benzofuro[2,3-b]pyridin-5-one 2-[1,3-benzothiazol-2-yl(methyl)amino]acetamide 2-(4-chlorophenyl)-N'-[N'-(3,5-difluoropyridin-2-yl)carbamimidoyl]propanimidamide N-ethyl-2,6-difluoro-N-[(3R)-piperidin-3-yl]benzamide (3R)-1-[4-(1,2-dihydroxyethylamino)-6-phenyl-1,3,5-triazin-2-yl]pyrrolidin-3-ol 5-methyl-2,4-diphenyl-1H-pyrimidin-6-one 2-[(3S)-1-(4-acetamidobenzoyl)pyrrolidin-3-yl]-N-[5-(2,2,2-trifluoroethoxy)pyridin-2-yl]acetamide (E)-2-[2-[[5-chloro-4-fluoro-7-morpholin-4-yl-1-(4-phenoxyphenyl)benzimidazol-2-yl]oxymethyl]pyrrolidine-1-carbonyl]hept-2-enamide 3-(4-aminocyclohexyl)-N,N-dimethylimidazo[1,5-a]pyridine-6-carboxamide 5-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-2-carbonyl)-1H-pyrrole-3-sulfonamide N-cyclopropyl-3-[2-(difluoromethoxy)pyridin-4-yl]-5-[3,6-dihydro-2H-pyran-4-ylmethyl(methylsulfonyl)amino]benzamide [4-[(2S)-6,15-dibromo-13-methyl-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl]piperazin-1-yl]-pyridin-3-ylmethanone 5-[[3-(4-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]methyl]pyridine-3-carboxylic acid N-(5-acetyl-2,4,6-trimethylphenyl)sulfonyl-1H-indole-3-carboxamide 6-(5-acetyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-2-yl)-8-chloro-1H-quinolin-2-one 1-phenyl-4-(10,12,20-triazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1,3(11),4,6,8,12,14,16,18-nonaen-21-yl)cyclohexane (E)-3-[3-amino-5-(2,4-difluorophenyl)pyridin-2-yl]prop-2-enoic acid 5-[[4-(1-methylindol-6-yl)pyrimidin-2-yl]amino]-N-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]cyclohexa-1,5-diene-1-carboxamide N-[3-(2-chlorophenyl)prop-1-en-2-yl]-5-cyclohexa-1,5-dien-1-yl-4-methanimidoyl-6-morpholin-4-ylpyridin-2-amine (2S)-2-[4-chloro-3-(trifluoromethyl)phenyl]-1-[4-(4,5-dihydro-1H-imidazol-2-ylamino)piperidin-1-yl]propan-1-one 6-fluoro-5-[(3S)-3-propan-2-yloxypyrrolidin-1-yl]pyridine-3-carbonitrile 2-cyclopentyl-1'-(1H-pyrrole-3-carbonyl)spiro[4,5-dihydrothieno[2,3-c]pyran-7,4'-piperidine]-2-carboxylic acid (4E,5Z)-4-[3-amino-6-(3,5-dimethylpyrazol-1-yl)-2H-pyrazolo[3,4-b]pyridin-4-ylidene]cyclohexane-1-carboxylic acid 2-[3-(4-oxo-7,8-dihydropyrido[1,2-a]pyrimidine-6-carbonyl)phenyl]propanamide 5-(1H-pyrrol-2-yl)benzene-1,3-dicarboxylic acid N-[5-(1,3-benzodioxol-5-yl)pyridin-2-yl]-4-[2-(trifluoromethoxy)anilino]cyclohexane-1-carboxamide (3S,4R)-1-[3-(4-chlorophenyl)-2-oxopropyl]-N'-hydroxy-2-oxo-5-piperidin-1-ylpyrrolidine-3'-carboximidamide N-benzyl-2-[4-(diethoxyphosphorylamino)phenyl]acetamide (3Z,5E)-1-(4-aminophenyl)-7-phenylhepta-3,5-dien-2-one 6-(4-methoxyphenyl)-3,4-dihydrobenzo[h]chromene (5S)-6,11-dihydroxy-1-methoxytetracene-5-carboxylic acid (3Z)-3-[3,5-difluoro-4-[2-(oxan-4-ylamino)ethoxy]phenyl]-1-N'-[1-[1-[4-(trifluoromethyl)phenyl]piperidin-4-yl]ethenyl]hexa-3,5-dienehydrazide N-benzyl-N-(2,3-dihydroxypropyl)nonanamide 1-methyl-2-[(4-propan-2-ylcyclohexa-1,3-dien-1-yl)methoxy]benzene 2-[[6-(4,4-dimethylpiperidine-1-carbonyl)pyridin-3-yl]methylamino]acetic acid 2-(1H-benzimidazole-5-carbonyl)-7-[4-cyano-3-(trifluoromethyl)phenyl]-N,N-dimethyl-2,7-diazaspiro[4.4]nonane-8-carboxamide (1S,3R,4S)-3-azido-N'-(2,5-difluorophenyl)-4-methylcyclopentane-1-carbohydrazide 1-(azidomethoxy)-2,3,5-trichlorobenzene N'-hydroxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indazole-1-carboximidamide 6-[(4-chlorophenyl)methyl]-2-cyclopropyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-[3-(4-chlorophenyl)-6,7-dihydroindazol-1-yl]benzamide 5-amino-4-[2,3-dihydro-1H-indene-5-carboximidoyl(methyl)amino]-N-pyridin-2-ylthiophene-2-carboxamide 1,4-bis(3-fluoropropoxy)-2-methylbenzene 3-[(Z)-(2-oxochromen-5-yl)methylideneamino]quinazolin-4-one N-(4-methylsulfonylphenyl)-6,7-dihydroquinoline-5-carboxamide N-(3-azidophenyl)cyclohexanecarboxamide 4-(4-azidobutyl)-3,5-dichloroaniline 1-(3,4-dimethoxyphenyl)hexan-2-ol 2,5-difluoro-4-[7-methyl-6-(1H-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-N-[(2S)-2-pyrrolidin-1-ylcyclopentylidene]benzamide 4-[3-(1,6a-dihydrocyclobuta[a]inden-5-yl)phenyl]-2-methyl-6-[(Z)-prop-1-enyl]pyrimidine 2-[1'-cyclobutylspiro[4,7-dihydrotriazolo[5,1-c][1,4]oxazine-6,3'-piperidine]-3-yl]ethanamine;dihydrochloride 3-[1-(1,4-diazepan-1-yl)-2-methoxyethoxy]-5-propan-2-yloxypyridine 2-[1-azido-3,3-di(propan-2-yl)inden-4-yl]ethanamine (2E)-2-[1-(2,3-dihydro-1H-inden-2-ylamino)ethylidene]-N'-ethyl-4,5-difluorohexanimidamide 2-methyl-N-(1,3-thiazol-5-yl)butanamide 2-[1-(benzenesulfonyl)azetidin-3-yl]-4,5-diphenylimidazole (5Z)-2-ethenyl-4,7-dimethylidene-1-propan-2-yl-5H-3-benzazepine 1-(4,6-dimethylcyclohexa-2,4-dien-1-yl)ethenylbenzene;ethane N-(2,6-dimethoxypyrimidin-4-yl)-1H-imidazole-5-sulfonamide 2-[3-(4-hydroxyphenyl)pyrazol-1-yl]-N-methoxy-5,6,7,8-tetrahydroquinoline-3-carboxamide 5-benzylsulfanyl-2-pyridin-3-yl-4H-pyrimidine 2-[(1R)-2-methylcyclohexyl]oxy-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one 5-chloro-4-[(2,3,6-trifluorophenyl)methoxy]pyrimidine N-[3,4-dimethyl-5-(1,2-oxazol-5-yl)phenyl]pyridine-2-carboxamide 4-chloro-6-[2,5-dimethyl-3-(1-methylpyrazol-4-yl)phenyl]pyrimidin-2-amine 2-amino-4,5-dichlorobenzenecarboximidamide 6-chloro-N-[4-(pyridine-3-carbonyl)-1,2,5-oxadiazol-3-yl]pyridine-3-carboxamide 4-aminobenzenesulfonic acid;3-[(6-ethylpyridin-2-yl)methoxy]-N,N-dimethylpropan-1-amine (2S)-3-[6,8-difluoro-5-methyl-7-[4-oxo-1-[(2-phenylacetyl)amino]pyridazin-3-yl]quinolin-3-yl]oxypropane-1,2-diol N-[4-fluoro-5-[3-[7-(3-methylpyrazol-1-yl)-3H-imidazo[4,5-c]pyridin-2-yl]-1H-indazol-5-yl]pyridin-3-yl]propanamide 3,4-bis(ethenyl)-2-fluoro-1H-indole;ethane 3-[4-(5-chloro-1H-imidazole-2-carbonyl)piperazin-1-yl]oxolane-3-carboxamide 5-[4-(azidomethyl)pyrazol-1-yl]-6,8-dichloroimidazo[1,2-a]pyridine 4-[(3R,4S)-1-[2-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4-yl)ethyl]-4-fluoropiperidin-3-yl]oxybenzoic acid N-[3-[3-(2,6-dioxopiperidin-1-yl)-4H-thieno[3,4-b]pyrazin-7-yl]phenyl]ethenesulfonamide 7-azidooxy-1,3,4,5,9-pentamethylxanthene 4-[4-[5-(2,6-dichlorophenyl)-4,5-dihydro-1,2-oxazol-3-yl]piperidine-1-carbonyl]-3-methoxybenzoic acid [2-(6-fluoropyridin-3-yl)phenyl]methanol 1-[5-chloro-6-(3,3,3-trifluoropropoxy)pyridin-3-yl]sulfonyl-4-(dimethylamino)piperidine-2-carboxamide 3-[6-[[(1S)-4-hydroxycyclohexa-2,4-dien-1-yl]amino]purin-9-yl]benzoic acid N-(2,3-dichlorophenyl)-9H-thioxanthene-1-carboxamide 1-(6-methoxyquinolin-3-yl)pentan-2-ol 5-(6-bromopyridin-3-yl)hexanoate 3-(3,5-ditert-butylphenyl)-2,4,8,9-tetrahydrocyclohepta[d][1,3]thiazole 2-[5-(2,3-dichlorophenyl)sulfanyl-4-propyl-1,3-thiazol-2-yl]-N-hydroxyacetamide (2-benzylcyclopentyl)methanol 5-(7-chloroimidazo[1,2-a]pyridin-3-yl)sulfonyl-N-diazonaphthalene-2-sulfonamide 2-[N-(benzenesulfonyl)-3,5-dichloroanilino]acetamide N-[1-(2,5-dimethylpyrazole-3-carbonyl)pyrrolidin-3-yl]-N-[2-(5-methylthiophen-3-yl)ethyl]acetamide 4-[7-(2,3-dihydroxy-3-methylbutoxy)-1,3-benzothiazol-2-yl]phenol N-[4-[1-(cyanomethyl)-3,5-dimethylpyrazole-4-carbonyl]phenyl]acetamide (2S)-5-[4-amino-3,6-bis(trifluoromethyl)-9H-carbazol-1-yl]-N'-phenylmethoxy-2,3-dihydrofuran-2-carboximidamide 6-(1H-benzimidazol-2-yl)-4-cyclopenta-1,3-dien-1-yl-2-fluorophenol N-[3-(2,6-difluorophenyl)oxetan-3-yl]pyrazine-2-carboxamide 4-azido-2-cyclohexyloxy-1,3-thiazole 2-N,4-N-bis(2-butoxyethyl)-6-[(Z)-[(E)-4-thiophen-3-ylpent-3-en-2-ylidene]amino]pyrimidine-2,4-diamine 6-[(2-methyl-5,6-dihydro-4H-cyclopenta[c]pyrazole-3-carbonyl)amino]hexanoic acid N-(2,6-dichloro-4-nitrophenyl)-N-ethylsulfonylbenzenesulfonamide 4-hydroxy-N-[(3S,5R)-1-[6-(2-methoxyphenoxy)hexyl]-5-pyridin-2-ylpyrrolidin-3-yl]benzamide N-[3-(2,4-dimethoxyphenyl)propyl]-3-ethynyl-5,6,7,8-tetrahydroquinoline-2-carboxamide (6R,9S)-2-amino-6-thiophen-3-yl-8-oxa-4,5,7-triazadispiro[2.6]nonan-3-one 6-fluoro-1-methyl-N-[(4-phenylcyclohexa-2,5-dien-1-ylidene)amino]-2H-pyridine-3-carboxamide N-[4-(3,5-dichlorophenyl)pyridin-2-yl]-6-methyl-2-morpholin-4-ylpyridine-3-carboxamide 4-[2,6-difluoro-3-(trifluoromethyl)phenyl]piperidine 1-[5-amino-3,4-bis(2,6-dichlorophenyl)furan-2-yl]butan-1-one 1-[7-[2,4-bis(trifluoromethyl)anilino]-3-hydroxyiminonaphthalen-2-ylidene]ethanolate N-azido-1-phenylmethoxycyclopentan-1-amine (E)-N-[1,3-dihydroxy-1-[4-(4-methylsulfonylphenyl)piperazin-1-yl]propan-2-ylidene]-3-(6-phenylpyridin-3-yl)prop-2-enamide N-(3,4,5-trimethoxyphenyl)quinazoline-2-carboxamide 5-[6-(4,6-diphenyl-1,3,5-triazin-2-yl)pyridin-2-yl]pyrido[3,2-b]indole (5Z)-2-[2-methoxy-4-(1,3-thiazol-4-ylsulfonylamino)phenyl]imino-N-(3-phenoxyphenyl)-1,3-thiazinane-6-carboxamide [3-[(4,5-dimethylthiophen-2-yl)methoxy]pyrrolidin-1-yl]-naphthalen-2-ylmethanone 2-[2,2-diethoxyethyl(octyl)amino]benzenesulfonic acid (2E,4Z)-2-[1-(cyclopentylmethylamino)ethenyl]-N,5-dimethylhepta-2,4,6-trienamide;(E)-N'-[(3,4-dichlorophenyl)methoxy]-N,3-dimethylhex-4-enehydrazide 4-(4,5-diethyl-1H-pyrazol-3-yl)phenol 5-(difluoromethyl)-N-[2-(dimethylamino)pyridin-3-yl]-4-ethylpyrimidine-2-carboxamide 3-[[4,6-diamino-5-(2-fluoro-4-hydroxybenzoyl)pyridine-2-carbonyl]amino]propanoic acid [5-(3,4-difluorophenyl)sulfonyl-2-methylphenyl]carbamic acid N-[(Z)-3-amino-4,4,4-trifluorobut-1-enyl]-5-[3-cyano-6-(hydroxymethyl)pyridin-2-yl]-2-fluorobenzamide 3-[2-ethyl-5-(1,6-naphthyridin-8-yl)pyrazole-3-carbonyl]-3-azabicyclo[3.1.0]hexane-1-carbonitrile (2Z)-3-cyclopentyloxy-2-[3-(N-phenylanilino)propylidene]-1,3-diazatricyclo[6.4.1.04,13]trideca-4,7,9(13),11-tetraen-12-one N-[6-(4-fluorophenyl)pyridazin-3-yl]butanamide 4-[2,6-dichloro-3-(1,2,4-triazol-1-yl)phenyl]-2H-benzotriazole 1-(cyclohexylmethyl)-2,6-difluoro-4-hydroxybenzimidazole (3S)-5,5-dimethyl-1-[3-(4-propoxyphenyl)quinolin-6-yl]pyrrolidine-3-carboxylic acid 5-[4-(bromomethyl)phenyl]-2H-tetrazole 2-fluoro-5-[4-(trifluoromethyl)pyrimidin-2-yl]oxybenzaldehyde 2-azido-4,5-difluoro-1H-indole 3-[(1R)-2,4-dinitrocyclohexyl]-5-methoxyquinoxalin-2-amine 2-bromo-1H-indole-3,5-dicarboxylic acid (2R)-3,4-dihydroxy-N-[[1-(5-methylpyridine-3-carbonyl)piperidin-3-yl]methyl]-2-propan-2-ylbutanamide 2-amino-N'-[1-(4-tert-butylphenyl)ethyl]-5,6-dimethanimidoylpyrimidine-4-carboximidamide 5-amino-4,7-dioxo-2-(pyridine-3-carbonyl)thieno[3,2-b]pyran-3-carbonitrile 1-[2-methyl-6-(6-oxobenzo[c]chromen-9-yl)oxyhexan-3-ylidene]guanidine 4-chloro-N-ethyl-3,5-dimethoxyaniline 3-[2-(4-ethoxyphenyl)imino-5,6,7,8-tetrahydro-1H-pyrido[3,2-d]pyrimidin-4-yl]aniline 5-[(2-methylpropanoylamino)methoxy]pyridine-3-carboxamide ethane;6-methyl-7-(5,6,7,8-tetrahydronaphthalen-2-yl)imidazo[1,2-a]pyrimidine 2-[1,3-dioxolan-2-ylmethyl(2-hydroxyethyl)amino]-4-fluorobenzoic acid 4-azidooxy-2-[(3-chlorophenyl)methyl]-1,3-thiazole (4R)-3,7-dimethyl-N-[2-[2-(trifluoromethoxy)phenoxy]ethyl]-8,9-dihydro-7H-imidazo[4,5-f]quinoline-6-sulfonamide 2-amino-4,5-bis(ethenyl)-6-methylpyran-2-ol N-[2-(3,4-dimethoxyphenyl)ethyl]-3,5-bis(3,3,3-trifluoropropoxy)aniline 2,6-dimethoxy-4-[5-(1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]phenol 1,5-diphenylnaphthalene;ethane 3-chloro-4-[[2,5-difluoro-3-(trifluoromethyl)phenyl]methyl-[2-[[[1-(ethoxymethoxy)-1-oxopropan-2-yl]amino]methyl]cyclohexanecarbonyl]amino]benzoic acid 3-(3,5-dichlorophenoxy)-1,1-dimethylurea [(3aR,6aS)-5-hydroxy-3a-methyl-2-[6-(trifluoromethoxy)-1H-benzimidazol-2-yl]-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl]-(furan-3-yl)methanone 7-azido-4-phenylcyclohept-2-en-1-one 3-cyclohexyloxy-2,3-dihydrochromen-4-one 6-(8,9,11-triazatetracyclo[7.7.0.02,7.010,15]hexadeca-1(16),3,5,7,10,12,14-heptaen-8-ylmethyl)quinoline (NE)-N-[1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)piperidin-3-ylidene]hydroxylamine 5-[1-(2,4-dihydroxyphenyl)propylideneamino]pentanoic acid (7R)-2,5-dimethyl-7-phenyl-3-propanoyl-N-(2,4,6-trichlorophenyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-6-carboxamide 3-[1,2-dimethyl-4-(4-propan-2-ylphenyl)-6H-phenanthridin-9-ylidene]propane-1,2-diol 2-[5-[(Z)-3-amino-4,4-dimethylpent-1-enyl]thiophen-3-yl]acetic acid (Z)-3-[4-[[(E)-2-[(1R,3S)-2,6,7-trichloro-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]ethenoxy]methyl]phenyl]prop-2-enoic acid (3aR)-N'-[5-[4-(2,6-dichlorophenyl)piperazine-1-carbonyl]pyridin-2-yl]spiro[1,3a,4,5,6,7,8,8a-octahydroquinazoline-2,4'-piperidine]-4-carbohydrazide 1-[4-(2,5-dimethylpyrrole-1-carbonyl)-3-propan-2-ylphenyl]-6H-pyrazolo[3,4-d]pyrimidin-4-one [4-(2,4-dihydroxy-5-propan-2-ylbenzoyl)piperazine-1-carbonyl]-phenylazanium 2-[4,6-bis(2,5-dichlorothiophen-3-yl)-1,3,5-triazin-2-yl]phenol 1-[4-(2,3-dimethyl-5,6-dihydro-[1,3]thiazolo[5,4-b]pyridin-7-yl)phenyl]-5-[3-ethoxy-5-(trifluoromethyl)phenyl]imidazolidine-2,4-dione 3-[(2,6-dioxopiperidin-1-ium-4-ylidene)amino]oxy-N,N-diethylbenzenesulfonamide;chloride 5-(2-acetylindol-1-yl)-1,3-dihydrobenzimidazole-2-thione 3-[1,5-bis(4-chlorophenyl)triazol-4-yl]cyclopentan-1-one N-(2-chloropyridin-4-yl)-5,6-difluoro-N'-methyl-1H-benzimidazole-2-carboximidamide 3-cyclohexylpropanal;(Z,2E)-N-methoxy-1-phenyl-2-propylidenepent-4-en-1-imine 4-(3,3-difluorocyclobutyl)-2-methoxypyridine 1-(4,5-diethylpyrimidin-2-yl)piperidine-3-carboxamide (2S)-4-[4-chloro-7-(4-ethylthiophen-3-yl)quinoline-2-carbonyl]-1-(4,5-dimethoxycyclohexa-1,5-dien-1-yl)piperazine-2-carbonitrile 3-(2,4-dichlorophenyl)-N'-[(Z)-ethylideneamino]propanehydrazide 2-azido-5-[1-[(2S)-pyrrolidin-2-yl]ethylamino]-1,3-benzothiazole-4,7-diol 7-(3-bromophenyl)-2,5,6,8-tetrahydroimidazo[1,2-a]pyrimidine 3-N,4-dimethylbenzene-1,3-disulfonamide 2-[(1R)-2,2,2-trifluoro-1-phenylethyl]naphthalene N-[2-[4-(6-methylquinoxalin-2-yl)piperazine-1-carbonyl]phenyl]-3,3a,5,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrole-1-carboxamide 2-methyl-5-(3-morpholin-4-ylphenyl)furan-3-amine 3-[4-(6-aminopyridine-2-carbonyl)piperazin-1-yl]propanoic acid N'-[(4-fluorophenyl)methyl]-2,6-dihydroxybenzenecarboximidamide ethane;N-[2-methyl-5-(3,4,5-trifluorophenyl)pyrazol-3-yl]formamide [5-(aminomethyl)-2-[8-methoxy-2-(trifluoromethyl)quinolin-4-yl]-1,3-oxazol-4-yl]-spiro[1H-2-benzofuran-3,4'-piperidine]-1'-ylmethanone 5-[4-[2-(3,4-dichlorophenyl)ethyl]piperazine-1-carbonyl]thiophene-3-carboxylic acid [(3R,5S)-3-amino-4,5-dihydroxypiperidin-1-yl]-[2-(5H-pyrrolo[3,2-d]pyrimidin-7-ylmethyl)cyclopenten-1-yl]methanone 2-chloro-5-phenylmethoxypyridine;ethane N-[2-[methyl(thiophene-2-carbonyl)amino]ethyl]pyrazine-2-carboxamide N-(2,6-dimethylphenyl)-4-[5-ethoxy-1-(6-fluoropyridin-3-yl)-1,3,4-triazol-2-yl]-5-fluoropyrimidin-2-amine 3-butylsulfanyl-2,6-dimethoxyquinoxaline 7-chloro-5-cyclopropyl-N-methylpyrido[2,3-d]pyrimidin-4-amine 1-cyclopropyl-3-[6-(furan-2-yl)isoquinolin-3-yl]urea 4-[(2R)-1-(cyclohexylmethoxy)propan-2-yl]-3-[(6-methoxypyridin-3-yl)sulfonylamino]benzoic acid 5-(2,6-dichlorophenyl)sulfanylpyrimidine-4,6-diamine 4-[(3R)-3-aminopiperidine-1-carbonyl]-7-(6-chloropyridin-2-yl)-9-fluoro-2,3-dihydro-1,4-benzoxazepin-5-one (E)-3-[4-[6-chloro-8-fluoro-7-[(2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]oxyquinazolin-4-yl]pyrazol-1-yl]prop-2-enoic acid 6-ethyl-5,8-dihydroxynaphthalene-2,3-disulfonic acid 4-(5,6-dimethoxypyridin-3-yl)-N-[[4-[ethenyl(propyl)amino]phenyl]methyl]aniline 1-[3,4-dihydroxy-5-(pyridin-2-ylmethoxy)oxolan-2-yl]-5-fluoropyrimidine-2,4-dione N-[4-(2,5-dimethylfuran-3-yl)phenyl]sulfonyl-6-piperidin-1-ylpyridine-3-carboxamide 5-(2,4-diaminoquinazolin-6-yl)pyridine-3-carboxylic acid N-(3,4-dimethylphenyl)-2-[(6-oxo-1H-pyrimidin-4-yl)amino]acetamide 1-(3,4-dihydronaphthalen-2-yl)pyrrole 2-bromo-1-[5-(4-chlorophenyl)naphthalen-2-yl]ethanol 2-[(2Z)-2-[(E)-(3,5-difluorophenyl)methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 3-[7-(azidomethyl)-1,2-dihydroquinoxaline-2-carbonyl]oxypropanoic acid (4R)-N'-[2-[3,5-bis(trifluoromethyl)phenyl]sulfanylethyl]-N-hydroxy-1,2-oxazolidine-4-carboximidamide (7-bromoquinolin-3-yl)methanol 4-[3,5-difluoro-N-(2-hydroxyethyl)anilino]benzenesulfonic acid 3-[(4-hydroxyphenyl)methyl]-4,5-dimethoxyphenol N-[2,6-dichloro-4-(trifluoromethyl)phenyl]-3-methyl-5-oxopentanamide (Z,3E)-1-[4-[3-bromo-5-(2H-tetrazol-5-yl)phenyl]phenyl]-N'-hydroxyhexa-3,5-dienethioamide 2-methyl-3-(4-propan-2-ylpyrazol-1-yl)but-2-enenitrile 5-[7-(3,4-dimethylphenoxy)heptoxy]-2-ethylquinoline 2-(3-hydroxyazetidine-1-carbonyl)-7-methoxy-5H-indeno[1,2-b]pyridine-9-carboxylic acid [(2Z)-2,5-dimethylhexa-2,4-dienoxy]methylbenzene 3-bromo-2,5-dimethylpyridine;ethane [1-(azidomethyl)-3,5-bis(trifluoromethyl)pyrazol-4-yl]-[4-[2-(cyclopropylamino)ethyl]piperidin-1-yl]methanone 1-[4-[2-(1H-imidazol-5-yl)ethynyl]phenyl]-N-methylmethanamine N-[3,5-dichloro-4-(2-oxopyrrolidin-1-yl)phenyl]acetamide N-cyclopropyl-2,5-difluoro-3-methoxybenzamide 3-(4,6-diphenyl-1,2,5-triazin-3-yl)naphthalene-1,5-disulfonate N-[(4R)-1-[1-(2,6-dichlorophenyl)ethenyl]pyrrolidin-3-yl]-5-(trifluoromethyl)pyridin-2-amine 3-(diethylamino)-N'-hydroxypyrazine-2-carboximidamide N-(1,3-benzodioxol-5-yl)-2-[7-[4-chloro-N-[(2S)-1-methoxypropan-2-yl]anilino]-[1,3]thiazolo[5,4-d]pyrimidin-2-yl]acetamide 2-azido-4,5-bis[(6-chloropyridin-3-yl)methoxy]benzene-1,3-dicarbonitrile 1-(1,3-benzodioxol-5-yl)-N-[4-chloro-2-[5-methyl-6-(trifluoromethoxy)pyridin-3-yl]phenyl]cyclopropane-1-carboxamide N'-hydroxy-1H-thieno[3,2-c]pyrazole-5-carboximidamide N-(3-aminopropyl)-6,7-dimethoxy-2-phenylimidazo[1,2-a]pyridine-3-carboxamide N-[1-[6-(2-cyano-3,4-difluorophenyl)pyridin-3-yl]ethyl]acetamide N-[3-(2,4-dimethylphenyl)-4-methylidene-6,7-dihydroquinazolin-8-yl]propanamide N-[3,5-bis(trifluoromethyl)phenyl]-2-methylsulfonylethanimidate 3-[1-[2-(4-methoxyphenyl)ethylamino]ethylidene]heptan-2-one 2-N,6,7-trimethylquinoline-2,5-diamine 2-[4-(1,3-benzothiazol-6-ylcarbamoylamino)piperidine-1-carbonyl]-6-fluoro-5H-furo[2,3-b]pyridine-3-carboxylic acid 1-(azidooxymethyl)-2,3-difluoro-4-(trifluoromethylsulfanyl)benzene [(1R,2S)-1-cyclohexyloxy-3-fluoro-2,4-dimethylpentyl]benzene N-[4-[(2S)-5-amino-1-methylpiperidin-2-yl]phenyl]acetamide 5-fluoro-4-[7-fluoro-3-[(2S)-pyrrolidine-2-carbonyl]quinolin-4-yl]oxy-6-methylcyclohexa-1,4-diene-1-carboxamide [2-(3,5-dimethylanilino)pyrimidin-4-yl]-[(2S,4R)-4-hydroxy-2-phenylpyrrolidin-1-yl]methanone 4-(3,5-dichlorophenyl)-6-methylsulfanylpyrimidine N-[2-[(6-chloropyridin-3-yl)amino]ethyl]acetamide 4-[[5,6-bis(ethenyl)pyridin-3-yl]methoxy]-2-piperidin-1-ylquinazoline 2-[(3,4,5-trichloropyridin-2-yl)methylidene]-1H-imidazole N-(diaminomethylidene)-6,7,8,9-tetrahydro-5H-carbazole-3-carboxamide 2-(1,3-dimethyl-5,6-dicyano-8H-carbazol-4-yl)acetate N-[4-(carbamoylsulfamoyl)phenyl]-2,3-dihydroxybenzamide N-[2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl)ethyl]piperidine-4-carboxamide 1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]propan-1-one N-(2,6-difluorophenyl)-4-[5-methyl-7-oxo-3-(trifluoromethyl)-2-[4-(trifluoromethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-6-yl]benzamide 4-chloro-N-[(E)-2,3-dihydropyridin-5-ylmethylideneamino]benzamide 4-[azidooxy(butoxy)methyl]benzenesulfonic acid N-(2,6-difluorophenyl)-7-methylimidazo[1,2-c]pyrimidine-8-carboxamide N-(4-aminophenyl)sulfanyl-3,6-dibromo-2-fluoroaniline 4-[(Z)-1-cyano-2-cyclopentylethenyl]benzenesulfonamide [4-[2,6-dichloro-4-(trifluoromethyl)phenoxy]cyclohexa-1,3-dien-1-yl]urea 2-cyclopropylimino-5-[(4,6-dichloro-1H-indol-3-ylidene)methyl]-3-ethyl-1,3-thiazol-4-ol 2-[1-(benzenesulfonyl)piperidin-4-yl]-6-(oxan-2-yloxymethyl)pyridine 3-(benzylamino)-6-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]pyrazine-2-carboxamide;cyclohexane 2-[2-azidooxy-1-[2-(4-chlorophenyl)ethyl]-1H-inden-4-yl]furan 5-(6-methoxynaphthalen-2-yl)-3,3a,4,5,6,7a-hexahydro-1H-furo[3,4-c]pyridine 1-butyl-3-[(E)-(2,4-dihydroxyphenyl)methylideneamino]thiourea 1-cyclopropyl-2-[4-[6-(3,5-dimethylpyridin-2-yl)oxynaphthalene-2-carbonyl]piperazin-1-yl]ethanone 3-chloro-N-[(2,5-dimethylpyrazol-3-yl)methyl]-N-propan-2-ylpyridine-4-sulfonamide 4-[3-chloro-5-(trifluoromethyl)phenyl]-N-cyano-2,6-dioxo-1H-pyrimidine-5-carboxamide 4-(1,3-dimethylpyrazolo[3,4-c]pyridin-5-yl)phenol 3-azido-2,4,6-trichlorobenzoic acid 1-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-5-yl]-3-(4-methoxyphenyl)urea 4-(3,3-difluoropyrrolidin-1-yl)-6-methoxypyrimidine 2-[3,5-dichloro-4-(4-hydroxycyclohexyl)oxyphenyl]propanoate 4-[(3S)-5-fluorospiro[2H-1-benzofuran-3,3'-azetidine]-1'-carbonyl]-N,N-dimethylbenzamide 2-(3,5-difluorophenyl)sulfonyl-N-hydroxy-1,3,4,6,7,8a,9,10,11,12b-dodecahydropyrazino[2,1-d][1,5]benzodiazocine-10a-carboxamide 1-[(3S,4R)-4-[[(1R)-1-naphthalen-1-ylethoxy]carbonylamino]oxolan-3-yl]pyrrole-2-carboxylic acid N-[(4-cyanophenyl)methyl]-3-hydroxy-9,9-dimethylfluorene-2-carboxamide 6-methoxy-2,3-dimethyl-7H-imidazo[1,5-f]phenanthridine [5-(5,6-dimethoxybenzimidazol-1-yl)pyridine-3-carbonyl]carbamic acid 1-(4,4-difluorocyclohexyl)-3,5-bis(triazol-2-yl)benzimidazol-2-one 2-(difluoromethoxy)-N-[6-[4-[[5-ethyl-3-methanimidoyl-4-(oxetan-3-ylamino)pyridin-2-yl]amino]piperidine-1-carbonyl]pyridin-2-yl]benzenesulfonamide 3-(dimethylamino)-2-fluoro-4-phenylbenzoate 1-[3-[5-chloro-2-(trifluoromethyl)phenyl]cyclopentyl]-N,N-dimethylmethanamine 3-cyclopropyl-1-phenylpyrazolidine 6-[2,6-difluoro-4-(4-hexylcyclohexyl)phenyl]-1,3-difluoro-7-isothiocyanatoisoquinoline 2-[3-[3-(4,6-diphenylpyrimidin-2-yl)phenyl]sulfanyl-2,4-dihydroimidazol-1-ium-1-ylidene]propanedinitrile N'-(4,5-diethoxy-2-nitrobenzoyl)-3-nitrobenzohydrazide N-[4-(4-aminophenyl)sulfanyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-7-id-7-yl]formamide;cyclopentane;uranium(2+) 4-[5-(furan-2-ylmethylidene)-1,3-diazinane-2,4-diylidene]-N,N'-bis(2-methoxyethyl)cyclohexa-2,5-diene-1-carbohydrazide N-(8-fluoroquinolin-3-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carboxamide 2-(4,5,6,7-tetrahydro-1H-indole-3-carbonyl)-5,7-dihydrofuro[3,4-b]pyridine-4-carboxylic acid 4-[(6S,9aR)-8-[2-methoxyethyl(methyl)amino]-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]benzonitrile N-[(2E)-2-[3,4-bis(ethenyl)-6-oxocyclohexa-2,4-dien-1-ylidene]ethyl]-3-phenyl-4H-pyrido[1,2-a]pyrimidine-2-carboxamide 3-[4-hydroxybutyl(phenacyl)amino]propane-1,2-diol N-[(2,4-difluorophenyl)methyl]cyclopropanamine;7-fluorospiro[1H-2-benzofuran-3,4'-piperidine] N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]naphthalene-2-carboxamide 3,5-dimethyl-2-methylidene-1-[(4E)-4-[2-(trifluoromethoxy)phenyl]hepta-2,4-dien-6-yn-3-yl]indole;ethane N-[[3-[[2-(4-chlorophenoxy)acetyl]amino]phenyl]methyl]pyridine-4-carboxamide 6-[(E)-3,3-difluoroprop-1-enyl]-5-[4-[2-(4-pentanoylphenyl)ethynyl]phenyl]naphthalene-2-carboxylic acid 2-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfonylbenzamide 4-(3,5-dichlorophenyl)-2-ethyl-6,6-dimethylheptan-4-ol;1H-pyridine-2,4-dione 1-[3-(1H-indol-2-yl)propyl]piperidine-4-carboxylic acid 2-chloro-N-[(1R,2S)-1-hydroxy-1-phenylpentan-2-yl]-4-methoxypyrimidine-5-carboxamide 7-amino-5-(4,5-dibromo-2-methylphenyl)-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile [2-(3,5-dimethylbenzoyl)-1H-indol-6-yl]carbamic acid (2R)-3-(4,7-dihydroxy-1H-indol-6-yl)-2-methylpropanoic acid;hydrochloride 2-[(1,3,5-trimethylpyrazol-4-yl)sulfonylamino]thiophene-3-carboxylate 1-[2-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-3-yl]ethanone 2-(6,8-diethylthieno[2,3-e]benzimidazol-1-yl)acetohydrazide N-[(4-methoxyphenyl)methyl]-1,1-bis(5-methylfuran-2-yl)ethanimine N-[(2S)-4,5-bis(dibenzylamino)-1-hydroxypentan-2-yl]carbamate N-[(1,6-dimethylpyrazolo[3,4-b]pyridin-4-yl)methoxy]benzenesulfonamide 6-[[4,5-di(propan-2-yl)pyridin-3-yl]amino]sulfanyl-1H-benzimidazole-2-sulfinic acid 2-fluoro-N,N-dimethyl-4-[3-[5-(trifluoromethyl)pyridin-2-yl]piperidine-1-carbonyl]benzamide (2E)-5-(3,4-dimethoxyphenyl)penta-2,4-dienoic acid (2R)-2-methyl-3-[4-methyl-1-(4-methylphenyl)sulfonylpyrrolo[2,3-b]pyridin-5-yl]propanoic acid 3-azido-5-(3,3-difluorocyclobutyl)oxypyridine N-(2,5-dichlorophenyl)-2-[4-methyl-6-oxo-1-[3-(trifluoromethoxy)phenyl]pyrimidin-5-yl]acetamide 3-hydroxy-4-[1,2,2-trifluoro-1-[3-(trifluoromethyl)phenyl]ethoxy]butanoic acid (2R)-2,4-dimethyl-N-[1-(2-propan-2-ylsulfonylbenzoyl)pyrrolidin-3-yl]morpholine-3-carboxamide 4-[4-(benzylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenol 2-(3,4-dimethoxyphenyl)-5-(1,3,5-triazin-2-ylsulfanyl)phenol 2-[[6-(3,5-dichlorophenyl)pyridine-3-carbonyl]amino]acetic acid N-benzyl-2,3,5,6-tetrafluoropyridin-4-amine 4-(2,6-dimethoxybenzoyl)-1H-pyrazole-5-carboxylate 6-[4-(2,3-dihydroimidazo[1,2-a]pyridin-7-yl)phenyl]-5H-1,6-naphthyridine N-(5-tert-butylpyridin-2-yl)-3,4-difluorobenzenesulfonamide (E)-1-[2-methoxy-5-(trifluoromethyl)phenyl]but-1-en-3-one 2-amino-N-[(3R)-1-[4-benzyl-5-(N'-hydroxycarbamimidoyl)thiophen-2-yl]sulfonylpyrrolidin-3-yl]acetamide 4-[2,3-bis(methylamino)phenyl]butanamide 1-azido-4-cyclopentyloxynaphthalene 2,3-difluoro-1-N',7-N'-bis[(4-methylphenyl)methylideneamino]-5-N-piperidin-4-ylbenzene-1,4,7-tricarboximidamide;dihydrochloride [1-(3,5-difluorophenyl)cyclopropanecarbonyl]urea 2-(4,6-diphenylpyrimidin-2-yl)-5,6-dimethoxy-1-benzofuran-3-ol 2-fluoro-N-[4-(8,9,10,11-tetrahydro-3H-pyrazolo[3,4-a]phenanthridin-7-yl)cyclohexyl]benzamide (Z)-3-[4-(cyclopentylamino)-5-methanimidoylpyrimidin-2-yl]iminoprop-1-en-1-amine;6-cyclopenta-1,3-dien-1-yl-N-(cyclohexylmethyl)pyrimidin-4-amine 7-bromo-4,5,6-trimethyl-2,3-dihydro-1H-indene;ethane [(1R,4S)-4-methyl-2-(pyridin-2-yloxymethyl)cyclopentyl]carbamic acid 2-[(4S)-4-[4-fluoro-3-(trifluoromethyl)phenyl]-5-hydroxyimidazolidin-1-yl]-N,N,6,7-tetramethyl-3H-benzimidazole-5-carboxamide N-[3-cyano-4-(pyridin-2-ylamino)phenyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 6-bromo-3-[(2-methylimidazo[1,2-b]pyridazin-6-yl)amino]pyridine-2-carbonitrile 1-[[2,3-bis(trifluoromethyl)phenyl]carbamoyl]cyclopentane-1,4-dicarboxylic acid 2-methyl-4,6-dinitro-N-[(E)-1H-pyrrol-3-ylmethylideneamino]benzamide 2,3-difluoro-4-[(E)-2-(6H-pyrido[1,2-a]indol-5-yl)ethenoxy]benzoic acid 2-(N-(4-bromo-2,5-dimethylphenyl)-3-hydroxyanilino)acetamide 2-[2-bromo-N-(2,2-dimethoxyethyl)anilino]acetic acid (3S,5R)-6-amino-5-[4-fluoro-2-[2-methoxy-3-(1,3-thiazol-2-ylsulfamoyl)phenyl]phenoxy]-N'-hydroxy-3-methylhexanimidamide 2-(1H-indazol-3-yl)-6,7-dimethoxy-1,2-benzoxazol-3-one N-[(4R)-7-fluoro-3,4-dihydro-2H-chromen-4-yl]-6-methoxy-1,5-naphthyridine-4-carboxamide N-cyclohexyl-2,4-dihydroxy-6-(methylamino)benzamide 4-[3-(1H-pyrazol-5-yl)phenyl]-6,7-dihydroquinoline N-cyclopropylsulfanyl-3-[4-(1,4-diazepane-1-carbonyl)phenyl]propanamide 6-amino-4-(3,5-dibromophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 3-[4-[2-(1,8,11-triazacyclododeca-9,14-dien-10-yl)-1H-indol-5-yl]phenyl]propan-1-amine 2-(4,5-dihydroimidazol-1-ylmethyl)naphthalene 4-(azidomethyl)-5-methoxy-1-phenylpyrazole 2-chloro-N-ethylsulfonyl-5-[4-(3,5,6-trifluoropyridin-2-yl)oxyphenyl]sulfanylbenzamide 4-[2-(3,5-dimethylphenoxy)pyridin-3-yl]pyrimidine 1-[4-(aminomethyl)phenyl]piperidine-2,6-dione;hydrochloride 1-[(E)-2-[4,5-dimethoxy-2-[(3,4,5-trifluorophenyl)methylsulfanyl]phenyl]ethenyl]-2,5-bis(ethenyl)-3-methylbenzene;formic acid 2-[(4-azidooxynaphthalene-1-carbonyl)amino]-4,6-dimethylpyrimidine-5-carboxamide (3R)-N'-[1-[4-(1,3-benzoxazol-2-ylamino)phenyl]ethenoxy]pyrrolidine-3-carboximidamide N-(2,5-dichlorophenyl)-4-nitro-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]benzamide N-[2-(3,5-dimethylphenyl)ethyl]-3-thiophen-3-ylpropanamide N-(7-azaspiro[3.5]nonan-2-ylmethyl)-4,6-difluoro-1H-indole-2-carboxamide;hydrochloride 4-[[7-fluoro-3-(2,4,6-trimethylphenyl)imidazo[1,2-a]pyridin-8-yl]amino]-N-hydroxybenzamide 4-[(3,5-dichloropyridin-2-yl)methoxy]-6-(trifluoromethoxy)-1H-indole 1-(3,4-dimethoxyphenyl)-4-[5-ethyl-6-[ethyl(propan-2-yl)amino]pyridine-3-carbonyl]piperazin-2-one;ethane N-[3-(4-ethylpiperazine-1-carbonyl)phenyl]thiophene-2-carboxamide N-(4-ethenoxycarbonyl-2-methylphenyl)benzenecarboximidate 2-[3-(4-methoxybutylamino)cyclopentyl]isoindole-1,3-dione 4-[(2-aminophenyl)diazenyl]naphthalene-1,5-disulfonic acid 4-[(5-azido-2,3-dihydroindol-1-yl)methyl]phenol 2-methyl-3-phenyl-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine;hydrochloride N-(2,6-dichlorophenyl)-2-[4-[(2E)-2-[1-(1H-indol-3-yl)ethylidene]hydrazinyl]-2-methoxyphenoxy]acetamide 3-amino-N'-[1,4-dimethyl-2-(thiophen-2-ylmethoxy)indol-5-yl]-3-thiophen-3-ylpropanimidamide (3S,4R)-1-benzyl-4-pyridin-2-ylpyrrolidine-3-carboxylic acid [4-amino-2,5-dichloro-3-methylsulfanyl-6-(trifluoromethyl)phenyl]methanol 2-amino-7-[1,3-bis(4-chlorophenyl)propyl]pyrrolo[3,2-d]pyrimidine-6-carboxylic acid 4-(5,5-dimethylhexyl)benzoic acid N-methyl-1-(2-methylphenyl)-3-phenyldiazenylindol-6-amine 2-(3,5-dimethylpyridin-4-yl)propanamide;ethane (3R,4S)-1-[3-bromo-5-(trifluoromethyl)pyridin-2-yl]-N-[2,6-difluoro-4-[2-[(2R)-oxolan-2-yl]ethoxy]phenyl]-4-fluoropiperidine-3-carboxamide [3-amino-4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-pyrrolidin-1-ylmethanone 4-(1,5-dihydropyrazole-2-carbonyl)-N-[(E)-(2-hydroxyphenyl)methylideneamino]benzamide N-[(4-chlorophenyl)methyl]-2-[3-(6-cyanonaphthalen-2-yl)propanoylamino]-3-methylbutanamide 1-(3,5-dimethyl-2H-pyrrol-4-yl)-N-[2-(methylideneamino)ethyl]-N-phenylethenamine;ethane 1-[3-[2-[(5-methylfuran-2-yl)methylidene]hydrazinyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyrazole-3-carboxylic acid (3S)-4,6-dichloro-3-hydroxy-2,3-dihydrochromen-4-ol 4-[N-(1-carboxyheptyl)anilino]benzoic acid [4-[3-(hydroxymethyl)-4-phenylmethoxyphenyl]-1,3-thiazolidin-2-ylidene]cyanamide N-[(5R,7S)-2-azido-6-ethoxycarbonyl-9-oxa-1,3,9-triazatricyclo[8.4.0.02,7]tetradeca-10,12-dien-5-yl]-3-methoxybenzamide 2-(hydroxymethyl)butanedioate;1-[4,5,7-tris(sulfanylidene)-3H-pyrimido[4,5-d]pyrimidin-2-yl]piperidine 5-(2,3-dimethoxyphenyl)-N'-hydroxyhexanimidamide 2-(4-azido-3-chlorophenoxy)-N,N-diethylacetamide 4-(3,4,5-trifluorophenyl)cyclohexane-1-carboxamide 5-(4,6-dimethoxypyrimidin-2-yl)-3-hydroxy-1H-pyridin-2-one 4-[3,5-bis(trifluoromethyl)phenyl]-3-cyanopyrrole-1-carboxylic acid N-[3,4-dihydroxy-5-(2-iodooxyphenyl)pentyl]formamide 2-[1-(2,3-dimethylphenoxy)propan-2-yl]-1H-imidazole 2-[3,5-dichloro-4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1-(4-ethoxycyclohexa-1,3-dien-1-yl)-3-[2-(trifluoromethyl)pyridin-4-yl]urea 4-[7-(1,3-benzodioxol-5-yl)-2-ethylimidazo[1,2-a]pyrimidin-3-yl]-N,N-dimethylaniline 4-amino-2-[1-(cyclopenten-1-yl)ethylsulfanyl]-1H-pyrimidin-6-one 2-[3,5-bis(4-fluorophenyl)-1H-pyrrol-2-yl]ethanol N-[(2-imidazol-1-ylphenyl)methyl]-3,4,5-trimethoxybenzamide 3-(4,5-dichloro-1H-benzimidazol-2-yl)propan-1-amine N-[(4Z)-4-[3-aminopropan-2-ylidene-(2,6-dichlorobenzoyl)azaniumyl]hexa-1,5-dien-2-yl]-4-fluorobenzenesulfonamide 4-cyclopentyl-2,6-diphenyl-1H-1,3,5-triazine [5-chloro-4-(2,3-dihydroindol-1-yl)pyrimidin-2-yl]hydrazine 4-azidooxy-3-chloro-2,6-dimethylaniline 4-[[6-(cyclohexa-1,5-dien-1-ylmethoxy)pyridine-3-carbonyl]amino]-2-(3-hydroxy-4-oxopiperidine-1-carbonyl)benzoic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-chloro-5-[4-[(2-chloroacetyl)amino]phenoxy]benzamide (4-chlorophenyl)-[3-methyl-2,6-dimethylidene-4-[3-oxo-7-[[1-(pyridine-4-carbonyl)piperidin-4-yl]amino]-4H-quinoxalin-2-yl]piperazin-1-yl]methanone 2-ethoxy-N-[4-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-3-yl)cyclohexyl]acetamide (2S)-5-methoxycarbonyl-6-[3-(4-nitrophenyl)sulfonylpropanoylamino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid 6-butyl-5-(2,4-dimethoxyphenyl)-3-[2-(4-nitrocyclohexa-1,3-dien-1-yl)ethyl]pyrimidin-4-one 5-chloro-4-[(2S)-3,3,3-trifluoro-2-hydroxypropoxy]pyridazine-3-carboxamide 2-[1-[3,5-bis(trifluoromethyl)phenyl]ethoxycarbonylamino]-4-(ethoxycarbonylamino)-5-fluoropyridine-3-carboxylic acid 5-azido-2,3-dimethyl-6-phenylpyridine 4-[3-ethenyl-2-fluoro-6-(triazol-1-yl)pyridin-4-yl]piperazine-1-carboxylic acid 2-[4,6-bis(3,4,5-trimethoxyphenyl)-1,2,3,4-tetrahydro-1H-pyridine-2-carbonyl]benzoic acid 4-(3-methoxyphenyl)-2-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-1H-pyrimidin-6-one 2-(5-chloro-1H-indole-3-carbonyl)-6,7-dimethoxy-4H-benzo[f]isoindole-1,3-dione 2-azido-4,5,6-trimethyl-1H-indole 4-hydroxy-N,2,5-trimethylpyrazolo[1,5-a]pyridine-3-carboxamide 3,6-dichloro-2-(4-propan-2-ylcyclohexa-1,5-dien-1-yl)phenol (E)-3,7-bis[2-(benzylamino)ethyl]-6-(furan-3-carbonylamino)non-5-enoic acid 1,3-dimethyl-6-[2-(2-methylbutanoyl)pyrrolidine-1-carbonyl]pyrimidine-2,4-dione 2-(6-bromopyridin-3-yl)-N,3-diphenylpropanamide 4-(cyclobutylmethylamino)-5-iodo-1H-pyrimidin-6-one 1-(2,4-dichlorophenyl)-N-[2-(5,6-dimethoxypyridin-3-yl)-4-morpholin-4-ylquinazolin-7-yl]ethanesulfonamide 3-(6-chloronaphthalen-2-yl)sulfonyloxy-5,7-difluoronaphthalene-1-sulfonate N'-(9H-fluoren-1-yl)hexanediamide 2-amino-6,7-dichloro-3H-quinazolin-4-one (2S)-6-[4-[2,6-dimethoxy-4-(phenylcarbamoylamino)phenyl]piperazine-1-carbonyl]-2,3-bis(phenylsulfanyl)heptanamide 3-(4-chlorophenyl)-5-[1-[cyclopropylidene-(pyridin-4-ylamino)methyl]piperidin-2-yl]-N,N-dimethylimidazole-4-carboxamide 5-chloro-2-[[(3S)-pyrrolidin-3-yl]amino]pyridine-3-carboxylic acid;hydrochloride 2-(dimethylamino)-1-[2-(8-nitroquinolin-4-yl)piperazin-1-yl]ethanone 2-azido-3-(2,3,4-trichlorophenyl)imidazo[1,2-a]pyridine 2-(3,4-dimethoxyphenyl)-1H-imidazo[4,5-b]pyridine 1-[4-(furan-3-yl)-5-methylpyrrolo[3,2-d]pyrimidin-7-yl]ethanone 3-(3,4-dimethoxyphenyl)-N-[2-(N'-hydroxycarbamimidoyl)pentyl]propanamide 5-[(4-chlorophenyl)methyl]-6-(4-hydroxycyclohexyl)oxy-N-[2-(1-iodoethoxyamino)-2-oxoethyl]-4-oxothieno[3,2-c]quinoline-8-carboxamide 4-methyl-N'-[3-(4-methylpiperazin-1-yl)propanoyl]benzohydrazide 6-[(4,5-dimethoxycyclohexa-1,3-dien-1-yl)amino]pyrimidine-2,4-dione 3-[(4R)-1-tert-butyl-4,5-dimethyl-2-phenyl-6H-triazolo[4,5-d]pyrimidin-7-ylidene]-1H-indol-2-one N-ethyl-2,3-dihydro-1H-indene-5-carboxamide 2-[4-(1,3-benzodioxol-5-yl)phenyl]-7,10-dimethoxy-6H-[1,3]benzothiazolo[5,6-c]chromene 6-[5-(4,5-dihydro-1H-imidazol-2-yl)pyridin-3-yl]oxy-N-ethyl-4H-azepine-7-carboxamide 1-[(Z)-2,3-dihydro-1H-1-benzazonin-7-ylmethylideneamino]-3-ethylthiourea 5-azidooxy-4-bromo-N-(2,3-dihydrofuro[2,3-b]pyridin-4-yl)pyridine-2-carboxamide N-[1,4-di(butanoyl)isoquinolin-7-yl]-3,5-bis(trifluoromethyl)benzamide 1-[4-(N'-hydroxycarbamimidoyl)phenyl]-3-pyridin-2-ylurea 1-(2,3-dihydroindol-1-yl)-5,6-bis[(4-methoxyphenyl)sulfanyl]pyrazolo[3,4-d]pyrimidine 3-chloro-4,5,6-trifluorobenzene-1,2-disulfonic acid 1-azidosulfanyloxy-2,3,4,5,6-pentafluoronaphthalene 5-amino-4-[3-methyl-2-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 4-[2,5-dimethylhexyl(propan-2-yl)amino]benzamide N-[5-(2,3-dihydro-1H-pyrrol-4-yl)-1-methylpyrazol-3-yl]formamide;2-formamido-1-phenylcyclopropane-1-carboxamide 2-tert-butyl-6-(cyclohexatrienyl)-4-methylpyridine N-[(1S)-1-cyclopropylethyl]-2-methoxy-6-[(3R,4R)-4-[(5-methylpyridine-2-carbonyl)amino]oxan-3-yl]pyrimidine-4-carboxamide 4-(4-nitrophenyl)piperidine-1,4-dicarboxylate (2Z,3E)-3-ethylidene-4H-1-benzothiocine 6-bromo-3-[1-(6-bromopyridin-2-yl)ethoxy]-2-methanimidoylaniline 3,6-dibromo-4-(4-chlorophenyl)benzene-1,2-disulfonic acid 2-[2-amino-3-(2-methylpropanoyloxy)propanoyl]benzoic acid N-[5-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-2-yl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-2-carboxamide 4-N-[5-(difluoromethyl)pyridin-2-yl]pyrimidine-2,4-diamine;hydrochloride 3-[3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)propoxymethyl]benzonitrile 5-[(E)-2-(4-chlorophenyl)ethenyl]-6,7-dihydro-1H-indazole [2-(1H-indol-3-yl)ethyl-(4-methoxybutanoyl)amino]carbamic acid 2-methylsulfanyl-6,7,8,9-tetrahydropyrido[3,4-b]indolizine 3-amino-5-[2-(4,6-dimorpholin-4-yl-1H-triazin-2-yl)phenyl]-N-piperidin-4-ylimidazole-4-carboxamide (3E)-5-bromo-N-[2-bromo-4-[[2-[1-hydroxyethenyl(methyl)amino]acetyl]amino]phenyl]-2,2,6-trimethylhepta-3,5-dienehydrazonate 4-[1-(2,5-dichloropyrimidin-4-yl)oxyethyl]benzoic acid 2-[5-(3,4-dihydroquinolin-6-yl)-1H-imidazol-2-yl]propanamide 5-[4-amino-6-[methyl-[2-(1-morpholin-4-ylethoxy)ethyl]amino]pyrimidine-5-carboximidoyl]benzene-1,3-diol 2-[[4-(1,3,3a,4,6,6a-hexahydrofuro[3,4-c]pyrrole-5-carbonyl)phenyl]methyl]pyridazin-3-one 4-(2,4-difluorophenoxy)-6-(7H-pyrrolo[2,3-d]pyrimidin-4-yloxy)pyridine-3-carboxamide 1,4-bis(2-methylphenyl)piperidine-4-carbodithioate ethane;1,2-difluorobenzene;N-(3-methoxyphenyl)sulfanylpyridin-4-amine 2-[4-amino-5,6-bis(4-chlorophenyl)pyrimidin-2-yl]phenol 2-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-ylmethyl)pyridine-2,4-dicarboxamide;hydrochloride 2-N,6-N-dimethyl-4-[2-(2-methylphenyl)ethyl]pyridine-2,6-dicarboxamide 4-[(1R)-2,3-dihydro-1H-inden-1-yl]cyclohexan-1-amine 1-[(3S,4R)-3,4-bis(phenylmethoxycarbonyl)cyclopentyl]-5-oxopyrrolidine-2-carboxylic acid N-(2-methylpropanoyl)-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxamide 2-chloro-7-[(4R)-3,4-dihydroxypyrrolidine-1-carbonyl]-10H-phenothiazine-1-carboxamide N-[1-(3,4-dichlorophenyl)ethyl]-N'-hydroxyheptanediamide 4-tert-butylbenzaldehyde;2-(dimethylamino)-5-[[6-ethoxy-2-[(1Z,3E)-3-methoxy-2-methylidenepenta-1,3-dienyl]-1H-indole-3-carbonyl]amino]benzoic acid N-[(1R,2R)-2-methoxycyclohexyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 4-(2,6-dichlorophenyl)-5H-1,3-thiazol-2-one 3-[4-[4-(2,2-difluoroethoxy)phenyl]piperidin-1-yl]sulfonylpyridine 1-[3-(6,7-dichloro-1H-indol-2-yl)-5-(trifluoromethoxy)phenyl]ethenol 2-[4-(aminomethyl)phenyl]sulfanyl-6-chloro-7,8-dihydropyrimido[1,2-a]pyrazin-4-one;hydrochloride 1-(5-tert-butyl-4-chlorothiophene-2-carbonyl)-2,3-dihydroindole-6-sulfonic acid 1-[2,4-bis(phenylmethoxy)-5-propan-2-ylphenyl]ethyl-butylphosphinic acid 6-[2-(3,5-difluorophenyl)morpholine-4-carbonyl]-1H-pyrimidine-2,4-dione N-(2-chlorophenyl)-5-methyl-7-oxo-8H-[1,3]thiazolo[4,5-h]chromene-6-carboxamide 2-methyl-5,6-dioxo-7-[(1R)-1-phenylethyl]-3,8-dihydropyrrolo[3,2-f]quinazoline-9-carbonitrile 4-(2-methylpyridin-3-yl)-1,3-dihydrofuro[2,3-f]benzimidazole 2-(1,3-benzothiazol-2-ylsulfanylmethyl)-4-[(4-bromophenyl)diazenyl]-5-phenyl-1H-pyrazol-3-one 5-[1-(2-phenylethyl)piperidin-3-yl]imidazolidine-2,4-dione [4-[5-(hydroxymethyl)-4-oxo-7-phenylpyrano[3,2-c]pyrazole-3-carbonyl]piperazin-1-yl]-methylborinic acid ethane;1-[(4-ethylphenyl)methyl]cyclohepta-1,3,5-triene 6-(4-cyclohexylphenyl)-3,6-dimethoxy-1,2,8,8a-tetrahydroindolizine;ethane (4R)-3-[5-(2-chlorophenyl)sulfanyltetrazolo[1,5-c]quinazolin-8-yl]-1-(6-methoxypyridin-2-yl)-4-phenylimidazolidin-2-one N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-4-(3-phenylpropyl)benzamide (3E,5Z)-6-chloro-2,4-dimethylidenehepta-3,5-diene;ethane;methanol;N-[2-[2-[5-methyl-3-oxo-7-propyl-1-[4-(trifluoromethoxy)phenyl]-1H-2,6-naphthyridin-8-yl]ethyl]pyridin-4-yl]formamide 2-[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]oxyacetamide 1-[2-cyclopropyl-6-(oxan-4-yloxy)pyridin-3-yl]cyclobutane-1-carboxylate (NE)-N-[5-(2-chlorophenyl)thiophen-3-yl]propanamide 2-[3-(1,4,5,7-tetrahydropyrrolo[2,3-c]pyridin-6-yl)-2H-pyrazolo[3,4-b]pyrazin-6-yl]phenol 2-[(E)-(4-methoxy-3,5-dimethylpyridin-2-yl)iminomethyl]phenol 2-(N,6-dibenzoyl-1,3-benzothiazol-5-yl)acetamide 3-azido-5-methylbenzenesulfonamide N-cyclopropylsulfanylaniline;ethane;1,4-xylene 3-[2-(5-chlorofuran-2-yl)pyrimidin-4-yl]-1,4,6,7-tetrahydropyrano[4,3-c]pyrazole (2S)-N-[[5-[4-fluoro-3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]methyl]butanamide 3-[4-(2,3-dihydro-1H-pyrrol-5-ylmethoxy)phenyl]propanamide 4-[2-hydroxyethyl(propan-2-yl)amino]-3-nitrobenzoic acid 2-[(3Z)-5-fluoro-3-methylhexa-1,3,5-trien-2-yl]furan 2-[3,5-bis(2-pyridin-4-ylethynyl)phenyl]propanamide 1-[4-(N'-hydroxycarbamimidoyl)phenyl]pyrrolidine-3-carboxylic acid;hydrochloride 2-[4-bromobutan-2-yl(prop-2-enyl)amino]phenol 2,3-bis(5-methylfuran-2-yl)quinoxaline [4-methyl-5-[3-[2-(trifluoromethoxy)phenoxy]propoxy]pyridin-2-yl]methanimine 6-[2,4-bis(trifluoromethyl)phenyl]imidazo[1,2-a]pyridine 2-[4-azido-1-(5-fluoropyridin-3-yl)cyclohexa-2,4-dien-1-yl]acetonitrile (2R)-4,4-difluoro-5-oxo-N-[1-(piperidine-1-carbonyl)-3-phenylcyclopentyl]pyrrolidine-2-carboxamide 1-[2,3-bis(4-methoxyphenyl)phenyl]-N'-methylethane-1,2-diimine 3-[2-(3,4-dihydroisoquinolin-1-yl)ethynyl]-4-methoxy-N-[3-[(2S,4R)-2-methylpiperidin-4-yl]phenyl]benzamide 2-(4-chlorophenyl)-1,3-dioxoisoindole-5-carboxylate 1-methyl-2-[(2Z,4E)-5-phenylhexa-2,4-dienylidene]indole N-(1-hydroxyethyl)-3-[2,4,6-trimethyl-5-(3-oxobutanoylamino)cyclohexa-2,4-dien-1-ylidene]benzamide 4-[7-[3-(aminomethyl)phenyl]imidazo[1,2-a]pyridin-3-yl]quinoline-8-carbonitrile 2-methyl-1-(7H-purin-6-yl)benzimidazole N-(3,4-difluorophenyl)-6-ethylsulfanylpyrimidin-4-amine 4-N-[3-(1,2,4-triazol-1-yl)cyclobutyl]pyrimidine-2,4-diamine 1-[2-amino-3,5-bis(trifluoromethyl)phenyl]propan-1-one 5-tert-butyl-2-(4,6,7-trimethylspiro[1H-indole-3,3'-oxetane]-2-ylidene)-1,3-dihydroindole N-[3,5-bis(4-fluorophenyl)-1,2,4-triazol-1-yl]cyclopropanecarboxamide 2-amino-5-[(4-methoxypyridin-3-yl)carbamoyl]benzoic acid 4-cyclopropyl-2-[4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazin-1-yl]quinoline-8-carboxamide N-(2,3-dihydroindol-1-yl)-4-methoxybenzamide 6-fluoro-8-methoxy-2,3-diphenyl-1H-quinolin-4-one 5-[4-chlorobutyl(hexylamino)amino]naphthalene-2-sulfonic acid 1-[2,6-dichloro-3-fluoro-4-(iodomethyl)phenyl]piperidine 3-(2,5-difluorophenyl)-1-methylpiperidin-2-one [3-(4-chlorophenyl)-2,6-dimethyl-2,3-dihydroindol-1-yl]-(7H-purin-6-ylamino)methanol (2-azidooxy-1,3-benzodioxol-4-yl)methanamine 5-[4-(2-propan-2-ylphenoxy)phenyl]sulfonylpentanoic acid 5-chloro-4-[2-methyl-6-(1,3-thiazol-2-yl)pyridin-4-yl]pyrimidin-2-amine 4-[1-(benzenesulfonyl)azetidin-3-yl]benzoic acid N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-ylmethyl)-1H-indole-7-carboxamide 2-[2-(4-fluorophenyl)piperazine-1-carbonyl]oxyethyl-dimethylsulfanium 1-[(3S,4R)-3-methoxy-4-(1-methyltriazol-4-yl)pyrrolidin-1-yl]propan-2-one 1-[(2,4-dichlorophenyl)methyl]-3-methoxybenzene;ethane 5-[(3S)-1,2-dioxo-1-phenylpentan-3-yl]-N-hydroxythiophene-2-carboxamide 4-[(3S)-1-[2-(3,5-dimethoxyphenyl)acetyl]piperidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-6-one N-[1-methyl-2-oxo-3-[4-(trifluoromethoxy)phenyl]benzimidazol-5-yl]formamide 2-[5-(4-carbamoylphenyl)thiophen-3-yl]oxyacetic acid 5-[(2S)-2-aminopropoxy]quinazoline-8-carboxylic acid N-(2,6-dichlorophenyl)sulfonylspiro[1H-4,6-naphthyridine-3,1'-cyclohexane]-7-carboxamide 1,1-dioxo-6H-benzo[e]indazole-3-carboxylic acid 1-[(6S)-2,6-dimethylmorpholin-4-yl]-4-(2-ethoxypyridin-3-yl)butan-1-one 1-[(4R,5S)-5-(3-methoxyphenyl)azocan-4-yl]propan-1-one 2-[2-(difluoromethoxy)-4-methylphenyl]-5-ethoxyphenol N-[[3,5-bis(trifluoromethyl)phenyl]-phenylphosphoryl]hydroxylamine 2-chloro-1-(2,3-dimethylphenyl)naphthalene 2-(N-methylsulfonylanilino)-1-phenylethanone 5-bromo-2,3-diphenylquinoxaline 1-ethyl-3-[2-(2-oxo-1H-cyclohepta[b]pyridine-3-carbonyl)-2,10-diazabicyclo[9.4.0]pentadeca-1(15),11,13-trien-12-yl]thiourea 4-amino-2-(3,5-dimethylimidazol-4-yl)sulfanyl-1H-pyrimidin-6-one [1-[(E)-4-phenylbut-3-enoxy]cyclopropyl]methanol N-[(2,5-dimethylphenyl)-[2-(trifluoromethoxy)phenyl]methyl]propanamide [4-methoxycarbonyl-3,6,7,8-tetrahydro-2H-furo[3,2-e]indol-5-yl]boronic acid (7S)-2-[3,4-bis(phenylmethoxy)phenyl]-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carbonitrile 3-[4-(difluoromethoxy)phenyl]-2-(3,5-difluoropyridin-1-ium-1-yl)-6-(methanesulfonamido)benzoate 2-[3-fluoro-4-(1,1,2,2,2-pentadeuterioethoxy)phenyl]-5-(trifluoromethyl)-1H-pyridazine 4-azidooxy-2,6-dimethyl-3-phenoxyaniline 7-[3,5-dimethoxy-4-(trifluoromethyl)phenyl]heptan-1-amine 5-azido-1-[(3,4,5-trichlorophenyl)methyl]pyrrolidine-2,4-dione [4-(3,5-difluorophenyl)cyclohexyl]methanol;4-(1-ethyl-2-hydroxyindol-6-yl)phenol N-[2-amino-4-(1,1,1,3,3,3-hexafluoropropan-2-yl)phenyl]-2,2-dimethoxyacetamide 3-(2,4-dichlorophenyl)-N,4,5,6-tetrahydro-1H-cyclopenta[c]pyrazole-4-carboxamide 2-[3,5-bis(trifluoromethyl)phenyl]sulfanylbenzene-1,4-diamine 2-[3-(cyclopropylmethoxy)-4-fluorophenyl]acetic acid 3-[(2,4-dihydroxyphenyl)-(9H-xanthen-9-ylmethoxycarbonylamino)methylidene]oxolane-2,5-dione 2-[3-[(4R)-1,8-diamino-6-fluoro-7H-imidazo[4,5-g]quinazolin-4-yl]phenoxy]acetic acid 1,3-difluoro-5-[4-(4-hexylcyclohexyl)phenyl]-2-(trifluoromethoxy)benzene 1-[4-[2-(3,5-dimethylphenyl)propan-2-yl]cyclohexa-1,5-dien-1-yl]ethanethiol (4-azidooxy-3,6-dimethylpyridazin-1-yl)hydrazine 4-chloro-5,5a-dimethyl-6a,7-dihydrocyclopenta[c]indole;ethane 4-(3,6-dimethylimidazo[1,2-b]pyridazin-2-yl)phenol 2-[1-azido-4-(6,7-difluoroquinoxalin-2-yl)piperazin-2-yl]propan-2-ol 3-chloro-N,5-dimethylbenzamide;ethane 2-methoxy-6-[4-(trifluoromethyl)phenyl]-1,5-naphthyridine (3R)-1,3-bis[2,6-di(propan-2-yl)phenyl]-2H-imidazole;cadmium(2+);ethoxymethane;oxygen(2-) 2-[[1-(2-chlorophenyl)-5-(dimethylamino)pyrazole-4-carbonyl]amino]-2,3,3a,9b-tetrahydrofuro[3,2-b]chromene-6-carboxamide 2-[3-(carboxymethyl)-5-ethenylphenyl]acetic acid N-(5-azidopyridin-2-yl)-6-methoxypyrazin-2-amine N-(4,5-dihydro-1H-pyrazol-2-yl)-6-[[4-(trifluoromethoxy)phenyl]methylamino]pyridine-3-carboxamide [3-chloro-2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)phenyl]methanamine;hydrochloride 1-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-3-ethylurea 5-[4,6-bis(4-fluorophenyl)pyridin-2-yl]oxy-3,4-dimethoxycyclohexa-1,3-diene-1-carboxylic acid 6-(4-hydroxyphenyl)imidazo[2,1-b][1,3]thiazole-5-carboxylic acid 3-(4-chlorophenyl)-6,8-dimethoxy-2H-chromene 1-[1-ethylsulfonyl-7-(2-methoxyphenyl)sulfanylindole-4-carbonyl]piperidine-4-carbonitrile 1-(2,5-diphenylphenyl)-3,7-bis[2,6-di(propan-2-yl)phenyl]benzotriazol-1-ium 1-[3,4-dimethoxy-5-(trifluoromethyl)phenyl]propan-2-one N-(4-methoxypyrimidin-2-yl)piperidine-1-carboxamide 2-amino-6-(4,5,6,7-tetrahydrothieno[3,2-c]pyridine-3-carbonyl)-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one 2-[4-(azidomethyl)phenoxy]-1,3-benzothiazole (2S,4S)-2-methyl-5-oxo-4-[(4-phenylphenoxy)methoxy]pyrrolidine-1-carboxylic acid N-(4-azidophenyl)-4-methylpyridine-2-carboxamide 2-(4-methylphenyl)-3H-imidazo[5,1-f][1,2,4]triazin-4-one N-(2-cyanoethyl)-3,4-dimethyl-2-[1-[4-(pyridine-2-carbonylamino)phenyl]butylcarbamoylamino]pentanamide [4-[(5-cyclohexylpyrrolo[3,2-d]pyrimidin-4-yl)amino]piperidine-1-carbothioyl]azanide 6-(hydroxymethyl)-3,9-dimethoxybenzo[c]chromene-2,11-diol 2-[5-(1-azidopiperidin-4-yl)oxypyridin-3-yl]-1H-indole 3-[7-fluoro-6-methoxy-2-(4-methoxyphenyl)-1H-indol-3-yl]-N-[(2R,3S)-3-hydroxy-4-oxooctan-2-yl]propanamide (6S,9R)-2-amino-6-[4-methoxy-3-(naphthalen-1-ylmethoxy)phenyl]-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 5-methyl-1-[[2-(oxan-3-yl)-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl]sulfonyl]pyrrole-3-carbonitrile N-[1,3-dihydroxy-2-(2-methylpropanoylamino)propan-2-yl]-4-phenylbenzamide 2-chloro-N-methyl-5,6-dihydrobenzo[h]quinazolin-10-amine 2-(3,4-dimethoxyphenyl)-1-[3-(1H-imidazol-5-yl)propanoyl]piperidine-3-carboxylic acid;2,2,2-trifluoroacetic acid 2-[4-(cyclobutanecarboximidoyl)phenyl]-6,7,8a,9-tetrahydropyrido[1,2-a]pyrimidin-4-one 2-[3-[(1R)-3,6-dimethylcyclohepta-2,4,6-trien-1-yl]propoxy]-N'-hydroxypyrimidine-5-carboximidamide 3-azido-4,5-dimethylbenzo[g]indazole (2S,3S)-N-[(1R,2R,4S)-4-[(Z)-5-hydroxypent-2-enoxy]-2,3-dihydro-1H-inden-2-yl]-1-methylpyrrolidine-2-carboxamide;hydrochloride ethane;5-[3-(2H-pyrazolo[3,4-b]pyridin-3-yl)phenyl]pyrimidine (3-methoxy-1-methylpyrazol-4-yl)-(4-phenylpiperidin-1-yl)methanone 3-[(2,5-difluorophenyl)methyl]-1-(5-ethoxypyrimidine-4-carboximidoyl)piperidin-3-amine (4Z)-4-ethylidene-8,9-dimethoxybenzo[f][1]benzothiole N-[2,5-dimethyl-4-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]-7-[[5-fluoro-3-methoxy-4-(2-morpholin-4-ylethoxy)benzoyl]amino]-9H-carbazole-1-carboxamide 4-chloro-2-[4-(5-hydroxypyridine-3-carbonyl)piperazin-1-yl]benzonitrile 2-[[2-[4-(methylamino)anilino]acetyl]amino]-5-oxo-5-thiophen-3-ylpentanamide 5-(4-fluorophenyl)-1-propan-2-ylpyrazole 2-hydroxy-5-[[4-(3-phenylmethoxyanilino)pyrimidin-2-yl]amino]benzoic acid 2-[4-methyl-6-oxo-3-(phenylsulfanylmethyl)-1H-pyridazin-5-yl]acetic acid N-(2-chloropyridin-4-yl)-7-cyclopropylimidazo[1,5-a]pyridine-6-carboxamide 1-(1,2-dimethylindole-3-carbonyl)piperidine-4-carboxamide 3-[(1E,3Z)-4-fluoro-5-methylhexa-1,3,5-trienoxy]-N'-hydroxybenzenecarboximidamide (3S)-3-azido-N-(4,5,6,7-tetrahydro-1H-indazole-5-carbonyl)pentanamide N-[2,5-dimethyl-4-(trifluoromethyl)pyrazol-3-yl]-2-iodobenzenesulfonamide 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-hydroxypyrimidine-4-carboximidamide N-[4-fluoro-5-[6-(2,3,3-trimethylbutan-2-yloxy)pyridin-3-yl]oxy-1H-benzimidazol-2-yl]-3-methylpyrazole-1-carboxamide 7-[3,4-difluoro-2-(trideuteriomethoxy)phenyl]thieno[3,2-c]pyridine N-[2,6-difluoro-3-(hydroxymethyl)phenyl]-1-propan-2-ylpyrazole-4-sulfonamide 2-(6-bromocyclohexa-1,3-dien-5-yn-1-yl)oxy-N-methoxypyridine-4-carboxamide 2-[(7R)-1-methyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-7-yl]benzamide 7-(4-hydroxypiperidine-1-carbonyl)-2-phenylquinoline-3,6-dicarbonitrile 4-[5-(3,5-dimethoxyphenyl)thiophen-2-yl]-2-methyl-1H-pyrazole-3-thione 4-[(2S)-1-benzoyl-5,7-dimethoxy-6-propan-2-yloxycarbonyl-3,4-dihydro-2H-quinolin-2-yl]-2-phenylpyrazole-3-carboxylic acid (2S)-1,4-dibenzylsulfanylbutane-1,2-diol 6-azido-1-(2,4-dimethoxyphenyl)hexan-3-one (5R,7S)-N-[[(3S,4S)-1-methyl-2-oxopiperidin-4-yl]methyl]-5,6,7,8-tetrahydroquinoline-5-carboxamide 3-methyl-4-[2-(4,5,7-trifluorobenzotriazol-1-yl)ethoxy]aniline N-[(4-nitrophenyl)methyl]-2,4-dioxo-3H-pyrimido[1,2-a]benzimidazole-5-carboxamide (5S)-2-[4-(2,3-dichlorophenyl)piperazin-1-yl]-N-(2-methoxyphenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 2-[azido-(3-fluorophenoxy)methyl]furan 3-(5,8-dichloroimidazo[1,2-a]pyridine-3-carbonyl)piperidine-4-carboxylic acid 3-(2,6-dichloropyridin-4-yl)-1-[2-(dimethylamino)phenyl]propan-1-one (3,5-dibromophenyl)methylsulfanylformohydrazide N-ethyl-1,4-bis(5-methylthiophen-2-yl)butane-1,3-diimine N-(2-methylpropyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide 4-N,6-N-bis[(2E)-2-ethenylpenta-2,4-dienyl]-4-N-methylpyrimidine-2,4,6-triamine N-(2-cyclopropyloxyphenyl)-1,4-dimethyl-5-(6-pyridin-3-ylimidazo[1,2-b]pyridazin-3-yl)pyrrole-3-carboxamide;ethane 1-(2,4-dichlorophenyl)sulfonyl-3,6-dihydro-2H-pyridine [1-aminooxy-3,4,5,6-tetramethyl-2-(trifluoromethyl)inden-1-yl]phosphane [2-(5,6-dimethoxy-3H-indol-2-yl)quinolin-4-yl]hydrazine 2-(1H-indol-4-yl)-N-[3-[6-[2-(methoxyamino)ethylamino]quinazolin-2-yl]phenyl]acetamide 5-azido-N-methylnaphthalene-1-sulfonamide (2S,5R)-N-[4-[5-chloro-6-[5-[difluoro(iodo)methyl]pyridin-3-yl]pyrazin-2-yl]phenyl]-1-cyano-N'-cyclopropylsulfonyl-2,5-dimethylpiperazine-1-carboximidamide 1-[5-tert-butyl-2-(4,6-dimethoxypyrimidin-2-yl)pyrazol-3-yl]-3-naphthalen-2-ylurea 4-(3,5-dinitrophenyl)sulfanylphenol N-(3,5-dibromo-4-hydroxyphenyl)hexanamide 5-[4,6-bis(trichloromethyl)-1H-benzimidazol-2-yl]-2-fluorophenol 2-amino-4-[3,6-bis(ethenyl)carbazol-9-yl]phenol 4-[3-fluoro-5-(2,2,6,6-tetramethylpiperidin-4-yl)oxyphenyl]-N'-(6-oxo-1H-pyridin-3-yl)butanimidamide 5-fluoro-1,4a-dimethyl-7-(3-propanoylphenyl)-10aH-acridin-9-one N-(1-benzothiophen-2-ylsulfonyl)cyclopentanimine (2S,5R)-N-[1-(3-chlorophenyl)ethyl]-4-(2-fluorophenoxy)-1,7-dioxo-2,6-dipropyl-2,9-diazaspiro[4.5]decane-9-carboxamide;formic acid ethane;4-[2-(3-formylphenyl)-7-oxo-6H-[1,2,4]triazolo[1,5-a]pyrimidin-5-ylidene]cyclohexa-2,5-diene-1-carboxylic acid 6-azido-8,9-difluorophenanthridine (2S)-1-[[2-fluoro-6-[5-(trifluoromethyl)pyridin-3-yl]oxyphenyl]methylamino]propan-2-ol N-[[4-chloro-2-(trifluoromethyl)phenyl]methoxy]-1-[(3S,5R)-5-ethylpyrrolidin-3-yl]-3,3-dimethylbutan-1-imine 2-(6,8-dimethoxy-1,5-naphthyridin-4-yl)-1H-indole-3-carboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[(1S,5R)-6,7-dihydro-5H-cyclopenta[a]pyridin-3-yl]acetamide (Z)-N'-[2-[6-methyl-5,7-bis[4-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidin-2-yl]propanoylamino]but-2-enediamide 2-(dimethylamino)-4-oxo-2,3-dihydrochromene-8-carboxamide 5-[(3Z,5E)-5-chlorohepta-1,3,5-trien-2-yl]-N-phenylpyridine-3-carboxamide 4-[5-methoxy-6,7-di(propan-2-yl)phthalazin-1-yl]morpholine N-[5-(2-methoxyphenyl)-3,4-dihydropyridin-6-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine 2-(7,8-dimethoxy-5H-1,6-naphthyridin-3-yl)benzamide 3-[1-(cyclopropylmethylamino)-2,6-naphthyridin-7-yl]-4H-1,2,4-oxadiazol-5-one 7-azido-4,5-dimethoxy-3H-quinazoline 7-(4-chlorophenyl)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-6-imino-4,5-bis(sulfanylidene)-1H-pyrrolo[3,4-d]pyrimidine-2-carboxamide 4-[3,5-bis(hydroxymethyl)phenyl]sulfonylphenol 1-(4-bromophenyl)sulfanyl-2,3-dimethylcyclopropane-1-carboxylic acid 3-(5-tert-butyl-1,2-oxazol-3-yl)benzoate 4-[5-methyl-2-(2-phenylethynyl)benzimidazol-1-yl]sulfanylbenzenesulfinate ethane;8-methylanthracene 6-chloro-4,5-dideuterio-2-(trifluoromethyl)benzimidazole 3-chloro-5-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]sulfanylbenzonitrile 3-fluoro-4-methylsulfonylbenzenesulfonic acid 3-[2,6-dichloro-4-(2-ethylimidazo[1,2-b]pyridazin-5-yl)phenyl]-2H-1,3,4-oxadiazole 1-methyl-2-propan-2-yl-5-[4,4,4-trifluoro-3-(4-pentanoylphenyl)but-1-enyl]pyridin-4-one 4-[azido(cyclohexyl)methyl]-N,N-bis(2-chloroethyl)aniline 4-[6-(4-fluorophenyl)thieno[2,3-b]pyrrol-5-yl]cyclohexa-1,3-dien-5-yne-1-carboxylic acid N'-hydroxy-5,6-dimethyl-3-[methyl(propan-2-yl)amino]pyridazine-4-carboximidamide N-[4,6-bis(propan-2-ylsulfanyl)pyrimidin-5-yl]benzenesulfonamide N-[(E)-[(4Z,6Z,8Z)-9-methoxyundeca-1,4,6,8-tetraen-5-ylidene]amino]-N,2,6-triphenylaniline N-[(2R,3S)-1-methyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]-1H-pyrrolo[3,2-b]pyridine-3-carboxamide 1-[3,5-difluoro-4-(trifluoromethyl)phenyl]ethanone;ethane;propane N-(5-bromopyridin-2-yl)-1-cyclopropylcyclopropane-1-carboxamide N-[2-(4-methylpiperazin-1-yl)phenyl]thieno[3,2-d]pyrimidine-7-carboxamide [4-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]oxycyclohexyl]carbamic acid 1-[3,5-dimethyl-4-(1H-pyrazol-5-ylsulfanyl)phenyl]-N,2-dimethylpentan-2-amine N-(5,6-dimethylpyridin-2-yl)oxybenzenesulfonamide [(2S)-5-chlorospiro[1H-indole-3,4'-piperidine]-2-yl]-cyclopropylmethanone (2S)-3-[5-[2-amino-4-[2-(dimethylamino)ethoxy]phenyl]-1H-imidazol-2-yl]pyrrolidine-1,2-dicarboxylic acid 2-(2,6-dichlorophenyl)-4-methyl-5-[3-(1H-pyrazol-5-yl)propanoyl]-1H-pyrimidin-6-one 4-[2-(1,3-benzothiazol-2-yl)ethenyl]benzenesulfonamide N-[2-(dimethylamino)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide;formic acid N-(4,5-dichloropyridin-2-yl)-2-(4-methoxyphenyl)-2-oxoacetamide 4-(1,3-benzoxazol-2-ylamino)-N-cyclohexyloxy-6-methoxypyridine-3-carboxamide N-[3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl)phenyl]acetamide 4-[7-chloro-1'-(4-fluorophenyl)sulfonyl-5-methylspiro[3H-1,4-benzodiazepine-2,4'-piperidine]-6-yl]-N,N-dimethylbenzamide (3,4-difluorophenyl)methyl-[5-(2H-pyrimidin-1-yloxy)pyrimidin-2-yl]carbamic acid 4-[3-(diethylamino)propylsulfanylmethyl]benzenediazonium 1-[(2S)-3,3-dimethylbutan-2-yl]-4-nitrobenzene (2Z,4E)-6-ethenylimino-N-[1-(3-methoxyphenyl)sulfanylethenyl]-5-(oxolan-2-ylmethylideneamino)pyrimidin-2-amine 2-[1-(6,7-dimethoxyquinazolin-4-yl)piperidin-3-yl]-N-ethyl-N-[(1E)-1-(methylideneamino)buta-1,3-dienyl]acetamide 2-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6H-pyrrolo[3,4-b]pyrrol-2-yl]benzonitrile 4-[3,5-dimethyl-2,6-dioxo-4-[3-(trifluoromethoxy)phenyl]pyrimidin-1-yl]-N-hexylbutanamide 2-methyl-N,2-diphenylpropanamide 4-[azido(3,5-dimethylanilino)amino]benzoic acid N-(2,6-dimethylphenyl)spiro[4.5]decane-8-carboxamide [1-(1,3-benzothiazol-2-yl)pyrrolidin-2-yl]-(4-pyridin-4-ylpiperazin-1-yl)methanone 5-bromo-2-(3,4-dihydropyridin-6-yl)-N-[1-(methoxymethyl)cyclopentyl]-1H-indole-7-carboxamide N-methylformamide;(E)-2-[4-[(Z)-3-oxobut-1-enyl]thiophen-3-yl]ethenesulfonic acid (NE)-N-[1'-[3-(4,6-dimethylpyrimidin-2-yl)oxyphenyl]spiro[chromene-2,4'-piperidine]-4-ylidene]hydroxylamine 4-(5-azidopentyl)aniline 1-(4-benzylpiperidine-1-carbonyl)cyclopropane-1-carboxylic acid 1-(azidomethyl)-3-chloro-5,6-difluoroindole 7-[[4-(diethylamino)cyclohexa-1,5-dien-1-yl]amino]-N'-hydroxypyrene-2-carboximidamide 7-[3-(trifluoromethyl)anilino]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid 3-(benzylamino)naphthalene-2,7-dithiol ethane;(4E,6Z)-5-methoxy-3,8-dimethylnona-1,4,6-triene;6-oxospiro[3H-chromene-2,4'-oxane]-4-carboxylate 5-butyl-2-methyl-3-pyridin-4-ylimidazo[1,2-a]pyridine N-methyl-3,7-diphenylbicyclo[4.1.0]hepta-2,5-dien-8-amine (3R)-1-[(2S)-4-amino-1,2,5-trideuteriopentan-3-yl]-3-[6-ethoxy-5-fluoro-2-(propoxymethyl)benzimidazol-1-yl]piperidine-2,6-dione 1-benzyl-3,4-dimethylimidazolidin-2-one N-[(E)-[5-hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl]methylideneamino]-4-nitrobenzenesulfonamide N'-[3,4-bis(phenylmethoxy)cyclohexa-1,3-dien-5-yn-1-yl]ethanimidamide 1-[2-(5-ethyl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-2-yl)-3-methoxyphenyl]-3-[4-fluoro-3-(trifluoromethyl)phenyl]urea (2-cyclopropyloxyphenyl)methanesulfonic acid 1-(2-azidooxyethyl)sulfonyl-4-methylbenzene 4-[2,3-dihydroxypropyl(2H-tetrazol-5-yl)amino]butan-1-ol 1-[3,5-dichloro-4-(trifluoromethyl)phenyl]-3,3-dimethoxypropan-2-one 2-(1-azidoethyl)-5-nitroindazole N-(2,5-dimethylphenyl)-N'-[(Z)-(4-hydroxy-3-iodophenyl)methylideneamino]oxamide 5-azido-1,2-bis(trifluoromethyl)naphthalene 2-(azidomethyl)-6,6-dimethyl-5H-1,4-benzothiazine 1-(4,5-difluoro-3-methylthiophene-2-carbonyl)-N-pyridin-2-ylpiperidine-4-carboxamide 1-(5-tert-butyl-2,3-dihydro-1H-indene-4-carbonyl)pyrrolidine-2-carboxylic acid 2-methyl-N-(3-pyrrolidin-1-ylpropyl)furan-3-carboxamide 1-(3,4-dihydroisoquinoline-1-carbonyl)piperidin-2-one 1-[4-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]cyclohexa-1,3-dien-1-yl]propan-2-one 3-amino-2,4,5-trifluoro-6-(tribromomethyl)benzenesulfonic acid 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethoxy)benzonitrile 5-(4-methylphenyl)sulfonyl-3-pyridin-2-yl-1H-indole 1-[(E)-but-2-enoxy]-4-[2,3-difluoro-4-(trifluoromethyl)phenyl]-2-prop-2-ynoxybenzene 2-[4,6-bis(phenylmethoxy)-1,3,5-triazin-2-yl]butanoate 2-[4-(trifluoromethyl)phenyl]-3,5,6,7-tetrahydropyrrolo[3,4-d]pyrimidin-4-one (6aR,10aS)-5-chloro-10a-methyl-1,4-dihydroanthracene;2-chloroethanol N-[[2,6-dichloro-4-(trifluoromethyl)phenyl]methylideneamino]-3-phenylpropanamide 4-(2,3-dihydrofuran-5-yl)-1-methoxybutan-1-amine;1-[6-(3-methylpyridine-2-carbonyl)-6-azaspiro[3.4]octan-8-yl]ethanone N-[[1-(6-fluoroquinolin-2-yl)piperidin-3-yl]methyl]ethanesulfonamide 5-(azidomethyl)-1-N,2-N-bis[3-chloro-4-[2-(diethylamino)-6-oxocyclohexen-1-yl]phenyl]pyrrolidine-1,2-dicarboxamide 2-N-(3,4-dimethoxyphenyl)benzene-1,2-diamine;1-[3-[4-fluoro-3-(trifluoromethyl)phenyl]propanoylamino]cyclobutane-1-carboxylic acid 2-[(6R,9R)-6-pyridin-3-yl-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-ylidene]acetaldehyde ethane;4-(5-methylthiophen-2-yl)cyclohepta-3,6-diene-1,2-dione (3-fluoropyridin-4-yl)-[3-hydroxy-3-(triazol-1-ylmethyl)piperidin-1-yl]methanone N-[3-(2,3-dihydro-1H-pyrrol-5-yl)-3-methoxypropyl]aniline (5-amino-1H-pyrazol-4-yl)-[2-fluoro-6-methoxy-3-methyl-6-(trifluoromethyl)phenyl]methanone 4-[[2-(butanoylamino)phenyl]methylamino]quinazoline-8-carboxamide 4-(4-amino-3-methanimidoylphenyl)sulfanyl-2-propan-2-yloxybenzonitrile 1-(5-chloro-6-oxo-3,4-dihydro-2H-pyridin-1-yl)-N-[1-(2,6-difluorophenyl)propan-2-yl]isoquinoline-7-carboxamide 2-[4-chloro-3,5-dimethyl-1-(oxan-4-yl)pyrazol-4-yl]-N-(4-cyanophenyl)acetamide 1-(2-amino-3H-benzimidazol-5-yl)-4,5-dihydropyrazolo[3,4-c]pyridin-6-one [3-(2,4-difluorophenyl)pyrrolidine-1-carbonyl]-[1-(pyridin-3-ylmethyl)piperidin-4-ylidene]azanium 6-methyl-3-[4-(3,4,5-trifluorophenyl)cyclohexa-1,3-dien-1-yl]-2H-pyrazolo[3,4-d]pyrimidine 5-(2,2-dimethylpropyl)-4-fluoro-2-methoxyaniline 1-[(E)-3,4-diphenylbut-2-enyl]imidazole N-[4-(2,4-dimethylphenoxy)butyl]formamide 2-(1-azidoethyl)-5-methoxyquinoxaline (E)-1-[4-[7-chloro-8-methoxy-3-(2-propan-2-ylphenyl)pyrazolo[3,4-c]quinolin-1-yl]piperidin-1-yl]but-2-en-1-one 2-[3-bromo-4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonylamino)phenyl]acetic acid [1-(2-chloro-5-fluorophenyl)sulfonylpiperidin-3-yl]methanol 4-[2,6-bis(2,4,5-trimethylphenyl)cyclohexa-1,3-dien-1-yl]-3H-pyrrole 2-[2,4-dichloro-6-(5-ethyl-1,3-dimethylpyrazole-4-carbonyl)phenyl]sulfanyl-4-methoxybenzonitrile 2-[(4-bromophenyl)sulfonylamino]-5,6,7,8-tetrahydroquinoline-3-carboxamide 1-(2,3-difluorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]butan-1-ol N-(4-chlorobutyl)-6-nitro-N-propyl-1,3-benzothiazol-2-amine 4-chloro-N-[1-[(2E)-2,5,7-trimethylhepta-2,6-dienoxy]propan-2-ylideneamino]aniline 1-[1,3-dioxo-2-(4-phenylphenyl)isoindol-5-yl]propane-1-sulfonate N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-4-[5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]benzamide 1-[[5-(4-fluorophenyl)-2,3-dihydro-1,3,4-oxadiazol-2-yl]methoxymethylamino]-N-hydroxycyclopropane-1-carboxamide (6S,9aR)-2-[2-(3-chlorophenyl)ethenyl]-N'-hydroxy-6-methoxy-1,4-dioxospiro[5.5]undecane-8-carboximidamide 1-cyclopropyl-3-[4,4-difluoro-2-(hydroxymethyl)pyrrolidin-1-yl]-6,7,8,9-tetrahydrobenzo[g]isoquinoline-5-carbonitrile 4-methyl-6-(5,6,7,8-tetrahydronaphthalen-2-yloxy)pyrimidine (3,5-dimethylpiperazin-1-yl)-[1-(1,2-oxazol-4-ylmethyl)pyrrol-2-yl]methanone 1-(2-methyl-3-propoxyphenyl)ethanone 2-bromo-3-(3,4-difluorophenyl)-3H-1,2-oxazol-5-amine 1-[(2S,4R)-4-fluoro-1-(5,6,7,8-tetrahydro-[1]benzothiolo[3,2-d]pyrimidin-4-ylamino)pyrrolidin-2-yl]-N-methylcyclopropane-1-carboxamide 5-ethyl-7-[[3,4,6-tris(trifluoromethoxy)phenyl]methoxymethyl]-2,3-dihydro-1-benzofuran 1,2-difluoro-6-[2-(3-fluorophenyl)ethynyl]naphthalene 4-[(6E,8Z)-9-aminonona-1,5,7-trienyl]-2-ethoxyphenol 4-[4-[(1S,2R)-2-phenylcyclopropanecarbonyl]piperazine-1-carbonyl]piperidine-1-carboxylic acid 4-(4,5,6,7-tetrachloronaphthalen-2-yl)sulfonylpyridine N-[2,6-difluoro-3-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)phenyl]acetamide 1-cyclobutylsulfonyl-4-[(2R)-6,15-dibromo-13-methyl-4-azatricyclo[9.5.0.03,8]hexadeca-1(11),3(8),4,6,12,14-hexaen-2-yl]piperazine;ethane N-azido-5-[(dimethylamino)methyl]-2-fluorobenzamide 1-(azidomethyl)-5-bromonaphthalene N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-8,9-dimethoxy-5-oxo-10H-benzo[b][1,6]naphthyridine-2-carboxamide (2-aminophenyl)-[4-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazine-1-carbonyl]piperidin-1-yl]methanone 2-[4,5-bis(ethenyl)-1H-pyrrol-3-yl]-N-benzylidenepropanediamide 5-(4-fluoro-2,6-dimethylphenyl)-7-[3-fluoro-5-[(1S,2R)-2-hydroxycyclohexyl]pyridin-2-yl]oxy-6-methylpyrrolo[3,4-b]pyrazine-3-carbonitrile 2-[4-[(3R,4S)-1-benzylsulfonyl-4-[[2-(cyclopropen-1-yl)pyrimidine-5-carbonyl]amino]pyrrolidin-3-yl]oxyphenyl]acetic acid (4-nitrophenyl)-[(E,3S)-1-phenylpent-1-en-3-yl]azanium (2S,3R)-3-ethyl-N-[1-(4-fluorophenyl)pyrrolidin-3-yl]morpholine-2-carboxamide 3-(2,4,5-trimethoxyphenyl)cyclopropane-1,1,2,2-tetracarbonitrile 5-(2,6-dimethoxyphenyl)furan-2-carboxamide N-[5-(4-fluorophenyl)sulfonyl-2,3-dihydro-1H-inden-1-yl]-1-methoxyethanethioamide 1-[(3S)-2,6-dioxopiperidin-3-yl]-2-ethynyl-5,8-dimethoxybenzo[f]benzimidazole-4,9-dione 3-chloro-2-[5-(4,5-dihydro-1H-imidazol-2-yl)thiophen-2-yl]-5-iodobenzonitrile N-[4,5-dimethoxy-2-nitro-3-(trifluoromethyl)phenyl]acetamide 3-butyliminoindole-6,8-disulfonic acid 4-[[6-amino-5-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)pyridin-2-yl]amino]cyclohexan-1-olate ethane;N-methyl-4-[2-(morpholin-4-ylmethyl)imidazo[1,2-a]pyrimidin-6-yl]aniline (1S,2R)-6-amino-3-hydroxy-1-phenyl-7,8-dihydro-2H-anthracene-2-carboxamide N-[2-(4-oxo-3H-quinazolin-2-yl)ethyl]-5,6,7,8-tetrahydroisoquinoline-1-carboxamide [2-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-1,1,1,3,3,3-hexafluoropropan-2-yl]phosphane 3-[5-(3,4-dimethoxyphenyl)-1H-pyrazole-4-carbonyl]benzoic acid 5-bromo-1H-pyrrolo[2,3-b]pyridine-3-carboxylic acid 2-benzylsulfanyl-4,6,8,10,11-pentazatricyclo[7.3.0.03,7]dodeca-1(9),2,4,7,11-pentaen-5-amine 2-[(5S)-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl]-4-thiophen-3-ylbenzamide [4-(2,3-dihydropyrrolo[2,3-b]pyridine-1-carbonyl)anilino]thiourea 1,2-bis(3-nitrophenyl)-3H-imidazo[1,5-a]pyrazine (4S)-2-[3-(2,6-dimethylphenyl)-1,2,4-oxadiazol-5-yl]-4-methoxypyrrolidine-1-carboximidamide 3-[2-(4-chlorophenyl)ethenyl]benzamide 3-[6-[4-(cyclohexa-1,5-dien-1-ylmethoxy)phenyl]sulfanylpyridin-2-yl]hexanamide 1,3-bis[4-(hydroxyamino)-6-phenylpyridin-2-yl]urea N-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethyl)-5-(trifluoromethoxy)pyridine-3-carboxamide 1-benzyl-5,6-dichloro-3-propanoylindole-2-carboxylic acid 3-[4-(2,6-dichlorophenyl)-5-methyl-1H-imidazole-2-carbonyl]hexanenitrile 1-ethyl-3,4-diphenylpyrrole 2,4-diphenyl-1H-1,3,5-triazine (2S)-4,5-difluoro-N-[(4-methoxyphenyl)methyl]-1-methyl-3-oxospiro[indole-2,4'-piperidine]-2'-carboxamide 1-(4-butylphenyl)sulfonyl-2-fluoropiperidine 2-methyl-1-[3-(trifluoromethoxy)phenyl]propan-1-one (3S)-3,4,4a,6-tetramethyl-2,5,10b-trioxo-7-propanoyloxy-9H-indeno[1,2-b]pyridine-3-carboxylic acid N-[1-(4,5-dimethylthiophen-2-yl)ethenyl]-4-methoxyaniline (3-azido-1,2-oxazol-4-yl)-phenylmethanone N'-methyl-2,3-bis(propan-2-yloxy)benzenecarboximidamide N-azido-3-(3-oxomorpholin-4-yl)benzamide 1-(4-amino-3,5-dichlorophenyl)-2-azidoethanone 3-[8-fluoro-5-(4-fluorophenyl)-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl]-N-(3-hydroxypropyl)-2-oxoimidazolidine-1-carboxamide 2-(4-butoxyphenyl)sulfinyl-3,6-diethylphenol 1,4-diamino-N'-[2,3-bis(trifluoromethyl)phenyl]-6-methanimidoylpyrrolo[3,2-c]pyridine-7-carboximidamide 4-[(3-chlorophenyl)methyl]-2H-pyrrole 1-[2-bromo-4,5-bis(ethenyl)imidazol-1-yl]-3-bromo-6-fluorohexan-1-ol 4-[azido(methyl)amino]oxypyridine-2-carbonitrile 4-chloro-2-[(1E,3Z)-hexa-1,3,5-trienyl]aniline (2S,5R)-5-phenyl-1-(2-phenylethylamino)heptane-3,4-diol 4-azidooxy-6-chloro-5,8-dihydropyrimido[4,5-d]pyrimidine 2-[7-(diethylamino)-5,10-dimethylphenazin-5-ium-2-yl]oxyethanol N-[(1S)-2,3-dihydro-1H-inden-1-yl]-1-ethyl-6-hydroxy-5-oxo-4H-pyrazole-3-carboxamide 1-(4,6-dichloropyrimidin-5-yl)cyclopropane-1-carboxylate 4-[(1S)-1-[[2,5-dioxo-3-[(E)-2-phenylethenyl]cyclopentan-1-ylidene]amino]propyl]benzamide 1-(4-bromophenyl)-2-[4-(4,5-dihydroimidazol-1-ylmethyl)piperidin-1-yl]ethanone;formaldehyde 4-[(1-cyclobutylpyrazol-3-yl)methyl]-5-(1,2,3,6-tetrahydropyridin-4-yl)thiadiazole 7,8-dimethoxy-5-oxo-1H-pyrido[2,3-b]indole-4-carboxylic acid 3-[2-(diethylamino)acetyl]-7,8-dimethoxychromen-4-one;ethane 5-(4-butyl-3,5-difluorophenyl)-2,3-difluorophenol 1-methyl-6,7,8-trioxoquinoline-2-carboxamide 5-[[(2R,3S)-2-(1H-pyrazol-4-yl)oxan-3-yl]methoxy]pyrazine (4-butylsulfanylphenyl)-[5-(6-methoxypyridin-3-yl)thiophen-2-yl]-pyridin-3-ylmethanol (3S)-N'-hydroxy-2,2-dimethyl-4-[1-[4-(4-pyrrolidin-1-ylpiperidin-1-yl)phenyl]pyrazolo[3,4-d]pyrimidin-3-yl]oxybutanimidamide (3,4-dichlorophenyl)methylcarbamic acid 1-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]-5,6-difluoroindole N-[(5-bromopyridin-3-yl)methyl]-2,6-difluoro-4-(pyridin-2-ylmethoxy)benzamide 1-[2-(3,5-dimethylpiperidin-1-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-(3-ethoxypropanoylamino)cyclobutane-1-carboxylic acid 3-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(4-hydroxyphenyl)iminomethyl]benzenesulfonic acid N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)spiro[1,3-dihydroindene-2,2'-cyclopropane]-1'-carboxamide 1-[(4R)-4-(cyclohexylmethoxy)-5-fluoro-2-methylpentan-2-yl]-3-(3,5-dichlorophenyl)urea 5-[(2R,4S)-1-acetyl-2-cyclopropylpiperidin-4-yl]oxy-N-cyclopropyl-8-methyl-2-oxochromene-3-carboxamide 2,4-diphenylbutanehydrazide 4-[7-chloro-3-(2,6-difluorophenyl)quinolin-2-yl]piperazine-1-carboxylic acid 4-chloro-N-[(Z)-1,3-diaminobut-2-enylidene]-5-(3-methoxyazetidin-1-yl)sulfonylthiophene-2-carboxamide 4-(3,5-dimethylphenyl)-2-[(4Z)-2-methylidenehepta-4,6-dienoxy]pyridine 2-methylsulfonyl-1-[4-(thiophen-2-ylmethyl)piperidin-1-yl]propan-1-one 1-[(3-hydroxyphenyl)methylamino]-3-(thiophen-2-ylmethylidene)thiourea N-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]-6,8-difluoro-7-morpholin-4-ylquinoxaline-5-carboxamide 2-azidosulfanyl-6-methoxynaphthalene 2-(6,8,9,10,11-pentamethyl-3,7,12-triazaspiro[5.8]dodeca-1,4,6,11-tetraen-3-yl)quinoline 1-methyl-4-[2-(3-nitrophenyl)sulfonylpropan-2-yl]benzene (2R)-N,3-diethyl-1-oxo-2-pyridin-4-yl-2H-imidazo[1,5-a]indole-8-carboxamide 5-(2,2-diethoxyethylamino)naphthalene-1,4-disulfonic acid 4-[5-amino-6-(1H-pyrazole-4-carboximidoyl)pyrazin-2-yl]-3-fluorophenol 1-(4-butoxyphenoxy)sulfonyl-2,3-dihydroindole-2-carboxylic acid 3-[(2S)-1-benzoyl-5-(methanesulfonamido)-4-oxo-2,3-dihydroquinolin-2-yl]propanamide 2-[1-(6-chloropyrimidin-4-yl)piperidin-3-yl]propan-2-ol N-[4-fluoro-3-(7-oxo-2-oxa-5,8-diazabicyclo[11.4.0]heptadeca-1(17),13,15-trien-16-yl)phenyl]acetamide 3-[2-(trifluoromethyl)quinoline-6-carbonyl]benzamide [(3R)-1,2-dihydroxy-5-phenylpentan-3-yl]carbamic acid (2R)-N-[6,7-dichloro-1-oxo-2-phenyl-8-(trifluoromethylsulfonyloxy)isoquinolin-3-yl]pyrrolidine-2-carboxamide (1-azidocyclopentyl)methoxymethylbenzene N-[(E)-1,5-diphenylpent-4-enyl]-3-methoxy-2H-pyran-2-amine 1,2-dimethoxy-4-[(2E)-5-(trifluoromethylsulfanylamino)penta-2,4-dien-3-yl]benzene 4-[5-(3,3a,4,5,6,7,7a-octahydro-2H-furo[2,3-c]pyridine-2-carbonyl)thiophen-2-yl]-2-amino-6-(1H-pyrazol-5-yl)pyridine-3-carbonitrile N-azido-2-tert-butyl-4-fluoropyridine-3-carboxamide 5-benzyl-N-ethenyl-2,3-dimethylaniline (3R)-N'-hydroxy-2,2-dimethyl-4-[(Z)-3-(pyridine-4-carbonylamino)prop-1-enyl]-3H-1-benzofuran-7-carboximidamide 3-[(2-chloroacetyl)-phenacylamino]propanoic acid N-[4-(2,3-dihydro-1H-pyrrol-5-yl)phenyl]-5,7-bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide (4-amino-2,5-dihydroxyphenyl)-[3,5-bis(trifluoromethyl)phenyl]methanone 4-(1,3-benzothiazol-2-yldiazenyl)phenol 4-[2-(2-hydroxyethoxy)phenyl]benzoic acid 2-[4-(2-aminopyridin-3-yl)thiophen-2-yl]-N'-hydrazinylidene-6-phenylthieno[3,2-d]pyrimidine-5-carboximidamide N-methyl-6-[(3-methylfuran-2-carbonyl)amino]pyridine-3-carboxamide N-[[4-[2-[(3R)-4-hydroxy-1-methylpyrrolidin-3-yl]ethynyl]phenyl]methyl]naphthalene-2-carboxamide 4-[[5-fluoro-2-(triazol-1-ylmethoxy)benzoyl]amino]cyclohexane-1-carboxylic acid [[2-amino-4,5-bis(trifluoromethyl)phenyl]carbamoylamino]carbamic acid 4-[(2R)-2,3-dihydroxypropyl]-5-(4-fluoro-1H-indole-6-carbonyl)piperazin-2-one 4-[3-[[4-(cyclopenten-1-yl)phenoxy]methyl]-5-fluorophenyl]pyridine 1-(4,5-dimethoxy-2-nitrophenyl)piperazine;3H-furo[3,2-d]pyrimidin-4-one 1-[4-(3,5-dichlorophenyl)piperazin-1-yl]-2-[4-[(Z)-prop-1-enoxy]pyridin-2-yl]sulfanylethanone 1-(4-methylphenyl)-5-[5-(trifluoromethoxy)pyridin-2-yl]pyrazole-3-carboxylic acid N'-hydroxy-5-[(4,4,4-trifluorobutylamino)methyl]pyridine-2-carboximidamide (2S)-2-amino-3-[3-[(4-fluorophenyl)methyl]imidazol-4-yl]propanoic acid 4-[3,5-bis(trifluoromethyl)phenyl]cyclohexan-1-amine;N-(3,4-dihydro-2H-chromen-6-ylmethyl)propanamide 1-(azidomethyl)anthracene 2-(azidomethyl)-6-[4-[(3-fluorophenyl)methoxy]phenyl]pyridazin-3-one 6-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5H-benzo[h]quinoline (4-iodopiperidin-1-yl)-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]methanone 2-[3-(4-methoxyphenyl)cyclobutyl]ethanol [4-(4-acetylphenyl)phenyl]-(5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)methanone 1-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-N-methyl-1-(2-methylphenyl)ethanimine;(Z)-pent-2-ene 3-[N'-(diethylamino)carbamimidoyl]-1H-indole-2,4-dicarboxylic acid [7-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)carbazol-9-yl]boronic acid 6-(5-chloropentyl)naphthalen-2-ol 2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)-N-[(E)-ethylideneamino]aniline [1-(3,5-dichlorophenyl)sulfanyl-2-hydroxyindol-4-yl]-(2-fluoropyridin-3-yl)methanone N-[(2,4-dimethoxyphenyl)methyl]-5-(furan-2-yl)pyrimidin-2-amine 6-methyl-4-oxo-N-(1,3-thiazol-2-yl)-1H-pyridine-3-carboxamide 1-[4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl]prop-2-en-1-one (5-chloroquinoline-8-carbonyl)-phenylazanium (3R)-4-(4-methylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine N-[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]benzamide 2-(3,4-dichlorophenyl)-N'-hydroxy-6-(2-methoxyethylsulfanyl)pyrimidine-4-carboximidamide 4-(1-hydroxynaphthalen-2-yl)-6,8,9-triazatricyclo[5.3.0.02,4]deca-1(10),6,8-trien-7-one 2,4-dimethyl-6-[1-(6-phenylpyridazine-3-carbonyl)piperidin-2-yl]pyridine-3-carbonitrile 2-[3-(4-bromophenyl)-1,2,4-oxadiazol-5-yl]benzenesulfonamide 6,7-dimethoxy-N-[(E)-2-quinolin-5-ylethylideneamino]quinazolin-4-amine N-(2,5-dimethylphenyl)-2-[[6-oxo-4-(propan-2-ylsulfanylmethyl)-1H-pyrimidin-2-yl]sulfanyl]acetamide 2-[(3aR,6aS)-5-[(5-methoxypyridin-2-yl)methyl]-3a-(5-methyl-1H-1,2,4-triazol-3-yl)-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-2-yl]-N,N-dimethylacetamide;formic acid 6-[4-(3,5-dichlorophenyl)sulfanylpiperazine-1-carbonyl]pyridine-2-carboxamide (E)-N-[2,6-dimethoxy-4-(1H-pyrazole-5-carbonylamino)phenyl]sulfonylprop-2-enamide 5-bromo-2-(dipropylamino)pyrimidine-4,6-dicarbonitrile 2-(1,3-benzodioxol-5-yl)-1-[4-(4-chlorobenzoyl)piperazin-1-yl]ethanone 6-[4,5-bis(ethenyl)-1H-pyrrole-2-carbonyl]cyclohex-3-ene-1-carboxylic acid 5-[3-methylbutyl(propyl)amino]naphthalene-2-sulfonic acid 3-[(3R)-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]pyrrolidin-3-yl]-N-(2,5-dimethoxyphenyl)sulfanylpyridine-4-carboxamide (2S,3R)-4-[4-hydroxy-6-[[4-(5H-tetrazol-1-ylmethyl)phenyl]methoxymethyl]oxan-2-yl]-3-methylsulfonyl-1-[4-(trifluoromethoxy)phenyl]butan-2-ol 2-(2,5-dichloro-N-ethenylsulfonylanilino)acetic acid N-[4-(3,5-dimethoxyanilino)quinazolin-6-yl]-2-pyrrolidin-1-ylacetamide 4-[3-[1,3-dioxo-2-(trifluoromethyl)inden-5-yl]sulfonyl-6-phenyl-2H-indazol-5-yl]benzonitrile 2-[(3S,4R)-3-amino-4-fluoropiperidin-1-yl]-N-[1-(dimethylcarbamoyl)-2,5-dimethylpyrrol-3-yl]-7-ethoxyquinazoline-6-carboxamide 2-[4-[(Z)-[2-(3-chlorophenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]phenoxy]acetamide [4-(1H-indol-3-yl)piperidin-1-yl]sulfonylhydrazine 2,4-dihydroxy-3-methoxy-N-(4-phenylbutyl)benzamide 3-(2,4-difluorophenyl)sulfinyl-5H-benzo[c][1]benzazepine 7-[1,5-dimethyl-3-(trifluoromethyl)pyrazole-4-carbonyl]-2-pyridin-4-yl-2,7-diazaspiro[4.4]nonan-3-one N-(3,4-dichlorophenyl)-4-[(E)-hydroxyiminomethyl]benzenesulfonamide 2-cyclopropyl-5,7-dimethoxy-1-(methoxymethyl)benzimidazole 3-[(4,5-dimethoxy-2-nitrophenyl)iminomethyl]-1H-indol-2-ol [2-(3,5-dimethylphenyl)morpholin-4-yl]-(1,7-naphthyridin-8-yl)methanone (2Z)-3,3-dimethyl-2-[5-[4-[1-(2-morpholin-4-ylethoxy)naphthalen-2-yl]-1,3,5-triazin-2-yl]pentylidene]butanoic acid [(5R,7S)-2,5,7-trimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazol-3-yl]urea 6-chloro-2,3-diiodobenzoic acid 3-[(E)-2-methoxyethenyl]-6,11-dihydrobenzo[c][1]benzoxepine ethane;2-[3-fluoro-4-(methylamino)phenyl]-7-(propylamino)indazole-5-carboxamide (6R,9S)-6-methyl-2-methylsulfanyl-9-pyridin-3-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 3-[7-(4,6-diphenyl-1,3,5-triazin-2-yl)naphthalen-2-yl]benzonitrile 1-(azidomethyl)-3-[4-(trifluoromethoxy)phenyl]sulfanylbenzene 3-[4-bromobutan-2-yl(prop-2-enyl)amino]phenol 2-azido-3,4-dichloro-5-(trifluoromethyl)aniline 1,3-dimethyl-2-(4-phenylphenyl)sulfonylbenzene 4-[(3R)-1-[(3,5-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one 3-(1,5-dimethylpyrazole-4-carbonyl)-2-methoxybenzamide 1-[4-methyl-2,6-di(propan-2-yl)phenyl]sulfanylimidazole [2-(4-aminophenyl)hydrazinyl]-oxoazanium 5-(azidomethyl)-3,3-difluoro-1H-indol-2-one (Z)-3-[4-amino-2,5-dimethyl-3-[[1-[(6-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-yl)sulfanyl]cyclobutyl]methoxy]phenyl]prop-2-enoic acid 4-(5,6-dichloropyridin-3-yl)oxybutan-2-one 1-[2,3-difluoro-4-(trifluoromethyl)phenyl]pyrazole-3-carboxamide;ethane 2-(2-bromo-4-fluorophenyl)-3-hydroxy-6,6-dimethylcyclohex-2-en-1-one 2-(5,6-dimethylpyridine-3-carbonyl)cyclohexane-1-carboxylic acid (2S)-1-[3-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)propanoyl]pyrrolidine-2-carboxylic acid 2-[5-[(E)-1-butylsulfanylprop-1-enyl]-1,3-thiazol-2-yl]ethanamine;5-methoxythiophene-2-carboxylic acid 4-azido-5-methylsulfonylpyrimidine 6-azidooxy-N,7-dibutylnaphthalene-2-carboxamide 6-[2,3-bis(ethenyl)phenyl]-9-methoxy-3H-furo[3,4-b]quinoline [(3aS,6aR)-5-propanoyl-2,3,4,6,6a-hexahydrofuro[2,3-c]pyrrol-3a-yl]-(4-methoxyphenyl)methanone;formic acid 2-methyl-4-[(E)-1,3,3-trifluorobut-1-enyl]sulfanylbenzoic acid 5-[2-[4-(1,3-benzoxazol-6-yl)piperazin-1-yl]ethyl]-7-methoxy-N-methylidenethieno[3,2-b]pyridine-3-carboxamide 5-(3,4-dihydronaphthalen-2-yl)-3-methyl-1H-imidazole-2-thione 6-methoxy-5-phenylcyclohexane-1,3-diamine 2-(methoxymethyl)-1-methylpyrrolo[3,4-b]quinoline 3-chloro-1,2,4-trimethyl-7H-pyrrolo[2,3-d]pyrimidine N-[4-(8-bromo-4-oxochromen-2-yl)phenyl]propanamide 4-[3,4-bis(phenylmethoxy)pyridin-2-yl]benzoic acid (2S)-N-hydroxy-1',2,3,4',5',7',8-octamethyl-6'-oxospiro[2-benzofuran-3,9'-xanthene]-1-carboxamide 1-bromo-2-[(1S,2R)-3-chlorocyclohexa-2,4-dien-1-yl]benzene 2-[4-[5-(3-chloro-4-fluorophenyl)-6-methoxypyridin-2-yl]butanoylamino]propanoic acid N'-[6-(3,4-dimethoxyphenyl)-9H-pyrido[3,4-b]indol-8-yl]thiophene-2-carboximidamide [(2S)-5,6-diamino-4-oxohexan-2-yl]-ethoxyphosphinate 2-amino-4,6-bis[[3-hydroxy-5-(hydroxymethyl)phenyl]methylidene]cyclohexa-1,3-diene-1-carbonitrile 7-[1,4-dimethyl-2-(4-nitrophenyl)-3H-pyrazol-5-yl]-1-[4-(morpholin-4-ylmethyl)phenyl]heptan-2-one 1-(4,6-dimethylpyrimidin-2-yl)-3-[5-fluoro-2-(methylamino)phenyl]urea 2-[5-(4-fluorophenyl)pyrazol-1-yl]-N'-hydrazinylethanimidamide N-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-1,4-dihydropyrimidine-2-carboxamide N-[4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]phenyl]-N-phenacylnonanamide ethane;N-(4-hydroxy-3-methoxyphenyl)-2-oxo-1,3-dihydropyrido[2,3-b]pyrazine-6-carboxamide 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]-5-ethoxypyridine 5-(2-fluorophenyl)-1-methyl-4,6,7,8-tetrahydropyrazolo[3,4-b][1,4]diazepine;(E)-N'-hydrazinylideneethanimidamide 3-[4-chloro-2-(fluoromethyl)anilino]-5-methylthiophene-2-carboxylic acid 2-[6,7-dimethyl-3-(trifluoromethyl)thieno[2,3-b]pyridin-2-yl]-5-hydroxyindene-1,3-dione N-azido-4-morpholin-4-ylaniline N-butyl-4-phenyl-1,2,3,6-tetrahydropyridine-5-carboxamide 1-(3,5-dimethylphenyl)-2,4-diethoxybenzene 2-[1-[4-(6-aminopyridin-3-yl)phenyl]ethylidene]-1,3-thiazolidine-3-carboxylic acid (2S,3R)-N-[1-(4-methoxybutylsulfonylamino)ethenyl]-5-oxo-3-phenylpyrrolidine-2-carboxamide 5-phenylmethoxy-4-propyltriazole N'-amino-5-[1-[4,6-dimethyl-2-(trifluoromethoxy)cyclohexa-1,3-dien-1-yl]oxyethyl]naphthalene-2-carboximidamide (2S)-4,4-dimethyl-6-[5-(2,2,2-trifluoroethoxy)pyridin-3-yl]heptane-2-thiol ethane;2-[4-(hydroxymethyl)phenoxy]acetic acid 4-(6,7-dimethylimidazo[1,2-a]pyridin-3-yl)-2-nitrophenol 1-[3-(4,4-dimethylcyclohexen-1-yl)phenyl]ethanone 4-bromo-2-[(3Z)-2-ethylpenta-1,3-dienoxy]benzoic acid 6-chloro-3-(2-methylpentan-2-yl)-2,4-dihydroisoquinolin-1-one 2-(N-benzyl-4,5-dimethyl-2-phenyldiazenylanilino)acetonitrile N-azido-2-[(4-carbamimidoylphenyl)methoxy]acetamide 3-(2,4,6-trichloroanilino)phenol 4-azido-6,7-diethoxyquinazoline 4-[(3R)-1-[(2S,5R)-6-azabicyclo[3.2.0]heptane-2-carbonyl]piperidin-3-yl]-N-methylbenzamide [3-(2,4-dihydroxyphenyl)-1H-pyrazol-5-yl]-[2-(trifluoromethyl)phenyl]iminoazanium N-[3-(1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]oxazin-10-yl)phenyl]formamide 1-[(2,5-dimethylpyrazol-3-yl)sulfonylamino]cyclopentane-1-carboxamide N-(2,3-dimethylphenyl)-4,5-bis[4-(dimethylamino)-2-fluoroanilino]-1,3-thiazole-2-sulfonamide N'-(2,6-diethylphenyl)benzenecarboximidamide 2-[5-(3,4-dimethoxyphenyl)pyridin-2-yl]-6-(1H-indazol-6-ylamino)-8-propan-2-ylpteridin-7-one N-[2-(4,5-dihydro-1H-imidazol-2-yl)phenyl]methanesulfonamide (2S)-3-hydroxy-N-[4-[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]-1,1-dimethylcyclobutane-1-carboxamide (2-ethyl-1,3-dioxoisoindole-5-carbonyl)azanium (2R,4S)-2-[[1-[(3,5-dimethylphenyl)sulfonylamino]-2-fluoro-7-oxo-6H-pyrrolo[2,3-c]pyridin-4-yl]oxy]-4-ethylhexanoic acid (3S,4R)-1-[5-fluoro-2-(5-methylfuran-3-yl)pyrimidin-4-yl]-N-methyl-4-(triazol-1-yl)pyrrolidine-3-carboxamide N'-hydroxy-5-(3,4,5-trimethoxyphenyl)pyridine-2-carboximidamide (E)-2-(4,5-dimethyl-1H-imidazol-3-ium-2-yl)-N-methylethenamine 2-(4-methylpiperazin-1-yl)quinoline;dihydrochloride 7-[5-amino-4-(5-bromo-2-hydroxyphenyl)-1,3-thiazol-2-yl]-N'-hydroxy-3H-azepine-4-carboximidamide 4-[(3R)-4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N-(oxan-4-yl)piperidine-1-carboxamide 2,4-dioxo-6-[4-(trifluoromethylsulfanyl)phenyl]-1,3-diazinane-5-carbonitrile 2-amino-3-[4,7-bis(carboxylatomethoxy)naphthalen-1-yl]propanoate;tin(4+) 3-(2,4-dihydroxyphenyl)-N-[[1-[3-fluoro-4-(4-methylimidazol-1-yl)benzoyl]pyrrolidin-3-yl]methyl]propanamide 1-azidooxy-2,3-bis(fluoromethyl)benzene N-methylspiro[chromene-2,4'-piperidine]-1'-carboxamide 5-[(4S)-6,8-dimethylspiro[3H-pyrano[2,3-c]pyridine-4,1'-cyclohexane]-2-carbonyl]-N,N-diethylpyridine-2-carboxamide N-(2,3-dichlorophenyl)-5-hydroxy-6-oxo-1H-pyrimidine-4-carboxamide 2-[3-methylbut-2-enyl(octyl)amino]phenol 2-(cyclohexyliminomethyl)phenol 2-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-3,4-dimethoxybenzoic acid N-(2,3-dihydro-1H-inden-5-yl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 2-(3,4-dimethylphenyl)sulfanyl-N'-hydroxypyrimidine-4-carboximidamide 3-(5,6-dichloro-2-methoxyquinoline-8-carbonyl)imidazolidine-1-carboxylic acid 2-[(1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-8-carbonylamino)methyl]-N-[2-(2-oxopyrrolidin-1-yl)ethyl]pyridine-4-carboxamide 1-(5-ethylfuran-2-yl)sulfonyl-3,4,6,7,8,9-hexahydro-2H-pyrimido[1,2-a]pyrimidine 4-azidooxy-5,7-dichloro-2H-isoquinoline N-[3-(4,5-dimethylimidazol-1-yl)propyl]-7,8-dihydroxyquinoline-2-carboxamide;hydrochloride 5-methyl-3-phenyldioxepine 2-methylbutanamide;N-(5-methyl-1,3-thiazol-4-yl)formamide;3-phenyl-5-[2-[2-[6-(trifluoromethoxy)quinolin-2-yl]ethynyl]pyridin-4-yl]-1H-pyridazine 3-(3,4-dimethoxyphenyl)-5-[(3E)-hexa-1,3,5-trien-3-yl]-N-methylthiophene-2-carboxamide 6-[5-[(dimethylamino)methyl]furan-2-carbonyl]-N-[2,4-difluoro-3-[(7S)-1,2,5-triazabicyclo[3.2.0]heptane-5-carbonyl]phenyl]-7,8-dihydro-5H-2,6-naphthyridine-3-carboxamide (E)-2,3,4-trimethyl-N-[5-methylidene-4-[4-(6-propanoylpyridin-2-yl)-1H-pyrazol-5-yl]piperidin-1-ium-1-ylidene]pent-2-enamide (7S)-N-(4-chlorophenyl)-7-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 2-cyclopropyl-5,6,7,8,9,10-hexahydrocycloocta[b]pyridin-4-amine N-(2,5-dimethoxyphenyl)-4-methylsulfanylquinoline-3-carboxamide;1-N-methylpropane-1,2-diamine 3-[3-chloro-4-[(3R)-1-[2-[4-methoxy-1-(trifluoromethyl)cyclohexa-2,4-dien-1-yl]acetyl]piperidin-3-yl]oxyphenyl]-5-(trifluoromethyl)-1,2,4-oxadiazole 1,3-bis(4-hydroxyphenyl)-2-[(4S)-4-(hydroxymethyl)cyclohexa-2,5-dien-1-ylidene]propane-1,3-dione 3-(6,7-dimethyl-1H-indol-2-yl)-4H-1,2,4-oxadiazol-5-one 3-benzyl-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine 5-[5,6-di(propan-2-yl)pyridin-3-yl]-3,4-bis(4-methylphenyl)benzonitrile 4-[(8-hydroxyquinolin-2-yl)methylideneamino]benzenesulfonic acid (1-azido-4,5,6-trimethylcyclohexa-2,4-dien-1-yl)benzene 2-[6,6-dimethyl-4-oxo-3-(5-propanoylpyridin-2-yl)-5,7-dihydroindazol-1-yl]-N-(4-fluorophenyl)acetamide 2-(1H-indol-3-ylmethylidene)-1,3-dioxoisoindole-4,6-dicarbonitrile 4-chloro-2-[4-(3,5-difluorophenyl)-1-bicyclo[2.2.2]octanyl]-N-methyl-N-piperidin-4-ylbenzamide 1-(2,4-diethoxyphenyl)pentan-3-one 2-[1,4-bis(sulfanyl)cyclohexyl]-3H-isoindol-1-one 2-[[(5S)-3-[4-fluoro-3-[[1-(3-oxobutyl)triazol-4-yl]methoxy]phenyl]-4,5-dihydro-1,2-oxazole-5-carbonyl]amino]acetic acid 1-[(2R)-4-[3-[6-(difluoromethyl)imidazo[1,2-a]pyridin-3-yl]-6-propan-2-ylidenepyridazin-1-yl]butan-2-yl]pyrazolo[3,4-d]pyrimidine 2,4-dichloro-N-hexyl-N-(1,2,4-triazol-4-yl)pyrimidin-5-amine N-(4-chlorophenyl)sulfonyl-1-cyclopentylpyrazole-3-carboxamide N-[(5S,7R)-2-(2-ethoxyphenyl)-5-methyl-7-thiophen-3-yl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]furan-2-carboxamide 2-(4-aminophenyl)-1-[4-[3-[(E)-2-[6-[4-chloro-3-(trifluoromethyl)phenoxy]pyrazin-2-yl]ethenyl]phenyl]piperidin-1-yl]ethanone 4-methyl-1,2-dihydrophenanthrene 1-[(6R)-2,6-dimethylcyclohexyl]-4-methoxybenzene 1-azido-5-methyl-2-(4-propan-2-yloxyphenoxy)benzene 2-(3,5-dimethylphenyl)-4,4-difluoro-1H-[1]benzofuro[2,3-a]indene 1-[[(2S)-2-ethylpyrrolidin-1-yl]methyl]-3,4-dihydroquinolin-2-one (3S,4R)-N'-[5-chloro-2-fluoro-4-(trifluoromethyl)phenyl]-4-(dimethylamino)pyrrolidine-1-carboximidamide 2-chloro-N-[(1R)-6,7-diethoxy-4-oxo-3H-quinazolin-2-yl]acetamide 3-[1-(dimethylamino)propan-2-yl]-1,7a-dihydroindole-6-carboxylic acid 3-(2,5-dimethylphenyl)imino-2-[[4-(hydroxyamino)phenyl]methylidenehydrazinylidene]propanoic acid N-(2,6-dimethylphenyl)-4-methoxy-3-[(6S)-1-methyl-8-oxo-6,7-dihydro-5H-isoquinolin-6-yl]benzamide;ethane 4-cyclopropyl-6-[6-(3,5-dimethoxyphenyl)pyridin-2-yl]oxypyrimidine 4-amino-1-[(E)-2-azidoethenyl]-5-fluoropyrimidin-2-one (1S)-N-[[4-[(Z)-1-amino-3-iminoprop-1-en-2-yl]phenyl]methyl]-2,2-difluorocyclopentane-1-carboxamide N-[4-(2,3-dihydro-1H-indol-5-yloxy)pyrimidin-2-yl]benzamide [4-(3,5-dimethylphenyl)piperazin-1-yl]-(oxan-4-yl)methanone [4-(4-chlorocyclohexa-1,3-dien-1-yl)oxy-2H-pyridin-1-yl]-(5-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl)methanone (2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl)-[1-[(Z)-3-propan-2-ylidenehept-1-enyl]piperidin-3-yl]methanone 2-(4-methylsulfonylphenyl)-1,3-benzothiazole 3-(1,3-benzothiazol-2-ylmethyl)-4-hydroxynaphthalene-2-carboxamide;1H-imidazole 3-[2,5-dioxopyrrol-1-yl(phenyl)methyl]benzenesulfonamide 5-bromo-4-N-[(2E,3Z)-3-ethylidene-1-methylpiperidin-4-yl]pyrimidine-2,4-diamine 6-(4-nitrophenyl)-3,7,8,9-tetrahydropyrimido[5,4-e]indolizin-4-one 4-[(3S,5R)-3-azido-2-oxo-5-phenylpyrrolidin-1-yl]benzaldehyde 7,9-dibromoperylene-3-carboxylic acid 1-methyl-4-[3-(trifluoromethoxy)phenyl]piperidine;N,2,6-trimethylpyrimidin-4-amine 3-amino-5-methyl-1-[[4-(2-pyrrolidin-1-ylethoxy)phenyl]methyl]pyrazole-4-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-6-(4-pyrrolidin-1-ylquinazolin-2-yl)spiro[2.5]octane-2-carboxamide (Z)-3-(4-acetyloxy-2,6-dimethoxyphenyl)prop-2-enoic acid N-[2,4-difluoro-3-(5-thiophen-2-yltetrazol-1-yl)phenyl]-1H-indole-6-sulfonamide 1-(5-tert-butyl-2,3-dimethylphenyl)sulfonylpiperidine 1-(7-chloroquinolin-4-yl)pyrrolidine-3,4-diamine;2,2,2-trifluoroacetic acid 3-(4,7-dimethoxynaphthalene-2-carbonyl)oxypropanoic acid 5-(1,3-benzothiazol-2-yl)-4-[2-[3-methoxypropyl(methylsulfonyl)amino]ethyl-methylamino]pyridine-2-carboxylic acid (2S)-2,5-diamino-6-oxo-3-phenylhexanamide N'-[2-chloro-3-(2,6-dioxopiperidin-3-yl)-1H-indol-5-yl]oxamide N-(2-methylphenyl)-1,3-bis[2-oxo-2-(propan-2-ylideneamino)ethyl]thiourea 2-[2-(1,3,2-dioxaborolan-2-yl)phenyl]-4-methoxypyrimidine 2-azido-3-methylsulfanylacridine 1-chloro-3-methylbenzene;2,4-difluoro-N'-(oxan-4-yl)benzenecarboximidamide 1-chloro-2,3-diphenylcyclohexa-2,4-dien-1-amine 6-bromo-1'-[2-[1-(5,6-dimethoxypyridin-3-yl)ethylamino]thieno[3,2-d]pyrimidine-4-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one N-[(2S)-1-oxo-3-phenyl-1-pyrrolidin-2-ylbutan-2-yl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxamide 2-(2,4-dichloro-6-methylphenyl)benzoic acid N-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-ylmethyl)-N-(5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-yl)acetamide;hydrochloride 3-[4-(2,5-dioxopyrrolidin-1-yl)phenyl]sulfonyl-N'-(2-phenylethyl)propanimidamide N-[6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]propane-2-sulfinamide 4-[3,5-bis(4-cyanophenyl)pyridin-2-yl]-3,5-dinitrobenzonitrile 6-hydroxy-5-(indole-2-carbonyl)-1,3-dimethylpyrimidine-2,4-dione N-[1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-3-yl]prop-2-enamide 3-[2-[3-(dimethylamino)azetidine-1-carbonyl]-4-propan-2-ylphenyl]piperidine-2,6-dione (4R)-1-[3,5-bis(trifluoromethyl)phenyl]-7,8-dichloro-6-fluoro-4-hydroxy-N-propan-2-yl-3,4-dihydro-2H-quinoline-3-carboxamide N-[[5-(2,4-dimethoxyphenyl)pyridin-3-yl]methyl]ethanamine ethane;5-[(1Z,3E)-4-fluorohexa-1,3,5-trienyl]-4-methyl-3H-1,2,4-thiadiazole 3-[(5S)-5-amino-5-methylpiperidin-2-ylidene]-4H-1,4-benzoxazin-7-amine 5-phenyl-8H-cyclohepta[d]pyrimidine 4-(azidomethyl)-2-[5,6-bis(phenylsulfanyl)pyrazin-2-yl]phenol (3S,4R)-3-fluoro-N-[(2S)-1-[[(2R)-1-hydroxy-3-phenylpropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]piperidine-4-carboxamide (E)-N'-[(1S)-2-[4,7-dimethoxy-1-[3-(trifluoromethyl)phenyl]sulfonylindole-3-carbonyl]cyclohexyl]-N-ethylprop-1-ene-1,3-diamine N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]oxane-2-carboxamide;5-fluoropyridine-3-carbonitrile 6-[2,4-difluoro-3-(trifluoromethoxy)phenyl]sulfonyl-N-hydroxyhexanamide 2-tert-butyl-4-chloro-6-methyl-3-phenylpyrrolo[1,2-a]indole 3-[4-(1,3-benzothiazol-2-yl)phenyl]hexanoic acid N-[4-(1-benzothiophen-7-yloxy)phenyl]acetamide 2-[2-ethoxy-4-(1,3,4-oxadiazol-2-yl)phenyl]benzotriazole N-[4-bromo-2-(1,1-dioxothiolan-3-yl)pyrazol-3-yl]pyridine-3-sulfonamide 1-cyclopropylsulfonyl-3,4-dihydro-2H-1,5-benzodiazepine 2-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-(2-ethoxy-2-oxoethyl)amino]decanoic acid 3-[4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]-N-prop-2-enylanilino]butanoic acid 1-(4,5-dichloro-2-methoxyphenyl)sulfonylpiperidine 2-[2-(trifluoromethyl)pyridin-3-yl]pyrimidine 5-hydroxy-4,6-dimethylpyrimidine-2-carboxamide;1-[2-(3,4,7,8-tetrahydronaphthalen-1-yl)ethyl]pyrrolidine (3S,4R)-N-(2-methoxyphenyl)-1-pyridin-3-ylsulfonylpyrrolidine-3,4-dicarboxamide 2-amino-9-[(4R,5S)-3-fluoro-1-methylpiperidin-4-yl]-8-propanoylpyrido[2,3-b]indole-7-carboxamide (3R)-7-methoxy-2,4,5,8-tetraphenyl-1,3,4a,9b-tetrahydroindeno[2,1-b]pyridine 4-chloro-N-[(2R)-2,3-dihydroxypropyl]benzenesulfonamide 6-chloro-7-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl)-N-ethyl-4-oxochromene-2-carboxamide;methane 2-cyclohexyl-1,3,5,6-tetrahydrobenzo[e]azulene 1-(4-amino-1,2,5-oxadiazol-3-yl)-N-[(Z)-butan-2-ylideneamino]-5-[(5E)-3,6-dimethylideneocta-5,7-dienyl]triazole-4-carboxamide 4-(dipropylamino)-3-ethoxybenzenesulfonic acid 3,4-dimethyl-6-phenyl-8,10-dihydro-7H-chromeno[2,1-c]pyrazole 1-cyclopentyl-5-(4-fluorophenyl)-2,3-dihydrotetrazol-1-ium 3-[4-(2,5-difluorophenyl)-1H-indol-2-yl]-5-pyridin-4-yl-2H-pyrazolo[3,4-b]pyridine 1-(3,4-difluorophenyl)sulfonyl-2-[(E)-5-prop-2-enylundec-9-enoxy]pyrrolidine 7-methyl-6-(1,3,5-triazin-2-yl)indolo[2,3-c]quinoline 5-bromo-4-[4-(methoxymethyl)piperidin-1-yl]-1H-pyrimidin-6-one N-(2,5-dichlorophenyl)-2-[3-oxo-4-[[(E)-3-pyridin-3-ylprop-1-enyl]amino]-1H-isoindol-2-yl]butanamide 4-(2,5-dimethylphenyl)-1-(1H-inden-1-id-2-yl)piperidine;zirconium 2-amino-4,5-dimethylbenzamide;3-N-[2-(7-carbamoyl-2,3-dihydroindol-1-yl)-2-oxoethyl]-6-propan-2-ylidenecyclohexa-1,4-diene-1,3-disulfonamide 6-[(2R)-2-azido-4,4-dimethylcyclopenten-1-yl]-N-benzylimidazo[2,1-b][1,3]thiazol-5-amine (4-azidopyrimidin-5-yl)-[3-ethoxy-2-[(1R,2S)-2-methoxycyclohexyl]oxyphenyl]methanone 2-methyl-5,6-didehydropyrene 4-cyclopropyl-N-[(2,3,5,6-tetramethoxyphenyl)methyl]-1H-pyrrole-3-carboxamide (Z)-N'-ethenyl-3-[2-methylidene-3-[6-methyl-2-propan-2-yl-5-(trifluoromethoxy)indol-1-yl]cyclopentyl]but-2-enehydrazide 2-[5-(4-fluorophenyl)-1-phenylpyrazol-3-yl]-N,N-dimethoxyethanamine 1-[3-[[4-(2,2-dimethylpropoxy)phenyl]methylideneamino]phenyl]ethanone 4-[(3R)-3-azidopyrrolidine-1-carbonyl]benzonitrile 6-(9,10-difluorodecoxy)-2-methyl-3H-isoindol-1-one (2R,4S)-N-[4-[(3,5-dimethylpyridin-2-yl)amino]phenyl]-4-fluoropyrrolidine-2-carboxamide 1-[4,6-bis(ethenyl)-5H-naphthalen-2-yl]-N-methylmethanamine;ethane;2-methylpropane 1-(5-chlorothiophen-2-yl)sulfonyl-3,4-dihydroisoquinoline N-(4-chlorophenyl)-6,7-dihydroisoquinolin-5-amine (Z)-3-[3,5-bis(trifluoromethyl)phenyl]prop-2-enoic acid;methane N-[2,3-difluoro-4-(1H-pyrrolo[3,2-b]pyridine-6-carbonyl)phenyl]-5-(dimethylamino)pentanamide N-[3-(dimethylamino)propyl]-6-methoxypyrimidine-4-carboxamide (5E)-1-ethenyl-5-[(Z)-prop-1-enyl]-2,3-dihydropyrido[2,1-a]isoindole N-methyl-1-(6-propan-2-ylpyridin-3-yl)methanimine 4-methyl-N-[(1S,2R)-2-pyridin-3-ylcyclopropyl]pyrimidine-5-carboxamide 1-[3-(1H-imidazol-2-yl)propanoyl]-5,7-dimethoxyisoquinoline-6-carboxylic acid (3S,4R)-3-ethoxy-1-[4-[2-fluoro-5-methyl-4-(trifluoromethyl)phenyl]-6,7-dihydrothieno[3,2-d]pyrimidin-6-id-6-yl]piperidine-4-carboxylic acid;uranium N-(4,6-dimethylpyrimidin-2-yl)-4-[3-nitro-N-(1,3-thiazol-5-yl)anilino]benzenesulfonamide [6-(4,5-dimethylcyclohexen-1-yl)pyrazin-2-yl]methanamine 1-[(2-methyl-5,6,7,8-tetrahydroquinolin-3-yl)amino]ethanol 4-hydroxy-3,6-dimethyl-1-benzofuran-2-carboxylic acid 2-amino-5-[3,4-dichloro-6-(4-iodophenyl)quinolin-8-yl]benzenesulfonamide 2-methyl-6,6a,7,11b-tetrahydrochromeno[4,3-b]chromene (4-aminophenyl)sulfonyl-[4,5,6-trimethoxy-3-(4-methylpiperazin-1-yl)pyridazin-4-yl]azanium 2,4-dichloro-N-[5-[(6-fluoro-3H-indol-2-yl)amino]pyrazin-2-yl]benzenesulfonamide (3S,5R)-5-[(2S)-4-hydroxybutan-2-yl]-1,3,4,6,7,8-hexahydrocyclohepta[c]pyridine-3a-carboxylic acid 2-[4-(5,6-diphenylpyridin-3-yl)-1,3,5-triazin-2-yl]-5-fluorophenol 3-methoxycarbonyl-5-nitrobenzoic acid (2R)-3,4-dihydroxy-1-[(4S,5S)-2,4,7-trimethyl-6-oxo-8H-pteridin-5-yl]butan-2-one 1-[4-(aminomethyl)phenyl]sulfanyl-3-azidopropan-2-amine 2-[4-(dimethylamino)phenyl]-N-(3-hydroxypropyl)quinoline-4-carboxamide 2-(2,2-difluoroethyl)-N-[4-[1-methoxypropan-2-yl(2-oxoethyl)amino]phenyl]benzamide 2-(4,6-diphenyl-1,3,5-triazin-2-yl)-9H-fluoren-1-ol (2R)-N-[1-(3,5-difluorophenyl)-4-(ethylamino)butan-2-yl]-4-oxopyrrolidine-2-carboxamide N-[2-(2,3-dihydro-1H-inden-5-yloxy)pyrimidin-4-yl]-6-methylpyridine-3-carboxamide 4-(2,6-dimethoxyphenyl)-3-methyl-1H-pyrrole-2-carboxylic acid 1-cyclopentyloxy-4-methoxy-2-propan-2-ylbenzene 1-[4-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridine-7-carbonyl)piperazin-1-yl]butan-1-one N-benzylsulfonyl-2-[5-(2,3-difluorophenyl)-6-ethoxypyridin-2-yl]-1H-indole-7-carboximidate 2-(6-azidopyridin-3-yl)-7-(4-fluorophenyl)imidazo[1,2-a]pyridine (1S)-5,6-dimethyl-N-[1-[4-(trifluoromethoxy)phenyl]ethylideneamino]-2,3-dihydro-1H-indene-1-carboxamide 2-[(1R)-5-[2-chloro-6-(trifluoromethoxy)phenyl]-3,4-dihydro-2H-chromen-2-yl]ethanamine;ethane 1-[[4-(3,5-dimethylbenzoyl)morpholin-2-yl]methyl]pyrrolidine-2-carboxylic acid N-cyclopropyl-2-[4-(2,3,6-trifluorophenoxy)piperidin-1-yl]-7,8-dihydropyrido[2,3-d]pyrimidine-5-carboxamide;hydrochloride 4-[(E)-2-(3,4-dihydroxyphenyl)ethenyl]benzenesulfonamide (3E)-4-amino-3-[[4-hydroxy-3-[(2-phenyl-5-propan-2-ylphenoxy)methyl]phenyl]methylidene]azete-2-thione (2R)-2-[4-chloro-3-[1-methyl-5-(1,2-thiazol-4-yl)pyrazol-4-yl]phenoxy]propanoic acid 4-(2,6-difluorophenoxy)-3H-pyrido[2,3-b]pyrazine 3-[4-[2-(2-chlorophenyl)ethoxy]phenoxy]cyclobutan-1-amine 4-[[8-(2,3-dichlorophenyl)quinazolin-5-yl]methylidene]pentanal;ethane 1-[6-azidooxy-2,3,5-trimethyl-4-(4-nitrophenoxy)phenyl]-4-chlorobutan-1-one N-(3,4-difluorophenyl)-3-methoxybenzamide N-[4-(2,4-dimethylphenyl)-1H-pyrazol-5-yl]-3,6-difluorocyclohexa-1,3-diene-1-carboxamide 2,6-dimethylpyridine;ethane;4-phenylquinolin-5-amine 1-(2,4-difluorophenyl)-3-(1H-indol-5-ylmethylideneamino)thiourea ethane;2-[1,4,7-tris(methoxymethoxy)isoquinoline-3-carbonyl]cyclohexene-1,3-dione 2-[3,5-bis(trifluoromethyl)phenyl]-N,4,6-trimethylaniline;1-cyclohexa-1,5-dien-1-ylnaphthalene;2-methylidenecyclopentane N-(3,4-difluorophenyl)-7-methyl-2-(1H-pyrazol-5-yl)quinoline-4-carboxamide 2-methylsulfanyl-3,10b-dihydro-1H-imidazo[4,5-b]indazole;hydrochloride 3-(3-aminophenyl)sulfonylbenzaldehyde 5-(2-azidocyclohexyl)oxy-2,3-dihydroinden-1-one 4-[(5S)-2-amino-5,6-dimethyl-8-(2-morpholin-4-ylethoxy)-9-oxo-1H-imidazo[1,2-b]isoquinolin-3-yl]cyclohexane-1-carboxylic acid 4-[5-(5-methoxypyridin-2-yl)furan-2-yl]sulfonylpiperazine-1-carboxylate 4-[2-(3,5-dichlorophenyl)propyl]phenol 2-[3,5-bis(trifluoromethyl)phenyl]-N-(4-cyclohexa-1,5-dien-1-yl-6,7-dihydronaphthalen-1-yl)-N-ethylacetamide (2Z)-3-methyl-2-[(Z)-2-methylbutan-2-ylidenehydrazinylidene]-1,3-thiazolidin-4-one;3-methylbenzonitrile 3-chloro-4-[3,5-difluoro-2-(methylamino)phenyl]sulfanyl-1H-pyrrolo[2,3-b]pyridine-6-carbonitrile;ethane N-[2-(2,3-dihydroindol-1-yl)ethyl]-3-methoxy-4,6-bis(phenylsulfanyl)pyridine-2-carboxamide N-(2-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 4-[8a-(2,6-difluorophenyl)-2-methyl-1H-imidazo[1,5-a]pyrimidine-7-carbonyl]-3-cyclopropylpiperazin-2-one N-(3,5-dimethylphenyl)-2-[(2Z)-4-oxo-2-pyrimidin-2-ylimino-1,3-thiazolidin-5-yl]acetamide N-(2,5-dimethylphenyl)sulfonyl-1-methylpyrazolo[4,3-c]pyridine-6-carboxamide 4-(methylamino)-3-[(E)-2-(1,2,3,6-tetrahydropyridin-5-yl)ethenyl]benzaldehyde (4S)-2-ethyl-8-phenylmethoxyspiro[4,7-dihydrochromene-5,3'-oxetane] 4-fluoro-N,1-dimethylindole-6-carboxamide 1,3-diphenylpropane-2-sulfonate 4-[3-fluoro-5-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)phenyl]piperazin-2-one;dihydrochloride 2-(4,5,6,7-tetrahydro-1H-indazole-3-carbonylamino)pentanedioic acid 2-[5-(5-chloro-2,3-dihydro-1H-inden-4-yl)pyridin-3-yl]sulfonylpropanoic acid 2-[4-ethoxy-6-[(5S)-2-(methylamino)-2,7-dioxo-1,3-diazabicyclo[3.2.0]heptan-3-yl]pyrimidin-2-yl]sulfanyl-N,N-dimethylacetamide 2-(4,5-dihydro-1H-imidazol-2-yl)-N-[3-(2,6-dimethoxyphenyl)imidazo[4,5-c]pyridin-7-yl]propanamide 5-chloro-2,4-dimethoxy-N-(6-oxo-1H-pyridin-3-yl)benzenesulfonamide 2-[(1S)-1-[4-[7-(4,5-dimethyl-6-oxocyclohexa-1,3-dien-1-yl)oxythieno[3,2-b]pyridin-2-yl]phenyl]ethyl]isoindole-1,3-dione [6-bromo-1-ethyl-7-(trifluoromethoxy)imidazo[4,5-c]pyridin-2-yl]methanol N-[4-methoxy-2-(1,3-thiazol-5-yl)phenyl]-1-morpholin-4-ylcyclopropane-1-carboxamide (5E)-3,6-dimethyl-4-[2-oxo-2-(1,2,3,6-tetrahydropyridin-4-yl)ethoxy]-5-propylidenepyridine-2-carboxylate (2-chlorophenyl)methyl-diethoxyphosphoryloxyphosphane 1-[4-[2,5-difluoro-6-(2-hydroxypropan-2-yl)pyridin-3-yl]-3-methoxyphenyl]-3-[(Z)-1H-indol-3-ylmethylideneamino]urea 2-(4-butylphenoxy)-3H-pyrido[3,4-d]pyrimidin-4-one [4-[5-chloro-7-(2,3-dihydro-1H-imidazol-2-ylmethoxy)-4-oxoquinazolin-3-yl]-3-fluorophenyl]oxidanium 1-[4-[3-chloro-5-methyl-2-[[3-[(2,4,6-trifluorophenyl)methoxy]piperidin-1-yl]methyl]imidazo[1,2-a]pyridin-7-yl]piperazin-1-yl]ethanone 6-(4-chlorophenyl)-N-[2-methyl-2-(naphthalen-1-ylsulfonylamino)propyl]pyridazine-3-carboxamide N-ethyl-2,5-difluorobenzenesulfonamide 4-azido-5-chloroquinoline (1R,2S)-N-[8-amino-6-(5-methylpyrazine-2-carbonyl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide [2-amino-4-(pyridin-3-ylmethoxy)-1,5-dihydroimidazol-4-yl]methanol 7-[(3R,4S)-4-(2-methoxyethylamino)oxolan-3-yl]pyrrolo[2,3-d]pyrimidine-6-carboxylic acid 3-azido-1-(2,5-difluorophenyl)pyrrolidine [5-[(4-chlorophenyl)sulfonylmethyl]-2,3-dihydro-1H-inden-1-yl]carbamic acid N-[(3E)-hexa-1,3,5-trien-3-yl]oxybenzenesulfonamide 3-(4-chlorophenyl)-1-methyl-1-[2-oxo-5-(trifluoromethyl)pyrimidin-1-yl]urea 3-[(2Z)-3,4-dimethylhexa-2,6-dien-2-yl]-1,2,5-trimethylbenzene;ethane 1-(3,5-dichlorophenyl)sulfinylpyrrolidine;2,4,6,8-tetramethylquinolin-7-amine N-(2,6-difluorophenyl)-1,2-benzothiazole-3-carboxamide;3-[4-(trifluoromethoxy)phenyl]oxolane 2-[3-(3,5-dimethoxyphenyl)pyrazol-1-yl]benzamide N'-[4-(7-chloroquinolin-4-yl)oxyphenyl]ethanedithioamide 3-(benzenesulfinyl)-2-methylsulfonylphenol 4-[2,5-bis(trifluoromethyl)phenyl]-4-(N'-methylcarbamimidoyl)piperidine-1-carboxylic acid (4R)-4-(3-bromophenyl)-1,3-dimethyl-6,7,8,9-tetrahydro-4H-pyrazolo[3,4-b]quinolin-5-one 5-(4,5-dihydroxy-2,3,7-trimethylnaphthalene-1,2-dicarbonyl)-N,N,2-triethylbenzenesulfonamide 2-[4-(2,3-dihydroindole-1-carbonyl)phenyl]sulfanyl-N-(3-hydroxypropyl)-2-methylpropanamide 2-[4,6-bis(2,3,4,5,6-pentafluorophenyl)-1H-1,3,5-triazin-2-yl]phenol 7-chloro-3-methyl-N-(2-morpholin-4-ylethyl)isoquinoline-1-carboxamide;cyclohexane 2-[(4S)-1-[3-bromo-5-ethoxy-4-[(3-nitrophenyl)methoxy]benzoyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-4-carbonyl]-1,3-benzothiazole-6-carbonitrile 2-chloro-6-[(2R,3S)-1-methyl-5-oxo-2-thiophen-3-ylpyrrolidin-3-yl]benzoic acid 6-[(1,5-dimethylpyrazol-3-yl)methyl]-2-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (2Z)-N,4-dimethylpenta-2,4-dien-1-imine;3-methylcyclohexa-1,5-diene;2-[2-(2-phenylphenoxy)ethoxy]ethanamine 1-(4-nitrophenyl)sulfanylpyrrolidine [(4S)-6-hydroxy-2,3-dihydrochromen-4-yl]carbamic acid (2Z)-1-methyl-2-propylidenequinoline-3-carboxylic acid 4-(aminomethyl)-N-[2-oxo-2-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)piperidin-1-yl]ethyl]benzamide 3-[1-(4,5-dimethylpyrimidin-2-yl)azetidin-3-yl]-1-phenyl-1,8-naphthyridin-2-one 2-(5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-yl)phenol 4-[2,2-dimethoxyethyl(3-methylbut-2-enyl)amino]-N-thiophen-2-ylbenzenesulfonamide 1-[(4-chlorophenyl)methyl]piperidine N-[(1R)-1-phenylethyl]pyridine-3-carboxamide 2-[3-[4-(4,7-dimethoxy-1H-benzimidazol-2-yl)pyridine-2-carbonyl]phenyl]-N-phenylpropanamide 1-azido-2,4-dichloroanthracene 4-[4-(3,5-dimethylanilino)pyridin-2-yl]piperazine-1-carboxamide (6R)-7-acetyl-3-ethylsulfanyl-6-methyl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 5-[3,5-bis(trifluoromethyl)phenyl]-N-dichlorophosphorylpentan-1-amine 5-[(E)-2-[4-chloro-3-(trifluoromethyl)phenyl]ethenyl]-N'-[(Z)-1,3-diaminobut-2-enylidene]-1-(oxan-4-yl)imidazole-4-carboximidamide 2-[4-(1,3-dioxoisoindol-2-yl)piperidin-1-yl]-N'-hydroxyethanimidamide 2-(7-chloro-3,4-dimethyl-5H-1,2,4-benzotriazin-6-yl)benzene-1,4-disulfonate N-(4-amino-3,4-dioxo-1-pyridin-2-ylbutan-2-yl)-4-pyrazin-2-yl-1H-imidazole-5-carboxamide 1-(5-azido-2-fluorophenoxy)-4-(trifluoromethoxy)benzene 2-(2-ethoxyethyl)benzo[g][1,3]benzothiazole N-[3,5-dimethyl-4-[2-[(3R)-oxolan-3-yl]oxyethyl]pyridin-2-yl]sulfanylcyclopropanecarboxamide 1-(4,5-dichlorothiophen-2-yl)sulfanyl-3-[4-[(E)-4,6-dioxohept-2-enoxy]phenyl]urea 6-[4,4-dimethylpentanoyl(methyl)amino]pyridine-3-carboxylic acid 2-[4-(aminomethyl)phenyl]-1-[4-hydroxy-3,5-bis(hydroxymethyl)piperidin-1-yl]ethanone (2R,3S)-5,7-dibenzyl-6-methoxy-N-methyl-2-phenyl-1,3,4,9-tetrahydropyrido[2,3-b]indole-3-carboxamide 6-[4-(6-methoxypyrimidin-4-yl)piperazine-1-carbonyl]pyridine-3-carbonitrile N-[1-(2,4-difluorophenyl)ethyl]-6-(methoxymethyl)-3,4-dihydro-1H-pyrrolo[2,1-c][1,4]oxazine-8-carboxamide 2-[6,7-dichloro-1-(4-hydroxyphenyl)-4-[3-(trifluoromethyl)phenyl]sulfonylindol-5-yl]acetamide 2-[4-(5,6-difluoronaphthalen-1-yl)phenyl]-5-(trifluoromethyl)pyridine 1-cyclopropylsulfonyl-3,4,6,7,8,9-hexahydro-2H-pyrido[2,3-b]indolizine 5-(cyclopropanecarbonylamino)-3,4-dihydroisoquinoline-1-carboxamide 2-(5,7-dimethylbenzimidazol-1-yl)-6H-[1]benzofuro[3,2-b]pyridin-6-ide;iridium;trimethyl-(6-phenyl-4H-thiopyran-3-id-2-yl)silane (2R)-2-amino-3-[4-(2,5-difluorophenyl)-3-methoxy-1H-indol-7-yl]propanoic acid (2R,3S)-1-cyclohexyl-N-[(4-methoxyphenyl)methyl]-N'-methylsulfonylpiperidine-2,3-dicarbohydrazide N-[(2S)-3-hydroxy-1-oxo-1-piperidin-4-ylpropan-2-yl]-7,10,11-triazaspiro[5.6]dodecane-10-carboxamide 5-(1,2,3,4-tetrahydroisoquinoline-7-carbonyl)pyrimidine-2-carboxylic acid 1-azido-N-phenyl-6,7,8,9-tetrahydroimidazo[4,5-c]quinolin-2-amine 4-bromo-6-ethyl-2-[[4-(trifluoromethoxy)phenyl]iminomethyl]phenol 4-[4-azidooxy-1-(9H-fluoren-2-yl)hexan-3-yl]pyridine 1,3-diamino-1-[4-(2,4-dimethoxyanilino)cyclohexa-2,4-dien-1-yl]urea [(3S,5R)-4-benzyl-3,5-dimethoxycyclohexa-1,5-dien-1-yl]-phenoxyphosphinic acid 3-[[4,5-bis(2-methylphenyl)-1H-imidazole-2-carbonyl]amino]-4-[methyl(prop-1-enyl)amino]butanoic acid;ethane N-(2-bromo-6-chlorophenyl)-5-methyl-4-(morpholine-4-carbonyl)-1,3-thiazole-2-carboxamide 5-(2,6-difluorophenyl)-3H-1,4-benzodiazepine 2-chloro-6,11-dihydroindolo[1,2-c]quinazoline 3-(azepane-1-carbonyl)-4-hydroxybenzaldehyde 3,6-ditert-butyl-8-(2-propan-2-yloxyethoxy)quinoline 5-methylsulfonyl-1,2-dihydropyrazolo[1,2-a]pyridazine 4-[(E)-1,2-bis(4-hydroxy-3-nitrophenyl)ethenyl]benzenesulfonic acid [3-chloro-2-(trifluoromethyl)phenyl]-diphenylphosphane 2-[5-(methoxyamino)pyrazin-2-yl]sulfanyl-4-propyl-1H-pyrimidin-6-one 4-(2,3-dichlorophenyl)-2,5-dimethylfuran N-[(1S)-3-[5-ethylsulfonyl-6-[4-(trifluoromethyl)phenyl]pyridin-2-yl]cyclohexyl]propanamide N-methyl-6-[3-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazol-1-yl]pyridazine-3-carboxamide 4-(cyclobutylamino)-6-[(2,5-dimethoxyphenyl)methyl]-1H-1,3,5-triazin-2-one 2-[6-[[6-(cyclopropanecarbonylamino)pyridin-3-yl]sulfonylmethoxy]-4,5,6,7,8,9-hexahydrocarbazol-2-yl]acetic acid 5-(2-butyl-4,6-dioxothieno[3,4-c]pyrrol-5-ium-1'-carbonyl)pyridine-2-sulfonamide N-[1-cyclohexyl-2-(2,4-dioxocycloheptylidene)-2-methoxyethyl]-N-(3,5-dimethylpyridin-4-yl)formamide 4-(2,3-dimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidine 4-N,4-dimethyl-6-N-(2-methylprop-1-enyl)pyrimidine-4,6-diamine 2-[5,8-difluoro-3-methyl-7-(2-methylpyrazol-3-yl)naphthalen-1-yl]propan-2-ol;ethane 4-[6-[(2-ethylpyrimidin-5-yl)amino]pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexan-1-ol 4-cyclohexa-1,5-dien-1-yl-1,3-diphenylazetidine N-[2,5-difluoro-4-(3,4,5,6-tetradeuteriopyridin-2-yl)phenyl]ethanesulfonamide (2S)-2-[[4-(3,5-dimethoxyphenyl)benzoyl]amino]-N-hydroxy-6-(prop-1-en-2-ylamino)hexanamide (6-methoxypyridin-2-yl)-[(5S,7R)-2-methyl-6-oxa-2-azaspiro[4.5]decan-7-yl]methanone;2,2,2-trifluoroacetic acid 1-methyl-2,3,5-trinitro-4-phenylbenzene 2-chloro-N-[4-chloro-3-(trifluoromethyl)phenyl]acetamide 5-(4-aminophenyl)-N'-[1-hydroxy-3-methyl-2-methylidene-6-(trifluoromethoxy)pyrimidin-4-yl]sulfanylpyridine-2-carboximidamide N-[[3,4-bis(trifluoromethyl)phenyl]methoxy-pyridin-2-ylmethylidene]hydroxylamine 2-[(4-bromophenyl)methyl]-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-4-one 3-[(2,4-dioxo-1H-pyrimidin-5-yl)methylideneamino]-N-[(1R)-1-(3,5-dimethylphenyl)ethyl]propanamide 5-methyl-2,4,6-triphenoxypyridine 2-(2,3-dihydrothiophen-5-yl)-1,7-naphthyridine 1-(4-methoxyphenyl)-N-[(3S)-1,1,3,2-tetramethyl-6,7-bis(trifluoromethyl)-1,3,5,2,4,9-hexahydrobenzo[f]isoquinolin-8-ylidene]methanesulfonamide 1-bromo-2-(4-butylcyclohexyl)benzene 7-methoxy-2,3-dihydrochromene-4-thione 1-[4-[2-fluoro-5-(6-methyl-7,8-dihydroquinolin-3-yl)phenyl]piperidin-1-yl]ethanone (2S)-N-[1-amino-3-(4-azidophenyl)propan-2-yl]-2-methoxy-3-phenylpropanamide 3,5-dimethyl-1-[2,4,6-tri(propan-2-yl)phenyl]pyrazole;ethane 3-[4-[(3R)-pyrrolidine-3-carbonyl]piperazin-1-yl]pyridazine-4-carbonitrile;hydrochloride 4-[2-(1,3-benzodioxol-5-yl)ethoxy]-N-[5-[[2-methyl-6-(2-methylpropoxy)pyridine-4-carbonyl]amino]-2-bicyclo[4.1.0]hepta-1,3,5-trienyl]benzamide 2-methylsulfinyl-3-[4-(trifluoromethyl)phenyl]oxirane (3Z,5E)-5-amino-N'-[(2S)-1-hydroxypropan-2-yl]-7-phenylmethoxyhepta-3,5-dienimidamide 7-(4-chlorophenyl)-5,6-diethyl-2-[(3-methoxypyrazin-2-yl)amino]-8H-pteridin-7-ol ethane;5-methyl-2,4-diphenyl-6H-furo[3,4-d]pyrimidine 4-[(Z)-2-amino-3-[methyl-[1-oxopropan-2-yl(phenyl)carbamoyl]amino]-3-pyridin-4-ylprop-1-enyl]-N-phenylbenzamide N-[2-methyl-4-(1,2,4-triazol-1-yl)phenyl]-3-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)propanamide (4R)-4-[6-[5-(2,6-dimethylpyridin-3-yl)-1H-imidazol-2-yl]-7,8-dihydro-5H-1,6-naphthyridin-2-yl]-N-methylcyclopentan-1-imine 1-(2,4-dimethoxyphenyl)sulfonyl-3-(5-fluoro-2,3-dihydroindol-1-yl)propan-2-ol 2-chloro-4,7-dimethyl-5H-pyrido[3,4-d]pyrimidine;ethane 3-bromo-N-[5,7-difluoro-1-[(2R)-1-hydroxypropan-2-yl]-6-methoxybenzimidazol-2-yl]cyclohexane-1-carboxamide N-[(2R)-3,4-dihydro-2H-chromen-7-yl]-3-methoxy-2,5,6-trimethylcyclohex-2-ene-1-carboxamide 4-N-(3-chloro-2-methylphenyl)-6-phenylpyrimidine-4,5-diamine;dihydrochloride N-[1,3-dimethyl-7-(3,4,5-trifluorophenyl)-2H-azepine-6-carbonyl]pent-4-ynamide 5-[2-(6-fluoro-1H-indol-3-yl)ethyl]-4-N,4-N-dimethylpyrimidine-2,4-diamine 2-[2,6-difluoro-4-(trifluoromethyl)phenyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one 3-[(4E,5Z)-4-ethylidene-3-methyl-6-methylidenehepta-1,5-dien-2-yl]-2H-chromene 2-[1-(4-chlorophenyl)-3-hydroxycyclohexyl]acetic acid 6-bromo-4,5-dimethylpyridine-3-carboxylic acid;ethane 3-(2-azidophenyl)sulfanylaniline 2-(4-chlorophenyl)-7-methylsulfanyl-5,6,8,9-tetrahydropyrido[2,3-d]azepine 1-(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)-N-propan-2-ylmethanesulfonamide 2-(5,6,7,8-tetrahydronaphthalene-1-carbonylamino)spiro[1H-indole-3,4'-piperidine]-5-carboxylic acid N-[(6-methoxy-2,3-dihydroinden-1-ylidene)amino]-7H-purin-6-amine 5-chloro-4-[1-[3-(cyclopropylmethoxy)-5-fluorophenyl]cyclopentanecarbonyl]pyridazine-3-carboxylic acid 3-(7,11,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),9,11-trien-10-yloxymethyl)benzonitrile 3-ethyl-N,4-dihydroxy-5-methoxybenzamide 4-[(2S)-1-azidoazetidine-2-carbonyl]-3,5-dichlorobenzonitrile 2-(cyclopropylmethylamino)-N-[4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl(pyridin-3-yl)methylidene]ethanimidamide 4-[3-(2-chlorophenyl)pyridin-4-yl]-6-propan-2-yloxypyrimidine 1-[2-(5-azido-1,3-benzodioxol-4-yl)ethyl]piperazine N-(2,6-difluorophenyl)-1-[4-[3-(dimethylamino)propoxy]benzoyl]piperidine-4-carboxamide 2-[4,6-bis(3,5-dimethylpyrazol-1-yl)pyridin-2-yl]-8H-[1]benzofuro[2,3-b]pyridin-8-ide;iridium;trimethyl-[4-(2-methylpropyl)-6-phenylpyridin-3-yl]silane (2R)-2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-N-[(1S)-1-phenylethyl]propanamide N-[(1S,2R)-3-hydroxy-5-oxocyclopentyl]-4-[2-methoxyethyl(methylsulfonyl)amino]benzamide N-(3-chlorophenyl)-2,4-dihydroxybenzenecarbothioamide N'-(3,4-dimethylphenyl)-N-hydroxy-3-pyridin-2-yl-1H-pyrazole-5-carboximidamide 1-[4-(2,3-difluorophenyl)piperidin-1-yl]-5-hydroxy-3-methoxypentan-1-one 1-[(3R)-3-fluoropyrrolidin-1-yl]-2-(7-methoxyspiro[1,2-dihydroquinoline-4,4'-piperidine]-2-yl)ethanone 4-[7-(diethylamino)-3-methoxyquinolin-2-yl]benzene-1,2-diamine 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-1H-pyridine-2-thione 4-[2-chloro-5-(3,6-dihydro-2H-pyran-4-yl)pyridin-3-yl]morpholine 2-[6-(dimethylamino)pyridin-3-yl]-N-[5-ethoxy-4-fluoro-2-(2,2,2-trifluoroacetyl)phenyl]-N,5-dimethylpyrazole-3-carboxamide 1-(6-methylpyridin-3-yl)-N-[2-(oxan-4-yl)-2,2-dithiophen-2-ylethyl]pyrazole-3-carboxamide ethane;6-[1-(4-propylpiperazine-1-carbonyl)pyrazol-3-yl]pyridine-2-carbonitrile 3-ethenyl-N-[[4-(fluoromethoxy)phenyl]methyl]pyridine-2-carboxamide 3-[2-(4,5-dimethylimidazol-1-yl)phenyl]-4H-1,2,4-oxadiazol-5-one 4-chloro-2,6-dimethoxy-N-(3-methylbut-1-en-2-yl)aniline;ethane 5-bromo-2-(3,3-difluoro-2H-pyridin-6-yl)-1,3-thiazole;methane 2-hydroxy-5,6-dimethoxy-3-[(4-nitrophenyl)methyl]-1H-indole 4-[3,3-dimethylbutanoyl(2-phenylethyl)amino]-N-hydroxy-2-phenylsulfanylbenzamide 5-methyl-8-(2,4,6-trifluorophenyl)-3H-imidazo[1,5-a]pyrazine 3-(1H-imidazol-2-yl)-2,4-di(propan-2-yloxy)pyridine 3-(5,6-dimethyl-[1,2]oxazolo[4,5-d]pyrimidin-7-yl)oxybenzonitrile [2-(3,5-difluoro-4-methylphenyl)-2-(6H-pyrido[1,2-b]pyridazin-7-ylidene)acetyl]azanium N-[4,6-bis(2-methoxyphenyl)pyrimidin-2-yl]-2-phenylacetamide 5-[1-[5-cyclopropyl-4-(2,3-difluorophenyl)pyridine-3-carbonyl]piperidin-4-yl]-2-ethoxybenzonitrile ethane;1-[5-(2-fluoro-4-methylphenoxy)pyridin-3-yl]pyrrolidine-3,4-diol 1-(azidomethyl)-2,3-dibromo-4-propan-2-yloxybenzene N-benzyl-5-(4,4-dimethylcyclohexen-1-yl)-2-ethenyl-N'-ethyl-4-methoxybenzenecarboximidamide 3-[2-oxopropyl(pyridin-2-yl)amino]butanoic acid (2S,3R)-1-(1,5-dimethylpyrazole-4-carbonyl)-N-[6-(trifluoromethoxy)-1,3-benzothiazol-2-yl]piperidine-3-carboxamide 2,3-bis(cyclohexyloxycarbonyl)benzoic acid N-methylsulfonyl-2,3-dihydro-1H-indole-5-carboxamide 6-(2-azidopropan-2-yloxy)-7-methoxyquinoline 3-(4-methoxyanilino)propyl-(2,4,6-tribromophenyl)azanide (3R)-3-N-cyclopropyl-1-methyl-6-oxo-4,5-dihydropyridazine-3,7-dicarboxamide 4-(1,3-benzodioxol-5-yl)-N-methoxy-N,2-dimethylbutanamide;hydrochloride 2-[4-(dipropylamino)phenyl]-1,3-thiazole-5-carboxylic acid;ethane 2-(dimethylamino)ethanol;ethane;3-[2-fluoro-4-hydroxy-3-(trifluoromethyl)phenyl]propanamide N-[2-(3,5-dimethylphenoxy)propanoyl]carbamate 1-[5-(2,3-dihydro-1H-inden-4-yl)-2-methylpyridin-4-yl]ethanone 2-[5-(2,6-dimethylphenyl)pentyl]-1H-imidazole 4-[(3R)-1-[2-(diethylamino)acetyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one 1-[(3R)-2,5-dioxopyrrolidin-3-yl]-7-fluoroindazole-4-carboxylic acid N'-[1-[2-(4-chlorophenyl)ethylamino]ethenyl]-N,N-dimethylpropane-1,3-diamine (4S)-2,5-diphenyl-8,9-dihydropyrazolo[3,4-h]quinazoline-4-carboxylic acid 6-chloro-3-[(2,4-difluorophenyl)methyl]-1,3-benzothiazol-2-one 2-[2-(3,5-dimethylphenyl)ethynyl]-4-ethenoxybenzoic acid 2-[4-(3,4-dihydropyridin-2-yl)phenyl]naphthalene (2S)-N-[(2R)-1-[(4,5-dimethylfuran-3-carbonyl)amino]propan-2-yl]pyrrolidine-2-carboxamide 2-(4,7-dioxobenzo[g][1,3]benzothiazol-2-yl)-N-(furan-2-ylmethyl)-4-methoxybenzenesulfonamide 1-amino-3-[(4,5-dimethyl-6H-phenanthridine-8-carbonyl)amino]thiourea 3-chloro-N-[5-[1-(4-methylphenyl)sulfonylpyrrolo[2,3-b]pyridin-4-yl]-6-(trifluoromethoxy)pyridin-3-yl]benzamide 2-[5-ethylsulfonyl-6-[7-methoxy-2,3-dioxo-1-(trifluoromethyl)pyrrolo[2,3-c]pyridin-4-yl]pyridin-2-yl]-N-methylacetamide N-[3,5-dichloro-4-(1H-pyrrole-2-carbonyl)phenyl]-7-azaspiro[3.5]nonane-7-carboxamide (4S)-2,3-dimethyl-1-[4-[4-[4-(4-phenylpiperidine-1-carbonyl)phenoxy]butoxy]benzoyl]azetidine-3-carboxylic acid 3-(2,3,4a,5-tetrahydro-1H-pyrido[4,3-b]indol-7a-ylamino)propanal 4-[[4-(trifluoromethoxy)phenyl]sulfonylamino]piperidine-1-carboxamide 6-hydroxy-5-[(2R)-2-phenyl-1H-indol-3-yl]cyclohexa-2,4-diene-1-carboxylic acid 2-[(5Z)-5-[(3,4-dimethylphenyl)methylidene]-1-methyl-6-oxopiperidin-3-yl]acetic acid 4-[5,6-bis(ethenyl)pyridin-3-yl]phenol 2-[6,8-dibromo-4-ethyl-3-(hydroxymethyl)imidazo[1,5-a]quinoxalin-1-yl]acetaldehyde 6-[(2,4-dihydroxyphenyl)methyl]-3-methyl-5-propan-2-ylidenecyclohexa-1,3-diene-1-sulfonic acid 3-benzylsulfanyl-N'-hydroxypyrazine-2-carboximidamide 3-azido-N-[3-(2H-tetrazol-5-yl)phenyl]pyridine-2-carboxamide 4-[(3R)-3-aminopyrrolidin-1-yl]-6-cyanoquinoline-3-carboxylic acid 5-bromo-2,6-difluoro-1-benzothiophene 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-indol-3-yl)ethyl]propanamide 6-chloro-4H-1,3-benzoxazine;ethane (3S)-3-[[5,6-bis(4-chlorophenyl)pyrazine-2-carbonyl]amino]-4-[[2,6-difluoro-4-(trifluoromethoxy)benzoyl]amino]butanoic acid N-(8,8a-dihydroquinolin-3-yl)-2,6-diphenyl-1,4-dihydropyrido[2,3-d]pyrimidin-7-amine 1-benzyl-2-cyclopropylidene-4-(trifluoromethyl)pyrimidine 1-[3,4-bis(4-methylphenyl)-2H-naphthalen-2-id-1-ylidene]guanidine;[cyclopenta-1,3-dien-1-yl(methyl)silylidene]zirconium(2+) 6-(3,4,5-trimethoxyphenyl)pyrrolo[3,4-c]pyrrole 1-(2-methylpentan-3-ylamino)-3-[(4-phenoxyphenyl)methyl]thiourea (7S)-N-[2-fluoro-3-methoxy-4-(tetrazol-1-yl)phenyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine-7-carboxamide 5-azidosulfanyl-2,3-dimethoxyaniline 2-[3-(azepan-1-ylmethyl)phenyl]-4-cyclopropyl-5H-1,3-thiazole 1-[(3R,6S)-3-ethenyl-6-hydroxycyclohexa-2,4-dien-1-ylidene]propan-2-one;iron 5-chloro-3,7-dimethyl-2,4-dihydro-1H-pyrrolo[1,2-a]pyrazine;N-(3,4-dihydroquinolin-6-yl)formamide 3-(4,5-dimethyl-1H-imidazole-2-carbonyl)benzonitrile 4-amino-2-(5-methylcyclohepta-1,3,6-trien-1-yl)pyrimidine-5-carbonitrile N'-[2,5-dimethyl-4-(methylideneamino)phenyl]ethanimidamide 6-bromo-5-fluoro-N-[(2S)-3-hydroxy-1-phenylbutan-2-yl]-8-oxo-2,7-naphthyridine-4-carboxamide (2Z)-2-[5,6-diamino-4-[1-[6-amino-5-(4-chlorophenyl)pyrazine-2-carbonyl]azetidin-3-yl]oxypyridin-2-yl]-N-methylidenebutanamide 3-(4,5-dichloro-2-nitrophenyl)propanamide (2S)-1,1,1-trifluoro-N'-[6-(2H-indazol-3-ylmethoxy)naphthalene-2-carbonyl]methanesulfonohydrazide N-[2-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]cyclohexa-1,3-diene-1-carboxamide (1R,3R)-N-[4-[2-fluoro-5-methyl-6-[(2-methyl-3,4-dihydro-2H-quinolin-1-yl)sulfonyl]cyclohexa-1,3-dien-1-yl]phenyl]-2,2-difluorocyclopropane-1-carboxamide N'-hydroxy-5,7-dimethoxy-6-(2-pyrrolidin-1-ylethoxy)naphthalene-2-carboximidamide 2-(2-hydroxyphenyl)-3,4,5,6,7,8-hexahydroquinazoline-6-carboxylic acid 2-chloro-6-methoxy-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)benzoic acid N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-5-pyridin-3-ylfuran-2-carboxamide 4-amino-N-(3,5-dichlorophenyl)sulfonylpyridine-2-carboxamide;3-methylbut-1-ene 7-[5,6-dimethyl-2-(4-pyrrolidin-1-ylphenyl)sulfanylpyrimidin-4-yl]oxyisoquinoline (4R)-1-(4,6-dimethylpyrimidin-2-yl)-3-methyl-4-thiophen-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one [5-[(2-methylpropan-2-yl)oxycarbonyl]-1H-indazol-6-yl]boronic acid 1-azido-3,5-bis(9H-fluoren-1-yl)-1-methoxyurea 1-[3-cyclohexyl-2-[(dimethylamino)methyl]quinolin-8-yl]ethanone 3-cyclobutyloxy-N'-hydroxy-5,6-dimethylpyridazine-4-carboximidamide (3R)-1-(2-amino-4,5,6,7-tetrahydrobenzotriazol-5-yl)-N'-[(2S)-1-hydroxypropan-2-yl]oxy-N-phenylmethanediamine 2-azido-5,5,6-trimethyl-3-(4-nitrophenyl)-1H-indole 6,8-dichloro-N'-hydroxyisoquinoline-3-carboximidamide 7-[4,6-bis(trichloromethyl)pyrimidin-2-yl]-3-iodo-1-pentan-3-ylquinazoline-2,4-dione N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]cyclohexanecarboxamide 4-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]cyclohexan-1-one (4-aminopiperidin-1-yl)-[2-methoxy-5-[3-morpholin-4-yl-5-(trifluoromethyl)anilino]phenyl]methanone (6R)-N,6-dimethyl-1,2,3,4,5,8,9-heptahydrocarbazole-1-carboxamide 4-amino-3,5,6-trichlorobenzene-1,2-disulfonic acid 3-(3,4-dichlorophenyl)hexanoic acid 3-azido-5-bromo-1-ethylindole 1-(2,3-dihydro-1H-indene-5-carbonyl)pyrrolidine-2,5-dione (E)-3-[1,4-dimethyl-2-(propan-2-ylideneamino)cyclohexa-2,4-dien-1-yl]-N-[2-[2-(trifluoromethoxy)phenyl]ethyl]but-2-enamide 4-[2,6-dibromo-N-(2-hydroxyethyl)anilino]phenol 3-N,2-dimethyl-4-N-phenylpyrimidine-2,4,6-triamine 1-azidooxy-3-phenylbenzene 4-[3,5-bis(4-methoxyphenyl)-2-propylpyrrol-1-yl]benzenesulfonamide 2-(9,10-dimethoxy-3-propanoylanthracen-1-yl)acetic acid 4-N-ethyl-5-methanimidoylpyrimidine-2,4-diamine;1-(2-fluoro-6-formamidophenyl)piperidine-3-carboxylic acid N-[2,3-difluoro-4-(8-methoxyquinolin-7-yl)phenyl]-2-hydroxypropane-1-sulfonamide 3-cyclohexyl-N-(1,4-dimethyl-2H-benzo[h]quinolin-7-yl)sulfanylpropanamide 2-(3,4-dichlorophenyl)ethylcarbamothioylazanide 7-fluoro-6-methoxy-2,4a-dihydrodibenzofuran 5-benzyl-2-(2-morpholin-4-ylethoxy)benzoic acid 3-(1,2,4-triazol-1-yl)cyclohexan-1-amine 3-[(1R)-6,7-dimethoxy-2-[(2S)-oxan-2-yl]-1,4-dihydroisoquinoline-1-carbonyl]cyclopentane-1-carboxylic acid (5S,6R)-1-(2,3-difluorophenyl)-5-methyl-4-sulfanylidene-6-[(pyridine-3-carbonylamino)methyl]piperidine-3-carboxylic acid 4-bromo-2-[(6,7-dichloro-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl)amino]benzoic acid 4-[2,2,3-trifluoro-1-hydroxy-2-(methylamino)ethyl]phenol 7-chloro-5-[2-(methylamino)ethyl]pyrrolo[1,2-a]quinoxalin-4-one N-[4-(5-methyl-1,3-benzoxazol-2-yl)cyclohexyl]carbamate 2-[(2E,5S)-2-[(Z)-1-naphthalen-1-ylethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid ethane;5-(2-fluoro-4-methylphenoxy)-6-[1-(4-fluorophenyl)propan-2-yl]pyridine-3-carboxylic acid 3-[(4-nitrophenyl)methoxycarbonyl-nonanoylamino]butanoic acid 2-azidooxy-5,6,7-trimethyl-1H-indole 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;3-ethyl-8-(6-methoxypyridin-3-yl)-2-phenylisoquinolin-1-one (5S)-3-cyclopropyl-2,4,5,6-tetrahydroxy-N-[[1-[(1R)-1-phenylethyl]piperidin-4-yl]methyl]heptanamide 4-(1,3-benzothiazol-2-yl)-5-imino-1-phenylimidazolidin-2-one 2-(4-bromobutyl)-7-methoxy-3,4-dihydro-1H-isoquinoline 2-[3,4-bis(propylsulfanylmethyl)phenyl]pyridine 3-[5-cyclobutyl-2-(4-ethenylphenyl)-6-methylidenepyrimidin-1-yl]propanoic acid 2-(3,4-diethoxyphenyl)-4-(4-methylsulfonylphenyl)-1H-imidazole 3-[[2,6-difluoro-4-(triazol-1-yl)phenyl]methoxy]-5-pyrimidin-5-ylpyridin-2-amine N-[(E)-1-amino-3-(dimethylamino)prop-2-enylidene]-3-[4-oxo-5-(trifluoromethyl)quinazolin-3-yl]benzamide;ethane 2,3-dimethylbut-2-ene;ethane;6-ethylidene-1-ethylcyclohexa-1,4-diene;formaldehyde;N-[2-methoxy-5-(oxan-4-yl)pyridin-3-yl]acetamide 1-methyl-2-[(2E)-6-nitrohexa-2,4-dien-3-yl]naphthalene 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethanone 4-amino-1-(difluoromethoxy)pyridin-2-one [4-[3-methoxy-4-(6-methylsulfonylpyridin-2-yl)oxyphenyl]pyrrolidin-1-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone 1-[5-(4-chlorophenyl)-2-propylthiophen-3-yl]ethenol N-(4,5-dimethyl-2-phenyldiazenylphenyl)-1H-indole-3-carboxamide 5-cyclopropyl-4-[(2,6-difluorophenyl)methoxy]-N-methylidenepyridine-3-carboxamide 7-[4-(dimethylamino)phenyl]-5,5-difluoro-3H-1,4-benzothiazepine-2-thione (5S)-3-benzylsulfanyl-7,8-dihydro-2H-[1,4]dioxino[2,3-e]indole 3-[2-(4-methylpiperazin-1-yl)-6,7,8,9-tetrahydropyrimido[5,4-b]indolizin-4-yl]-5-propan-2-yloxy-1H-quinolin-2-one 2-(N-(5-nitro-1,3-thiazol-2-yl)-4-propylanilino)decanoic acid 3-bromo-4-[(E)-2,5-dimethylhex-1-enoxy]phenol 6-(5,5-dimethyl-4,7-dihydrothieno[2,3-c]pyridin-6-yl)-N-[[6-(3-hydroxy-3,4-dihydropyridin-5-yl)pyridine-2-carbonyl]amino]pyridazine-3-carboxamide 4-[2-[(4,6-dimethylpyrimidin-5-yl)sulfonylamino]ethoxy]benzoic acid 2-(2-bromophenyl)imino-5-[(1,3-dimethylindol-4-yl)methylidene]-1,3-thiazolidin-4-one N-[(2S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl]quinoline-8-carboxamide 1-[2-(2,6-dichlorophenyl)ethyl]-N-(1,3-thiazol-4-ylmethylideneamino)indole-5-carboxamide (E)-3-[4,7-dimethyl-5-(2-phenylethynyl)-1H-indol-3-yl]prop-2-enoic acid N-[4-(dimethylamino)phenyl]-2,4-dihydroxy-N-methylbenzenesulfonamide 2-(3,4-dichloroanilino)-6-(7-methylimidazo[1,5-a]pyridin-3-yl)-8H-pyrido[2,3-d]pyrimidin-7-one 6-(7,8-dihydronaphthalen-2-yl)cyclohexa-1,5-dien-3-yne N-[(2S)-2-aminopropoxy]-2-methyl-4,5,6,7-tetrahydroindazole-3-carboxamide 4-[3,6-dimethyl-2-(triazol-1-yl)phenyl]butanal 2-chloro-N-[1-(3,4-dimethoxyphenyl)ethyl]benzenesulfonamide (3-azido-1,4-dioxan-2-yl)-phenylmethanone [2-(cyclopropylmethylamino)phenyl]-[4-hydroxy-3-[6-(trifluoromethyl)pyridin-3-yl]piperazin-1-yl]methanone 1-(2-methoxyethyl)-2-oxoindole-3-carboxylic acid (2R,3S)-5-[4-chloro-N-(cyanomethyl)anilino]-2-(hydroxymethyl)-1-methoxycarbonylpyrrolidine-3-carboxylic acid (2R,5R)-1-tert-butyl-5-methylspiro[3H-indole-2,4'-piperidine] 6-(2,3-dihydropyridin-5-yl)-2-(4-fluorophenyl)-3-(2-propoxyethylamino)quinazolin-4-one (4aS,9bS)-5-methyl-7-(3-nitrophenyl)-1,2,9b-trihydroazirino[2,1-a]isoindole N-[3-(2,4-dihydroxyphenyl)-5-methyl-1H-pyrazol-4-yl]cyclopentanecarboxamide 3-(N-phenacylanilino)propanenitrile (4R)-3,8-dimethyl-1-(6-pyrrolidin-1-ylpyridazin-3-yl)-4-pyridin-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 2-(4,6-diphenylpyridin-2-yl)-1H-imidazole;iridium(3+) 2,7-dimethoxy-3-methylquinoline 1-[4-(2,3-dihydro-1H-inden-5-yloxy)phenyl]ethanone 2-(3,5-dimethylpyridin-4-yl)oxy-7-(1-ethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidine 2-bromo-5-[1-(trifluoromethyl)cyclohexa-2,4-dien-1-yl]benzonitrile 1-[2,6-dimethyl-4-(trifluoromethoxy)phenyl]-3-[2-[(3R)-3-ethoxypyrrolidin-1-yl]phenyl]urea;hydrochloride 2-[3-bromopropyl(2,2-diethoxyethyl)amino]benzoic acid 2-(3,4-dihydro-1H-isoquinolin-2-yl)-6-oxo-N-[3-(propan-2-ylamino)phenyl]-1H-pyrimidine-4-carboxamide N-[[4-bromo-5-[2-(cyclohexylamino)ethoxy]pyridin-2-yl]methyl]-N',N'-diethylpropane-1,3-diamine 2-[1-[(4-chlorophenyl)methyl]imidazol-2-yl]ethanamine;dihydrochloride 6-(diethylamino)-3-hexylsulfanyl-4H-1,2,4-triazin-5-one (2Z)-3-(4,5-dichlorothiophen-2-yl)-N-hydroxy-2-[(2E,5Z)-octa-2,5-dienylidene]-1H-pyrido[2,1-b]quinazoline-9-carboxamide 4-chloro-N-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]benzamide 3-[(5S,7R)-2-hydroxy-5-methyl-7-phenyl-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazole-4-carbonyl]-2-methoxybenzonitrile 6-[2,4-bis(phenylmethoxy)phenoxy]hexylphosphonic acid 1-[6-(4-hydroxyphenyl)benzotriazol-2-yl]ethanone 5-phenylmethoxypyridine-2,3-dicarboxylic acid 1-[(3,5-dimethylphenyl)sulfonylamino]cyclohexane-1-carboxylic acid 7-hydroxy-5,6-dimethoxy-2H-chromene-3-carboxamide 5-[3-(4-hydroxy-2,6-dioxocyclohexyl)-1-methoxybutan-2-yl]sulfanyl-4-methylpyridine-3-carboxamide 1-[4-(2,3-dihydropyridin-2-yl)phenyl]-N-ethoxypentan-1-imine 2-(4,5-dichlorothiophen-3-yl)oxyacetic acid 2-methyl-1'-phenylspiro[1H-indole-3,4'-piperidine] N-[5-(furan-2-ylmethylamino)-3-[4-(4-hydroxypiperidine-1-carbonyl)phenyl]imino-5,6-dioxocyclohexa-1,4-dien-1-yl]pyridine-3-carboxamide N-(6-chloro-2,4-dimethoxypyrimidin-5-yl)-5,7-dimethylpyrrolo[2,3-d]pyrimidin-4-amine 1-[4-(azidomethyl)-2,3,5-tribromophenyl]-N-[[4-(trifluoromethoxy)phenyl]methyl]piperidin-4-amine N-[[3,5-bis(trifluoromethyl)phenyl]methyl]methanimine 3-hydroxy-2,5,7-trimethyl-6-[(E)-prop-1-enyl]pyrazolo[4,3-b]pyridine (2R,3S)-4-[[1,7-dimethyl-6-(2-oxopropylamino)benzimidazole-5-carbonyl]amino]-2-hydroxy-3-methoxybutanoic acid 1,2-dimethylbenzimidazole;4,4'-spirobi[fluorene]-2',3',5'-trione 3-[2-(1H-indol-3-yl)ethenyl]benzenesulfonamide N-(2,6-difluorophenyl)-3-(4-hydroxy-5-methylpyrimidin-2-yl)sulfanyl-N-(2-hydroxyethyl)propanamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-6-[2-(4-ethylcyclohexyl)ethynyl]-1-fluoronaphthalene 4-[3-(1,2-diphenylethyl)imidazolidin-1-yl]benzaldehyde 1-[4-[2-(7,8-dichloroquinolin-5-yl)oxyethoxy]piperidine-1-carbonyl]pyrrolidine-3-carboxylic acid 3-(3-methylphenyl)-2H-pyrazolo[3,4-b]pyridine N-(2,4,6-trimethylphenyl)-3H-benzimidazole-5-carboxamide 3-butoxy-N'-hydroxypyridine-2-carboximidamide (E)-3-[2,5-bis(trifluoromethyl)phenyl]-N-[4-oxo-2-sulfanylidene-1-[[4-(trifluoromethoxy)phenyl]methyl]pyrimidin-6-yl]prop-2-enamide N-(4-carbamimidoylphenyl)-1-[6,7-dimethoxy-2-[3-methyl-5-(trifluoromethyl)anilino]quinoline-3-carbonyl]pyrrolidine-2-carboxamide;formic acid 4-[2-(4-methoxycarbonylphenyl)ethyl]piperazine-1,3-dicarboxylate 1-[[2-[(3S)-4-(cyclopropylmethoxy)piperidin-3-yl]oxyphenyl]methyl]pyrrolidine 6-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)-N-[3-(trifluoromethoxy)phenyl]pyridine-2-carboxamide 2-azido-5-(3,4-dichlorophenyl)-1H-pyrrole 3-[(4-chlorophenyl)methoxy]pyridine 1-butanoyloxynaphthalene-2,3,6-tricarboxylic acid [3-(2,6-dimethoxyphenyl)-3-iminopropyl]carbamic acid 2-(5-chloro-1H-indol-3-yl)ethanimine;1-[(Z)-2-[(Z,2E)-2-hydroxyiminopent-3-enoxy]but-2-enyl]-4,6-dimethylpyridin-2-one 3-(2,4-dichlorophenyl)sulfanyl-2-(difluoromethylsulfonylamino)benzamide 2-chloro-4-[2-(dimethylamino)ethyl]aniline 6-(3,5-difluoro-4-hydroxyphenyl)-4-[ethyl-(1-methylpiperidin-4-yl)amino]quinoline-3-carbonitrile 2-[N-(1-carboxyethyl)-4-chloroanilino]propanoic acid 3-[2-(1-methylpyrazol-4-yl)ethyl]pyridine N-[4-[2-(4,5-difluorocyclohexa-1,3-dien-1-yl)ethynyl]phenyl]benzamide N-(3,5-difluorophenyl)sulfonyl-2-[1-(6-methylpyridin-2-yl)pyrrolo[2,3-b]pyridin-2-yl]acetamide 2-[4,5-dichloro-3-(4-phenylmethoxyanilino)isoindol-1-ylidene]propanedinitrile 3-(4-cyclohexyloxyphenyl)pentan-2-one 2-amino-3,5-bis(benzenesulfonyl)benzoic acid 2-amino-4,4-dimethoxy-6-[4-(4-pentanoylphenoxy)phenyl]-3-azabicyclo[3.1.0]hex-2-ene-1,5-dicarbonitrile 6-(4-bromophenyl)-8-methoxyquinazoline (2R,5S)-5-[[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]oxolane-2,3-diamine 3-amino-5,6-dimethylthieno[2,3-b]pyridine-2-carboxamide;4,4-difluorocyclohexane-1,3-diol 1-[4-methoxy-3-(4-oxo-5,6,7,8-tetrahydro-3H-quinazolin-2-yl)phenyl]pyrrole-2,5-dione (2R)-N'-methyl-1-methylideneanthracene-2-carbohydrazide 4-(1,3-dimethylpyrazol-4-yl)-2-propan-2-yl-1H-pyrimidin-6-one 6-(3,4-difluorophenyl)-N-[(2-propylpyridin-4-yl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-3-amine 2-(azepan-1-yl)-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-3-one (6E)-3-[(2S,4R,5S)-4,5-bis(phenylmethoxy)oxan-2-yl]-1,5-dihydroimidazo[4,5-g]quinoxaline-2,8-dione 7-(1,3-thiazol-2-yl)-5H-pyrrolo[3,4-b]pyridin-6-one 3-(4-bromophenyl)-7-methyl-5,6-dihydrobenzimidazolo[1,2-a]quinazoline N-[(Z)-1H-indol-2-ylmethylideneamino]-4-nitrobenzamide 3-[[2,5-bis(4-fluorophenyl)pyrrolidine-1-carbonyl]amino]indole-1-carboxylic acid 2-[4,5-bis(4-methoxyphenyl)-1H-imidazol-3-ium-3-yl]ethanamine 3-butoxy-2-[(E)-2-(4-phenylphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one 1-(cyclohexylmethoxy)-4-phenylbenzene 1-phenyl-6-(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)cyclohexa-2,4-diene-1-carbonitrile 2-fluoro-1,3,5-trimethyl-4-[[2-methyl-6-(trifluoromethyl)pyridin-4-yl]methoxy]-2H-pyridine 2-(2,4-difluorophenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide (1R)-2,2-difluoro-N-[4-(3-morpholin-4-ylpropoxy)phenyl]cyclohexane-1-carboxamide 2,3-diamino-N'-[(5S)-7-[3-(dimethylamino)propoxy]-6-methoxy-1,2,4,5-tetrahydro-3-benzazepin-5-yl]benzenecarboximidamide N-methyl-3-(2,4,6-trimethylphenoxy)propanamide 2-[4-(trifluoromethoxy)phenyl]-1,2,3,4-tetrahydroquinoline N-(4,6-dimethylpyrimidin-2-yl)-5-[2-ethoxy-3-hydroxy-3-(1-propanoyltetrazol-5-yl)prop-2-enyl]pyridine-2-carboxamide 4-azidooxy-1-chloronaphthalene 3,5-diamino-6-chloro-N'-methylpyridine-2-carboximidamide (2S,3R)-4-[5-(2,6-dimethoxyphenyl)imidazol-1-yl]-N-ethylbutane-2-sulfonamide;hydrochloride 2-(1,3-benzodioxol-5-ylmethoxycarbonyl)benzoate N-[2-hydroxy-4-(trifluoromethyl)phenyl]-N',4,5-trimethoxycyclohexa-1,3-diene-1-carboximidamide 2,4-dibutyl-1-hexylbenzene ethane;methanol;4-[(3E,5Z)-2-methylhepta-1,3,5-trien-4-yl]sulfonylcyclohepta-1,3,6-triene 2-(3,4-dichlorophenyl)-1-[4-[2-hydroxyethyl(methyl)amino]piperidin-1-yl]-5-methylpentan-1-one 2-[4-(3,5-dimethoxyphenyl)piperazin-1-yl]acetamide 2-benzyl-4,5-dimethoxyphenol 1-bromo-2,3-dimethyl-4-(3-nitrophenyl)benzene 2-(4,5-dimethylpyrimidin-2-yl)propanedioic acid (2S)-1-cyclopropylsulfonyl-4-methylsulfanyl-N-[3-(1,1,2,2,2-pentafluoroethoxy)phenyl]pyrrolidine-2-carboxamide 3-[(2,4-dimethylphenyl)carbamoylamino]benzamide 4-[5-[2-(diethylamino)ethyl]-1,3-thiazol-2-yl]phenol 2,3-dichloro-N-diazobenzenesulfonamide N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-3-hydroxypyridine-2-carboxamide N-(3,4-dichlorophenyl)-1H-[1]benzofuro[3,2-c]pyrazole-7-carboxamide 2-azidooxy-5-[3-chloro-4-(trifluoromethyl)phenyl]pyridine [6-(4-hydroxyphenyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl]methanol 3-[3,4-dihydroxy-2-(3-methylbut-2-enylidene)oxan-4-yl]benzoic acid 4-[2,5-difluoro-6-(methoxymethyl)phenyl]-N-(1,2-thiazol-3-ylamino)sulfanylcyclohexane-1-carboxamide 1-[6-(2,5-dimethylphenyl)-4H-pyran-3-yl]-N'-hydroxypyrrolidine-2-carboximidamide 1-[6-methoxy-2-(4-phenylmethoxyphenoxy)pyridin-3-yl]propan-1-one 1-[(3,5-difluorophenyl)methyl]indole-4-carboxylic acid 2-(4,5-dihydro-1H-imidazol-2-yl)-3,6-bis(pyridin-2-ylmethylideneamino)phenol 2-[4-amino-3-methyl-6-(propanoylamino)pyridin-2-yl]oxyacetic acid N-(5,6-difluoro-3-methylpyridin-2-yl)piperidine-4-sulfonamide 2-methyl-5-[(1S)-3,3,4-trimethoxy-1H-2-benzofuran-1-yl]tetrazole 2-azido-5,6-dihydropyrano[2,3-b]indole 1-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridin-5-yl)-5-(trifluoromethoxy)indole-7-carbonitrile 1-[2,6-di(propan-2-yl)phenyl]-3-[5-methoxy-2-(4-methoxyanilino)pyrimidin-4-yl]urea 1-chloro-2,3-dimethylbenzene;N'-(4-cyanophenyl)-N-[2-methoxy-5-[[(Z)-prop-1-enyl]sulfanylamino]pentyl]butanediamide 2,6-bis[(1R)-1-hydroxypropyl]benzoate;manganese(3+);hydrate 2-[(4-methoxy-6,7-dihydrothieno[3,2-c]pyridine-5-carbonyl)amino]acetic acid N-methyl-4-[2,3,4-tris(sulfanylidene)cyclobutyl]benzenecarbothioamide 6-chloro-N,2-dimethyl-5-(pyridin-3-ylamino)pyridazine-4-carbothioamide (3R,4R)-1-ethyl-4-[[3-fluoro-5-(trifluoromethoxy)phenyl]methylamino]pyrrolidin-3-ol (5Z)-3-[4-(2,6-dichlorophenyl)-1,3-thiazol-2-yl]-5-[[3-(trifluoromethoxy)phenyl]methylidene]-1,3-oxazolidine-2,4-dione 4-[(2,3,4,5-tetramethoxycyclopenta-1,4-dien-1-yl)methoxy]aniline N-[2-fluoro-5-(2,3,4,6-tetramethylphenyl)-1H-indol-7-yl]-3-piperidin-1-ylcyclobutane-1-carboxamide 1-[4-(2,4-dimethylphenyl)piperazin-1-yl]propan-2-ol 5-methyl-2-(2,3,4-trifluorophenyl)pyrimidine N-[2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-3,3,3a,4,5,6,6a-octahydro-1H-cyclopenta[c]pyrrole-2-carboxamide 4-[(E)-3,3-diphenylprop-1-enyl]-N,N'-diethyl-5-methoxypyridine-2-carboximidamide (2R,3S)-N-[2-(5-chlorothiophen-2-yl)ethyl]-1-methyl-2-pyridin-4-ylpiperidine-3-carboxamide [2-chloro-4-(trifluoromethyl)phenyl]-[3,5-diethyl-6-hydroxy-4-(pyridine-4-carbonylamino)cyclohexa-1,5-dien-1-yl]azanium (1S,2R)-1-[(4-chlorophenyl)methyl]-3-isoquinolin-1-yloxy-1-[(2E,4Z)-3-methylhepta-2,4,6-trienoxy]propan-2-amine N-[(4-amino-6-oxo-1H-pyrimidin-2-yl)methyl]-1,3-thiazole-5-carboxamide N-(4-methylphenyl)benzenesulfinamide 1-N,1-N-dimethyl-2-N-[4-[4-(trifluoromethoxy)anilino]phenyl]cycloheptane-1,2-dicarboxamide 1,3-bis[(2E)-penta-2,4-dienoxy]benzene;ethane 5-[2-azidooxy-3,4-bis(phenylmethoxy)phenyl]pyrimidine (6-methoxypyridin-2-yl)-[5-[2-(trifluoromethyl)pyridin-3-yl]pyridin-2-yl]methanone 5-(4,7-dioxabicyclo[3.2.0]hepta-1(6),8-dien-2-ylmethyl)-9-oxopyrido[4,3-b]indole-7-carboxylic acid (6-methoxy-4,5,7,8-tetrahydropyrazolo[1,5-d][1,4]diazepin-2-yl)-(3-phenyl-2H-[1,2,4]triazolo[4,3-a]pyridin-3-yl)methanone 3-[(3S)-1-cyclobutylpiperidine-3-carbonyl]benzonitrile 3-hydroxy-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carboximidamide 4-[5-(1-hydroxypyridin-1-ium-2-yl)-1,3,4-oxadiazol-2-yl]phenol N-[3-(diethylamino)propyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxamide;hydrochloride (2Z,4E)-N-[5-[[4-chloro-6-(trifluoromethyl)pyrimidin-2-yl]sulfamoyl]pyridin-3-yl]oxy-2-ethenyl-3-(4-fluorophenyl)hexa-2,4-dienamide (5Z)-2-[1-[4-chloro-2,3-bis(prop-1-en-2-yl)phenyl]ethylidenehydrazinylidene]-5-[[1-(4-methoxybutyl)indol-3-yl]methylidene]-1,3-thiazolidin-4-one 1-methyl-3-[1-(5-phenylpent-2-enyl)piperidin-4-yl]-5,6-dihydro-4H-pyrrolo[3,2-c]pyrazole [4-(3-amino-1H-indazole-5-carbonyl)piperazin-2-yl]-thiomorpholin-4-ylmethanone 2-(3-methylthiophen-2-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine (E)-3-[(2S,3R)-4-(2-ethoxyphenoxy)-1-oxo-1-phenylpentan-2-yl]undec-9-enoic acid 3-[1,1,1,2,3,3,4,5,5,6,7,8,8a-decafluoro-4-(2-phenylethenyl)dec-2-enyl]benzonitrile N-methyl-1'-(2-phenylethyl)spiro[6,8-dihydrofuro[3,2-g][1]benzofuran-7,4'-piperidine]-5-amine 1-[5-(1H-indazole-4-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]ethanone (2-aminopyridin-3-yl)-[3-hydroxy-3-[[4-methoxy-5-(1H-pyrazol-4-yl)cyclohexa-2,4-dien-1-yl]iminomethyl]pyrrolidin-1-yl]methanone N-(3,4-difluorophenyl)-8-methyl-5-oxo-2-pyridin-4-ylimidazo[1,2-a]pyrimidine-6-carboxamide;ethane 2-(4,6-dimethoxypyrimidin-5-yl)-N-methylsulfonylimidazole-1-carboxamide (1R,3S)-3-[[6-amino-5-[4-(6-phenoxypyridine-2-carbonyl)benzenecarboximidoyl]pyrimidin-4-yl]amino]cyclohexane-1-carboxylic acid (1S,4aR)-6-(benzylamino)-3-phenyl-2,3,4,4a,5,6,7,8,8a-octahydro-1H-naphthalene-1,4-diol (4R)-3-benzyl-4-[2,6-dichloro-4-nitro-N-(2-phenylethyl)anilino]azetidine-1-carboxylic acid (E)-1,2-diamino-3-methyliminoprop-1-en-1-ol;(5R)-7-[[3-fluoro-4-(pyridin-2-ylmethoxy)phenyl]methyl]-5-methyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-one 1-(3,5-dichlorophenyl)-4-oxo-7H-pyrazolo[3,4-b]pyridine-6-carbonitrile 3-azido-2,6-dichloro-5H-imidazo[1,2-b]pyrazole 1-N',3-N'-bis(4-methylphenyl)propanedihydrazide 6-(2-cyclopropyl-4,6-difluorophenyl)-4-N-[1-(3,4-dimethoxyphenyl)pyrazol-3-yl]pyrimidine-2,4-diamine N-[1-(4-phenylphenyl)ethyl]piperidin-3-amine (2Z,4E)-3-[5-(2,6-dimethylphenyl)-7-(4-fluorophenyl)-1H-pyrrolo[2,3-f]indazole-6-carbonyl]hexa-2,4-dienedinitrile 4-amino-2-fluoro-5-[3-(4-hydroxypiperidin-1-yl)propyl]benzoate 2-[(4-oxochromene-3-carbonyl)amino]pentanedioic acid 2-[4-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indazol-1-yl]ethanol ethane;5-(2,4,5-trifluorophenyl)pyrazine-2-carbonitrile 4-[2-[(2S)-4-methyl-2,3-dihydro-1H-inden-2-yl]ethoxy]-2-methylidenepiperidine 3-[(2S,4R)-1-acetyl-6-methoxy-5-oxo-3,4-dihydro-2H-1,4-benzodiazepine-2-carbonyl]pyridine-4-carbonitrile 4-[(8aS)-7-[3-hydroxy-4-(2-phenylethynyl)benzoyl]-1,5,6,8-tetrahydroimidazo[1,5-a]pyrazin-3-yl]benzonitrile 1-[(3-fluorophenyl)methyl]-N-(2H-tetrazol-5-yl)indole-6-carboxamide 3-(9,10-dihydrophenanthren-4-yl)-9-phenylcarbazole 7-(azetidine-1-carbonyl)-3H-quinazolin-4-one (1S,5R)-8,15-dimethoxy-9-phenyl-2-oxa-10,13-diazatricyclo[14.4.0.06,11]icosa-3,6(11),7,12,17,19-hexaen-18-ol 1-phenyl-N-[2,3,6-trifluoro-4-(4-pyridin-4-ylpyrrolo[2,1-f][1,2,4]triazin-7-yl)phenyl]methanesulfonamide [3,5-dichloro-2-hydroxy-4-(trifluoromethyl)phenyl]methylideneazanium 3-azidooxy-4,6-dichlorobenzene-1,2-disulfonic acid N-[2-(4-chlorophenyl)ethyl]-4-[5-[5,6-difluoro-1-(4-fluorophenyl)benzimidazol-2-yl]-1H-pyrrol-3-yl]butan-1-imine N-(1,3-benzodioxol-5-yl)formamide;ethane 6-[(2R,3S)-2,3-dihydroxypyrrolidine-1-carbonyl]isoquinoline-7-carbonitrile 7-(4-bromobutoxy)-3-(1,2,4,5-tetrahydro-3-benzazepin-3-ylmethyl)quinazolin-4-one;hydrochloride 1-(5,8-dihydropyrido[3,4-d]pyrimidin-6-yl)propan-2-one 5-[(2-fluorophenyl)methyl]-N,4-dimethylpyridin-2-amine 3-[4-(2,6-difluorophenyl)piperazine-1-carbonyl]-2H-pyridine-3-carbonitrile N-[(4-aminophenyl)methyl]-2-azido-3,6,7,8-tetrahydrocyclopenta[g]quinazolin-4-amine (NE)-N-[1-[[4-[6-(1,1-difluoroethyl)pyridine-2-carbonyl]phenyl]methoxymethyl]pyrimidin-2-ylidene]nitramide 5-[3-(azidomethyl)cyclohexen-1-yl]-2-methoxypyridine N-benzyl-5-hydroxy-4,6-dimethyl-8-[4-(methylideneamino)phenyl]-3-propan-2-yl-7H-1,8-naphthyridine-2-carboxamide 1-[(Z)-[3,4-bis(ethenyl)-2H-naphthalen-1-ylidene]amino]ethenamine 4-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-N-[4-(hydroxycarbamoyl)cyclohexa-1,3-dien-5-yn-1-yl]-2H-quinoline-1-carboxamide 4-(3-fluorophenyl)-5-nitro-2-[3-(trifluoromethyl)pyrazol-1-yl]pyridine N-(1,3-benzodioxol-5-ylmethyl)-6-bromoquinoline-7-carboxamide 2-azido-1,5-dichlorobenzotriazole 2-methoxyimino-2-(2,3,4,5-tetrachlorophenyl)acetic acid 2-[4-(3,6-dimethylcyclohepta-1,4,6-trien-1-yl)phenyl]ethanimidamide [3-methyl-2-(1H-pyrrol-2-yl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]-[3-(triazol-1-ylmethyl)phenyl]methanone N-[(4S)-4-(2,3-dihydroindole-1-carbonyl)-6-methoxyspiro[2.5]octan-8-yl]pyridine-3-carboxamide 6-amino-3-[(4,5-difluoro-2-sulfophenyl)diazenyl]-7-methylnaphthalene-1-sulfonate 6-[[1,3-benzothiazol-2-yl(methyl)amino]methyl]imidazo[1,2-a]pyridine-3-carboxamide 2-(4,5-dimethyl-N-octyl-2-phenyldiazenylanilino)octanoic acid 4-(1,3-benzothiazol-2-ylmethoxy)cyclohexan-1-amine 4-benzylsulfanyl-3-(2,6-dimethoxyphenyl)-5-ethyl-1H-pyrazole N-[[6-chloro-3-fluoro-2-(2,4,5-trifluorophenyl)phenyl]methyl]pyrrolidine-1-carboxamide 1-[4-(4,4-dimethylcyclohexen-1-yl)phenyl]-2-methylbenzene N-[4-[2-(2,6-dimethylanilino)-1H-indol-3-yl]phenyl]-4-morpholin-4-ylbenzamide 1-[2,4,6-trimethyl-N-(3-morpholin-4-ylpropyl)anilino]propan-2-one N-ethyl-2-[4-[3-(1H-indazol-5-ylamino)quinoxalin-6-yl]pyrazol-1-yl]acetamide 4-methyl-2,3-dihydroindole-1H-1-benzothionine N-(3,5-dimethoxyphenyl)-1,7-naphthyridine-8-carboxamide (1-methylpiperidin-4-yl)methanimine;2,5,7-triphenylpyrrolo[2,3-d]pyrimidine (6S)-2,8-dichloro-6-[(4R)-3,7-dimethylheptyl]-5-fluoro-6H-quinoline N-[(E)-1H-indol-3-ylmethylideneamino]-2-(6-methoxyquinolin-4-yl)acetamide 4-chloro-2,5-dimethoxy-N-[(1S)-2-oxocyclohexyl]benzenesulfonamide 3-(3-fluoro-4-methoxyphenyl)-1,2-diphenylpyrrolo[2,3-b]pyridine 3-[4-(1,2-benzothiazol-5-ylamino)piperidine-1-carbonyl]piperidin-2-one N-azido-4-chloronaphthalen-1-amine 3-[2-methylpropyl(propyl)amino]-4-sulfanylidenecyclobut-2-en-1-one;1-propylnaphthalene 7-(3,6-dihydro-2H-pyran-4-yl)-N-[(1S)-1-(5-fluoro-1H-indol-3-yl)ethyl]quinazolin-2-amine 7-[(2Z)-1,4-diphenylpenta-2,4-dienyl]-9H-fluorene 3-[3-[5-(azetidine-1-carbonyl)pyridin-2-yl]-4,5-dihydrooxepin-6-yl]benzoic acid N-[1-(1,3-benzothiazol-2-yl)ethylideneamino]-4-methoxy-2-methylaniline 3-(4,5-dimethylthiophen-2-yl)sulfonyl-2-oxopropanoic acid N-(3,4-dimethylphenyl)-2-[(6S)-2-ethylsulfanyl-5-oxo-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]acetamide 5-[(Z)-2,3-dihydroinden-1-ylidenemethyl]pyrimidine 2-ethyl-7,8-dimethoxy-3H-cyclopenta[c]chromene 3-[4-chloro-2-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)phenyl]-N'-ethoxypropanimidamide N-(cyclohexylmethyl)-3,4-dihydronaphthalene-1-carboxamide 2-(4-oxopyridin-1-yl)-N-[3-[[6-methyl-5-(1H-pyrazol-4-yl)-1,2-dihydropyrimidin-7-yl]oxy]phenyl]acetamide N-[4-(3,5-dimethylphenyl)pyridin-2-yl]cyclohexanecarboxamide 3,5-dimethyl-1-(2-phenoxyethyl)pyrazole 5-(3,4-dimethoxyphenyl)-3-[1-(7H-purin-2-yl)piperidin-4-yl]triazolo[4,5-d]pyrimidine 2-[[3-[4-(carboxymethylcarbamoyl)phenoxy]benzoyl]amino]acetic acid N-[2,6-dichloro-4-(trifluoromethyl)phenyl]-3-ethynyl-5-fluorobenzenesulfonamide 5-(6-bromopyridin-2-yl)sulfanyl-3H-1,3,4-thiadiazol-2-one 1-butanoyl-N-[2,6-di(propan-2-yl)phenyl]piperidine-4-carboxamide (E)-3-[5-[(2S,4R,6R)-4-methoxy-6-methyloxan-2-yl]furan-2-yl]prop-2-enoic acid 6-[(E)-1-amino-3-methyliminoprop-1-en-2-yl]-N-(5-cyclohexylpyridin-2-yl)-3,4-dihydro-1H-isoquinoline-2-carboxamide 6-tert-butyl-1,3-dimethylimidazo[4,5-c]pyridin-2-one (2Z,3E)-N,4-dimethyl-1-phenylhexa-2,5-dien-3-amine;2-ethylbenzenethiol N-[[3,5-bis(trifluoromethyl)phenyl]carbamoyl]-2-benzylsulfanylacetamide (4aS,8aR)-6-[3-[2-(5-chloropyridin-3-yl)ethynyl]azetidine-1-carbonyl]-4,4a,5,7,8,8a-hexahydropyrido[4,3-b][1,4]oxazin-3-one 6-(cyclopentylamino)pyridazine-3-carboxamide 5-[2-(difluoromethyl)pyridin-4-yl]-3H-indole N-[2-[(2S,3R)-5-amino-2,6-dimethylheptan-4-ylidene]-1-cyclopentylpropyl]-7-fluoro-1-benzothiophene-2-carboxamide [2-fluoro-5-(trifluoromethyl)phenyl]sulfanium 1-[[2,6-di(propan-2-yl)phenyl]iminomethylideneamino]naphthalene-2,7-diol (3S,4R)-1-cyclohexyl-3-methoxycarbonyl-4-[4-[(4-propan-2-ylphenyl)sulfonylamino]butanoylamino]pyrrolidine-2-carboxylic acid 7-chloro-3-hydroxy-2,4-dimethyl-5-nitrochromene-2-carboxylic acid 4-methyl-N-[6-(3-pyrrolidin-1-ylpropoxy)pyridin-2-yl]quinoline-6-carboxamide 1-[4-azidooxy-3,5-bis(trifluoromethyl)phenyl]-2H-azete 1-(3,4-dimethoxyphenyl)sulfonylpiperidine;hydrochloride 1-bromo-2,4-bis(1H-pyrazol-5-yl)piperazine 4-(2,3-dihydro-1H-inden-5-yl)-N-[1-hydroxy-2-methoxy-1-[(4-methoxyphenyl)methylamino]propan-2-yl]benzamide 1-(2-cyclohexa-1,5-dien-1-yloxyethyl)-3-[4-(trifluoromethyl)pyridin-2-yl]urea [1-[(4-aminopyrimidin-2-yl)methyl]piperidin-3-yl]-[4,5-bis(ethenyl)furan-3-yl]methanone;ethane N-[5-(7,8-dihydronaphthalene-1-carbonyl)-4,6-dimethylpyridin-2-yl]-3-[(dimethylamino)methyl]benzamide;ethane N-[6,7-dichloro-2-(trifluoromethyl)quinolin-4-yl]formamide 4-N,3-bis(4-chlorophenyl)-2-methyl-6-N-propan-2-ylisoquinoline-1,4,6-triamine (4Z)-2-methyl-4-[(3,4,5-trihydroxyphenyl)methylidene]-1,3-oxazol-5-one 4-azidosulfanylthieno[2,3-d]pyrimidine 3-[(6,8-dichloronaphthalen-2-yl)sulfanylamino]-4-fluoro-5-nitrobenzoic acid 4-(1,2,3-triazatricyclo[7.3.1.05,13]trideca-5,7,9(13)-trien-8-ylsulfanylamino)phenol 3-[4-(1,3-benzodioxol-5-yl)-6-oxo-2-pyridin-3-ylsulfanyl-1H-pyrimidin-5-yl]propanoic acid N-[5-(4-methoxyphenyl)sulfonyl-1,3,4-thiadiazol-2-yl]-2-piperidin-1-ylacetamide 1-[(3S)-6-fluoro-2,3-dihydroindole-1-carbonyl]-N-[4-(trifluoromethylsulfanyl)phenyl]cyclopropane-1-carboxamide 3-[4-(dimethylamino)anilino]benzaldehyde;ethane;N'-ethylpropanimidamide N-[(Z)-1,2-diphenylethylideneamino]-4-[(E)-[4-methyl-5-oxo-3-propan-2-yl-1-(3-propoxyphenyl)pyrazol-2-ium-2-ylidene]methyl]benzamide 1-but-2-ynylsulfanyl-3-[5-(4-chlorophenoxy)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carbonyl]pyrrolidin-2-one 4-[2,4-dimethyl-6-oxo-5-[(E)-2-(oxan-2-yloxy)ethenyl]pyrimidin-1-yl]-3-iodobenzamide 2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonylamino]benzoic acid 2-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-N-ethylquinazoline-8-carboxamide 4-N,7-N-dimethylisoquinoline-3,7-diamine;ethane N-(3-chlorophenyl)-N'-[4-[2-fluoro-5-(2,2,2-trifluoroethylsulfanyl)phenyl]-1H-pyrazol-5-yl]oxamide 3-(4,5-dihydro-1H-imidazol-2-ylamino)benzenesulfonamide 6-(3-methoxypropyl)-1H-quinazoline-2,4-dione 5-[2-(3,4-difluorophenyl)pyrrolidin-1-yl]-3-propan-2-ylsulfanyl-1H-1,2,4-triazole 7-amino-5-[4-fluoro-2-(oxan-2-ylmethoxy)phenyl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 3-[4-amino-2-(2,6-difluoroanilino)-5-fluorobenzoyl]-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxylic acid 4-[2-(cyclopropylmethoxy)-5-fluorophenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile 2-[2,4-bis(trifluoromethyl)phenyl]-N'-hydrazinylidene-1H-imidazo[4,5-b]pyridine-7-carboximidamide 2-[4-(1,3-benzodioxol-5-ylmethoxy)piperidin-1-yl]-5-[(2-methylphenyl)sulfonylamino]pyridine-3-carboxylic acid;2,2,2-trifluoroacetic acid 4-(2-amino-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperazine-1-carboxylate 5-chloro-N-[4-[2-[5-methyl-3-(trifluoromethoxy)pyrazol-1-yl]ethoxy]cyclohexyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 4-[(Z)-1-amino-2,3-dimethylbut-1-enyl]-N-[(2S)-1-amino-1-oxopropan-2-yl]benzamide;(3R)-8-azaspiro[3.5]nonane 5-(3,4-dichlorophenyl)-1-methylsulfonylpyrrolidin-2-one N-(2,6-difluorophenyl)-1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carboxamide 5-tert-butyl-1,4-bis(ethenyl)-3,8-dimethylquinolin-2-one 5-bromo-3-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)pentanoate N-[3,5-bis(trifluoromethyl)phenyl]-1-cyano-N'-(4-fluorophenyl)sulfonylcyclopropane-1-carboximidamide 3-(ethoxymethyl)-N'-hydroxypyridine-2-carboximidamide (4R)-1-phenylsulfanylcarbonylazepane-3,4-dicarboxylic acid 3-[5-(2,4-dihydroxyphenyl)tetrazol-1-yl]benzoic acid 2-[3-(1,3-benzoxazol-6-yl)butanoylamino]acetic acid 1-(5-bromothiophen-2-yl)-3,4,4a,6,7,8,8a-octahydro-1H-quinazolin-2-one (3aR)-2,10-dimethoxy-9,10-dihydrobenzo[a]acridine 2-[3,5-bis(trifluoromethyl)phenyl]propanoic acid 2-[3-(methylamino)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carbonyl]benzonitrile 2-[4,6-bis(5-bromofuran-2-yl)-1,3,5-triazin-2-yl]-N,N-diethylaniline (E,1Z)-N'-(aminomethyl)-2-ethoxy-3-[5-(trifluoromethyl)-2H-tetrazol-3-ium-2-yl]but-2-enehydrazide N-[4-chloro-2-[4-(1H-pyrrole-3-carbonyl)piperazin-1-yl]phenyl]-3-(trifluoromethyl)benzamide (1S,2R)-1-azido-3-bromo-6-[(4-chlorophenyl)methyl]-N-methoxy-4,5-dihydro-2H-inden-1-amine 5-[(3E)-4,5-dimethylhexa-1,3,5-trien-2-yl]-3-[(3Z,5Z)-hepta-1,3,5-trien-2-yl]pyridine 5-[2,6-dimethyl-4-[3-(4-methylpiperazin-1-yl)azetidine-1-carbonyl]phenyl]-1,3-diethylpyridin-2-one N-[3-(2,6-difluorophenyl)phenyl]-1-methyl-5-(methylaminosulfanyl)pyrazole-4-carboxamide;ethane N-[(3S,7R,8aS)-3-propan-2-yl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-5-oxo-1,4-diazepane-1-carboxamide 4-(2,5-dimethoxyphenyl)-3-(3-ethylpyridin-4-yl)furan-2-one;ethane [4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-[5-(2,6-difluorophenyl)-1H-pyrazol-3-yl]methanone N-[3-[2-(5-methoxy-1H-indazol-4-yl)acetyl]cyclobutyl]pyridine-2-carboxamide 4-(3,5-difluorophenyl)sulfanyl-2-[3-(4-methoxyphenyl)prop-1-enyl]-1H-pyrrole [3,6-dimethoxy-2-(4-propan-2-ylphenyl)pyridin-4-yl]carbamic acid 5-(4-bromophenyl)-1,3-dimethylpyrazole 2-chloro-N-(2,3,4,5,6-pentadeuteriophenyl)cyclopentene-1-carboxamide 2-(4-cyanophenyl)-N,4-dimethylpentanamide 5-fluoro-1,3-dimethylindazole;2-hydroxyethyl-methylidene-[1-[(6-propan-2-ylpyridin-3-yl)amino]pentyl]azanium 2-methyl-1'-(6-methylpyridazin-3-yl)spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,4'-piperidine]-4-one 3-fluoro-5-(2-hydroxyethyl)-6-methoxypyrimidin-4-one [3-(4-chlorophenyl)-1,2-oxazol-5-yl]-[(Z)-(4-hydroxy-3-methoxyphenyl)methylideneamino]azanide;tungsten(2+) 6-[1-(4-methylsulfanylbutoxy)propoxy]naphthalen-2-ol 5-(1,1,2,3,3a,4,5,6,7,7a-decahydroinden-5-ylmethoxy)-1H-indole (Z)-1-[2,3-difluoro-6-methoxy-4-[(E)-pent-3-enyl]phenyl]prop-1-ene-2-thiol (Z)-[N'-[[4,5-bis(difluoromethyl)furan-2-yl]methyl]carbamimidoyl]carbamic acid (E)-1,2-dicyanoethenesulfonic acid;palladium(2+);triphenylphosphane 2-[(7R)-7-methyl-5-thiophen-2-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidin-6-yl]ethanamine N-[(5S)-2,4-dioxospiro[4.5]decan-1-yl]-2-(1H-imidazol-2-yl)benzamide;2-hydroxyacetic acid 2-N-ethenyl-1-(4-methylsulfonylphenyl)-4-N-[4-[3-(trifluoromethyl)phenoxy]cyclohexa-2,4-diene-1-carbonyl]pyrrolidine-2,4-dicarboximidamide 2-azido-N-[3,5-difluoro-4-(3-piperidin-1-ylpropoxy)phenyl]-4-methylsulfonylbutanamide 2-(N,2-dimethylanilino)-3H-quinazolin-4-one 4-(dimethylamino)benzaldehyde;N-ethenylcyclopropanamine;4-[5-(2-methoxypyridin-3-yl)pyridin-3-yl]oxy-2-methylbutanal (5R,7S)-N-[3-(2,4-dichlorophenyl)cyclobutyl]-5-methyl-1,5,7-triazaspiro[3.4]octan-7-amine;2,2,2-trifluoroacetic acid 3-[(4-methylpiperazin-1-yl)methyl]-N-[3-(2H-quinolin-1-yl)propyl]benzamide 2-methyl-N'-(4-methylsulfanylphenyl)quinoline-3-carboximidamide 2-[4-[[1,3-dimethyl-5-(pyrrolidine-1-carbonyl)pyrazol-4-yl]carbamoylamino]-1H-pyrazol-5-yl]acetamide 1-(azidomethyl)-5-chloro-3-(4-fluorophenoxy)benzene 3-[1,2-difluoro-2-(5-methylthiophen-2-yl)ethenyl]-4-ethynyl-N,4-diphenylcyclohexa-1,5-dien-1-amine N-[4-methoxy-7-(1H-pyrazol-5-yl)-[1,3]thiazolo[4,5-c]pyridin-2-yl]-1,3-dimethylpiperidine-4-carboxamide;hydrochloride 7,9,10-trioxotetracene-5,12-dicarboxylate 5-methoxy-2-(3-methylbutan-2-ylidene)-3,4-dihydroquinoline 1-[(2-methylpyrazol-3-yl)amino]-3-[[4-[(5-piperidin-1-ylpyridin-2-yl)carbamoylamino]phenyl]methyl]urea 1-[3-(methylideneamino)phenyl]sulfonyl-4,5,6,7-tetrahydroindazole-3-carboxamide 2-(5-nitro-2,3,4-triphenylimidazol-1-ium-1-yl)-N-[2-[5-[(E)-1H-pyrrol-2-ylmethylideneamino]oxypentoxy]ethyl]acetamide;chloride 4-(1,3-benzodioxol-5-ylmethoxy)butan-2-ylidene-(3,5-ditert-butyl-4-hydroxyphenyl)azanium 2-chloro-1H-indole;4,5-diethoxypyridine-3-sulfinamide 2-[4-[[(3R)-1-benzoylpiperidine-3-carbonyl]amino]-3-fluorophenoxy]acetic acid (E)-3-[2,5-bis(trifluoromethyl)phenyl]-N,4,4-trideuterio-1-[4-(difluoromethoxy)-3-[(4-methylpiperazin-1-yl)methyl]phenyl]-N-methyl-3-(methylideneamino)but-2-en-2-amine 2-[azido-[4,5-dichloro-1-(2-methylpropyl)pyrazole-3-carbonyl]amino]propanoic acid (2S)-2-acetamido-5,8-dimethoxy-9-oxo-N-[2-phenyl-1-(2H-tetrazol-5-yl)ethyl]undecanamide 2-(6-fluoro-1,3-benzothiazol-2-yl)-5,8-dihydroxy-7-methoxy-4a,9,10,11b-tetrahydro-3H-benzo[d][2]benzoxepin-1-one 2-[2,4-dichloro-5-(3-cyano-1-methylpyrazol-4-yl)anilino]ethanesulfonic acid 2-N,7-N-di(propan-2-yl)-[1]benzofuro[3,2-e][1]benzothiole-2,7-diamine 1-(2,6-diethylphenyl)sulfonyl-3-[4-hydroxy-7-[2-(trifluoromethoxy)phenyl]heptyl]urea [5-methyl-3-(2-phenylethynyl)furan-2-yl]-spiro[3,4-dihydroisochromene-1,1'-cyclopropane]-7-ylmethanone 2-(3-azidophenyl)sulfanyl-1,4-dimethoxybenzene 4-[[4-methoxy-3,5-bis(trifluoromethyl)phenyl]methyl]piperazine-1-carboxylic acid 6-methoxy-7-phenyliminoquinoline-5,8-dione 2-[3,4-dichloro-1-(1,2,4-triazol-4-yl)buta-1,3-dienyl]-5-propan-2-yloxypyridine ethane;2-[1'-(3-methylbenzoyl)spiro[3,4-dihydrochromene-2,4'-piperidine]-6-yl]oxyacetic acid (4S)-5'-bromospiro[1,3-dihydroisochromene-4,3'-azetidine] (4S)-5-[3,6-difluoro-2-[[1-[[4-fluoro-2-[(2-methylpropan-2-yl)oxycarbonyl]phenyl]carbamoyl]cyclobutyl]amino]phenoxy]-4-hydroxypentanoic acid 4-N-azido-2-N,6-dimethylpyridine-2,3,4-triamine 2-[4-(2,3-difluorophenyl)-7-hydroxy-3-propylnaphthalen-1-yl]oxypentanoic acid 5-chloro-2,3-dimethyl-1H-indazole;2,4-dinitroaniline (2R,3S)-N-[cyclopropylmethoxy(phenyl)methyl]-N'-[(5-methylfuran-2-yl)methyl]-2-phenylpyrrolidine-1-carboximidamide;hydrochloride 4-[7-chloro-6-fluoro-2,4-dioxo-1-(2-piperidin-3-ylethyl)quinazolin-3-yl]benzoic acid 2-[3-(4,5-difluoro-3-methyl-1H-indol-2-yl)phenyl]propanoic acid 3-[2-(2,6-dioxopiperidin-4-yl)-1,3-dihydroxyisoindol-5-yl]oxypiperidine-2,6-dione 1-[(4R)-3,6-diazabicyclo[3.2.0]heptan-3-yl]-2-[5-hydroxy-3-(2-methoxyphenyl)pyridin-2-yl]ethanone N-methyl-4-oxo-5,7,8,9-tetrahydrothieno[3,2-h]quinazoline-6-carboxamide (5Z)-2-imino-5-[(3-phenoxyphenyl)methylidene]-1,3-thiazolidin-4-one (4-methoxy-2,6-dimethylphenyl)-[8-(6-propan-2-ylpyridin-3-yl)-1,11-dioxa-4,7,10-triazacyclododec-4-yl]methanone N-[4-[2-azidooxy-1-(3,4-difluorophenyl)ethyl]pyridin-3-yl]-2-methylpropanamide 6-benzylsulfanyl-N,2-dimethoxypyrimidine-4-carboxamide N-(4,5-dimethyl-2-phenyldiazenylphenyl)-2-methoxy-N-octylacetamide 3-[[4-(2-chloroanilino)pyrimidin-5-yl]amino]benzamide 6-(3,5-dimethoxyphenyl)-1-[4-[3-fluoro-5-(2,2,2-trifluoroethyl)phenoxy]butyl]pyrazolo[3,4-d]pyrimidine 6-amino-4-(2,3-dihydro-1H-inden-5-yl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide (E)-2-(1,3-benzothiazol-5-ylsulfonylamino)-3-[4-ethenyl-3-methoxy-6-[3-(trifluoromethyl)phenyl]pyridin-2-yl]prop-2-enethioamide 4-amino-3-bromo-5-ethylsulfonylbenzoic acid [2-(3,5-dimethylpyridin-1-ium-1-yl)propanoyloxy]-(6-ethyl-8-oxo-7H-naphthalene-1-carbothioyl)azanide;uranium(2+) 4-(6,7-dimethylquinolin-3-yl)oxy-N-[2-hydroxy-3-(1H-indol-3-ylmethylideneamino)propyl]benzamide 2-(difluoromethyl)-N-[4,4-bis(ethoxysulfanyl)cyclohexa-1,5-dien-1-yl]benzamide 4-(methylamino)-5-nitro-2-propoxybenzaldehyde 5-[7-chloro-1-(2,4-difluorophenyl)-6-fluoro-4-hydroxy-3-methylisoquinoline-8-carbonyl]-1H-pyrrole-3-carboxylic acid 1-[3-[4-(1,6-dimethylindazol-5-yl)phenyl]azetidin-3-yl]ethanone 1-(3,5-dimethylphenoxy)ethanesulfonate 3-[2-(4-fluorophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2,1-benzothiazole;hydrochloride 3-[2,4-dimethyl-5-(1-tritylimidazole-4-carbonyl)phenyl]propanoic acid 4-(2,3-dihydro-1H-inden-1-yl)benzene-1,3-diol N-[[1-(4-hydroxybenzoyl)piperidin-3-yl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-6-carboxamide N-[(2S)-3,3-dimethylbutan-2-yl]-1-[5-[2-(2-hydroxyethoxy)propan-2-yl]pyridin-3-yl]cyclohexane-1-carboxamide N-[5-(3-methoxyphenyl)pentyl]formamide 4-(2,3-dimethoxyphenyl)-6-ethyl-1H-quinazoline-2,7-dione 1-[(2R,4S)-4-methoxy-6-(pyridin-3-ylmethylcarbamoyl)oxan-2-yl]-3-methylpyrazole-4-carboxylic acid 5-(azidomethyl)-3-(trifluoromethoxy)pyridine 2,5-dimethyl-N-[2-(4-methylphenyl)ethyl]pyrazole-3-carboxamide ethane;5-methyl-2-(3-phenylbutan-2-yl)phenol 5-methyl-7-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)spiro[2.4]heptane-6-carboxamide N-[2-(4,5-dimethylfuran-2-yl)oxolan-3-yl]-1H-pyrrolo[3,2-c]pyridine-6-carboxamide 2-(3,4,5-trimethylphenyl)pentanedioic acid 6-benzyl-1,2-benzothiazol-3-one 1,3-bis[2-chloro-4-(trifluoromethyl)phenyl]-5H-pyrazolo[4,3-c]pyridin-4-one N'-ethyl-2,6,7-trimethoxyquinazoline-4-carbohydrazide 3-[1-[6-(furan-2-yl)pyridin-2-yl]piperidin-4-yl]quinazolin-4-one [6-fluoro-2-(trifluoromethyl)-3H-benzimidazol-5-ium-1-yl]-(4-hydroxyphenyl)methanone [3-(5,6-dihydrobenzo[b]carbazol-11-yl)phenyl]boronic acid 4-methyl-6-(oxan-2-yl)pyrrolo[3,4-d]pyrimidine 1-(6,7-dihydro-1H-indol-3-yl)-2-[2-ethoxy-4-[[hydroxy-[1-(4-methylphenyl)piperidin-4-yl]amino]methyl]phenoxy]ethanone 2-[4,5-bis(4-methoxyphenyl)-1H-imidazol-2-yl]ethanol 3-chloro-5,6,7-triphenylnaphthalene-2-carboxylic acid 4-[3,5-dichloro-N-(2-methylpropanoyl)anilino]benzoic acid 2-[3-fluoro-4-(3,4,5-trifluorophenyl)phenyl]-6-methyl-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene (4R)-1-ethyl-2,2-dimethyl-6-phenyl-3,4-dihydroquinoline N-[1-(2,4-dimethylcyclohexanecarbonyl)piperidin-3-yl]-2-methoxy-6-(trifluoromethyl)pyridine-4-carboxamide (1R)-N-[3-[4-amino-2-methyl-5-[(E)-[(2Z,4E)-2-(trifluoromethoxy)hexa-2,4-dienylidene]amino]phenyl]prop-2-ynyl]-4-ethylcyclohexane-1-carboxamide 1-[2-(diethylamino)ethyl]-3-[4-fluoro-3-(trifluoromethyl)phenyl]-1-(4-sulfamoylphenyl)urea 5-(cyclopropylmethoxy)-2,3-dihydroinden-1-one (2R)-1,1-dimethyl-2-[4-(5-propylbenzimidazol-1-yl)phenyl]hydrazine 2-[1-(1,3-benzodioxol-5-ylsulfonyl)piperidin-4-yl]oxyacetic acid 4-[2-[(6-but-3-enyl-1,2,3,4-tetrahydronaphthalen-1-yl)methoxy]phenyl]benzonitrile 2-bromo-1,4-difluoro-3-[4-(4-methylphenyl)buta-1,3-dienyl]benzene (2S,3R)-N-[[3-(2-methylpyrazol-3-yl)phenyl]methyl]-2-(1H-pyrazol-4-yl)oxolan-3-amine (E)-4,8-bis(4-bromophenyl)oct-5-enal;N-(3-chlorophenyl)propanamide 6-[3-methyl-1-(4-methylphenyl)-5-(3,3,3-trifluoropropoxy)pyrazol-4-yl]-2-pyrimidin-2-ylimidazo[2,1-b][1,3,4]thiadiazole 4-(4-fluorophenyl)-2,3-dimethyl-5H-1,5-benzothiazepin-8-ol 1-(1H-benzimidazol-2-yl)-6,7-dimethoxy-2-[4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]phenyl]sulfanylhepta-4,6-dien-3-one 1-(3,5-dimethylphenyl)-N-[(2R,4E)-4-hydroxycycloocta-1,4-dien-6-yn-1-yl]cyclopropane-1-carboxamide 5-[(2,3-dimethylimidazol-4-yl)sulfonylamino]thiophene-2-carboxylic acid (5R)-2,3-dimethyl-5-(4-nitrophenyl)-1,3-oxazolidine N-methylsulfonyl-2,4-dinitrobenzenecarboximidate 1-(4-iodophenyl)-2H-pyrimidine N-[5-(azepan-1-yl)pentan-2-ylidene]-2-(cyclopropanecarbonylamino)-1,3-thiazole-4-carboxamide 2-(1,3-benzothiazol-2-yl)-6-[5-(4-methoxyphenyl)thiophen-2-yl]phenol N-cyclohexyl-2-[4-hydroxy-5-(indol-3-ylidenemethyl)-2-oxo-1,3-thiazol-3-yl]acetamide [4-(3,5-dichlorophenyl)piperazin-1-yl]-(2-methoxy-6-methylpyridin-3-yl)methanone;2,2,2-trifluoroacetic acid [7-chloro-5-(2,6-difluorophenyl)-1H-indol-3-yl]-(2-methylpyrazol-3-yl)methanone [2-amino-5-(1,3-benzothiazol-2-ylmethylcarbamoyl)phenyl]carbamic acid 5-(2,3-dimethylphenoxy)-N'-hydroxypyridine-2-carboximidamide 4-(2,5-dichlorophenyl)sulfonyl-5,7-diethyl-1H-pyrrolo[3,4-c]pyrazole 5-bromo-4-N-[2,5-dimethyl-1-(3,5,6,7-tetrahydropyrrolo[3,4-d]pyrimidin-4-ylidene)piperidin-3-yl]-2-N-(2-methoxyethyl)pyrimidine-2,4-diamine;ethane 4-[6-amino-5-(4-methylphenyl)pyridazin-3-yl]phenol 6-[2,3,5,6-tetrafluoro-4-(trifluoromethyl)phenoxy]pyridazine-3-carboxamide 2-[(1E,3Z)-5-hydroxyhexa-1,3,5-trienyl]benzene-1,4-diol 2,5-difluoro-3-[(4S)-4-methyloxolan-2-yl]sulfanylaniline 3-[4-(cyclohexylmethoxy)phenyl]oxirane-2,2-dicarbonitrile 1-(2,3-dihydroindol-1-yl)pentan-1-one [2-[(6-chloropyridine-3-carbonyl)amino]phenyl]methylazanium 3-[(4,5-dichlorothiophene-2-carbonyl)amino]-2-methylpropanoic acid 1-(3,5-dichloropyridin-4-yl)pyrrolidine-2-carboxylic acid N-benzylsulfanyl-1-[4-chloro-2-[(E)-2-nitroethenyl]phenyl]methanamine 7-ethyl-3,5-bis(2-methoxyphenyl)pyrazolo[1,5-a]pyrimidine N-(3,5-dimethoxyphenyl)-6-ethyl-2-[[4-oxo-5-(pyridine-3-carbonylamino)pyrazolo[1,5-a]pyrazin-2-yl]methylamino]pyrimidine-4-carboxamide 1-(3,5-dichlorophenyl)butane-2-thione 2-[(4R,5S)-2-[2-[3-fluoro-4-(trifluoromethoxy)phenyl]ethyl]-1-oxo-3-azabicyclo[3.1.0]hexan-6-yl]acetic acid [2-(2,6-dimethylanilino)-2-oxoethyl]-diethyl-[1-(2-hydroxyphenyl)ethylideneamino]azanium;chloride (6-bromo-2,3-dihydroindol-1-yl)-[5-methyl-6-(oxolan-3-yloxy)pyridin-3-yl]methanone 3-(6-chloropyridin-3-yl)-1-[1,4-dimethoxy-2-(5-nitrothiophen-2-yl)naphthalen-1-yl]propane-1,2-dione 2-(3,5-dichlorophenyl)sulfanyl-N'-hydroxypyrimidine-4-carboximidamide 2-[4-bromobutan-2-yl(prop-2-enyl)amino]-1,3-thiazole-5-carboxylic acid 2-[3-(hydroxymethyl)-5-oxo-1-phenylpyrrolidine-3-carbonyl]-1,3-dihydroisoindole-4-carboxamide 2-tert-butyl-6-cyclopropylidene-3-[(5E)-4,7-dimethylocta-1,5,7-trien-3-yl]-1H-pyridine 2-[4-methyl-3-(methylamino)phenyl]naphthalene-1,5,7,8-tetracarboxylic acid 1-(4-fluorophenyl)indazole;N-propylcyclobutanamine 1-[4-chloro-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propan-2-one (2R)-2-azido-N-[(3,4-dimethylphenyl)methyl]-1-ethoxypropan-1-amine 2-[(3-fluorophenyl)methyl]-9H-fluoren-1-amine 2-N,4-N-bis(9H-fluoren-1-yl)-3,5-dimethoxybenzene-1,2,4-triamine 3-(7,8-dimethyloctoxy)benzenesulfonate 4-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-8-methyl-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-9-one 2,5-dichloro-4-nitrothiophene;ethane 1-[(3,5-dimethylphenyl)methyl]-4-(2-fluoroanilino)sulfanylpiperidine-4-carboxylic acid 3-(2,6-dimethylmorpholine-4-carbonyl)pyrazolo[1,5-a]pyridine-7-carboxylic acid 2-[5-(3,4-dichlorophenyl)-1,2-oxazol-4-yl]acetaldehyde;methoxyethane 1-azidooxysulfanylnaphthalene 3-[(3R)-5-acetyloxypentan-3-yl]-4-nitrobenzenesulfonate (4-methylphenyl)-[4-(thiophene-3-carbonylamino)phenyl]azanium 5-(2,4-difluorophenyl)-1H-pyrrolo[3,2-b]pyridine 5-methyl-N-[[3-(2-methylpropoxy)phenyl]methyl]pyrazolo[1,5-a]pyrimidine-7-carboxamide 2-[3-methoxy-4-(4-methylpiperazin-1-yl)phenyl]acetamide [(2S,4R)-2-benzylpiperidin-4-yl]-[7-(2-propan-2-yloxypyridin-3-yl)thieno[3,2-b]pyridin-2-yl]methanone ethane;1-[(3E)-hexa-1,3,5-trien-3-yl]-4-[6-(4-phenylcyclohexa-1,3-dien-1-yl)pyridin-2-yl]benzo[f]quinoline 3-azido-5-chloro-N-[2,4-dimethoxy-6-(trifluoromethyl)phenyl]pyridin-2-amine N-methyl-1-phenyl-4,6-bis(2H-pyridin-3-ylidene)pyrimidine-5-carboxamide 5-[(3R)-1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-3-yl]-2-oxa-6-azaspiro[3.4]octan-7-one 2-[4-[[4-(hydroxymethyl)phenyl]methoxy]anilino]-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one 1-[(4,5,6-trimethylpyrimidin-2-yl)amino]piperidine-3-carboxamide 2-(N-hexadecyl-4-methoxyanilino)-4-methylpentanoic acid 5-(dibenzylamino)-7,8-dimethoxyquinoline-3-carboxamide 5-[[1-(5-hydroxypentyl)piperidin-4-ylidene]methyl]-1-(6-methoxypyridin-3-yl)-2H-pyrazolo[1,5-a]pyrimidine-7-thione 1-azidosulfonylsulfanyl-4-benzylbenzene [5-(2,2-difluoroethoxy)pyridin-3-yl]methanediol (2Z,3E)-6-amino-5-[[2-[[2-(dimethylamino)ethylamino]-hydroxymethylidene]-1,3-benzothiazol-3-ium-3-yl]oxy]hexa-2,4-dienal 5-[2,6-dichloro-4-(5-methylpyridin-3-yl)phenoxy]-2-nitrophenol N-[3,5-dichloro-4-[(2E)-2-ethenylpenta-2,4-dienoxy]phenyl]acetamide 1-[5-[4-(3,5-dichlorophenyl)piperazine-1-carbonyl]indol-1-yl]ethanone 5-[1-(4,6-dichloro-2H-pyrimidine-1-carbonyl)piperidin-3-yl]-2H-triazole-4-carbonitrile N-[[2-amino-4-[(6-chloro-1,3-benzothiazol-2-yl)sulfonyl]phenyl]methylidene]propanamide 5-(3,4-dichlorophenyl)sulfanyl-1-(4-ethoxyphenyl)-2H-pyridine 3,4-dimethyl-2,7-bis(phenylsulfanyl)pyrene 2-(2,3-dihydroindol-1-yl)-N'-hydroxypyridine-4-carboximidamide 2-[2-(3,4-dimethoxyphenyl)ethynyl]-5-hydroxybenzaldehyde 7-(6,8-dichloro-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-2-iodoheptanoate N-[3,5-bis(trifluoromethyl)phenyl]-1,2-difluoroethenamine 6-[3-fluoro-4-[2-(trifluoromethyl)pyrimidin-5-yl]phenyl]-4-hydroxy-1H-pyridin-2-one N-[2,5-dimethyl-4-(morpholine-4-carbonyl)phenyl]-4-(4-oxo-1H-quinazolin-3-ium-2-yl)butanamide 3-methyl-N-[(1-phenylpiperidin-4-yl)carbamoyl]pyridine-2-carboxamide N-[(1R)-6,7-dimethoxy-3,4-dihydro-2H-chromen-4-yl]-N',N'-diethylpropane-1,3-diamine 2-[4-fluoro-5-(methoxymethyl)-1H-benzimidazol-2-yl]phenol 4-[(4-butyl-N-ethenyl-3-methoxyanilino)methylidene]benzonitrile N-[3,4-bis(2-methylpropoxy)phenyl]acetamide N-(4-chlorophenyl)-2-cyclopropylpyrazolo[1,5-a]pyrazine-3-carboxamide 1-(4-hydroxy-3,5-dimethoxyphenyl)-5-methyldodecan-2-one N-[(Z)-(3,5-dibromo-2,4-dihydroxyphenyl)methylideneamino]propanamide 3-[N-(2,2-diethoxyethyl)-4-methylanilino]propane-1,2-diol 3-methyl-5-[4-(trifluoromethoxy)phenyl]-1H-indole (3-bromophenyl)methylcarbamodithioic acid 6-methoxy-N'-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyridine-2-carboximidamide 4-[5-(1,3,3-trimethylindol-2-ylidene)penta-1,3-dienyl]quinoline ethane;1-[(5S)-9-methoxy-2,3,4,7,12b-hexahydro-1H-indolo[2,1-a]isoquinolin-6-yl]butan-1-one 1-[5-ethylsulfonyl-6-[7-methoxy-3-(trifluoromethyl)imidazo[4,5-c]pyridin-2-yl]pyridin-3-yl]cyclobutane-1-carboxamide [2-(3,5-ditert-butylphenyl)-3-methoxyphenyl]boronic acid 2-(3,4-dimethoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine 1,5-ditert-butyl-3-(1-phenylethenoxy)pyrazole 4-amino-2-(2,5-dimethoxyphenyl)benzoic acid (7S)-N-[2-(4-chlorophenyl)ethyl]-11,14-dioxo-4-oxa-1,8-diazatricyclo[8.4.0.03,8]tetradeca-10,13-diene-13-carboxamide 2-[(1-methylimidazole-4-carbonyl)amino]propanedioic acid 2-[[4-(4,5-dihydrobenzo[g][1]benzoxepine-2-carbonyl)phenyl]methyl-methylcarbamoyl]benzenesulfonic acid 5-chloro-4-[1-ethyl-3-(1-methylpyrazol-3-yl)azepan-3-yl]oxy-2,6-difluoropyrimidine (5S,7R)-2-benzylsulfanyl-N-(3,4-dichlorophenyl)-5-methyl-7-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide N-(3-chlorophenyl)-2-[6-ethyl-7-(4-fluorophenyl)-2-oxo-1,3-dihydroimidazo[1,2-b]pyrazol-3-yl]acetamide 3-bromo-4,5-dimethoxy-N'-methyl-6-(trifluoromethyl)pyridine-2-carboximidamide N-(furan-2-ylmethylideneamino)-4,5-dihydro-1H-imidazole-5-carboxamide 3-methyl-2,6-dioxo-N-[1-(4-propan-2-ylphenyl)cyclopropyl]piperidine-3-carboxamide 1,6-dimethyl-3-(3-nitrophenyl)pyrazolo[4,3-c]pyridine N-[6-(4-aminophenyl)pyrido[3,2-d]pyrimidin-4-yl]hydroxylamine 1-[(4Z)-5,6-dichloro-2-methylhepta-2,4,6-trien-3-yl]oxyethenamine;ethane 5-[(2E,3Z)-1-methylsulfanylhexa-2,3-dien-2-yl]oxypyridine-2-carboxylic acid 4-[(E)-3-[5-[5-fluoro-2,6-dimethyl-4-[[1-(oxan-4-yl)pyrazol-4-yl]amino]pyridin-3-yl]thiophen-2-yl]prop-2-enimidoyl]phenol 3-(1,3-dihydroisoindol-2-yl)pyrazine-2-carbonitrile 4-(2,6-dichlorophenyl)-5-methyl-1H-pyrazole N-(cyclopropylmethoxy)-2-[4-fluoro-3-(trifluoromethyl)phenyl]-5-methylsulfonyl-1,3-dihydroisoindole-1-carboxamide 4-[8-amino-3-[1-(pyridine-3-carbonyl)pyrrolidin-2-yl]imidazo[1,5-a]pyrazin-1-yl]cyclohexan-1-ol 2-[(3Z)-4-bromohexa-1,3-dien-3-yl]oxy-N-methylaniline 4-[(1R)-1-azidoethyl]-2-methoxy-6,7,8,9-tetrahydrobenzo[g]quinazoline N-(1,3-dimethylindazol-5-yl)-2,4-dihydroxybenzamide 2-methylsulfonylethanamine;3,4,5-trimethoxy-N-[(E)-[5-(methylideneamino)pyridin-3-yl]methylideneamino]benzamide 2-(furan-3-yl)-N'-hydroxypyrimidine-4-carboximidamide 6-methyl-4-(trifluoromethyl)-5,7-dihydro-1H-furo[3,4-c]pyridin-3-amine 2-[(5R,10bR)-9-chloro-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 1-(3-hydroxypropyl)-N',6-dimethylindole-5-carbohydrazide N'-[4-(1-methoxyethenyl)phenyl]-N,2-dimethyl-N-(thiophen-2-ylmethyl)butanimidamide 4-[1-(2,3,5,6-tetrafluorophenyl)ethyl]benzenesulfonic acid 1,3-diamino-1-[2-[[4-(benzylcarbamoyl)cyclohexyl]oxymethyl]phenyl]urea;ethane (2S)-N-[[4-(1H-benzimidazol-2-ylmethoxy)phenyl]methyl]-5-ethylsulfanylpyrrolidine-2-carboxamide 2-amino-4-[3-(5-methylimidazol-1-yl)propoxy]benzaldehyde 2-benzyl-3,5-dinitrobenzoic acid 2-[(E)-1-cyclopropylidene-4,4,4-trifluorobut-2-enyl]-6-piperidin-3-ylpyridine 3-ethyl-5,6-dimethyl-2-phenylbenzo[f]benzimidazole 4-[2,6-dichloro-N-(3-methylbutyl)-4-nitroanilino]butan-1-ol 4-[3-fluoro-4-(2-propan-2-yl-1H-imidazole-5-carbonyl)phenyl]benzoic acid 4-(3-amino-2,4,6-trimethylphenyl)butan-2-ol 3-[[2-fluoro-5-(1,4,6,7-tetrahydropyrano[4,3-c]pyrazole-3-carbonyl)phenyl]carbamoyl]-1H-pyridazin-6-one 1-[[4-amino-3,5-di(butanoyl)phenyl]methyl]-2H-isoquinoline-3-carboxylic acid (6S)-N-[(1R,2R)-1-hydroxy-1-(3-methoxyphenyl)propan-2-yl]-6-methyl-4-oxo-6,7-dihydro-5H-triazolo[1,5-a]pyrazine-3-carboxamide 6-methyl-8-[(5R)-5-methylpiperazin-1-yl]-2,3-dihydro-[1,4]oxathiino[2,3-c]pyridine 6-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-N-[5-methanimidoyl-1-methyl-2-(6-morpholin-4-ylpyridine-3-carboximidoyl)pyrrol-3-yl]pyrazin-2-amine 4-[(2,6-dichlorophenyl)methyl]-N-ethylaniline;hydrobromide 2-(2,4-dichloro-5-fluorophenyl)-1H-imidazole;dihydrochloride 1-(5-azidopentyl)-2,4-diethylbenzene (2S)-1,3-diamino-4-phenylbutan-2-ol 4-[3-(hydroxymethyl)phenyl]benzoic acid 5-amino-4-[3-fluoro-2-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione N-[5,6-diethyl-3-(1H-pyrazole-4-carbonyl)pyridin-2-yl]-N'-methanimidoylpropanediamide 1-azido-2,4-dimethylindole-5-carbonitrile 1-methyl-N-[4-(2H-tetrazol-5-yl)phenyl]pyrrole-3-carboxamide 6-methyl-4-[(1-propan-2-ylcyclobutyl)amino]-5,6,7,8-tetrahydroquinoline-3-carboxylic acid 4-[(2,6-difluorobenzoyl)amino]-1H-pyrazole-5-carboxamide (4S)-1,3-dimethyl-2,4-diphenylpyrrolidine 1-[3-[4-[(E)-2-[7,7a-dimethyl-7-[4-(trifluoromethoxy)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-ylidene]ethyl]piperidine-1-carbonyl]phenoxy]propan-2-one 4-chloro-3,7-dinitro-1H-quinolin-2-one 2-[4-[[(4-chlorophenyl)carbamoylamino]methyl]piperidin-1-yl]acetic acid 5-[4-(4-carboxyanilino)phenyl]-2,3-dihydrothiophene-2-carboxylic acid 3-[(Z)-aminomethylideneamino]-6-bromo-N-methylpyridine-2-carboxamide 3-bromo-1,4-dihydroquinoxaline 2-(3,4-dichlorophenyl)-N-[[5-methylsulfanyl-1-[6-oxo-1-propan-2-yl-5-(trifluoromethyl)pyridazin-4-yl]pyrazol-4-yl]methyl]acetamide 3-butanoyloxypropyl-[4-[(E)-4-chloropent-1-enyl]phenyl]sulfonylazanide 5-[3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-indazole-3-carboxylic acid 2-methoxy-4,6-di(propan-2-yl)phenol 2-[N-[(4,5-dimethyl-1H-pyrazol-3-yl)methyl]-3,5-bis(trifluoromethyl)anilino]-N-methylacetamide;ethane N-(4,5-dimethylpyrimidin-2-yl)-1H-indol-6-amine 5-bromo-4,6-difluoro-N'-methylpyridine-2-carboximidamide 2,7-bis(2,6-dimethylphenyl)-9,10-dihydrophenanthrene;ethane 1-[4,5-dimethyl-2-(methylamino)phenyl]-2-(6-ethylpyridin-3-yl)imidazole-4-carboxamide N-[2-(1H-indol-3-yl)ethyl]-N-(4-propylphenyl)benzamide 1-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-3-ylmethyl)-3-[3-fluoro-4-(5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl)phenyl]urea 7-azido-4,5-dichloro-2H-pyrazolo[3,4-b]pyridine 2-[4-(3-methyl-1,2,4-oxadiazol-5-yl)anilino]-N-propan-2-ylpyridine-4-carboxamide N-[(E)-1,3-benzodioxol-5-ylmethylideneamino]pyridine-4-carboxamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-6-[(E)-pent-3-enyl]-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 4-[N'-(3,5-dimethylphenyl)carbamimidoyl]-N-ethylbenzamide 5-methyl-3-[1-(5-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]quinazolin-4-one (E)-1-[4-(5,6-dimethylquinolin-8-yl)phenyl]but-2-en-1-one 4-ethyl-2,5-difluoro-N-[1-(3-methoxypropyl)pyrazol-4-yl]benzamide 5-[4-[[(2R)-1-hydroxybutan-2-yl]amino]quinazolin-6-yl]pyrazine-2-carboxylic acid 3-[3,4-dimethyl-6-(1H-pyrazol-5-ylamino)cyclohepta-2,4,6-trien-1-ylidene]-N'-propan-2-yl-2-[1-(2,2,2-trifluoroethylamino)ethenyl]propanehydrazide N-[(4-methyloxan-4-yl)methyl]-1,2-benzothiazol-3-amine N-(3,4-dimethylphenyl)-5-methoxy-2H-pyrimidine-1-carboxamide 2-[7,8-dimethoxy-3-(4-methylphenyl)sulfonylquinolin-4-yl]phenol 1-[2,6-di(propan-2-yl)phenyl]-2-methylimidazole;ethene 5-[5-chloro-1-[4-(3,7-dimethyloctyl)phenyl]pyrazol-3-yl]-2H-tetrazole 2,6-dichloro-3-(pyridine-4-carbonyl)benzaldehyde (6S,9R)-6-methyl-2-(4-nitrophenyl)sulfanyl-9-thiophen-3-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 5-(2,3-dihydro-1H-pyrrolo[2,3-b]pyridin-4-ylmethyl)-N,N-diethylpyridin-2-amine N-[(3,4-dichlorophenyl)methyl]piperidine-2-carboxamide 4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-ethylsulfanylbenzamide (2S)-1-[3-(4-azidophenyl)propylamino]-3,3-dimethylbutan-2-ol 2-[[3,4-dihydronaphthalene-1-carbonyl(methyl)amino]methyl]benzamide (2R)-N-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-2-methoxy-2-phenylpropanamide 1,4-difluorobenzene;1-[5-[(Z)-3-(2-ethylphenyl)but-2-enylidene]-6H-phenanthridin-9-yl]piperidine-4-carboxylic acid 4-(3,5-dichlorophenyl)sulfanyl-2-methylbutanenitrile (E)-2-cyano-3-[4-(ethoxycarbonylamino)phenyl]prop-2-enoic acid 4-[3-(furan-2-yl)-4H-quinazolin-2-yl]phenol 4-[4-(methoxymethyl)phenyl]-1H-pyridine 1-[5-(3,4-dichlorophenyl)-2-oxopentyl]pyrrolidine-2,5-dione 2-(6-methylheptan-3-yl)pyridine N-ethenyl-2,5-bis(3-methoxyphenyl)aniline 2-[4-(1,3-dioxol-2-yl)phenyl]-5H-pyrido[2,3-b]pyrazine 2-[4-(ethylamino)-2-nitrophenyl]sulfanyl-4-propyl-1H-pyrimidin-6-one 2-cyclohexyloxycarbonylbenzoic acid 4-[2,3,5-trifluoro-6-methyl-N-(propylamino)anilino]piperidine-1-carboxylic acid 2-[6-[(4-methylphenyl)methoxy]pyridin-3-yl]-5H-[1,3]oxazolo[3,2-a]pyrimidine 2,3-dibromoanthracene 2-(4,4-dimethylcyclohexen-1-yl)-3-methoxy-4-nitropyridine N-[2-(5,7,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),3,6,9,11-pentaen-13-yl)ethyl]acetamide 3-azido-7-chloro-1H-pyrazolo[4,3-b]pyridine 4-chloro-3,8-dimethylnaphtho[1,2-f][1]benzothiole (2Z,4E)-3-[3-cyclohexyloxy-4-(trifluoromethyl)phenyl]hepta-2,4,6-trienoic acid 4-N,4-N-diphenyl-6-N-(2H-1,3-thiazol-2-id-5-ylmethylideneamino)pyrimidine-2,4,6-triamine N-(diaminomethylidene)-3,5-difluoro-4-methoxybenzamide;ethane 2-chloro-4,8-dimethyl-7H-furo[3,2-e]indole 5-methoxy-N-[(3S)-3-methyl-2,3-dihydro-1H-inden-1-yl]-3,4-dihydro-2H-chromene-8-sulfonamide N-[[5-[(4,6-dichloropyrimidin-2-yl)sulfamoyl]thiophen-2-yl]methyl]benzamide N'-[amino(methyl)carbamoyl]-4-(4,5-dihydrobenzo[g][1,2]benzoxazol-7-yl)piperidine-1-carboximidamide;ethane 1-[2-(4-fluorophenyl)ethyl]piperidine;2,3,5-trimethylcyclohexa-1,3-diene (2S)-1-azido-2-methylsulfonyl-3-(4-phenylphenyl)propan-2-ol 7-[(2S)-1-cyclopentylpropan-2-yl]-8-methoxy-N,4-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide 3-[3,5-difluoro-2-methyl-4-(6-oxo-1H-pyridin-3-yl)phenyl]-3-[[(2R)-4-[2-(oxan-4-yloxy)ethyl]morpholin-2-yl]methylcarbamoylamino]propanoic acid 4-(ethylamino)-N-[2-(methylsulfanylamino)phenyl]benzamide 6-ethyl-7,8-dihydrobenzo[h]quinoline N-[5-chloro-2-[(3S)-4,6-difluoro-3-propyl-1-[(E)-3,3,3-trifluoro-2-methylprop-1-enyl]sulfonyl-2H-indol-3-yl]phenyl]acetamide ethane;N-[4-fluoro-5-(2-fluoropropan-2-yl)pyridin-3-yl]formamide 2-[[5-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]pyrimidin-2-yl]amino]-N-[(3R)-1-propan-2-ylpyrrolidin-3-yl]benzamide 5-[3,4-dimethyl-2,6-bis(sulfanylidene)cyclohexa-1,3-dien-1-yl]oxy-N-phenylpentane-1-sulfinamide 3-[6-(6-aminopyridin-2-yl)imidazo[1,2-a]pyrazin-8-yl]phenol 6-methyl-N-[5,7-dioxo-4-(2-phenylethyl)octan-3-yl]pyridine-3-carboxamide 4-(azidomethyl)-N'-(2,3-dihydro-1H-inden-5-ylsulfonyl)benzohydrazide N-[4,5-dimethyl-2-phenyldiazenyl-4-(trifluoromethoxy)penta-1,3-dienyl]methanimine 2-bromo-6-[3-(4-hydroxyphenyl)piperazine-1-carbonyl]spiro[cyclohexane-1,5'-imidazo[2,1-c][1,4]benzodiazepine]-11'-one 6-(3,5-dichloropyridin-4-yl)-7-methyl-N-[[1-(1-propan-2-ylazetidin-3-yl)triazol-4-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amine 1-[2-fluoro-3-(trifluoromethyl)phenyl]pentan-1-one 6-[4-ethoxy-3-(trifluoromethyl)phenyl]-2,5-dimethylcyclohepta-1,3,6-triene 1-[4-(azidomethyl)phenyl]-3-[2,4-bis(trifluoromethyl)anilino]pyrrolidin-2-one N-ethenyl-1-[3-(5-methylpyridin-2-yl)phenyl]ethanamine [2-[3,6-bis(4-methylphenyl)carbazol-9-yl]-1-cyanoethenyl]azanium N-[2-hydroxy-1-(3-propan-2-ylphenyl)ethylidene]hydroxylamine 4-(2,5-dimethylphenyl)sulfanyl-3-(7H-purin-6-ylamino)butan-1-ol;hydrochloride 4-[2-(1H-indol-3-yl)ethenyl]benzamide 2-amino-8-[4-(1,3-dioxoisoindole-5-carbonyl)piperazin-1-yl]-7-ethoxy-N,N-dipropyl-10H-1-benzazecine-3-carboxamide;ethane N-(1-azidoimidazol-4-yl)-2-(hydroxyamino)pyridine-3-carboxamide (2R)-4-[(2S,6R)-5-deuteriooxycarbonyl-6-hydroxyoxan-2-yl]oxy-1-(2-fluorophenyl)butane-1,2-dione 5-N,5-N,4-trimethyl-2-[(Z)-1H-pyrrol-3-ylmethylideneamino]furan-3,5-dicarboxamide N-benzyl-2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)propanamide;hydrochloride (3-chloropyridin-4-yl)-[2-(3,5-dimethoxyphenyl)piperazin-1-yl]methanone 5-(3-nitrophenyl)pentacyclo[6.6.6.02,7.09,14.015,20]icosa-1,4,6,8,10,12,15,17,19-nonaene 2-[(3S)-1-(4,6-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-9-hydroxy-1H-purin-6-one 2-[5-(4-bromophenyl)thiophene-3-carbonyl]-N'-methyl-3,4-dihydro-1H-isoquinoline-5-carbohydrazide;ethane 5-[5-(dimethylamino)pyridin-3-yl]-N-[4-fluoro-2-(2,2,2-trifluoroethoxy)phenyl]-1H-indazole-3-carboxamide (5S,7R)-N-(4-fluorophenyl)-7-(3-methoxy-2-prop-2-enylphenyl)-5-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide N-[[4-(methylamino)phenyl]methyl]-3-[2-oxo-8-(trifluoromethyl)chromen-3-yl]propanamide N-[2-(4-chloroanilino)-5-nitrophenyl]acetamide 2-amino-N-[[4-(3,5-difluorophenyl)cyclohexyl]methyl]pyridine-3-carboxamide 3-(2,4-dihydroxyphenyl)-N'-hydroxybenzenecarboximidamide 1-[(4aS,8R)-2-benzylsulfanyl-3,4a,5,7,8,8a-hexahydropyrano[4,3-d][1,3]thiazin-8-yl]propan-1-one ethane;2-[7-(4-fluorophenyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]-N-methylpyridine-3-carboxamide 6-(dichloromethyl)imidazo[1,2-b]pyridazine 3-[(4-azidocyclohexyl)methyl]-5-fluoropyridine 3-[2,3-dichloro-5-(6-methoxypyridin-2-yl)phenyl]propanamide 1-(2,5-diethylphenyl)-3,4-difluoro-9H-fluorene 2-(ethylamino)-4,6-dimethyl-5-[(4-nitrophenyl)hydrazinylidene]pyrimidine-7-carbonitrile [2-(2-hydroxyphenyl)pyridin-3-yl]urea [4-(2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrole-5-carbonyl)-4-phenylpiperidin-1-yl]-[6-methoxy-2-(trifluoromethyl)pyrimidin-4-yl]methanone 1-[3-[(E)-1,1-difluorobut-2-enyl]-4-(4,6-dimethoxypyrimidin-5-yl)phenyl]ethanone N-[4-[(3,5-difluorophenyl)methylamino]butyl]naphthalene-1-carboxamide 1-cyclopropylsulfonyl-2,3-dihydroindole 2-amino-4,6-dibromobenzo[g]quinoline-3-carbonitrile N-(2,6-dibromopyridin-4-yl)-N-methanesulfonamide N-(2,6-difluorophenyl)-4-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]benzamide 3-azidooxy-1,2,4,5-tetrafluoronaphthalene (2R)-2,6-diamino-N-[4-[4-[2-(1,3-thiazol-5-ylmethoxy)ethyl]phenyl]but-1-en-2-yl]hexanamide 6-[4-(3,5-dimethylpyridine-2-carbonyl)piperazin-1-yl]pyridazine-3-carbonitrile [6-[(4,4-dimethylcyclohexyl)amino]-1H-indazole-3-carbonyl]iminoazanium 2-chloro-N'-ethyl-6-hydroxybenzenecarboximidamide N-(5-bromopyridin-2-yl)-N-ethenylsulfonylnonanamide N-methyl-1-[4-(2,3,5,6-tetrafluorophenyl)pyridin-2-yl]ethanamine N-(2-ethoxypyridine-3-carbonyl)-1,3-benzothiazole-5-carboxamide 5-(2,3-difluorophenyl)-4-oxoimidazolidine-1-sulfonate 4-[2,5-diamino-3-(4-chlorophenyl)-6-(trifluoromethyl)pyridin-1-ium-1-yl]benzamide N-[(4-chlorophenyl)methyl]-2-[6-(3-morpholin-4-ylpropoxy)indazol-1-yl]acetamide 4-(2,6-dimethylmorpholine-4-carbonyl)spiro[1H-indole-3,4'-piperidine]-2-one;propane [(1S)-2,2,3,3,4,5,6-heptadeuterio-7-methyl-1-[2,2,2-trifluoro-1-(hydroxymethoxy)ethyl]-9H-fluorene-9-carbonyl]oxidanium 3-[(2S)-1-amino-6-hydroxy-5,5-dimethylhexan-2-yl]oxycarbonylbenzoate 2-[[4-(trifluoromethyl)phenyl]methoxymethyl]piperidine 2-methyl-7,10,10a,11,12a-hexahydro-6aH-indolo[2,3-b]quinolizine 3-fluoro-5-[2-(5-pyrazin-2-yl-1H-indazol-3-yl)-1H-pyrrolo[3,2-c]pyridin-4-yl]phenol 1-cycloheptyl-2,3,3a,4,5,6-hexahydroindole 1-[2-[(3-fluorophenyl)methyl]-4-methoxypyrrolidin-1-yl]-2-(3-methylcyclohexa-1,5-dien-1-yl)ethanone (4R)-1-[(2S,3S)-2-[[(2R)-3-hydroxy-2-[5-[(E)-4-oxopent-2-enyl]thiophen-2-yl]propanoyl]amino]-3-methylpentanoyl]-N-naphthalen-1-yl-4-(phenylcarbamothioylamino)piperidine-2-carboxamide N-[1-(4,6-dimethylpyrimidin-2-yl)pyrazol-3-yl]-5-fluoropyridine-2-carboxamide 1-[(1R,5S)-6-phenylmethoxy-3-azabicyclo[3.2.0]heptan-3-yl]-2-pyrrolidin-1-ylethanone 2,4-dibromo-6-[(E)-[(5-nitropyridin-2-yl)hydrazinylidene]methyl]phenol 2-[5-(3,4-dimethoxyphenyl)-6-ethyl-7-oxofuro[2,3-c]pyridin-2-yl]-N-methylacetamide (2E,4Z)-N,5-dimethylhepta-2,4,6-trien-3-amine;methanol;1-[2-[[4-[5-(trifluoromethoxy)pyridin-2-yl]-1H-indazol-7-yl]oxy]ethyl]pyrrolidine N-benzyl-1,2-dimethoxy-7H-purin-6-imine 4-N-(2-butyl-6,7-dihydro-1H-benzimidazol-5-yl)-5-chloro-2-N-[3-fluoro-4-(piperazin-1-ylmethyl)phenyl]pyrimidine-2,4-diamine 3-[(2R)-2,4-dimethylpentoxy]-4-ethynyl-7-hydroxychromen-2-one 2-(4-azidopiperidin-1-yl)-N,N-diethylpyrimidin-5-amine (E)-2-[2,6-dimethyl-4-(trifluoromethyl)phenyl]-N'-ethylbut-1-ene-1,4-diamine;ethane (1S)-3-[2-[(1S,5R)-7-chloro-6-ethyl-3-azabicyclo[3.1.0]hexan-3-yl]ethyl]-1-methyl-1,4-benzodiazepine 3,5-dichloropyridine;N-[[2-(1H-imidazol-5-yl)acetyl]amino]-2-(5-oxopyrrolidin-3-yl)acetamide 3-N-[(2R)-4-amino-1,5-dioxopentan-2-yl]-5-phenyl-1H-pyrazole-3,4-dicarboxamide;dihydrochloride 4-(2-chlorophenyl)-1-[3-ethoxy-5-(6-methylpyrazin-2-yl)oxyphenyl]butan-1-one;ethane N-[1-(5-ethylsulfonylpyridin-2-yl)propan-2-yl]acetamide 6-(4-aminocyclohexyl)imino-1,3-dihydro-2-benzofuran-5-one (3R,4S)-4-[1-(2,6-dimethylphenyl)piperidin-4-yl]oxypyrrolidine-3-carboxamide 1-N,3-N-bis(2-methoxyethyl)benzene-1,3-diamine 3-[(6R)-2-tert-butyl-7-oxo-4,5,6,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-6-yl]propanamide 5-[2-(4-methylphenyl)ethynyl]pyrimidine [2-(aminomethyl)-4-iodophenyl]boronic acid 6-chloro-4,8-dimethyl-2,3-dihydro-1H-quinoxaline 2-cyclohexylsulfanyl-6-[(3,5-difluorophenyl)methyl]-8-ethylpyrido[2,3-d]pyrimidin-7-one 2-(N-propylanilino)decanoic acid 2-[(1,4-dichloronaphthalene-2-carbonyl)amino]acetic acid 4-[6-(3,5-difluorophenoxy)pyridine-2-carbonyl]morpholine-3-carbonitrile (7-fluoroquinolin-2-yl)-[4-methoxy-1-(pyrazin-2-ylmethyl)piperidin-4-yl]methanol 2-methyl-5,6-bis(2-methylphenyl)-3H-thieno[2,3-d]pyrimidin-4-one [(3R,4S)-1-[(2-chloro-3-fluorophenyl)methyl]-4-hydroxypyrrolidin-3-yl]-piperidin-1-ylmethanone 3-(difluoromethoxy)-4-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]benzoic acid (Z)-N-[3,5-bis(2,4,6-trimethylphenyl)sulfonylpyridin-4-yl]-N'-phenylethene-1,2-diamine [4-(3-propoxypyrrolidin-1-yl)phenyl]azanium N-cyclopentyl-5-[(E)-2-ethenylbut-2-enoxy]pyrimidine-4-carboxamide N-[4-[[2-[(3R)-4-(cyclopropanecarbonyl)-3-methylpiperazine-1-carbonyl]phenyl]sulfamoyl]phenyl]acetamide 3-[2-(5-amino-2-chlorophenyl)ethynyl]-N-cyclopenta-1,4-dien-1-yl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carboxamide 2-[3-ethoxycarbonyl-1,2-dihydroimidazol-5-ylmethylidene]propanedioic acid 3-(dimethylamino)-2,4,6-triiodobenzoic acid 4-[2-methoxy-5-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-2-carboxylic acid 5-(dimethylsulfamoylamino)-6-[1-ethyl-3-(trifluoromethyl)pyrazol-4-yl]oxypyridine-3-carboxamide 5-[4-amino-2-(trifluoromethyl)anilino]-3-bromo-1,2-thiazole-4-carboxylic acid N'-(4-azido-2,5-difluorophenyl)ethane-1,2-diamine 3-[2,4-difluoro-N-(2-methylpropyl)anilino]butanoic acid 2-ethyl-1,4-dimethoxynaphthalene 3-[7-(2,4-dichlorophenyl)-5-methyl-9H-fluoren-1-yl]piperidine 1-(2,4-dichlorophenyl)-7,11,12-trimethyl-3-thia-8,9,11-triazatricyclo[6.3.0.02,6]undeca-1(8),2(6),4,10-tetraene N-[3-(4-cyclohexylbutanoyl)phenyl]-2-methoxypropane-1-sulfonamide 5-[2,6-difluoro-4-(3-methylbutan-2-yloxy)phenyl]-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidine-2,4,7-trithione 2-(1,3-dioxoisoindol-2-yl)-4-methoxy-N-(2H-pyrazolo[3,4-b]pyridin-3-ylimino)butanamide (3-methyloxetan-2-yl)-[4-[[1-methyl-5-[4-(trifluoromethyl)phenoxy]cyclohexa-2,4-dien-1-yl]amino]piperidin-1-yl]methanone 4-(4-methoxyphenyl)sulfanyl-2-methylpyrimidine 3-fluoro-2-(4-propan-2-ylphenyl)quinoline 1-[(E)-3,4-dihydro-2H-naphthalen-1-ylideneamino]-3-[2-methyl-4-(6-morpholin-4-ylpyrimidin-4-yl)oxyphenyl]thiourea 1-(2,5-dioxopyrrolidin-1-yl)oxycarbonylpyrazole-3-carboxylic acid 3-[[(2S)-1,4-dioxan-2-yl]methoxy]-2-hydroxy-6-(N-phenylanilino)benzaldehyde 3-[5-[[2-chloro-4-(trifluoromethyl)phenyl]carbamoylamino]-1H-pyrrol-2-yl]-N,N-diethylbenzamide 2-[4-(4-aminobenzoyl)piperidin-1-yl]-3H-quinazolin-4-one 2-[(E)-3-ethylhex-4-enoxy]naphthalene-1,4-dione 2-(4-ethoxyphenyl)-N',N'-bis[4-methyl-3-(4-propan-2-ylphenyl)phenyl]ethanedithiohydrazide 2-[(7Z)-3,5-bis[(1R)-1-cyclopropylethyl]deca-7,9-dienoyl]benzoic acid 1-[4-(2,5-dimethoxyphenyl)piperazin-1-yl]propan-2-ol N-[(3S)-1-cyclohexyl-4,5-dihydro-2H-pyrrol-3-yl]-6-methoxynaphthalene-2-carboxamide 1-(2,4-dichlorophenyl)sulfinyl-3-[5-methyl-6-[3-methyl-4-(methylideneamino)oxyanilino]pyrimidin-4-yl]urea 5-azido-N-(4,4-difluorocyclohexyl)pyrimidin-2-amine 3-ethenyl-2,4,5-triphenyl-1H-pyrrole 4-[(3S)-1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one 1-(4-chlorobutyl)-3,5-dimethoxybenzene 1-[[2-chloro-4-(cyclopropanecarbonyl)phenyl]methyl]quinazoline-2,4-dione (1R,2S)-N-[8-amino-6-[4-(hydroxymethyl)pyridin-3-yl]isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 2-methyl-6-[(Z)-4,4,4-trifluoro-1-hydroxy-3-(4-iodo-3-oxocyclohexa-1,5-dien-1-yl)but-2-en-2-yl]imidazo[1,2-a]pyridine-8-carbonitrile N-(6-chloro-1,3-benzothiazol-2-yl)-4,5-dimethoxy-2H-thiopyran-2-amine 5-methyl-N-(4-phenylquinazolin-2-yl)cyclohexa-1,5-diene-1-carboxamide N-[3-chloro-5-[methyl(prop-2-enoyl)amino]phenyl]-1,3-thiazole-4-carboxamide 4-(1,3-diethoxypropan-2-ylamino)benzenesulfonamide [3-(cyclopenten-1-yl)-2H-indazol-4-ylidene]hydrazine 6-(2,4,5-trimethylphenoxy)carbonylcycloheptene-1-carboxylic acid (3R,4S)-4-methoxy-1,1-dioxo-N-[[2-[4-(2-phenylethylamino)piperidine-1-carbonyl]phenyl]methyl]thiane-3-carboxamide 2-[(2S)-1-(4-methylphenoxy)propan-2-yl]pyrimidine 2-[4-(2-fluorobenzoyl)piperazin-1-yl]-N-(2H-tetrazol-5-ylmethyl)-6-azaspiro[3.4]octane-7-carboxamide 2-[(7S)-6-[2,6-dimethyl-4-(oxetan-3-yloxy)phenyl]-5,7-dihydropyrrolo[3,4-b]pyrazin-7-yl]acetic acid 6-[2,3-bis(ethenyl)phenyl]hexanoic acid 2-bromo-N-[4-methoxy-5-(naphthalene-1-carbonyl)-1,3-thiazol-2-yl]acetamide N-[(E)-3-hydroxy-4,6-diphenylhex-1-enyl]-2-[2-(trifluoromethoxy)ethoxy]acetamide ethane;7-methoxy-3-methyl-1,4,8,9-tetrahydropyrido[3,2-b]indole 3-[1-methyl-4-(2-phenylethynyl)cyclohexa-2,4-dien-1-yl]propanoic acid 1-(7,8-dihydronaphthalen-2-yl)pent-4-yn-3-one 1-azidooxy-4-[(2,6-dichlorophenyl)methyl]piperidine 2-[1-(3,4-dichlorophenyl)ethoxy]-8-fluoroquinazoline 6-[3-(4-methylpiperidine-1-carbonyl)pyrrolidin-1-yl]pyridine-2-carbonitrile 2-[4-[3,5-dimethyl-1-(oxan-2-yl)pyrazol-4-yl]pyridin-2-yl]phenol (Z)-1,3-bis(4-tert-butylphenyl)prop-2-en-1-one 5-[[4-(dimethylamino)phenyl]methoxy]-2,3-dihydroisoindol-1-one (3S,4R)-1-benzyl-4-(3,5-difluorophenyl)pyrrolidine 4-(dimethylamino)-2-[6-methyl-3,5-bis(trifluoromethyl)pyridin-2-yl]sulfanylacetic acid 4-[2-(hydroxymethyl)phenyl]-3,8a-dihydro-1H-quinolin-2-one 3-[6-(2,4-difluorophenyl)pyridin-3-yl]propanoic acid 6-chloro-2-methyl-4-[(3R)-1-(3,3,3-trifluoropropanoyl)piperidin-3-yl]pyridine-3-carbonitrile 5-[[3,5-dichloro-2-hydroxy-4-(trifluoromethyl)phenyl]methylideneamino]naphthalene-1-sulfonamide 3-(5-chlorothiophen-2-yl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-2-[5-nitro-6-oxo-1-[[2,4,6-tri(propan-2-yl)phenyl]methyl]pyridin-2-yl]prop-2-enamide 6-[3-amino-4-(piperidin-2-yliminomethyl)phenyl]-1,5-dimethyl-7H-pyrrolo[2,3-d]pyridazin-4-one;propane [3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)azetidin-1-yl]-(6-ethoxypyridin-2-yl)methanone 1-[5,6-dimethyl-2-(trifluoromethyl)pyridin-3-yl]butane-2,4-dione (3R,4S)-1-benzyl-4-[2-methoxyethyl(methylsulfonyl)amino]piperidine-3-carboxylic acid 3-aminosulfanyl-4-(6-hydroxyhexoxy)benzoic acid 2-[(1R)-6-oxocyclohexa-2,4-dien-1-yl]benzamide 3-[2,6-di(propan-2-yl)phenyl]-4-hydroxypent-3-en-2-one 1,3-dichloro-2-[(2E)-4-ethylpenta-2,4-dien-2-yl]benzene;ethane 2,2-diphenylethenoxymethylbenzene (3R,4S)-1-ethoxycarbonyl-N-[5-methyl-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]sulfonylpiperidine-3-carboxamide N-[1-[4-[2-chloro-3-(trifluoromethyl)anilino]phthalazin-6-yl]pyrrolidin-3-yl]carbamate 3-(2,2-dichlorocyclopropyl)-2-methoxypyridine 4-[(2Z,4E)-5-oxo-6-thiophen-3-ylhexa-1,4-dien-2-yl]benzaldehyde 1-[2,4-difluoro-3-[6-methyl-5-(1H-pyrazolo[3,4-b]pyridin-3-yl)cyclohexa-1,5-dien-1-yl]oxyphenyl]ethanone 1-(2,3-dihydro-1H-indol-5-yl)-4-[2-fluoro-5-methoxy-6-(2-phenylethynyl)phenyl]butane-1,4-dione 2-[4-(benzimidazole-1-carbonyl)piperidin-1-yl]-N-methylpyridine-3-sulfonamide 1,5-bis[3-(dimethylamino)propyl]pyrazole-4-carboxamide [7-(4-aminobutylcarbamoyl)-2,2-dimethylchromene-6-carbonyl]azanium 3-[2-(1H-indol-4-yl)ethenyl]-N,5-dimethylaniline 6-[[4,5-bis(ethenyl)imidazol-1-yl]methyl]-2-butan-2-yl-3H-quinazolin-4-one N-(2,3-dihydro-1H-inden-5-yl)-4-methoxy-6-oxo-5H-benzo[b][1,4]benzoxazepine-3-carboxamide 3-hydroxy-2,5-diphenylbenzenesulfonic acid N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-N-methyl-5,6-dihydroquinoline-7-carboxamide 5-chloro-6-(trifluoromethyl)spiro[3,4-dihydrochromene-2,4'-piperidine] 7,8-dihydropyrimido[4,5-g][1,3]benzoxazin-2-one 1-[2,4-dimethyl-3-(phenylmethoxycarbonylamino)pentyl]cyclopropane-1-carboxylic acid 3-[(4,6-dimethyl-2-oxopiperidin-3-yl)carbamoyl]-5-[ethanimidoyl(oxan-4-yl)amino]thiophene-2-carboxylic acid 1-[5-(methoxymethyl)oxolan-2-yl]pyrimidine-2,4-dione N-(4,5-dichloropyridin-2-yl)-5-fluoro-1H-indole-7-carboxamide N'-(benzenesulfonyl)benzohydrazide (2R)-1-[4-[2,6-difluoro-N-(3-methylbutanoyl)anilino]-3-methylphenyl]propane-2-sulfonamide N-(2,3-dihydro-1H-inden-1-yl)-2-[4-fluoro-5-(trideuteriomethoxy)pyridin-2-yl]-6-oxo-1H-pyrimidine-4-carboxamide 4-(4-methylphenyl)-3-nitrobenzenethiol (2R)-1-[[3-bromo-5-methyl-6-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]methyl]-N'-hydroxy-4-oxo-1,8-naphthyridine-2-carboximidamide 3-(N-tert-butyl-2,4,6-trichloroanilino)propane-1,2-diol 2-[(6-chloropyridin-3-yl)-(2,4-dichloropyrimidin-5-yl)amino]-2-methylpropanoic acid 3-ethyl-2,6-dimethoxy-4-(5-oxo-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-4-yl)benzenesulfonic acid 3-methylsulfonylbenzamide;propane 1-[[5-(cyclohexylmethylamino)-4-propanoylthiophen-3-yl]methyl]pyrazole-3-carboxylic acid N-benzyl-4-(2,6-difluorophenyl)piperidine-1-carboxamide 3-[7-(2,4-dichlorophenyl)-5-methyl-2-oxo-1,3-oxazepane-3-carbonyl]piperidine-1-carboxylic acid (4S)-4-[3-[3,5-bis(trifluoromethyl)phenyl]propanoylamino]pyrrolidine-2-carboxylic acid 6-[4-(dimethylamino)butyl]-2,3,8-trifluoro-10H-acridin-9-one;hydrochloride N-[(E)-6,6-dimethylhept-3-enyl]-4-ethylbenzamide N-(4,5,6-trimethylpyrimidin-2-yl)acetamide 2-[[(3S)-oxolane-3-carbonyl]amino]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxylic acid (2S,3R,4S)-1-[5-cyano-7-cyclopropylimino-9-[(2-fluorophenyl)methyl]-6-[4-methoxy-3-(trifluoromethyl)anilino]pyrazolo[1,5-a][1,3,5]triazin-2-yl]-N,N-diethyl-4-hydroxypyrrolidine-3-carboxamide N-(3,4-dihydro-2H-pyran-6-yl)-2-hydroxy-1,2-benzothiazol-5-imine (6R,7S)-6-hydroxy-7-[(2S)-4-(2-methylphenoxy)butan-2-yl]oxyoxepane-3,4-dione (2S)-1-acetyl-N-[(3R,5S)-5-amino-4,6-dioxoheptan-3-yl]-2,3-dihydroindole-2-carboxamide N-[5-(2,6-dimethylmorpholine-4-carbonyl)pyridin-2-yl]-2-phenylacetamide (3aR,7aS)-2-[6-[2-hydroxyethyl(methylsulfonyl)amino]pyridin-3-yl]-N-(1H-indazol-5-yl)-1,3,4,6,7,7a-hexahydropyrano[3,4-c]pyrrole-3a-carboxamide (3S,4R)-1-[1-[4-(dimethylamino)phenyl]piperidine-4-carbonyl]-N-(oxan-2-yloxy)-4-[[4-(trifluoromethoxy)benzoyl]amino]pyrrolidine-3-carboxamide 1-[4-(3,5-dimethylphenoxy)butyl]-2-oxopyridine-3-carboxylic acid 4-[2,3-bis(ethenyl)phenyl]-6,7-dichloroquinazoline;5-cyclohexa-1,3-diene-1-thiol 7-chloro-1-methyl-3-phenyl-6,8,9,10-tetrahydro-5H-cycloocta[b]pyridine 6-chloro-N-[4-[(3S)-1-methylpyrrolidine-3-carbonyl]phenyl]imidazo[1,2-a]pyridine-8-carboxamide (1E,3Z)-4-[2-(7-methyl-1H-indol-5-yl)ethynyl]hexa-1,3,5-trien-1-amine 6-[1,4-di(propan-2-yl)pyridin-1-ium-3-yl]naphthalene-2,7-disulfonate;manganese(3+);propan-2-one [2-(1-cyanopropan-2-yl)pyridin-4-yl]methanesulfonate 2-(5-ethylpyrimidin-2-yl)oxy-N'-hydroxy-6-methylpyridine-4-carboximidamide (NE)-N-[1-(2,5-dimethoxyphenyl)-3-[4-[(5,7-dimethylcyclohepta-1,6-dien-1-yl)methyl]piperazin-1-yl]propan-2-ylidene]hydroxylamine;ethane 1-[(3S)-1-[2-[6-(hydroxymethyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-3-yl]acetyl]piperidin-3-yl]pyrrolidin-2-one 5-[4-[2-(methylamino)ethyl]phenyl]thiophene-3-carboxylic acid (3R,4S)-1-[4-cyano-2,6-di(propan-2-yl)phenyl]-N-methyl-4-(trifluoromethoxy)piperidine-3-carboxamide 4-[2-[(3R)-piperidin-3-yl]ethyl]benzenesulfonamide 1-[1-(3-fluorophenyl)propyl]-5H-pyrazolo[4,3-d]pyrimidin-7-one 5-[4-fluoro-3-(4-pyridin-3-yl-1H-benzimidazol-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]-N-propan-2-ylidenepyridine-3-carboxamide [4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonylamino)phenyl]carbamic acid 3-methyl-7-[(4Z)-2,3,5-trimethylideneocta-4,7-dienoxy]-1H-quinoxalin-2-one 6-N,2-dimethyl-5-pyridin-2-yl-4H-pyrrolo[3,2-d]pyrimidine [4-(6H-benzotriazol-1-yl)phenyl]methylphosphonic acid N-(4,6-diamino-1,3,5-triazin-2-yl)acetamide 1-(4-chlorophenyl)sulfinyl-2-ethyl-3,4-dihydro-2H-quinoline 2-[6-ethenyl-3,4-dimethoxy-5-(piperazine-1-carbonyl)pyridin-2-yl]-5,7-difluoro-3H-isoindol-1-one 2-(N-acetyl-4-fluoroanilino)acetamide (E)-3-[4-ethenyl-5-methylidene-1-phenyl-2-propan-2-ylpyrrol-3-yl]-N-[(2-fluoro-6-methoxyphenyl)methyl]prop-2-enamide 3-(1,2,4-oxadiazol-5-yl)-6H-benzo[c]chromen-8-ol 2-cyclohexyl-5,7-dimethoxy-3H-quinazolin-4-one 2-[2-azidooxy-1-(4-ethylphenyl)propan-2-yl]phenol 2-chloro-N-(4-methoxyphenyl)-5-nitropyrimidin-4-amine (2S)-2-[8-[4-[(7-chloroquinolin-4-yl)amino]butoxy]-6-methoxy-3H-quinazolin-5-ium-4-ylidene]propanal 5-azidooxy-3-tert-butyl-1H-indole 5-(3,3a,4,6a-tetrahydro-1H-furo[2,3-c]pyrrole-2-carbonyl)pyridine-2-carboxamide;dihydrochloride N-[1-(5-chloropyridin-3-yl)ethenyl]-1,7-naphthyridin-2-amine 1-(2,6-dimethylpyridin-4-yl)-3-(oxan-4-yl)imidazolidine-2,4-dione 1-methylsulfanyl-4-(2,2,3,5,5-pentafluoropentoxy)benzene ethane;1-[4-fluoro-3-(trifluoromethyl)phenyl]sulfanyl-N,2-dimethylindole-6-carboxamide 2,6-ditert-butyl-4-(3H-furan-2-ylidenemethyl)phenol 5-cyclopropyl-4-[7-(trifluoromethoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidine 5-chloro-N'-(1,4-dimethylpiperidin-3-yl)sulfanylpyridine-2-carboximidamide 3-[(1R,4S)-2-carboxy-6-oxocyclohexyl]benzoic acid 1-[4-chloro-5-(methylideneamino)-2-(trifluoromethyl)phenyl]ethanone N-[6-(methylamino)pyridin-2-yl]sulfonyl-6-[3-(1,3-oxazolidin-3-ylsulfanylamino)phenyl]-2-propan-2-ylpyridine-4-carboxamide (2-ethoxy-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl)-[(3R,4S)-1-methyl-4-thiophen-3-ylpyrrolidin-3-yl]methanone 4-[2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)ethynyl]cyclohexan-1-ol 2-[(1R)-3,4-dihydro-1H-isochromen-1-yl]-6-fluorophenol N-[1-(3,5-dimethylphenyl)ethenyl]-4-(5,6-dimethylcyclohexa-2,4-dien-1-yl)aniline 4-[[4,5-bis(ethenyl)-6-methylidenepyridine-3-carbonyl]amino]benzoic acid;methanethiol 4-[[2,4-bis(trifluoromethyl)phenyl]sulfonylamino]-N-(1,4,5,6-tetrahydropyrimidin-2-yl)benzamide N-[5-(2-hydroxypropan-2-yl)pyridin-3-yl]acetamide N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]-3-nitrobenzenesulfonamide 4-(2-ethenylsulfonylphenyl)-6,7-dimethoxyquinazoline 2-[6-tert-butyl-4-[(2E,3Z)-2-ethylidenehexa-3,5-dienoxy]cyclohepta-1,3,5-trien-1-yl]-N'-methyl-1H-indole-6-carboximidamide N-[4-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-1H-pyrazol-5-yl]-2-chlorobenzamide 4-(2,3,5,6-tetrafluorophenoxy)benzaldehyde (5Z)-2-[3-chloro-4-(trifluoromethoxy)phenyl]imino-5-[[3,5-dibromo-2-hydroxy-6-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidin-4-one 2-[N-(4-bromobutan-2-yl)-4,5-dimethyl-2-phenyldiazenylanilino]benzenesulfonic acid 4-[5-(azidomethyl)-6-(5,6,7,8-tetrahydronaphthalen-1-yloxy)pyridin-3-yl]morpholine (5Z)-2-[2,6-dimethyl-4-(3-piperidin-1-ylpropoxy)phenyl]imino-5-[(3-hydroxyphenyl)methylidene]-1,3-thiazolidin-4-one N-methyl-1-[3-(4-pentan-2-ylphenoxy)propoxy]ethanamine 1-(4,5-dichlorocyclohexa-2,4-dien-1-yl)sulfonyl-N-[4-[2-[3-[(2S)-6,15-dibromo-13-chloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl]piperidine-1-carbonyl]pyrrolidin-1-yl]-4-oxobutyl]piperidine-4-carboxamide 6-N-[4-(trifluoromethoxy)phenyl]pyrimidine-2,5,6-triamine 4-[(4E,5Z)-2,6-dimethylhepta-1,3,5-trien-4-yl]-2-ethynylpyridine N-(2-aminophenyl)-4,4,5,6-tetrahydro-1H-cyclopenta[b]pyrrole-3-carboxamide 2-[3,4-bis(9H-fluoren-1-yl)phenyl]ethanamine (3R,4S)-1-[2-(cyclobutylmethoxy)ethyl]-4-[1-[2-(trifluoromethoxy)phenyl]piperidin-4-yl]pyrrolidine-3-carboxylic acid 2-[2,6-dichloro-N-(3-methylbut-2-enyl)-4-nitroanilino]acetamide 4-(2,6-dimethylphenoxy)-3-fluorobenzamide 7-(4-ethoxyphenyl)-3-[(2E,4Z)-hepta-2,4,6-trien-2-yl]-1H-quinoline-2,4-dione 1-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1]benzazepin-11-yl)-3-propan-2-yloxypropan-2-ol 3-methyl-7-pyridin-2-yl-4H-pyrazolo[1,5-a]pyrimidine-5-carboxylic acid 1-azidooxynaphthalene-2,6-disulfonic acid 2-[4-(benzylamino)-6,7-dihydroquinazolin-2-yl]phenol 3-(2,4-dimethylphenyl)-1-iodopyrrolidine 2-[2-(4-cyclopropylphenyl)ethynyl]-5,6-dimethoxy-1H-indole N-[4-[(E)-2-[5-[1-(cyclohexylmethoxyamino)propan-2-yl]pyridin-3-yl]ethenyl]phenyl]sulfanylacetamide 2-bromo-3,4,5-trimethoxyaniline 2-ethyl-8,9-difluoro-1,4,5,6-tetrahydrothiopyrano[3,4-b]indole 6-amino-7-[(2,4-dichlorophenyl)methylamino]-3H-quinazolin-4-one 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethanol 2-[4-bromobutan-2-yl(1,3-thiazol-5-yl)amino]benzenesulfonic acid 7-amino-6,8-difluoro-4-oxo-1H-quinoline-3-carboxylic acid N-[1-(2,4-dichloropyrimidin-5-yl)sulfanylethenyl]hydroxylamine 4-[N-(2,3-dihydroxypropyl)anilino]benzenesulfonic acid 1-[7-(2,4-dichlorophenyl)-5-methyl-6H-[1,3]thiazolo[5,4-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide 1-[4-(6,8-dichlorospiro[3H-quinazoline-2,4'-piperidine]-4-yl)oxyphenyl]ethanone 3-bromo-N-[1-(3,4-dimethoxyphenyl)cyclopropyl]quinoline-2-carboxamide 2-(4,6-dimethoxypyridin-3-yl)pyridine-4-carboxamide 2-[(2S)-4-azidomorpholin-2-yl]-5,6-dihydrothieno[3,2-d]pyrimidine 2-[8-methylsulfonyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)-6H-benzo[c]chromen-9-yl]acetamide 3-amino-6-(4-fluorobenzoyl)-1H-pyridazin-5-one 3-[(3,5-dibromophenyl)methyl]-1-propan-2-ylpiperazine 7-chloro-5,6-dihydroindeno[1,2-b]quinoline 2-chloro-4-[(E)-[[6-[3-ethoxy-5-(methanesulfonamido)phenyl]-4-oxoquinazolin-3-yl]-hydroxymethylidene]amino]oxybenzoic acid N-[4-(cyclopropanecarbonyl)-2,6-dimethylphenyl]-2-(4-fluorophenyl)piperidine-1-carboxamide 1-(3,4-dichlorophenyl)-5-[5-(3-hydroxypyrrolidine-1-carbonyl)thiophen-2-yl]pyrazole-3-carbonitrile 2-(N-(4-nitrobenzoyl)anilino)benzenesulfonic acid 7-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-1,2,8-trifluoro-3-propylnaphthalene 1-benzyl-N-(3,4,5-trichlorophenyl)pyrrole-3-carboxamide (5S)-N-(1,3-benzothiazol-2-ylmethylidene)-6-oxo-2-propan-2-ylidene-4,5-dihydro-1H-pyrimidine-5-carboxamide 5-N,8-N-dimethylnaphthalene-2,7-diamine 2-[(6,8-dimethoxyquinazolin-4-yl)amino]-N-[2-hydroxyethyl(methyl)carbamoyl]-1H-benzimidazole-5-carboxamide N-methyl-3-oxo-N-[(3,4,5-trifluorophenyl)methyl]piperazine-1-carboxamide [1-[2,4-di(propan-2-yl)phenyl]pyrrolidin-3-ylidene]cyanamide 6-chloro-5-[3-(4-cyclobutylpiperazine-1-carbonyl)azetidin-1-yl]pyridine-2-carbonitrile (5S)-3-ethyl-5-[2-[4-(trifluoromethylsulfonyloxy)phenyl]propan-2-yl]pyrrolidine N-cyclopropyl-2-[3-[4-methoxy-6-(trifluoromethyl)pyridin-3-yl]-1,1-dioxothietan-3-yl]acetamide 2-(4-methoxyphenyl)-N-[(1R)-6-nitro-4,9-dioxo-3H-indeno[5,11b]pyrazin-2-yl]acetamide 2-[2-(3,4-dimethoxyphenyl)morpholin-4-yl]-N-[1-(4-hydroxycyclohexa-1,3-dien-5-yn-1-yl)ethyl]acetamide 1-cyclobutyl-3-[(5S,7R)-5-[4-(2-hydroxyethoxy)phenyl]-9-oxa-2-azaspiro[4.6]undecan-7-yl]propan-1-one (4R)-6-chloro-8-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-ylidene]-4-propan-2-yloxy-3,4-dihydro-2H-chromene;hydrochloride 2,3-diamino-5-[4-[(2-fluorophenyl)methoxy]phenyl]benzoic acid 5-(4,6-difluoro-3-methoxy-2H-1,3-benzothiazol-7-yl)-1-methanimidoylnaphthalen-2-amine 2-[(5-chloroquinoline-8-carbonyl)amino]-4,6-difluorobenzoic acid;1-[6-oxo-5-(2-phenylethynyl)pyridazin-1-yl]-3-[2-(trifluoromethoxy)phenyl]urea 3,5-difluoro-N-[2-[methyl(pyridin-4-yl)amino]ethyl]pyridine-4-carboxamide (5S,7R)-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-5,7-dimethyl-1,4,5,7-tetrahydropyrano[3,4-c]pyrazole-3-carboxamide ethane;1-[4-[(2E,4Z)-hexa-2,4-dien-3-yl]phenyl]ethanone N-[2-[4-(4,5-dihydroimidazol-1-yl)phenyl]ethyl]-3-(trifluoromethyl)benzamide (4R)-1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-4-phenyl-3-thiophen-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 2-[1-acetyl-4-(7-fluoro-5-methyl-1H-indole-2-carbonyl)piperazin-2-yl]-N,N-dimethylacetamide 5-(cyclohexylmethyl)-3-[6-(trifluoromethyl)pyridin-2-yl]imidazolidine-2,4-dione N-[4-(1,3-benzodioxol-5-ylmethylsulfonyl)phenyl]-3-morpholin-4-ylpropanamide 5-(azidomethyl)-N-methoxy-2,3-dihydroindole-1-carboxamide 3-[4-[(2,6-dichlorobenzoyl)amino]phenyl]-2-methoxypropanoic acid 2-[3-(2-chlorophenyl)propanoyl]cyclopentane-1,3-dione 2-[1-(3,5-dimethylbenzotriazol-4-yl)isoquinolin-6-yl]-8-[5-isocyano-4-phenyl-2-(4-isocyanophenyl)-1H-imidazol-5-yl]-[1]benzofuro[2,3-b]pyridine 6-methoxy-4-[(1S)-1-[4-[5-methyl-4-(2,2,2-trifluoroethylamino)pyridin-3-yl]phenyl]ethyl]phthalazin-1-amine 4-(4-tert-butylphenyl)sulfanyl-3,5-dimethoxy-N'-[(E)-1-pyridin-2-ylethylideneamino]benzenecarboximidamide 1-[2,5-difluoro-4-(4-methylphenyl)phenyl]-N,N-diethylpiperidine-3-carboxamide 6-[7,10a-dihydrobenzo[b]fluoren-5-yl(methoxy)phosphoryl]-2-methylidenecyclohexan-1-one 2-methylsulfinyloxypyridine-3-carboxylic acid 2-(1,3-benzodioxol-5-yl)-6,7-dimethoxy-3,4-dihydro-2H-chromene;hydrate (2S,4R)-1-[2-chloro-3-[(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)oxy]benzoyl]-N-methoxypiperidine-4-carboxamide (3S)-5,7,10-trimethyl-3-phenyl-2H-phenazin-1-one 7-bromo-6-chloro-4H-1,3-benzodioxine 4-(3,6-difluorocarbazol-9-yl)-5,6-dimethylhexanoic acid 3-[[8-chloro-6-(2-hydroxyphenyl)imidazo[1,5-a]pyridin-3-yl]methoxy]pyrrolidine-1-carboxylic acid 2-[1,3-benzodioxol-5-ylmethoxyimino-(2-hydroxyphenyl)methyl]phenol 4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)benzoic acid N-cyclohexyl-4-[1-(3,5-difluorophenyl)cyclopentanecarbonyl]piperazine-1-carboxamide 1-[3-azidooxy-4-ethylsulfonyl-2,6-di(propan-2-yl)phenyl]-9H-fluorene 1-[4-azidooxy-3,5-di(propan-2-yl)phenyl]-2,2-bis(4-chlorophenyl)ethane-1,1-diol 5-(furan-2-yl)-N'-hydroxypyrazine-2-carboximidamide 4-(5-methylsulfanyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-8H-carbazole-7-carboxamide (2R)-6-[5-chloro-3,7a-dimethyl-4-oxo-6-(trifluoromethoxy)indol-1-yl]-N-formyl-4-oxo-N-propan-2-ylhexanamide 4-[(2,6-dichlorobenzoyl)amino]-N-ethylpiperidine-1-carboxamide;2,2,2-trifluoroacetic acid 5-hydroxy-3-(3-methyl-4-nitrophenyl)-2H-pyrazolo[3,4-d]pyrimidine-4-thione 3-(2,5-dioxo-4-sulfanylpyrrolidin-1-yl)naphthalene-2-sulfonic acid 1-[2,6-difluoro-4-(4-fluorophenyl)sulfanylphenyl]ethanone 2-[2-(3,4-dimethoxyphenyl)-1H-imidazol-5-yl]-N-ethylethanamine 2-[4-(1,3-benzodioxol-5-ylsulfonylamino)-N-ethylanilino]-N-(1H-indol-6-ylmethyl)acetamide 5-[2-[4-(1,3-benzoxazol-2-ylmethoxy)phenyl]ethyl]pyrimidine-4,6-diamine 4-[1-[(2S)-3,5-dioxopyrrolidine-2-carbonyl]piperidin-4-yl]oxybenzonitrile 5-[4-(6-methoxypyridin-3-yl)phenyl]sulfonyl-2,5-diazaspiro[3.4]octane (3R)-1-[2,6-dichloro-4-[1-(dimethylamino)ethenyl]phenyl]-N-[5-fluoro-4-(7-fluoro-2-hydroxy-1H-indol-4-yl)pyridin-2-yl]piperidine-3-carboxamide 2-[2-amino-3-(4-chlorophenyl)benzenecarboximidoyl]sulfanylacetic acid 1-(3,4-dimethoxyphenyl)sulfonylpiperidine 2-[2-(6,7-dihydrobenzo[d][1]benzazepin-5-yl)ethyl]isoindole 1-(6-methyl-5-pentanoylpyridin-2-yl)cyclopropane-1-carboxamide N-[(2S)-1-amino-3-methyl-1-oxobutan-2-yl]-1,3-difluoro-5-propanoylpyrazole-4-carboxamide 1-(3,3-dichloroprop-2-enoxy)ethenylbenzene N-(2,6-dioxopiperidin-3-yl)-4-[3-(methoxymethyl)pentanoyl]benzenesulfinamide 1,3-dihydrobenzo[b][1,4]benzothiazepine 3-(2-hydroxy-4,6-dimethylphenyl)-1,2-oxazol-5-ol 2-[(1S,5R)-3-azabicyclo[3.1.0]hexan-6-yl]-6-pyridin-4-ylpyrimidine-4-carboxamide N-azido-6-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-2-amine 4-cyclopentyloxy-N,6-dimethoxyquinazolin-7-amine;piperidine 6-[(3,4-dimethoxyphenyl)methyl]-1H-indazole 4-hydroxy-3,5-dimethoxy-2-(1H-indol-2-yl)-6-phenylbenzenesulfonamide N-[(4,5-dichloro-1H-benzimidazol-2-yl)methoxy]formamide N-(azidomethyl)-1,3-diethylimidazol-1-ium-2-carboxamide (3aR,6aS)-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-5-pyridin-3-yl-3,3a,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-4-one N-(4-methylpyrimidin-2-yl)-N-phenylmethanesulfonamide 2-[(4-benzylpiperazin-1-yl)methyl]-3-ethyl-6,7-dihydrothieno[3,2-c]pyridine N-[1-[5-[3,5-bis(trifluoromethyl)phenyl]-3,4-dihydropyrazole-2-carbonyl]piperidin-4-yl]-2-phenylacetamide 4-[1-(5-methylthiophen-2-yl)ethyl]morpholine 3-[2,4-dimethyl-1-(2-piperidin-1-ylethoxy)benzimidazol-5-yl]sulfanylpropanenitrile 6-(1,2-dihydropyrazin-3-yl)-N-methylpyridine-2-carboxamide [(2R)-4-[3,5-bis(trifluoromethyl)phenyl]-1-[[3-tert-butyl-5-[hydroxy-[6-(methoxymethyl)quinolin-8-yl]sulfanylamino]-2-methylphenyl]methyl-methylcarbamoyl]pyrrolidine-2-carbonyl]oxidanium 2-[3-(1,4-dimethylbenzotriazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-N-(4-fluorophenyl)acetamide 4-(4,5-dimethylpyrimidine-2-carbonyl)-N-[3-(4-ethyl-6-oxo-1H-pyrimidin-2-yl)phenyl]piperazine-1-carboxamide 4-(2,3-dihydro-1H-inden-5-yl)-N-[[(2S)-oxolan-2-yl]methoxy]pyrimidine-5-carboxamide [(4R,5S)-1-[2,6-dimethoxy-4-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl]-3,8-bis(trifluoromethyl)-6-azabicyclo[3.2.0]heptan-6-yl]methanesulfinate 2-(8,14,22-trioxa-1-borahexacyclo[11.7.1.13,19.02,7.09,21.015,20]docosa-2,4,6,9(21),10,12,15(20),16,18-nonaen-5-yloxy)pyrimidine 2-(2,3-dihydroxyphenyl)cyclopentane-1-carboxylic acid (2S,4R)-N-hydroxy-1-[(5S)-3-phenylmethoxy-6-azabicyclo[3.2.0]heptane-6-carbonyl]-4-propylpyrrolidine-2-carboxamide N-[4-(2,4-difluorophenyl)oxan-4-yl]methanesulfonamide 2-azido-4,6-bis(methylsulfonyl)pyrimidine 3-(4,5-dimethoxy-2-methylphenyl)-1H-pyrazole 3-[4-(4-methylphenyl)piperazin-1-ium-1-ylidene]propane-1,2-diamine;4-phenylmethoxybenzaldehyde 3-[2-(2-methoxyethylimino)-5,6,7,8-tetrahydro-1H-quinazolin-4-yl]-N,N-dimethylaniline 4-bromo-6-[[2-chloro-5-(trifluoromethyl)phenyl]iminomethyl]benzene-1,3-diol 2-(5-cyclopropylpyrimidin-4-yl)-N-[2-hydroxy-3-[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]acetamide [4-(7H-pyrrolo[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]-[(4S)-4-thiophen-3-ylcyclohexyl]methanone (7S)-5-(4-chlorophenyl)-3-[(3R)-1-propanoylpiperidin-3-yl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one 2-[4-(1H-indazol-5-ylamino)piperidin-1-yl]acetaldehyde 1-(4-methoxyphenyl)-3,6,7,8-tetrahydro-2H-cyclopenta[e]indole 1-(3,5-dichlorophenyl)-N-[2-methyl-4-(phenylsulfamoyl)phenyl]-6-oxopiperidine-3-carboxamide N-(1,3-benzodioxol-5-yl)-7-[[2-(4-chlorophenyl)cyclopropen-1-yl]methoxy]-1H-indole-6-carboxamide 2-(N-cyclohexyl-4-nitroanilino)acetonitrile 4-[7-(dimethylamino)-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]bicyclo[2.2.2]octane-1-carboxylic acid N-[3-(4-propan-2-ylphenyl)pyrazin-2-yl]acetamide (2S)-N-[(Z)-(4,5-diphenylfuran-2-yl)methylideneamino]-3-methoxy-1-naphthalen-2-ylsulfonylpyrrolidine-2-carboxamide N-(3,4-dimethylphenyl)-1,2,4-triazol-4-amine;6-propoxy-3H-quinazolin-4-one [2-methyl-3-(3,5,6-trimethylpyrazin-2-yl)oxyphenyl]boronic acid ethane;5-[2-(6-methylpyrazin-2-yl)propan-2-yl]pentanenitrile N-(2,3-dihydro-1H-inden-5-yl)-4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidine-3-carboxamide (4-butoxyphenyl)sulfanylazanide (2S,6R)-4-[5-fluoro-7-methoxy-3-[6-methyl-1-[(4-propan-2-ylphenyl)methyl]indazol-4-yl]quinoxalin-2-yl]-2,6-dimethylmorpholine N-[4-(cyclohexylcarbamoyl)phenyl]propanamide 2-(3,5-dimethylphenyl)pentanethioamide N-[3-(4-chlorophenoxy)phenyl]-6-(2-propoxyethyl)-7-(1,3-thiazol-5-ylmethylsulfanyl)-2H-pyrrolo[3,2-d]pyrimidin-4-amine 5-[4,6-bis(difluoromethoxy)-1,3,5-triazin-2-yl]-N-tert-butylthieno[3,2-b]thiophene-2-sulfonamide 2-cyclohexyloxy-4-[(E)-[[4-(3,5-dimethylpyrazol-1-yl)benzoyl]hydrazinylidene]methyl]benzoic acid 4-(1H-indol-3-ylmethylamino)thieno[2,3-d]pyrimidine-5-carboxylic acid N-butyl-4-[[2-(N'-hydroxycarbamimidoyl)phenyl]methoxy]-1,5-dimethylpyrazole-3-carboxamide 1-butyl-3-[4-[2-(6,8-dichloro-4-oxochromen-3-yl)-5-methoxy-3-methylphenoxy]butyl]thiourea 2-[4-cyano-3-(trifluoromethyl)phenyl]-8-(cyclobutanecarbonyl)-N,N-dimethyl-2,8-diazaspiro[4.5]decane-4-carboxamide N-[5-[(3E)-hexa-1,3,5-trien-3-yl]sulfanyl-3-phenylsulfanylpyridin-2-yl]acetamide 3-[4-(hydroxycarbamoyl)-2,6-dimethylphenoxy]-N-[1-(6-hydroxynaphthalen-2-yl)ethyl]pyrrolidine-2-carboxamide 2-N,6-N-diphenylphenanthrene-2,6-diamine 2-bromo-N-(3-methylbutoxy)aniline 2-(1-fluoroethenyl)-6-[5-methyl-3-(trideuteriomethyl)-4H-1,3-oxazol-5-yl]aniline [2-methyl-4,5-bis(phenylmethoxy)phenyl]boronic acid 4-(4,4a,8a-dihydroquinoline-2-carbonyl)-3H-1,3-thiazol-2-one 2-[1-methyl-6-(3,4,5-trifluorophenyl)pyrazolo[3,4-b]pyridin-4-yl]oxyacetic acid [5-[4-(1H-indol-3-yl)phenyl]pyrimidin-2-yl]azanium 2-amino-3-phenylbenzene-1,4-disulfonic acid 5-chloro-1-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]indole-2-carbonitrile;1-N'-(2-chlorophenyl)ethane-1,1-diamine 1-[[4-(4-propan-2-ylpiperazin-1-yl)sulfonylphenyl]methyl]-3H-indol-2-one 2-(2,6-dimethylpyridin-4-yl)-1-ethoxy-N-[3-fluoro-5-(1H-indole-2-carbonyl)phenyl]indolizine-6-carboxamide 5-(3,4-dihydro-2H-chromen-6-yl)-N-[(Z)-1-(methylideneamino)prop-1-enyl]cyclooctane-1-sulfonamide 2-[N-hexyl-4-(thiophene-3-carbonyl)anilino]octanoic acid 6-(2,5-dimethyl-3,4-dihydro-1H-pyrido[4,3-b]indole-8-carbonyl)-1-cyclobutyl-5-(1-oxo-7-propan-2-yloxy-6,7-dihydro-2H-isoquinolin-6-yl)pyridin-2-one 4-[2-(methylamino)ethyl]-N-phenylpiperidine-1-carboxamide 4-[2,5-bis(ethoxymethyl)phenyl]butanal 2-(1H-indol-4-ylmethylamino)pyrimidine-5-carboxylic acid 5-chloro-N-[(1R,2S)-2-ethylcyclopropyl]pyrimidin-4-amine 7-(3-fluorophenyl)-2,4-dimethyl-8H-pyrido[2,3-d]pyrimidine 4-(5-azidopyridin-2-yl)piperazine-1-carboxylic acid 3-[2-(aminomethyl)pyrimidin-5-yl]oxy-N-azidobenzamide 4-(1,3-benzothiazol-2-yl)cyclohexa-1,5-diene-1-thiol 1-[3-(dimethylamino)-2,6-dioxopiperidin-3-yl]pyrrole-2-carboxamide;5-(4,5-dihydro-1H-imidazol-2-ylamino)-2-hydroxybenzoic acid [1-(3,4-dichlorophenyl)pyrrol-2-yl]-(3,3-dimethyl-6-morpholin-4-ylazepan-1-yl)methanone 1-(4-azidophenyl)sulfonyl-2,3,4,9-tetrahydro-1H-carbazole N-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butyl]tricyclo[4.3.0.02,4]nona-1,4,6,8-tetraene-7-carboxamide 7-bromo-6-chloroisoquinoline-3,4-diamine 3-[5-(dimethoxyphosphorylmethylamino)pyridin-2-yl]-1H-inden-4-ol 5-[(3S)-1-(4-chlorophenyl)sulfonylpiperidin-3-yl]-1,2-oxazole 1-[(2E,3Z)-3-ethylidene-4-methylhepta-2,5-dienyl]-N-methylcyclohexa-2,4-diene-1-carboxamide;(3Z)-penta-1,3-diene 2-methyl-4-[[[6-oxo-1-(pyridin-3-yloxymethyl)pyridazin-4-yl]amino]methyl]benzonitrile 2-[4-chloro-N-(5-nitro-1,3-thiazol-2-yl)anilino]propanoic acid 5-[2-(2,3-dihydroindole-1-carbonyl)cyclopropyl]-1H-imidazole-4-carboxylic acid [2-amino-5-[(Z)-1,3-diaminopent-1-en-4-ynyl]phenyl]methanol 1-(4,6-dimethoxypyrimidin-2-yl)pyrazole-3-carboxylic acid 1-[(4-bromophenyl)methyl]-N-ethylpiperidine-2-carboxamide 2-[2,4,6-tris(3-methylbutyl)phenoxy]acetic acid 6,7-dihydroxynaphthalene-2-sulfonic acid 4-chloro-1,2-dimethoxyphenanthrene N-(4,5-dimethoxy-2-propan-2-ylphenyl)-6,7-bis[4-(trifluoromethyl)anilino]quinazoline-2-carboxamide N-cyclopropyl-4-methyl-2-(3,4,5-triethoxyphenyl)butanamide 2-[[5-(3,4-dichlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-quinazolin-4-one 7-[4-(difluoromethoxy)cyclohexyl]-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine 2-[(2Z)-4,6-diphenylhepta-2,6-dienyl]phenol N-[(1R,3S)-3-[benzylcarbamoyl-[(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethylamino)methyl]amino]cyclohexyl]oxolane-2-carboxamide;dihydrochloride 1-(3,5-dimethoxyphenyl)sulfonyl-4-piperazin-1-ylpyrrolo[2,3-b]pyridine;ethane N-[2-[5-cyano-6-(methylamino)pyrimidin-4-yl]oxyphenyl]acetamide 1-(6,7,8,9-tetrahydrodibenzofuran-3-yl)ethanimine 4-amino-2,6-dichloro-N-[(1R)-1-phenylethyl]pyrimidine-5-carboxamide 2-[3,6-bis(aminomethyl)-4-benzyl-2H-quinazolin-1-yl]acetic acid N-[(2S)-1-[4-(3,4-dichlorophenyl)piperidin-1-yl]propan-2-yl]acetamide 3-[2,2-diethoxyethyl(3-methylbutyl)amino]phenol 3-(4-butanoyloxyphenyl)propyl-trimethylazanium 2-[3-[4-(1,3-benzoxazol-2-yl)phenyl]imidazo[4,5-b]pyrazin-2-yl]sulfanylacetic acid 1-(5-fluoro-2,3-dihydroindol-1-yl)-2-[4-[6-[4-(4H-pyrazol-3-yl)anilino]pyridin-2-yl]phenyl]ethanone 1-[[2,5-difluoro-4-(triazol-2-yl)phenyl]methylamino]ethanol 2-(4-chlorophenyl)-6,7,8,9-tetrahydro-[1]benzothiolo[3,2-d]pyrimidine 1-bromo-4-[(E)-2,3-dimethylbut-1-enyl]benzene;propane 2-[5-[5-(3,4-dichlorophenyl)pyridin-2-yl]tetrazol-1-yl]acetic acid 6-chloro-2,4-diiodoquinoline 6-methoxy-1,5-diphenylhexan-3-one 1-[3,5-dichloro-4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2-(3,3-difluoroazetidin-1-yl)ethane-1,2-dione 1-[4-chloro-2,3-difluoro-6-(2-hydroxyethyl)phenyl]-N-methoxymethanimine (4aS,8R)-7-[5-(2-phenylethyl)triazol-1-yl]-6-(pyridine-3-carbonyl)-3,4a,5,8,8a-hexahydro-2H-pyrido[4,3-b][1,4]oxazin-4-one N-[4-amino-5-(1,2-oxazole-3-carboximidoyl)pyridin-3-yl]cyclopropanecarboxamide 1-(3,5-diphenylpyrazole-1-carbonyl)piperidine-4-carboxamide N-[3-(4-hydroxyphenyl)heptan-2-yl]acetamide 1-(2,4-dichlorophenyl)ethyl-[4-[3-(hydroxymethyl)anilino]piperidin-1-yl]sulfonylazanide 1-[(E)-(4-bromophenyl)methylideneamino]-3,3-dimethyl-2H-indole-6-carboxamide 2-[3-(oxan-4-yl)phenyl]acetic acid 3-(hydroxymethyl)-6,8,11-trioxatetracyclo[7.4.0.02,5.010,15]trideca-1(9),12-dien-4-one 7-fluoro-6-[(2E,4Z)-hepta-2,4-dienoxy]-1H-quinolin-2-one (5-chlorothiophene-2-carbonyl)-[(4-methoxyphenyl)methyl]azanium 3-[[1,3-bis(2-methylphenyl)imidazol-1-ium-4-yl]sulfonylamino]propanethioamide N-[2-(azidomethoxy)-4,5-dimethylphenyl]acetamide (1-chlorocyclohexa-2,4-dien-1-yl)sulfonylbenzene (4R)-3,4,5-trihydroxy-2-[3-(2-phenylethynyl)benzoyl]oxane-4-carboxylic acid (2R)-N',N'-dimethyl-2-[3-(5-oxo-1H-tetrazol-4-yl)propanoylamino]butanehydrazide N-[5-cyclopropyl-2-(4,6-dimethylpyridine-3-carbonyl)furo[3,2-b]pyridin-7-ylidene]-2-fluorobenzamide 3-methyl-2-(4-phenylmethoxyphenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-8-amine 1-(2-bromophenyl)-N'-hydrazinylidenepyrrolidine-3-carboximidamide N-(2,4-dimethoxyphenyl)sulfonyl-1-[6-fluoro-3-(2-pyridin-4-ylethynyl)cyclohexa-1,5-dien-1-yl]benzimidazole-5-carboxamide 2-[[8,9-bis(4-fluorophenyl)-7H-purin-6-yl]methyl]isoindole-1,3-dione 3-[5-[2-chloro-4-(6-oxononyl)phenyl]pyridin-3-yl]propanoic acid 2-[2-(2,3,4,5-tetrahydro-1H-inden-1-yl)phenyl]ethanamine 1-[2-(diethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]cyclopentane-1-carboxamide 4-[2-chloro-5-(trifluoromethoxy)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile 2-(4-bromophenyl)-N,N'-dimethylpropanediamide (2Z)-N'-[4-cyano-3-(trifluoromethyl)phenyl]-2-(1H-indol-5-ylmethylidene)propanediamide N-[3-(2,5-dimethylphenoxy)propyl]piperidine-1-carboxamide;formic acid [4-[1-(2,3-dihydro-1H-inden-5-ylamino)ethenyl]-4-hydroxypiperidin-1-yl]-[(2S)-oxolan-2-yl]methanone (5S)-4,7-dioxo-2-piperidin-1-yl-N-(3,4,5-trimethoxyphenyl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide N-[1-(5,7-dimethoxy-1H-indole-2-carbonyl)piperidin-4-yl]-2-methylpyridine-3-carboxamide 1-[4-[(6S)-3,6-dimethyl-5,6-dihydrobenzo[b][1]benzoxepin-7-yl]phenyl]cyclobutan-1-amine 2-(4-tert-butylphenyl)pyridine;iridium(3+);2,3,5,6-tetrapyridin-2-ylpyrazine;trihexafluorophosphate 2,3-dihydro-1H-indene;N-[1-(2-methyl-5-phenylpyrazol-3-yl)ethylideneamino]naphthalen-1-amine 4-[2,5-dimethyl-1-(4-pentoxyphenyl)pyrrol-3-yl]benzoic acid [4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-[2-[5-methoxy-8-(2-propan-2-ylpyrazol-3-yl)-3,4-dihydro-1H-isoquinolin-2-yl]cyclohexyl]methanone 4-[6-(6,6-dimethyl-1H-pyridazine-3-carbonyl)-8,9-dimethoxy-5H-benzo[c][2]benzazepin-11-yl]benzonitrile 2-(4-tert-butyl-1,3-thiazol-5-yl)-2-methoxypropanoic acid N-(3,5-dichlorophenyl)-2-[(6S)-2-methyl-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 6-ethyl-2,2-dimethyl-5-[1-(4-propan-2-ylpiperazin-1-yl)ethenyl]imidazo[1,2-a]pyrazin-3-imine 2-[4-(2,3,4,5-tetramethylcyclopenta-1,4-dien-1-yl)phenoxy]-N-(2,4,6-trimethylphenyl)acetamide 4-[2,6-dimethoxy-4-[(E)-5-oxopent-3-enyl]phenyl]butanoic acid 3,6-dichloro-5-[(3E)-4-phenylbuta-1,3-dien-2-yl]pyrido[4,3-b]indole (E)-3-[2-[[[1-[1-[1-[cyclohexyl(hydroxy)methoxy]-4,4-difluorocyclohexanecarbonyl]piperidine-4-carbonyl]azetidin-3-yl]amino]methyl]phenyl]prop-2-enoic acid 2-(3,4-dimethoxyphenyl)-6-[1-[ethyl(oxan-4-yl)amino]butan-2-ylamino]pyrazine-3-carboxamide;methane (2R)-5-benzylsulfanyl-2-[(4,6-dimethoxypyrimidin-2-yl)amino]pentanenitrile N-[3-fluoro-4-(tetrazol-1-yl)phenyl]-2-(4-oxoquinazolin-3-yl)acetamide 2-(4-fluorophenyl)imino-5-[(7-fluoroquinolin-6-yl)methylidene]-1,3-thiazolidin-4-one N-(2,6-dimethoxypyrimidin-4-yl)-4-[2-methylpropanoyl(1,3-thiazol-5-yl)amino]benzenesulfonamide 2-(6,7-dimethoxyquinazolin-4-yl)-N-[2-oxo-1-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl]benzamide 2-(3-ethynylphenyl)-N-methylcyclopropan-1-amine 2-[(6-azido-3,4,5-trimethylpyridin-2-yl)sulfanylmethyl]-4,6-bis(trichloromethyl)pyrimidine 3-[(2R,3R)-2,6-diaminohexanoyl]-4H-1,2,4-oxadiazol-5-one 4-(2,5-difluorophenyl)butanamide;ethane N-ethyl-4,5-dimethyl-2-phenyldiazenyl-N-propylaniline 2-(2,6-dioxopiperidin-3-yl)-5-[4-[[3-fluoro-1-(2,2,2-trifluoroethyl)azetidin-3-yl]methoxy]cyclohexylidene]isoindole-1,3-dione N-[3-[(2S,4R)-1-benzyl-2-methylpiperidin-4-yl]oxyphenyl]propanamide N-[3-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-4-(methylamino)pyridine-3-carboxamide N-[(4S)-2,2-dimethylpiperidin-4-yl]-5-(1H-pyrrolo[3,2-b]pyridin-6-ylmethylamino)pyrazine-2-carboxamide 6-[2,5-difluoro-4-(3-methoxypropyl)phenyl]-1H-indazole 2-[(1R)-7-chloro-6-fluoro-5-hydroxy-4,8b-dihydro-3aH-indeno[1,2-d][1,3]thiazol-1-yl]acetic acid [2-[5,6-di(propan-2-yl)benzimidazol-1-id-2-yl]phenyl]-trimethylsilane;iridium N-(3,3a,4,5,6,7,7a-octahydro-2H-indol-1-ylmethylideneamino)-2-morpholin-4-ylbenzamide N'-[[6-(2-morpholin-4-ylethoxy)quinolin-3-yl]methyl]-N'-phenylethane-1,2-diamine 2-[[(5Z)-4-oxo-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-2-ylidene]amino]acetic acid 2-[1-[[2-(azidomethyl)phenyl]methoxymethyl]cyclopropyl]ethanamine 2-(3-tert-butylcarbazol-9-yl)ethanol 6-[3,5-dichloro-4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]spiro[1H-indole-3,2'-oxetane]-2-one 4-(3,5-dimethoxyphenyl)benzenecarboximidamide 3-[6,7-dichloro-1-[4-(methylsulfanyloxyamino)butyl]-5-(2-phenylmethoxyphenyl)sulfonylindol-3-yl]propanoic acid 5-bromo-N,N-dimethyl-3-phenyl-1H-indole-2-carboxamide N-[1-(2-hydroxycyclohexa-2,4-dien-1-yl)-3-oxobutan-2-yl]furan-2-carboxamide 2-[1-(3-amino-4,6-difluoro-5-methoxycarbonylpyridin-2-yl)piperidine-4-carbonyl]cyclobutane-1-carboxylic acid 1-[4-azidooxy-2,6-di(propan-2-yl)phenyl]ethanone N-[(E)-2-(1,3-benzodioxol-5-ylmethylideneamino)but-2-enyl]-4-[(2-fluorophenyl)sulfonylamino]benzamide 2-[2-(4-carboxyphenyl)acetyl]benzenesulfonate [2-(4,5-dichlorocyclohepta-1,3,6-trien-1-yl)-1-(4-methoxyphenyl)butan-2-ylidene]oxidanium N'-[2-methyl-1,3-bis(oxan-2-yl)propanoyl]-5,6-dihydroquinoline-8-carbohydrazide 4-[3-(4-propoxyphenyl)-2H-imidazol-1-yl]butanenitrile 1-[[2-(dimethylamino)-5,7-dihydro-4H-thieno[2,3-c]pyran-6-yl]sulfonyl]cyclopropane-1-carboxylic acid 3-[3-bromo-5-[(1S)-1,2-dihydroxyethyl]pyridin-2-yl]oxypyrrolidine-2,5-dione 1-[2,6-di(propan-2-yl)phenyl]-N-(pyridin-4-ylmethylideneamino)methanimine 5-bromo-3,4-dimethyl-2-[1-(4-methylphenyl)ethoxy]quinoline 1-methylsulfonylindole-2,3-dicarbonitrile 2-[(3R,4S)-3-amino-4-propan-2-ylpyrrolidine-1-carbonyl]-6-methoxy-3H-quinazolin-4-one 2-(4,5-dimethyl-1H-pyrazol-3-yl)-1-hydroxy-6,7-dihydrocyclohepta[c]pyridin-9-one 1-[4,4-dimethyl-5-(1H-pyrrolo[2,3-b]pyridine-6-carbonyl)-1,3-thiazolidin-3-yl]propan-1-one 6-(4-azidophenyl)-N,N'-dimethylpyridine-3-carbohydrazide 1-azidooxy-5,8-dibromonaphthalene 1-[3-[(5-chloropyrimidin-2-yl)amino]cyclobutyl]-N-(2,6-dioxopiperidin-4-yl)pyrrolidine-3-carboxamide 2-[4-[5-(trifluoromethyl)pyridin-3-yl]phenyl]propanoic acid 4-[2-(3-ethoxyphenyl)quinolin-6-yl]benzenesulfonamide 5-amino-2,4-dimethoxybenzenethiol;N-[(Z)-1-(2,3-dimethylphenoxy)butan-2-ylideneamino]-N-ethylaniline 4-[2,6-dimethyl-3-(2-oxopropanoyl)-5,7-dihydropyrrolizine-1-carbonyl]piperazine-1-carboxylic acid 1-amino-1-phenylheptane-1,3,4-triol;ethanol 2-[1-(6,8-dichloro-3-phenylimidazo[1,2-a]pyridine-7-carbonyl)piperidin-4-yl]acetic acid N-[1-[2,4-dimethyl-5-(methylideneamino)phenyl]ethenyl]-3-propoxyaniline 3-[(3-chloro-4-fluorophenyl)methyl]pyrazine-2,5-diamine 2-(hydroxymethyl)propane-1,3-diol;3-[1-[2-(trifluoromethoxy)phenyl]imidazol-4-yl]-5H-imidazo[1,2-b]pyrazole 1-azido-4-[(E)-3,7-dimethyloct-6-en-2-ynoxy]benzene (2R)-N,N-dimethyl-4-oxo-1-[2-[2-(trifluoromethoxy)phenyl]acetyl]pyrrolidine-2-carboxamide 4-(cyclopropanecarbonylamino)-N,2-dimethylbenzamide ethane;4-methylpentanenitrile;3-(4-propan-2-ylphenyl)-4H-chromene 2-(1,3-benzothiazol-4-yloxy)-N-[3-fluoro-4-(methylamino)phenyl]acetamide N-(4,4-dimethylcyclohexyl)-1-[7-[(Z)-2-fluoro-3-iminoprop-1-enyl]imidazo[1,2-a]pyridin-3-yl]ethanimine (5Z)-2-sulfanylidene-5-[[4-[3-(trifluoromethyl)phenyl]phenyl]methylidene]imidazolidin-4-one 4-tert-butyl-6,7-dihydropyrazino[2,3-b]pyrazin-8-one N-(3,5-dimethylphenyl)-2-[3-methoxy-4-(6-methylpyridin-3-yl)phenyl]-3H-benzimidazole-5-carboxamide 2,4-dimethyl-6-(3-pyridin-2-ylpyrrolidine-1-carbonyl)-[1]benzofuro[3,2-d]pyrimidine 2,7-dibromo-9H-fluorene N-[[(5S)-3-[3,4-bis(trifluoromethyl)phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]acetamide 3-[4-(2,6-dimethylphenyl)-5-methoxypyridin-2-yl]benzoate 1-(4-tert-butylphenyl)ethanethiol;3-[2-chloro-5-[[6-methoxy-7-(piperidine-1-carbonyl)quinolin-4-yl]amino]phenoxy]propan-1-ol 4-(5-amino-2-pentylphenyl)benzenethiol;methane;4-methoxy-N,2-dimethylaniline 4-[1,2-difluoroethyl(pyridin-3-yl)amino]piperidine-1-carboxylate 2-[1-[[(3Z,5E)-6-chloroocta-3,5-dienoxy]methyl]cyclopentyl]sulfanyl-4-(trifluoromethyl)pyrimidine 2-[[(3S)-1,3-dimethylcyclohexanecarbonyl]amino]pyridine-4-carboxylic acid N-(cyclopropylmethyl)-1'-(furan-2-ylmethyl)spiro[7,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyridine-6,4'-piperidine]-3-carboxamide;2,2,2-trifluoroacetic acid (2S)-2,6-bis[4-chloro-5-(trifluoromethyl)pyrimidin-2-yl]-1,2,3,4-tetrahydronaphthalene 2-(4-nitropyrazol-1-yl)aniline [(1R)-2,5-dihydroxycyclohexa-2,4-dien-1-yl]-phenylmethanone 4-[2-[(3-cyanophenyl)methylamino]propyl]piperidine-1-carboxylate 4-[5-(3,6,6-trimethylcyclohexa-2,4-dien-1-yl)pentanoyloxy]benzenesulfonic acid (2R)-N-methyl-4-phenyl-1-[4,5,7-trifluoro-6-(4-fluorophenyl)-1H-indole-3-carbonyl]piperazine-2-carboxamide 1-[3-(1H-indole-2-carbonyl)imidazolidin-1-yl]-3,3,3-trifluoropropan-1-one 2-(N-amino-4-tert-butylanilino)-3,5-dichlorobenzoic acid 1-[2-(7-chloro-4-oxo-3H-quinazolin-6-yl)ethyl]-5,6,8,9-tetrahydropyrazolo[3,4-c]isoquinoline-7-carboxylic acid 1-[3-(methylamino)phenyl]indole-2,5-dione 1-[5,6-bis(ethenyl)pyridin-2-yl]ethanone;cyclohexane;ethene;2-methylpropane N-(3,4-dimethoxyphenyl)-6-ethylthieno[2,3-d]pyrimidin-4-amine (3-hydroxy-2,2-dimethylpyrrolidin-1-yl)-(4-pyrimidin-5-ylphenyl)methanone 3-[(2E,4Z)-hexa-2,4-dien-3-yl]sulfonylbenzenethiol 4-(5-bromopyridine-3-carbonyl)-1,4-oxazepane-6-carboxylic acid 2-[4-(2-ethoxypyridine-3-carbonyl)piperidin-1-yl]-1,3-thiazole-5-carboxylic acid 1-chloro-3-(5,6,7,8-tetrahydronaphthalen-2-yl)propan-2-ol;methanamine 2-[1-carboxypropan-2-yl(3,5-dichlorophenyl)amino]octanoic acid 2-benzyl-6,7-dihydrobenzo[d][1]benzoxepine (5Z)-5-[(3,4-dibromophenyl)methylidene]imidazolidine-2,4-dione 1,3-dichlorobenzene;N-[2-(4-formylphenoxy)ethyl]-5-methyl-3H-indole-2-carboxamide (3-cyclopropyl-1,2-oxazol-4-yl)-[3-hydroxy-3-(triazol-1-ylmethyl)piperidin-1-yl]methanone 3-[4-azidooxy-1-methylsulfonyl-2-(oxan-2-yloxy)indol-3-yl]propanenitrile (3S,4S)-4-[2-fluoro-5-(4-methylphenyl)sulfonylphenyl]-1-iodopyrrolidine-3-carboxylic acid 2-(3,4-dimethoxyphenyl)-6-methylchromene N-(4-chlorobutyl)-2,6-difluoroaniline [(1R,2S)-3-chloro-1-(4-cyclohexyloxyphenyl)-1,1-difluoropropan-2-yl]carbamic acid 1-[4-(3,3-dimethylbutan-2-ylidene)cyclohexa-1,5-dien-1-yl]-7-(3-pyrrolidin-1-ylpropoxy)naphthalene N-[2-(1,4,6-trimethylpyrazolo[3,4-b]pyridine-5-carbonyl)phenyl]formamide 3-[5-(trifluoromethyl)pyrazol-1-yl]aniline (6R)-4,4,6-trimethyl-3-pentanoyl-1,4-dihydroquinazolin-2-one N-[(1S)-1-aminoethyl]-2-(2,3-dihydro-1H-inden-5-yloxy)thieno[3,2-d]pyrimidin-4-amine;hydrochloride N-[(2R,3S)-2-methylsulfanylhexan-3-yl]-4-nitrobenzamide 3-N,5-dibenzyl-1H-indole-2,3,6-triamine 4-[2,6-difluoro-N-(2,2,2-trifluoroethyl)anilino]benzoic acid 1-(2,3-dihydroindol-1-yl)-2-methoxyethanone (3R,5S)-2-[2-hydroxyethyl(phenylmethoxycarbonyl)amino]-6-methylheptanoic acid 3-(2,5-dihydroxyphenyl)-N-[3-methyl-4-(trifluoromethoxy)phenyl]benzamide 2,6-diamino-N'-(1,3-benzothiazol-4-yl)pyridine-3-carboximidamide 6-[1-(2,5-dihydroxyphenyl)ethylideneamino]-1-(3-hydroxyphenyl)heptan-4-one 6-(dimethylsulfamoyl)-3-iodopyridine-2-carboxylic acid N-(4,5-dichlorothiophen-2-yl)sulfanyl-6-fluoro-7-methoxyquinolin-3-amine N-[(E)-4-aminobut-2-enyl]-5-[[3-[3,5-bis(trifluoromethyl)phenyl]-1H-pyrazole-5-carbonyl]amino]pyridine-3-carboxamide 3-azido-5-[4-(2,2-diphenylethenyl)phenyl]-1H-pyrazole 4-[2-(dimethylamino)pyrimidin-5-yl]sulfonylpiperazine-1-carboxylic acid 2-(1-benzylpiperidin-3-yl)oxy-5-ethanimidoylpyridine-4-carboxylic acid 2-[(3R,4S)-4-azidooxolan-3-yl]oxypyridine 2-azido-3-phenyl-1H-pyrrole ethane;1-[4-(3-methylphenyl)cyclohexa-2,4-dien-1-ylidene]ethanol 2-[2-hydroxyethyl(methylsulfonyl)amino]benzenesulfonic acid (E)-3-[5-[(4-tert-butylphenyl)methoxy]spiro[1,2-dihydroindene-3,2'-cyclopropane]-1'-yl]-N-hydroxyprop-2-enamide (6S)-7-[[1-[[4-chloro-2-fluoro-3-(3-hydroxypropoxy)phenyl]methyl]piperidin-4-ylidene]amino]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-3-carboxamide 7-methyl-3,4-diphenylchromene 2-[(Z)-1-aminobut-1-enyl]-N-[2,4-bis(trifluoromethyl)phenyl]-N'-[3-chloro-5-(trifluoromethyl)phenyl]-5-methanimidoyl-3H-pyrrole-4-carboximidamide (5S,7R)-2-[[1-(4-methylphenyl)pyrazol-3-yl]methylamino]-5,7-dihydropyrano[4,3-d]pyrimidine-8-carboxylic acid 1-(4-cyclohexyloxyphenyl)ethanethiol 2-[(4E,5Z)-2-methyl-6-(3-methylanilino)octa-1,4,5,7-tetraen-3-yl]oxy-N-(1-pyridin-2-ylethylidene)acetamide 4-[(3,5-dimethylphenyl)methylamino]-6-(2H-pyrrole-4-carbonylamino)quinoline-7-carboxylic acid 2-(4-chlorophenyl)-1-[7-(3,5-dimethylpyrazole-1-carbonyl)-9,11-dioxa-2-azaspiro[5.6]dodecan-2-yl]ethanone 4-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)aniline 2-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-ylamino)-1-[4-(oxan-2-yloxymethyl)piperidin-1-yl]ethanone 2-[6,7-dichloro-1-(4-methoxyphenyl)sulfonylindol-3-yl]propan-2-ol (E)-2,4-difluoro-N'-(7-methoxyquinolin-3-yl)pent-1-ene-1,5-diamine 4-[4-(3-phenylmethoxypropanoyl)piperazine-1-carbonyl]benzenesulfinamide 1-[4-chlorobutyl(naphthalen-2-yl)amino]propan-2-one 4-[[1-(3,5-dichlorophenyl)sulfonylpiperidin-2-yl]methoxy]-5-cyclopropyl-N'-hydroxypyridine-2-carboximidamide 2-(4-amino-3-methoxyphenyl)sulfonyl-1,3-benzoxazol-6-amine;ethane 2-ethyl-5-[(6-hydroxycyclohexa-1,3-dien-1-yl)methylideneamino]benzene-1,4-diol 2-[3,5-dichloro-4-(4-hydroxypiperidin-1-yl)anilino]-N-propan-2-ylacetamide 4-[7-amino-3-methyl-2-(methylidenehydrazinylidene)azepin-1-yl]-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-ylmethyl)benzamide;6-chloro-4H-chromene 2-(4-fluorophenyl)sulfanyl-N-[2-oxo-1-(trideuteriomethyl)pyrrolidin-3-yl]acetamide 3-(4-chloro-2-nitrophenoxy)-N'-hydroxypyridine-2-carboximidamide 1-cyclohexyl-4,7-dimethyl-2,3-dihydropyrrolo[2,3-c]pyridine (2S)-2,3-dimethylbutane;4-[4-[3-[3-[[5-ethoxycarbonyl-6-hydroxy-1-(pyridine-4-carbonyl)benzimidazol-2-yl]methyl]phenyl]prop-1-enyl]phenyl]benzoic acid N-[2-(2,5-difluorophenoxy)propanoyl]cyclobutanecarboxamide 2-(3,4-dimethoxyphenyl)-5-ethyl-N,N,6-triethylpyrimidin-4-amine;hydrochloride 6-bromo-3-(1H-indol-2-ylmethylideneamino)-1H-quinazoline-2,4-dione ethane;5-[4-[2-(3-methoxyphenyl)propyl]piperazine-1-carbonyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 2,4-dichloro-N-[6-(5-chloro-1H-indazol-7-yl)pyridin-3-yl]benzamide 3-[5,6-dimethyl-1-(2-morpholin-4-ylethoxy)indol-3-yl]oxirane-2,2-dicarbonitrile 4-(3-methylpentan-3-yl)-1-phenylcyclohepta-1,3,5-triene 1-[4-(trifluoromethoxy)anilino]butan-2-one 5-[2-chloro-6-(trifluoromethyl)phenyl]-3H-1,3,4-oxadiazole-2-thione 1-(2,4-dihydroxyphenyl)-2H-pyrimidine-5-carbonitrile 6-[1-cyclopropyl-3-(oxan-4-ylmethoxy)pyrazol-4-yl]sulfonyl-2,5,7,8-tetrahydro-2,6-naphthyridin-1-one 3-(2,4-difluorophenyl)pyridine-1-carboxylic acid;ethane ethane;4-(3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazol-2-yl)phenol (2R)-3-cyclopropyloxy-N'-[(5S,7S)-5-methyl-8-oxo-6,7-dihydropteridin-2-yl]butanimidamide 2-ethyliodanuidyl-N'-hydroxypyrimidine-4-carboximidamide 1-(difluoromethyl)-4-[2-(difluoromethoxy)ethoxy]-3-fluoro-2-(3,3,5,5-tetrachloropropN,2-dimethyl-6-phenylcyclohexa-1,3-dien-1-yl)benzene 1-(5-ethylthiophen-2-yl)sulfonyl-3,4-dihydro-2H-quinoline [4-[5-[1,3-bis(methylsulfonyl)indol-2-yl]thiophen-2-yl]phenyl]hydrazine N-cyclohexyl-6-(4,5-difluoro-2-methoxyphenyl)imidazo[1,2-a]pyridin-8-amine N-[(1S)-1-[5-chloro-1-benzofuran-2-ylsulfonyl-[(3R,4S)-4-phenylpyrrolidine-3-carbonyl]amino]propyl]-6-oxo-1H-pyridazine-3-carboxamide 4-[(3R)-3-aminopiperidine-1,4-dicarbonyl]-2-methyl-7H-pyrazolo[3,4-d]pyrimidin-6-one 4-[2,4-di(propan-2-yl)phenyl]-3-oxobutanenitrile 4-[3-azidooxy-5-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-1-yl)pentan-3-yl]aniline 4-azido-N-[1-(3,5-dichlorophenyl)ethyl]benzamide 3-(4,5-dimethyltriazol-2-yl)-7-fluorobenzonitrile (E)-N-benzylsulfanyl-1-cyclohexylmethanimine 6-(2,3-dihydrothiophen-4-yl)-2-ethylsulfanylthieno[2,3-d]pyrimidine ethane;N-[4-(2-hydroxypropan-2-yl)pyridin-3-yl]pyrrolidine-1-carboxamide 2,3-bis(ethenyl)-1,5-dimethylquinolin-4-one 4-[(5-methyl-2-propan-2-ylimidazo[1,2-a]pyridin-3-yl)diazenyl]benzene-1,3-diamine 3-(1,3-benzodioxol-4-yl)-N-[[2-[(2R,5S)-4-[(2-fluorophenyl)methyl]-2,5-dimethylpiperazine-1-carbonyl]-4,6-dimethoxyphenyl]methyl]propanamide 3-methylbutanoic acid;4,9,10-tris(2-nitrophenyl)anthracene 1-(2,5-difluorophenyl)-3-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]propan-1-one 3-hydroxy-1-(2,5,6,7-tetrahydro-[1]benzofuro[2,3-d]pyrimidin-4-yl)azepan-2-one 2-[4-[(5-cyclohexylpyridine-3-carbonyl)amino]-1H-pyrazol-5-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine-3-carboxylic acid 2-ethoxy-6,8a-dihydrobenzo[g]quinoxaline 2-chloro-N-[5-ethylsulfonyl-6-[3-(trifluoromethoxy)phenoxy]pyridin-3-yl]acetamide (2S)-N-[(4R,5S)-3-methyl-6-oxo-7-oxa-1,5-diazaspiro[5.5]undecan-9-yl]-6-oxo-7-thiatricyclo[15.4.0.02,4]henicosa-1(21),12,14,16,18-pentaene-5-carboxamide 2-amino-6-[3-bromo-4-(hydroxymethoxy)phenyl]-4,4-dimethoxy-3-azabicyclo[3.1.0]hex-2-ene-1,5-dicarbonitrile 6-methyl-2-(pyridin-4-ylamino)-3H-thieno[3,2-d]pyrimidin-4-one 2-[4-(3,5-dimethoxyphenyl)piperazine-1-carbonyl]-6H-thieno[2,3-b]pyrrole-5-carboxamide 3-cyclopentyloxy-N'-hydroxypyridine-2-carboximidamide 4-benzamido-3,5-difluorobenzoic acid 3-[(E)-3,5-diaminopent-2-enyl]-4-ethoxyphenol 4-bromo-2-[5-(3,5-dibromophenyl)pentyl]phenol 3-[2-(5-methylfuran-2-yl)ethyl]-4H-1,2,4-oxadiazol-5-one N-(furan-2-ylmethyl)-5-oxo-1-(6-phenoxypyridin-3-yl)pyrrolidine-3-carboxamide 5-(2,4-difluoro-6-methoxyphenyl)imidazolidine-2,4-dione 1,5-dimethyl-2-[3-(trifluoromethoxy)phenoxy]benzene;ethane 2-(5,5-dimethylcyclohepta-1,3,6-trien-1-yl)-N-[4-(trifluoromethoxy)phenyl]quinoline-4-carboxamide 7-(4,4-dimethylpiperidin-1-yl)-2-ethylsulfanyl-N-(3-imidazol-1-ylphenyl)quinazolin-5-amine N-[(2,6-dichlorophenyl)methyl]-5-ethyl-3,4-dihydropyrazole-2-carboximidate 2-[(5-methylfuran-2-yl)methylamino]thieno[3,2-d]pyrimidine-4,6-diamine N-cyclopropylsulfanyl-4,5-difluoro-2-(3H-pyrazolo[3,4-c]pyridin-6-yl)aniline N-[1-[3-[2-(dimethylamino)ethyl]phenyl]-5-methoxy-4-methylpyrazol-3-yl]formamide (2-benzo[g][1,3]benzothiazol-2-ylphenyl)-phenyldiazene 1-chloro-2,3-dimethylbenzene;ethane;formaldehyde 2-(1,4-dimethoxybutan-2-ylamino)benzenesulfonic acid 3-(4-fluorocyclohexa-2,4-dien-1-yl)oxybenzoic acid 5-azidooxy-1H-cyclopenta[a]naphthalene (2E,4Z)-3-chloropenta-1,4-dien-3-ol;(Z,2R,6S)-2-ethyl-5-methylidene-7-phenyloct-6-enal N-[(2R)-2-azido-2,3-dihydro-1H-inden-5-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide (2R)-2-amino-N-[[1-[3,4-difluoro-5-(6-methylpyridin-3-yl)oxyphenyl]ethylamino]carbamothioyl]pentanamide 2-[3-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-N-(4-pyridin-2-yloxycyclohexa-2,4-dien-1-ylidene)acetamide 2-[(1R,5S)-3-[1-(difluoromethyl)cyclopropanecarbonyl]oxy-6-oxo-3-azabicyclo[3.2.0]heptan-9-yl]-2-(4-methoxyphenyl)acetic acid 2-[2-[(5S)-2-oxo-3-phenyl-1,4-diazepane-1-carbonyl]cyclohexyl]acetic acid ethane;1-methyl-4-propan-2-yloxynaphthalene 4-[3-(4-ethylpiperidin-1-yl)propoxy]aniline ethane;5-methylnaphthalene-1,7-disulfonic acid 5-(2,3-dihydro-1H-inden-2-yl)-4-(2-fluorophenyl)imino-1-propylimidazolidin-2-one 1-[5-amino-6-(2,4-difluorophenoxy)pyridin-3-yl]ethanone N-[2,3-difluoro-4-[3-[(1S)-1-[5-(trifluoromethyl)pyridin-2-yl]oxyethyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]phenyl]propane-1-sulfonamide 1-[2-(4,5-dihydro-1H-indole-7-carbonylamino)ethyl]-N-(4-methoxyphenyl)piperidine-3-carboxamide 7-[4-(2,6-diphenylpyrimidin-4-yl)phenyl]quinoline [2-(cyclopropylmethoxy)phenyl]-pyrrolidin-1-ylmethanone 4-[1-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylcarbamoylsulfonyl)azetidin-3-yl]oxybenzoic acid 5-[1-(4-azidophenyl)ethyl]-2H-triazole-4-carboxylic acid 2-(4,5-dimethylthiophene-2-carbonyl)oxyacetic acid 2-azido-7-(trifluoromethyl)quinoxaline 2-[1-(3,4-difluorobenzoyl)pyrrolidin-2-yl]-6-methyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 5-[3-(2,6-dimethylphenoxy)phenyl]pentan-1-ol;ethane 5-methylsulfanyl-4-(2,3,6,7-tetrahydroazepin-1-yl)pyridine-3-carbonitrile 1-methyl-3,4,5,6-tetrahydro-2H-quinoline;N,8,10-trimethoxy-2,12-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,11-trien-4-amine N-(2,2-diethoxyethyl)-4-nitro-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]benzamide 3-(4-chlorophenyl)propanoate 2-fluoro-4-[(3R)-3-[4-(6-phenylpyridine-3-carbonyl)piperazin-1-yl]pyrrolidin-1-yl]benzonitrile 4-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-N,N-dimethylaniline N-[3-[[6-(1,2,3,5,7-hexahydro-s-indacen-4-ylamino)pyrimidin-4-yl]sulfanylmethyl]cyclobutyl]acetamide 6-(5,7-dimethylimidazo[1,2-c]imidazol-2-ylidene)cyclohexa-2,4-dien-1-ol N-[6-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)pyridin-3-yl]acetamide 5-[3,4-di(propan-2-yl)phenyl]-8-[3-methoxy-4-(4-methylpiperazin-1-yl)anilino]imidazo[1,2-c]pyrimidine-7-carboxamide 3-[5-methyl-4-(2,6,6-trimethylcyclohexen-1-yl)furan-2-yl]propanoic acid 3-(4-methylpiperazine-1-carbonyl)-N-[(4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methyl]piperidine-1-carboxamide 1-azidosulfanyl-2,3-di(propan-2-yl)benzene 3,5-bis(3,3,4,4,5,5,6,7,8,8-undecafluorooctyl)aniline 4-benzylsulfanyl-2,3-dihydroisoindol-1-one 3-[3-(1,3-benzothiazol-2-yl)phenyl]-N,N-dimethylaniline 3-(3,4-dimethoxyphenyl)sulfanylpropanenitrile;1-phenylethylbenzene 1-[(3R,4S)-3-phenyl-1-propan-2-ylpiperidin-4-yl]-2H-pyrrolo[3,2-b]pyridine 2-amino-6-(3,4-dimethylpiperazin-1-yl)-N'-hydroxypyridine-4-carboximidamide 5-fluoro-3,4-dimethoxy-6-[(3E)-penta-1,3-dien-3-yl]pyridine-2-carbonitrile 1-[(E)-2,3,5-trimethyloct-4-enoxy]naphthalene 2-methyl-N-[5-(4-phenoxyphenyl)-1,3,4-thiadiazol-2-yl]propanamide [2-[6-(4-butylcyclohexen-1-yl)naphthalen-2-yl]ethynyl]boronic acid [2,3-diamino-6-(1H-indole-2-carbonyl)phenyl]-methylcarbamic acid 4-[2-(1H-indol-5-yloxy)ethyl]-9H-pyrido[3,4-b]indole 4-(2,6-dichloropyridine-4-carbonyl)-5,8-dimethyl-1,3,3a,4,7,9b-hexahydropyrrolo[3,4-h]isoquinolin-2-one N-[2-methyl-4-(tetrazolo[1,5-b]pyridazin-6-yl)pyrazol-3-yl]formamide (E)-3-[4-(dimethylamino)naphthalen-1-yl]-2-sulfanylprop-2-enal 6-(3,5-dimethylpyridin-2-yl)hexanamide 2-azido-4,5-dimethylbenzenesulfonic acid (2R,4S)-2-tert-butyl-4-[3-(2-methoxyethoxymethyl)phenyl]pyrrolidine 1-(2,6-difluorophenyl)-N-[5-methyl-6-(triazol-2-yl)pyridin-3-yl]-4H-pyrimidine-5-carboxamide N-(2,6-dioxopiperidin-3-yl)-6-methoxy-1H-indole-7-carboxamide (7S)-N-(2,4-dimethylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 3-[(4S)-1-hydroxyheptan-4-yl]sulfanyl-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-8-one N-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]butanamide 1-[(4R)-1-azido-2,5-dioxoimidazolidine-4-carbonyl]pyrrole-3-carbonitrile 1-(4-ethylsulfonylphenyl)-2,3-difluorobenzene;2-(2,6,7-trimethoxyheptyl)-3H-isoindol-1-one [4-(5-chloropyridin-2-yl)piperazin-1-yl]-[1-[(6,7-dimethoxyquinazolin-4-yl)amino]cyclobutyl]methanone (3E,5Z)-5-[3-[5-methyl-4-[(1E)-1-thiophen-2-ylbuta-1,3-dienyl]-1H-pyrrol-2-yl]-1H-indazol-5-yl]hepta-1,3,5-triene-3-thiol 5-amino-7,8,9,10-tetrahydrophenanthridin-6-one 6-chloro-2-[[1,3-dihydroisoindol-2-yl(methyl)amino]methyl]-3H-thieno[3,2-d]pyrimidin-4-one 2-[azido(methoxy)amino]sulfanylbenzonitrile 2-[3-(4-hydroxyphenyl)-5-methyl-1,2,4-triazol-4-yl]acetic acid 4-[7-(4,6-diphenyl-1,3,5-triazin-2-yl)dibenzothiophen-4-yl]benzene-1,2-dicarbonitrile 4-(2-aminoethoxy)naphthalene-1,7-disulfonic acid;hydrochloride 2-[2-bromo-4-(2,3,5,6-tetrafluorophenoxy)phenyl]acetamide 2-benzyl-3,4-dihydrophthalazin-1-one [5-methoxy-3,4-di(propan-2-yl)thiophen-2-yl]carbamic acid [5-chloro-2-(ethylaminomethyl)phenyl]boronic acid 4-hydroxy-3,5-dimethyl-N-(2-nitrophenyl)sulfanylbenzamide (5R,7S)-N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)phenyl]-5,7-dihydrofuro[3,4-d]pyrimidin-2-amine;dihydrochloride N-[4-(N'-hydroxycarbamimidoyl)-1H-pyrazol-5-yl]-5-methoxypyrimidine-2-carboxamide (5E)-2-(4-methylphenyl)imino-5-[[5-(naphthalen-1-ylmethoxy)-1-(3,4,5-trifluorophenyl)pyrazol-4-yl]methylidene]-1,3-thiazolidin-4-one N-(2,6-dichloro-4-nitrophenyl)-N-(4-hydroxybutyl)benzamide 3-[[1-(2,2-dimethylpropanoyl)piperidin-4-yl]methoxy]-5-[(E)-3-oxo-1-phenylbut-1-en-2-yl]benzonitrile 2-(N-[4-chloro-3-(trifluoromethyl)phenyl]sulfonylanilino)acetamide N-[(1S,2R)-2-hydroxycyclooctyl]-4-phenylbenzamide (5E)-2-cyclohexylimino-5-[[4-(dimethylamino)phenyl]methylidene]-1,3-thiazolidin-4-one N-[4-chloro-2-(hydroxymethyl)phenyl]-3-[3-fluoro-5-(trifluoromethoxy)phenoxy]-1H-pyrazole-5-carboxamide 4-[2-(5-fluoropyridin-2-yl)phenyl]butanoic acid 1-[4,5-difluoro-2-(methylamino)phenyl]ethanone 2-(3,4-dimethoxyphenyl)-5-ethyl-7-oxo-6H-[1,3]thiazolo[4,5-d]pyrimidine-7a-carboxylic acid 4-[2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-4-yl)phenyl]butanoic acid [4-(2,5-difluorophenyl)piperazin-1-yl]-[(5R,7S)-5-methyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]methanone ethene;4-[(E)-1-[ethyl-[(Z)-prop-1-enyl]amino]prop-1-enyl]-6-fluoro-2,3-dihydrothiochromen-4-ol [2-bromo-5-(trifluoromethyl)phenyl]methanamine 5-[4-(5,7-dichloro-1-hydroxy-1H-isoindole-2-carbonyl)piperidin-1-yl]pyridine-3-carboxamide 6-chloro-2-[4-fluoro-3-(trifluoromethyl)phenyl]pyrimidine-4,5-diamine 3-[5-(2,4-difluorophenyl)cyclohexa-1,5-dien-1-yl]-N-ethyl-N-methylpropanamide;ethane 4-(2-bromoanilino)-6-[(3,5-dimethoxyphenyl)methyl]pyrimidine-5-carbonitrile 2-methylsulfonyl-N-[(1-propan-2-ylimidazol-2-yl)methyl]-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine-4-carboxamide 2-(3,6-dimethylpyrazin-2-yl)oxyphenol N-[(1R)-3,4-dihydro-2H-chromen-7-yl]-3-methyltriazole-4-carboxamide 4-chloro-7-[[(2S)-1,3-dihydroxypropan-2-yl]methoxy]chromen-2-one 4-[(3S)-3-phenylpiperidin-1-yl]quinazoline (E)-3-[3,5-dimethoxy-4-[2-(1H-pyrrolo[3,2-b]pyridin-2-yl)ethynyl]phenyl]-N-methoxy-N-methylprop-2-enamide 2,3-bis(ethenyl)quinoxaline;ethane 3,5-dihydroxy-1-methylquinoline-4-thione;2-[2,6-di(propan-2-yl)phenyl]guanidine 3-[2-(cyclopropylmethylamino)pyrimidine-4-carbonyl]-1,1-dimethylurea 5-(2,3-dichlorophenyl)-1-methyl-3-pyridin-3-ylpyrazole 2-[(3-methylphenyl)methyl]-7-piperidin-1-yl-4H-pyrazolo[1,5-a]pyrimidin-5-one 1-N',1-N'-dicyclohexyl-5-(hydroxymethyl)-2H-naphthalene-1,1'-dicarboxamide N-butyl-1-[4-[2-(3,5-dimethoxyanilino)pyrimidin-4-yl]phenyl]-4-methylpiperidine-3-carboxamide;ethane (Z)-N-[2-fluoro-4-methyl-5-(trifluoromethyl)phenyl]-3-hydrazinylidenebutan-1-imine 3-[2-(7-methyl-1H-indazol-5-yl)ethenyl]-N-(2-propan-2-ylpyridin-4-yl)-4-[2-(trifluoromethoxy)phenyl]benzamide 2,4-di(propanoyl)benzenecarboximidamide 4-(4-fluorophenyl)sulfanyl-2-[5-methoxy-6-(2-piperidin-1-ylethoxy)pyridin-3-yl]quinoline 1-[2-(3,4-dimethoxyphenyl)ethyl]-3-[2-(2-propan-2-ylimidazol-1-yl)ethyl]urea 1-[2,3-dihydroxypropyl(pyridin-4-yl)amino]propan-2-one 4-[2,3-bis(aminomethyl)anilino]-N'-hydroxypyridine-2-carboximidamide 4-[(4,5-dichloropyridin-2-yl)amino]-N-[(3-fluorophenyl)methyl]benzamide 3-(2,4-dioxopyrimidin-1-yl)cyclohexane-1-carboxylic acid N-(1-aminopropan-2-yl)-4-[4,5-bis(ethenyl)-3-methylidene-6-oxopyridazin-2-yl]benzamide (2S,3aS,8bR)-N-benzylspiro[1,2,3a,4,5,6,7,8,8a-decahydroisoquinoline-3,2'-cyclopropane]-1'-carboxamide 1-[4-[(2S,6R)-1,3,6-trimethylpiperidin-2-yl]phenyl]pentan-1-imine 2-[4-[4-[6-(hydroxymethyl)pyridine-3-carbonyl]piperazine-1-carbonyl]phenyl]acetonitrile 1,3-diamino-1-[2-[[6-(cyclohexylmethoxy)-5-methylpyridin-3-yl]methylsulfanyl]-3-methylphenyl]urea 2-hydroxy-N-[(Z)-(6-oxocyclohepta-1,3,5-trien-1-yl)methylideneamino]benzamide (4-azido-3,6-dihydro-2H-pyridin-1-yl)-(5,6,7,8-tetrahydronaphthalen-1-yl)methanone (2-phenylphenyl)-[3-[4,4,5,5-tetramethyl-1-(1H-pyrrole-2-carbonylamino)pentan-2-yl]phenoxy]borinic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-[4-oxo-5-[[2-(trifluoromethoxy)phenyl]methylsulfanyl]pyrazolo[3,4-d]pyrimidin-1-yl]acetamide 5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]furan-3-carboxylic acid [6-[[(2R,5S)-1-(4-fluorophenyl)sulfonyl-5-methylpyrrolidin-2-yl]amino]pyridine-3-carbonyl]carbamic acid N-[(3S,7R,8aS)-3-[2-(dimethylamino)ethoxy]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-5-ethylpyridine-3-carboxamide 2-(4,5-dihydro-1H-imidazol-2-yl)-4-[4-(trifluoromethoxy)phenyl]pyrimidine N-azido-4,5-dimethylthiophene-2-carboxamide 3-[4-(2-methylpropoxy)phenyl]-5-piperidin-3-yl-1,2,4-oxadiazole;hydrochloride 2-methylsulfanylethylidene-[4-[(5R)-7-oxo-8,9-dihydro-6H-pyrimido[1,2-a]pyrimidin-3-yl]phenoxy]-propylazanium 3-(1H-indol-2-yl)-N-[6-(4-methoxyphenyl)pyridazin-3-yl]benzamide 2-methyl-3-[4-(trifluoromethoxy)phenyl]propanoic acid 2-[4-[(3,6-dichlorocarbazol-9-yl)methyl]triazol-1-yl]-N-[[2-ethoxy-4-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]methylideneamino]acetamide N-(2,6-dichloro-4-nitrophenyl)-2,5-dimethyl-N-octylaniline 6-(4-aminocyclohexyl)-2,5-dimethoxypyridine-3-carboxylic acid 4-(5-nitrothiophen-2-yl)butanal 5-[4,6-dichloro-3-(trifluoromethyl)imidazo[1,2-a]pyridine-7-carbonyl]-N'-(4-methoxyphenyl)-1,2-oxazole-3-carbohydrazide 5-(trifluoromethyl)-2-[1-[2,4,6-tris(trifluoromethoxy)phenyl]ethylamino]pyridine-3-carboxylic acid 2-(4-methoxyphenyl)-6-propan-2-yl-N-pyridin-3-ylpyrimidine-4-carboxamide 7-bromo-N'-(4,6-dimethylpyrimidin-2-yl)spiro[3H-chromene-2,1'-cyclobutane]-4-carbohydrazide;ethane 3-(4,5-dichloro-2-hydroxyphenyl)cyclopropane-1,1,2,2-tetracarbonitrile 2-[(5-cyclopropylsulfonylpyridin-2-yl)methyl]-6,7-dihydropyrrolo[1,2-c]imidazole 3-[(2S,4R)-4-fluoropyrrolidine-1-carbonyl]-N'-hydroxy-5,6-dimethylpyridazine-4-carboximidamide (2R,5S)-5-[[3-chloro-4-(trifluoromethylsulfanyl)phenyl]methyl]-2-(4-fluorophenyl)oxolane 1-[3-[[(1Z)-buta-1,3-dienyl]iminomethyl]phenyl]-5,6-dihydro-4H-cyclopenta[c]thiophen-4-amine 2-[1-(3-bromophenyl)sulfonylazetidin-3-yl]-4-methyl-6-(2,2,2-trifluoroethoxy)pyrimidine (3S)-4,5-dimethylhexanenitrile;1-[3-[2-(3,4-dimethylphenyl)ethoxy]propyl]pyrrolidine 3-[7-(4-fluorophenyl)sulfonyl-5,6,8,9-tetrahydropyrido[2,3-d]azepin-3-yl]propanoic acid N-[4-chloro-2-(diethylamino)phenyl]sulfanylpropanamide 2-methoxy-1-phenylindole [2-(4-bromophenyl)pyrazol-3-yl]methanamine N-[(3E)-penta-1,3-dien-2-yl]-4-phenylbenzenesulfonamide 4-[(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)diazenyl]benzoic acid (2-azidooxyphenyl)methylphosphonic acid 4-[2-(5,6-difluorobenzimidazol-1-yl)ethoxy]phenol (2S,4R)-1-benzyl-N-hydroxy-4-[methoxy(diphenyl)methyl]pyrrolidine-2-carboxamide 1-(2,3-dihydroxypropyl)-N-[5-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-6-oxo-6-[[4-(trifluoromethyl)cyclohexa-2,4-dien-1-ylidene]methyl]pyridin-3-yl]pyrrolidine-3-carboxamide 6-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-sulfonamide 4-methyl-2-phenyl-5,6,7,8-tetrahydroisoquinolin-1-one 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-N-methoxypyridine-3-carboxamide 4-[4-(2,6-dimethylphenyl)piperazin-1-yl]pyridine-3-carboxylate 4-(azidomethyl)-5-phenoxypyridazine 1-[2-ethoxy-5-fluoro-4-(8-fluoroquinolin-3-yl)phenyl]-N,N-dimethylethanamine 5-[2,6-dichloro-4-(trifluoromethyl)phenoxy]pyrazine-2-carboxylic acid 4-methyl-2-[[5-(1H-pyrrol-3-yl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-thieno[3,2-d]pyrimidine ethane;N'-ethyl-N-methyl-N-propan-2-ylbenzenecarboximidamide 4-(methylideneamino)benzaldehyde;3-(2,6,8-trimethylimidazo[1,2-a]pyridin-3-yl)oxetane 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-[7-(ethylideneamino)-6-fluoroquinolin-4-yl]propanehydrazide 2-[4-(3,5-dimethylphenyl)piperazine-1-carbonyl]-1H-pyridin-4-one 4-methoxycarbonylnaphthalene-2,6-disulfonic acid N-[(E)-but-2-enyl]-3-methylbutanamide;7-ethoxy-6-methoxy-4,4-dimethyl-1H-3,1-benzoxazin-2-one (5S,7R)-5-(4-ethylphenyl)-N-[3-methoxy-2-(pyrazol-1-ylmethyl)phenyl]-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 2-[4-ethyl-1-(3,5,6-trimethylpyrazin-2-yl)azepan-3-yl]-N-[[1-(trifluoromethyl)cyclobutyl]methyl]acetamide 3-benzyl-5-N,7a-dihydropyrene-1,2,6-triamine 4-[5-(2,3-dichlorophenyl)furan-2-yl]pyridine 1-(3,4-dimethoxyphenyl)decan-1-one N-[1-(oxan-4-yl)pyrazol-3-yl]-2,5-dioxopyrrolidine-3-carboxamide N-(6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-3-ylsulfonyl)-2-ethylbenzamide N-(5-chloropyridin-2-yl)-N',N'-diethylethane-1,2-diamine 4-[3-(5,6-dimethylpyrazin-2-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-N,N-diethylpiperazine-1-sulfonamide 4-[5-[(Z)-2-(7H-cyclohepta[b]pyridin-11-yl)ethenyl]-1,3-oxazol-2-yl]phenol N-(5-fluoropyridin-2-yl)oxyquinoline-3-carboxamide (2S)-1,5-diamino-N'-azido-3,4,6-trihydroxy-2-phenylmethoxyheptanehydrazide 2-methyl-3-phenylsulfanylpyrazine 1-[(2R,4S)-2-benzyl-5-oxooxolan-3-ylidene]-N'-phenylmethoxymethanediamine 4-[(E)-2-amino-1,3-bis(2-hydroxyphenyl)prop-2-enoxy]benzenesulfonic acid 4-[5-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-3-propan-2-yl-1H-pyrazol-4-yl]pyrimidine 7-(cyclohexylamino)-4-oxo-3H-pyrimido[5,4-b]indole-2-carboxylic acid 5-fluoro-2-methyl-N-(1H-pyrrolo[3,4-c]pyridin-6-yl)pyrimidine-4-carboxamide [4-(3,5-dimethylpyrazol-1-yl)phenyl]-phenyldiazene 1-(3,4-dichlorophenyl)-5-(2-hydroxyethyl)triazole-4-carboxylic acid 4-methyl-2-[(1E,3Z)-4-methylidenehepta-1,3-dienyl]furan;N-methyl-5-(2-methylpropoxy)pyridin-2-amine 1-(1,3-benzodioxol-5-ylmethoxy)-2-[4-[[6-[cyclopentyl-(4-fluorophenyl)sulfanylamino]pyridin-3-yl]methyl]piperidin-1-yl]propan-2-ol [2-(3-fluorophenyl)pyrrolidin-1-yl]-piperidin-4-ylmethanone;dihydrochloride 6-methylsulfinyl-2-thiophen-3-ylquinoline 3-amino-2,4,6-trimethylimidazo[1,5-a]pyridine-7-carboxylic acid 2-cyclopentyloxy-3-phenylquinoxaline 3-benzyl-5,6-dichloro-1H-indole 5-[4-methyl-3-(trifluoromethyl)phenyl]-N,N-bis[(2-methylpyrazol-3-yl)methyl]-1H-pyrazole-4-carboxamide (3-azidooxypiperidin-1-yl)-phenylmethanone [3-fluoro-4-(2-quinolin-6-ylethynyl)phenyl]azanide 4-[6-azido-2,3-dichloro-5-(4-methoxyphenoxy)phenyl]-2-pyridin-4-yl-1H-pyrimidin-6-one 4-[[3-(4-hydroxyphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]-N'-methanimidoylbenzenecarboximidamide N-(2,3,5,6-tetrachloropyridin-4-yl)acetamide 2-amino-4-(5,6-diethoxypyridin-3-yl)-N'-hydrazinylidenepyrimidine-5-carboximidamide 4-[7-(2-methoxyethyl)spiro[3.5]nonan-1-yl]-3,5-dimethyl-1H-pyrazole 4-[2,5-bis(trifluoromethyl)phenoxy]butanoate 3-(2,6-diethylphenyl)imino-5-(furan-3-ylmethylidene)piperidin-4-one [[2-(8-aminoquinoline-3-carbonyl)-5-chlorophenyl]-piperidin-1-ylmethylidene]azanium 1-(3,5-dimethoxyphenyl)dodecane-2,4-dione 5-chloro-3,4,5,6-tetradeuterio-2-(3-hydroxyphenyl)phenol (5S)-5,7,8-trimethyl-2-[3-methyl-4-(4-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-ium-2-yl]-5H-benzo[f]quinoline 1,2-difluoro-6-[4-(propylsulfanylmethoxy)phenyl]naphthalene N-(2,6-dichloro-4-nitrophenyl)-N-pyridin-2-ylacetamide N-[6-amino-3,5-bis(2-pyridin-4-ylethoxy)pyrazin-2-yl]-4-methyl-1H-pyrrole-3-carboxamide 1-[2-(4-bromocyclohexa-2,4-dien-1-yl)ethynyl]-2-(3,5-difluorophenyl)benzene 1-[(1R)-1-phenylethyl]cyclopropane-1,2-diamine 5-[(3R)-5,8-dichloro-7-hydroxy-1,2,3,4-tetrahydroisoquinolin-3-yl]quinoline-8-carboxylic acid N-[5-[4-methyl-2-(trifluoromethoxy)phenyl]-1H-pyrazol-3-yl]-4-[(2S,6R)-2-propanoyl-6-propan-2-ylmorpholin-4-yl]benzamide 5-chloro-2-[5-(1-cyclopropyltriazol-4-yl)-1,3-thiazol-2-yl]phenol 7-cyclopropyl-6-(1H-indazole-4-carbonyl)-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,8,11-tetraen-12-one 2-(4-methyl-N-octylanilino)acetamide 2-[(2S)-1,4-dioxan-2-yl]-N-[3-(5-methyl-1H-pyrazol-4-yl)propyl]ethanamine [4-(2-aminoethyl)-2,6-dimethoxyphenyl]methanol 4-[[6-ethyl-5-(4-fluorophenyl)pyrazin-2-yl]methoxy]benzamide 3-amino-N'-(5,7-difluoroquinolin-2-yl)-4-methoxybenzenecarboximidamide 2-[4-(bromomethyl)phenoxy]-5-fluorobenzonitrile 3-[(4,6-diamino-1,3,5-triazin-2-yl)sulfanyl]propanenitrile 4-[(2S)-6,15-dibromo-13-chloro-2-methyl-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-5-yl]piperidine-1-carboxylic acid N-[4-chloro-2-(6,7-dimethoxyquinolin-4-yl)phenyl]acetamide 2-[4-(bromomethyl)phenyl]-3,5-bis(trifluoromethoxy)quinoline (Z)-3-amino-1,2-bis(4-chlorophenyl)-N'-[4-[1-cyclohexyloxyethenylsulfanyl(methyl)amino]phenyl]prop-2-enediamide;ethane N-[4-[(1E,3Z)-4-[2,5-bis(trifluoromethyl)phenyl]buta-1,3-dienyl]cyclohexa-1,5-dien-1-yl]-6-chloro-2-methylpyrimidin-4-amine 3-[(2-cyclopentylsulfanylacetyl)amino]-5,7-dihydrobenzo[d][1]benzazepine-6-carboxamide (E)-N-[2,3-bis(ethenyl)phenyl]-N'-[5-(3H-benzimidazol-5-yl)pyrazin-2-yl]prop-1-ene-1,3-diamine 5-chloro-2-fluoro-N-[(1R,3S)-3-hydroxycyclopentyl]-4-(1H-pyrazolo[3,4-c]pyridin-6-ium-5-yloxy)benzamide 4-(3,5-dimethylphenyl)-2,3-bis[1-(2-hydroxyethoxy)ethyl]phenol N-[3,5-bis(trifluoromethyl)phenyl]-1-hydroxynaphthalene-2-carboxamide 1-N',3-N',2,4-tetrahydroxyanthracene-9,10-dione 1-[4-(N'-hydroxycarbamimidoyl)-2-nitrophenyl]pyrrolidine-3-carboxylic acid N-methyl-1-[4-(2,3,6-trifluorophenyl)-3,8-dihydropyrimido[5,4-d]pyrimidin-2-ylidene]methanamine N-(2,6-dioxopiperidin-3-yl)-1,4-dimethylindole-5-carboxamide 2-[(3-cyclopropylphenyl)methylidene]butanedinitrile (NE)-4,4-difluoro-5-hydroxy-2-oxopentanoic acid;[1,3-thiazol-3-ium-5-ylmethylideneamino]methanethiol N-[6-azidooxy-2,4-dichloro-3-(hydroxymethyl)phenyl]acetamide 2,6-bis[(Z)-1-aminoprop-1-enyl]pyridine-4-carboxylic acid 2-[2,5-dimethyl-4-(5-oxo-1H-tetrazol-4-yl)phenyl]acetic acid 3-azidooxy-N,2,4-trimethylbenzamide 3-[(4-fluorophenyl)methyl]-N,1-dimethylpyrazole-4-carboxamide 5-(3,4,5-trifluorophenyl)-2H-[1,2,4]triazolo[1,5-a]pyridin-8-amine 3-[4-(azidomethyl)phenyl]-N,N-dimethylpropan-1-amine 7-[2-(3,4-dimethoxyphenyl)propanoyl]-N-hydroxy-1-propanoyl-3,6-dihydro-2H-azepino[2,1-b]quinazoline-5-carboxamide 4-[4-(3-aminopiperidin-1-yl)pyridine-2-carbonyl]benzonitrile 3-[(5R)-2,4-dioxospiro[7H-thieno[2,3-d]pyrimidine-5,1'-cyclopropane]-6-yl]benzoic acid N-[3-chloro-4-(dimethylsulfamoyl)phenyl]acetamide;(2S,5R)-2-[5-(hydroxymethyl)pyrimidin-2-yl]oxy-5-nitrosooxolane-3,4-dione 5-(2,3-difluorophenyl)-N-[3-methylsulfonyl-1-oxo-1-[(4-pyrazol-1-ylphenyl)methoxy]butan-2-ylidene]-1H-pyrrole-3-carboxamide 1-[4-[[5-amino-2-(benzylamino)thieno[3,2-d]pyrimidin-4-yl]amino]piperidin-1-yl]prop-2-en-1-one 6-bromo-7-chloroquinoline-4-carboxylic acid ethane;[6-(2,4,5-trifluorophenyl)pyridin-3-yl]methanol [1-benzyl-2,4-dioxo-6-(trifluoromethyl)pyrido[3,2-d]pyrimidin-3-ium-7-yl]phosphane;bromide 3-[[5-[5-(azetidine-1-carbonyl)pyridin-2-yl]pyridin-2-yl]amino]cyclobutane-1-carboxylic acid 2-(4-chlorophenyl)sulfanyl-7H-purine 2-cyclohexyl-1-(2,4,6-trichlorophenyl)ethanone 2-[(3S,4R)-1-[2-chloro-6-methyl-5-(trifluoromethoxy)benzoyl]-4-phenylpyrrolidin-3-yl]-N-ethyl-N'-methanimidoylpropanediamide 4-ethenyl-N,2-dimethoxyaniline;7-fluoro-6-(3-fluorophenyl)-1H-quinazolin-2-one 4-[2-(3,6-dihydro-2H-pyran-4-yl)ethynyl]benzoic acid N'-hydroxy-6-[methyl(2,4,4-trimethylpentan-3-yl)amino]pyridine-2-carboximidamide (3aR,6aS)-5-(1H-indole-2-carbonyl)-N-pyridin-4-yl-3,4,6,6a-tetrahydro-1H-furo[3,4-c]pyrrole-3a-carboxamide 3-(1,3,2-benzodioxaborol-5-yl)-7-propan-2-ylidene-4H-naphthalene-1-carbonitrile 2-[4-(4-butylcyclohexen-1-yl)phenyl]-7-fluoro-6-pentoxynaphthalene 7,7-bis(3,4,5-trimethoxyphenyl)bicyclo[2.2.1]heptane 4-[2-methoxyethyl(pyridin-3-yl)amino]benzenesulfonamide N-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-6,7-dihydro-1H-indazole-4-carboxamide N-[2-(4,6-dimethoxypyridin-2-yl)ethyl]-2H-triazole-4-carboxamide [2-(5,6-dimethylpyridine-3-carbonyl)morpholin-4-yl]-[1-[2-(trifluoromethoxy)benzoyl]piperidin-3-yl]methanone 2-[5-(4-butylcyclohexyl)thiophen-3-yl]-3H-imidazo[4,5-c]pyridine 4-(4,6-dimethoxypyrimidin-2-yl)sulfanylbenzenecarboximidamide (2S,3R)-4,6,6-triethyl-5-methoxy-7-pent-1-ynyl-2,3-dihydro-1H-indene-2,3-diol N-(1,3-dimethylindazol-4-yl)-1-(2-fluorophenyl)triazole-4-carboxamide 7-(3,4-dichlorophenyl)-5-methyl-N-[2-(methylideneamino)cyclohexa-1,5-dien-1-yl]-6-oxo-8H-imidazo[1,2-a]pyrimidine-2-carboxamide 2-(2,4-difluorophenyl)-3-hydroxybutanoate 5-methylsulfanyl-3,4-bis(prop-1-enoxy)benzoic acid 3-ethoxycarbonyl-2,6-dimethylbenzoic acid (2E)-N-methyl-2,3-diphenylpenta-2,4-dienamide N'-[1,3-bis(4-methoxyphenyl)prop-2-enyl]-2H-pyridine-5-carbohydrazide 6-(5,7-dimethylfuro[3,2-c]pyridin-2-yl)-5H-pyrazolo[1,5-b][1,2,4]triazole 2-[3-[[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]sulfonyl]phenoxy]propanoic acid N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)formamide;[(E)-1-iminobut-2-en-2-yl]azanide;yttrium [6-(1,2,3,4-tetrahydroisoquinolin-7-yl)pyrazin-2-yl]methanol 1-[3-(4,5-dihydroimidazol-1-ylmethyl)-1H-indol-2-yl]ethanol 4-[3,5-dimethyl-2-[2-methyl-3-(2H-tetrazol-5-yl)phenyl]imidazo[1,2-a]pyrimidin-7-yl]morpholine [2-fluoro-4-(triazol-1-yl)phenyl]-[3-methoxy-6-(trifluoromethoxy)pyridin-2-yl]methanone 2-[1-(methylamino)propan-2-yloxy]-1,3-thiazole-5-carboxamide N'-[(Z)-(2-hydroxynaphthalen-1-yl)methylideneamino]-N-(5-methoxy-2-nitrophenyl)oxamide 6-[4-[1-(dimethylamino)ethyl]phenyl]-2-pyridin-3-ylquinazolin-4-amine 2-[4-bromobutan-2-yl(methoxycarbonyl)amino]benzoic acid (5S)-6-[4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]oxyphenyl]hexanoic acid;methane 2-(4-bromo-5,6,7,8-tetrahydronaphthalene-1-carbonyl)-3-(dimethylamino)propanoate 4-[2,3-dihydroxypropyl(1-phenylethyl)amino]benzenesulfonic acid 2-[4-(2,3-dihydro-1H-inden-5-yl)-2-ethylpyrrolidin-1-yl]pyridine 1-(2-chlorophenyl)-N-[2-fluoro-4-(2-morpholin-4-ylethoxy)phenyl]methanesulfonamide 6-chloro-7-(2-fluorophenyl)pyrido[3,4-b]pyrazine;ethane 5-(3-propan-2-ylphenyl)-1,2,4-oxadiazole 2-amino-9-[(3S,4R,5S)-3-hydroxy-4,5-dimethoxyoxolan-2-yl]-1H-purin-6-one;2,2,2-trifluoroacetic acid 2-bromo-N-(furan-2-ylmethyl)-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]benzamide 4-[5,8-dichloro-7-(3-fluorophenyl)-1H-indole-2-carbonyl]-N-[(3S)-pyrrolidin-3-yl]piperazine-1-carboxamide;hydrochloride 1-benzyl-3-[1-(2-fluorophenyl)ethyl]piperazine;methanamine 5-[2-(4,4-difluorocyclohexyl)phenyl]imidazolidine-2,4-dione (2S,5R)-1-benzyl-5-hydroxy-N'-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboximidamide;hydrochloride 2-[4-chloro-5,6-difluoro-1'-(oxan-3-yl)spiro[indole-3,4'-piperidine]-2-yl]acetonitrile 2-[5-azidooxy-3,4-di(propan-2-yl)pyridin-2-yl]-6-pyrazol-1-ylpyrimidine (2S)-1-[[4-[3,5-bis(trifluoromethyl)phenoxy]phenyl]sulfonylamino]-N-hydroxy-N'-methyl-N'-propan-2-ylazetidine-2-carboximidamide 1-azidooxy-2,3,4-tris(trifluoromethyl)benzene N-[1-cyclobutyl-3-(4-ethenylphenyl)-2H-pyrimidin-6-ylidene]hydroxylamine N-[1-(4-methylphenyl)pyrazol-3-yl]formamide 3-[4-[4-[(2S)-1,1,1-trifluoropropan-2-yl]pyridin-2-yl]pyrimidin-2-yl]oxetan-3-ol 3-[1-(6,7-dimethoxyquinazolin-4-yl)-2,5-dihydropyrrole-2-carboximidoyl]cyclobutan-1-amine;formaldehyde (5S)-4,7-dimethyl-5-propanoyl-2-[[1-[3-(trifluoromethyl)phenyl]cyclohexyl]amino]-6H-pyrazolo[1,5-a]pyrazine-3-carbonitrile N-(2,4-dinitrophenyl)-1,3-benzothiazol-6-amine 4-[3-(3-ethenylnaphthalen-2-yl)propoxy]butanal 2-[(2S)-1-(cyclopropanecarbonyl)pyrrolidin-2-yl]-6-(pyridine-3-carbonyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 1-(3-aminophenyl)-N-(diethylcarbamoyl)-4-methylcyclohexane-1-carboxamide 6-fluoro-8,9-dimethylacridine-4-carbonitrile N-(3-methylbutanoyl)-4-nitrobenzenesulfonamide 4-[2-(dimethylamino)ethyl]-N-[2-[2,6-bis(2,2,2-trifluoroethoxy)pyridin-3-yl]pyrazol-3-yl]morpholine-3-carboxamide 3-[4-(azidomethyl)phenoxy]-1,2-thiazole 1-[3,5-dimethoxy-4-(2-pyrrolidin-1-ylethoxy)phenyl]-N-ethylpentan-3-amine N-[2-amino-6-(methyliminomethyl)pyridin-3-yl]-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxamide N-(3,4-dimethylphenyl)-N'-methanimidoylbenzenecarboximidamide N-[3-(1,2,4,5-tetrazin-3-ylmethoxy)pyridin-2-yl]acetamide N-(2,5-dimethylphenyl)formamide;ethane ethane;4-(2-methylbutyl)-N-[4-(trifluoromethoxy)phenyl]benzamide 5-bromo-6-(cyclohexylamino)pyridine-3-carboxylic acid 5-[3,4-bis(trifluoromethyl)phenyl]-2-hydroxy-N-[4-(pyridine-2-carbonylamino)phenyl]benzamide;methoxycyclobutane [2-amino-3-ethylsulfonyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-[2-[(2S)-oxetan-2-yl]pyridin-3-yl]methanone 5-azidooxy-2,3-difluoro-1H-indene N-(2,2-dimethoxyethyl)-2-nitro-N-[4-(thiophen-2-ylsulfamoyl)phenyl]aniline 1-[2,3,5,6-tetrafluoro-4-(4-phenylphenyl)phenyl]propan-1-amine 2-[(Z)-3,4-dichlorohept-1-enyl]-5-phenyl-1H-imidazole (2S)-1-(2,4-dichlorophenyl)sulfinyl-N-[(4-methylpiperazine-1-carbothioyl)amino]pyrrolidine-2-carboxamide 2-[[4,5-dichloro-1-(3-fluorophenyl)-6-(trideuteriomethylamino)cyclohexa-2,4-dien-1-yl]-hydroxymethyl]phenol 1-(2,5-dichloroanilino)sulfonyl-3-[4-fluoro-2-(1-methoxybutan-2-ylcarbamoyl)phenyl]urea 2-chloro-4-phenylheptanoate 2-[2,6-dimethyl-4-(3-nitrophenoxy)phenyl]acetic acid 3-cyclopentyloxy-2-[[1-(4,6-dimethylpyrimidin-5-yl)sulfanylpiperidin-4-ylidene]amino]propanoic acid 3-[(6,7-dimethoxy-1,2,4,5-tetrahydro-3-benzazepine-3-carbonyl)amino]propanoic acid N-[4,5,6,7-tetrafluoro-2-(4-methoxyphenyl)sulfonyl-3-methylindol-1-yl]benzenesulfonamide N-[4,6-diamino-1-(cyclopropanecarbonyl)indol-3-yl]imino-3,4-dihydroxybenzamide 3-(4-bromobutyl)-N'-hydroxypyridine-2-carboximidamide 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-ethyl-5-[4-methyl-4-(methylaminosulfanyl)cyclohexa-1,5-dien-1-yl]-1,2-oxazole-4-carboxamide (3,4-dimethoxyphenyl)-[5-hydroxy-2-(trifluoromethyl)phenyl]methanone 5-[3-[7-(4-methylimidazol-1-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl]-N-propan-2-ylpyridin-3-amine 2-[(4R)-4-methyl-5,6-dihydrothieno[2,3-b]pyrrol-4-yl]ethanol 2-azido-1,6-ditert-butyl-4-(methoxymethoxy)naphthalene 3-azidooxypropylsulfanylbenzene (1S)-2,2,2-trifluoro-1-[3-(1H-indol-3-ylmethylideneamino)phenyl]ethanamine N-benzyl-N'-[4-(1,3-benzothiazol-2-yl)cyclohexa-1,5-dien-1-yl]hexane-1,6-diamine 2-[4-chloro-2-(1H-indol-3-yl)-N,5-dimethoxyanilino]-2-(oxolan-2-ylmethyliminomethyl)propanedioic acid 2-(5-ethylpyridin-3-yl)-6-[(E)-1-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)prop-1-enoxy]pyrazolo[1,5-a]pyrimidine 6-(aminomethyl)-N'-[2-(1,3-benzothiazol-2-yldiazenyl)pyridin-4-yl]pyridine-2-carboximidamide 3-(4-chlorophenyl)-N'-[[6-methyl-5-(3,4,5-trifluorophenyl)pyridin-2-yl]methyl]-1H-pyrazole-5-carbohydrazide 3-bromo-2-(bromomethyl)benzoate 1-[3-(4,4-diphenylpiperidin-1-yl)propyl]cyclohexan-1-ol;1-[4-methyl-5-(2,2,2-trifluoroethoxy)pyridin-2-yl]azepane 2-[4-(2,5-dimethylfuran-3-carbonyl)piperazine-1-carbonyl]-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-4-one 7-methylsulfanyl-4,4a-dihydroquinoline N-[2,3,5,6,7,8-hexahydro-1H-pyrrolizin-5-yl(phenyl)methylidene]hydroxylamine N-azido-3-(4-chlorophenyl)furan-2-amine 4-(4-chlorophenyl)-N'-[2,5-dimethyl-1-[4-(trifluoromethoxy)phenyl]pyrrol-3-yl]sulfonyl-3,3-dimethylbutanimidamide 3-[4-(2,3-dichlorophenyl)piperazine-1-carbonyl]pyrrolidine-1-carboxylate 1-(5,6,7,8-tetrahydroquinolin-2-yl)pentane-1,5-dione N-[3,5-bis(trifluoromethyl)phenyl]-2-[4-bromo-2-(trifluoromethoxy)phenoxy]acetamide 6-hydroxy-4,5-bis(4-nitrophenyl)-7-oxabicyclo[4.1.0]hepta-2,4-dien-3-one 3-(2,4-dichlorophenyl)-5,7-dihydropyrrolo[3,4-b]pyridin-6-one 4-cyclohexyl-6,7-dihydro-5H-1,2,3-benzotriazol-4-amine 4-[2,3-dihydroxypropyl(1,1,1,2,3,3,3-heptafluoropropan-2-yl)amino]-N-quinoxalin-2-ylbenzenesulfonamide 2-azidooxy-5,7-dimethylquinoline 1-[3,5-bis(trifluoromethyl)phenyl]pyrrolidine-2,4-dione N-[4-chloro-3-(trifluoromethyl)phenyl]-1-[2,5-dihydroxy-1-[3-methylsulfonylpropyl(sulfinoamino)carbamoyl]cyclohexyl]methanimine 3-azido-N,4-dimethylbenzamide 2,3-dichlorobenzaldehyde;1-[(E)-2-fluoroprop-1-enyl]azepane (5Z,7E)-4-[5-(aminomethyl)furan-2-carbonyl]-1H-1,4,8-triazecin-7-one 3-[5-(3,4-dichlorophenyl)-1-[2-methyl-6-(oxan-4-yl)pyridine-3-carbonyl]pyrazol-3-yl]propanoic acid 4-amino-2-methyl-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide;1-ethyl-3-phenylbenzene 2-azido-6,7-dimethoxyquinazolin-4-amine 4-[1-(4-chlorophenyl)propan-2-yl]benzoate 4-(dimethylamino)-N-[(2E,3Z,5Z)-5-ethylidene-2-hydroxyhepta-3,6-dienyl]pyridine-3-carboxamide 5-(2-nitrophenyl)-3,6-dioxatetracyclo[12.4.0.02,7.08,13]octadeca-1(18),2(7),8,10,12,14,16-heptaene 4-[[3-[3,5-bis(trifluoromethyl)phenyl]pyrrolidine-1-carbonyl]amino]benzoic acid 5-chloro-4-[2,3-difluoro-5-(1H-pyrazolo[3,4-b]pyridin-6-yl)phenyl]pyrimidine N-[2-(5-chloro-1,3-benzothiazol-2-yl)propan-2-yl]-2-methyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-5-carboxamide 2-[(6-chloro-1,3-benzothiazol-2-yl)amino]-N-cyclohepta-1,4,6-trien-1-ylacetamide 1-(3,4-dimethylcyclohex-2-en-1-yl)sulfonyl-4-[(E)-pent-3-enyl]benzene N-[(4S)-3,4-dihydro-2H-chromen-4-yl]-4,5-dimethylfuran-2-carboxamide 1-[(5S,7R)-2,5-dimethyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]ethanone [1-(2,6-difluorophenyl)-2-hydroxyethylidene]carbamic acid ethane;5-[2-fluoro-4-(5-hydroxypentoxy)phenyl]-2,3-dihydrothieno[3,4-c]pyrrole-4,6-dione N-butyl-1-(6,7-dihydro-4H-pyrano[3,2-d][1,2]oxazole-3-carbonyl)-N-methylpyrrolidine-3-carboxamide (2R)-2-amino-3-[3-[1-[2-hydroxy-4-[(3-oxomorpholin-4-yl)methyl]phenyl]-2-methyl-5-oxopyrazol-4-yl]indol-1-yl]propanal 2-(2,4-dimethylphenyl)-N,2-diethoxy-2-phenylacetamide N-(2,5-dimethylphenyl)-1-(6-oxo-1H-pyrimidine-4-carbonyl)piperidine-3-carboxamide 2-(1,3-benzothiazol-6-ylamino)-7-oxo-8H-[1,2]oxazolo[5,4-b]quinoline-3-carbonitrile 5-(2,3-dichlorophenyl)sulfanyl-4-methyl-1H-pyrazole (Z)-3-[4-(1-acetyloxyethenylsulfanyl)phenyl]prop-2-enoic acid 5-amino-4-(3,4-difluorophenyl)-2-ethylsulfanyl-1H-pyrimidin-6-one 2-(benzylamino)-6-methylbenzaldehyde 6-(1H-benzimidazol-2-yl)-5,7-dihydropyrazolo[3,4-d]pyrimidine 1-[2-[2-(5-chloronaphthalen-2-yl)cyclopropyl]-4-fluorophenyl]ethanone 7-azido-2,3,5,6,8,9-hexamethylbenzo[g]quinoxaline N-(5-chloropyrimidin-2-yl)-4-[1-(2,6-difluorophenyl)ethylamino]piperidine-1-carboxamide 2-azido-1,3-bis(difluoromethyl)-5-methoxybenzene [4-(3,5-dimethylphenyl)piperazin-1-yl]-phenylmethanone 1-[(2S,4R)-4-hydroxy-2-phenylpiperidin-1-yl]-2-[3-methoxy-6-(3-methyl-1,2,4-triazol-1-yl)pyridin-2-yl]ethanone N-(5-acetylpyridin-2-yl)-3,4-difluorobenzamide N-[(2,5-difluorophenyl)methyl]-6-[3-(trifluoromethoxy)pyridin-1-ium-2-yl]pyridine-2-carboxamide N-[(3,4-dimethoxyphenyl)methyl]-1,6-naphthyridine-2-carboxamide 1-(2,4,5-trifluorophenyl)sulfanylpiperidine (4R)-1-[3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-N-methyl-4-propan-2-ylpyrrolidin-3-amine (3R)-1-[2-(4-benzylpiperidin-1-yl)acetyl]-N-[1-(3,4-dichlorophenyl)ethyl]pyrrolidine-3-carboxamide 2-[4-[(3S)-1-[(3,5-dimethylpyridin-4-yl)methyl]piperidine-3-carbonyl]piperazin-1-yl]acetic acid N-(2-methoxyethyl)-4-[2-[6-oxo-3-[1-phenyl-5-(trifluoromethyl)pyrazole-3-carbonyl]pyridazin-1-yl]propoxy]benzamide 3-azido-4-methoxy-2,6-dinitroaniline N-[(3R,4S)-1-tert-butyl-4-phenylpyrrolidin-3-yl]-3,5-dimethoxybenzamide 3-[2-[4-(ethylamino)phenyl]quinolin-6-yl]-N,N-dimethylpropanamide 1-azido-2,3-dichloro-4-(3-nitrophenyl)benzene (2S)-N'-benzyl-N-[3,5-dichloro-4-(1H-indol-3-yl)phenyl]-2-hydroxybutanehydrazide (Z,3E)-3-[1-amino-2-methyl-4-(3-piperidin-1-ylpropoxy)iminobutylidene]-5-chloro-N'-[5-(3-chlorophenoxy)pyrimidin-2-yl]-2-hydrazinylpent-4-enimidamide (2S)-3-(N'-hydroxycarbamimidoyl)imino-2-naphthalen-1-ylpropaneperoxoic acid N-(3,3-dimethylbut-1-en-2-yl)-5-[7-fluoro-3-[4-(4-fluorophenyl)-1H-imidazo[4,5-c]pyridin-2-yl]-2H-indazol-5-yl]pyridin-3-amine 3-(1H-indol-5-yl)-7-methoxychromene-2,4-dione (E,2S)-N-[3-(1H-indazol-6-ylmethyl)phenyl]-4-(4-methoxypiperidin-1-yl)-2-propan-2-ylidenebut-3-enamide 5-amino-2-(2,4-dioxopyrrolidin-1-yl)-N-[[3-[[methoxy(methyl)carbamoyl]amino]phenyl]methyl]pentanamide 2-amino-4,8-dichloropyrazolo[1,5-a]quinoxaline-3-carbonitrile;ethane 2-[(E)-5-chloro-6-methylhept-4-en-3-ylidene]-1,6-dihydropyrrolo[2,3-b]pyrrole;propane 2-[3-(4,5-dihydroimidazol-1-yl)propoxy]-N-methylbenzamide 3-[2-[4-(4,5-dihydro-1H-imidazol-2-ylamino)benzoyl]anilino]propanoic acid (2R,3S)-N,2,3-trimethyl-1,4-bis[(4-nitrophenyl)sulfonylamino]butanamide N-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide N-[3-fluoro-2,4-di(propan-2-yl)phenyl]-5-(2-hydroxypropan-2-yl)pyridine-3-carboxamide 3-(2,6-dimethylpyridin-4-yl)-5-[1-(4-fluorophenyl)indazol-5-yl]-N-propan-2-ylaniline 3-[[2-[4-(4,6-dimethoxypyrimidin-2-yl)piperazine-1-carbonyl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]amino]benzonitrile 7-[3-(hydroxymethyl)pyrrolidin-1-yl]-4-oxo-N-pentylchromene-2-carboxamide N-[4-[2-(3,6-dihydro-2H-pyran-5-yl)ethynyl]phenyl]pyridine-3-carboxamide N-[4-(2,5-dioxopyrrolidine-1-carbonyl)-3-fluorophenyl]-2-propan-2-ylbenzamide 3,6-difluoro-N-[1-[[4-(trifluoromethyl)phenyl]methyl]pyrazol-3-yl]pyridine-2-carboxamide 5-[(3S)-1-benzoylpyrrolidin-3-yl]oxypyridine-2-carboxylic acid (3R)-N-benzyl-2-(2,4-dimethoxyphenyl)-6-methylidenecyclohexan-1-amine N-(2,4-dichloropyrimidin-5-yl)-N-[6-(4-methoxyphenyl)pyridazin-3-yl]nonanamide 1-benzylpiperidine;2-[(3R)-2,6-dioxopiperidin-3-yl]-4-methoxyisoindole-1,3-dione 2-ethyl-7-[(E)-2-methoxyethenyl]sulfanylquinoline N-(3,4-difluorophenyl)-2-methylpiperidine-1-carboxamide N-[2-amino-4-(1H-pyrazole-5-carbonyl)phenyl]-7,8-dimethoxyquinoline-6-carboxamide [2-(3,4-dimethoxyphenyl)azepan-1-yl]-(6-methylcyclohexa-2,4-dien-1-yl)methanone 1,3-diethyl-5-(2-nitrophenyl)benzene 2-[[3-(3,5-difluorophenyl)piperidin-1-yl]methyl]-6-ethoxy-3H-quinazolin-4-one 4-ethyl-2-methyl-N-(3-pyridin-3-ylphenyl)pentanamide N-[4-[(5-bromopyridin-2-yl)-propan-2-ylamino]phenyl]sulfonylbenzamide 1-methylsulfanyl-3-[4-(trifluoromethoxy)phenyl]benzene 1-(4-hydroxy-5,6,7,8-tetrahydroquinazolin-2-yl)piperidine-3-carboxylic acid 1-[4,4-diamino-5-oxo-2-(3,3,3-trifluoropropyl)imidazolidin-1-yl]ethanone 6-methyl-1,5-dihydropyrazolo[3,4-d]pyrimidine-2-sulfonic acid N-[2,6-difluoro-4-(1H-indazol-5-yl)phenyl]-8-methoxyquinoline-3-carboxamide 1-(2,3-dihydrofuran-5-yl)-6-(4-methylsulfanylphenyl)-2H-quinazoline 4-bromo-2,6-dichloro-N-(2-hydroxyethyl)benzenesulfonamide 1-N,2-N-dimethyl-3-[2-(1-pyridin-3-ylethenoxy)ethoxy]benzene-1,2-diamine 2-[4-(4-benzylpiperazine-1-carbonyl)piperidin-1-yl]-N-[3,5-difluoro-4-(trifluoromethylsulfonyl)phenyl]-N'-hydroxy-2-oxoethanimidamide ethane;4-(5-methylpyridin-3-yl)oxybenzamide 1-[4-[4-[(3R)-3-aminopyrrolidine-1-carbonyl]phenyl]sulfonylpiperazin-1-yl]ethanone;2,2,2-trifluoroacetic acid 2-[(5R)-4-oxo-2-[5-(4-phenoxybutylsulfonylamino)pyridin-3-yl]imino-1,3-thiazolidin-5-yl]acetic acid (6S)-2,6-dimethyl-3-methylidene-8,9-dihydropyrano[3,4-f]quinoline 1-[(2R)-4,5-dihydroxy-7-oxo-3-phenylnonyl]pyrrolidine-2-carboxylic acid 6-azido-2-(3,4-dichlorophenyl)-[1,2,4]triazolo[4,3-a]pyrazin-3-one N-[6-(4-fluorophenyl)imidazo[1,2-b]pyridazin-3-yl]-5-methoxypyridine-2-carboxamide N-[(1R,3S)-3-[1-[3-chloro-4-(trifluoromethoxy)phenyl]-5-hydroxytriazol-4-yl]cyclohexyl]-2,6-dimethoxypyridine-4-carboxamide (2R)-1-acetyl-N'-[5-chloro-4-cyano-6-(trifluoromethoxy)pyridin-3-yl]-N,N,2-trimethylpyrrolidine-2-carbohydrazide 4-[2-bromo-N-(3,5-dichlorophenyl)anilino]benzenesulfonic acid [4-(2-morpholin-4-ylethoxy)phenyl]boronic acid 4-[2,2-dimethoxyethyl(propyl)amino]benzenesulfonamide N-(furan-2-ylmethyl)-3-phenylbutanamide 1-azidooxy-3-phenylpropan-2-amine 1-(4,5-dimethylfuran-2-carbonyl)-N-methylpiperidine-3-carboxamide 4-[(2,6-difluorophenyl)methylamino]pyridazine-3-carboxamide N-[6,7-bis(ethenyl)-4,5,10,11-tetrahydro-3H-azepino[2,1-c][1,4]benzoxazin-8-yl]benzenesulfonamide (5Z)-2-(3,4-dimethylphenyl)imino-5-[(1,2,2,4,7-pentamethylquinolin-6-yl)methylidene]-1,3-thiazolidin-4-one 4-[1-(2,5-dimethylthiophene-3-carbonyl)piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one 1-(4,5-dichlorocyclohexa-2,4-dien-1-yl)oxy-3-[4-(naphthalen-2-ylsulfanylamino)butyl]urea (1S,2R)-4-fluoro-4-phenylmethoxycyclohexane-1,2-diol 3-[2-(butanoylamino)phenyl]-N-cyclopropyl-N-methylpropanamide 1-[2,2-diethoxyethyl(1H-inden-5-yl)amino]propan-2-one 2-methylsulfanyl-6-[(E)-2-pyridin-4-ylethenyl]quinazolin-4-amine 1-[(1R,2R)-2-fluorocyclobutyl]-3-(pyridin-4-ylmethoxy)pyrazolo[3,4-d]pyrimidin-4-amine 5-(4-ethylphenyl)-3H-furan-2-one 6-tert-butyl-N-[3-(4,5-dihydro-1H-imidazol-2-ylmethoxy)naphthalen-2-yl]thieno[2,3-d]pyrimidine-4-carboxamide 5-(2,4-difluorophenyl)sulfanyl-1H-indazole N-azido-5-tert-butyl-2,4-dimethoxyaniline 2-[(3S)-4,5-dimethylpyrrolidin-3-yl]-N-[1-oxo-1-(4-phenylpiperidin-1-yl)propan-2-yl]acetamide 1-(4,5,6,7-tetramethylnaphthalen-2-yl)ethanone 6-(cyclopropylmethoxy)-7-ethyl-1,2,3,4-tetrahydronaphthalene 4-[[6-(3,4-dihydropyridin-4-yl)pyridine-2-carbonyl]amino]piperidine-1-carboxylic acid 3-(4-amino-N-azidoanilino)benzonitrile ethane;3-methyl-1,4-bis[(E)-2-(3,4,5-trihydroxyphenyl)ethenyl]pyridin-2-one 4-[(2S)-1,3-dihydro-2-benzofuran-5-yl]morpholine 4-(2,4-dichlorophenyl)sulfinyl-N,3-diethyl-1H-indole-2-carboxamide (4aS,7S,8aS)-6-ethyl-N-[(2R)-2-hydroxypropyl]-1-methyl-4,4a,5,7,8,8a-hexahydro-3H-1,6-naphthyridine-2-carboxamide;dihydrochloride [3-[(1,5-dimethylpyrazole-4-carbonyl)amino]phenyl]boronic acid 5-(2,6-dichlorophenyl)-N-[2-[4-(3-oxomorpholin-4-yl)cyclohexanecarbonyl]phenyl]furan-2-carboxamide 2-[(4-benzylphenyl)methylideneamino]acetohydrazide 3-chloro-1-methyl-5H-pyrrolo[2,3-b]pyrazine;(Z)-N-ethylidenebut-2-enamide N-[(3S)-7-benzyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]carbamate [3-(difluoromethyl)azetidin-1-yl]-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-2-yl)methanone [1-[1-[4-(azetidin-3-yloxy)phenyl]piperidin-4-yl]cyclopropyl]carbamic acid 2,5-difluoro-4-(7-hexylsulfanylheptylamino)-N-phenylmethoxybenzamide N-[4-fluoro-3-(trifluoromethyl)phenyl]-1,3-dihydroxy-6-oxopyridazine-4-carboxamide 2-(1-benzylpyridin-1-ium-4-yl)sulfanylacetamide 3-methyl-4,5,6,7-tetrahydroindazole-1-carboxylic acid 3-(4-acetyloxyphenyl)-2,2-dichlorocyclopropane-1,1-dicarbonitrile 1-azidooxy-4,5-dimethyl-2-(3-phenylprop-2-enoyloxy)benzene N-cyclopentyl-4-[2-methoxyethyl(methyl)amino]-2,6-dimethylpyrimidine-5-carboxamide 1-(3,4-dihydroxybutyl)-6-iodo-2-oxoquinoline-5-carboxylic acid N-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-propan-2-ylpyrimidin-2-yl]-1H-indole-4-carboxamide 4-[2-(5,6-difluoroindol-1-yl)ethoxy]benzonitrile 3-(2-phenylethyl)-N-[1-(4,5,6,7-tetrahydro-1H-indazole-4-carbonyl)piperidin-4-yl]benzamide 2-tert-butyl-N'-[(4-methylphenyl)-dipyridin-2-ylmethylidene]propanediamide 3-(5-methyl-2,4-dioxopyrimidin-1-yl)sulfanylbenzonitrile 2-amino-3,4-dihydronaphthalene-1-sulfonic acid 2-(5-phenyl-3,4-dihydropyrazol-2-yl)-1H-indole 1-(4-bromophenyl)-3-(1H-indol-2-ylamino)thiourea 2-methyl-3H-benzo[e]indole-4,9-dione [2-[6-(hydroxymethyl)pyridin-3-yl]pyrrolidin-1-yl]-[5-propan-2-yloxy-4-[3-(trifluoromethyl)pyrazol-1-yl]pyridin-2-yl]methanone 3,4-dichloro-N-[(1S,2S)-1-phenylbut-3-en-2-yl]benzenesulfonamide 6-bromo-2-chloro-5-ethynylpyridine-3-carboxylic acid 5-chloro-6-[4-(trifluoromethyl)pyrazol-1-yl]pyridin-3-ol N-[4-[2-(cyclohexylamino)ethyl]phenyl]-2,5,11,13,15-pentazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),3,5,7,9,11,16-heptaen-10-amine (2S)-2-[4-[2,6-bis(3,5-dimethylpyrazol-1-yl)pyridine-4-carbonyl]piperazin-1-yl]propanoic acid 3-[4-(3,5-dimethoxyphenyl)-1H-benzimidazol-2-yl]-5-pyridin-2-yl-2H-pyrazolo[3,4-b]pyridine N-[4-cyano-1-(cyclopentylcarbamoyl)pyrazol-3-yl]-2,6-dimethoxypyridine-4-carboxamide N'-[4-(2,3-dihydro-1H-inden-5-yloxy)pyridin-3-yl]-4-[4-(hydroxymethyl)phenyl]piperidine-1-carboximidamide 2-amino-4,5-bis[(Z)-1-phenylprop-1-enyl]thiophene-3-carbonitrile 2-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one 2-bromo-5,6-dimethoxybenzo[g][1]benzothiol-7-ol 3-[(E)-hydroxyiminomethyl]-2-propan-2-ylpyrido[1,2-a]pyrimidin-4-one 4-[(2R,4S)-1-tert-butyl-4-fluoropyrrolidine-2-carbonyl]piperazin-2-one 2-(N-ethenylsulfonylanilino)benzenesulfonic acid 2-[(4,6-dihydroxycyclohexa-1,5-dien-1-yl)methylidene]propanedinitrile;rhenium 2-(4,5-difluoro-1H-indol-3-yl)-6-methoxyquinoline 3-(2-butoxyethyl)-5-methoxy-1H-indole 4-[(3-methoxyphenyl)methyl]-2-methyl-6-propan-2-ylpyrimidine 2-(4-methoxyphenyl)-6-methylsulfanylnaphthalene 4-azido-2,3,5-trimethylbenzenesulfonic acid 2-[(3R,4S)-3-amino-4-fluoropiperidin-1-yl]-7-butan-2-yl-5H-pyrrolo[2,3-b]pyrazine-6-carboxamide 3-[4-(2,6-diphenylpyrimidine-4-carbonyl)piperazin-1-yl]sulfonylphenol 5-chloro-3,6-dimethylpyrimidine-2,4-dione;ethane [4-(5-amino-2H-tetrazol-1-ium-1-yl)phenyl]-bis(3-methoxyphenyl)sulfanium 1-[3-chloro-5-(3-hydroxypentoxy)phenyl]ethanone;propane 1-N',4-N-dibutylbenzene-1,4-dicarboximidamide [3-(2,4-dihydroxy-5-propan-2-ylphenyl)-1H-phenanthro[9,10-b]pyrrol-6-ylidene]azanide;uranium(2+) 6-methoxy-4,10-dihydropyrazolo[3,4-c][1]benzazepine 5-(1,4-diazepan-1-yl)-N'-hydroxypyridine-2-carboximidamide 1-[(2,4-difluorophenyl)methyl]-3-[4-(trifluoromethoxy)benzenecarbothioyl]quinolin-4-one 2-[4-(1,1-dihydroxythiolan-3-yl)sulfonylphenyl]benzoic acid (1S,5R)-2-[4-[4-chloro-3-(trifluoromethyl)phenyl]sulfonylpiperazine-1-carbonyl]-N-hydroxybicyclo[3.1.0]hexane-1-carboxamide (3R)-3-(2,4-dioxo-1H-quinazolin-3-yl)piperidine-1-carboxylic acid 1-[2-(4-propan-2-ylphenyl)acetyl]piperidine-3-carboxamide N-[(5E)-1-[2-[3-(4-methoxybenzoyl)indol-1-yl]acetyl]-5-[(2Z,4Z,6Z)-nona-2,4,6-trienylidene]pyrazol-4-ylidene]methanimidamide 2,6-dichloro-4-(tribromomethyl)phenol 2-[3,5-dibromo-4-(3-cyclobutyl-1H-indol-5-yl)phenyl]propan-2-ol 2,3-diaminopropanoic acid;1-[4-(furan-2-carbonyl)phenyl]-2-methylpropan-1-one (2S)-1-[2,6-bis(trifluoromethyl)benzoyl]-N-(oxan-4-yl)pyrrolidine-2-carboxamide 6-hydroxy-5-[(2-hydroxynaphthalen-1-yl)diazenyl]-4-methoxynaphthalene-2-sulfonic acid 2-(4,5-dihydrobenzo[g][1]benzoxepin-3-yl)ethanol 4-fluoro-N,2-dimethylbenzamide;6-(5-methoxypyridin-3-yl)-2-[(Z)-(2-oxo-1H-indol-3-ylidene)methyl]-4-piperidin-4-ylpyridazin-3-one (3R)-N-[2-[(E)-N'-hydroxycarbamimidoyl]pyridin-4-yl]oxolane-3-carboxamide 5-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]furo[2,3-c]pyridine 6-bromo-1,2,3a,4,5,9b-hexahydrobenzo[e]indole 3-[4-amino-1-(2-methoxyethyl)pyrazolo[3,4-d]pyrimidin-3-yl]-N-(3,5-difluorophenyl)-N'-methylcyclopentane-1-carbohydrazide (2S,3aS)-N-[6-(dimethylamino)pyridazin-3-yl]-1-[(4-methoxyphenyl)methyl]-5-oxo-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrole-2-carboxamide 2-[5-fluoro-6-(1,3-thiazol-4-yl)pyridin-3-yl]acetamide 3-[4-(cyclohexylcarbamoyl)phenyl]-N-ethoxy-N-propan-2-ylpyrrolidine-1-carboxamide;hydrochloride 3-[1-azido-2,4-bis(trifluoromethyl)cyclohexa-2,4-dien-1-yl]phenol (Z)-1-(6-chloro-4-cyclopropyloxypyridin-2-yl)but-2-en-1-imine 4-[2-(4-hydroxyphenyl)ethyl]-5-iododithiol-3-one N-[4,5-dihydroxy-2-(hydroxymethyl)phenyl]methanesulfonamide 2-[azido(bromo)methyl]naphthalene 2-[2-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-ylmethyl)piperidin-4-yl]oxyethylamino]quinoline-3-carbonitrile;dihydrochloride 4-N-[2-(1,3-benzodioxol-5-yl)ethyl]-6-N-methylpyrimidine-4,6-diamine N-(4-fluorophenyl)-3,8,10-triazatricyclo[7.4.0.02,6]trideca-1(9),2(6),3,11-tetraene-12-carboxamide 4-[(E)-2-nitroethenyl]benzenesulfonic acid (5R,7S)-N-[[2-chloro-3-[(1-cyanocyclopentyl)methoxy]phenyl]methyl]-1,4,5,7-tetrafluoro-2,5-dihydropyrano[3,4-c]pyrazole-6-carboxamide 4-[6-(2,3-dichlorophenyl)-5,6-dihydropyrimido[4,5-d]pyrimidin-1-yl]benzenesulfonamide 3-[6-(difluoromethyl)pyridine-2-carbonyl]-1H-pyridazin-6-one 1-(2,3-dihydro-1H-inden-5-yl)ethanone;propane 3-chloro-N,7-dimethylimidazo[1,2-a]pyridine-6-carboxamide N-ethyl-3-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)benzenesulfonamide;hydrochloride 4-[4-(2,3-dimethylbutanoylamino)anilino]piperidine-1-carboxylic acid 7-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]-N-[(3S)-oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide N-(3-acetamido-5-methylphenyl)-2-[4-[2,6-dichloro-4-(trifluoromethylsulfanylamino)phenoxy]phenoxy]acetamide [[5-(aminomethyl)pyrimidin-2-yl]-[4-fluoro-3-methoxy-2-(1-methylcyclopropanecarbonyl)phenyl]methylidene]azanium N-[[4-(3,5-difluorophenyl)cyclohexyl]methyl]piperidine-1-carboxamide 1-N,5-N,2-trimethyl-5-N-[(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)methyl]piperidine-1,5-dicarboxamide 5-azido-4-(3,6-dihydro-2H-1,4-oxazin-5-yl)pyrimidin-2-amine N-[4-(dimethylamino)phenyl]-4-nitro-N-propylbenzamide 1-[2-(5-azidopyridin-3-yl)phenyl]ethanone N-[(Z)-1H-indol-3-ylmethylideneamino]-5,6,7,8-tetrahydronaphthalene-2-carboxamide N-(1,3-benzothiazol-6-yl)-2-(3-methoxyphenoxy)-5-sulfanylbenzamide 2-[4-[(3S)-3-ethyl-4-methoxypiperidine-1-carbonyl]pyrazol-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxylic acid 6-chloro-3-[2-(4,5-diethyl-1H-imidazol-2-yl)ethyl]-1,2-benzoxazole N-[6-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-7,8-dihydronaphthalen-2-yl]-1-methylindole-4-sulfonamide 1-[(3,5-difluorophenyl)methyl]-3-[(2R)-4-hydroxybutan-2-yl]-6-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)pyridine-2-carbonitrile 4-(2,6-difluorophenoxy)-N-[1-[5-(5-methoxypyridin-3-yl)pyrimidin-2-yl]butylideneamino]aniline;ethane 6-butyl-3-methoxy-N,N-dimethylpyridazine-4-carboxamide 1-[4-(2-cyclohexylethynyl)phenyl]-3-cyclopenta-1,4-dien-1-ylurea 5-(4-fluorophenyl)sulfanyl-1,2,3,6-tetrahydropyrrolo[3,4-c]pyrrol-8a-amine;hydrochloride 3-aminosulfanyl-N'-(5,6-difluorocyclohexa-1,5-dien-1-yl)-4,5-dimethoxybenzenecarboximidamide 1-(2,6-dimethylphenyl)-5-[[4-[[3-(2-methoxyphenyl)phenyl]carbamoylamino]phenoxy]methyl]pyrazole-3-carboxylic acid 6-(3,5-dimethoxy-4-propan-2-ylphenyl)-1H-benzimidazole [2-(6-chloropyridin-3-yl)-1,4-oxazepan-4-yl]-[3-(trifluoromethyl)phenyl]methanone 7-chloro-N-[2-(6,7-dimethoxyquinazolin-4-yl)ethylidene]quinoline-3-carboxamide 5-tert-butyl-3,4,6-trichloro-1H-indole N-[3,6-dimethyl-2-(3-propan-2-ylcyclobutyl)oxyphenoxy]ethanethioamide 1-cyclobutyl-N-[(3R)-piperidin-3-yl]thieno[2,3-c]pyrazole-5-carboxamide;hydrochloride 1-[2-(3,5-difluorophenyl)ethyl]piperidine;hydrochloride 3-bromo-6-[2-(3,4-dimethoxyphenyl)ethyl]quinoxaline 3-cyclohexyloxynaphthalene-2,7-disulfonic acid N-(2,3-dichlorophenyl)-4H-1,2,5-oxadiazol-5-imine 6-methyl-7-[4-(6-phenylpyrimidin-4-yl)piperazine-1-carbonyl]pyrazolo[1,5-a]pyridine-3-carbonitrile 2-methoxy-6-[[6-(trifluoromethyl)pyridin-3-yl]iminomethyl]phenol 3-amino-4-[2-hydroxyethyl(methyl)amino]cyclobut-3-ene-1,2-dithione;N'-amino-4-(3-fluoroanilino)thieno[3,2-c]quinoline-7-carboximidamide 2-[7-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)furo[3,2-c]pyridin-2-yl]-4,5-dihydro-1H-imidazole 1-[2,4-dichloro-5-methoxy-3-[[(Z)-prop-1-enyl]sulfanylamino]phenyl]ethanone N-[6-(3,4-dichlorophenyl)pyridin-2-yl]-1H-pyrrole-3-carboxamide 3-[[5-[(2E,4Z)-6,6-dimethylhepta-2,4,7-trien-3-yl]furan-2-carbonyl]amino]-N-[1-[4-[1-[1-(trifluoromethoxy)ethenylsulfanyl]ethenyl]phenyl]ethyl]azetidine-1-carboxamide 1-cyclopropyl-4-(3,6-diphenylcarbazol-9-yl)benzimidazole 2-N,4-N-bis[3-(dimethylamino)phenyl]thiophene-2,4-disulfonamide 2-azido-5-tert-butyl-4-chloro-N-(4-methoxyphenyl)aniline 2-[(5Z)-5-[(6-hydroxynaphthalen-1-yl)methylidene]-4-oxo-3-sulfanylidenethiolan-2-yl]acetic acid 4-chloro-2,6-dimethoxypyrimidine-5-carboxamide (5E)-2-(4-chlorophenyl)imino-5-[(1,3-dimethylindol-6-yl)methylidene]-1,3-thiazolidin-4-one 1,4-bis[(4-fluorophenyl)methyl]benzene;ethane 6-[1-[2,6-dimethyl-4-(methylideneamino)phenyl]ethenoxymethyl]pyridine-2-carboxylic acid 1-(3,3,4,6-tetramethylheptan-2-yl)imidazole [2-hydroxy-3-(morpholine-4-carbonyl)phenyl]urea 3-[4-(pyridine-3-carbonyl)piperazin-1-yl]benzoic acid [1-(cyclohexylmethyl)pyrazol-3-yl]-(7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)methanone;2,2,2-trifluoroacetic acid 2-methyl-2-[2,3,5,6-tetrafluoro-4-(trifluoromethyl)phenyl]oxirane 3-azido-N'-[2-(cyclopropanecarbonylamino)pyrimidin-5-yl]-1,4-dihydroindeno[1,2-c]pyrazole-6-carboximidamide (4-chlorophenyl)-(2,5-dihydrofuran-3-ylmethylidene)azanium 5-(9H-fluoren-1-yl)-4,6-dimethoxypyrimidine 4-(1,3-benzoxazol-2-ylsulfanyl)butanenitrile 6-(4-chlorophenyl)-2,3-dihydroimidazo[1,2-a]pyrimidine 2-[(3R)-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfonylpyrrolidin-3-yl]-3H-benzimidazole-5-carboximidamide (4S)-3,6-dichloro-5-[2-(3,4-dimethoxyphenyl)ethyl]-4-propan-2-yl-1,4-oxazepane 2-[(2,6-dichlorophenyl)methylsulfanyl]-4-propyl-1H-pyrimidin-6-one 1-(2,3-dihydro-1H-inden-2-yl)-4-[7-(trifluoromethoxy)imidazo[1,2-a]pyridine-3-carbonyl]piperazin-2-one N-methyl-5-[3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-amine 2-(ethylamino)-N-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]benzamide 6-[(2,3-dichlorophenyl)methyl]-1H-pyrimidine-2,4-dione 4-[4,6-bis(6-hydroxyhexoxy)-1,3,5-triazin-2-yl]phenol 4-[2-[3-chloro-4-(morpholin-4-ylmethyl)phenyl]-1,3-thiazol-5-yl]pyrimidin-2-amine 3-[[5-(2,6-dioxopiperidin-3-yl)-6-oxo-4H-thieno[3,4-c]pyrrole-4-carbonyl]amino]pyrrolidine-1-carboxylate 3-(N-(2,4-dioxo-1H-pyrimidin-5-yl)-2-methoxyanilino)propanoic acid 2-[5-(3,4-dichlorophenyl)furan-2-yl]-N'-hydroxy-1H-imidazo[4,5-b]pyridine-7-carboximidamide 2-[2,3,5,6-tetrafluoro-4-(furan-2-yl)phenyl]-1H-pyrrole N-[(3R)-1,1,2,3,4-hexamethylinden-5-yl]thiohydroxylamine 2-(3,4-dimethoxyphenyl)-1-iodoindole 5-[2,4-bis(3,4-dichlorophenyl)piperazine-1-carbonyl]-N,N-dimethyl-2H-pyridine-1-sulfinamide 4-[3-(cyclopropylmethoxy)phenyl]butanenitrile N-[2,4-dichloro-3-(pyridine-2-carbonylamino)phenyl]-5-oxopentanamide 3-bromo-7,8-difluoroquinoline 5-methyl-N,2,4-triphenyl-1H-pyrrole-3-carboxamide 2-methylsulfonyl-6H-pyrido[1,2-d]pyrimidine 1-(3,6-dimethylpyrazin-2-yl)-N-(4-thiophen-3-yloxan-4-yl)piperidine-3-carboxamide 1-(3,4-dihydroquinoxalin-2-ylmethoxy)butan-2-one;N-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)cyclohexanecarboxamide 5-fluoro-2-(9-methoxycarbonyl-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)benzoic acid 2-aminoacetaldehyde;2-N,5-N-dimethyl-1H-indene-1,2,6-triamine;ethane 5-N-cyclopropylsulfanyl-6,7-difluoroquinoxaline-2,3,4,5-tetramine 6-[[(2Z)-2-[[4-bromo-2-(trifluoromethylsulfanylamino)phenyl]methylidene]hydrazinyl]methyl]pyridine-3-carboxylic acid 2,4-diphenyl-1H-pyrazol-5-one 2-(5,6-difluoro-1H-indol-3-yl)-4-N-pyrimidin-5-yl-6-N-[4-(trifluoromethoxy)phenyl]-1H-pyrimidine-4,6-diamine 1-(3,5-dichlorophenyl)-6-hydroxy-5-[[2-(4-methylpiperazine-1-carbonyl)quinolin-8-yl]diazenyl]pyrimidine-2,4-dione N-[4,6-dimethyl-2-[(1Z)-1-methylsulfanylbuta-1,3-dienyl]pyrimidin-5-yl]-5-ethoxy-2-iodopyridine-3-carboxamide N-[3-[(1Z)-buta-1,3-dienyl]-2-methylphenyl]propanamide 3-amino-4,5-dichlorobenzoate 5-butyl-2-(4,6-diphenylpyrimidin-2-yl)oxy-1H-benzimidazole 1-(4,5,6,7-tetrahydro-1H-indol-2-yl)benzimidazole 4-[1-[(3,5-dimethylphenyl)-phenylmethoxy]ethyl]benzoic acid 3-[(E)-[4,5-dimethyl-1-(2-pyrrolidin-1-ylethoxycarbonyl)pyrrol-2-yl]methylideneamino]-6-methylquinoline-8-carboxylic acid 3-[6-[(4-methylsulfonylphenoxy)methyl]pyridin-2-yl]cyclopropane-1,1,2,2-tetracarbonitrile 2-(4-oxopiperidin-1-yl)-N-[3-(pyrrolidine-1-carbonyl)phenyl]acetamide 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-4-[[4-(1-methylpiperidin-4-yl)oxycyclohexa-2,4-dien-1-yl]amino]-1H-1,2,4-triazole-5-thione (4-cyclopropylmorpholin-2-yl)-(7,8-difluoro-6H-pyrano[3,2-c]pyrazol-3-yl)methanone (3-chloro-5,6-dihydrobenzo[b][1]benzoxepin-8-yl)methanol 2-chloro-N-cyclobutyl-7,9-difluoroimidazo[1,2-c]quinazoline-3-carboxamide 2-N-(6-methoxypyrimidin-4-yl)-1-N,2-N-dimethylbenzene-1,2-disulfonamide (1S)-2,3-dihydro-1H-indene;formic acid 1-[(2S,5R)-3-amino-4-hydroxy-5-methyloxolan-2-yl]pyrimidine-2,4-dione 2-[2-(3-ethylpyridin-4-yl)cyclopropyl]-N,N'-dimethylethanimidamide (3S)-N-benzyl-1-[3,5-bis(trifluoromethyl)phenyl]sulfonyl-N-methylpyrrolidine-3-carboxamide 1-(3-nitrophenyl)sulfonyl-2,5-dihydrotetrazol-1-ium;chloride 3-(5,6-dihydronaphthalen-1-yl)cyclohexan-1-amine 2-benzyl-1-[2,5-dimethyl-4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]butan-1-one 1-[(3,5-dimethylphenyl)methyl]-6-hydroxy-N'-(2-piperidin-4-ylethyl)-7-[(Z)-prop-1-enoxy]benzimidazole-2-carboximidamide 1-[4,6-difluoro-5-hydroxy-3-(1-methylcyclopropyl)pyridin-2-yl]piperidine-4-carboxylic acid (E)-2,4-dimethyl-1-phenyl-3-[propan-2-ylidene-[2-[1-(2-sulfoethoxy)ethenyl]pyridin-4-yl]methylidene]pent-4-en-2-olate;palladium(2+) 6-(3,4,4a,5,7,8,8a-octahydro-2H-pyrano[3,2-b]pyridine-1-carbonyl)pyridine-3-carboxamide (2-ethylsulfonylphenyl)methylidenehydrazine (1S,2R)-N-[(E)-3-hydroxyprop-1-enyl]-2-methoxy-N'-(4-phenylphenyl)cyclohexane-1-carbohydrazide 1,2-diamino-4-[3-(6-methylpyridin-2-yl)oxyphenyl]-6-oxopyridine-3,5-dicarbonitrile 7-azidonaphthalene-1,6,8-triol 1-ethyl-3,4-dimethoxy-2H-pyridine;1-(4-ethynylphenyl)-2-fluoro-4-propan-2-ylbenzene 4-fluoro-3-[6-(2,2,2-trifluoroethoxy)pyridin-3-yl]benzaldehyde 2-[3-(1,3-benzothiazol-4-yloxy)phenoxy]ethanol;propanoic acid 3-[(1-methylimidazol-2-yl)methylamino]benzoic acid (E)-3-[4-methoxy-2,6-dimethyl-1-[(4-nitrophenyl)methoxy]-7H-cyclohepta[d]imidazol-8-ylidene]prop-1-en-1-amine 3-[[5-(4-fluorophenyl)tetrazol-2-yl]methyl]-4-oxothieno[3,2-d]pyrimidine-7-carboxylic acid 3-ethenyl-2,4,9,10-tetrahydronaphtho[1,2-g][1]benzofuran-6,11-dione [3-(2,5-dimethylpyrrol-1-yl)phenyl]phosphane N-[(3R)-1-[6-chloro-7-(4-fluorophenyl)-2H-quinoline-1-carbonyl]pyrrolidin-3-yl]acetamide 3-cyclobutyloxy-4,5-difluoroaniline 4-[(4,5-diphenyl-1H-imidazol-2-yl)methoxy]benzamide 2-[3,5-bis(trifluoromethyl)phenyl]sulfanylacetic acid (5R)-6,9-diazaspiro[4.5]decane;3,8-dimethyl-11-oxo-7-thia-1,2-diazecine-2-carboxylic acid (4-azidophenyl)-(5-methylsulfonylpentyl)diazene (3S)-5,5,8,9,10,11-hexafluoro-2,6,7,11,12,13,14,15,16-decamethyltricyclo[8.4.0.03,8]tetradeca-1(10),3,6,12-tetraene N-[1-(2-aminoacetyl)pyrrolidin-3-yl]-4-cyclopropylbenzamide N-[(3R)-1-[(1-tert-butyltriazol-4-yl)methyl]pyrrolidin-3-yl]-2,6-difluoro-8-methoxyquinoline-5-carboxamide (4S,6R)-5-[[amino-(6-fluoro-2,3-dimethylindazol-5-yl)methylidene]amino]-1-cyclobutyl-6-methyl-4-propan-2-yloctan-4-ol 5-phenyl-1H-indazole;2,3,4,5-tetramethylcyclopenta-1,3-diene 2-(2,6-dichlorophenyl)-N-[2,4-bis(trifluoromethyl)-1H-pyrrol-3-yl]acetamide 4-azido-2-propan-2-yloxypyrimidine (2R)-4-amino-1,5-diphenylpentane-2,3-diol (1S,2R)-1-hydroxy-4-methylsulfanyl-N-phenylmethoxypentane-1-sulfinamide 1-butyl-4-[(E)-3,3-dimethylbut-1-enoxy]benzene;2,6-dichloro-4-phenylpyridine 4-[(4-bromophenyl)methyl]benzenesulfinate 2-azido-6,8-bis(trifluoromethyl)quinoline 2,6-dibromo-4-[1-[2,4-di(propan-2-yl)phenyl]tetrazol-5-yl]phenol 3-(2,4-difluorophenyl)-6-(trifluoromethyl)pyridine-2-carbonitrile 1-[6-(2,5-dimethylthiophene-3-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]azetidin-2-one (E)-3-[5-[(2,6-dichlorophenyl)methylsulfanyl]-4-(pyridin-3-ylmethoxy)thiophen-2-yl]prop-2-enoic acid [4-(2,3-dichlorophenyl)sulfanylpiperidin-1-yl]-(5-pyrrolidin-1-ylsulfonylthiophen-2-yl)methanone ethane;3-(4-fluorophenyl)-6-methyl-2,3-dihydroinden-1-one 1-[3,4-bis(trifluoromethyl)phenyl]-N-[2-bromo-4-chloro-6-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methanesulfonamide (6S,9R)-2-methyl-9-pyridin-4-yl-6-thiophen-3-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one (5-fluoro-2-hydroxyphenyl)-[4-methyl-3-(2-morpholin-4-ylethoxymethyl)pyrrolidin-1-yl]methanone 4-[2,6-dichloro-3-fluoro-5-(2H-1,4-triazol-5-yl)phenyl]butanoic acid N-[1-(oxan-2-yloxy)cyclopropanecarbonyl]benzamide 2-[(3,4-difluorophenyl)methyl]-8-hydroxy-5,7-dihydropyrido[2,3-d]pyrimidine-6-carboxylic acid 3-[2-(benzylamino)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]-2,6-dimethylbenzoic acid 5-[2-(4-aminocyclohexyl)ethynyl]-N-(4,5-dimethylcyclohepta-1,3,6-trien-1-yl)pyridine-2-carboxamide N-[5-(2,4-dichlorophenyl)sulfonyl-1H-indazol-3-yl]-4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-(oxetan-3-ylamino)benzamide 1-N',3-N'-bis[(E)-(4-hydroxy-6-methoxy-2-oxo-1H-indol-3-ylidene)amino]propanedihydrazide 6-amino-2-[2,4,6-tri(propan-2-yl)phenyl]isoindole-1,3-dione 2-amino-3-[4-(2,5-dimethylphenyl)sulfanyl-1H-pyrrol-2-yl]propanoic acid 2-[(E)-3,6,7-trimethyloct-5-enyl]thiophene (3S,4R)-1-[(4-fluorophenyl)methyl]-4-hydroxy-N-[(2S)-1-[[(2S)-1-[[6-(trifluoromethyl)pyridin-3-yl]amino]propan-2-yl]amino]propan-2-yl]pyrrolidine-3-carboxamide 1-[4-(8-amino-2-ethoxypurin-9-yl)phenyl]cyclopropane-1-carboxamide 2-chloro-5-(1,3-dimethylpyrazol-4-yl)pyridine;N-[1-(4-methoxyphenyl)ethyl]cyclopropanesulfonamide 7-cyclopropyl-2,3,6,9,11,15,18-hexazatetracyclo[8.8.0.03,8.012,17]octadeca-1(10),4,6,8,11,13,16-heptaen-14-one 5-N,7a-dihydropyrene-2,5-diamine 4-[1-(2,6-dimethylphenyl)imidazol-2-yl]phenol [2-cyclohexyl-1,3-dioxo-5-(4-phenylmethoxybutan-2-ylamino)isoindol-4-yl]-dimethyl-sulfidoazanium 1-methylsulfonyl-N-[1-(2,4,6-trichlorophenyl)ethylideneamino]azetidine-3-carboxamide [(2R,3S)-4-amino-1-cyclopropyl-3-methoxybutan-2-yl]benzene 2-[(3R)-4-azidobutyl]isoindole-1,3-dione 1-(4-aminopyridin-3-yl)indole-5-carbonitrile 2-[1-hydroxy-4,5-dimethoxy-3-(4-phenylsulfanylphenyl)naphthalen-2-yl]propanenitrile N-[(2,3-dimethylphenyl)carbamoyl]benzamide 4-N-(2-cyclopropylpyrimidin-4-yl)-1-[3,5-bis(trifluoromethyl)phenyl]-6-methoxyquinoline-4,7-diamine 4-(azidomethyl)-1,2-diethoxybenzene 4-(4-amino-3-ethylphenyl)-N,N-diethyl-2H-furan-5-imine 3-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]-7-piperidin-4-yl-4H-pyrazolo[1,5-a]pyrimidin-5-one;hydrochloride 4-(6,7-difluoroquinoxalin-2-yl)sulfanyl-3-methoxybenzoic acid (5R)-5-[4-(2,6-dichloro-3,5-dimethoxyphenyl)-7-oxopyrido[2,3-d]pyrimidin-6-yl]oxyhexanoic acid (1R)-N,N-dimethylspiro[1H-2-benzofuran-3,4'-piperidine]-1'-carboxamide (5E)-2-[(Z)-(3,4-dimethoxyphenyl)methylidenehydrazinylidene]-5-[[1-[(4-fluorophenyl)methyl]indol-3-yl]methylidene]-1,3-thiazolidin-4-one N-[(3R)-piperidin-3-yl]-2H-quinolin-1-amine 5-methoxy-2-[(Z)-[4-[[3-(trifluoromethyl)phenyl]methylsulfanyl]-1,3-thiazol-2-yl]iminomethyl]phenol 2-chloro-N-cyclobutylquinazoline-8-carboxamide N-(2,4-difluorophenyl)-5-oxopyrrolidine-3-carboxamide 2-[(4,4-difluorocyclohexyl)methoxy]-3H-pyrido[3,4-d]pyrimidin-4-one 4-methoxy-3-[(Z)-5-methyl-2-[methyl(naphthalen-1-ylsulfonyl)amino]hex-2-enoyl]benzenesulfonic acid (E)-3-[5-methoxy-2-[4-methyl-2-(trifluoromethylsulfonyl)phenoxy]phenyl]prop-2-enoic acid [2-azido-1-(4-fluorophenyl)ethyl]carbamic acid (Z)-2-[N'-(3,5-dimethoxyphenyl)carbamimidoyl]-3-(4-ethylsulfanylphenyl)prop-2-enoic acid N-[5-(7-fluoro-3,4,8,9-tetrahydro-1H-pyrido[3,4-b]indole-2-carbonyl)pyridin-3-yl]-3,4-dimethoxybenzamide 2,5-dichloro-4-(3-propan-2-yloxyanilino)sulfanylbenzoate 5-[1-(2,2-dimethylpropyl)pyrazol-3-yl]-3H-1,3,4-oxadiazol-2-one;6-piperidin-1-ylpyrimidine-4-carbonitrile [3-methoxy-4-(2,2,2-trifluoroethoxy)pyridin-2-yl]urea 4-[3-(2,6-dimethylmorpholine-4-carbonyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]benzonitrile 5-[(5,6-dimethylpyridin-3-yl)methoxy]-N'-hydroxypyrazine-2-carboximidamide 5-[(3Z)-3-ethenylhexa-1,3,5-trien-2-yl]oxypyrazine-2-carboxylic acid N-(2,3-dimethylphenyl)-4-[5-fluoro-6-(1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)pyridin-3-yl]benzamide 6,7-difluoro-3-propanoylquinoxaline-2-carboxylic acid 4-[1,3-dihydroisoindol-2-yl(methoxy)methyl]-N'-hydroxypyridine-2-carboximidamide N-[1-(2-ethenylcycloprop-2-en-1-ylidene)-3,3-dimethylbutan-2-ylidene]-4-fluorobenzamide (E)-3-[4-[(2R,6S)-6-[2-(4-fluorophenyl)ethynyl]oxan-2-yl]oxy-3-methoxyphenyl]-1-pyrrolidin-1-ylprop-2-en-1-one 5-[(E)-2-phenylethenyl]-1,3-benzodioxole 2-(4-chloroanilino)ethanol;5,7-diphenyl-1H-pyrrolo[3,2-c]pyridine 4-[(6-chloro-2,3-dihydroindole-1-carbonyl)amino]benzenesulfonic acid 1-[2-(cyclopropylmethoxy)ethylamino]-3-(thiophen-2-ylmethyl)urea 2-[(5E)-4,6-dihydrocycloocta[b]thiophen-9-yl]propanoic acid N-[5-chloro-2-(diethylamino)phenyl]-5-methylfuran-3-carboxamide;hydrochloride 1-[(4R)-6,9-dimethyl-8,10-dihydro-7H-cyclopenta[h]quinolin-4-yl]ethanone 3-[4-[(1R)-1-[[4-[2-[2-fluoro-5-methyl-6-(triazol-2-yl)pyridin-3-yl]ethynyl]pyrimidin-2-yl]amino]ethyl]phenyl]propanoic acid 3-[(E)-2-methylbut-1-enyl]sulfanyl-6-[5-propan-2-yloxy-1-[4-(trifluoromethyl)phenyl]pyrazole-4-carbonyl]-1H-pyrazin-2-one [4-amino-6-(butylamino)pyrimidin-5-yl]-methoxy-oxoazanium 2-methylsulfonylnaphthalene-1,4-dione 2-azido-4-[(1R)-3,3-difluorocyclohexyl]pyridine (E)-3-hydroxy-2-[4-nitro-5-[1-(oxan-2-yloxymethoxycarbonylamino)ethyl]pyridin-2-yl]prop-2-enoic acid 1-[3-(2,5-dihydroxypentylsulfanyl)phenyl]-3-phenylurea N-[1-(3,5-dichlorophenyl)ethenyl]pentan-2-imine 3-(6-amino-2,4-dichlorobenzo[b]carbazol-11-yl)benzoic acid [4-(4-aminophenyl)piperazin-1-yl]-[3,3-bis(4-fluorophenyl)azetidin-1-yl]methanone 4-ethyl-3-hydroxy-2,5-dioxodiazinane-1-carboxylic acid 5-chloro-6-methoxycarbonylpyridine-3-carboxylic acid (2R)-3-cyclopropyl-2-[6-methoxy-7-[(1-phenylethylideneamino)oxymethyl]-1,4-dihydroindeno[1,2-c]pyrazole-3-carbonyl]butanoic acid N-(2,4,6-trimethylphenyl)sulfonylpropanamide 4-bromo-2,3-dichlorobenzamide;ethane N'-[3,4-bis(ethenyl)phenyl]-N-[1-[2-(methylamino)phenyl]ethenyl]benzenecarboximidamide;methanamine N-butyl-2,6-dichloro-N'-(3,4,5-trimethoxyphenyl)-1H-indole-3-carboximidamide 2-(3,5-dimethylpyrazol-1-yl)-1-[4-(piperidine-1-carbonyl)-8-oxa-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,6-trien-11-yl]ethanone [1-[5-(2-cyanophenyl)pyridine-3-carbonyl]azetidin-3-yl]carbamic acid 2-azido-3-N,4-N-diphenylpyridine-1,3,4-triamine 3-[4-methoxycarbonyl-N-(2,3,4,5,6-pentafluorophenyl)sulfonylanilino]butanoic acid 5-methoxy-2-(3,4,6-triethylpyridin-2-yl)phenol 6-chloro-2-ethyl-4-(4,4,5,5-tetramethyloxaborolan-2-yl)pyridazin-3-one 4-[5-fluoro-2-(4-fluorophenyl)phenyl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 6-tert-butyl-1,8a-dihydropyrene 3-[5-(2-cyanopyridin-4-yl)-1,3-thiazol-2-yl]propanamide 3-(4-fluoro-1H-benzimidazol-2-yl)-N-[(2S,3S)-1-imidazol-1-yl-3-methylpentan-2-yl]propanamide 4-(7-fluoroimidazo[1,2-a]pyridine-3-carbonyl)-6-methylpiperazine-2-carbonitrile 3-chloro-N-(4,5-dimethylpyrimidin-2-yl)sulfanylpyrazin-2-amine N-(2-tert-butylpyrazol-3-yl)-4-[5-methyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]pyrimidin-2-amine 2-amino-4-[(1R,3S)-3-[1-cyclohexylbutyl-(5-methoxypyridine-2-carbonyl)amino]cyclopentyl]benzoic acid 1-aminoethylidene(pentan-3-yl)azanium;2,4,5,6,7,8-hexachloronaphthalene-1,6,8-trisulfonate 1-[4-(1,2,3a,4,6,7,8,8a-octahydrocyclopenta[d]pyrimidin-5-ylmethoxy)phenyl]-N'-(2-aminoethyl)cyclopropane-1-carboximidamide;dihydrochloride 2-[[4-(3,5-dichloropyridine-4-carbonyl)piperazin-1-yl]methyl]-8-fluorochromen-4-one 2-[(1R)-1-[(4-chlorophenyl)methylamino]propyl]phenol 2-ethoxy-1-[(6R)-3-methyl-4,5,6,7-tetrahydropyrazolo[3,4-b]pyridin-1-yl]propan-1-one 2-[1-(4-fluorophenyl)sulfonylpiperidin-4-yl]oxy-N,N-dimethylethanamine 2-[(5Z)-5-[[3,4-dimethoxy-6-[3-(trifluoromethylsulfanyl)phenoxy]pyridin-2-yl]methylidene]-2-oxo-1,3-thiazolidin-3-yl]acetic acid 2-[1-(3,5-dichlorophenyl)ethenyl]pyrrolidine;2-methoxyquinoline 4-[8-(2,6-dioxopiperidin-3-yl)-5H-indeno[1,2-b]pyridin-3-yl]-N'-hydrazinylidenecyclohexane-1-carboximidamide 3-[4-(1H-benzimidazole-2-carbonyl)piperazin-1-yl]pyrrolidin-2-one N-[(2S)-5-amino-1-oxo-5-phenylpentan-2-yl]-4-cyclobutylidenebut-2-ynamide N-(5-methoxy-1,3,4-thiadiazol-2-yl)-6-oxopiperidine-2-carboxamide 6-(3,4-dihydro-2H-1,5-benzodioxepine-7-carbonyl)-10-ethyl-2-oxa-6,10-diazaspiro[4.6]undecan-7-one 5-[2-(2,4-difluorophenoxy)phenyl]imidazolidine-2,4-dione 1-cyclopropylsulfonyl-4-fluorobenzene 1-azidooxy-4-nitronaphthalene N-[2,3-bis(ethenyl)phenyl]-5-methoxy-1-(4-morpholin-4-ylphenyl)benzimidazol-4-amine 2-[[3-(4,5-difluorocyclohexa-1,3-dien-1-yl)oxypyrrolidin-1-yl]methyl]benzonitrile 4-[5-[[(2,6-dichlorobenzoyl)amino]methyl]-1H-imidazo[4,5-b]pyridin-2-yl]benzenesulfinate N-azido-1,2,3,4-tetrachlorocyclopenta-2,4-diene-1-carboxamide 2-(3,6-dimethyl-4H-azepin-7-ylidene)cyclohexa-1,5-diene-1-carboxamide N-[(4R,5S)-1-[6-methoxy-5-(4-methylimidazol-1-yl)pyridine-2-carbonyl]-3-methyl-2-oxo-5,7-dihydropyrrolo[3,4-b]pyridin-4-yl]cyclopropanecarboxamide 5-[4-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)phenyl]-N'-pyrrolidin-3-ylpentanimidamide (3R)-7-[[2,6-bis(4-methoxyphenyl)pyridine-4-carbonyl]amino]-6-oxo-N-[(1S)-1-phenylpropyl]-1,3,4,5-tetrahydropyrrolo[3,4-c][1,6]naphthyridine-8-carboxamide N-benzyl-2-[(4E)-4-[[3,5-bis(difluoromethoxy)phenyl]methylidene]-3,3-dimethylpiperidin-1-yl]acetamide 5-phenyl-6H-phenanthridine [[2-amino-5-(1,3-benzodioxol-4-yl)phenyl]-(1H-indol-5-ylamino)methylidene]azanium 1-[(5S,7R)-2-benzylsulfanyl-5-phenyl-7-thiophen-2-yl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]ethanone 2-methyl-3H-benzo[g]chromene-4,9-dione (4S)-1-[2,6-difluoro-4-(5-methyl-1H-pyrazol-3-yl)benzoyl]-N-ethyl-N'-[(Z)-(2-fluorophenyl)methylideneamino]-4-hydroxypyrrolidine-2-carboximidamide N-azido-6,7-dichloronaphthalene-2-sulfinamide 2-azidooxy-1,3,5-tri(propan-2-yl)benzene 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-[2-[4-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]pyridin-2-yl]phenyl]propan-2-one N-methyl-3,6-dihydro-2H-pyridine-1-carboxamide;4-[(3-methylphenoxy)-phosphanylidenemethyl]benzonitrile 1,2,3-trimethylquinoxaline-6-carboxylic acid 2-azidooxy-N-(3-methylbutanoyl)benzamide 4-[2-(3,5-dimethyltriazol-4-yl)piperidin-1-yl]-6-ethoxypyrimidine 2-[3-fluoro-4-(oxolane-3-carbonyl)piperazin-1-yl]quinoline-5,8-dione 2-[2-(4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carbonyl)-2H-indol-3-yl]acetonitrile 1-azido-4-cyclohexyloxybenzene 3-butanoyl-5-pyridin-2-ylhex-4-enoic acid 3-(3,4-dihydroquinolin-8-yl)-2-methoxypropanamide 5-methyl-2,3,6-triphenylaniline N-(3,5-dimethylphenyl)-2-(3-methyl-6-oxo-2H-purin-7-yl)acetamide [4-[2,4-dimethyl-5-(2,3,4,5,6-pentafluorophenyl)sulfanylhexyl]-2,5-dimethoxyphenyl]-ethoxyphosphinic acid 2-amino-9-[(4S)-1,1,1,3,3,6,6-hexadeuterio-4-hydroxyhexan-3-yl]-8-[[2-fluoro-5-methoxy-4-(morpholine-4-carbonyl)phenyl]methyl]purin-6-olate N-(cyclopropylmethyl)-3-hydroxy-4-[(6Z,8E,10E)-10-[(4-iodophenyl)methylidene]-3-methoxy-2,3,5,9,11-pentazatricyclo[7.4.0.02,6]trideca-1(13),5,8,10-tetraen-12-yl]butanamide 5-(2-methylpyrazol-3-yl)sulfanyl-1H-pyrrolo[2,3-b]pyridine (E)-1-[4-hydroxy-3,5-di(propanoyloxy)phenyl]pent-2-en-1-one 4-(ethylamino)-3,6-diiodobenzene-1,2-diol 4-(5,6-dichloro-1H-benzimidazol-2-yl)-N-[3-[2-[4-(hydroxymethyl)anilino]ethoxy]phenyl]butanamide N-[3,4-bis(1,2,3,4,5,6-hexahydronaphthalen-2-ylmethoxy)phenyl]acetamide;ethane [1-amino-4-(4-ethenylpiperazin-1-yl)pentan-3-ylidene]azanium;1,2,5-trifluorobenzene N-[1-(4-chlorophenyl)sulfonylpyrrolidin-3-yl]-3,5-dimethoxy-2-morpholin-4-ylbenzamide 5-butylsulfanyl-6H-[1,2]oxazolo[4,5-d]pyrimidine 4-[(1S)-1-azidoethyl]-2,6-dibromophenol 3-chloro-N-[2,4-difluoro-3-(2-methyl-5,6-dihydropyrrolo[1,2-b]pyrazole-3-carbonyl)phenyl]-1-oxidopyridin-1-ium-2-carboxamide (2S)-3-[6-[4-[1,5-bis(trifluoromethyl)pyrazol-3-yl]phenyl]imidazo[1,2-b]pyridazin-2-yl]oxypropan-1-ol N-[2-[(6-amino-1,3-benzothiazol-2-yl)disulfanyl]ethyl]decanamide 3-methyl-5-(2-methylidenepyrrolidine-1-carbonyl)benzenethiol 5-chloro-4-N-[(2,3-dimethylindazol-6-yl)methyl]pyrimidine-2,4-diamine 6-(1,3-benzodioxol-5-yloxy)-2-(4-phenylpiperazine-1-carbonyl)-[1]benzofuro[3,2-b]pyridine-3-carboxamide 3-[(1E,3Z)-4,5-dimethylhexa-1,3,5-trienyl]-1-(2-hydroxyethyl)imidazo[4,5-b]pyridin-2-one;ethane 2,3-dihydro-1H-indene;ethane;(2E)-N-[5-methyl-4-(7-methyl-3,4-dihydro-1H-isoquinolin-2-yl)pyridin-3-yl]penta-2,4-dienamide 2-[(1S)-1-cyclopentylethyl]imino-5,6,7,8-tetrahydro-3H-pyrido[4,3-d]pyrimidin-4-one 2-(4-methyl-6-oxo-1H-pyrimidin-5-yl)-N-[(1S,3R)-3-morpholin-4-ylcyclopentyl]acetamide [3-(4-fluorophenyl)-1,2-oxazol-5-yl]-[4-(1H-imidazol-5-ylmethyl)piperazin-1-yl]methanone 1-[4-(ethylaminomethyl)cyclohexyl]-3-[4-(4-oxo-5H-pyrazolo[4,3-c]pyridin-1-yl)phenyl]urea [3-[5-(2,6-diphenylpyridine-4-carboximidoyl)-1H-pyrrol-3-yl]phenyl]-(4-methoxyphenyl)sulfonylazanium 4-(1H-indazole-5-carbonyl)-3,5-dimethyl-6-[3-(trifluoromethyl)phenyl]piperazin-2-one (3R)-4,5,6,7-tetrahydroxy-3-(phenyliminomethyl)chromen-2-one N-(4-chloro-3,5-dimethylphenyl)-2-methoxyiminoacetamide 5-[(2,4-dichloropyrimidin-5-yl)-ethylamino]-3H-1,3,4-thiadiazole-2-thione 3,8-bis[(dimethylamino)methyl]naphthalene-1,2-dione 2-(3,5-dimethylphenyl)-1-[5-(4-fluorophenyl)-2H-pyrrol-4-yl]ethanone 2-(6-aminopurin-9-yl)butanamide;but-1-ene (2S)-5-[(4-methoxyphenyl)methyl]piperidine-2-carboxylic acid 1-benzyl-5-[6-bromo-7-(2,5-dihydropyrrole-1-carbonyl)imidazo[4,5-b]pyridin-3-yl]pyridin-2-one N-[2-chloro-6-(trifluoromethyl)pyridin-4-yl]-5,7-difluoro-1H-indole-3-sulfonamide 2-[4-(diethylamino)phenyl]-2-[1,3-oxazol-5-ylmethyl(propan-2-yl)amino]acetamide 2-[4-(3-propan-2-yloxyanilino)-1,5-dihydropyrrolo[2,3-b]pyridin-3-yl]acetic acid 4-[(1R)-2,3-dihydro-1H-inden-1-yl]-N-(6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepin-3-ylmethyl)aniline (E)-3-methyl-1,1,1-triphenylpent-4-en-2-one 6-[(2R)-2-(4-tert-butylphenyl)pyrrolidin-1-yl]pyridine-3-carbonitrile [3-(9H-fluoren-1-yl)pyrrolidin-2-ylidene]cyanamide 2-azido-6-(3,5-dimethylpyrazol-1-yl)pyridine N'-[2-(2,4,5-trimethylphenyl)ethylideneamino]ethanimidamide 2-chloro-4-(6,8-dioxo-7H-imidazo[1,5-a]pyrazin-5-yl)benzonitrile 3-(6,8-dichloro-2H-chromene-5-carbonyl)sulfanylpropanoic acid 2-(5,7-difluoronaphthalen-1-yl)-N-[(E)-3-methoxyprop-1-enyl]acetamide 3-chlorosulfonyloxyphthalic acid 1-butan-2-yl-4-[(4-pentoxyphenyl)disulfanyl]benzene;ethane 2-amino-4-[[(1R)-cyclohexa-2,4-dien-1-yl]methoxy]naphthalene-1,3-disulfonic acid 2-amino-4-[3,5-dichloro-4-(1H-indole-2-carbonyl)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile 3,5-ditert-butyl-N'-hydroxybenzenecarboximidamide 3-(5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-1-carbonyl)-N,N-diethylbenzamide 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]octanoic acid 5-amino-N,N'-dimethyl-6-(2-oxopyrrolidin-1-yl)pyridine-3-carboximidamide N-(5-tert-butyl-2-hydroxyphenyl)sulfonyl-6-chloropyridine-3-carboxamide 1-(2,4-dimethoxyphenyl)-3-[2-(2-methylimidazol-1-yl)pyridin-3-yl]urea N-cyclohexa-1,5-dien-1-ylsulfanyl-2-methoxyaniline 2-(3-bromopropoxy)-4-ethylpyridine 2-(2,6-dioxopiperidin-3-yl)-5-[4-(morpholine-4-carbonyl)phenyl]isoindole-1,3-dione 1-(4-chlorophenyl)-N-[[(2R,3S)-6-oxopiperidin-3-yl]methyl]triazole-4-carboxamide (2R)-2-[4-[(1-ethylcyclohexyl)amino]butanoylamino]-3-phenylpropanoic acid 6-[[4,5-bis(ethenyl)-2-methylphenyl]diazenyl]-3,9a-dihydropyrene-1-carboxylic acid 2-[(Z)-3-amino-1-hydroxy-4,4-dimethylpent-2-enylidene]sulfanyl-6-(6-chloro-1H-benzimidazol-2-yl)pyridine-3-carbonitrile N-(1,3-benzodioxol-5-ylmethyl)-N'-[(Z)-(2-chlorophenyl)methylideneamino]oxamide 2-[4-(methylaminomethyl)phenyl]sulfanylbenzamide 3-chloro-N-[(2R,4S)-6-fluoro-1-[3-(6-methoxyquinolin-4-yl)propyl]-4-methylpiperidin-2-yl]benzamide N-cyclopropylformamide;ethane;1,3,5-trimethyl-2-[(E)-prop-1-enyl]benzene N-[4-(1,5-dimethylpyrazol-3-yl)phenyl]propanamide N-[5-(1H-indole-3-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]-1,2-thiazole-5-carboxamide 2-(2,6-dibromophenoxy)acetaldehyde (3S)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide 4-[[(E)-3-(2,3,5-trimethoxyphenyl)prop-2-enoyl]amino]benzoic acid 7,8-dichloro-5-ethyl-2,4-dimethyl-1H-[1]benzofuro[3,2-c]quinoline N-[[6-(difluoromethyl)pyridine-3-carbonyl]amino]formamide 6-[(2Z,4E)-5-methylhepta-2,4-dien-3-yl]sulfanylpyrimidine-4-carbonitrile 2-[(3R,4S)-1-azidopyrrolidin-3-yl]oxy-5-propan-2-ylpyrazine 2-[(Z)-1,3,4-oxadiazol-2-yliminomethyl]benzoate 5-[2-chloro-4-(diethylamino)phenyl]-5-(6,8-dihydro-5H-1,7-naphthyridine-3-carbonylamino)pentanoic acid 1-(9,10-dioxoanthracen-2-yl)piperidine-4-carboxylic acid N-[(E)-3,4-dioxopent-1-enyl]benzamide [1-(5-bromopyrimidin-2-yl)piperidin-4-yl]-trimethoxyboranuide 7-(4-bromophenyl)-2,3-dichloroquinoline 2-(6,11-dihydropyrrolo[2,1-c][1,4]benzothiazepine-8-carbonyl)-N',4-dimethylbenzenecarboximidamide 2-[[6-(4-chlorophenyl)pyridin-3-yl]methylideneamino]oxy-N-ethyl-N-(5,6,7,8-tetrahydroquinolin-8-ylmethyl)acetamide 5-amino-2,6-dimethyl-4-[(4-propan-2-yl-1H-indazol-6-yl)oxy]pyridine-3-carbonitrile 1-[2-fluoro-4-(trifluoromethyl)phenyl]ethanone;3,4,5-trifluoro-N-(3,4,5,6,7,8-hexahydronaphthalen-2-yl)benzamide (4Z)-2-cyclopentyl-4-[[4-methoxy-3-(morpholine-4-carbonyl)phenyl]methylidene]-1,3-oxazol-5-one 1-phenyl-2,3-dihydroindole-4,7-disulfonic acid 2-(3,4-difluorophenyl)-1H-pyrrolo[3,2-b]pyridine 6-[2-(2,3-dihydrothiophen-4-yl)phenyl]pyridine-2-carboxylic acid (2R)-2-[2-(4-fluorophenyl)-1H-inden-1-yl]propanamide N-methyl-4-[(2-thiophen-3-yl-5,6,7,8-tetrahydroquinazolin-4-yl)oxy]aniline 1-[2-(4,6-dimethylpyrazolo[1,5-a]pyridine-3-carbonyl)spiro[3.3]heptan-6-yl]propan-1-one 1-[2-azidooxy-3,5-diethyl-6-(methoxymethyl)phenyl]-N,N',N'-trimethylpropane-1,3-diamine 4-[(2-chloroquinolin-3-yl)methylidene]-2-cyclohexyloxycyclohexa-1,5-dien-1-ol 6-bromo-3,3-difluoro-1,2-dihydroindene 1-bromo-3-chloro-2-[2,4-di(propan-2-yl)phenoxy]benzene;ethane 5-(6-fluoroquinolin-4-yl)oxy-N',1-dimethylpyrazole-3-carbohydrazide N-[3,5-bis(trifluoromethyl)phenyl]-1-[3-(4-chlorophenoxy)propanoyl]piperidine-4-carboxamide N'-tert-butyl-4-[5-(3,7-dimethoxynaphthalen-2-yl)-1H-imidazol-2-yl]benzenecarboximidamide;dihydrochloride 4-[(3S)-1-(4,6-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one (6S)-5,6-dimethyl-3-[1-[4-(trifluoromethoxy)phenyl]ethylsulfanylmethyl]cyclohexa-2,4-dien-1-one 6-[(3-chlorophenyl)methoxy]-N,4-dipropylquinoline-2-carboxamide 1,4-bis(bromomethyl)-2,5-difluorobenzene N-[4-(4-phenylphenyl)cyclohexa-2,4-dien-1-yl]propanamide (2S)-3,4-bis(phenylmethoxycarbonylamino)pyrrolidine-2-carboxylic acid (E)-N-[(Z)-3,6-dimethylhept-2-en-4-ylidene]-3-(5-ethenylpyridin-3-yl)-4-iminopent-2-enamide N-[(Z)-1H-indol-3-ylmethylideneamino]-3-methoxyquinolin-2-amine 2-[3,5-bis(trifluoromethyl)phenyl]-N,6,6-trichloro-1H-pyrimidine-2-carboxamide N'-amino-6-[4-(1H-imidazol-5-yl)piperidin-1-yl]pyridine-2,3-dicarboximidamide 1,3-bis(2-hydroxyphenyl)-5-(4-nitrosophenyl)pyrazol-4-ol (2S)-3-methyl-1,1-dioxo-N-[[4-(trifluoromethylsulfanyl)phenyl]methoxy]-1,2-benzothiazole-6-carboxamide 1-N',1-N'-dimethylethane-1,2-diamine;(E)-3-[4-(8H-carbazol-4-yloxymethyl)triazol-1-yl]prop-2-enal N-(2,3-dihydro-1H-inden-5-ylmethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 4-(1,3-benzodioxol-5-ylmethylamino)-2-propan-2-yl-1H-pyrimidin-6-one 1-[4-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethoxy)phenyl]azetidine-3-carboxylic acid 6-[(4-benzylbenzoyl)amino]-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide;2,2,2-trifluoroacetic acid 5-(azidomethyl)-2-(3,4-dichlorophenoxy)-1H-imidazole (3S)-1-ethyl-5'-methoxy-8',9-dimethylspiro[3H-pyrido[2,1-b]quinazoline-11,3'-benzo[g]quinoline]-2'-one N-ethyl-2-(4-methoxyphenoxy)butanamide 2-(4-bromophenyl)-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one 4-amino-1-[(3S,5R)-4-benzyl-3,5-dimethylpiperazin-1-yl]-2-(4-hydroxyphenyl)-7-methylsulfanyloxypyrido[2,3-d]pyrimidin-6-one 2-[N'-(4-chlorophenyl)carbamimidoyl]sulfanyl-1,3,6,7,8,9-hexahydropyrrolo[1,2-a]azepine-5-carboxamide 2-[1-(6,7,8,9-tetrahydro-5H-carbazole-3-carbonyl)piperidin-4-yl]oxybutanoic acid 2,2-dimethylpropane;5-[1-(3-fluorophenyl)ethoxy]pyridine-3-carboxamide 2-(4-amino-3,5-dimethylphenyl)-1-[(3R,4S)-3-hydroxy-4-pyridin-2-ylpyrrolidin-1-yl]ethanone N-[(Z)-1-aminoethylidenecarbamothioyl]-4-(2-cyclopentyloxyphenyl)pyridine-3-carboxamide 1-[2-[5-(4-chlorophenyl)-1H-imidazol-2-yl]piperidin-1-yl]-3,3-dimethylbutan-1-one 2-[4-[5-fluoro-6-[(3S)-1-[3-methyl-2,5-dioxo-1-(pyridin-4-ylmethyl)imidazo[4,5-c]quinolin-8-yl]pyrrolidin-3-yl]oxy-2H-pyrimidin-1-yl]piperazin-1-yl]acetamide N-[4-(2,3-dihydro-1H-benzotriazol-4-yl)phenyl]sulfanyl-N',N'-dimethylpropane-1,3-diamine 2-[4-(3,5-dimethyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]-N-methylacetamide 4-(4,5-dihydro-1H-imidazol-2-yl)-6-iodobenzo[f]isoquinoline 4-[[4-methyl-3-(2-pyridin-3-ylethynyl)phenyl]methoxy]oxane-4-carboxamide N-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]-4-tert-butylbenzamide N-[(Z)-4,5-dimethylhex-2-enoxy]sulfanyl-4-(4-ethylphenyl)aniline 1-azido-4-[4-(2,6-dimethoxyphenyl)-5-(4-fluoropyridin-3-yl)-1,2,4-triazol-3-yl]piperidine 3-[2-[(3Z)-7,8-difluoro-6-methoxy-4-methyl-1H-5-1,5-benzodiazocin-2-ylidene]hydrazinyl]-N-(trihydroxymethylsulfanyl)benzamide 2-[4-(trifluoromethyl)phenoxy]thiophene 2,7-diazaspiro[4.5]decan-7-yl-(2-propan-2-yl-1H-imidazol-5-yl)methanone 3-[4-(5-methylfuran-2-carbonyl)piperazine-1-carbonyl]cyclohexa-1,3-diene-1-carbonitrile 1-cyclobutylsulfonyl-3,4-dihydro-2H-quinoline 4-(3,5-dimethylanilino)-N-[(E)-1H-indol-7-ylmethylideneamino]benzamide N-[4-(1,3-dihydroisoindole-2-carbonyl)cyclohexyl]pyrazine-2-carboxamide 2-[3,4,5-tris(trifluoromethyl)phenyl]cyclohexan-1-one 1-(4-chlorophenyl)sulfonyl-3-[4-[(E,3Z)-5-methoxy-3-propylidenehex-1-enyl]phenyl]urea 5-methyl-8H-pyrido[2,3-d]pyrimidine-6-carboxamide 5-[2,3-bis(ethenyl)phenoxy]pyridine-2-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-piperidin-4-ylpropanamide (2S)-N,N'-dibenzyl-3-[4-methylsulfonylbutanoyl(pentyl)amino]-2-propanoylbutanediamide (4Z)-4-[(6-methylpyridin-3-yl)methylidene]-2,5-diphenylpyrazol-3-one 2-[3-(dimethylamino)propoxy]-5-[6-methyl-7-oxo-1-[[4-(trifluoromethoxy)phenyl]methyl]pyrazolo[3,4-d]pyridazin-3-yl]benzamide 4-(3,7-dimethylocta-2,6-dienoxy)-1-methoxy-10-(3,5,8,11-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,10-pentaen-3-yl)decan-1-ol N-[(3,5-dimethoxyphenyl)methyl]-2-oxo-1H-pyrazine-4-carboxamide N-[2-[4-[(1,3-dihydroxy-2H-isoindol-5-yl)oxy]piperidin-1-yl]ethyl]-2-methylpropanamide 4-(1,3-benzodioxol-5-yl)-3H-1,2,4-oxadiazole;ethane 2-[3-(2,5-dioxopyrrolidin-1-yl)propoxy]-6-[4-(oxan-4-yl)pyrazole-1-carbonyl]pyridine-3-carbonitrile (3S)-1,2,3-trimethoxy-4-phenylbutan-2-amine N-butyl-N-hexyl-6-nitro-1,3-benzothiazol-2-amine N-(2,5-dioxopyrrolidin-3-yl)-5-(4-methoxyphenyl)sulfonylspiro[1H-indole-3,3'-azetidine]-2-carboxamide 6-amino-4-(2,3-dibromo-5-ethoxy-4-prop-2-enoxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 3-(dibutylamino)benzenesulfonamide 6-[2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-5-yl]-8-methoxy-3,4-dihydro-2H-quinoline-1-carboxylic acid 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-pyridin-3-ylbenzamide 2-[1-(2,6-dimethylphenyl)-4-hydroxy-5-(oxetan-3-yl)pyrazol-3-yl]isoindole-1,3-dione 2-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(3-methylbutyl)amino]benzoic acid [4-(2,6-difluorophenoxy)phenyl]sulfonylazanide N-[2-(1,3-benzodioxol-5-yl)ethyl]-1-phenylpropan-2-amine 1-[(E)-2-[6,7-bis(ethenyl)-9H-pyrido[3,4-b]indol-8-yl]ethenyl]-N'-[4-chloro-6-(2-methoxyphenyl)-1,3,5-triazin-2-yl]cyclopropane-1-carbohydrazide 5-[[(3S,4R)-3-benzylpiperidin-4-yl]amino]quinoline-8-carbonitrile 2-cyclopropyl-6-[(1-ethylimidazol-4-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 6,7-dimethyl-3,4,5,8-tetrahydropyrano[2,3-c]isoquinoline 6-azido-2-ethylsulfanylquinazoline 4-[3-[[4-(4-fluorophenyl)piperazin-1-yl]methyl]phenoxy]pyridine-2-carboxylic acid 6-[(2,4-dihydroxyphenyl)methyl]-2-thiophen-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one [3-(diethylamino)azetidin-1-yl]-[4-fluoro-6-[[(1S,2R)-2-fluorocyclopropanecarbonyl]amino]pyridine-3-carboximidoyl]borinic acid (2R,3S)-3-benzyl-4-oxo-N-(5-phenylpentyl)azetidine-2-carboxamide N-[1-(4-fluorophenyl)piperidin-3-yl]-2-phenylimidazole-1-carboxamide (7R)-6-N,5-dimethyl-7-[4-(2-methylpropoxy)phenyl]-3-N-(3-nitrophenyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide 3,6-bis(2,5-dimethylphenyl)-4-methylidenehexanamide [4-(2,6-difluorophenoxy)phenyl]methanol N-[4,4-difluoro-3-hydroxy-1-(hydroxyamino)-3-methylbutan-2-yl]-7-(methanesulfonamido)imidazo[1,5-a]pyridine-1-carboxamide 2-(3,6-difluorocarbazol-9-yl)acetamide 3-(5,6,7,8-tetrahydronaphthalen-1-yloxy)oxolane (E)-4,8-dihydroxy-3-methoxy-5,6-dihydronaphtho[2,1-f]isoquinoline-9,10-dione;5-(3-dodecan-4-ylthiophen-2-yl)-2H-tetrazole (E)-1-(2,6-diethoxy-4-methylphenyl)-3-[5-(disulfanylamino)naphthalen-1-yl]prop-2-en-1-one 4-(2,3-dihydroxypropoxy)-1H-indole-2-carboxylic acid N-[2,4-difluoro-3-(2-oxospiro[1H-indole-3,4'-oxane]-6-yl)oxyphenyl]propane-1-sulfonamide 4-[(2,2-dimethylcyclopentylamino)methyl]phenol 1-[2,4-dichloro-6-(trifluoromethyl)phenyl]propan-1-one 2-bromo-4,8-bis[(4-methoxyphenyl)methyl]pteridine 6-tert-butyl-2,3-dihydrofuro[2,3-b]chromene 2-methyl-N-[3-methyl-4-(5H-[1,2]oxazolo[4,5-b]pyridine-7-carbonyl)phenyl]benzamide 1-benzyl-3,4-bis(phenylmethoxy)quinolin-2-one N-[6,7-dihydro-4H-thieno[3,2-c]pyran-2-yl(propan-2-yl)amino]acetamide 6-[(2R)-3,3-difluorobutan-2-yl]oxynaphthalene-1-carbonitrile;propane ethane;(2S)-2-[5-(4-nitrophenyl)pentyl]piperidine (3R,4S)-2-[4-fluoro-2-(trifluoromethyl)phenyl]sulfanyl-6-(hydroxymethyl)oxane-3,4-diol 5-(azidomethyl)-3-(4-chlorophenyl)-1,2,4-oxadiazole 2-[[1-(3,4-dichlorophenyl)triazol-4-yl]methoxy]-N'-[6-ethylsulfonyl-5-(2,2,2-trifluoroethylsulfanyl)pyridin-2-yl]-2-methylpropanehydrazide 4-[4-methoxy-3-(2,2,2-trifluoroethylsulfanyl)phenyl]butanoic acid 2-chloro-4,6-dinitroaniline 2-hydroxy-3-[3-(methylamino)propanoylamino]-N-phenylnaphthalene-1-carboxamide 4-(3,6-difluorocarbazol-9-yl)butanenitrile (2E)-N-[[1-[1-(4,6-dimethylpyrimidin-5-yl)cyclobutyl]triazol-4-yl]methoxy]-4-oxopenta-2,5-dienamide 2-(4-bromophenyl)imino-5,6-dimethoxycyclohexan-1-one N-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-1,3-dimethylpyrazolo[3,4-b]pyridine-5-carboxamide N-(1,5-dimethyl-3-oxo-2-phenylpyrazolidin-4-ylidene)benzamide 2-[(5R,10bR)-9-chloro-5-thiophen-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 4-[3-cyclopropyloxy-6-(2,5-dimethyl-1H-imidazol-4-yl)-7,8-dihydro-5H-pyrido[3,4-b]pyrazin-2-yl]piperazine-1-carboxylic acid (1E)-1-[3-amino-4-[[2,5-dimethyl-3-(trifluoromethyl)phenyl]methoxy]cyclohexa-2,4-dien-1-ylidene]butan-2-one 1-(5-benzylthiophene-2-carbonyl)-3-piperidin-4-ylpyrrolidine-3-carboxamide 2-N-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-5-nitropyridine-2,4-diamine N-(1,3-thiazol-2-yl)thieno[2,3-c]pyridine-7-carboxamide (3,5-dichlorophenyl)sulfonylformaldehyde 4-ethenyl-3-methylidene-5,6-diphenyl-1H-pyrazin-2-one 1-methyl-3,6-diphenylpyrazin-2-one 5-cyclopropyl-N-(2,6-dimethoxypyridin-4-yl)pyridazine-3-carboxamide 2-[(2,3,4,5,6-pentachlorophenyl)methyl]propanedinitrile 2-[(3S)-6,9-difluoro-5-hydroxyiminotriazolo[4,5-c][1]benzimidazol-7-yl]sulfanyl-N-phenylpropanamide 4-[(1E,3Z)-3-amino-1-phenylhexa-1,3-dienyl]piperidine-4-carboxamide 4-(2,6-dimethylmorpholin-4-yl)-N'-hydroxypyridine-2-carboximidamide 1-[4-(3,5-difluorophenoxy)cyclohexyl]-N,2,2-trimethylpropan-1-amine 1-(2,6-dichlorophenyl)-3-[4-methyl-5-(methylideneamino)pyridin-2-yl]urea 3,4-difluoro-N'-[1-(methylamino)ethenyl]benzenecarboximidamide;4-[2-[2-[[2-(6-ethynylpyridin-3-yl)-5-ethoxypyrazol-3-yl]amino]pyrimidin-5-yl]ethynyl]benzaldehyde N-(2,5-difluorophenyl)-1-ethyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidine-5-carboxamide 1-N',2-N'-dimethyl-3-(propan-2-ylideneamino)benzene-1,2-dicarboximidamide (1R,2S)-N-[8-amino-6-(4-methylpyridin-3-yl)isoquinolin-3-yl]-2-cyclopropylcyclopropane-1-carboxamide 6-amino-4-[4-methoxy-3,5-bis(trifluoromethyl)phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 3-(6-bromoquinolin-2-yl)oxycyclobutane-1,1,2-triol 2-[(4,5-dichloro-1H-imidazole-2-carbonyl)amino]acetic acid 4-ethyl-3,5,6-trifluorobenzene-1,2-disulfonic acid N-(3,4-dihydroxyphenyl)-2-[1,2-dimethyl-5-oxo-6-[3-(trifluoromethoxy)phenoxy]imidazo[1,2-a]pyrimidin-7-yl]acetamide 4-[3-[4-(5-fluoropyridin-2-yl)piperazine-1-carbonyl]phenoxy]benzaldehyde N-azido-3-[[4-(2-chlorophenoxy)-5,6,7,8-tetrahydroquinazolin-2-yl]amino]benzenesulfonamide 3-(2,4-dichlorophenoxy)propane-1-sulfinic acid 3-(8,9-dihydro-5H-pyrimido[4,5-c]azepine-7-carbonyl)-2,6-dimethylbenzenesulfonamide;ethane N-(3-aminopropyl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamide;hydrochloride (E)-3-[4-amino-3-[4-hydroxy-2,6-dimethyl-3-(trifluoromethyl)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]prop-2-enal 5-[2,4-bis(phenylmethoxy)phenyl]-3-(4-chlorophenyl)-N-cyclopropyl-1H-pyrrole-2-carboxamide 1-[2,3-bis(ethenyl)indol-4-ylidene]piperidine 1-[(3-tert-butyl-2,6-dimethoxyphenyl)methyl]-5,6-dimethylpyrimidine-2,4-dione 2-(3,4-difluorophenyl)-5-oxo-1H-pyrazole-3-carboxylic acid 2-amino-4-(1,3-benzodioxol-5-yl)-6-[[3-(hydroxymethyl)phenyl]methoxy]pyridine-3-carbonitrile (2R)-5,6-dihydroxy-2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]-3,3a,4,9b-tetrahydro-1H-benzo[e]indole-7-sulfonic acid 1-[2-[4-(3-chlorophenyl)cyclohexyl]ethylamino]ethenol 4-N-(3,5-dimethylphenyl)-2-N-[4-(1H-pyrrol-2-ylmethylideneamino)phenyl]pyrimidine-2,4-diamine (3S,4R)-1-(9H-carbazole-2-carbonyl)-3-fluoropiperidine-4-carboxylic acid 1-[(E)-2-(4-butoxyphenyl)ethenyl]-3,5-bis(trifluoromethyl)benzene 2,4-bis(2-aminoethyl)-6-benzylaniline 3-[1-[4-amino-3-[5,7-difluoro-2-(methyliminomethyl)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-5-chloro-8-methoxy-2H-isoquinolin-1-one ethane;2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-4-pyridin-3-yl-1H-pyrimidin-6-one (2-chloro-5,6-difluoro-3H-1,4-benzothiazin-2-yl)-phenylmethanone N-cyclohexyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide [5-(2,6-difluorophenyl)sulfanyl-6-methoxypyridine-3-carbonyl]azanium (2S)-3,4-dihydroxy-2-(phenylmethoxycarbonylamino)butanoic acid 4-(3,5-dimethylphenyl)sulfonylbutanenitrile 4-methyl-6-[4-(1H-pyrazole-5-carbonyl)piperidin-1-yl]pyrimidine-2-carbonitrile 5-chloro-2-[4-(4-ethoxyphenyl)cyclohexyl]-6,7-dihydro-4H-[1,3]thiazolo[4,5-c]pyridine 3-[2-(1-benzothiophen-5-yl)pyrimidin-4-yl]phenol 2-[(4-methoxyphenyl)methylamino]-N-[[4-(1H-pyrazol-5-yl)phenyl]methyl]benzamide (2S,3R)-5-[(4-aminopiperidin-1-yl)methoxy]-N-[(2R)-7-fluoro-2-(hydroxymethyl)-3-methylheptyl]-2-[(3-methylphenyl)methyl]-6-oxo-3,4-dihydro-2H-pyran-3-carboxamide;hydrochloride 1-(4-bromophenyl)-5-[2-methylbutanoyl(propyl)amino]pyrazole-3-carboxylic acid 5-[[4-amino-2-(3,5-difluorophenyl)quinazolin-6-yl]methyl]-1H-pyridin-2-one 1-(5-ethoxycarbonylthiophene-2-carbonyl)pyrrolidine-2,4-dicarboxylic acid N-cyclohexyl-4,5-dimethoxy-2,3-dihydroinden-1-imine N-[2,2-dimethoxyethyl(1,3-thiazol-5-yl)amino]-4-nitrobenzamide N-(4-acetamidophenyl)-3-[[(Z)-2,4,6-trimethylhepta-1,3,5-trienylidene]amino]benzamide N-(1,3-benzothiazol-2-yl)-N-[4-(ethylsulfonylamino)-2-methoxyphenyl]formamide 2-fluoro-4-(5,6,7,8-tetrahydro-4H-[1,3]thiazolo[5,4-d]azepine-2-carbonyl)benzonitrile 3-[4-(2,6-dichloro-3-fluoroanilino)cyclohexyl]oxy-1,5,6,7-tetrahydroindol-4-one 4-azido-2-bromo-1-tert-butylsulfonylbenzene 5-[(4-nitrobenzoyl)amino]hexanoic acid 2-ethenylimino-N',N'-dimethyl-1H-indole-3-carboximidamide;(6S)-5-hydroxy-8,9-dihydro-6H-[1]benzofuro[2,3-e]benzimidazole 2-[4,5-dimethoxy-6-[[(1R)-3-oxospiro[cyclohexane-1,1'-isoindole]-1'-yl]methyl]pyridazin-3-yl]acetamide 1-(3,4-dihydro-2H-pyrrol-5-yl)-2-methylidene-5-pyridin-2-ylimidazolidine 5-azidosulfanyl-2-chloro-1,3-difluorobenzene 2-[4-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-1-ethylcyclohexa-2,4-dien-1-yl]-5-[4-hydroxy-3-(3-methoxypropyl)piperazin-1-yl]pyrazine-2-carboxamide 2-[5-[3-(3,6-dihydro-2H-pyridine-1-carbonyl)phenyl]-4-phenoxypyridin-2-yl]benzonitrile 2-[4-(aminomethyl)phenyl]-5,8-dihydroxy-3H-chromene-4,7-dione 5-cyclopentyl-N,1-dimethyl-6H-pyrrolo[2,3-c]pyrazole-4-carboxamide N-[(6R,7S)-3-methylsulfanyl-5-oxo-7-thiophen-2-yl-4H-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]benzamide 1-[(4R)-3,3-dimethylpiperidin-4-yl]-N-(6-methoxypyridin-2-yl)indole-5-carboxamide 4-N-[2-(furan-3-yl)ethyl]-6-methylpyridine-2,4-dicarboxamide N-[4,4-difluoro-1-hydroxy-2-(hydroxymethyl)butan-2-yl]-3-iodobenzamide 2-[(E)-hex-4-enoxy]-1,3,5-triazine 1,3-dichloro-5-[4-ethenyl-2,6-bis(trifluoromethoxy)phenoxy]-2-fluorobenzene 2-[3,5-bis(trifluoromethyl)phenyl]-N,4-di[(2-methoxyethylamino)methylidene]-6-(trifluoromethyl)piperidine-1-carboxamide (4aR,6S,8aS)-2-ethylsulfanyl-N-[3-(tetrazol-1-yl)phenyl]-6-(2,4,5-trimethoxyphenyl)sulfonyl-1,3,4,4a,5,6,7,8-octahydroisoquinoline-8a-carboxamide (2-butyl-1,3-thiazol-4-yl)-[4-[5-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl]methanone (E)-3-(5-fluoro-2-iodophenyl)but-2-enal 4-[(4Z)-2-chlorohexa-1,4-dienyl]-6-methoxy-5-propylpyrimidine 2-[4-chloro-2-[4-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)piperidine-1-carbonyl]phenyl]acetic acid 2-(1,3-dimethylpyrazol-4-yl)-5-iodoiodanuidyl-4-propan-2-yl-1H-pyrimidin-6-one 5-[4-amino-3-(6-chloro-2,7-naphthyridin-1-yl)phenyl]cyclopentene-1-carboxylic acid 5-methoxycarbonyl-2-(trifluoromethyl)benzenesulfinic acid 3-methyl-6,7-dioxo-4H-thieno[2,3-c]pyridine-5-carboxamide (2E)-1,3-dimethyl-N'-[3-(trifluoromethoxy)phenyl]hexa-2,4-dien-1-imine ethane;3-[2-[(Z)-1-phenylbut-1-enyl]quinolin-6-yl]propanoic acid 6-(dimethylamino)-N-[(2-ethyltriazol-4-yl)methyl]pyridine-3-carboxamide (2E,3Z)-1,5-bis[2,6-di(propan-2-yl)phenyl]-3-ethylidene-4-methylidenepyrrolidine;ethane (2R)-3-azido-1-[4-(2,6-dimethoxypyrimidin-4-yl)piperazin-1-yl]propan-2-ol 2-[2,3-dihydroxypropyl(methylsulfonyl)amino]benzenesulfonic acid (E)-2-[5-amino-6-(quinolin-8-ylmethoxy)pyridine-3-carboximidoyl]pent-1-en-1-ol N-[3,5-dichloro-4-(9H-pyrido[2,3-b]indole-7-carbonyl)phenyl]acetamide 3-[2-(4-chlorophenyl)ethynyl]-1,2-benzoxazole 5-methyl-2,4-dipentoxyaniline 2-chloro-N-[[4-(1H-pyrazol-5-yl)phenyl]methoxy]acetamide (2S)-2-amino-5-[[8-butyl-4-methoxy-6-phenylmethoxy-7-[2-(1,3-thiazol-2-yl)ethynyl]quinoline-2-carbonyl]amino]pentanoic acid [3-[4-(1,3-benzodioxol-5-yl)phenyl]sulfanyloxetan-3-yl]methanamine 3-[3,5-dichloro-4-(2-fluorophenyl)phenyl]-1-methyl-5-methylideneimidazolidine-2,4-dione;ethane 1-[3-amino-4,5,6,7-tetradeuterio-2-(difluoromethyl)phenyl]pentan-1-one (2S)-1-[4-[3-fluoro-4-(trifluoromethyl)phenyl]pyridin-2-yl]-N-propylsulfonylpyrrolidine-2-carboxamide [3-amino-6-(2,4-difluorophenyl)-1-benzofuran-2-yl]methylideneazanium N-(4-bromobutan-2-yl)-N-[6-(4-methoxyphenyl)pyridazin-3-yl]acetamide 6-chloro-3-methyl-5-nitropyridine-2,4-diamine (4E)-2-[2-(3,5-dimethoxyphenyl)ethynyl]-4-[(3-nitropyridin-1-ium-1-yl)methylidene]-6,7-bis[(4-nitrophenyl)sulfanyl]-8H-quinazoline 1,2-difluorobenzene;5,8-dimethyl-4-[3-(6-propan-2-yloxypyridin-3-yl)phenoxy]pyrrolo[2,3-g]quinoline 4-(N-cyclohexylanilino)benzenesulfonic acid 7-methylsulfonyl-1,3,4,5-tetrahydropyrido[2,3-e][1,4]diazepine 4-(3-fluoro-2,4-dimethylphenyl)sulfinyl-1,5-dihydropyrazole 2-amino-6,9-dibromo-5-(2,3,4-trimethoxyphenyl)nonanoic acid 3-N,5-dicyclopropylpyridine-2,3-disulfonamide 4-[5-(6,7-dihydro-1H-benzimidazol-2-yloxymethyl)triazol-1-yl]phenol N-butyl-2,4-dichloro-N-(2H-tetrazol-5-yl)pyrimidin-5-amine N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]-4-methoxybenzamide N-[2,3-dihydroxypropyl(pyridin-2-yl)amino]benzenesulfonamide 2-(4,5-dihydro-1H-imidazol-2-yl)benzenecarboximidamide (7R)-4,8-dimethyl-2-[[1-[(3S)-oxolan-3-yl]pyrazol-4-yl]amino]-5,7-dihydropteridin-6-one 7-(2-chloro-3,5-dimethoxyphenyl)-12-[2-[4-(3,4-difluorophenyl)piperazin-1-yl]ethylamino]-N-(2,6-dioxopiperidin-3-yl)-5-methyl-9-thia-3,4,6,10-tetrazatricyclo[8.3.0.02,6]trideca-1(13),2,4,11-tetraene-11-carboxamide 3-[(4-chlorophenyl)methyl]-N-piperidin-4-ylidene-1,2,4,5-tetrahydro-1,5-benzodiazepine-7-carboxamide;formic acid N-[1-(3-methoxyphenyl)ethenyl]-N',2-dimethylbenzenecarboximidamide 7-[5-[4-(2-hydroxyethyl)phenyl]-4,6-dihydro-1H-pyrimidin-2-yl]-8a-methyl-3a,4-dihydrobenzo[g]isoquinoline-1,10-dione (Z)-2-[5-chloro-3,4-difluoro-2-(trifluoromethyl)phenyl]-3-(cyclopropylamino)-3-hydrazinylidene-N-[4-hydroxy-2-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]prop-1-enamide 3-[[4-[(2S,3R)-5-benzyl-3-methyloxan-2-yl]phenoxy]methyl]pyridine 4-[(E)-3,3-dimethylbut-1-enyl]-2-fluoro-N'-(5-methyl-3-phenyl-1H-pyrazole-4-carbonyl)benzohydrazide;methanamine [1-(6,7-dimethoxyquinazolin-4-yl)piperidin-3-yl]-pyrrolidin-1-ylmethanone 3-(2,3-dihydroindol-1-yl)-5-(2-piperidin-4-ylethyl)oxolan-2-ol 1-[3-(dimethylamino)propyl]-2,4-bis(methoxymethyl)-5-methylpyrrole-3-carboxylic acid 1-[3-(methylamino)propyl]-2,3-dihydropyrrolo[3,4-c]isoquinolin-5-one 5-[4-fluoro-3,3,6-trimethyl-1-(2,4,6-trichlorophenyl)-2H-pyrrolo[2,3-b]pyridine-2-carbonyl]-1H-pyridin-2-one N-[1-(4-tert-butylphenoxy)pyridin-3-ylidene]hydroxylamine 5-[(1E,3Z)-4-methoxybuta-1,3-dienyl]-6-propan-2-ylidenecyclohepta-1,3,7-triene 7-(1,3-benzodioxol-5-yl)-2-[(2E)-2-ethenylpenta-2,4-dienoxy]imidazo[2,1-f][1,2,4]triazin-4-amine 2-[3,5-dichloro-4-(7-oxo-6H-[1,3]oxazolo[4,5-d]pyrimidin-6-yl)phenyl]-3,5-dioxo-1,2,4-triazinane-6-carbonitrile 6-[1-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzoyl]piperidine-4-carbonyl]oxypyridine-3-carboxylic acid 2-[4,6-bis(trifluoromethyl)pyridin-2-yl]-1H-pyrazole-3-thione 4-(2,5-dimethylphenyl)sulfonyl-6-[3-fluoro-5-(trifluoromethyl)pyridin-2-yl]-2,3-dihydro-1,4-benzoxazin-7-amine 6-[2-(3-methoxyphenyl)pyrimidine-4-carbonyl]-8a-methyl-1,5,7,8-tetrahydro-[1,3]oxazolo[3,4-a]pyrazin-3-one (4Z)-2,3-bis[(4-methoxyphenyl)methyl]hexa-2,4-dienamide 1-chloro-2-methylbenzene;5,7-difluoro-N-(2-hydroxyethoxy)quinoline-8-carboxamide;uranium(2+) 2-[3-methoxy-4-(propylcarbamoylamino)phenyl]acetamide (E)-3,4-diamino-N-[(1S)-2,2-difluorocyclopropyl]-5-quinolin-8-ylpent-2-enamide ethane;7-fluoro-2,3-dimethyl-5-[4-(trifluoromethoxy)phenyl]-1H-indole 4-[(5R)-4-cyclohexyl-2,5-dioxoimidazolidin-1-yl]benzonitrile;ethane N-(2,3-dihydro-1H-inden-5-yl)-2-[[6-oxo-4-(propan-2-ylamino)-1H-pyrimidin-2-yl]sulfanyl]acetamide N'-[(E)-4,5-dimethylideneoct-1-enyl]-N-methylidenepyridine-2-carboximidamide N-[1,2,3,5,6,7-hexahydropyrrolizin-8-ylmethyl(phenyl)phosphanyl]ethanamine 2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3H-quinazolin-4-one N-[(1R,3S)-3-azidocyclopentyl]-6-phenylthieno[2,3-d]pyrimidin-4-amine 2-azido-6-methylsulfanyl-1,3-benzothiazole 2-[(5-benzyl-1H-pyrrole-3-carbonyl)amino]acetic acid N-(4,5-dimethylpyridin-2-yl)-3-fluoropyridine-4-carboxamide 2-(3,5-dimethoxyphenyl)-4-(methylamino)quinazoline-7-carbonitrile [4-(3,5-dimethylpiperidine-1-carbonyl)phenyl]urea 3-fluoro-4-methylsulfanylbenzaldehyde;2,2,6,6-tetramethylpiperidin-1-amine 1-[2,2,3,3-tetrafluoro-4-(2,2,3,3,5,5,6,6-octadeuteriomorpholin-4-yl)oxybutanoyl]oxynaphthalene-2-carboxylic acid 6-(2,5-dimethylpyrazol-3-yl)-7H-purine (2-chloro-6-ethoxyphenyl)methyl-diethoxyphosphane N-ethylsulfonyl-3,5-dinitrobenzenecarboximidate 2,3-bis(ethenyl)-6-methylidene-1,4-dihydropyrido[1,2-a]benzimidazole;ethane N-[2-[3-[1-(aminomethyl)cyclopentyl]phenyl]ethyl]formamide 3-[4-methyl-2-[4-(3-phenylpropyl)piperazine-1-carbonyl]-1,3-thiazol-5-yl]indole-1-carboxamide 2-methyl-6-propan-2-ylimino-3-pyridin-4-yl-5H-pyrimidin-4-one 5-[6-(ethylamino)pyrimidin-4-yl]oxy-1,3,3a,4,5,6,6a-octahydropyrrolo[2,3-c]pyrrole-2-carboxylic acid N-[2-(3,5-difluorophenyl)ethyl]-4-[6-methyl-4-(trifluoromethoxy)cyclohexa-1,3-dien-1-yl]aniline 1-azidooxy-4-methoxy-2,3,5,6-tetramethylbenzene 4-(2,3-dimethylphenyl)piperidine-4-carboxylic acid 1-[2,2,2-trifluoro-1-(2-methylphenyl)ethyl]pyrazolidin-3-one 4-amino-3,5-dibromobenzoic acid;1,4-dimethylbicyclo[2.2.2]octane 1-chloro-4-(1,1-difluoroethyl)benzene;5-[3-[cyclohexa-2,4-dien-1-ylidenemethoxy-[(Z)-1-iminobutan-2-ylideneamino]methyl]-5-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazol-1-yl]pyridine-3-carbonitrile 2-[6-[(3S)-oxolane-3-carbonyl]-5,7-dihydro-4H-thieno[2,3-c]pyridin-2-yl]-1,8-naphthyridine-4-carboxamide (1-amino-4-propan-2-ylcyclohexa-2,4-dien-1-yl)-phenylmethanone N-[6-[2-fluoro-4-(trifluoromethyl)phenoxy]pyridin-3-yl]-1H-indole-5-carboxamide N-(1H-benzimidazol-2-ylmethyl)-5-chloro-1H-pyrrolo[3,2-b]pyridine-2-carboxamide;ethane 1-[4-(4-azidophenyl)cyclohexyl]-6,7-dihydro-5H-indol-4-one N-[(1R,2S)-1-azido-2-methylcyclohexyl]-3,5-dichloro-4-fluorobenzamide 2,4-ditert-butyl-6-(3-methoxy-6-phenylpyridin-2-yl)phenol 2-[3-methylbut-2-enyl-(6-nitro-1,3-benzothiazol-2-yl)amino]propanoic acid 2-amino-1-(4,4,5,5-tetramethylhexan-3-yl)pyrimidin-4-one [3-(cyclopropylmethoxy)pyrrolidin-1-yl]-imidazo[2,1-b][1,3,4]thiadiazol-6-ylmethanone ethane;1-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrrolidine 2-[1-(3-ethylsulfonylpropanoyl)piperidin-4-yl]oxy-5,6-dimethylbenzonitrile 3-[2-(2,4-dimethoxyphenyl)ethylamino]-5-[3-(methyliminomethyl)phenyl]pyrazine-2-carboxamide;ethane N'-ethyl-4-oxo-3,10-diazatricyclo[5.2.0.01,6]undeca-2(6),7-diene-9-carbohydrazide (5Z)-2-(4-bromophenyl)imino-5-[[3,5-diiodo-4-[(4-nitrophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one 2-(5,6-difluorobenzimidazol-1-yl)-1-[4-[3-[(7S)-7-hydroxycycloocta-2,4,6-trien-1-ylidene]aziridin-2-yl]-1,3-thiazol-2-yl]ethanone 2-bromo-1,4,5-trifluoro-3-methoxybenzene [2-(1,3-benzothiazol-6-yl)morpholin-4-yl]-[5-methoxy-1-[2-(trifluoromethyl)phenyl]sulfonylpyrazol-3-yl]methanone 1-azidosulfanyl-3,5-dichlorobenzene 2-[[3-[4-(1H-benzimidazol-2-ylsulfanylmethyl)triazol-1-yl]phenyl]methoxy]-5-methylbenzoic acid 1-[4,6-bis(trifluoromethyl)pyrimidin-2-yl]naphthalene-2-sulfonate 2,5-dichloro-N-[4-[(3-methylphenyl)carbamoyl]phenyl]benzamide (1E,6E)-4-N-[5-bromo-2-[3-(dimethylamino)propoxy]phenyl]-6-methoxy-4-N,4-N-dimethylcyclodeca-1,6-diene-1,4-diamine 3-amino-N-ethylsulfonyl-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-2-carboxamide 2-methoxycarbonyl-6-(4-octylsulfanylphenyl)hex-3-enoic acid 3-[(1,5-dimethylpyrazol-4-yl)sulfonylamino]-5-propan-2-ylthiophene-2-carboxylic acid 4-amino-N-(3,6-dihydroxyxanthen-9-ylidene)benzamide (3R)-7-[(3S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-3-methoxy-3-(phenylsulfanylmethyl)-1H-indol-2-one N-(2,6-dimethylphenyl)-4-[[(1S)-3-oxocyclohexyl]carbamoylamino]benzamide 2-(difluoromethyl)-N-[4-(4,6-dioxo-1H-1,3,5-triazin-2-yl)phenyl]benzamide 6-(1,3-thiazol-2-ylamino)hexanoic acid 1,1-difluoro-2H-benzo[e][1]benzoxepine 6-(4,4-dimethylcyclohexyl)-3-ethoxy-5H-pyrrolo[3,2-d]pyrimidin-1-ium 2-azido-N,N',2-trimethyl-N-(4-phenylbutyl)propane-1,3-diamine 4-(1,2,3,6-tetrahydropyridin-4-ylmethoxy)benzonitrile (2R)-N,3-bis(4-chlorophenyl)sulfanyl-1-phenylpropane-1,2-diamine 3-(2,4-difluorophenyl)-N,5-bis[(4-hydroxypiperidin-1-yl)methyl]-3a,4,5,6,7,7a-hexahydro-1-benzofuran-2-carboxamide N-[2-(2-methoxyethyl)pyrazol-3-yl]-4-methylidenepiperidine-1-carboxamide 2-[3-bromo-4-(trifluoromethyl)phenyl]-1,3-dioxolane N-[4-(3,3-difluoroazetidin-1-yl)phenyl]-5-methylthieno[2,3-d]pyrimidin-4-amine [6-(methoxymethyl)pyridin-3-yl]-(4-pyridazin-3-ylpiperazin-1-yl)methanone 1-[2-(1,3-benzothiazol-6-yloxy)ethyl]-4-hydroxypiperidine-4-carboxylic acid 3-[5-(3,4-dichlorophenoxy)-7-nitro-2H-indazol-3-yl]-1-methylcyclohexane-1-carboxylic acid N-ethylsulfonyl-N-[4-methoxy-2-(5-oxo-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-4-yl)phenyl]acetamide 3-hydroxy-N-[5-(2-morpholin-4-ylethoxy)-1H-indol-7-yl]propanethioamide 4-methylsulfonyl-6,11-dihydrothiochromeno[2,3-b]indole 1-(azidooxymethyl)-3,5-bis(trifluoromethyl)benzene 4-[(4-fluoro-5,6,7,8-tetrahydronaphthalen-1-yl)methoxy]-2,3-dihydroinden-1-one (2Z,4E)-5-(methylideneamino)-N-[(1S)-6-(2-phenylethylcarbamoyl)cyclohex-3-en-1-yl]penta-2,4-dienenitrilium 4-[3-(2,5-dimethylphenyl)cyclopenta-1,4-dien-1-yl]aniline 3-[4-(4-chlorophenyl)-5-cyclobutyl-1,2-oxazol-3-yl]-5-ethoxycarbonylbenzoic acid 4-[[1-(2,5-difluorophenyl)ethylamino]methyl]benzamide 3-fluoro-2-(4,5,6-trimethoxypyridin-3-yl)quinoline 2-(5-ethyl-6,8-dihydro-5H-imidazo[1,5-a]pyrazin-7-yl)-N-methylpyrimidine-4-carboxamide;2,2,2-trifluoroacetic acid 4-[7,8-difluoro-2-[3-fluoro-5-(trifluoromethyl)phenyl]-6-propan-2-yloxyquinazolin-4-yl]morpholine 2-(1H-benzimidazol-2-ylmethoxy)benzoic acid 4-[1-(2,3-dihydroimidazo[1,2-a]pyridin-5-yl)ethoxy]benzaldehyde 4-[(2S)-1-(5-methylthiophen-3-yl)sulfonylpyrrolidin-2-yl]-6-phenylpyrimidine N-ethyl-N,1-dimethyl-4,5-dihydroindazole-6-carboxamide 6-amino-4-(1,3-benzothiazol-2-yl)-7-methoxy-2-piperidin-4-yl-1H-indole-5-carbonitrile 2-(4-methylpiperazin-1-ium-1-ylidene)-N,3-diphenyl-1H-quinazolin-7-amine 2-amino-3-[4-(dibutylamino)phenyl]propanamide N-[(1R,2S)-2-aminocyclohexyl]-6-hydroxyimidazo[1,5-a]pyridine-3-carboxamide 1-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]pyrazole-3-carboxamide N-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]-3-oxobutanamide 2-[4-(azidomethyl)phenyl]-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one 1-[4-amino-5-(4-aminophenyl)pyrrolo[2,3-d]pyrimidin-7-yl]hexan-1-one (2R)-3-[4-amino-3,5,6-trifluoro-2-(methoxymethyl)phenyl]-N-[3-oxo-7-(1,1,4-trioxo-1,2,5-thiadiazolidin-2-yl)heptanoyl]propane-1-sulfonamide 5-ethylsulfanyl-2-methoxy-3-methylpyrazine 5-(2,2-difluoroethoxy)-1-[4-[(4-oxocyclohexyl)methyl]phenyl]indole-3-carboxylic acid (2S)-2-[[[5-chloro-2-[5-fluoro-6-(methylamino)pyridin-3-yl]pyrimidin-4-yl]amino]methoxy]butanamide N-[(1S)-4,5,6,7-tetrahydro-2,1-benzoxazol-3-yl]methanesulfonamide 6-[(6S)-2,7-dimethyl-3H-imidazo[4,5-c]quinolin-1-ium-8-yl]oxyhexanoate N-[4-[6-(methylamino)pyrido[3,2-d]pyrimidin-7-yl]phenyl]acetamide;propane (3S,5R)-2-[4-chloro-3-[[3-methyl-1-(6-oxo-1H-pyridazin-3-yl)pyrazol-4-yl]methylamino]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol 1-(1-azidopropan-2-yl)-4-(trifluoromethoxy)benzene 2-methyl-4-[4-(2-oxopiperidin-1-yl)phenyl]piperazine-1-carboxylic acid 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[5-(methoxymethyl)-1-methyl-1H-pyrazol-3-yl]sulfonylurea N-[2-(2-cyano-4,4-difluoropyrrolidin-1-yl)-2-oxoethyl]pyridine-3-carboxamide 1-(7-bromo-4H-1,3-benzodioxin-5-yl)propane-2,3-dione 2-(3,4-dimethoxyphenyl)sulfanyl-1H-indole 3-amino-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide;3-ethyl-8-[(E)-2-(6-methoxypyridin-3-yl)prop-1-enyl]-2H-isoquinolin-1-one 2-[(5S,8aS)-7-(1-methylpyrazole-4-carbonyl)-5-phenyl-3,6-dihydro-2H-furo[3,2-e]indol-5-yl]-N-cyclopropylacetamide 2-[4-hydroxy-3-(2H-naphthalen-1-ylideneamino)phenyl]propanedioic acid (E)-3-[4-(dimethylamino)phenyl]prop-2-enehydrazide 2-(7,8-dihydronaphthalene-1-carbonylamino)butanoic acid;hydrochloride 7-bromo-6,8-dichloro-4H-1,4-benzoxazin-3-one 1-[(4Z)-hepta-2,4,6-trienyl]-2,7-dimethyl-5,6-bis[(E)-pent-3-enyl]naphthalene (2S,4R)-1-[(2E,3Z)-2,3,6-diethylnona-2,5,8-trienoyl]-4-hydroxy-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide;N-(3,5-difluorophenyl)formamide 3-(3,5-difluorophenyl)-2-[(4-methylpyrazol-1-yl)amino]propanal 3-[[6,8-bis(3-chlorophenyl)imidazo[1,2-a]pyrazin-2-yl]amino]-N-hydroxypropanamide 6-(1H-pyrazol-5-yl)imidazo[2,1-b][1,3]benzothiazole 6-hydroxy-5-[(2-methoxyquinolin-4-yl)methyl]-3-phenylmethoxypyran-2-one 4-[8-(1H-pyrazol-5-yl)imidazo[1,2-a]pyrazin-6-yl]phenol [4-(6,7-dihydro-2H-1,3-benzoxazol-3-yl)piperidin-1-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone 1-[6-(methylsulfanylamino)pyridine-3-carbonyl]piperidine-4-carboxylic acid 4-[(1R)-1-azidoethyl]-2,6-bis(trifluoromethoxy)benzonitrile (5S)-3-[4-methoxy-3-(2-oxopyrrolidin-1-yl)phenyl]-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxamide N-cyclohexyl-4-nitro-2,5-diphenylpyrazole-3-carboxamide 6-[4-amino-3-(2,5-dihydrofuran-3-yl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohepta-1,3,5-triene-1-carboxamide (2S)-N-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]piperidine-2-carboxamide 3-[[[4,5-bis(ethenyl)-6-oxo-1H-pyrimidin-2-yl]amino]methyl]benzamide 4-N-ethyl-5-(2-fluorophenyl)-6,7-dimethyl-2H-pyrrolo[1,2-a]quinazoline-3,4-diamine 4-ethyl-3,5-dinitrophenol 1-[1-(oxan-2-yl)pyrazol-4-yl]indole 3-(4-methylphenyl)-6,7,8a,9-tetrahydro-5aH-pyrrolo[2,1-c][1,4]benzodiazepine N-[(4-chlorophenyl)methyl]-5,6-difluorocyclohexa-2,4-diene-1-carboxamide 7-methoxy-1,2-dihydro-[1]benzothiolo[3,2-f]benzimidazole (4E)-4-[(5,7-dihydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)methylidene]pentanoic acid 1-cyclopropyl-4-[(2,3-difluorophenyl)methyl]pyrrolidine;ethane N-[1-(4-chlorophenyl)ethenyl]-2,6-dimethylaniline 1-[4-(azidomethyl)phenyl]-N-[3-chloro-2-methoxy-5-(trifluoromethyl)pyridin-4-yl]sulfanylcyclopropane-1-carboxamide 2-ethyl-N-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yloxy)cyclohexyl]imidazo[1,2-a]pyrimidine-3-carboxamide 5-[1,3-bis(methylsulfanylamino)propoxy]-1-propylbenzimidazole-2-carboxylic acid 3-chloro-1-[4-fluoro-2,6-di(propan-2-yl)phenyl]-5-methoxypyrazole [4-(4-chlorophenyl)piperazin-1-yl]-[3,5-dihydroxy-7-methyl-2-(2-morpholin-4-ylethoxy)-1H-imidazo[1,2-a]pyrimidin-8-ium-6-ylidene]methanolate 3-(2,2-dimethylpentanoylamino)oxybenzenesulfonic acid (2S)-4-hydroxy-1-[4-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyloxymethyl)benzoyl]pyrrolidine-2-carboxylic acid (2R,3S)-N'-[(2R)-1-[(5-bromothiophen-2-yl)methylamino]propan-2-yl]-2-hydroxy-4-phenylbutanediamide 1-(4,6-dimethylpyridine-2-carbonyl)-N-ethylazetidine-3-sulfonamide 1-[(2S)-4-(7-fluoro-2,3-dihydro-1H-indole-5-carbonyl)-2-methylpiperazin-1-yl]-2-(1-oxo-8,9-didehydroisoquinolin-2-yl)ethane-1,2-dione N-(4-aminocyclohexyl)-2-methoxybenzenesulfonamide 5-[(4,6-dichloro-1,3,5-triazin-2-yl)methyl]-1-methylindole 4-[3,5-bis(2-cyanopropan-2-yl)phenyl]benzonitrile 3-[6-azidooxy-2-(furan-3-yl)-1,4-dimethylindol-3-yl]propanoic acid N-(diaminomethylideneamino)benzamide 5-(2,6-dimethoxyphenyl)-N-[1-[4-[(3R)-3-pyrrolidin-1-ylsulfonylpyrrolidin-1-yl]benzoyl]azetidin-3-yl]-1H-pyrazole-4-carboxamide 4-[2,6-bis(hydroxymethyl)phenyl]-3,5-dibromophenol 4-amino-6-[(6,7-dimethoxy-1,5-naphthyridin-4-yl)oxy]-1H-benzimidazole-2-carboxamide 2-[4-(3,5-dimethylphenyl)-6-[(2E,3Z,5Z)-hepta-2,5-dien-2-yl]pyridin-2-yl]aniline 2-[4-(4-ethylphenyl)phenoxy]ethanol 6-(4-hydroxyphenyl)-2,3,5,8-tetrahydroimidazo[1,2-a]pyrimidine-7-thione 2-(3-chlorophenyl)-3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-ylidene]-5-ethylquinazolin-4-one 5-methoxy-N-(1,3,4-thiadiazol-2-yl)quinoline-6-carboxamide 2-[(3S,4R)-1-cyclobutylsulfonyl-4-methoxypyrrolidin-3-yl]-5-methylpyridine (5S)-5-[2-[1,4-dimethyl-3-(trifluoromethyl)pyrrol-2-yl]pyridin-4-yl]oxyhexanoate 3-(1-phenylethylamino)naphthalene-2,7-disulfonic acid (2R,3S)-4,4-difluoro-N-[5-methyl-6-(8-methylimidazo[1,2-a]pyridin-6-yl)oxyisoquinolin-3-yl]-3-(trifluoromethyl)pyrrolidine-2-carboxamide 1-azidooxy-4-[2,6-di(propan-2-yl)phenoxy]benzene 3-(N-acetylanilino)propanoic acid 5-chloro-N-[3-(2,6-dimethylmorpholine-4-carbonyl)-4-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide 2-N,4-diphenylquinazoline-2,6-diamine 3-azidooxy-2,4-dichlorobenzoic acid 4-[2,3-dihydroxypropyl(methoxycarbonyl)amino]benzenesulfonic acid 1,3-bis[2,6-di(propan-2-yl)phenyl]-2H-imidazol-2-ide;1-methanidylbenzimidazole;tin(2+) (2S)-N-[4-fluoro-5-(1H-indole-2-carbonylamino)-3,6-dihydro-2H-pyridin-1-yl]oxolane-2-carboxamide 5-chloro-4-[(3R,6S)-1-methylazepan-3-yl]oxypyrimidine N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-hydroxypyridine-2-carboxamide 2-[(3,5-dichlorophenyl)methyl]decanoic acid ethane;N'-[5-(trifluoromethyl)pyridin-2-yl]ethane-1,2-diimine 5-[3,4-di(propan-2-yl)furan-2-carbonyl]-N,1-diethyl-2,6-dihydropyridine-3-carboxamide ethane;7-[(E)-2-(3-methylphenyl)ethenyl]-2,3-dihydropyrido[1,2-a]pyrimidin-4-one 5-[(3-chlorophenyl)methyl]-4-methoxypyrimidine 5-[2-[4-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]phenyl]ethynyl]pyridin-2-amine 1-(3,4-dichlorophenyl)-N'-[3-methylsulfanyl-5-(trifluoromethoxy)phenoxy]ethane-1,2-diamine (3Z)-N-[2-(4-ethylpiperazine-1-carbonyl)cyclohexa-2,4-dien-1-yl]-5-fluoro-6-[(E)-2-pyrrolidin-1-ylprop-1-enyl]hepta-3,5-dienethioamide 2,4-dimethoxybenzimidazole-1-carboxamide 2-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide 2-azido-6-methylsulfonylpyrazine 5-[3,5-bis(methylamino)phenyl]-1H-indole-2-carbonitrile N-[4-(dimethylamino)phenyl]-2-(7-fluoroquinolin-4-yl)oxyacetamide 6-[(1S)-2,2,5-trimethyl-4-[6-(trifluoromethoxy)pyridin-3-yl]cyclohexyl]quinoline 4-chloro-5-(1,3-dioxoisoindol-2-yl)-N-[(4S,5R)-4-hydroxy-8-oxabicyclo[10.4.0]hexadeca-1(12),13,15-trien-5-yl]pentanamide 2-[[1-(5,7-dimethoxyquinazolin-4-yl)piperidin-3-yl]methylideneamino]-5H-pyrimidin-6-one 6-butoxy-5,7-difluoro-2-(4-methylcyclohexen-1-yl)-2H-chromene-3-carboxylic acid (2-bromoimidazo[1,2-a]pyridin-3-yl)methanamine (4S,6R)-2-[2-methyl-4-[(3-nitrophenyl)diazenyl]phenoxy]-4,5,6,7-tetrahydroisoindole-1,3-dione (5-benzylsulfanyl-1,3-thiazol-4-yl)methanediol 6-tert-butyl-8H-cyclohepta[d]pyrimidine 1-(2-fluorophenyl)-3,5-dimethyl-7-oxabicyclo[4.1.0]heptane 4-bromo-3-[[5-methyl-1-[(2E)-penta-2,4-dien-2-yl]pyrazol-4-yl]sulfonylamino]benzoic acid 2-[(4S,6Z)-3-methyl-8-(1H-pyrazol-5-yl)deca-4,6,9-trienyl]phenol 3-azidooxy-5,6,7,8-tetrahydronaphthalene 7-(6-methylpyridin-3-yl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine 5-azidooxysulfonylnaphthalene-2-sulfonic acid ethane;N-[(Z)-1H-indol-3-ylmethylideneamino]-4-nitrobenzamide N-(2-hydroxyethyl)-4,5-dimethoxy-3-[[(E)-octadec-9-enoyl]amino]naphthalene-1-carboxamide 5-[3-(2,6-dimethylpyridin-4-yl)phenyl]-4-ethyl-1H-pyrimidin-6-one N-[1-(5-azidopyridin-2-yl)piperidin-4-yl]cyclopentanecarboxamide [3-[4-(benzenesulfonyl)phenyl]pyrrolidin-1-yl]-(6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl)methanone 1-[5-(2-azidoethyl)-6-nitropyridin-3-yl]piperidine-4-carboxamide N-(4-chlorophenyl)sulfonyl-1,3-dimethylpyrazolo[3,4-b]pyridine-5-carboxamide N-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-2-yl)butanamide 5-methyl-N'-[2,3,4-trimethyl-6-(methylideneamino)phenyl]pyridine-2-carboximidamide 3-fluoro-5,11a-dihydro-6H-benzo[c][1]benzazepine (2S)-4-hydroxy-N-[[(6R,7aS)-2-methyl-1,3,3a,5,6,7,7a-octahydroisoindol-4-yl]sulfonyl]-1-phenylazetidine-2-carboxamide 2-(4-cyclopropylphenyl)imino-6,7-dihydro-3H-[1]benzofuro[3,2-d]pyrimidin-4-amine N-(3-amino-5,6,7,8-tetrahydronaphthalen-2-yl)-4-phenylthiophene-3-carboxamide 2-[4-(4-azidophenoxy)piperidine-1-carbonyl]benzonitrile 1-(4-chlorophenyl)-4-methoxycyclohexa-2,5-diene-1-carboxylic acid (2Z)-3-[2-(5-chloro-2-methoxyphenyl)ethyl]-2-propylidene-6,7-dihydroquinoline N-[4,5-dichloro-2-(methylamino)phenyl]-3,4,5-trimethoxybenzenesulfonamide N-(8,8a-dihydronaphthalen-1-yl)dibenzofuran-4-amine 3,4-diethyl-5-fluoropyridine-2-carboxylate 2-(3,4-dimethylphenyl)-N-[1-(4,6-dimethylpyridine-2-carbonyl)piperidin-4-yl]acetamide 3-[(E)-(2,4-dihydroxyphenyl)methylideneamino]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one (2S)-2-[[(2Z,4E)-5-amino-3-cyanohepta-2,4,6-trienyl]amino]-4-methylsulfanylbutanoic acid;ethane 4-[2,5-dimethyl-3-oxo-6-(trifluoromethyl)pyridazin-4-yl]benzonitrile 1-amino-3-[6-methyl-2,4-bis(trifluoromethyl)benzoyl]indole-5-sulfonamide 1-(6,7-dihydronaphthalene-2-carboximidoyl)-4,10-dihydrophenanthren-9-amine N-[3,6-di(butanoyl)imidazo[1,2-b]pyridazin-8-yl]-4-nitrobenzamide 1-(2,5-dichlorophenyl)-4-(dimethylamino)pentan-3-one (4R,5S)-2-[3-fluoro-4-[3-methyl-6-(trifluoromethyl)-1H-indol-2-yl]phenyl]-4,5-dihydroxy-N-methyl-1,3-oxazolidine-3-carboxamide 2,6-diiodo-N'-phenylbenzenecarboximidamide N-(2,6-dichloropyridin-4-yl)sulfanylquinolin-2-amine 6-bromo-3,7-dimethylquinoxaline [(2R)-3-cyclohexyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-2,3'-piperidine]-1'-yl]-pyridin-3-ylmethanone N-[5-(2,6-difluorophenyl)-1H-pyrazol-4-yl]-3,7a-dihydro-[1,2,4]triazolo[4,3-a]pyridine-8-carboxamide (6R)-3,4,8-trihydroxy-7,11b-dimethyl-6-(2H-tetrazol-5-ylmethoxy)-9-(trifluoromethoxy)-1,2-dihydrobenzo[b]quinolizine-10-carboxylic acid N-butanoyl-4-chloro-2-methylpyrazole-3-carboxamide 2-(azidomethyl)-4-[3,5-dichloro-4-[1-[1-(3,3-difluoropropyl)piperidin-4-yl]ethenoxy]phenyl]-6H-pyrrolo[3,4-b]pyrrole (3R)-N-(4,5-dichloro-2-fluorophenyl)-1,3-dimethyl-2-oxopyrrolidine-3-carboxamide 3-[(1R)-5,6,7,8-tetrahydronaphthalen-2-yl]cyclopropane-1,1,2,2-tetracarbonitrile N-[2,4-bis(3-chlorophenyl)phenyl]-6-[6-(ethylaminomethyl)pyridin-3-yl]oxypyrimidin-4-amine 3-(2,6-dichlorophenyl)-7-[4-(4-methylpiperazine-1-carbonyl)anilino]-2H-pyrimido[5,4-e][1,3]thiazin-4-one 4-[3-(4-hydroxypiperidine-1-carbonyl)phenoxy]benzonitrile 2-[(3R)-5-(4-ethoxyphenyl)-1-(2-methylpropanoyl)pyrrolidin-3-yl]-N,N-dimethyl-2-oxoacetamide 4-[3,5-bis(methylsulfanyl)benzoyl]oxybenzenesulfonate 1,2-bis[1-(2-hydroxyphenyl)ethylideneamino]guanidine;hydrochloride 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-propylaniline 1-(6-methoxyquinolin-2-yl)-5H-pyrazolo[4,3-c]pyridin-4-one N-[(5-bromopyridin-2-yl)methylidene]hydroxylamine N-methyl-3,4-diphenylpentan-2-imine N-[4-[(1R)-1-hydroxyethyl]phenyl]-2-(4-morpholin-4-ylanilino)-3H-benzimidazole-5-carboxamide N-[(3S,5R)-1-azabicyclo[4.2.0]octan-3-yl]-1H-indazole-7-carboxamide 2-(4-chlorophenyl)-N-[1-cyclopentyl-2,3-dioxopropan-2-yl]-2-methyl-4-oxo-7H-furo[2,3-b]pyridine-5-carboxamide N-(4,5,6-trimethylpyrimidin-2-yl)dodecanamide 2-[[7-(3,4-dichlorophenyl)-1,4-oxazepane-6-carbonyl]amino]acetic acid 1-(4-azidopyridin-3-yl)benzimidazole N-[4-(N'-hydroxycarbamimidoyl)-1H-pyrazol-5-yl]-2,3-dimethoxybenzamide 1-(4-chlorophenyl)sulfonylsulfonyl-N-[2-fluoro-3,6-dimethyl-5-[(Z)-1,3-oxazol-2-yliminomethyl]phenyl]piperidine-4-carboxamide 1,2-dimethyl-N-[4-[3-methyl-2-(trifluoromethyl)phenyl]cyclohexyl]-6H-pyrrolo[3,2-f]quinazolin-9-amine [3-(4-fluorophenyl)-1,2-oxazol-5-yl]methoxyphosphane 2-[4-[4-(2,3-difluoro-4-methylphenyl)phenyl]cyclohexa-1,5-dien-1-yl]-6-ethoxyoxane [4-(2-cyanopropan-2-yl)phenyl]boronic acid N-[4-amino-3,5-dioxo-2-(phenylcarbamoyl)pyrazolidin-1-yl]-2-chlorobenzamide 7-methyl-N,6-diphenylnonanamide 4-[5,6-bis(phenylmethoxy)pyridin-3-yl]sulfinylbenzoic acid 1-[1,3-bis(2,6-dimethylphenyl)imidazol-1-ium-4-yl]benzimidazole;ethane 6-N-[(4R)-7-chloro-1,2,3,4,5,8a-hexahydropyrido[3,4-b]indol-4a-yl]-7H-purine-2,6-diamine (5S)-2-benzylsulfanyl-N-(4-methoxyphenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide N-(3-cyanophenyl)-2,4,6-trimethyl-N-(3-nitrophenyl)benzenesulfonamide 2-(7,8-difluoro-3H-1,4-benzodioxin-5-yl)-4,5-dihydro-1H-imidazole 1-[5-fluoro-2,3-di(propan-2-yloxy)phenyl]ethanone 2-(4,5-diamino-1,3-thiazol-2-yl)propanoic acid;2-fluoroaniline (1R,3aR,7aS)-N-pyridin-2-yl-5-pyrimidin-5-yl-3,3a,4,6,7,7a-hexahydro-1H-furo[3,4-c]pyridine-1-carboxamide;2,2,2-trifluoroacetic acid (7S)-N-benzyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4-carboxamide 4-amino-N-(1,3-benzothiazol-2-yl)-5-methoxy-3H-indene-1-carboxamide [(2S)-1-(4,5-dichloropyrimidin-2-yl)pyrrolidin-2-yl]methanol 4-[3,5-bis(trifluoromethyl)phenyl]sulfonyl-3-(methoxymethyl)quinoline (5Z)-5-[[3-fluoro-4-[(2-methyl-1H-indol-3-yl)methylideneamino]phenyl]methylidene]imidazolidine-2,4-dione 2-(4-chlorophenyl)-6-ethynylsulfanylquinoline (4R)-1,3-dimethyl-4-[4-[2-oxo-2-[6-[5-(trifluoromethyl)pyridin-3-yl]oxyindol-1-yl]ethoxy]phenyl]-1,3-diazinan-2-one N-[(1,5-dimethylpyrazol-3-yl)methyl]-2-[4-(trifluoromethyl)pyrimidin-2-yl]aniline 3-[2-chloro-5-(trifluoromethyl)phenyl]iminobutanal;N'-methylmethanediamine 2-[2-methoxy-5-(4-propylpiperazine-1-carbonyl)phenyl]acetic acid (6R,7S)-3-chloro-8-oxo-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 1-[4-(3,3a,7a-tetrahydropyrrolo[2,3-b]pyridin-5-yl)phenyl]azetidin-3-ol 1-(1,3-benzodioxol-5-ylmethyl)-4-bromopiperidine 5-[(6S)-1,8,10-trioxo-2-azaspiro[5.5]undecan-4-yl]pyrazine-2-carbonitrile N-[4,5-dimethoxy-2-(1H-pyrrolo[3,2-b]pyridine-3-carbonyl)phenyl]prop-2-enamide 4-[3-(diethylamino)propyl]benzenesulfonamide (E)-N-[4-methyl-3-(morpholine-4-carbonyl)phenyl]hept-2-enediamide 3-[1-(2,3-dimethylphenyl)sulfonylpiperidin-4-yl]-5-[[4-(2-ethoxyphenyl)piperazin-1-yl]methyl]-6H-triazolo[4,5-d]pyrimidin-7-one 6-[(2,4-dimethylphenyl)iminomethyl]-3,7-bis(2-hydroxyethoxy)-1H-quinoline-2,4-dione N-[3-(2,6-difluoroanilino)-4-methoxyphenyl]-1-oxothiane-4-carboxamide 1-methyl-3-(5-methylsulfanylpyrimidin-4-yl)indole 6-(5,7-dimethylthieno[2,3-d]pyridazin-4-yl)-1,2,3,4-tetrahydroisoquinoline 5-[[3,4-bis(difluoromethoxy)phenyl]methyl]-2H-tetrazole N-[2-(4-methyl-6-oxo-1H-pyrimidin-2-yl)ethyl]-2-propan-2-ylidene-3,5-dihydro-1,4-benzodioxine-7-carboxamide 3-[4-(1,2,3,6-tetrahydropyridin-5-yl)phenyl]oxirane-2,2-dicarbonitrile 4-[(2S)-2,6-dimethylmorpholine-4-carbonyl]-2-phenyl-1H-pyrimidin-6-one 5-[(2,3-dimethoxyphenyl)sulfonylamino]-N'-hydroxypyridine-2-carboximidamide 2-[1,3-benzodioxol-5-yl-(2,4-difluorophenyl)methyl]morpholine 4-[5-methylsulfonyl-2,3,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),6,9,11-tetraen-4-yl]benzamide (Z)-N'-benzyl-3-[1-(2,5-difluorophenyl)piperidin-4-yl]prop-1-ene-1,3-diamine 2-(1,3-benzodioxol-5-yl)-4-phenylbutanal 1-[6-(2,3-difluorophenyl)-5-(4-methyl-2H-tetrazol-5-yl)pyridin-3-yl]-N-[(6-ethoxypyrimidin-4-yl)methyl]piperidine-4-carboxamide 2-(4-chlorophenyl)-7-ethylnaphthalene 1-[3-(2-azidoethynyl)phenyl]sulfonylpyrrolidine 1-[3-(2,6-dimethoxyphenyl)-4-(furan-2-yl)-1,2-oxazol-5-yl]ethanimine 4-(1-phenylcyclobutyl)-6-[7-(pyridine-3-carbonylamino)heptanoyl]quinoline-2-carboxylic acid 5-[[3,6-bis(trifluoromethyl)carbazol-9-yl]methyl]-3H-1,3,4-oxadiazole-2-thione 6-[2-fluoro-4-(methylamino)phenyl]-5,7-dihydroxy-9H-fluorene-1-carboxylic acid 7-(3-methyl-2,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-yl)-3-oxa-7,10-diazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,11-tetraene 2-methoxy-7,8,9,10-tetrahydrobenzo[f]quinoline [2-fluoro-3-[(4-methylphenyl)methoxy]phenyl]boronic acid 1-[2-(5,6-dihydronaphthalen-2-yl)ethyl]-3-methoxyazetidine;hydrochloride 2-[[(2S)-1-amino-3,3-dimethyl-1-oxobutan-2-yl]carbamoyloxy]-4-fluorobenzoic acid N-(1-amino-3-methylbutan-2-ylidene)-4-[[5-cyano-2-[2-ethoxy-4-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]anilino]pyrimidin-4-yl]amino]benzenecarboximidamide 1-(2,4-difluorophenyl)sulfonyl-N-ethylpyrrolidine-3-carboxamide (5Z)-2-cyclopentylimino-5-[(4-fluorophenyl)methylidene]imidazolidin-4-one 3-[1-(2-ethoxyethyl)benzimidazol-2-yl]butane-2,3-dione 3-[5,6-dimethyl-2-(methylamino)pyrimidin-4-yl]-1H-indole-6-carbonitrile 3,5-dibromo-1,2,4-triazine N-[(1R,2S)-3-cyclohexyliminospiro[1,4-dihydroquinoxaline-2,3'-piperidine]-1'-yl]pyrazine-2-carboxamide 2-[(5,6-diethylpyridazin-3-yl)amino]butanoic acid 2-(3,5-difluorophenyl)acetate;2-[1-(2-hydroxyethyl)pyrazol-4-yl]propanoic acid 2-[3-(4-chlorophenyl)phenyl]-1,3,5-triazine 1-cyclobutyl-N-[(3R)-5-methylsulfonyl-2,3-dihydro-1H-inden-4-yl]benzimidazole-5-carboxamide (2S,3R)-2-(1,5-dimethylpyrazol-4-yl)-N-[[2-ethylsulfanyl-6-fluoro-3-(trifluoromethyl)phenyl]methoxy]piperidin-3-amine N-[(1R,2S)-2-fluorocyclopropyl]formamide;8-fluoro-6-(5-fluoro-7-methoxy-1H-indol-4-yl)-1-methyl-3,4-dihydroquinolin-2-one N-[5,6-diethyl-1-(oxan-2-ylmethyl)imidazo[4,5-b]pyridin-2-yl]ethanesulfonamide [(3S,4R)-1-[2-amino-6-[(2-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)methyl]quinazolin-4-yl]-4-fluoropiperidin-3-yl]carbamic acid 6-bromo-2,3-dihydrochromen-4-one 2-(2,3-dihydro-1H-indene-5-carbonylamino)imidazo[1,2-b]pyridazine-6-carboxamide [4-(2,5-difluorophenyl)sulfonylphenyl]boronic acid 2-methyl-1H-indole;N'-(3-methylphenyl)naphthalene-1-carboximidamide 5-[4-(4,4-dimethylpiperidine-1-carbonyl)piperidin-1-yl]-2-(trifluoromethoxy)benzonitrile 2-(3-azidopropyl)-4,6-diphenylpyrimidine [4-(7,8,9,10-tetrahydrocycloocta[d]pyrimidin-4-yl)piperazin-1-yl]-[2-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-5-yl]methanone 3-bromo-5-fluoropyridine;2,2,2-trifluoroacetic acid 4-[(3,6-dichloroimidazo[1,2-a]pyridin-2-yl)methyl]benzenecarboximidate 3-[2,4-dichloro-5-(trifluoromethyl)phenyl]-2-oxopropanoic acid 5-[2-(azidomethyl)pyrrolidin-1-yl]quinoline 6-chloro-N-[5-[2-(4-fluorophenyl)ethyl]-1,3,4-thiadiazol-2-yl]pyridine-3-carboxamide 4-(6-propan-2-yl-1,3-benzothiazol-2-yl)-5H-1,3-oxazole 2,4-dimethylpentane;ethanamine;1-[(Z)-3-ethoxy-3-oxoprop-1-enyl]-4-[6-[4-[2-(oxolan-3-yl)ethynyl]phenyl]hexyl]pyrrole-2,5-dione 1-(4-hydroxyphenyl)sulfinylethylidenephosphanium 3-[2,6-dichloro-4-(trifluoromethyl)phenoxy]azetidine 2-azido-1,4-dibromoanthracene 3-[2,4-bis(ethoxycarbonyl)phenyl]propanoic acid 3-[3,4-dimethoxy-5-(2H-pyran-6-yl)phenyl]-2-oxopropanoic acid 5-[4-(3,4-dimethoxyphenyl)phenyl]sulfanyl-2H-triazole-4-carboxylic acid 3-[(E)-2-fluoro-3-propan-2-yloxybut-1-enyl]imino-N'-hydroxypyridazine-4-carboximidamide 4-[(4R,5S)-3,7-dimethyl-6,8-dihydro-2H-pyrano[2,3-e]indole-5-carbonyl]-N'-(1,3-thiazol-4-ylsulfonyl)benzenecarboximidamide (Z)-1,2-dipyridin-2-ylethenethiol;ruthenium(2+);tetraphenylboranuide 1-[4-[2,4-dimethyl-5-(4-methylidenecyclohexa-1,5-dien-1-yl)pent-4-ynoxy]phenyl]piperidine (2Z,5E)-3-[(2Z)-2-[1-(4-chlorophenyl)ethenylimino]-4-oxo-6,7-dihydro-5H-thieno[3,2-c]pyridin-5-yl]-2-ethylidene-N,4-bis[(4-fluorophenyl)methyl]hepta-2,5-dienamide N-[5-cyclopropyl-4-[(2R,3S)-2-methyl-1-propanoylpiperidin-3-yl]oxypyridin-2-yl]formamide 2-[3-(trifluoromethyl)phenyl]piperidine 3-[(Z)-2,5-dimethylhept-4-enyl]-2-methoxyphenol 6-chloro-4,5-dimethyl-2-[1-(3-oxopropyl)piperidin-4-ylidene]-1H-pyridine-3-carboxylate 2-[[4-[(5-tert-butyl-1H-pyrazole-3-carbonyl)amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]methyl]indole-1-carboxylic acid 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidin-2-ide;cyclopenta-1,3-diene;iron(3+);oxolane (2S)-N-benzyl-1,1,3,3-tetramethyl-5-(3-oxopyrazolidine-1-carbonyl)-2,4-dihydropyrrolo[2,3-b]pyrrole-6-carboxamide 2-methyl-6-(3-methylpyridin-4-yl)pyridine 5-methyl-2,3,7,10-tetrazatricyclo[6.4.1.04,13]trideca-1,4,6,8(13),9,11-hexaene;hydrochloride N-[4-(2,3-dihydro-1H-inden-5-yl)-4-ethoxybut-1-en-2-yl]hydroxylamine 2-(4,6-difluoro-1H-indole-3-carbonyl)pyrrolidine-2-carboxylate N-[3,5-difluoro-4-(trifluoromethylsulfanyl)phenyl]-2-formamido-1H-benzimidazole-4-carboxamide;methanol 3-[4-(1H-benzimidazol-2-ylmethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 4-cyclopentyloxy-N-[3-(1,2-oxazol-4-yl)phenyl]pyridine-2-carboxamide 4-(2-azidoethyl)-1-(4-chlorophenyl)pyrazole (4-cyclopropylpiperazin-1-yl)-[5-[6-fluoro-8-methoxy-7-(3,4,5-trifluorophenyl)quinolin-4-yl]pyridin-2-yl]methanone N-[(1R,2R)-6-ethylcyclohept-4-en-1-yl]-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide 1-methyl-2,6-dipyridin-3-yl-5H-pyrazolo[3,4-d]pyrimidin-4-one [(3S,4R)-4-[3-chloro-4-(5H-pyrrolo[2,1-a]isoindole-8-carbonylamino)benzoyl]-1-(4-methoxyphenyl)sulfonylpyrrolidine-3-carbonyl]azanium N-[(4R)-1-ethanimidoyl-6-methylidene-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-3-yl]-6-phenoxypyridine-2-carboxamide 2,5-ditert-butyl-3-(4-methoxyphenyl)thiophen-1-ium N-[1-(2,4-dimethoxyphenyl)ethyl]-2-hydroxy-2-[(2R)-3-oxo-5-sulfanylidene-1,2-dihydroimidazo[1,2-c]quinazolin-2-yl]acetamide 3-N,5-N,7-N,7-tetramethylspiro[cyclohepta-1,3,5-triene-6,9'-fluorene]-2,7-diimine 3-[[2,6-difluoro-4-[(1R)-1-[(2S,5S)-2,4,5-trimethylpiperazin-1-yl]butoxy]phenyl]iminomethyl]-N-methylidenebenzamide 3-(4-fluorophenyl)-5-(2-propan-2-yloxyphenyl)-1,2,4-oxadiazole 4-methyl-N-(3-methylbutoxy)benzamide 2-chloro-N-(3,3-diphenylpropyl)benzamide 1-benzyl-3,4-dimethoxy-5-phenylpyrrolidin-2-one 3-chloro-N-[1-(2,4-difluorophenyl)propan-2-yl]-4-hydroxybenzamide 2-[2-methyl-N-(1,3-thiazol-5-yl)anilino]decanoic acid (3S,4R)-4-(1H-imidazol-5-ylmethoxy)oxolan-3-ol 2-hydroxy-5,7-dimethylsulfanylnaphthalene-1,4-disulfonic acid 2-bromo-7,8-dimethoxyquinoline 1-[(3,5-dimethylphenyl)methylamino]-3-(2-phenoxyethoxy)propan-2-ol;hydrochloride N-[2-(cyclopropanecarbonylamino)ethyl]-5-methyl-1H-pyrazole-3-carboxamide 1-[(4-oxo-3H-quinazolin-2-yl)methyl]pyrrolidine-2-carboxylic acid (2R,3S)-2,3-dimethyl-1-phenylmethoxypentan-2-ol 3-[(4R)-1,2,4-trimethylpyrrolidine-2-carbonyl]-1H-quinolin-2-one 2-[3-[(4-chlorophenoxy)methyl]phenyl]-1,1,1-trifluoropentane-2,4-diol 3,5-dichloro-2-(4-fluorophenoxy)benzaldehyde 3-[2-(4-azidophenyl)ethenyl]-5,6-dimethoxypyridazine N-[2,6-difluoro-4-(methylamino)phenyl]sulfanyl-3-[4-(trifluoromethoxy)phenoxy]aniline 3-[4-(1-azidocyclopropyl)phenyl]-5-[2-(2,6-dimethylmorpholin-4-yl)ethoxy]benzoic acid 1-(4-methylphenyl)sulfonyl-3-[5-(trifluoromethoxy)pyridin-2-yl]urea 2-[(6,7-dimethyl-2H-chromene-3-carbonyl)amino]-5-(2-ethoxyethoxy)-1H-indole-4-carboxylic acid [1-(3,4-difluorophenyl)cyclopentyl]methanol 3-[2,6-dichloro-4-(methylsulfinylmethoxy)phenyl]-5-ethyl-1H-pyrazole 2-methoxy-6-(4-propan-2-ylphenoxy)phenol 2-[2-[4-[5-(acetamidomethyl)pyridine-3-carbonyl]-1,3-thiazol-2-yl]pyrrolidine-1-carbonyl]-6-azaspiro[2.5]octane-6-carboxylic acid 7-[[4,4-difluoro-1-[2-(5-methyl-1H-imidazol-4-yl)acetyl]piperidin-3-yl]oxymethyl]-5-phenyl-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one (2R,3S)-1-[1-(benzenesulfonyl)piperidin-4-yl]-N-[cyclopropylidene-[5-(methoxymethyl)-4H-pyridin-2-yl]methyl]-2-methylpyrrolidine-3-carboxamide 2-(N-methylsulfonylanilino)decanoic acid 4-[2,3-bis(4-fluorophenyl)quinoxalin-6-yl]aniline 4-hydroxy-2,6-dioxo-1H-pyrimidine-5-carboxamide N-[2-(5-acetylcycloocten-1-yl)ethyl]-4-chlorobenzenesulfonamide 3-[4-azido-2-(1H-indol-5-yl)butan-2-yl]-1,7-naphthyridine 2-[(1R,5S)-3-benzyl-8-fluoro-6-oxo-5H-naphthalen-2-yl]acetic acid 4-hydroxy-5,6-diphenylcyclohexa-2,4-dien-1-one 4-(1H-benzimidazol-2-yl)-5,6-dimethoxypyrimidine N-[2-(6-methylpyridin-3-yl)ethyl]-1H-benzimidazole-4-carboxamide N'-[6-chloro-2-fluoro-3-(1H-pyrazol-5-yl)phenyl]-4-(pyrimidin-2-ylmethylamino)-1,2,5-oxadiazole-3-carboximidamide 3,7-dimethyl-2-[(E)-pent-2-enoxy]naphthalene 1-[[4-[(5,6-dichlorobenzimidazol-1-yl)methyl]phenyl]methyl]pyrrolidine-2,5-dione N-cyclohexyl-1-[(4S)-3,4-dihydro-2H-chromen-4-yl]piperidine-4-carboxamide 3-(3-fluorocyclohepta-1,4,6-trien-1-yl)-N-[2-[4-(5-methoxy-4-oxopentanoyl)piperazin-1-yl]pyridin-3-yl]propanamide 3-[2-[6-[(1,4-difluorocyclohexa-2,4-dien-1-yl)methoxy]-5-fluoropyridin-2-yl]ethynyl]cyclobutan-1-amine (2R,3S)-N-[6-fluoro-1-[(4-methoxyphenyl)methyl]indol-3-yl]-3-methyl-5-oxomorpholine-2-carboxamide 2-cyclopropyl-7-methoxy-6-(6-pyrrolidin-1-ylpyridine-3-carbonyl)-5H-pyrrolo[3,4-b]pyridin-5-ol 4-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazole-4-carbonyl]-1,1-dioxo-2H-1,4-benzothiazin-3-one 1-(4-methylphenyl)sulfonyl-N'-pyrimidin-2-ylethane-1,2-diamine 2-[[4-bromo-3,5-diethoxy-2-(3-methylbutanoylamino)phenyl]carbamothioylamino]acetic acid 7-chloro-2-ethyl-N-[3-methoxy-4-(oxan-2-yloxy)phenyl]imidazo[1,2-c]pyrimidin-5-amine (3S)-4-[7-[4-(aminomethyl)-1,3-thiazol-2-yl]imidazo[1,2-a]pyridin-3-yl]-3-methoxypiperidine-1-carboxylic acid 4-(cyclobutylmethoxy)-N-[5,6-difluoro-1-methyl-3-(2-oxopyrrolidin-1-yl)indazol-5-yl]pyridine-2-carboxamide 5-[(4-chlorobenzoyl)amino]benzene-1,3-dicarboxylic acid 5-[(1E,3E)-4-aminobuta-1,3-dienyl]-2,4-bis(prop-1-ynyl)-6-sulfanylidenepyran-3-carbonitrile N-azido-2-(oxolan-3-ylamino)pyridine-4-carboxamide 2-[5-(1,3-benzothiazol-2-yl)pyridin-2-yl]oxy-N,N'-dimethylethanimidamide N-butyl-2-[4-[2-(diethylamino)ethoxy]phenyl]-5,6-dimethoxyquinoline-4-carboxamide 2-methyl-N-[(3S,4R)-1-pyridin-2-ylsulfonylpiperidin-3-yl]-1H-pyrrole-3-carboxamide 5-chloro-N-[4-ethoxy-3-(2-oxo-1,3-oxazolidine-3-carbonyl)phenyl]-2-methylbenzamide [2,6-difluoro-4-(6-phenylpyridin-3-yl)phenyl]boronic acid (2S,3R)-N-[4-(4-fluorophenyl)phenyl]-1-azabicyclo[2.2.2]octan-3-amine 2-(dichloromethyl)-3,5-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol 5-[(4-methylphenyl)sulfonylamino]naphthalene-2-sulfonic acid 1-[5-fluoro-6-(2,4,5-trifluorophenyl)pyridin-3-yl]-N-methoxyethanimine 6-(3-fluorophenyl)imidazo[1,2-a]pyridine N-methyl-1-[3-[6-(2-pyridin-4-ylpropanoylamino)pyridazin-3-yl]phenyl]cyclopentane-1-carboxamide 2-[(5S,10bR)-7-methoxy-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-methoxyphenol (4E)-2-cyclopentyl-3-(4,7-dimethoxy-1H-benzimidazole-5-carbonyl)-4-[hydroxy-(1-phenyltriazol-4-yl)methylidene]cyclohexa-1,5-diene-1-carboxylic acid N-[(1S,3R)-3-aminocyclopentyl]-2-(4-benzamidophenoxy)propanamide;hydrochloride 4-[1-(2,3,6,7-tetramethyl-2H-quinoxalin-1-yl)cyclopropyl]oxybenzonitrile 4-[4-fluoro-3-(7-hydroxyquinazolin-2-yl)phenyl]morpholine-2-carboxylic acid N-[(2S)-1-amino-3-methylbutan-2-yl]isoquinoline-3-carboxamide;hydrochloride 1-[7-(2,3-dihydro-1H-pyrrolo[1,2-a]indole-6-carbonyl)-9H-pyrido[4,3-b]indol-2-yl]-N',N'-dimethyloxamide N-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide N-[5-(cyclobutylcarbamoyl)-1,3,4-thiadiazol-2-yl]piperidine-3-carboxamide N-[2-amino-3,5-bis(methanesulfonamido)phenyl]acetamide 2-[4-(3,4-dihydro-1H-isoquinoline-2-carbonyl)phenoxy]benzoic acid N-(cyclohexylmethyl)-N',N'-dimethylethane-1,2-diamine;5-[7-(3-ethenoxyprop-1-ynyl)furo[3,2-c]pyridin-5-yl]-4-fluoropyrimidin-2-amine N-[4,5-dimethyl-2-(4-oxo-1-phenyl-6H-pyrazolo[3,4-d]pyrimidin-5-yl)pyrazol-3-yl]-3,4-difluorobenzamide 2-(3,4-dichlorophenyl)-N-[4-hydroxy-1-methyl-6-oxo-5-[(E)-2-pyridin-4-ylethenyl]pyridin-3-yl]acetamide 2-bromo-4,5-dimethoxy-N-phenylbenzamide (Z)-2-amino-4-[3-fluoro-4-[3-[2-methyl-5-oxo-7-(trifluoromethyl)imidazo[1,2-a]pyrimidin-6-yl]propoxy]phenyl]but-2-enoic acid 7-[(1S,2R)-2-ethylcyclopropyl]oxy-4-fluorochromen-2-one N-[(3R,4S)-3-hydroxyoxan-4-yl]-2,5-dimethoxybenzamide;hydrochloride 1-(2,4-dichlorophenyl)-N-methylpyrazole-3-carboxamide (2R)-4,5-diamino-1-[3,3-dimethyl-6-(4-phenylcyclohexa-2,4-dien-1-yl)-2H-pyrrolo[2,3-b]pyridin-1-yl]-2,3-dihydro-1H-indene-2-carboxylic acid 5-(1,3-benzothiazol-6-ylsulfonyl)-N-[4-fluoro-2-(propanoylamino)phenyl]-4,6-dihydropyrrolo[3,4-c]pyrazole-2-carboxamide 6-(1,3-benzodioxol-5-ylmethylideneamino)-N-[2-(1H-indol-4-yloxy)ethyl]-N-[(2E,6Z)-octa-2,6-dien-3-yl]hexanamide 1-[2,6-dimethyl-4-(3-phenylpentanoyl)phenyl]ethenol 7-amino-2,4-dioxo-5-[2,3,5-trifluoro-6-hydroxy-4-(morpholine-4-carbonyl)phenyl]-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 4-amino-2-[6-(ethylaminomethyl)pyridin-3-yl]sulfanyl-1H-pyrimidin-6-one 2-amino-1,4-dibromoanthracene-9,10-dione (3R,4S)-4-[1-[5-chloro-7-[(2-fluorophenyl)methoxy]-2H-quinazolin-2-yl]piperidin-4-yl]-N,N-dimethylpyrrolidine-3-carboxamide 2-methyl-5,9-bis(4-nitrophenyl)sulfonylpyrrolo[3,2-b]carbazole-6,8-diol 5-(2,4-dihydroxyphenyl)-N-ethyl-4-[1-(pyridin-4-ylmethoxy)ethenyl]-1,3-thiazole-2-carboxamide 3-(2,6-dichlorophenyl)-7-[(4-methoxyphenyl)methylamino]-N-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5-carboxamide;ethane 2-[4-[(2-chloroacetyl)amino]phenyl]sulfanylpropanoic acid (2-methylcyclohexyl)benzene;N-[3-(1-propanoylpiperidin-4-yl)phenyl]formamide 5-N-[(4-aminophenyl)methyl]-1H-1,2,4-triazole-3,5-diamine 3-ethoxycarbonyl-4-[(1R,2S)-2-hydroxycyclohexyl]benzoate 1-(4-fluorophenyl)-N-[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]-5-(trifluoromethyl)pyrazole-4-carboxamide 2-[5-(diethoxyphosphorylmethylamino)-4,6-dioxo-1H-pyrimidin-3-ium-2-yl]acetic acid (4S)-5-[[(1R)-6-chloro-2,3-dihydro-1H-inden-1-yl]oxymethyl]-2,2-difluoro-4-phenylpentanenitrile 2-methoxy-5-(3,4,7-trihydroxy-9,9a-dihydro-6H-xanthen-1-yl)benzoic acid 1-[5-fluoro-2,6-dimethyl-3-[(2S)-2-[[5-(trifluoromethyl)pyridine-2-carbonyl]amino]butoxy]phenyl]cyclopropane-1-carboxylic acid 4-chloro-N-[(2S)-1-oxo-3-phenylbutan-2-yl]benzenesulfonamide 1-[6-cyclobutylidene-2,3-dimethoxy-5-(4-phenylpiperidine-1-carbonyl)pyridin-1-yl]ethanone 4-methoxycarbonyl-2-(phenylmethoxycarbonylamino)benzoic acid N-[(2,6-dichlorophenyl)methyl]-2-[2-ethoxy-4-[(Z)-1,3,3-trifluoroprop-1-enyl]phenoxy]acetamide 1-[6,7-bis(ethenyl)-9H-fluoren-2-yl]propan-2-one 2-(3,4-dimethoxyphenyl)-7-[2-(4-methylpiperidin-1-yl)pyrimidine-5-carbonyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide;2,2,2-trifluoroacetic acid 7-(1,3-benzothiazol-6-ylsulfonylamino)-N,4-dimethylisoquinoline-3-carboxamide 3-azido-5,7-dichloroquinoxaline 5-fluoro-3,4-dihydroisoquinoline;N-[2-(1H-indol-3-yl)ethyl]-6-piperidin-4-ylidenecyclohexa-2,4-dien-1-imine 2-ethyl-5-[(Z,4E)-4-methoxyiminooct-1-en-3-yl]-N-phenylbenzamide 1-[3,5-bis(trifluoromethyl)phenyl]-4-pyridin-2-ylbutane-1,4-dione 2,6-dichloro-3-methylsulfonyl-4-phenylbenzoic acid 4-(3,5-dichlorophenyl)sulfanyl-1H-pyrrole 2-[4-(1,3-benzodioxol-5-yl)-5-phenylpyrazol-1-yl]-N-[(Z)-1H-indol-3-ylmethylideneamino]acetamide 5-(2-hydroxyethyl)-N,N'-bis[[2-methoxy-4-[(1E,3Z,7E)-3-methylidenecycloocta-1,7-dien-1-yl]phenyl]methyl]heptanediamide (NZ)-N-[amino-[2,3-dichloro-4-methoxy-6-[(2R)-2-[(4-nitrophenyl)methyl]piperazine-1-carbonyl]phenyl]methylidene]-3-bromobenzenesulfonamide N-[(5S,7R)-3-chloro-5-(4-fluorophenyl)-10-iodo-11-oxa-2,4,6,7,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,10,12-tetraen-12-yl]benzamide 1-[2-(3-amino-4-cyclopropylpyrrolidin-1-yl)-2-oxoethyl]-N,N-dimethyl-6-[6-(trifluoromethyl)pyridin-3-yl]indazole-5-carboxamide [1-(2,4-dichlorophenyl)-3-phenylpropyl]azanium 5-chloro-2-(1,4-dioxan-2-yl)pyrimidine 4-[(5E)-5-(7H-cyclohepta[b]pyridin-9-ylidenemethyl)-2,3,4,8,9,10,11-hexahydro-1-benzoxocin-6-yl]benzoic acid 3-methyl-N-[4-(5-oxo-1H-pyrazole-3-carbonyl)phenyl]benzamide 2-[2-(benzenesulfonyl)ethyl]-7-pyridin-3-yl-5,6,8,9-tetrahydropyrido[2,3-d]azepine;2,2,2-trifluoroacetic acid 2-(2-phenylethyl)-5-[1-propylsulfanyl-4-(trifluoromethyl)benzimidazol-2-yl]oxypyrazine 5-methoxycarbonylbenzotriazole-1,3-dicarboxylate (7R)-5-chloro-N-[4-cyano-2,6-di(propan-2-yl)phenyl]-7-hydroxy-6,8-dihydroimidazo[1,2-a]pyrimidine-2-carboxamide 1-[(2S,5R)-4-hydroxy-5-(hydroxymethyl)-3-methylideneoxolan-2-yl]pyrimidine-2,4-dione (6Z)-2,4-diamino-5-[[4-[(4-aminophenyl)diazenyl]-3-hydroxynaphthalen-1-yl]diazenyl]-6-methylbenzenesulfonic acid 1-butyl-2,5-diphenyl-3H-pyrazole 4-[(E)-2-cyclobutylprop-1-enyl]-2,6-dimethoxyphenol 4-methoxy-3-[(2Z)-4-(2-methylphenyl)sulfonylpenta-2,4-dienoyl]quinoline-8-carboxamide 1-azido-3,4-dimethoxy-2-nitro-5-(trifluoromethyl)benzene 2-[4-[(5-phenylfuro[3,2-b]pyridin-7-yl)amino]phenoxy]acetonitrile 1-(6-ethoxy-5-nitropyridin-2-yl)pyrrolidine-2,4-dione 3-azido-5,7-dimethylsulfonylimidazo[1,2-a]pyridine 4-(4-chlorophenyl)-2,5-dimethyl-3,4,6,7-tetrahydropyrrolo[3,4-c]pyridine 3-methoxycarbonylquinoline-2,4-dicarboxylic acid 1-[7-methoxy-8-(3-morpholin-4-ylpropyl)imidazo[1,5-c]quinazolin-3-yl]ethanamine;hydrochloride (7E)-2,4-dimethylcycloocta-1,3,7-triene;1-[3-[6-(dimethylamino)pyridin-2-yl]azetidine-1-carbonyl]-4H-pyridin-4-id-3-one;uranium(2+) 5-[(4,7-dioxo-1,3-benzothiazol-2-yl)methoxycarbonyl]pyridine-2-carboxylic acid 5-[2,3-dihydroxypropyl(hexadecanoyl)amino]-2-hydroxybenzoic acid (2R)-N-[(Z)-1H-indol-3-ylmethylideneamino]-2-(3,4,5-trimethoxyphenyl)propanamide 3,4-bis(3-ethylsulfanylphenyl)pyrrole-2,5-dione 1-[[6,7-dichloro-4-(cyclopropanecarbonyl)-2H-isoquinolin-3-ylidene]methyl]-5-hydroxyindole-2,3-dione 1-[5-fluoro-6-(2,3,4,5,6-pentadeuteriophenyl)pyridine-3-carbonyl]piperidine-3-carboxamide N'-[(Z)-2-cyano-3-oxobut-1-enyl]benzenecarboximidamide 2-(1,3-benzothiazol-2-ylsulfanyl)-N'-hydroxyethanimidamide 2-[3-(pyridine-4-carbonyl)phenyl]pyridine-4-carboxamide N-[(E)-2,3-dimethylbut-1-enyl]-5-fluoro-4-[3-[7-(3-hydroxypropyl)imidazo[1,2-a]pyridin-3-yl]phenyl]pyrimidin-2-amine 4-[2,6-di(propan-2-yl)phenyl]-1H-imidazole 2-amino-N'-[3-[4-(3-aminopropyl)-5,6,7,8-tetrahydropyrido[3,2-d]pyrimidine-2-carbonyl]phenyl]ethanimidamide 5-[[2,4-dimethoxy-6-(1H-pyrrol-3-yl)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one 1-(2-azidooxy-5-nitrophenyl)sulfonylpiperidine 3-amino-4-cyclopentyloxybenzenecarboximidamide 5-[4-amino-3-(methyliminomethyl)phenyl]-6-(2,6-difluoro-4-hydroxyphenyl)imidazo[1,2-a]pyrazine-8-carbonitrile 2,3-bis[(1S)-3-ethylcyclopent-2-en-1-yl]-4-phenylquinoxaline ethane;N-(4-fluorophenyl)-1,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-2(6),4,7,9,12-pentaen-10-imine 4-(2,3-dihydro-1H-inden-5-ylmethoxy)pyrimidine N-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]-4-methoxybenzamide 2-[[1,3-benzothiazol-5-yl(2H-tetrazol-5-yl)methoxy]-methylphosphoryl]acetic acid 1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)hexan-1-one 1-[2,4-di(cyclobutyloxy)phenyl]ethanol 2-[4-chloro-3-(trifluoromethyl)phenyl]sulfanyl-N'-hydroxypyrimidine-4-carboximidamide (2-ethyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl)-(1H-pyrrol-2-yl)methanone;hydrochloride 3-[4-(1,3-dioxolan-2-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 3-(3,4-dihydro-2H-quinolin-1-yl)-N'-hydroxypyrazine-2-carboximidamide 4-(1-methoxycyclobutyl)-2H-benzotriazole 4-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-N-methyl-1-(oxan-2-yl)-3-phenylbut-2-en-1-imine 1-bromo-2,5-dimethyl-3-[(Z)-pent-3-enyl]benzene (Z)-3-[5,7-bis(3,4-dimethoxyphenyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl]prop-2-enenitrile N-[1-[4-(aminomethyl)phenyl]ethenyl]-3-(1H-imidazol-5-yl)cyclobutan-1-amine 2-chloro-N,3-dimethylaniline;3-ethoxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]benzaldehyde (Z)-3-amino-4,4,4-trifluoro-1-[3-methyl-4-[[2-(4-methylphenoxy)ethylamino]methyl]phenyl]but-2-en-1-one 1-[7-methyl-5-(2-methylbutan-2-yl)-1H-inden-2-yl]naphthalene 1-(6,7-dimethoxyisoquinolin-3-yl)ethanol 5-methoxy-2-[1-[(4R,5R)-4-phenyl-3,6-dihydro-2H-pyran-5-yl]azetidin-3-yl]-N,N-dipropylpyrimidin-4-amine (6R)-8-[2-(1,3-benzothiazol-5-yl)ethyl]-1-propanoyl-3-sulfanylidene-6-undecyl-7H-purine-2,9-dione 3-[(Z)-[3,4,5-trihydroxy-2-(hydroxymethyl)phenyl]methylideneamino]-1,5,6,7-tetrahydroindol-2-one N-azido-2,3-dichloro-5-(1H-pyrazol-4-yl)aniline 2-[(5,6-difluoropyridine-3-carbonyl)amino]propanoic acid (Z)-2-[[2,6-dichloro-5-(3-methylbutoxy)pyridin-3-yl]amino]-N'-ethylpent-2-enimidamide N-[(1S,2R)-2-hydroxycycloheptyl]-4-pyridin-3-yloxybenzenesulfonamide 4-[(6S)-1,7-dimethyl-3-phenyl-5,6-dihydropyrazolo[4,3-c]pyridine-8-carbonyl]-6-methoxycyclohexa-2,4-diene-1-carbonitrile 6-azidosulfanyl-3-methoxy-2H-benzotriazole 2-[3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)anilino]acetamide 5-bromo-2,3-dihydro-1H-quinolin-4-one ethane;N-[(1-hydroxycyclopentyl)methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide N-[(4-azidooxy-3,5-dimethylphenyl)methylidene]hydroxylamine N-[(2,5-dimethylpyrazol-3-yl)methyl]-3,4,5-trifluoro-6-methoxypyridine-2-carboxamide 2-[4-(3,5-dimethyl-1H-pyrazol-4-yl)-5-propan-2-ylsulfanyl-1,3-thiazol-2-yl]isoindole-1,3-dione 4-[5,6-dimethyl-2-(propylamino)pyrimidine-4-carboximidoyl]-N-[4-(trifluoromethoxy)phenyl]pyridin-2-amine (4-aminopyrimidin-5-yl)-[4-[(6-methoxypyridin-2-yl)methyl]piperidin-1-yl]methanone 4-azido-2-chloro-3,5-dimethyl-6-pyridin-2-ylpyridine 2,5-dichloro-4-(4-methylsulfinylanilino)phenol (1S,2R)-N'-hydroxy-4,4-dimethyl-3-[(4-propan-2-ylphenyl)sulfamoyl]cyclohexane-1-carbohydrazide 1-(4-bromophenyl)sulfonyl-3-fluoroazetidine 1-[(2S)-4,4-difluoro-2-(5-methoxypyridin-3-yl)pyrrolidin-1-yl]-2-methoxyethanone N-[1-(3,5-dimethoxyphenyl)ethenyl]-N-prop-2-enylbutan-1-amine (2-ethoxy-6-hydroxyphenyl)-[4-[4-(trifluoromethyl)phenoxy]piperidin-1-yl]methanone (4-anilinophenyl)methylphosphonic acid 2-[4-(3,5-dibromopyridin-2-yl)oxyphenoxy]butanoic acid 2-[6-chloro-4-(2,3-dimethylquinoxaline-6-carbonyl)-1H-indol-5-yl]-N,N-dimethylbenzenesulfinamide 3-[2,4-dihydroxy-6-(N'-hydroxycarbamimidoyl)phenyl]propanoic acid 5-[5-(3,4,4a,9b-tetrahydrodibenzofuran-4-yl)pyridin-2-yl]indolo[2,3-b]carbazole 3-amino-5-(3,4,6-trimethylcyclohexa-1,3-dien-1-yl)benzoic acid 3-[(5R)-1,5-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4H-pyrazolo[1,5-a]quinazolin-5-one 4-amino-5-[(3E)-2-fluorohexa-1,3,5-trien-3-yl]-6-(8-methoxyimidazo[1,5-a]pyridin-6-yl)pyrrolo[1,2-b]pyridazine-3-carbonitrile N-[(2S)-1-amino-3,3-dimethylbutan-2-yl]benzamide;hydrochloride (Z)-4-[(3Z,5E)-5-chlorohepta-1,3,5-trien-2-yl]-N-ethoxy-3-ethynyl-1H-pyrrole-2-carboxamide (5Z)-2-(3,4-dimethylphenyl)imino-5-[[4-[(2-nitrophenyl)methoxy]naphthalen-1-yl]methylidene]-1,3-thiazolidin-4-one 3,6-ditert-butyl-9H-fluoren-2-amine 1-azidosulfonyl-3-benzylurea 3-cyclopropyl-2,5-difluoro-6-[3-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazol-1-yl]pyrimidin-4-one (3S)-4,5,6,7-tetrahydroxy-3,9-dimethoxyanthracene-2-sulfonate 7-chloro-5,6-dihydroquinoline-4-carboxylate 2-[[5-chloro-6-(trifluoromethoxy)-1,3-benzoxazol-2-yl]amino]pentanedioic acid 2-[4-amino-5-(pyrrolidine-1-carbonyl)pyrrolo[2,3-d]pyrimidin-7-yl]-N'-propanoylbenzohydrazide N-(3,4-dichlorophenyl)sulfanylpiperidine-1-carbothioamide 2-[4-(3-amino-1H-pyrazolo[4,3-b]pyridin-5-yl)phenoxy]acetic acid 2-[2-(aminomethyl)-3,4-dihydronaphthalen-1-yl]ethanamine 3-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]-5,7-dihydropyrrolo[3,4-b]pyridine-6-carboxamide N-(5-bromothiophen-2-yl)sulfonyl-1-(cyclopropanecarbonyl)azetidine-3-carboxamide N-[1,3-bis(4-chlorophenyl)pyrazol-4-yl]-2-(2-methylpyrrolidin-1-yl)acetamide 2-(4-chlorophenyl)imino-3,6,8-trimethyloctan-1-amine N-(1H-benzimidazol-2-ylmethoxy)-3,4-difluorobenzenesulfonamide 1-methyl-3,5-bis(phenylsulfanyl)benzene (2R)-2-[5-chloro-4-oxo-6-[(1E,3Z)-5-phenylmethoxypenta-1,3-dienyl]pyrimidin-1-yl]-2-methylbutanoic acid 2-[1,4-dimethyl-6-(4-methylphenyl)-3-methylidenepiperazin-2-ylidene]propanenitrile N-[3-(4-chloro-2-methylphenyl)-1,2,4-thiadiazol-5-yl]-6-oxo-1H-pyridine-3-carboxamide 3-[4-(benzylamino)phenyl]pyrrole-2,5-dione (E)-4,5-dimethyl-3,7,8,11-tetrahydro-2H-azecine;7,10-bis(ethenyl)-9,13-dimethylidenenaphtho[1,2-c]acridine 2,4-bis(1H-imidazol-5-yl)butanoic acid N-(1,2-dihydropyridin-4-yl)-7-ethoxythieno[3,2-d]pyrimidin-4-amine 7-ethyl-4,4-dimethyl-1H-quinoline-2,3-dione 3-[2-(4,5-dihydro-1H-imidazol-2-ylmethylamino)-9-oxa-1,3-diazatricyclo[6.4.1.04,13]trideca-2,4(13),5,7-tetraen-6-yl]phenol 2-[[7-[(3,4-dimethylphenyl)methyl]-1,1-dioxothiepan-5-ylidene]amino]-N,N',2-trimethylpropane-1,3-diamine 2-(4-benzylpiperazin-1-yl)-8,9-dimethoxy-5-methylidene-6H-chromeno[3,4-c]pyridine-9-carboxamide 3-azido-4-(1H-indol-2-yl)benzenethiol 2,6-dimethoxy-4-[3-(4-naphthalen-1-ylsulfonylpiperidin-1-yl)propyl]phenol N-[(3-fluorophenyl)methyl]-4-phenoxy-N-phenylaniline 5-bromo-2-methyl-4-propan-2-ylidenecyclohexa-1,3-diene;ethane 3-[4,6-bis(ethylamino)-1,3,5-triazin-2-yl]-2,5-dimethoxyphenol 1-[4-(4-hydroxypiperidine-1-carbonyl)phenyl]-N,2-dimethylindole-5-carboxamide 5-[4-(azidomethyl)piperazin-1-yl]quinoline [4-(2-chlorophenyl)sulfonylpiperazin-1-yl]-[6,7-dimethoxy-2-[4-(trifluoromethyl)phenyl]quinolin-3-yl]methanone 1,3-dicyclopropyl-N-methyl-N-[(2-oxo-3H-1-benzofuran-5-yl)sulfonyl]pyrazole-4-carboxamide 7-[[2-(1,3-thiazol-5-yl)pyridin-4-yl]methoxy]chromen-2-one 4-[(3E)-5-aminopenta-1,3-dien-3-yl]-2-bromo-6-ethoxypyridine-3-carbonitrile 3-[4-(azidomethyl)phenyl]-5,6-dichloro-1H-benzimidazol-2-one 2-[4-methoxy-3,5-bis(phenylsulfanyl)cyclohexa-1,3-dien-1-yl]sulfanylacetic acid N-[1-(4-fluorophenyl)ethyl]-5-[3-hydroxy-2-oxo-6-(trifluoromethoxy)pyridin-1-yl]-2-methylidenepentanamide 4-methoxy-6,11-dihydro-5H-benzo[b][1]benzazepine 5-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-2,4-diphenyl-1H-pyrimidin-6-one 6-[(2E)-2-ethenylpenta-2,4-dienoxy]-3H-quinazolin-4-one 3-[2,3,4-tris(oxiran-2-ylmethoxy)phenyl]propanoic acid 4-azidooxy-6,8-dibromoquinazoline 3-fluoro-4-hydroxy-N-[(1R,2S)-2-phenylcyclopropyl]benzenesulfonamide 1,1-bis(4-fluorophenyl)-N-[(E)-prop-1-enyl]methanimine [2-(4-benzylpiperazin-1-yl)pyrimidin-5-yl]-[2-(5-methoxypyrazin-2-yl)pyrrolidin-1-yl]methanone 7-[(1S,2S)-2-(5,6-dichloroindol-1-yl)cyclohexyl]heptanoic acid N-ethyl-N',N'-dimethyl-3-(2,4,6-trifluorophenyl)benzenecarboximidamide 5-(2,4-difluorophenyl)-6-ethylsulfanylpyrazine-2-carboxylic acid ethane;1-[(3Z,5E)-4-methylhepta-1,3,5-trien-2-yl]-4-phenylbenzene 2,6-dimethyl-4-[[(1R)-1-naphthalen-1-ylethyl]amino]sulfanylaniline;2,6-dimethyl-4-piperazin-1-ylquinazoline 2-[(3S)-1-(2,5-dimethylthiophene-3-carbonyl)piperidin-3-yl]-6-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-tert-butyl-1-ethenyldibenzothiophene 2-[4-azido-3-fluoro-5-(trifluoromethyl)phenyl]-1,4-dichlorobenzene [1-[4-amino-3-chloro-5-(trifluoromethyl)phenyl]piperidin-4-yl]azanide 2-(4-cyclohexylphenyl)-5-methoxypyrimidine 2-[2-amino-4-(methylamino)pyrimidin-5-yl]-N-(1,3-benzoxazol-2-yl)acetamide N-ethenyl-2-[4-(2,5,7,9-tetrazatricyclo[6.3.1.04,12]dodeca-1(11),3,8(12),10-tetraen-6-ylidene)piperidin-1-yl]acetamide N-[1-(3-methoxyphenyl)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide (2R)-2-[3-[[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino]cyclobutyl]piperidine-1-carboxylic acid 1-[2-(5,8-dimethylnaphthalen-1-yl)ethynyl]cyclohexan-1-ol 2-(4-chlorophenyl)-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one 3-amino-N-[1-(2,4-difluorophenyl)ethyl]quinoline-7-carboxamide 4-amino-6-[(3,5-ditert-butyl-2-hydroxyphenyl)methylidene]-1-oxothiazinan-5-one N-[1-[3,5-bis(trifluoromethyl)phenyl]ethylideneamino]-4,5-dihydro-1H-imidazol-2-amine N-azido-6-methoxynaphthalene-1-carboxamide 2-amino-N'-[3,5-bis(trifluoromethyl)phenyl]-N-hydrazinylidenepropanimidamide 2-(6-bromopyridazin-3-yl)pyrrolidine-1,3-dione (2S)-2,6-diamino-4-[4-[(3,5-dioxopentanoylamino)methyl]phenyl]hexanoic acid 1-amino-1'-(2,2-diphenylacetyl)spiro[4H-isoquinoline-3,3'-azetidine]-2-one 2-(1-azidobutyl)-5-cyclopropylpyrimidine 6-fluoro-7-[1-methyl-3-(oxan-4-yl)pyrazol-4-yl]quinoline 1-N,1-N'-bis(2,4,6-trimethylphenyl)ethanedihydrazide [2-[2,4-difluoro-5-[[6-[6-(trifluoromethyl)pyridin-3-yl]pyrimidine-4-carbonyl]amino]phenyl]phenyl]sulfonylazanium 6-[2,3-dihydroxypropyl(pyridin-3-yl)amino]-4-hydroxynaphthalene-2-sulfonic acid 1-[6-(3,5-dimethylpyrazol-1-yl)pyridin-2-yl]piperazine 3-[(E)-2-hydroxyethenyl]-N-[2-(4-methoxyphenyl)ethyl]thiophene-2-carboxamide 3-(difluoromethoxy)-4-[4-[2-(3,5-difluorophenyl)ethynyl]cyclohexyl]benzaldehyde 1-[3,4-di(propan-2-yloxy)phenyl]sulfonyl-N-hydroxypiperidine-3-carboxamide 1-[4-chloro-3-(2,2-dimethylpropoxy)phenyl]ethanone;2-ethynyl-5-nitrofuran 5-(4-aminophenyl)-2-[2-(4-chloro-3,5-difluorophenyl)ethynyl]benzonitrile 1-[2-[1-(4,6-diphenyl-1,3,5-triazin-2-yl)indol-3-yl]quinoline-8-carbonyl]pyrrolidine-2-carboxylic acid 5-methyl-1,2-diphenylbenzimidazole (5R)-3-(3,4-dimethoxyphenyl)-N-methyl-6-oxo-2-piperidin-1-yl-1,2,4,5-tetrazine-5-carboxamide 2,3-dichloro-N-[4-chloro-5-[6-(ethylamino)-1H-benzimidazol-2-yl]-2-methoxyphenyl]benzamide 5-ethoxy-N'-[3-(2-fluoro-4-iodoanilino)cyclobutyl]pyridine-2-carbohydrazide 2-[3,5-bis(trifluoromethyl)phenyl]-4-[1-(4-methoxyphenyl)propan-2-ylideneamino]pentanenitrile 2-(4-azidophenyl)sulfanylpyrimidine N-(3-nitrophenyl)-N-octylpyridin-2-amine N-[2-(4-nitrophenyl)ethyl]-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide N-(2,4,6-trichlorophenyl)sulfonylcarbamate N-(1,3-benzothiazol-2-ylmethylideneamino)decanamide (E)-3-amino-2-ethenyl-N'-[1-oxo-4-phenyl-1-[[4-(trifluoromethoxy)phenyl]methoxy]butan-2-yl]-N-(1,3-thiazol-5-ylmethyl)hex-2-enediamide (1R,2S)-2-N-[5-chloro-4-(cyclohexylamino)pyrimidin-2-yl]cyclopentane-1,2-diamine 2-(4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridine-2-carbonyl)benzonitrile 6-[4,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-3-yl]-3H-pyrrolo[3,4-b]pyridin-7-one 6-[(2S,3R)-2-benzylpiperidin-3-yl]-1H-benzimidazole [4-(aminomethyl)-2,6-dichlorophenyl]carbamic acid [6-(4,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,9,11-pentaen-3-yl)pyridin-3-yl]methanol N-[(3S,7S,8aS)-3-phenyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-6-tert-butylpyridazine-3-carboxamide N-(2-hydroxyethyl)-4,5-dimethoxy-2-nitrobenzamide N-(2-aminophenyl)sulfanyl-3-chlorobenzenecarboximidate 1-[3-(2,6-dimethylphenyl)sulfonyl-5-methylphenyl]ethanone N-[(4S,5R)-1-cyclohexyl-3-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-5-yl]-2-phenoxyacetamide (2S,3R)-N-[(4-tert-butylphenyl)methyl]-2-fluoro-1-methylpiperidine-3-carboxamide 5-[2-(azidomethyl)phenyl]-1,3-dihydroindol-2-one N-benzyl-1-methoxy-9,10-dioxoanthracene-2-carboxamide 1-(2,6-dichlorophenyl)-3-[2-fluoro-4-[5-oxo-1-(trideuteriomethyl)pyrrolidin-3-yl]oxyphenyl]urea N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]-2-ethoxyacetamide 5-azidooxy-2-(4,5-dihydroimidazol-1-yl)aniline 1-(6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl)ethanone 2-tert-butyl-6-[(2,4,5-trimethoxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (2R,3S)-N-[4-(1-cyanocyclopropyl)phenyl]-2-(3,5-difluorophenyl)pyrrolidine-3-carboxamide 2,4-bis(3-phenylmethoxyphenyl)pentan-3-one (2E)-1-(3,4-dihydroxyphenyl)-2-[(E)-[7-(trifluoromethyl)quinolin-4-yl]methylidenehydrazinylidene]propan-1-one 3-[5-chloro-4-(difluoromethyl)-1,2-oxazol-3-yl]-1-[(1S,2R)-2-[(1R)-2-methoxycyclobutyl]cyclopropyl]-6,7,8,9-tetrahydro-5H-cyclohepta[d]pyridazine-8-carboxamide 2-(2,3-dimethoxyphenyl)-3-hydroxycyclohex-2-en-1-one N-[2-(1H-benzimidazol-4-yl)ethyl]formamide;ethane 1-[4-[4-(3,5-difluoropyridin-2-yl)piperazine-1-carbonyl]phenyl]pyrrolidine-2-carboxamide 3-[(4-chlorophenyl)-[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-1H-indol-2-one [3-chloro-2,4-dihydroxy-5-(trifluoromethyl)phenyl]-[(3R)-3-[(4-fluorophenoxy)amino]pyrrolidin-1-yl]methanone 5-chloro-3,4-dihydroquinoline-2,8-dione 2-[(4-amino-2-propylimidazo[5,1-f][1,2,4]triazin-7-yl)methoxy]ethanol;hydrochloride N-[4-(3-benzyl-5-but-2-ynoxyindole-1-carbonyl)phenyl]-N',N'-dimethylpropanediamide 1-chloro-6,8a-dimethyl-2-propylsulfanyl-4aH-quinazoline;ethane (3S)-5,6-difluoro-2-hexyl-2,3-dihydrothiochromen-4-one N-[2,4,6-trimethyl-3-[(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl]phenyl]-2-thiophen-2-ylacetamide N-cyclopropyl-3,4-dihydroxybenzenesulfonamide;hydrochloride 5-(2-chloropyridin-4-yl)oxy-1,3-dimethylpyrazole-4-carbonitrile 6-[4-[(2,3,5-trifluorophenyl)methyl]piperazin-1-yl]-2H-quinoline 2-[2-aminoethyl(methoxy)phosphoryl]oxyaniline 2-(6-bromoimidazo[1,2-a]pyridin-3-yl)-4-N-cyclopentyl-5-methylpyrimidine-4,6-diamine 5-[2-(1-hydroxycyclobutyl)ethynyl]-3H-1,3,4-thiadiazol-2-one 1,2-dimethyl-N-[(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)methyl]indole-3-carboxamide N-[2,5-di(propan-2-yl)phenyl]ethanesulfonamide 5-[2-(3,4-difluoro-5-isothiocyanatophenyl)ethynyl]-1H-pyrazole 4-(9H-fluoren-1-yl)-2,3,6-trifluorobenzoic acid N-(2,6-dimethylphenyl)-2,4-dioxo-1H-pyrimidine-5-sulfonamide 2-[1-(2,6-dichlorocyclohexa-1,3-dien-1-yl)ethoxycarbonyl]benzoic acid 1-azidosulfanyl-2-(4-chlorophenyl)-3-methoxy-5-nitrobenzene (2R)-6,8-dibromo-N-[2-(cyclohexylamino)ethyl]-4H-1,2,3,5-tetrazin-2-amine N-[4-cyano-3-(trifluoromethyl)phenyl]-2-(5,6-didehydropyridine-2-carbonylamino)-1H-benzimidazole-4-carboxamide 1-(cyclohexen-1-yl)-2,3,6-trimethoxynaphthalene (Z)-3,5-dihydroxypent-3-en-2-one;ethane;1-methyl-7-[(4-pyridin-2-yl-1H-pyrazol-5-yl)amino]indole-2,3-dione 4-chloro-N-[(3R)-1-[6-chloro-2,5-difluoro-4-[2-methoxyethyl(propanoyl)amino]benzoyl]pyrrolidin-3-yl]-2-(trifluoromethyl)benzamide (2S)-1-[3-(2,4-dimethyl-5,6-dihydronaphthalene-1-carbonyl)-1,7-naphthyridin-8-yl]pyrrolidine-2-carboxamide 7-azidooxy-2,3-dihydrochromen-4-one 4-[[3-(2,4-dichlorophenyl)-4-pyrimidin-6-yl-1H-pyrrol-2-yl]methylidene]cyclohexa-2,5-dien-1-one 1-[(E)-[(4,6-dimethylpyrimidin-2-yl)hydrazinylidene]methyl]naphthalen-2-ol 5-[5-methyl-6-(1H-pyrrol-2-yl)pyridin-3-yl]-N-(thiophen-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 3-[4-[2-(4,6-dimethylpyridin-3-yl)ethynyl]phenyl]-1,3-oxazolidin-5-ol 5-[3,4-bis(trifluoromethyl)phenyl]-N-[2-chloro-5-(2-cyclopropylideneethoxy)phenyl]-N'-ethenyl-1H-pyrrole-2-carboximidamide 5-[3,4-dimethoxy-2-(pyridine-4-carbonylamino)phenyl]-1H-pyrrole-2-carboxylic acid (1S,3R)-3-[2-chloro-5-[(3Z,6E)-7-methoxyocta-3,6-dienyl]-4-(piperidine-1-carbonyl)phenyl]cyclopentane-1-carboxylic acid 3-[6-amino-8-oxo-7-(4-phenoxyphenyl)purin-9-yl]benzamide 3-(methylamino)-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-6-carboxylic acid 1-[4-(4-chlorophenoxy)phenyl]-3,4-dihydro-2H-isoquinoline N-(3,4-dichlorophenyl)sulfanyl-2-methylpropanamide 2-[2-[(1S)-1-methoxypropyl]pyridin-4-yl]-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine 4-[(5R)-8-chloro-2,3-dioxo-5H-pyrimido[5,4-c]isoquinolin-1-yl]piperidine-1-carboxylic acid 6-[(2,5-difluorophenyl)methyl]-N'-hydroxypyridine-3-carboximidamide 6-[3-(4-azidooxy-5-chloropyridin-2-yl)phenyl]sulfonyl-N,N-diethylhexan-1-amine (5R)-2-[3,4-bis(2-methoxyethylamino)phenyl]-8-oxa-2-azaspiro[4.5]decan-1-one 1,3-difluoro-5-methylbenzene;[5-(2-hydroxyethyl)oxolan-2-yl]methanol N-[[4-(1,3-benzothiazol-2-yl)cyclohexa-1,5-dien-1-yl]methyl]-6-chloropyrazine-2-carboxamide 2-[(3S)-1-benzylpiperidin-3-yl]-6-methoxy-5,7-dihydropyrrolo[3,4-d]pyrimidine;ethane 4-chloro-6-[2,3,5,6-tetrafluoro-4-(trifluoromethyl)phenyl]-2-sulfanylidene-5,6-dihydro-1H-pyrimidine-5-carbonitrile 2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)acetate (2R)-N-[4-(benzylcarbamoylsulfamoyl)phenyl]-3,3,3-trifluoro-2-hydroxypropanamide 3-azidooxy-2-propan-2-yloxybenzonitrile 3-[N'-[2-(1H-indol-6-yl)ethyl]carbamimidoyl]propanamide 3-(1,4-dioxan-2-ylmethoxy)-5-fluorobenzoic acid 4-[3-(7,8-dihydronaphthalen-1-yl)phenyl]-2-(6-pyridin-4-yl-4-thiophen-3-ylcyclohexa-1,5-dien-1-yl)pyrimidine N-(1,5-dimethylpyrazol-4-yl)-5-(2-ethoxyphenyl)thiophen-3-amine 4-bromo-N,N-dimethyl-2-[(E)-1-phenylpropylideneamino]aniline 2-[2,6-dichloro-N-(1,3-thiazol-5-yl)anilino]decanoic acid 3-[1,3-diaminopropyl(methyl)amino]-6-phenylpyrazine-2-carboxamide [3-(dimethylsulfamoylamino)phenyl]azanide [4-(dimethylamino)phenyl]methanesulfinamide 1-azido-3,4,5-trimethoxy-9H-fluorene N-[3,5-dibromo-4-(6-chloro-2-methylsulfonylbenzimidazol-1-yl)phenyl]sulfanylaniline [(3S)-1-(5-chloro-4-methylpyridine-2-carbonyl)pyrrolidin-3-yl]-morpholin-4-ylmethanone N-[(4,5-dichloro-2-hydroxyphenyl)methylideneamino]-2-[4-fluoro-3-(trifluoromethyl)phenoxy]acetamide (2R)-4,4-difluoro-1-[3-[5-methyl-6-[5-methyl-2-(oxan-2-yl)pyrazol-3-yl]pyridin-3-yl]propanoyl]pyrrolidine-2-carbonitrile N-methyl-4-[2-(1,2-oxazol-3-yl)ethenyl]aniline ethane;3-methyl-2-(4-propan-2-ylidenephenyl)sulfanyl-1H-pyrrole (2S,4R)-1-[[4-(dimethylamino)phenyl]methoxycarbonyl]-4-(4-fluoro-3-prop-1-ynylphenyl)pyrrolidine-2-carboxylic acid 5-[4-(azidomethyl)phenyl]-1-benzothiophen-2-amine 2-[[1-[3,5-bis(trifluoromethyl)phenyl]sulfonylpiperidine-4-carbonyl]amino]-6-hydroxyquinoline-4-carboxylic acid 3,6-dichloro-1H-pyrazolo[3,4-d]pyrimidine 2-fluoro-3,4-dimethoxybenzenesulfonamide 4-[(3aR,6aS)-2,3a-dimethyl-1-oxo-5-phenyl-3H-pyrrolo[3,4-c]pyrrol-4-yl]benzonitrile [1-amino-2-(1H-indol-3-yl)ethylidene]azanium 2-(4-bromo-2,3,5,6-tetrafluorophenyl)sulfanylacetamide (5S)-2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-N-(3-methylphenyl)-6-oxopiperidine-4-carboxamide [1-(4,5-dimethylthiophen-2-yl)cyclopropanecarbonyl]azanium 5-N-[3-(difluoromethoxy)phenyl]pyridine-2,4,5-triamine 1-[(2S,4R)-4-hydroxy-2-phenylpiperidin-1-yl]hexan-3-one N-[6-(difluoromethoxy)pyridin-2-yl]sulfonylformamide 6-tert-butyl-3-(3-ethenoxyphenyl)sulfonyloxy-2,4-dihydroxybenzoic acid 2,7-dimethyl-N-[5-[3-(4-thiophen-3-yl-1H-pyrrolo[2,3-b]pyridin-2-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-yl]nonanamide 4-[5-(3,3a,4,6,7,7a-hexahydro-1H-pyrano[3,4-c]pyrrole-2-carbonyl)pyridin-2-yl]piperazine-1-carboxylic acid N-[(2R,3S)-1-acetyl-5-(1-methylpyrazol-4-yl)-2-(oxan-4-yloxymethyl)pyrrolidin-3-yl]methanesulfonamide 1-[4-(3,5-dimethylpyrazin-2-yl)piperazin-1-yl]ethanone N-(3,4-difluorophenyl)formamide;2-[(5Z,6E)-1-methyl-5,6-bis(prop-2-enylidene)pyridin-3-yl]oxy-N-(1-pyrrolidin-1-ylethenyl)ethanimine 2-cyclopentyl-4,5-bis(ethenyl)-1H-imidazole 5-[3-[4-(cyclopropylmethoxy)phenyl]-6,7-dihydroindazole-1-carbonyl]pyrazine-2-carbonitrile 6-[4-(3-fluorophenyl)sulfonylphenyl]-7-methyl-1H-imidazo[4,5-b]pyridine N-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-ylsulfonyl)-2-methylpropanamide 1-[(3aR,7aS)-2,3a-dimethyl-3,4,6,7-tetrahydro-2H-pyrrolo[3,4-c]pyridin-5-yl]-2-(furan-3-yl)ethanone;2,2,2-trifluoroacetic acid 2-(3-phenoxypropoxy)ethylphosphonic acid (5Z)-5-[[3-[2,6-dichloro-4-(trifluoromethyl)phenyl]phenyl]methylidene]imidazolidine-2,4-dione N-[1-(5-azidopyridin-2-yl)piperidin-4-ylidene]methanesulfonamide N-(2,3-dihydroindol-1-ylsulfonyl)pyrazine-2-carboxamide 3-amino-6-(2,5-dimethoxyphenyl)-4-methylthieno[2,3-b]pyridine-2-carboxylate N-[[3,5-bis(trifluoromethyl)phenyl]methoxymethyl]pyrimidin-2-amine N-(2,2-dimethoxyethyl)-N-[3-(trifluoromethyl)phenyl]methanesulfonamide (3R,4S)-1-[5-chloro-6-ethyl-2-[(2R)-pentan-2-yl]pyrimidin-4-yl]-4-methoxypyrrolidine-3-carboxamide 3-[3-azidooxypropyl(phenyl)amino]propanal N-[2-(3,4-dimethoxyphenyl)ethyl]-5-iodopyrimidin-2-amine 6-[2-[3-(4-fluorophenyl)propyl-methylamino]ethoxy]-1H-indole-2,3-dione (4E)-5-methoxy-4-[2-methoxy-1-phenyl-1-(3,4,5-trimethoxyphenyl)ethyl]hepta-4,6-dienal 2-methyl-3,4-bis(3-nitrophenoxy)benzoic acid 1-[2,4-dimethyl-6-(2-nitro-5-phenylphenyl)cyclohexa-1,3-dien-1-yl]ethanone N-[4-(benzylamino)phenyl]benzenesulfonamide 1-phenylnon-3-enylhydrazine 4-[(4S)-3,8-diethyl-1-oxo-2-phenylisoquinoline-4-carbonyl]piperazin-2-one 3-[4-amino-2-(ethoxymethyl)pyrimidin-5-yl]-N,N-diethylpropanamide;ethane 4-[(8,9-dihydroxy-9H-fluoren-2-yl)methylidene]hexanoic acid N-[3-(4-oxospiro[3H-chromene-2,1'-cyclopentane]-6-yl)propyl]benzamide 2-[3,4-di(butanoyl)phenyl]acetamide 4-tert-butyl-2-(3,5-difluorophenyl)-1H-pyrimidin-6-one 6,7-dibromo-4-hydroxynaphthalene-2-carboxylic acid 2-chloro-3-[4-[2,6-di(propan-2-yl)phenyl]imino-1,1-dioxo-1,2,5-thiadiazol-3-ylidene]-4H-indol-7-ol 3-[2,2-dimethylpropoxy(hydroxy)phosphanyl]benzoic acid N-[3-(difluoromethyl)-1-pyridin-3-ylpyrazol-4-yl]-5-piperidin-1-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide 4-(7,8-dimethoxyquinolin-2-yl)phenol 2-[1-(4,6-diphenylpyrimidin-2-yl)propan-2-ylideneamino]ethanol 4-(2,6-dichlorophenyl)sulfanyl-3-ethoxypyridine N-(2,3-difluorophenyl)-4-methyl-6-oxopyran-2-carboxamide (5R)-N-ethyl-7,8-difluoro-2-hydroxy-9-oxo-4-oxa-1,15-diazatricyclo[8.6.0.03,8]hexadeca-3(8),6,10,12,14-pentaene-5-carboxamide 3-benzyl-N-diazoisoquinoline-7-sulfinamide 2-amino-N'-hydroxy-5,7-dimethylpyrazolo[1,5-a]pyridine-3-carboximidamide (4R)-2,3,4a,5,6,10b-hexahydro-1H-benzo[f]quinoline 2-amino-4-[3-(2,6-dimethylpyridin-4-yl)phenyl]-4H-pyran-3,5-dicarbonitrile N-benzyl-2,4-dichloro-N-[(3R)-1-methoxypentan-3-yl]pyrimidine-5-carboxamide N-[5-[[3,4-dioxo-2-[(1S)-1-phenylethyl]cyclobuten-1-yl]amino]pentyl]acetamide 2-(3,4,5-trifluorophenyl)-6-(1,3,4-oxadiazol-2-yl)benzonitrile 2-(4-aminopiperidin-1-yl)ethanol;5-[3,5-bis(trifluoromethyl)phenyl]-1-pentanoylpyrrole-3-carbonitrile 3-(2,4-dihydroxy-5-propanoylphenyl)-N-[[1-methyl-6-(pyrrolidine-1-carbonyl)-2,3-dihydroindol-7-yl]methyl]-4H-1,2,4-oxadiazol-5-one;ethane 1-[2-(6-methoxy-3,4-dihydro-2H-chromen-7-yl)phenyl]ethanone 7-(2-fluorophenyl)-2,4-dihydropyrrolo[1,2-a]pyrimidine N'-hydroxy-6-[2-(4-methylphenyl)pyrrolidin-1-yl]pyridine-3-carboximidamide N-[(3S,5R)-1-benzylpiperidin-3-yl]-6-oxo-4H-imidazo[2,1-c][1,4]benzothiazine-9-carboxamide 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-pyridin-2-ylamino]benzenesulfonic acid 4-N,4-N-dimethyl-6-(2-piperidin-1-ylethoxy)pyridine-3,4-diamine 6-(4,5-diphenyl-1,3-oxazol-2-yl)-3-phenyl-4H-chromen-7-ol 5-[3-methyl-4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole 4-(3,4-dimethylphenyl)-N,5-bis(furan-2-ylmethylideneamino)-1H-pyrazole-3-carboxamide 4-[3-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)anilino]phenol 2-[4-[1,3-benzodioxol-5-ylmethyl(ethyl)amino]piperidin-1-yl]quinoline-6-carbonitrile 5-[(4-chlorophenyl)methyl]-1,3-thiazolidine 1,5-dimethyl-3-phenylpyrazole-4-carbonitrile ethane;5-[2-(1H-pyrazol-4-yl)pyridin-4-yl]oxyisoquinoline 2-[2-[4-(aminomethyl)phenyl]ethynyl]-4,6-bis(1,1,1,3,3,3-hexafluoropropan-2-ylidene)cyclohexa-2,5-dien-1-one N-[1-(difluoromethyl)cyclobutyl]-2,4-diethylpyrimidine-5-carboxamide 2-(3,4-dihydroquinolin-8-yl)propan-1-amine (2S,3aS)-1,2,3a-trimethyl-5-phenyl-2H-indole [2-(methylamino)pyridin-3-yl]-pyrrolidin-1-ylmethanone 4-(2,3,5,6-tetrafluorophenyl)benzoic acid (1R,2R)-1-(4-azidophenyl)-N-(isoquinolin-5-ylmethyl)butan-2-amine 3-[[(1R,2S)-4,5-dihydroxy-7-methyl-1-phenyloctan-2-yl]amino]cyclobutan-1-one 6-cyclopropyl-N,3-diethyl-2-(methylamino)-5-nitrobenzamide [(2S)-2-[1-carboxypropan-2-yl-(2-methoxyacetyl)amino]-3-phenylpropylidene]azanium 3-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrazine 1-[2,3-bis(ethenyl)cyclopentyl]-2-methoxybenzene 4-chloro-N-[2,3-difluoro-5-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)phenyl]benzenesulfonamide 4-[(1Z)-3-methylpenta-1,3-dienyl]benzenesulfinic acid 4-[3-(6-cyanopyrazin-2-yl)phenyl]-N,1-dimethylpyrazole-3-carboxamide 1-amino-3-[(5-fluoro-2,3-dihydrothiophen-4-yl)methylsulfanyl]propan-2-ol ethane;N-(2-propan-2-ylsulfonylphenyl)methanesulfonamide 2-[6-chloro-3,4-dimethyl-5-(1H-pyrazol-5-yl)pyridin-2-yl]propanoic acid 3-bromo-2,4-difluorobenzonitrile 2-[(2R)-1,1,1,3,3,3-hexafluoropropan-2-yl]oxy-5-nitropyridine (2S)-1,2-bis[3-(cyclopropylmethoxy)phenyl]piperazine (E)-3-[4-(dimethylamino)phenyl]-N,2-bis(hydroxyimino)but-3-enamide 2-(2,4-dimethylphenyl)sulfanylbutanenitrile 4-[(1S)-1-[(3,5-dichloropyridin-2-yl)amino]ethoxy]-2H-isoquinolin-1-one 2-[4-(1H-benzimidazole-2-carbonyl)phenoxy]-2-phenylacetic acid 1-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]ethanamine [4-(methyliodanuidylcarbamoyl)phenyl]boronic acid [4-(2-fluorophenyl)piperazin-1-yl]-[5-methyl-7-(trifluoromethoxy)-3,4-dihydronaphthalen-2-yl]methanone 2-[[4,5-bis(ethenyl)-1H-imidazol-2-yl]methoxy]-N-ethylethanamine 5-(furan-3-yl)-N-[1-methoxy-2-phenylethyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-3-carboxamide;hydrochloride 3-[6-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-2-methoxypyridin-3-yl]-N'-hydroxyprop-2-enimidamide 4-(2-chloro-6-ethylphenoxy)-N'-hydroxypyridine-2-carboximidamide 5-[3-(2,4-dihydroxyphenyl)-1,2,4-oxadiazol-5-yl]-7-methyl-1H-pyrrolo[2,3-c]pyridin-4-one [6-(aminomethyl)-9H-fluoren-1-yl]oxyphosphonamidic acid N'-(5,6-dimethylimidazo[1,2-a]pyridin-3-yl)sulfanylacetohydrazide 2-(1,3,4,5-tetrahydrocyclohepta[c]isochromen-6-yl)ethanol 1-azidooxy-2,3,5,6-tetrafluoro-4-(3,4,5,6-tetrachlorocyclohexa-1,3-dien-1-yl)benzene 4-hydroxy-3,5-dimethyl-2,6-dioxopyrimidine-1-carbothioamide 3-(azidomethyl)-1-[1-(4-methoxyphenyl)ethyl]pyrrolidine 3-(2,6-dioxopiperidin-4-yl)-5-propoxycarbonylbenzoic acid 2-(4-ethoxy-N-hexadecylanilino)acetamide (Z)-2,3,6-trifluoro-4-methylsulfonyl-1-phenylhept-3-en-1-one 4-[(3R)-1-[(2S)-3,3-dimethylbutan-2-yl]piperidin-3-yl]oxy-6-fluoroquinoline 4-(3,5-difluoro-2-hydroxyphenyl)butanoic acid 4-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(hexyl)amino]phenol 4-[(1S,5R)-3-benzyl-2,6-dioxabicyclo[3.1.0]hexan-2-yl]phenol 4-chloro-1,3-diethyl-5-(trifluoromethyl)pyrazole 1-phenylpentane-2,4-diol;propanoic acid (E)-N-[5-cyano-4-(dimethylaminosulfanyl)pyridin-2-yl]-3-[5-ethoxy-6-(1-propylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-ium-3-ylidene]prop-1-ene-1-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-2-methoxybenzamide 7-[2,6-di(propan-2-yl)phenyl]furo[3,4-b]pyridine 2-(1,3-benzodioxol-5-yl)-6-cyclopenta-1,4-dien-1-yl-1H-pyrazolo[1,5-a]pyrimidine 1-azido-N,4-diphenylmethanesulfonamide N-(4-anilinophenyl)-2,4,6-trimethylbenzenesulfonamide 3-[1-(2,4-difluorophenyl)ethyl]-6-methoxy-1-piperidin-4-yl-5H-pyrazolo[3,4-d]pyrimidin-4-one 1-azido-2-benzylsulfinylbenzene N-[4-chloro-3-(pyridine-2-carbonyl)phenyl]acetamide 3-[(4-fluorophenyl)methyl]-7-oxo-8H-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylic acid N-(2-butylquinolin-7-yl)-6-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]pyrimidin-4-amine (4R)-4-(3,5-dichlorophenyl)-1-phenylmethoxycarbonylpyrrolidine-2-carboxylate 4-(2-methoxyethylamino)-N'-[6-(3-methoxyphenoxy)pyridin-3-yl]-1,2,5-oxadiazole-3-carboximidamide (E)-2-cyano-3-[4-(dimethylamino)phenyl]-N'-hydroxyprop-2-enimidamide (E)-3-[3,4-dichloro-N-[1-(2,6-dimethylanilino)-5-methyl-1-oxohexan-2-yl]anilino]but-2-enal 4-[[(3S)-1,6-dioxopiperidin-3-yl]amino]-N'-hydroxypyridine-2-carboximidamide 1-[6-(dimethylamino)pyrimidin-4-yl]-3,4-dihydro-2H-quinoline-5,7-diamine 4-[5-(methylideneamino)-1,3-dihydroisoindole-2-carbonyl]naphthalene-1-carbonitrile 3-methoxy-5,6-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxylic acid 5-methyl-2,6-diphenylpyrrolo[3,4-d]pyrimidine 1-[4-(azidomethyl)cyclohexyl]-2,3,5-triiodobenzene 5-hydroxy-4,6-diphenylquinoline-2-carboxylic acid 2-(1,3-benzoxazol-5-yl)-N-[4-(1-hydroxyethyl)-9H-fluoren-1-yl]acetamide (Z)-N',1,3,5-tetramethyl-6-methylidene-2-phenylcyclooctene 3-(2,4-dimethylphenyl)-1-(1-methoxyethyl)pyrrolidine 3-[5-(2,6-diethylphenyl)-1H-imidazol-4-yl]pyridine (3S)-N,5-dimethyl-1-[(2R,6R)-6-phenylpiperidine-2-carbonyl]pyrrolidine-3-sulfonamide 3-[(1S)-2,2-dimethylcyclopropyl]-5-(2-fluoroethoxy)pyridine N-(3,4-diethoxyphenyl)-4-(dihydroxymethyl)azepane-1-carboxamide 3-amino-6-(4-bromophenyl)-N-methylpyrazine-2-carboxamide 2,3-dimethylpentane;5-(4-piperidin-1-ylphenyl)-1H-pyrrole-2-carboxylic acid (2R)-1,4-bis[4-fluoro-3-(trifluoromethyl)phenyl]butane-2,3-diol (E)-N,N-dimethyl-3-phenylmethoxyprop-1-en-1-amine 1-(4-methoxyphenyl)heptan-3-ol 2-[(Z)-2-methoxyethenyl]-1,3-dioxoisoindole-4-carboxamide N-[2,6-dichloro-4-(1H-tetrazol-1-ium-5-yl)phenyl]-2-methoxyiminoacetamide 2-[4,5-dimethoxy-N-(2-phenylethyl)-2-sulfoanilino]propanoic acid 2-[4-(1H-indole-2-carbonyl)piperazin-1-yl]-N-(1,3,5-trimethylpyrazol-4-yl)acetamide 1-(8,9-dihydrothieno[2,3-f]quinolin-10-yl)piperazine 1-amino-3-[2-(bromomethyl)phenyl]thiourea [5-hydroxy-3,4-dimethyl-1-(quinolin-8-ylmethyl)indol-2-yl]-phenylmethanone (2S)-3-amino-N-methyl-1-phenylbutan-2-amine;dihydrochloride N-(3,5-dichlorophenyl)-N-(2-hydroxyethyl)acetamide 3-[4-methylsulfonyl-6-(piperazine-1-carbonyl)cyclohexa-2,4-dien-1-yl]benzenesulfonamide N-[(3S,5R)-1-[6-[(6-bromopyridin-2-yl)methoxy]quinolin-2-yl]piperidin-3-yl]acetamide N-[6-amino-5-chloro-3-(difluoromethyl)pyridin-2-yl]cyclopropanecarboxamide 2-(3,4-dichlorophenyl)-N-[(1R,2S)-2-ethylcyclohexyl]acetamide 3-[5-amino-2,4-dihydroxy-3-(1H-indol-6-yl)phenyl]propanoic acid (2E)-2-[[4,6-bis(trichloromethyl)-1H-benzimidazol-2-yl]sulfanyl]-N-methoxyimino-2-phenylacetamide 1-[4,6-di(propan-2-yl)pyrimidin-5-yl]piperidine-3-carboxylic acid 2,4-dichloro-N-(3-nitrophenyl)benzenesulfonamide N-[5-[(2,4-dihydroxyphenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-phenylpropanamide;hydrochloride 2-[(6R)-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]-N-(2,3,4-trimethoxyphenyl)acetamide 7-phenyl-4,5,6,8-tetrahydro-3H-quinazoline 3-[(3Z,5E)-5-(4-cyanophenyl)hepta-1,3,5-trien-2-yl]cyclohexane-1-carboxylic acid (2R)-4-[(6-azidopyridin-3-yl)methoxy]-1,2,5-oxadiazole (3S)-4-[4-[4-(difluoromethoxy)phenoxy]phenyl]sulfonyl-2,8-diazaspiro[4.5]decane;hydrochloride 3-azido-2,4,5-trifluoro-6-(3-phenylpropyl)aniline N-(6,7-dimethylcyclohepta-1,3,6-trien-1-yl)-2-[4-[[5-fluoro-4-(6-hydroxy-5-methoxyindazol-2-yl)pyrimidin-2-yl]amino]phenyl]acetamide (2S,4R)-N-benzyl-5-oxo-4-[2-(1H-pyrrol-3-yl)ethynyl]pyrrolidine-2-carboxamide 3,4-bis(ethenyl)-6-phenyl-1H-pyridin-2-one 3-(2,5-dichlorophenyl)sulfanylpropyl-(methylideneamino)azanium (3Z)-4-methyl-3-[[2-(1,4-oxazepane-4-carbonyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]methylidene]piperazin-2-one 7-aminosulfanyl-2,4-difluoro-3-oxo-1H-indene-5-carboxylic acid 4-N-[(Z)-3,5,5-trimethylhexan-2-ylideneamino]benzene-1,4-diamine 6-amino-4-[2-bromo-3-(trifluoromethyl)phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 4-[5-[2-chloro-5-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl]phenol N-(2,4,6-trimethylphenyl)-1H-indole-3-carboxamide 3-amino-2-(4,5-dimethoxypyrimidin-2-yl)propanamide 5-(2,4-dichlorophenyl)furan 6-[4-(2-aminoethyl)piperazine-1-carbonyl]-5,7,8,9-tetrahydrothieno[3,2-h]quinolin-2-amine;dihydrochloride 5-[2,4-difluoro-6-(methoxymethyl)phenyl]-1,1,1-trifluoropentan-3-one (2Z,4Z)-5-[8-amino-1-[(3S)-oxolan-3-yl]pyrazolo[4,3-c]quinolin-5-yl]penta-2,4-dienoic acid 2-[(3-hydroxyphenyl)methyl]-5-(1H-indol-3-yliminomethyl)benzenethiol 1-(difluoromethyl)-4-[2-ethoxyethynyl(phenoxy)phosphoryl]oxybenzene N-azido-4-phenyl-1,3-thiazole-2-sulfonamide N-[3-(azepan-1-yl)propyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 6-(3-fluorophenyl)sulfonyl-1,4-dihydroquinazoline 1-(2,4-dibromophenyl)-5-ethylpyrazole 7-(3-methylsulfonylphenyl)pyrazolo[1,5-a]pyrimidine N-benzyl-2,5-dimethoxyaniline 1-(3-chlorophenyl)-N-[2-[[(E)-1-(6-oxopyridin-2-ylidene)propan-2-yl]iminomethyl]phenyl]cyclopropane-1-carboxamide 6-[2-(4-chlorophenoxy)acetyl]-N-(cyclopropylmethyl)-6-azaspiro[3.4]octane-8-carboxamide (2Z)-4,8a-dimethyl-2-[(3,5,6-trimethoxypyridin-2-yl)methylidene]-1H-quinazoline 3-(2,6-difluorophenyl)-4H-pyridine 5-(3,4-diethoxyphenyl)sulfonyl-6-fluoro-1H-indazole 2-(2,5-dioxoimidazolidin-4-yl)-N-(6-methoxypyridin-3-yl)acetamide 4-[[6-[2,3-difluoro-5-(methanesulfonamido)phenyl]quinazolin-2-yl]amino]-N-ethylpiperidine-1-carboxamide 3,5-dinitro-N-(2-oxo-1H-pyridin-4-yl)benzamide (2E,3S)-4,6,8-trifluoro-3-[(1-hydroxyisoquinoline-5-carbonyl)amino]-2-methylhepta-6,8-dienoic acid 2-methyl-3H-benzimidazole-5,6-dicarboxylic acid 3-[(E)-1,2-bis(4-chlorophenyl)ethenyl]-6-methoxyisoquinoline 1-[1-(3,4-difluorophenyl)ethyl]-6-(4-methoxyphenyl)sulfanylimidazo[4,5-c]pyridine 5-cyclopentyloxy-1,3-dimethylpyridin-2-one 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;8-chloro-3-ethyl-2-(2-oxoazetidin-1-yl)isoquinolin-1-one 5-amino-N-[2,6-dichloro-4-(trifluoromethyl)phenyl]-2-methoxypyridine-3-carboxamide 3-[4-[4-(dimethylamino)phenyl]piperazine-1-carbonyl]-5,6-bis[4-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidin-4-one 7-chloro-4-[(3S,5R)-4-cyano-3,5-dimethylpiperazin-1-yl]quinoline-6-carboxylic acid;ethane 7-(2-ethylbutyl)-1,3-dimethoxypyrrolo[3,4-b]quinoxaline 4-[2-[2,5-dimethyl-N-(oxan-4-yl)anilino]acetyl]benzoate 3-[(3R)-1-methylpiperidin-3-yl]-7-phenyltriazolo[4,5-d]pyrimidine;hydrochloride N-[3-(methylamino)pyridin-2-yl]acetamide 1-ethylsulfonyl-4-[4-(trifluoromethoxy)phenyl]piperazine 1-(4-butoxyphenyl)-6,7,8,9-tetrahydropyrazolo[3,4-c]quinoline 1-[4-amino-2,6-di(propan-2-yl)phenyl]ethanone 2-amino-3-[5,7-difluoro-1H-indole-2-carbonyl(methyl)amino]propanoic acid 1-[3-[5-(2,4-dichlorophenyl)oxolan-2-yl]piperidin-3-yl]-2,6-naphthyridine 4-N,5-diethyl-2-methoxybenzene-1,4-diamine 6-[3,5-dichloro-4-[(1R)-2,2-dimethylcyclopropanecarbonyl]oxyphenyl]pyridine-2-carboxylic acid (1R)-N-[2-(4-chlorophenyl)ethyl]-7,9,10-trihydroxy-9H-anthracene-1-carboxamide 4-(6,8-diamino-1-fluoroisoquinolin-3-yl)-2-methoxy-5-propan-2-ylbenzoic acid 3-(3,4-dimethoxyphenyl)sulfanyl-6-[5-(trifluoromethyl)pyridin-2-yl]-8H-[1,2,4]triazolo[4,3-b]pyridazine N-[(2R,4S)-1-(benzenesulfonyl)-6-methoxy-7-oxooctan-2-yl]acetamide 4-(3,6-dihydro-2H-pyran-5-yl)-N'-hydroxybenzenecarboximidamide 1-(2,6-dichlorophenyl)-3-[[4-[methylsulfonyl(oxolan-3-yl)amino]piperidin-1-yl]methyl]urea 6-[5-chloro-2-(difluoromethoxy)phenyl]-4H-thiopyran 3-benzyl-5-(trifluoromethyl)-1H-indole N-(4,5-dihydroimidazo[1,2-a]quinoxalin-7-yl)-2-methoxyacetamide 2-[5-[2,6-dichloro-4-(1H-1,2,4-triazol-5-yl)phenyl]-3-methoxy-10-oxo-8-thia-4,11-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,12-tetraen-12-yl]acetamide 4-ethenyl-N,2,6-trimethylbenzenesulfinamide 2-(3,4-dimethylphenoxy)ethylazanide 1-(9H-fluoren-3-yl)cyclohexa-2,4-dien-1-amine 6-[4-(2,3-difluorophenyl)piperazine-1-carbonyl]-3H-quinazolin-4-one N-[(2E,4Z)-hepta-2,4-dienyl]-6,8-dihydroxyquinoline-5-carboxamide N-ethyl-4,5-dimethylpyridine-3-sulfonamide 4-[(2-azidooxy-3,5-dichlorophenyl)methyl]-1H-indole 2-[(1,1-dioxothiolan-3-yl)methyl]isoindole-1,3-dione 4-azido-2-(2,3-difluorophenyl)-1,3-benzothiazole 4-(1,2,3-benzotriazin-4-yl)piperazine-1-carboxylic acid (E)-1,2-dipyridin-4-ylundec-1-en-3-one 6-chloro-3,4-dihydrodibenzothiophene;5-cyclohexyl-4-phenylcyclohexa-1,3-diene [2-(methoxymethyl)pyrrolidin-1-yl]-(6-nitronaphthalen-2-yl)methanone N-cyclohexyl-2-(4-ethoxyphenyl)-7,8-dihydro-[1,3]thiazolo[5,4-e]indazole-6-carboxamide 5-[(1R,3E)-6-bromohexa-3,5-dienoxy]-2-chlorophenol 3-(2,4-dimethoxyphenyl)propan-1-ylcarbamic acid [(4S)-3,4-dihydro-2H-1,5-benzodioxepin-7-yl]-[6-hydroxy-4-methoxy-3-(piperidine-1-carbonyl)quinolin-8-yl]iminoazanium 5-methyl-2-[(3S)-1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-3-yl]pyrimidine-4-carboxylic acid (2S)-N-[2-oxo-1-phenyl-2-[[2-(pyrrolidine-1-carbonylamino)acetyl]amino]ethyl]morpholine-2-carboxamide N-[4-(3-chloropropoxy)phenyl]acetamide 2-(5,6-dioxobenzimidazolo[1,2-a]quinolin-11-yl)-N-pyridin-2-ylacetamide (6R)-7-[[2-methylsulfanyl-2-(4-phenylmethoxyphenyl)acetyl]amino]-3,3a,4,5,6,7a-hexahydro-1H-isoindole-2-carboxylic acid 3-(dimethylamino)-4-[4-(ethylaminomethylsulfanyl)phenyl]benzoic acid 6-(3,4-dichlorophenyl)-2-oxo-1H-pyrimidine-5-carboxylic acid 2-[(E)-pent-3-enyl]-1,5-diphenylpentane-1,5-dione 6-amino-3-(cyclopropylmethoxy)-2-iodobenzoic acid N-[5-(azidomethyl)-2,4-difluorophenyl]-1H-indole-3-carboxamide 2,4-dichloro-N-[3-methoxy-5-(trifluoromethyl)phenyl]-N-(2-oxopropyl)benzamide 5-[3-[[4-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]methyl]phenyl]-[1,3]oxazolo[4,5-b]pyridine 2-chloro-3,6-diphenylbenzenethiol 4-[3-chloro-2,6-dimethoxy-5-(pyridine-3-carbonylamino)benzoyl]piperazine-1-carboxylic acid 1-[4-(6-methylsulfonylpyridin-3-yl)phenyl]butan-2-one 4-(2,6-dimethylphenyl)sulfanyl-3-methoxy-1,2-oxazole N-[4-(3,5-dimethylpyrazol-1-yl)butyl]-6-oxo-2,5-dihydro-1H-pyridine-4-carboxamide 4-N-(2-morpholin-3-ylethyl)-6,7-dihydro-5H-pyrrolo[1,2-b]pyrazole-2,4-dicarboxamide 2-bromo-N-cyclohexyl-4,6-bis(trichloromethyl)aniline (NE)-N-[2-amino-1,3-bis(4-ethynylphenyl)propylidene]hydroxylamine 4-[(2,6-dihydroxyphenyl)methyl]piperazine-1-carboxylic acid 2-[(1,3-dimethylpyrazol-4-yl)amino]oxycarbonylbenzoate 4-methyl-6-[2-oxopropyl(phenacyl)amino]-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 2-(3,5-difluorophenyl)-3-ethylsulfanylquinoline 4-(difluoromethyl)-N-[3,5-difluoro-2-(1H-imidazol-5-yl)phenyl]-2-methoxypyridine-3-carboxamide 6-[(3R)-5-[(2,4-difluorophenyl)methyl]-3-pyridin-4-ylimidazol-4-yl]imidazo[1,2-a]pyrazine 1-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]quinoxaline 2-cyclohexyloxy-N-methyl-N-(4-propan-2-ylphenyl)-5-(trifluoromethyl)pyrimidin-4-amine 4-chloro-N-[2-methoxy-6-methyl-5-(6,7,8,9-tetrahydropyrido[1,2-a]benzimidazole-3-carbonyl)phenyl]benzenesulfonamide 4-[5-(1,3-dioxolan-2-yl)thiophen-3-yl]-6-[(E)-2-methylbut-1-enoxy]benzene-1,3-diamine N-[4-(diethylamino)-2-methoxyphenyl]-3-methoxycarbonyl-6,7-dihydroindole-1-carboxamide 1-[1-(1,3-benzodioxol-5-ylmethyl)azetidin-3-yl]-4-(5-chloropyridin-2-yl)piperazine 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-6-(4-ethylcyclohexyl)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 2-ethylbutanedioate;tetraphenylphosphanium 2-[[4-bromo-3-(trifluoromethyl)phenyl]methylidene]propanedinitrile 6-azidooxy-4,4-dimethyl-1H-3,1-benzoxazin-2-one 4-amino-1-(9H-fluoren-2-yl)cyclohexane-1,3-diol N-[3-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazole-3-carbonylamino)phenyl]pyridine-4-carboxamide 1-[5-[(dimethylamino)methyl]furan-2-carbonyl]piperidine-4-carboxylic acid N-[(4-methylphenyl)sulfonylmethyl]-2,3-dihydro-1H-indene-5-carboxamide 2-(4,6-dichlorocyclohexa-1,5-dien-3-yn-1-yl)oxy-N-[4-(trifluoromethylsulfanyl)phenyl]acetamide 2-methyl-2-[4-[6-oxo-1-(2,3,5,6-tetrafluorophenoxy)hexan-2-yl]phenoxy]propanoate N-[(4E,5Z)-4-ethylideneocta-1,5-dien-3-yl]-2-piperidin-4-ylpyrimidine-4-carboxamide 6-amino-4-(2-hydroxy-3,5-dinitrophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide N-(2-fluoroethyl)-3,4-dihydro-1H-isochromene-6-carboxamide 4-(6,7-difluoroquinolin-2-yl)phenol N-(2-methylbutan-2-yl)-N,1-diphenylmethanesulfonamide N-methyl-4-[2-oxo-2-(2H-triazolo[4,5-b]pyridin-6-ylamino)ethoxy]benzenesulfonamide 4-[[(3aS,6aS)-2-ethylsulfonyl-1,3,3a,4,5,6,6a-octahydrocyclopenta[c]pyrrole-5-carbonyl]amino]benzoic acid 6-(4,5-dihydropyridin-2-yl)-1-phenyl-[1]benzofuro[3,2-c]isoquinoline N-[4-(dimethylamino)phenyl]-N',N'-diethylethane-1,2-diamine 4-methoxy-2-(N,4-dimethylanilino)benzoate 7-chloro-N-[(3S)-5-hydroxyhexan-3-yl]quinoline-4-carboxamide N-(3-methylbut-2-enyl)-N-phenylquinolin-8-amine (2Z,5E)-3-ethyl-6-[2-[(1S)-4-fluoro-6-methoxy-7-methylidenecyclohepta-2,4,6-trien-1-yl]ethynyl]-5-methoxy-N'-methylhepta-2,5-dienehydrazide 2-azido-6,7-dihydro-4H-furo[3,2-c]pyran 5-amino-3-(3,4-diethoxyphenyl)-2,3-dihydro-1,2-oxazole-4-carbonitrile 1-(4-methoxyphenyl)sulfonyl-3-[5,6,7,8-tetrahydropyrido[2,3-b]pyrazin-3-yl(thiophen-2-yl)amino]pyrrolidin-3-ol 1-[3,5-bis(trifluoromethyl)phenyl]-4-ethoxy-N-(fluoromethoxy)phthalazin-6-amine 2-(3-methylbenzotriazol-5-ylidene)propanedinitrile 1-[5-fluoro-2-(4,4,4-trifluorobutyl)benzoyl]piperidine-3-carboxylic acid 2-azido-4-fluoro-3,5-dimethyl-1H-indole (3S)-1-[(4-azidosulfanylphenyl)methyl]pyrrolidin-3-ol 4-[4-(N'-hydroxycarbamimidoyl)pyrazol-1-yl]piperidine-1-carboxylic acid ethane;1-[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]-3H-indole N-azido-4-pyridin-3-ylpyridine-2-carboxamide 1-[(3R)-4-azido-1,2,3,4-tetrahydroisoquinolin-3-yl]-N,N-dimethylmethanamine N-[4-[1-(2,2-dimethyloxan-4-yl)ethenyl]pyridin-2-yl]-5-hydroxycyclohepta-1,3,6-triene-1-carboxamide 5-(chloromethyl)-1,4-difluoro-2-methoxybenzene;ethane 2-[4-chlorobutyl(3,5-dimethoxypropanoyl)amino]benzenesulfonic acid 2-[[(3S,4R)-1-[5-chloro-2-(difluoromethoxy)benzoyl]-3-(hydroxymethyl)piperidin-4-yl]amino]pyridine-4-carbonitrile 5-[(2S,3R)-2-[(dimethylamino)methyl]-3-phenylmorpholine-4-carbonyl]-1H-pyrrole-3-carbonitrile 2,2-dimethyl-3-[3-(4-naphthalen-1-ylphenyl)sulfanyloxyphenoxy]propanoic acid N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide (2R,3S)-N-ethyl-3-methoxyimino-4-[4-(5-nitropyridin-2-yl)piperazin-1-yl]butan-2-amine 1,3-bis(methylsulfanyl)benzo[f]isoindole ethane;2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxy-N-(pyridin-4-ylmethyl)-6H-cyclohepta[d]pyrimidin-4-amine 4-(1,3-benzothiazol-2-yl)-N-ethylaniline ethane;2-(4-methylphenoxy)-N-[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]acetamide (1R,2S)-N-[[4-fluoro-3-(trifluoromethyl)phenyl]carbamoyl]-4-fluoro-2-pyridin-3-ylcyclohexane-1-carboxamide 2-[(7S)-3-cyano-5-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-7-yl]-N,N-dimethylacetamide N-[2-(4-amino-6,7-dimethoxyquinazolin-2-yl)ethynyl]oxolane-3-carboxamide (E)-2,3-diamino-N'-[(4R)-5-amino-4-methyl-1-phenylpentan-3-yl]prop-2-enimidamide 1-cyclopropyl-2-(difluoromethoxy)-4-iodobenzene 1-[(3R,4S)-1-azido-4-fluoropiperidin-3-yl]-N-cyclopropyl-5-methoxybenzimidazol-2-amine [2-(4-iodophenyl)-5,7-dihydro-4H-thieno[2,3-c]pyridin-6-yl]-[5-methoxy-2-(triazol-2-yl)phenyl]methanone 2-[(1R)-1-phenylethyl]iminoacetate 2-[(4R)-6-methylidene-1,3-bis(2-phenylethyl)-3,4-dihydro-2H-pyrido[1,2-a]pyrazin-7-yl]acetaldehyde;6-(methylamino)pyridine-2,5-dicarbonitrile 5-(3,4-dimethylphenyl)-2-N-[4-ethoxy-3-(3-fluoropropoxy)phenyl]-1H-pyrimidine-2,4-diamine 2-(dimethylamino)-1-[5-fluoro-6-[4-[(2S,3R)-4-propan-2-ylmorpholine-2-carbonyl]phenoxy]-1H-indole-2-carbonyl]piperidine-4-carboxylic acid 1,4-di(cycloheptylidene)naphthalene N-[[2,3,6-trifluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]carbamoyl]carbamate 4-(2,3-difluorophenyl)-2-methylsulfonylaniline 2-ethyl-N,3-dimethylbutanamide;5-[(E)-1H-indol-6-ylmethylideneamino]-4-piperidin-1-yl-7H-pyrrolo[2,3-d]pyrimidin-6-amine 2-[3-(5,8-difluoro-3,4-dihydroquinolin-6-yl)-1H-pyrazol-5-yl]-N'-pyridin-2-yl-3H-benzimidazole-5-carboximidamide 2-[(4-methylpiperidin-1-yl)methyl]benzamide N-azido-2,5-bis(phenylmethoxy)benzamide 2-[6,8-dibromo-7-(1H-indole-2-carbonyl)-3-methylpyrrolo[3,2-f]quinoxalin-5-yl]acetic acid (3S)-5,6,7,8-tetramethyl-2-[(E)-4-phenylbutylideneamino]-3H-quinazolin-4-one 3-(2,2-diethoxyethyl)-5H-imidazo[5,1-a]isoindol-6-amine 2-tert-butyl-4-[(E)-4,4-dimethylpent-1-enyl]-6-fluoropyridine 2-[2,4-bis(2,3-dimethylphenyl)phenoxy]aniline;ethane (4-chlorophenyl)-[5-cyclopropyl-3-methoxy-2-methyl-6-[2-[(1S,2R)-2-(trifluoromethyl)cyclohexyl]ethynyl]phenyl]methanone ethane;methoxycyclohexane;3-methylbutanoic acid;4-[2-(4-methylpiperazine-1-carbonyl)phenoxy]benzonitrile 2,4-dimethyl-8-pentoxyquinoline 4-[6-[methyl(pyrimidin-2-yl)amino]pyridine-3-carbonyl]piperazin-2-one (2Z,4E)-N-[1-(4-chlorophenyl)ethyl]-2-methoxy-4-phenylsulfanylhexa-2,4-dienamide 4-tert-butyl-1,6,7-trimethylnaphthalene 3-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]propanamide 2-[6-(2,4-difluorophenyl)-3-fluoronaphthalen-1-yl]pentanoic acid 7-(3-azidopentyl)naphthalene-2-carboxamide 2-[6-(4-fluorophenyl)-5,7-dihydrobenzo[d][1]benzazepin-9-yl]-N-methylethanamine 5-(1,3-thiazol-2-yldiazenyl)naphthalene-2-sulfonic acid (2S)-N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-1-(4-ethylbenzoyl)piperidine-2-carboxamide 7-[(2R)-2-cyclopropyl-3-[4-methoxycarbonyl-1-(1,1,1-trifluorobutan-2-yl)piperidin-4-yl]propanoyl]-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]diazepine-1-carboxamide N-[2-(3,5-dimethylcyclohexyl)ethyl]-1H-imidazole-4-carboxamide N-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]thiophene-3-sulfonamide [3-amino-6-(2,4-difluorophenyl)pyrazin-2-yl]-pyridin-4-ylmethanone 3-chloro-2,5-dimethoxybenzenesulfonic acid 6-butanoyloxynaphthalene-2,3,4-tricarboxylic acid 1-(6-azidohexyl)-N,2,3,4-tetrahydroquinolin-8-amine 1-[2-[(3E)-hexa-1,3,5-trien-3-yl]oxyethyl]-N'-hydroxyimidazo[4,5-b]pyridine-6-carboximidamide N-(2-methyl-3,4-dihydro-1H-isoquinolin-6-yl)-5-[[2-(2,4,6-trifluorophenyl)acetyl]amino]furan-2-carboxamide 5-bromo-N'-hydroxy-1H-indole-7-carboximidamide (5-ethylpyridin-3-yl)-[3-methoxy-4-(2H-tetrazol-5-yl)phenyl]methanone [2-[bis(cyclohexylmethoxy)phosphoryl]phenyl]-phenylmethanone 3-azido-6-chloro-2-methyl-4,5-dihydroindazole 5-[(2,3-difluorophenyl)iminomethyl]-6-hydroxy-1H-pyrimidine-2,4-dione 2-azido-6,7,9-trimethoxy-4-[(2S)-3-methylbutan-2-yl]-1H-benzo[f]isoindole 4-[[4-(6,7-dichloroquinazolin-2-yl)piperazin-1-yl]methyl]phenol 3-[4-[2-(4-methylsulfanylpiperazin-1-yl)ethoxy]phenyl]pyrazolo[1,5-a]pyrimidine 6-(2,2-dimethylpropanoylamino)pyridine-3-carboxylic acid 4-[(3-methyl-4-propylpyrrolidin-1-yl)methyl]benzamide 4-[(2S,3R)-3-azido-1-cyclopropylbutan-2-yl]benzene-1,3-diol 2-[(1S)-6-hydroxy-3,4-dihydro-1H-isochromen-1-yl]acetic acid 1-[2,4-dimethyl-5-(1H-pyrrol-3-yl)benzoyl]azetidine-3-carboxylic acid 4-chloro-3,5-difluoro-N'-hydroxybenzenecarboximidamide 1-[(4-fluorophenyl)methyl]-6-(pyridin-4-ylmethoxy)spiro[2H-indole-3,8'-3,7-dihydro-2H-furo[2,3-g][1,4]benzodioxine] 3,4-dimethyl-6-(trifluoromethoxy)-1H-quinolin-2-one 4-[5-chloro-2-(3,7-dimethyloctoxy)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile N-[(3R)-1,3-dimethylpiperidin-4-yl]-2-fluoro-6-(5-hydroxy-6-oxoheptoxy)benzamide;ethane (1S)-N'-[[2,6-dimethoxy-4-(5-morpholin-4-ylcyclohepta-1,3,6-trien-1-yl)phenyl]methyl]-2,2,2-trifluoroethane-1,1-diamine 2-chloro-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carboxylic acid N-(3-chlorophenyl)-4-[5-fluoro-4-(2,2,2-trifluoroethylamino)pyrido[3,2-d]pyrimidin-8-yl]benzamide 7-(2-methoxyethyl)-1,8-dimethyl-3-[4-(3-propan-2-ylphenyl)cyclohexyl]-6H-purin-1-ium (2R)-2-[4-[2-oxo-3-[1-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]phenyl]propanamide 3,5-dichloro-4-[4-(oxan-2-ylmethoxy)-1H-pyrrolo[3,2-c]pyridine-2-carbonyl]benzenesulfonamide (1Z,3E)-2-[2-(4-chlorophenoxy)ethyl]penta-1,3-dien-1-amine N-(2,4-dinitrophenyl)-N-hexylbutanamide 4-[[2,3-difluoro-5-(trifluoromethyl)phenyl]carbamoylamino]-N-ethyl-1H-pyrazole-5-carboxamide 1-[2,6-bis(2-methoxyethoxy)phenyl]ethanone 2-[(3S)-3-[4-[[5-chloro-6-(2,2-difluoroethoxy)pyridin-3-yl]methoxy]phenyl]-1-(4-cyanocyclohexanecarbonyl)pyrrolidin-3-yl]oxyacetic acid N-(2,4-dinitrophenyl)-N-ethylmethanesulfonamide (E)-2-cyano-3-[5-(2,4-dichlorophenyl)furan-2-yl]prop-2-enamide 5-(azidomethyl)-3-chloro-2,4-difluorophenol 1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]sulfonyl-4-phenylpiperazine 4-fluoro-6-methylbenzene-1,2,3,5-tetracarboxylic acid 3,5-dichloro-4-[(3S)-4-(1-methyltetrazol-5-yl)-2-oxopyrrolidin-1-yl]benzonitrile 1-(2-fluorophenyl)-5,6,7,8-tetrahydroquinolin-4-one;hydrochloride N-[5-cyclopropyl-3-(2,6-dichlorophenyl)-1H-pyrazol-4-yl]-6-phenylpyridin-3-amine N-[(E)-but-2-enyl]formamide;ethane;3-fluoro-6-(4-hydroxycyclohexyl)-4H-1,2,5-oxadiazine-7-thione 2,6-dichloro-4-[5-[(1S)-3-hydroxycyclopentyl]sulfonylpyridin-2-yl]phenol 6-azidosulfonyloxybenzene-1,3-dicarboxylic acid 2-methyl-4,7-dioxo-5H-pyrrolo[3,4-d]pyrimidine-6-carboxamide 1-[2-azido-3-methyl-4-(trifluoromethylsulfonyl)phenyl]pyrrolidine 4-[2,3-bis(ethenyl)indol-1-yl]butanoic acid 3-[3,4,5-trichloro-1-(2H-naphthalen-1-ylidene)cyclohexa-2,4-dien-1-yl]pyridine ethane;3-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]piperidine-2,6-dione N-[4-amino-5-(3,6-dichlorocyclohexa-1,3-dien-1-yl)sulfonylpyrimidin-2-yl]-3-bromo-4-methoxybenzamide 4-[3-fluoro-5-(2-methylpropyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-[4-[(5-oxopyrimido[4,5-b][1,4]benzothiazepin-6-yl)amino]phenyl]acetic acid ethane;4-[(6E)-6-ethylidene-3,4-dihydropyridine-2-carbonyl]pyridine-2-carbonitrile 2-(4-chlorophenyl)-6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-amino-1,5-dimethyl-4H-1,2,4-triazol-4-ium-5-carboxamide;5-[2-chloro-6-(trifluoromethoxy)phenyl]-3,3-bis(3,3-dibromoprop-1-en-2-yl)thiophene-2-carboxylate (1E,3Z)-2-[3-(7-methoxy-2-oxochromen-4-yl)-5-phenoxy-1H-indole-2-carbonyl]penta-1,3-diene-1-sulfonic acid [6-[[6-(4,5-dimethylpyrimidine-2-carbonyl)-3,7a-dihydroimidazo[1,2-a]pyrazin-1-yl]methoxy]pyridazin-3-yl]boronic acid 2-[4-[(3,4-dichlorophenyl)methylamino]pyrimidin-2-yl]phenol 7-(4-chlorophenyl)-2-[3,5-dimethyl-4-[6-(trifluoromethoxy)benzimidazol-1-yl]phenyl]-N,N,2-trimethylheptanamide 3-[[4-[3,5-difluoro-2-(hydroxymethyl)phenyl]-1,2-oxazol-3-yl]amino]piperidine-2,6-dione 2-(4-azido-1H-indol-3-yl)ethanamine 6-bromo-1,3,4,9b-tetrahydroindeno[2,1-c]pyridin-2-one;hydrochloride 3-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]-6H-triazolo[4,5-d]pyrimidin-7-one 2-tert-butyl-N'-[3,5-bis(trifluoromethyl)phenyl]-N'-[(2,6-dichloro-4-ethoxybenzoyl)amino]-1H-imidazole-5-carbohydrazide N'-amino-2-(3,4-dichlorophenyl)-5,6-bis(1H-imidazol-2-ylmethoxy)pyridine-3-carboximidamide [(E)-[(2S)-1-(4-bromophenyl)piperidin-2-yl]methylideneamino]thiourea 2-ethylsulfanyl-5,6-difluorobenzene-1,3-dicarboxylic acid N-[5-[3-(7-thiophen-2-yl-3H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-yl]cyclohexanecarboxamide (5Z)-2-(4-chlorophenyl)imino-5-[[3,5-diiodo-4-[(3-nitrophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one N-[3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]formamide 2-[3,5-dimethyl-1-(5-oxo-4H-1,2,4-oxadiazol-3-yl)pyrazol-4-yl]-N-[(E)-[(Z)-2-hydroxypentan-3-ylidene]amino]acetamide 2-(5,6-dimethoxypyridin-3-yl)-7H-purine 1-[3,5-bis(trifluoromethyl)phenyl]-N-[4-[2-methoxyethyl(methyl)amino]-6-methylpyrimidin-2-yl]cyclopentane-1-carboxamide 4-[1,3-benzodioxol-5-yl(methoxy)methyl]morpholine;hydrochloride 2-[3-(4-aminophenyl)sulfonyl-5-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]phenoxy]-N-benzylacetamide 3-[1-amino-2-(4-aminophenyl)ethyl]aniline (Z)-4-methyl-2-[3,5,7-tris(4-methoxyphenyl)-2H-pyrazolo[3,4-c]pyridazin-6-ium-1-carbonyl]pent-2-enenitrile 4-methyl-1,2-bis(phenylsulfanyl)benzene 3-[2-(cyclopropylsulfonylamino)pyrimidin-4-yl]-N-ethyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide 2-chloro-N-(1H-imidazol-2-ylmethyl)-5-[(3R,4S)-3-phenylpiperidin-4-yl]oxybenzamide;dihydrochloride 1-[2-(4-chlorophenyl)ethyl]-N-[(6-methyl-2-oxo-1H-pyridin-3-yl)methyl]-6,7,8,9-tetrahydro-5H-pyrazolo[4,3-c]azepine-3-carboxamide (2-cyclopropyl-1,3-oxazol-4-yl)-[6-[5-methanimidoyl-2-[(6-methoxypyridin-3-yl)amino]phenyl]-1H-indol-3-yl]methanone (E)-N-[3,5-bis(trifluoromethyl)phenyl]-2-nitro-3-[4-(3-nitrophenyl)pyridin-1-ium-1-yl]prop-2-enamide;chloride (2Z,4E)-5-[[(1S,3R)-3-[[2-hydroxy-2-phenyl-1-(4-pyridin-3-ylphenyl)ethyl]amino]cyclopentanecarbonyl]amino]-N-methylidenepenta-2,4-dienamide (7S)-7-[2-(azepan-1-ylmethyl)-5-fluorophenyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide 6-amino-4-(1H-indol-3-yl)-2,4-dioxo-1,3-thiazinane-5-carbonitrile N-cyclohexyl-3-(4,6-dimethoxypyrimidin-2-yl)sulfanylprop-2-enamide 4-(2-nitrophenyl)piperidine 1-azidooxy-2-propylnaphthalene [(2R,6S)-2-butyl-6-propan-2-ylmorpholine-4-carbonyl]-(3-methoxyquinolin-7-yl)-diphenylphosphane N-[(4-methoxyphenyl)methyl]-2,2,5-trimethyl-3-[(1Z)-penta-1,4-dienyl]pyrrole-1-carboxamide N-(2-methylpropyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-7-carboxamide;hydrochloride 2-methyl-N-(3-nitrophenyl)-N-phenacylpropanamide 1-(3,4-dihydro-1H-isoquinolin-2-yl)-3,3-bis[4-(trifluoromethylsulfanyl)phenyl]propan-2-one N-[(2,4-dimethoxyphenyl)methyl]-6-oxo-1H-pyrimidine-5-carboxamide N-[4-amino-6-[3-(trifluoromethyl)anilino]pyrimidin-5-yl]propanamide;ethane 3-[(E)-4,5-dimethylhex-2-enoyl]-N'-propan-2-ylpyridine-2-carbohydrazide 2-(4-fluorophenyl)-N-[3-hydroxy-1-[4-(6-hydroxyhexanoylamino)cyclohexyl]piperidin-4-yl]-5-methoxypyrazole-3-carboxamide 4-[2,3-dihydro-1H-perimidin-2-ylmethoxy(phenyl)methyl]benzonitrile [(2R,4S)-1-benzylsulfonyl-4-hydroxypyrrolidine-2-carbonyl]-benzylazanium 5-butyl-2,6-bis(trifluoromethyl)pyridine-3,4-diamine [2-(5-methylfuran-3-carbonyl)piperazin-1-yl]-(3,4,5-trifluorophenyl)methanone 2-[(Z)-2-(6-hydroxypyridin-3-yl)ethenyl]benzaldehyde 1,4-bis(2-methylprop-1-enoxy)anthracene N-butyl-1,3-diethoxy-2,3-dihydro-1H-indene-5-sulfonamide 4-[1,3-dideuterio-2-(trifluoromethoxy)propan-2-yl]benzoic acid 2-[(3-ethoxythiophene-2-carbonyl)amino]-4-[(1R,5S)-6-methyl-3-azabicyclo[3.2.0]heptan-3-yl]butanoic acid 4-chloro-6-[(2Z,5R)-2-[(3-ethoxyphenyl)methylidene]hydrazinyl]pyrimidine-2-carboxylic acid 3,5-ditert-butyl-4-cyclopropyl-1-methoxypyrazole [(2S,3R)-2-phenyloxolan-3-yl]carbamic acid 2-ethoxy-6,7-dimethylnaphthalene N-[[1-(4,6-dimethylpyrimidin-2-yl)pyrazol-3-yl]methyl]-1-methylsulfonylcyclobutane-1-carboxamide (1Z)-N-[1-(6,8-dihydrobenzo[c]chromen-9-yloxy)propan-2-ylidene]hydroxylamine 2-[6-chloro-4-(4-ethylphenyl)quinazolin-7-ylidene]propanedioic acid 5-fluoro-4,7-dimethyl-3-propan-2-ylthieno[2,3-c]pyridine (3S,5R)-5-[1-[4-(difluoromethoxy)phenyl]ethylcarbamoyl]piperidine-3-carboxylic acid 2-[(6S)-3-(4-chlorophenyl)sulfanyl-8-oxo-5,6,7,9-tetrahydro-4H-pyrazolo[5,1-b]quinazolin-6-yl]benzoic acid 2-amino-4,7-dioxo-N-[3-(pyrazol-1-ylmethyl)phenyl]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide (1R,2S)-2-[5-[5-[2-(4-methylpiperazin-1-yl)ethoxy]pyridin-3-yl]-1H-indazol-3-yl]cyclopropane-1-carboxylic acid N-(2,3-dihydro-1H-inden-5-yl)-7-methoxy-6-[4-[methyl-[2-(methylideneamino)ethyl]carbamoyl]cyclohexa-2,4-dien-1-yl]oxy-2,3-dihydrochromene-4-carboxamide 4-[5-[(2,3-difluorophenyl)methylamino]-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]cyclohexan-1-one 2-(5-chloropyridin-2-yl)-3-[1-methoxypentan-2-yl-(4-phenylbenzoyl)amino]propanoic acid N'-hydroxy-2-[(5-methylpyridin-3-yl)methoxy]pyrimidine-4-carboximidamide 3-methyl-4-phenyl-6-(2-sulfanylidene-1H-pyrimidin-5-yl)benzene-1,2-dicarbonitrile (2S)-3,3,4-trimethyl-N-[4-(2-oxoimidazolidin-1-yl)phenyl]pentane-2-sulfonamide N-[2,6-difluoro-4-(1H-pyrazol-5-yl)phenyl]hexanamide N-[2-(methylamino)ethyl]-4-[6-methyl-3-oxo-7-(2,2,2-trifluoroacetyl)quinoxalin-5-yl]piperidine-1-carboxamide 2-(7-methyldibenzofuran-3-yl)thiophene N-[(E)-but-1-enyl]-2,4-dichloroaniline 5-(3-cyanopentanoyl)-N-[6-[(2R,4S)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]pyridin-2-yl]-1H-pyrrole-3-carboxamide 2-(4-acetyl-N-hexylanilino)propanoic acid ethane;4-methyl-1,2-dihydronaphthalene;4-[(4-phenylphenyl)methyl]benzonitrile 1,2-bis[2-(4-chlorophenoxy)phenyl]ethanone 6,8-dichloro-9-methylpurine N-[(E)-(5-bromo-2-hydroxyphenyl)methylideneamino]naphthalene-1-carboxamide N-[(1R,2S)-2-hydroxycyclobutyl]-3-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide (2E)-3-[3,5-dibromo-4-[hydroxy(diphenyl)methyl]iminocyclohexa-1,5-dien-1-yl]oxy-2-ethylidenebutanoic acid 3,5-difluoro-4-[3-(fluoromethyl)phenyl]benzenethiol;methanamine 2-[6-(2,3-dihydroxypropoxy)-2,2-bis(4-methylphenyl)hexanoyl]benzoic acid [2-(4,5-dimethylcyclohexa-1,3-dien-1-yl)phenyl]methanol 2-chloro-4,5-diethoxy-N-[3-fluoro-4-(2-pyridin-2-ylthieno[3,2-b]thiophen-6-yl)oxyphenyl]benzenesulfonamide 3-[(2,4-dichloropyrimidin-5-yl)-hexadecanoylamino]propanoic acid (5Z)-2-[3,6-dimethyl-1-(4-phenylphenyl)pyrrolo[3,2-b]pyridin-5-yl]imino-5-ethylidene-1,3-thiazolidin-4-one N-[4-(1,3-benzodioxol-5-yl)phenyl]formamide (1R)-3,4,4-trimethyl-2-[4-[(2S)-2-phenylpropoxy]butylimino]cyclopentan-1-ol 1-(2-iodo-6,7,8,9-tetrahydrodibenzofuran-3-yl)ethanone 6-[2,4-dimethyl-5-(trifluoromethyl)pyrazol-3-yl]hexanamide 6-[2-(azepan-1-yl)ethoxy]pyridine-3-carbonitrile (2S)-4-[5-amino-6-[(1R,3R,4S)-4-hydroxy-3-methylcyclohexen-1-yl]pyrazin-2-yl]-N-tert-butylpyrrolidine-2-carboxamide 2,5-diamino-N'-[(2S)-3-phenylbutan-2-yl]pyridine-4-carboximidamide 2-(6-aminopyridin-3-yl)-4,5-dichlorothiophene-3-carboxylic acid [2-(8-chloro-4-oxochromene-2-carbonyl)phenyl]-dimethylsulfanium 2-[1-[4,5-diamino-6-(trifluoromethyl)pyridine-3-carbonyl]piperidin-4-yl]oxypyrimidin-4-amine 6-(4-fluorophenyl)-3-methylsulfinylimidazo[1,2-a]pyrazin-8-amine;hydrate 2-[5-(4,6-diphenyl-1,3,5-triazin-2-yl)spiro[fluorene-9,9'-xanthene]-4'-yl]benzonitrile N-(4-acetylphenyl)-2,2-dichloro-3-(3,5-dimethoxy-4-nitrophenyl)cyclopropane-1-carboxamide 2-[(2,6-dimethylphenyl)iminomethyl]-5-nitrophenol 5-chloro-6-cyclopentyloxy-N'-hydroxypyridine-2-carboximidamide 4-methyl-2,3-dioxopyrazine-1-sulfonic acid (3-amino-5,6,7,8-tetrahydronaphthalen-2-yl)-methoxyphosphane 4-(2,3-dihydro-1H-inden-5-yl)-6-[2-methoxyethyl(pentanoyl)amino]pyridine-3-carboxylic acid 2-chloro-3-[(4-methoxybenzoyl)amino]-N-(3,3,5,5,8,8-hexamethyl-6,7-dihydronaphthalen-2-yl)benzamide 2-(1,3-benzodioxol-5-yloxymethyl)-5-[2-chloro-4-(trifluoromethoxy)phenyl]pyridine ethane;2-[(5-oxopyrazolidin-1-yl)methyl]-1,3-thiazole-4-carboxylic acid N-[1-[5-(3,5-dichlorophenyl)-4H-pyrazol-3-yl]ethoxy]aniline 2,2-dimethyl-6-(2H-triazolo[4,5-b]pyrazin-5-yl)spiro[1-benzofuran-3,4'-piperidine];ethane 4-[5-(1,3-dioxol-2-ylmethoxy)naphthalen-1-yl]sulfonyl-1-oxa-4,8-diazaspiro[4.5]decane 2-[5-(4-cyclohexylpiperazin-1-yl)pyrazin-2-yl]oxyacetic acid (2R)-1-(3,4-dihydroxyphenyl)-3,7-diethyl-5-methoxynona-6,8-dien-2-one 2-[(4S)-6-chlorospiro[3H-chromene-2,1'-cyclobutane]-4-yl]ethanamine 3-chloro-N-[2,4-difluoro-5-[(3E)-penta-1,3-dien-3-yl]phenyl]-2-hydroxybenzenesulfonamide;ethane N-[6-fluoro-1,3-benzoxazol-2-yl(phenyl)methylidene]hydroxylamine (Z)-3-[4-[2-bromoethyl(methyl)amino]phenyl]prop-2-enoic acid N-benzyl-6-(2,4-difluorophenyl)-5-oxohexanamide (2Z,4E)-2-cyano-5-[1-[2-methoxyethyl(propanoyl)amino]pyrrol-3-yl]penta-2,4-dienoic acid 7-chloro-2,3-dihydrothieno[3,4-b][1,4]oxazine-4-carboxylic acid;ethane 3-(2,5-dimethoxyphenyl)-4-[[6-methyl-1-[3-(trifluoromethyl)phenyl]sulfonylindol-3-yl]methylideneamino]butanamide N-[4-chloro-2,5-difluoro-3-(2-methylpropanoylamino)phenyl]-2-fluorobenzamide N-[(Z)-1-amino-3-(methylamino)prop-2-enylidene]-4-[2-(4-cyclopentylpiperidin-1-yl)ethoxy]-5-methylthiophene-2-carboxamide 4-[(7-azidoquinolin-2-yl)methoxy]benzenecarboximidamide 3-methyl-1-(4-methyl-2-phenylquinolin-7-yl)-4H-pyridin-2-one 2-benzylimino-5,8-dimethylchromene-3,4-dione 4-ethyl-5-methyl-2-[2-[(2S)-pyrrolidin-2-yl]phenyl]-1H-pyrimidin-6-one 1-N,1-N'-bis(phenylmethoxy)spiro[cyclohexane-1,2'-indene]-1'-carboxamide 3-[(1-azidosulfonylcyclopropyl)methylamino]-1H-indole N-[(1S)-2-hydroxy-2,3-dihydroinden-1-ylidene]hydroxylamine 3-[3-[3,5-dimethyl-4-(oxan-4-yl)pyrazol-1-yl]phenoxy]pyrrolidine-1-carboxylic acid 4-(2-hydroxyphenyl)-N'-[5,6,7-tris(sulfanylidene)-3H-thiopyrano[3,2-d]pyrimidin-2-yl]benzenecarboximidamide 4-amino-2-(1H-imidazo[4,5-b]pyridin-7-yl)benzenesulfonic acid 4-chloro-5-fluoro-2-[(3R)-1,1,1-trifluoropentan-3-yl]aniline 2-(3,4-dihydrochromen-2-ylidene)indene 3-[5,6-dichloro-4-(ethylamino)pyridin-2-yl]-N'-hydroxybenzenecarboximidamide N-[3-(1H-pyrazol-4-yl)phenyl]propanamide N-[3-(7,8-dimethoxy-2-oxochromen-3-yl)-1H-indol-5-yl]acetamide 2,3-dihydro-1H-indol-7-yl-[(3S,4R)-3-hydroxypiperidin-4-yl]methanone;hydrochloride 2-[2-[3,5-di(propan-2-yl)phenyl]ethyl]benzonitrile 6-(diethylamino)-3-methoxypyrazine-2-carboxamide 2-[4-azido-3,5-difluoro-6-(1H-indazol-4-ylamino)pyridin-2-yl]sulfanyl-N'-hydrazinylethanimidamide N-(2,4-dibromopyrimidin-5-yl)-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethanimine 2,6-ditert-butylthieno[3,4-d]pyrimidine (6-amino-3,5-dimethylpyrazin-2-yl)urea 2-hydroxy-5,7-dimethyl-3-(3-oxobutanoyl)pyrido[1,2-a]pyrimidin-4-one 3-(azidomethyl)-N'-(3-chlorophenyl)-5-methyl-4-oxoimidazo[2,1-d][1,2,6]thiadiazine-7-carbohydrazide 2-[1-[3,4-bis(phenylmethoxy)phenyl]ethyl]-1H-imidazole (4R)-3-methyl-1-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)piperidine 5-methoxycarbonylthiophene-3-sulfonic acid (4-fluorophenyl)-[4-[2-(3,4,5-trimethoxyanilino)pyrimidin-5-yl]piperazin-1-yl]methanone N-[1,4-dimethyl-2-(4-phenylmethoxyphenyl)-6,7-dihydrobenzimidazol-5-yl]-2,3-dihydroxypropanamide 2-[(3,4-dichlorophenyl)methylimino]-5-[5-[(2R)-3,3-dimethylbutan-2-yl]oxypentyl]-1,3-thiazolidin-4-one 4-[2-hydroxyethyl(nonanoyl)amino]benzenesulfonic acid (5Z)-1-(4-phenoxyphenyl)-5-[[3,4,6-trihydroxy-2-(3-methylbut-2-enoxy)phenyl]methylidene]imidazolidine-2,4-dione 5-(1H-indazol-4-yl)-N-[3-methoxy-2-[(2R)-oxan-2-yl]propyl]pyridine-3-carboxamide 1-(5-methyl-1H-imidazole-4-carbonyl)-N-phenylpiperidine-3-carboxamide (2S)-3-methyl-N-[4-(trifluoromethoxy)phenyl]pentanamide 6-(3,4-dimethylphenyl)-5-propanoyl-1,2-benzothiazole-3,7-trione 5-cyclohexyl-4-methoxy-2,3,6-triphenylpyridine 5-azido-2-[1-(1,3-benzodioxol-5-yl)cyclopropanecarbonyl]pentanoic acid 2-ethoxy-N-[4-(3-piperidin-1-ylpropoxy)phenyl]acetamide N-[4-cyano-2,5-bis(trifluoromethyl)phenyl]-3-(1,2-dihydropyridin-6-ylsulfanylamino)pyrrolidine-1-carboxamide 2-hydroxy-5-[(3-methyloxiran-2-yl)methoxy]benzaldehyde 3-(2,4-dichlorophenyl)-6-fluoro-7-[3-methoxy-5-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]azetidin-1-yl]quinazolin-4-one ethane;2-[[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)piperidine-1-carbonyl]amino]acetic acid [1-[4-(1,3-oxazol-5-yl)anilino]cyclobutanecarbonyl]azanium 4-(azidosulfanylmethyl)-1,2-difluorobenzene 2-methyl-4-[2,3,5,6-tetradeuterio-4-hydroxy-5-(trifluoromethoxy)phenyl]butanal 4-azidosulfonyl-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1H-pyrrole-2-carboxamide 2-(4-chlorophenyl)-1,3-diethyl-7H-imidazo[4,5-e]diazepine (3aR,9bR)-1-[2-cyclopropyloxy-5-(2,2,2-trifluoroethoxymethyl)benzoyl]-3,3a,4,9b-tetrahydro-2H-chromeno[4,3-b]pyrrole-5-carboxylic acid (2-aminophenyl)methylcarbamic acid 5-[(2,4,5-trifluorophenyl)methoxy]pyrimidine 2-[3-(trifluoromethyl)pyridin-4-yl]-5H-1,2,4-oxadiazole-3-thione 5-bromo-2,3-dimethylbenzenecarboximidamide 3,6-dihydroxy-2-[4-(4-hydroxyphenyl)cyclohexa-1,5-dien-1-yl]benzoic acid N-(3-methylbut-1-en-2-yl)-5-[3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-amine N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]naphthalene-2-carboxamide 2-[3,5-bis(trifluoromethyl)phenyl]-4-iodo-1H-benzimidazole 5-(6-propoxypyridin-3-yl)pyrazole-1-carboxylic acid N-(2,6-dimethylphenyl)-1-methoxy-4H-thiopyran-4-amine 2-amino-5-[4-(2,3-dichlorophenoxy)phenyl]phenol 1-[2-[3-(2,5-dimethylphenoxy)propoxy]ethoxy]ethanol 4-[1,3-benzodioxol-5-ylmethyl(butanoyl)amino]-2-[(2,6-difluorobenzoyl)amino]thiophene-3-carboxylic acid N-ethylformamide;2-fluoro-5-methoxy-4-[5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-2-yl(thiomorpholin-3-yl)amino]benzaldehyde [[6-(2-chlorophenyl)-5H-imidazo[1,2-a]pyridine-7-carbonyl]amino]thiourea 3-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-quinolin-2-one 3-ethyl-7,8-difluoroisoquinoline 5-[4-[(2E,4Z)-6-methoxyhexa-2,4-dien-3-yl]pyrazol-1-yl]pyridine-2-carboxylic acid N-[4-(3,5-difluorophenoxy)-2,3-dihydropyrido[3,4-b]pyrazin-6-yl]formamide 2-(cyclohexylmethyl)-6-oxo-N-pyridin-3-ylpiperidine-4-carboxamide 5-ethyl-2-[(3Z,4Z)-hexa-1,3,5-trien-2-yl]furo[3,2-b]pyrrole [2-(1,3-benzodioxol-5-yl)propanoylamino]carbamodithioic acid N-(2,3-difluorophenyl)sulfonyl-1-[[4-hydroxy-5-(trifluoromethyl)cyclohexa-2,4-dien-1-yl]carbamoylamino]pyrazole-3-carboxamide 5-bromo-1,2,3a,9b-tetrahydrocyclopenta[l]phenanthrene 3-[1-(4-methylphenyl)cyclopentanecarbonyl]oxycyclobutane-1-carboxylic acid N-[4-(aziridin-1-ium-2-yloxy)phenyl]acetamide 2-methyl-N-[1,3]benzothiazolo[5,4-d]pyrimidine-7-carboxamide 6-(4-ethoxy-2,3-difluorophenyl)-2,7-difluoro-1,4-dihydronaphthalene (4R)-6-bromospiro[2H-indene-3,4'-piperidine]-1'-one 6-amino-N-[4,5-dimethyl-2-(3-methylcyclohexa-1,5-dien-1-yl)pyrazol-3-yl]hexanamide 2,6-dichloro-N-[(E)-[4-(diethylamino)-2-hydroxyphenyl]methylideneamino]benzamide N-cyclopropyl-1-[(3R,4S)-3-hydroxypiperidin-4-yl]indole-5-carboxamide;hydrochloride N-[1-[2-(3,5-dichloropyridin-4-yl)-2-oxoethyl]piperidin-4-ylidene]-7,8-dihydronaphthalene-2-sulfonamide 2-[4-(3,5-dimethylpyridin-1-ium-1-yl)phenyl]-5H-phenanthridin-6-one;chloride (2S)-1-azidooxy-3-phenylpropan-2-ol N-[[2,4-dichloro-6-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-2-hydroxyacetamide 2-[4-chloro-3,5-dimethyl-N-(pyridin-3-ylcarbamoyl)anilino]acetic acid N-[6,7-difluoro-8-(2-hydroxyethylimino)-7H-quinolin-5-ylidene]hydroxylamine 2-methyl-5-[4-(3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazole-2-carbonyl)piperazine-1-carbonyl]benzonitrile 1-(3-aminophenyl)sulfonyl-N'-[2-(2-chlorophenyl)ethyl]-4,5-dihydroimidazole-4-carboximidamide N-(2,4-dimethylphenyl)-N-[(3R)-1-ethylpyrrolidin-3-yl]formamide;ethane 4-(N-tert-butyl-2,5-dichloroanilino)benzenesulfonic acid 3-(3,5-dichlorophenyl)-2-(dimethylamino)-N-ethylpropanamide 3-[(2R,4S)-1-[2-[2-[(5-chloropyrimidin-2-yl)amino]ethoxy]ethylsulfonyl]piperidin-2-yl]benzonitrile (1S,2R)-2-[6-methyl-4-[5-(trifluoromethyl)pyridin-3-yl]pyridin-2-yl]cyclohexan-1-amine 7-(2,6-dichlorophenyl)-12-[4-methoxy-3-(2-piperidin-1-ylethoxy)anilino]-5-thia-2,10,11,13-tetrazatricyclo[7.4.0.02,6]trideca-1(13),3,6,8,11-pentaen-12-one;ethane 3-fluoro-2-[1-(furan-2-ylmethyl)piperidin-4-yl]oxypyridine 1-[3,5-di(butan-2-yl)phenyl]-N-methoxymethanimine;rhodium 1-[4-(1,3-dimethylcyclohexylidene)butanoyl]-N-ethylindolizine-7-carboxamide 5-[[4-(2,3-dihydropyrrole-1-carbonyl)pyrazol-1-yl]methyl]-2,4-dimethyl-1H-pyrimidin-6-one N-(3,4-dimethoxyphenyl)-2-[6-oxo-5-(trifluoromethyl)-1H-pyrimidin-4-yl]acetamide (1S,3R)-2,2-dichloro-N-[4-chloro-3-[2-oxo-6-[4-(trifluoromethyl)piperidin-1-yl]-1H-pyridine-3-carbonyl]phenyl]-3-(3-chloro-5-propan-2-yloxyphenyl)cyclopropane-1-carboxamide 3-[(4,5-dichlorothiophene-2-carbonyl)amino]hexanoic acid 1-[(2S)-3-cyclohexyl-2-hydroxypropyl]-N-[[4-methoxy-6-(1,3-oxazol-5-yl)pyridin-3-yl]methyl]pyrazole-4-carboxamide;ethane (E)-4-(2,6-dimethylphenyl)-1-[5-ethenyl-3-[1-(4-methoxyphenyl)ethenyl]pyridin-4-yl]but-3-en-2-imine;ethane 4-[(3R)-1-acetylpiperidin-3-yl]-2,6-dimethylpyridine-3-carboxamide N-(3,4-dimethylphenyl)-2-[6-(furan-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]acetamide 6-(4-chlorophenyl)-2-methyl-1,3-diazinan-5-one;ethane N-[3-(2,6-dioxopiperidin-3-yl)-5-methoxy-4-oxo-1H-quinazolin-2-ylidene]pyridine-3-carboxamide N-(3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[b][1]benzoxepin-10-ylmethyl)-2-hydroxy-3-nitrosobenzamide (4S)-N'-[2-methoxy-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonylamino)propyl]spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,3'-piperidine]-4-carboximidamide 4-(5-bromopyrimidin-2-yl)oxy-3,5-dimethylcyclohexane-1-carboxylic acid 2-azidooxy-5-methoxy-1,3-dihydroisoindole 3-[4-[(2,6-difluorophenyl)methoxy]phenyl]propanoic acid (6-propanoyl-2H-indol-3-yl)iminothiourea (4-chlorophenyl)sulfonyl-[3-(2,5-dihydroxypyrrol-1-yl)propyl]azanium 5-(azidomethyl)-4,5-difluoro-2,3-dimethoxycyclohexa-1,3-diene 5-[3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]pentanoic acid 6-(4,5-dihydroimidazol-1-yl)pyridine-3,4-dicarbonitrile 5-(3,4-dimethylphenyl)-2-ethenyl-N-(iodomethyl)aniline 1-[2,3-difluoro-4-(trifluoromethyl)phenyl]ethanone 3-(4-phenylpiperazin-1-yl)propanoic acid;hydrochloride 3-[[(4,5-dichlorothiophen-2-yl)sulfonylamino]methyl]benzoic acid N-[(3R)-1,7-dimethyl-6-oxopiperidin-3-yl]-3,4,5,6-tetrahydro-2H-carbazole-9-carboxamide 5-[[(2R,3S)-2-[1-[2-[di(propan-2-yl)amino]acetyl]piperidin-4-yl]oxolan-3-yl]methoxy]pyridine-3-carbonitrile 1,4-dimethylpiperazine;7-(2-morpholin-4-ylethoxy)quinazoline 1-(3,4-dichlorophenyl)-2H-pyridine 5-amino-7-chloro-3-(2,4-difluorophenyl)-1H-1,6-naphthyridine-2,8-dione 4-[7-fluoro-2-(propylamino)quinazolin-6-yl]oxybutane-1,2-diol 5-bromo-2-[(6-methoxy-1H-imidazo[4,5-b]pyridin-2-yl)sulfanyl]phenol 1-N,3-N-bis(4-butanoylphenyl)benzene-1,3-dicarboxamide 2-(1,4,5-oxadiazole-3-carbonyl)-3,4,6,7,8,9-hexahydropyrido[1,2-a]pyrazine-1-carboxamide N-ethyl-2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide N-[5,7-dimethyl-3-[(2-phenylethylamino)methyl]pyrazolo[1,5-a]pyrimidin-6-yl]formamide 2-(3-bromophenyl)-4-chloropyrazole N-[3-(2,4-difluorophenyl)oxan-3-yl]pyrazine-2-carboxamide N-[6,6,6-trifluoro-5-(2-methylphenyl)hexyl]-2H-benzotriazol-5-amine 2-[5-(5-aminopyridine-3-carbonyl)cyclohepta-1,4,6-trien-1-yl]benzonitrile 7-chloro-4,5-dimethyl-1-benzothiophene-2,3-dione N-[3-[4-(1,2-dimethylimidazol-4-yl)sulfonylpiperazine-1-carbonyl]phenyl]-5-nitrofuran-2-carboxamide 2,5-difluoro-N-[2-(4-hydroxyoxolan-3-yl)ethyl]benzenesulfonamide 3-[4-amino-6-(trifluoromethyl)pyridin-1-ium-2-yl]oxypiperidine-1-carboxylate N-[(Z)-3,3,6,6-tetramethyl-5-nitrohept-4-enyl]pyridine-2-carboxamide 1-(2,4-dimethylthiophen-3-yl)-N-[(5-oxo-1,4-oxazepan-6-yl)sulfonyl]cyclobutane-1-carboxamide N-(2,4-dimethylphenyl)-3-[2-[[1-[6-(4-hydroxyphenyl)pyridin-2-yl]pyrrolidin-3-ylidene]amino]ethoxy]benzamide 3-[2,4-difluoro-5-[2-(hydroxyamino)pyrimidin-4-yl]phenyl]propanoic acid (2R)-4-[2-chloro-5-fluoro-3-(3-methylpyridin-2-yl)phenyl]pentane-1,2-diol (2E,4Z)-4-[3-(dimethylamino)propoxy]-N-methyl-2-methylsulfanyl-6-methylidene-5-[4-(2-phenoxyethyl)piperazin-1-yl]hexa-2,4-dienamide 1-methyl-7,8-dihydroindeno[2,3-b]pyrazine;7H-purin-6-amine 3-(4-chlorophenyl)-5-cyclopropyl-1-[(E)-2,3-dihydroxy-1-phenylbut-1-enyl]pyrrolidine-2,4-dione ethane;2-(3,5,6-trimethylpyridine-2-carbonyl)oxybenzoic acid 6-[4-[2,4-bis(4-fluorophenyl)imidazol-1-yl]phenoxy]-5-methylidenecyclohexa-1,3-dien-1-ol 3-cyclopropylsulfonylquinoline 4-(3,5-dimethylphenyl)-N-(3,5-dimethylpyridin-2-yl)piperidine-1-carboxamide 3-[(2R)-6,8-dichloro-2-methyl-9-phenylnonan-4-yl]oxypropane-1,2-diol (5R,7S)-N-[2-(1H-imidazol-5-yl)ethyl]-N-methyl-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide N-[2-(3,5-dimethylphenyl)ethyl]-N'-hydroxypyridine-4-carboximidamide 3,7-dihydroxy-N-(2-hydroxyethyl)-4H-chromene-2-carboxamide (Z)-2-[3-[3,5-difluoro-4-(1-methoxycarbonylpiperidine-2-carbonyl)phenyl]pyridin-4-yl]-3-iminoprop-1-enyl]azanide 2-(3,5-dimethoxyphenyl)-4H-quinazoline (5E)-2-cyclopentylimino-5-[(4-fluorophenyl)methylidene]-1,3-thiazolidin-4-one 5-(4-ethylphenyl)sulfonyl-2-(2H-tetrazol-5-ylmethoxy)benzonitrile (E)-3-[4-[2,6-difluoro-N-methyl-3-[(E)-4-oxobut-2-enoyl]anilino]phenyl]prop-2-enal 6-azido-2,3,7-trimethylquinoline 6-butanoyl-2,3-dimethyl-5H-pyrimidin-4-one N-(5-chloropyridin-2-yl)-3-[2-[4-ethyl-6-(propan-2-ylamino)pyrimidin-5-yl]ethynyl]benzamide 5-(3,4,5-trimethoxyphenyl)pentanedinitrile N-[[(2S,3aS)-5-(oxan-4-yl)-1,2,3,3a,4,6,6a-octahydropentalen-2-yl]methyl]thieno[2,3-b]pyridine-3-carboxamide (3S,4R)-3-[4-amino-5-[(2R)-2-methyl-3-phenoxypropoxy]imidazo[5,1-f][1,2,4]triazin-7-yl]hexane-1,4-diol 4-(1-aminoethenyl)-2,5-dibromophenol N-[2-(1H-benzimidazol-2-yl)ethyl]-3,5-dibromopyrazolo[1,5-a]pyrimidin-7-amine 2-amino-4-(2,5-difluoro-6-hydroxyphenyl)-4H-pyran-3,5-dicarbonitrile N-[3,5-bis(trifluoromethyl)phenyl]-2-cyclopropylidene-1-hydroxy-7-methyl-6-oxo-5H-cyclohepta[b]pyrrole-3-carboxamide [1-(3-hydroxy-5-methylpiperidine-1-carbonyl)pyrazol-4-yl]-[2,2,6-trimethyl-4-[1-[3-(oxan-4-ylamino)pyridin-2-yl]oxybutyl]piperazin-1-yl]methanone 4-[5-(2-propan-2-ylsulfonylethylsulfanyl)pyrazin-2-yl]-1,3-thiazole [3-(5,6-dimethylpyrimidin-4-yl)oxypyrrolidin-1-yl]-(2-imidazol-1-ylphenyl)methanone 2-[4-(difluoromethoxy)-3-fluorophenyl]acetonitrile 3-[1,2,4-triazol-4-yl(1,3-thiazol-5-yl)amino]propanoic acid 3,4-dichloro-2-phenoxyaniline N-[1-methylsulfonyl-4-(trifluoromethoxy)cyclohexa-2,4-dien-1-yl]pyrimidine-5-carboxamide 2-[2,5-bis(trifluoromethyl)anilino]-5-cyclopropyl-4-phenyl-1H-pyrimidin-6-one [3-amino-2-[4-(pyridine-4-carbonyl)phenyl]prop-1-enyl]-[2-[(2R,6S)-6-azidooxan-2-yl]ethoxymethylidene]azanium 5-(2-cyclopentylethynyl)pyridine-3-carboxylic acid 5-chloro-2,4-difluoro-N'-(5,6,7,8-tetrahydronaphthalene-1-carbonyl)benzohydrazide 1-(1-azidooxypropan-2-yl)-4-phenylpiperidine (2-chloropyridin-4-yl)-[3,5-diamino-6-(1H-indol-3-yl)pyrazine-2-carboximidoyl]azanium 1-(7,9-dihydropurin-6-yl)-2-methoxyethanone 1-[2,6-di(propan-2-yl)phenyl]-3,4-bis[3,5-di(propan-2-yl)pyrazol-1-yl]-5-methylpyrrole-2-carbonitrile 2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-methylpyridine-4-carboxylic acid 3-(2,6-dimethylphenyl)benzenesulfonic acid;ethane (E)-3,4,5-trihydroxy-N-[2-(4-phenoxyphenyl)ethyl]benzamide [4-(2,6-difluorophenyl)sulfanylpiperazin-1-yl]-(3-phenylpyridin-4-yl)methanone 1-azido-2,3,4,5-tetrachloro-6-(9H-fluoren-1-yloxy)benzene 2-[1,3-dihydroxy-4-(2-phenylethyl)isoindole-6-carbonyl]-3,4,5,6-tetrafluorobenzenesulfonate (1S,3R,4R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-4-hydroxy-3-methoxycyclohexane-1-carboxamide 1-[3-(4-fluorophenyl)propyl]azetidine;formic acid 2-hydroxy-4-[3-(1,1,2,2,2-pentafluoroethyl)phenyl]-N'-pyridin-3-ylbenzohydrazide 2-[3-methyl-5-(3-morpholin-4-ylpropoxy)phenyl]benzo[g][1,3]benzothiazole 1-chloro-7-methylsulfonylphenanthrene 1-[[6-(5,5,8,8-tetramethyl-2,3,4a,9b-tetrahydroindeno[1,2-b]pyridin-10-yl)-1H-benzimidazol-2-yl]oxy]ethanol N-(2-methylprop-1-enoxy)methanamine;1-[3,4,5-tris[(E)-pent-1-enyl]phenyl]pyrrolidine 6-[2-(3,4-dimethoxyphenyl)ethynyl]-5H-cyclopenta[d]pyrimidine 2-[(3-chlorophenyl)sulfonylamino]-N-(4-ethylcyclohexa-1,5-dien-1-yl)acetamide N-[(2S)-3-methylbutan-2-yl]-4-phenyldiazenylbenzamide 3-(5,5-dimethylcyclohexa-1,3-dien-1-yl)-2,6-difluoroaniline (2R,4S)-N-[(3aR,6aS)-5-hydroxy-1,3,3a,4,6,6a-hexahydrocyclopenta[c]pyrrol-2-yl]-4-(4-bromophenyl)sulfonylpiperidine-2-carboxamide [1-(2,4-dichlorophenyl)cyclohexyl]carbamic acid 2-[4-[3-(3-chloro-4-fluorophenyl)-5,5-dimethyl-4H-pyrazol-1-yl]anilino]-N-(3,5-dihydroxy-5-methylhexan-2-yl)acetamide 4-N-[5-[3-(2,4-dichlorophenyl)propyl]-1H-pyrazol-3-yl]benzene-1,4-diamine 2-(1,3-benzothiazol-2-ylsulfanyl)-N-[(Z)-(4-hydroxyphenyl)methylideneamino]acetamide 3-[2,6-dibromo-4-(1,2-oxazol-5-yl)phenyl]sulfanyl-4H-1,2,4-oxadiazol-5-one (4S)-1'-ethylsulfonyl-1-methyl-N-(3-oxocyclohexen-1-yl)spiro[5,7-dihydropyrazolo[3,4-b]pyridine-4,3'-indole]-2'-carboxamide 2-[(2,4-difluorophenyl)methyl]-4-(hydroxymethyl)-5-sulfanylidene-1H-pyrazol-3-one 2-[1-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)piperidin-3-yl]acetamide [6-[2-ethyl-4-(1,2,4-triazol-4-yl)phenoxy]pyridin-3-yl]methanamine 1-phenylsulfanyl-2H-pyrimidine (6S)-5-[3-(4,6-diphenylpyridin-2-yl)oxybutyl]-6-ethylidenecyclohexa-1,3-dien-1-ol 5-methoxy-1,3-dimethylthieno[2,3-c]pyrazole-4,6-dione N-(4-oxo-2,3-dihydrochromen-7-yl)acetamide 2-(3,4-dibromophenyl)-1,3-benzothiazole N-(5-tert-butyl-1H-pyrazol-4-yl)-2-oxospiro[1H-indole-3,1'-cyclohexane]-6-carboxamide 2-[4-(5-bromopyrimidin-4-yl)piperazin-1-yl]-N,N-diethylethanamine;ethane 6-amino-4-[2,5-dimethyl-3-(trifluoromethoxy)phenyl]-4-methyl-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile 1-[(2S)-4,4-difluoro-2-methylpyrrolidin-1-yl]-3-[4-(2-methoxyphenyl)piperazin-1-yl]propan-1-one 1-azido-2,3-bis(4-methoxyphenyl)benzene 4-cyclopentyloxy-N-(3-ethynyl-4-methoxyphenyl)pyrimidin-2-amine 1-[4-[2,3-dimethyl-7-(3-methylphenyl)-2H-imidazo[1,5-a]pyrimidin-8-yl]piperazin-1-yl]propan-1-one;hydrochloride 4-[(5R)-3,6-diazabicyclo[3.2.0]heptan-3-yl]-3-methoxyaniline 1-benzyl-2,5-dimethoxybenzimidazole ethane;[1-[[4-[2-fluoro-3-(3-phenylpropoxy)phenyl]pyrimidin-2-yl]methyl]cyclohexyl]carbamic acid N-[1-(2,6-dichlorophenyl)ethenyl]ethanimine;ethane [3-amino-5,7-dichloro-2-(pyridine-4-carbonyl)indol-1-yl]sulfonylazanium 3-[(3S)-1-methyl-2,4-dioxo-3H-quinoxalin-3-yl]propanamide ethane;2-[4-(3-methylbutyl)phenyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine 3-(4-bromophenyl)-6-fluoro-3-methyl-1H-indol-2-one (E,2R)-4-[4-(cyclopropanecarbonylamino)phenyl]-2-methylbut-3-enoic acid (4R,5S)-2-[3-[5-(2-hydroxyethoxymethyl)pyridin-3-yl]phenyl]-6-oxaspiro[2.5]octane-7-carboxylic acid 1-methyl-5-phenylpentane-1,3-dione 5-[1-[5-bromo-4-(2,3,5-trichlorophenyl)pyridine-2-carbonyl]azetidin-3-yl]oxypyrimidine-2-carboxylic acid 1-[(3R,4S)-3-fluoropiperidine-4-carbonyl]-N-methyl-N-propan-2-yl-6-pyrazol-1-ylindazole-5-carboxamide N'-[4-(1,3-benzothiazol-2-ylsulfanylmethyl)-6-phenoxypyrimidin-5-yl]ethane-1,2-diamine 2-amino-N-[(5S)-3,4,4a,5-tetrahydro-1H-cyclohepta[c]pyridin-5-yl]-6,7,8,9-tetrahydro-5H-cyclohepta[d]pyrimidine-7-carboxamide 1-[3-[2-hydroxypropan-2-yl(methyl)amino]propoxy]anthracene-9,10-dione 3-cyclohexa-1,5-dien-1-ylpropanal;N-[(2Z)-5-methylhexa-2,4-dienoxy]-4-thiophen-2-ylaniline 5-bromo-2,3,4-trimethylbenzaldehyde 1-(2,3-dihydrofuro[2,3-b]pyridine-4-carbonyl)pyrrolidine-3-carboxamide 3-azidooxy-1,2,4,5-tetrafluorobenzene (2Z)-N-[1-(4-chloroanilino)ethenyl]-N,3-dimethylpenta-2,4-dien-1-amine 6-[4-(cyclopropylamino)piperidine-1-carbonyl]pyridine-3-carbonitrile 3-(4-methoxyphenyl)sulfonylpyridine 3,4-diphenyl-5-propylpiperidine 3-[2-hydroxyethyl-(6-sulfonaphthalen-1-yl)amino]butanoic acid (Z)-N-[(5S)-3,8,10-triazatricyclo[7.4.0.02,7]trideca-1,9,11-trien-6-yl]ethanesulfonamide 4-chloro-2-[(1,1-dioxothian-4-yl)amino]-5-(propylsulfamoyl)benzoic acid 3-[1-[4-(benzylamino)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-4-yl]propanal 5-[(2,4-dioxoquinazolin-1-yl)methyl]triazole-4-carboxylic acid 4-fluoro-2-N-[3-fluoro-5-(trifluoromethyl)phenyl]-7-N,6-N,7-N-trimethyl-1H-benzimidazole-2,7-diamine [6-fluoro-1-(3,4,5-trifluorophenyl)indol-3-yl]sulfanium N-(3-ethoxyphenyl)-6-(methylaminosulfanyl)-1,2,3,4-tetrahydronaphthalen-1-amine N-[2-methoxy-5-(1,3-oxazol-4-yl)phenyl]-5-oxo-2H-pyrrole-3-carboxamide (2-butylphenyl)-[5-chloro-4,6-dimethoxy-7-(3-piperidin-1-ylpropoxy)-1H-indol-2-yl]methanone N-[1-amino-3-(hydroxymethyl)pentan-2-yl]-4-morpholin-4-ylbenzamide;ethane 2-(azidomethyl)-5-phenoxypentan-1-ol N-[1-[4-(5,5-difluoropentyl)phenyl]ethenyl]-4-methoxy-3-[(E)-2-nitroethenyl]aniline 1-[(5R,7S)-3-chloro-5-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidin-7-yl]pyrazole-4-carboxylic acid (3S)-N'-[2-fluoro-4-iodo-6-methyl-3-(1H-pyrazol-5-yl)phenyl]-1-phenylpyrrolidine-3-carbohydrazide [4-(aminomethyl)phenyl]-[3-[4-[hydroxy(phenyl)methylidene]piperidin-1-yl]propyl]azanium 5-[4-(N-tert-butylanilino)phenyl]-2-hydroxybenzoic acid 4-[2-methylpropanoyl(1,3-thiazol-5-yl)amino]benzoic acid 1-(5,6-dimethylcyclohexa-2,4-dien-1-yl)-3-[(Z)-1H-indol-3-ylmethylideneamino]urea 1-phenyl-2H-thieno[2,3-d]pyrimidine 3-[(Z)-2-nitroethenyl]thiophene-2-sulfonic acid N-[3-[5-(2,4-difluorophenyl)pyrazolo[1,5-a]pyrimidin-3-yl]propyl]-2,6-bis(trifluoromethylsulfonyl)benzamide N-(2,4-difluorophenyl)-6-methoxyquinoline-8-carboxamide 4-[4-[[5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazol-4-yl]methoxy]-1-methylpyrazol-3-yl]pyridine-2-carbonitrile 3-(diethylamino)-1-(3,5-dimethoxyphenyl)propan-1-one;1-[4-(4-hydroxybenzoyl)piperazin-1-yl]ethanone 2-N-cyclopropyl-6-methoxy-4-N,4-N-dipropylpyridine-2,4-dicarboxamide 4-(aminomethyl)-1-[5-chloro-6-methoxy-2-(3,3,3-trifluoropropoxy)pyridine-3-carbonyl]pyrrolidin-2-one N-[1,3-di(propan-2-yl)-5-pyridin-4-ylpyrazol-4-yl]benzenesulfonamide 4-amino-N-[2-(4-chlorophenyl)ethyl]pentanamide 4-(N-(2,4-dichloropyrimidin-5-yl)-3-nitroanilino)benzenesulfonamide 2-[(3S)-7-bromo-1,4-dimethyl-5-oxo-2-phenyl-2H-pyrido[3,4-e][1,4]oxazepin-3-yl]acetic acid 2,7-dipyridin-4-ylthieno[3,2-c]pyridine [4-(6,7-dihydro-5H-cyclopenta[c]pyridin-2-yl)phenyl]methanamine;propane 1-cyclohexyl-3,6-dimethoxypyrrolo[2,3-b]pyridine 2-(2,6-dichloroanilino)-7-fluoro-4-methoxyquinoline-3-carboxamide (5Z)-2-[5-chloro-1-(4-hydroxyphenyl)ethylidene]heptanoic acid 5-(azidomethyl)-3,7-dichloro-2H-isoquinolin-1-one 2-(2-ethoxyphenyl)sulfonyl-N-[4-fluoro-3-(trifluoromethyl)phenyl]acetamide 1-(4,4-difluorocyclohexyl)-6-[3-[(4,4-dimethyl-2-oxopentanoyl)amino]phenyl]pyrazolo[3,4-b]pyridine-3-carboxylic acid 1-[(Z)-2,3-dihydro-1H-1,5-naphthyridin-4-ylideneamino]pyrrole-2-carbonitrile 2-[4-(3,5-dimethylphenyl)piperazin-1-yl]butanamide N-(cyclopentylmethyl)-2-[2-[(1R)-3,4-dihydro-1H-isochromen-1-yl]ethoxy]-6-[2-[4-(hydroxyamino)phenyl]propan-2-yl]pyridine-4-carboxamide 5-(5-pyridin-3-yl-1H-indazol-3-yl)-N,4-dipropoxypyridine-2-carboxamide (E)-4,5-dimethyl-N'-[1-(2-phenylphenyl)ethenoxy]oct-3-enimidamide N-methyl-2-[6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]propanamide 7-[6-bromo-3-(2,5-dichlorophenyl)sulfonylhexanoyl]-9H-fluorene-1-sulfonate (1S,3R,4R)-3-[(2-hydroxyphenyl)methylamino]-N-[2-(2H-triazol-4-yl)ethyl]-4-propoxycyclohexane-1-carboxamide 2-(4-fluorophenyl)sulfanylbenzoic acid N-[(2-hydroxyphenyl)methyl]-N-methylmethanesulfonamide (2S)-3-ethoxycarbonyloxy-1-oxo-5-thiophen-2-yl-6,7-dihydrobenzo[c]isoquinoline-8-carboxylic acid 2-(2-chlorophenyl)-N-[4-[4-(trifluoromethyl)phenoxy]phenyl]acetamide (E)-3-cyclopropyloxy-2-methanimidoyl-1,4,5,6-tetrahydrophenalene-9-carboxamide 7-bromo-4,6-dichloro-1H-pyrazolo[4,3-c]pyridine N-[(2R,3S)-1-(4-methylphenyl)sulfonyl-5-oxo-2-pyridin-3-ylpyrrolidin-3-yl]propane-1-sulfonamide 2-(4,5-diethyl-3-pyridin-4-yl-1H-pyrrol-2-yl)propanenitrile 2-amino-3-[(6-methylpyridine-3-carbonyl)amino]propanoic acid (E)-3-amino-2-(4-phenylbutyl)prop-1-en-1-ol (2Z)-3-chloro-1,6,7-trimethyl-2-[(4-nitrophenyl)hydrazinylidene]quinoline 1-(3,4-dimethylphenyl)-N'-hydroxyimidazole-2-carboximidamide (3S)-1'-methylsulfonylspiro[1H-indole-3,4'-5,7-dihydropyrazolo[3,4-b]pyridine]-2,6'-dione 4-N,4-N-diethyl-2-(2-methoxyethyl)quinazoline-2,4,6-triamine 4-(4-fluorophenoxy)-3,3a,5,6,7,7a-hexahydro-2H-furo[3,2-b]pyridine 2-(2,3-dimethylpyridin-1-ium-1-yl)-5-nitrobenzoic acid 1-[3-(2-chloroanilino)pyrido[4,3-b]pyrazin-6-yl]-3H-indole-3-carboxamide (4R,6S)-1,2,4,5,6,7-hexamethyl-3,4-dihydroquinoline;6-(4-phenoxyanilino)-1H-pyridin-2-one 2-[3,4,5-trimethoxy-N'-(methylideneamino)-6-(6-phenoxypyridin-2-yl)iminopyridin-2-yl]acetonitrile [4-[(2,3-dichlorocyclohepta-1,3,6-trien-1-yl)methoxy]phenyl]methanol 4-[(3aR,7aS)-2,3,5,6,7,7a-hexahydropyrrolo[3,2-b]pyridine-1-carbonyl]pyrazole-1-sulfonamide 2-[(4-chloro-3,5-difluorophenoxy)methyl]-1-(2,6-diethoxyphenyl)imidazole 1-[1-(5,7-difluoroquinazolin-4-yl)piperidin-3-yl]propan-2-amine 1-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-[1-(4-chloro-6-cyclopropyloxypyridin-2-yl)ethylideneamino]azetidine-3-carboxamide 6-(2-hydroxyphenyl)-3-methylsulfanyl-7H-[1,2]oxazolo[5,4-b]pyridin-4-one N'-[(E)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-N-propan-2-yloxamide 5-[4-(2-hydroxyethyl)piperazin-1-yl]-N'-[[3,5,7,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,8,11-hexaen-13-ylidene(phenyl)methyl]amino]pyridine-2-carboximidamide (2S)-3-[8-(5-aminopentylsulfonyloxy)-1,4-dimethyl-2-oxoquinolin-6-yl]-2-methylpropanoic acid 7-(4-chlorophenyl)spiro[6H-imidazo[1,2-a]pyrimidine-5,3'-pyrrolidine] 5-[1-(2,4-difluorophenyl)cyclopentyl]oxycarbonyl-3-methyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-4-carboxylic acid 5-fluoro-2-[5-(methoxymethyl)pyrimidin-4-yl]pyridine 1-[4-(azidomethyl)phenyl]-3,5-bis[2-(diethylamino)ethoxy]benzene 3-(4,5-dihydro-1H-imidazol-2-yl)-1,6-dimethylindole 2-amino-N,N-diethylquinoline-3-carboxamide 2-ethyl-N'-hydroxy-6-(trifluoromethoxy)benzenecarboximidamide (4S)-5-[3,4-bis(2-methylpropoxy)phenyl]-2-imino-1,3-thiazolidin-4-one N-(4-bromophenyl)-2-[7-(4-methoxyphenyl)-6-methyl-2-oxo-1,3-dihydroimidazo[1,2-b]pyrazol-3-yl]acetamide 3-[6-[1-(1-methoxybutyl)pyrazol-4-yl]pyrazolo[4,3-b]pyridin-2-yl]propanenitrile 2-bromo-N-(8-chloro-4,5-dihydrothieno[3,2-d][1]benzoxepin-6-ylidene)hydroxylamine N-[1-[2-(methylamino)-2,3-dihydrothiophene-5-carbonyl]piperidin-4-yl]-4-propan-2-ylbenzamide 1-(4-butylphenyl)-3-(2,2-dichlorocyclohexyl)-1,3,8-triazaspiro[4.5]decan-2-one 1-azido-2-(2,4-difluorophenyl)piperazine 6-[(2Z,4E)-2-methyl-1-phenylhexa-2,4-dien-3-yl]-8,9,10,11-tetrahydrophenanthridine ethane;4-(4-methyl-3,5-dihydro-2H-1,4-benzoxazepine-7-carbonyl)benzonitrile 2-[1-[4-(1,3-benzothiazol-6-ylamino)pyrimidin-2-yl]piperidin-4-ylidene]propanedinitrile 7,8-dichloro-N',N'-diethyl-6-fluoroquinoxaline-2-carbohydrazide 3-[[4-[2-[(5R)-4-amino-5,6,7,8-tetrahydroquinazolin-6-yl]ethynyl]-3-fluorophenyl]methyl]-1,3-oxazolidin-2-one 4-[1-[2,5-difluoro-3-(trifluoromethoxy)phenyl]ethylamino]pyrrolo[1,2-b]pyridazine-3-carboxamide 7-[2-methoxy-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoyl]-8a-methyl-1,5,6,8-tetrahydro-[1,3]oxazolo[3,4-a]pyrazin-3-one N'-(4,5-diphenyl-1H-imidazol-2-yl)propane-1,3-diamine 7-chloro-1-[2,6-difluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyrido[2,3-d]pyrimidine-2,4-dione N-(3,4-dimethoxyphenyl)-2-[(6R)-5-oxo-2-phenyl-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 2-[5-(3,4-difluorophenyl)-1H-indol-2-yl]ethanamine 2-cyclopentyloxy-1,4-dimethylbenzene;ethane (5R)-5-[2,4-bis(phenylmethoxy)-5-propan-2-ylphenyl]-4,5-dihydro-1H-imidazol-2-amine N-(2-aminophenyl)-4-[2-[3,5-difluoro-4-hydroxy-6-(4-methoxyphenoxy)oxan-2-yl]ethynyl]benzamide 5-[4-(2,6-dimethylphenyl)piperazine-1-carbonyl]piperidin-2-one 2-[5-[[4-[4-(2,3-dihydrothiophen-5-yl)phenyl]phenoxy]methyl]furan-2-yl]-1H-imidazole 1,2-diamino-4-[3-bromo-5-chloro-2-methoxy-6-(trifluoromethyl)phenyl]-6-oxopyridine-3,5-dicarbonitrile N-[3-(1H-indol-6-ylmethylamino)propyl]-2-oxoethanesulfonamide N-methyl-1-[2-[(4R)-4-phenylcyclohexyl]-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl]piperidin-4-amine 2-[(4R)-1-acetyl-6-(4-cyanophenyl)-3,4-dimethyl-2-oxopiperidin-3-yl]-N-[5-chloro-4-fluoro-3-(trifluoromethyl)pyridin-2-yl]-2-(6-fluorocyclohexa-1,5-dien-1-yl)propanamide N-(4-azidooxyphenyl)-2,3-dihydro-1H-inden-5-amine [(2S)-3-(4-chlorophenyl)pyrrolidin-2-yl]methanol N-benzyl-4,6-bis(trichloromethyl)cyclohexa-1,3-dien-1-amine 5-[[4-(2,3-dichlorocyclohexyl)oxyphenyl]methylidene]-2-imino-1,3-thiazolidin-4-one (2R)-N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-2-(4-ethylphenoxy)propanamide [3-[2,4,6-trihydroxy-3-(hydroxymethyl)phenyl]phenyl]phosphonic acid [7-(cyclopentylmethylamino)naphthalen-2-yl]urea 2-(N-benzyl-4-methoxyanilino)octanoic acid 2-(1,3-benzothiazol-2-yl)cyclopenta-1,4-dien-1-amine 3-butoxy-N-[2-(cyclopropylmethyl)pentanoyl]benzamide 4-[4,5,6-trichloro-3-(trifluoromethyl)pyridin-2-yl]sulfonylbutanoic acid N-[(1R)-1-(4-fluorophenyl)ethyl]-2-oxo-5,6,7,8-tetrahydro-3H-furo[3,2-c]azepine-4-carboxamide N-[2-(2,3-dihydroindol-1-yl)ethyl]-1',3',3'-trimethylspiro[5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-a]azepine-7,4'-piperidine]-4-amine;dihydrochloride 1-[[(2E,4Z)-hexa-2,4-dienyl]amino]naphthalene-2,5-disulfonic acid (2R)-4,8-dihydroxy-1-phenyloctane-2,3,5-trione 2-methyl-6-[4-(4-propan-2-ylphenyl)sulfonylpiperazine-1-carbonyl]-3H-isoindol-1-one (2S)-1-[3,4-bis(methoxycarbonyl)anilino]-N-(cyanomethyl)-5-methylpyrrolidine-2-carboxamide;hydrochloride N'-(4-tert-butylphenyl)-2,5-dimethylpyrazole-3-carbohydrazide 1-[2,3-di(propan-2-yl)phenyl]-4-methylpiperazine N-azido-4,6-dichlorothieno[2,3-d]pyrimidin-2-amine 2-(3,4-dimethoxyphenyl)-N'-hydroxypyrazolo[1,5-a]pyrimidine-7-carboximidamide 5-(3-cyclobutyl-2H-indazol-7-yl)pyrimidin-4-amine 2-(3,4-dimethylcyclohexyl)-1H-benzimidazole 2-[4-(1,3-benzothiazol-6-yl)-5-(6-morpholin-4-ylpyridin-3-yl)oxypyridin-2-yl]acetonitrile 1-(4,7-dichloroquinolin-2-yl)-N'-[5-methoxy-6-(trifluoromethylsulfonylamino)pyridin-3-yl]-1-propan-2-ylpiperidine-4-carboximidamide [6-(3,4-dimethoxyphenyl)-5-oxobenzo[c][2,7]naphthyridin-8-yl]boronic acid [1-hydroxy-2-(methylamino)ethyl]-phenylazanide 4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]benzonitrile 3-[1-amino-2,2-dimethyl-6-(trifluoromethyl)-3H-pyridin-4-yl]oxybenzonitrile 2-(dimethylphosphorylmethyl)-7,9-diethoxypyrido[1,2-a]indole N-[2-(dimethylamino)ethyl]-3-fluoro-5-morpholin-4-yl-N,2-di(propan-2-yloxy)benzamide 1-(2,6-diethylphenyl)-4-(trifluoromethyl)imidazole 2-[4-[1-(3,5-dimethoxyanilino)-5H-pyrrolo[2,3-b]pyrazin-6-yl]phenyl]ethanol 6,7-difluoro-4-(2-methoxyethylamino)quinoline-3-carboxylic acid N-(3,3-difluorocyclobutyl)-2-(1,2,4-triazol-1-ylmethyl)morpholine-4-carboxamide 2-[N-(4-chlorobutyl)-4-nitroanilino]acetic acid [[1-(2,3-dihydroindole-1-carbonyl)cyclopropyl]methylideneamino]urea 6-[(4R)-1-benzyl-3,4-dimethylpyrrolidin-3-yl]pyridine-2-carbonitrile 1-[(2R,5S)-4-azido-2,5-dimethylpiperazin-1-yl]-3-phenylpropan-1-one (3S)-4,4-dimethyl-7-phenylnonanoic acid 2-[5-(1,2,4-triazol-1-yl)pentoxy]butanoic acid 2-[azido(diphenyl)methyl]sulfanylnaphthalene (3E,5Z)-3,4-dimethylocta-1,3,5,7-tetraene;N-[(2R)-3,3-dimethylbutan-2-yl]-2-nitro-1H-imidazole-5-carboxamide 1-[(2,6-difluorophenyl)methyl]-4-[2-(1H-indol-5-yl)ethynyl]pyridin-2-one (5S)-2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-4,7-dioxo-N-[3-(trifluoromethoxy)phenyl]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 3-methyl-5-[[2,3,4-trifluoro-6-(4-propylcyclohexen-1-yl)phenyl]diazenyl]phenol 2-(3,5-diaminophenoxy)-N'-hydroxybenzimidazole-1-carboximidamide 4-methyl-2-[3-(2,2,5,5-tetradeuteriopyrrolidine-1-carbonyl)phenyl]phthalazin-1-one N-[(2-methylpropanoylamino)carbamothioyl]benzamide 2-[[5-(dimethylamino)-3,4-dihydropyridin-2-yl]amino]ethanol;ethane 5-(6-azido-3-methylpyridin-2-yl)oxypyrimidine 2-[2,3-dihydroxypropyl(pyridin-4-yl)amino]acetamide 2-amino-8-(cyclopropylmethoxy)-4-[(4,6-dimethylpyrimidin-2-yl)methyl]-N'-ethyl-7H-pteridine-6-carboximidamide 3-(4-methylphenyl)-2-phenyl-7,8-dihydroquinoline;1-methylpyrrolidine (7R)-2,4-dimethyl-7-[3-(trifluoromethoxy)phenyl]-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidine N-[2,5-dichloro-4-(trifluoromethyl)phenyl]-3-oxobutanamide N-[3-[2-hydroxy-4-(1H-imidazol-5-yl)phenyl]oxolan-3-yl]acetamide 2-[4-(1H-benzimidazol-2-ylmethylideneamino)phenyl]sulfanyl-N,N-diethylacetamide;hydrochloride 4-chloro-5,7-dimethoxy-2-[[3-(trifluoromethyl)phenyl]sulfonylamino]quinoline-6-carboxylate ethane;(2Z,4Z)-N-[[3-methoxy-5-(methylamino)phenyl]methyl]-2,3-dimethylhexa-2,4-dienamide 2-[(Z)-6,7-dimethylnon-3-enoxy]carbonylbenzoate 2-[(1S)-1-[4-amino-3-methanimidoyl-5-[(1R)-6-methoxy-2,3-dihydro-1H-indene-1-carboximidoyl]anilino]ethyl]-3H-quinazolin-4-one 4-[3-bromo-2,6-difluoro-5-(trifluoromethyl)phenyl]-1,5-dihydropyrazole 2-[4,5-bis(4-chlorophenyl)-1H-imidazol-2-yl]phenol 4-[(Z)-[5,7-dihydro-4H-thieno[2,3-c]pyran-5-yl(phenylcarbamothioyl)hydrazinylidene]methyl]-N'-hydroxybenzenecarboximidamide 2-[3-(4-bromophenyl)propyl]pyrrolidine 3-azidooxy-4-cyclohexylfuran 4-cyclopentyloxy-N'-hydroxypyridine-2-carboximidamide 1-[(2,4-dimethoxyphenyl)methyl]-3-(2-methoxyethylamino)thiourea N-[5-chloro-2-(difluoromethoxy)pyridin-3-yl]-2-[4-ethylsulfonyl-2-methyl-1-oxo-3-[6-(trifluoromethyl)pyridin-2-yl]pyrrolo[1,2-a]pyrazin-8-yl]acetamide N-[3-(difluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[2,3-c]pyrrole-5-carboxamide 5-(2-chlorophenyl)-6-[2-oxo-4-(trifluoromethyl)pyrimidin-1-yl]-3,4-dihydro-1H-1,8-naphthyridine-2-thione N-(2,5-dichlorophenyl)sulfonylpyridine-3-carboxamide N'-[(2-methoxyphenyl)methyl]-3-(1H-pyrazol-5-yl)cyclohexa-1,3-diene-1-carboximidamide N-[1-(cyclopropylmethyl)piperidin-4-yl]-5,6-dihydropyrazolo[3,4-b]pyridine-1-carboxamide [4-(3,5-dimethylpyrazol-1-yl)phenyl]methanamine;ethane 4-azido-1-(3,5-dimethylphenoxy)pyrrolidine 3-ethoxy-4-(2-methylpropoxy)aniline 7-[1,2-bis(4-methoxyphenyl)ethyl]triazolo[4,5-d]pyrimidine (4S,5S)-2,7,9-trihydroxy-1-(2-methoxyphenyl)-4-[[(3R)-pyrrolidin-3-yl]amino]-5H-pyrido[4,3-b]indole-6-carboxamide 1-methyl-4,5-diphenylpyrrole-2-carboxylate 2-(3-bromothiophen-2-yl)-6-tert-butylpyridine 2-(dimethylamino)-1,3-bis(ethenyl)benzimidazole-5-carboxylic acid 4-(benzylcarbamoylamino)-3,5-dimethoxybenzoic acid 3-[[4-(2-chloroanilino)-6-methoxyquinazolin-7-yl]amino]sulfanyl-N,N-diethylpropane-1-sulfinamide 3-chloro-1,2-diethyl-4,5-bis(methoxymethyl)benzene N-[(3S,4R)-1-tert-butyl-3-hydroxypiperidin-4-yl]-5-ethoxypyrazine-2-carboxamide 4-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[1-[(2-methoxyphenyl)methyl]azetidin-3-yl]benzamide N-[(2,4-dichlorophenyl)methyl]-7-formyl-6-hydroxy-5-oxo-2,3-dihydro-1H-imidazo[1,2-a]pyridine-8-carboxamide 5-fluoro-N,4-dimethyl-3-[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazole-4-carbonyl]benzamide 5-methyl-3-(3-phenylpyrazol-1-yl)pyridazine (2S,3R)-1-benzyl-3-(cyclobutanecarbonylamino)-N-methyl-5-oxopyrrolidine-2-carboxamide 3-[4-(1H-indazol-5-ylamino)thieno[2,3-b]pyridin-2-yl]piperidine-1-carboxylic acid N-[2,5-dimethyl-6-(1,1,1-trifluoropropan-2-ylamino)pyrimidin-4-yl]-1,3-thiazole-5-sulfonamide N-methyl-4-[2-[[1-(5H-pyrrolo[3,2-d]pyrimidin-7-yl)cyclohexanecarbonyl]amino]ethoxy]benzamide 3-amino-N-[(6,8-dimethyl-2,3,4,5-tetrahydro-1H-2-benzazepin-3-yl)methyl]butanamide;dihydrochloride 2-(2-aminobutanoylamino)-3-(9H-fluoren-1-ylmethoxycarbonylamino)propanoic acid 4-(3,5-diethylpyrazol-1-yl)-2,6-bis(2-methylbutan-2-yl)pyrimidine 2-chloro-6-fluoro-4-(1,3,5-trimethylpyrazol-4-yl)phenol 1-[3-(2,4-diaminopyrimidin-5-yl)phenyl]-2-fluorobutane-1,3-dione (E)-1-[6-(3,5-dimethylpiperidin-4-yl)oxypyridin-2-yl]-3-methanimidoylpent-3-en-2-one 5-(4,6-dichlorocyclohexa-1,3-dien-1-yl)sulfonyl-4,6-dihydrothieno[2,3-c]pyrrole (3R)-3,4-dimethylpentanoic acid;N-[2-[[4-[3-[2-(ethylamino)-1H-inden-5-yl]propanoylamino]phenyl]sulfonyl-methylamino]ethyl]-N-[2-oxo-2-(2-pyridin-3-ylethylamino)ethyl]carbamate N-[2-chloro-5-(1,3-dioxoisoindol-4-yl)phenyl]acetamide 2-[4-(4,5-dimethylpyrimidin-2-yl)pyridazin-1-ium-1-yl]ethanesulfonic acid 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]-5-ethoxypyridine N-cyclopropylsulfonylbenzamide 4-[4,5-di(propan-2-yl)furan-3-yl]-3-iodobenzonitrile (2S)-N-[(1R,3R)-3-[(4-chloronaphthalene-1-carbonyl)amino]cyclohexyl]piperidine-2-carboxamide 1-methyl-6-(5-methyl-4,10-dihydrothieno[2,3-c][1]benzazepine-7-carbonyl)indazole-3-carboxylic acid 6-N-methyl-2-[(3Z,5E)-4-(oxan-4-yl)hepta-1,3,5-trien-3-yl]-4-N-[4-(propanoylamino)cyclohexyl]pyrimidine-4,6-dicarboxamide 2-(3,5-dimethylphenyl)-N-[2-ethoxy-6-(4-hydroxypiperidin-1-yl)pyridin-3-yl]acetamide N-[(2S)-3-(4-acetylpiperazin-1-yl)-2-hydroxypropoxy]-5-cyclopenta-1,3-dien-1-yl-7-(2-fluorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamide N-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]-2-morpholin-4-ylacetamide [3-(2,5-dimethoxyphenyl)-1H-indazol-6-yl]azanide 2-(1,3-benzodioxol-5-ylmethylidene)-4,6-bis[(5-methoxypyridin-2-yl)amino]-3H-isoindol-1-one 2-amino-4,6-dimethyl-5-[3-(pyrrolidine-1-carbonyl)phenyl]benzene-1,3-dicarbonitrile 6-[4-(9,10-dihydrophenanthrene-1-carbonyl)piperazin-1-yl]pyridazine-3-carboxylic acid 4-[(6S)-6-[[5,7-dimethyl-3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-4-yl]methylcarbamoyl]-1,3-oxazin-3-yl]butanoic acid N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-ethyl-3-hydroxy-5-(1-piperidin-1-ylcyclopentyl)benzamide 3-(3,5-dimethoxyphenyl)cyclopentane-1-carboxylic acid 1-benzyl-4,4-dimethylpyrrolidine;2,2,5,8,9-pentamethylpyrano[3,2-g]chromene N-[4-[(3,5-dimethylphenyl)sulfamoyl]phenyl]-2-hydroxy-N'-[(E)-1H-indol-3-ylmethylideneamino]butanediamide 1-[5-(cyclohexa-2,4-dien-1-ylmethoxy)pyrazin-2-yl]ethanone 3-(5-amino-1,2-oxazol-3-yl)-5-[2-(trifluoromethoxy)phenyl]-6H-[1,2]thiazolo[4,5-d]pyrimidin-7-one N-[(4-nitrophenyl)methyl]-2H-triazole-4-carboxamide 2-[(3,5-dibromo-4-hydroxyphenyl)methylideneamino]benzoic acid 1-[(4aS,10aR)-7-methylsulfonyl-3,4a,5,6,10,10a-hexahydro-2H-benzo[g]quinolin-4-yl]-2-aminoethanone 3-[(6E)-2,4-diamino-7-methoxyocta-1,5,7-trien-3-yl]-N-methylbenzamide;ethane;propan-1-amine N-(5-ethyl-1,3-thiazol-2-yl)-2,7,8-triazabicyclo[4.2.0]octa-1(6),2,4-triene-7-carboxamide (2Z,5E)-3-ethyl-N-[4-(4,7,8-trimethoxyquinolin-6-yl)oxyphenyl]octa-2,5-dienamide [(4aR,9aS)-8a-hydroxy-1-(5-hydroxypentyl)-2,3,4a,5,6,7,8-heptahydroquinoxalin-6-yl]-[3-fluoro-2-methoxy-6-(tetrazol-2-yl)phenyl]methanone N-butanoyl-1,5-dimethylimidazole-4-carboxamide 1-[4-(3,5-dichloropyridin-2-yl)oxyphenyl]propan-1-amine;hydrochloride 3-(4,6-dichloro-1H-indole-2-carbonyl)sulfanylbenzoic acid N-[3-(1,2-dihydropyridin-4-yl)-6-phenylimidazo[1,2-a]pyrazin-8-yl]-5,6-difluoro-1H-benzimidazol-2-amine 2-[4-(cyclopropylmethoxy)phenyl]-2-pyridin-3-ylacetaldehyde 2,6-dibromo-N-(4-ethoxyphenyl)-N-octylpyridin-3-amine 2-(1,3-dimethyl-4-propan-2-ylpyrrol-2-yl)-5-[(4-hydroxyphenyl)methylidene]-1,3-thiazol-4-one 2-benzylsulfanyl-N-methyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carboxamide 3-[5-[6-(dipropylamino)pyridin-2-yl]-3-ethynylpyrazolo[3,4-b]pyrazin-1-yl]cyclobutan-1-one N-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-1,4-dioxane-2-carboxamide N-[4-cyano-2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]-7-(trifluoromethoxy)indole-1-carboxamide (2S)-2-[4-(dimethylamino)phenyl]-1-N,3-N-bis(2-phenylethyl)cyclobutane-1,3-dicarboxamide 5-[2,4-bis(sulfanyl)phenyl]pentanenitrile 5-amino-3-[2-[4-[(2,4-dichlorophenyl)methyl]piperazin-1-yl]pyrimidin-4-yl]-6-methoxy-2,3-dihydroisoindol-1-one;trihydrochloride 1-[4,6-difluoro-5-(3-piperidin-1-ylpropoxy)-2H-chromene-8-carbonyl]pyrrolidine-2-carboxamide 1-[(2,3-dichlorophenyl)methyl]-4-nitropyrrole-3-carbonitrile 2-azido-N,N-dibenzylethanamine 2-[(2Z)-2-[(Z)-(3,5-dichloro-4-hydroxyphenyl)methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 1-bromo-2-chloro-4-(trifluoromethyl)benzene;ethane 1-cyclopropyl-N,2-diethyl-5,6-dimethoxyindole-3-carboxamide (2S)-3-cyclohexyl-N-[(E,6R)-1,8-diphenylnon-7-en-5-ynyl]propanamide 4-azido-6,7-dichloroisoquinoline 3-chloro-N,5-dimethyl-4-[(Z)-1-(2-nitrophenyl)propylideneamino]sulfanylaniline 6-[2,5-dimethyl-4-[3-[(1S)-1-phenylethyl]imidazol-4-yl]-N-propan-2-ylanilino]hexanenitrile 4-[[(E)-3-[5-bromo-2,4-bis(methoxycarbonyl)phenyl]prop-2-enoyl]amino]benzoic acid 1-azidooxy-3-(2-methylpropanoylamino)naphthalene-2-sulfonic acid 2-(2,4-dimethylphenyl)imino-5-[(3-propan-2-yloxynaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one 3-[(2R,6S)-2-butyl-6-cyclopropylmorpholine-4-carbonyl]-5H-pyrido[3,2-b]indole-7-carboxylic acid 4-[1-(3,5-dimethyl-1,2-oxazol-4-yl)propan-2-yl]-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide 5-methylsulfonyl-7-[(4-phenylpiperazin-1-ium-1-ylidene)amino]pyrido[2,3-d]pyrimidin-8-one [2-[(E)-2-(1,3-benzodioxol-5-ylmethoxyimino)propanoyl]oxyphenyl]azanium (1R,2S)-N-[4-methoxy-6-(pyrazol-1-ylmethyl)-1,3,5-triazin-2-yl]-2-phenylcyclopropane-1-carboxamide 2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxylic acid 3-(2,5-dimethylanilino)-4H-1,2,4-oxadiazol-5-one 1-[6-ethyl-5-[4-(2-hydroxypropan-2-yl)phenyl]pyridin-3-yl]-3-methylidenecyclobutane-1,3-diol (2R)-4,4-difluoro-1-[4-methyl-5-(6-pentanoylpyridin-3-yl)oxy-7H-pyrrolo[2,3-d]pyrimidin-2-yl]pyrrolidine-2-carboxylic acid 5-(8,14,22-trioxa-1-borapentacyclo[11.7.1.02,7.09,21.015,20]henicosa-2,4,6,9,11,13(21),15,17,19-nonaen-11-yl)quinoline 2-chloro-3,4,5,6,7,8,9-heptafluorofluoren-1-ol N-[5-methyl-2-(1H-pyrrol-3-yl)pyrimidin-4-yl]formamide 7-[4-(1,3-benzodioxol-5-yl)-2H-pyridin-1-yl]-9-pentan-3-yloxycarbonylhept-6-enoic acid 1-azidosulfanyl-3,4-dichloro-2-(9H-fluoren-1-yl)-9H-fluorene 3-fluoro-5-[2-(4-methylpiperidine-1-carbonyl)-7,8-dihydroimidazo[1,2-a]pyridin-5-yl]benzonitrile 3-(6-chloroquinolin-7-yl)-4-hydroxy-2H-furan-5-one 2-amino-5,7-dibromoquinolin-8-ol 4-cyclobutyl-N,2-dimethyl-5-(4-piperidin-1-ylsulfonylphenyl)pyrazol-3-amine N-(6-methoxypyridin-3-yl)-2-methyl-4,5-dihydropyrimidine-4-carboxamide N-azido-4-[(3-hydroxyphenyl)methylamino]benzenesulfonamide N-[5-(3-cyanophenyl)-1,3-thiazol-2-yl]-4-(trifluoromethoxysulfanyl)benzamide 1-N,3-N-diethylbenzene-1,2,3-triamine (3R)-N-ethyl-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-3-carboxamide;hydrochloride 3-chloro-N-[[4-[2-methyl-6-(oxetan-3-ylamino)pyrimidin-4-yl]cyclohexyl]methylidene]benzamide 3-[4,5-diamino-2-(2-methoxyethoxy)phenyl]sulfanyl-1H-indole-7-thiol 6-chloro-5-(5-methyl-3,4-dihydropyridin-2-yl)-N-(2-morpholin-4-ylethyl)pyrazin-2-amine 1-methyl-3,5-bis(phenylmethoxy)-4-propan-2-yl-1H-indene 2-(difluoromethyl)-4-(3,5-dimethyl-1,2-oxazol-4-yl)-5-nitrobenzaldehyde 4-azido-2,3-bis(difluoromethyl)phenol (7R,9aS)-2-[(4-ethylphenyl)methyl]-7-(hydroxymethyl)-5-[[(1R)-2-hydroxycyclohexyl]carbamoyl]-8-oxo-N-[(3,4,5-trifluorophenyl)methyl]-1,3,4,7,9,9a-hexahydropyrrolo[1,2-a][1,4]diazepine-9-carboxamide 4-(1,5-dimethylpyrazole-3-carbonyl)-3-[(2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one 1-[3-[3,5-difluoro-4-(trifluoromethyl)phenoxy]propoxy]-6-ethoxy-2-fluoronaphthalene 2-[2,4-dinitro-N-(2H-tetrazol-5-yl)anilino]octanoic acid 5-[(Z)-1-amino-3-methyliminoprop-1-en-2-yl]-N-[6-(piperidine-4-carbonyl)-7,8-dihydroimidazo[1,2-a]pyridin-2-yl]furan-2-carboxamide 1-phenyl-2-(6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-2-ylamino)ethanol 4-(5-amino-1,3,4-oxadiazole-2-carbonyl)-2,6-dimethylmorpholin-3-one 1,4-diamino-2-naphthalen-2-ylanthracene-9,10-dione 4-[4-(5,6-diaminopyrimidin-4-yl)-1,2-oxazol-3-yl]phenol N-[(2R)-1,1,1-trifluorobutan-2-yl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide N-[(2S)-1-amino-3-phenylpropan-2-yl]formamide;5-(4-ethylphenyl)-3-methoxy-N,N-dimethylbenzenecarboximidamide 3-[3-methoxycarbonyl-6,8-dioxo-7-(trifluoromethyl)pyrido[2,1-f][1,2,4]triazin-2-ium-2-yl]benzenesulfonic acid 2-[[4-(hydroxymethyl)cyclohexanecarbonyl]amino]-N,N-dipropylbenzamide 3-[7-[(3,4-dichlorophenyl)methoxy]-6-fluoro-2H-chromene-3-carbonyl]-1-azabicyclo[2.2.2]octane-2-carboxylic acid 4-[(2,3-diethylphenyl)-phenylmethoxy]benzenecarboximidamide 2-(4,6-dichloropyrimidin-5-yl)oxybenzonitrile 5-(4-ethoxyphenyl)-3-methyl-1,2,4-thiadiazole 1-[6,7-dichloro-9-(methylamino)-3,4-dihydro-2H-pyrano[2,3-b]indol-4-yl]ethanone 3-(7,8-dioxabicyclo[4.2.0]octa-1,3,5-trien-2-yl)propanenitrile 1-(6,11-dihydrobenzo[c][1]benzazepin-5-yl)-2-phenylethanone 1-[2-(cyclopropylmethoxy)phenyl]-N-hydroxy-6,7-dihydro-4H-imidazo[4,5-c]pyridine-5-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]-cyanomethylidene]methanesulfonamide 2-[5-(carbamoylamino)pyridin-3-yl]-N,N-dimethyl-1H-imidazo[4,5-b]pyridine-7-carboxamide (4Z)-4-[[5-(2,4-dichlorophenyl)furan-2-yl]methylidene]pyrazolidin-3-one 4-(8-iodoimidazo[1,2-a]pyridine-5-carbonyl)piperazine-1-carboxylic acid [2-[(3,4-diethylphenyl)methoxy]pyrimidin-5-yl]methanamine 4-N-(2,4-dichlorophenyl)-5-methyl-3H-1,3-benzoxazole-2,4-diimine (2S)-1,2-bis(4-methoxyphenyl)-3-[(E)-1,4,4-trifluoro-3-oxobut-1-enyl]-2H-quinazolin-4-one 4-[3-(4,6-diamino-1,3,5-triazin-2-yl)-4-hydroxyphenoxy]benzenesulfonic acid ethane;2-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)phenyl]acetonitrile 2-[5-methyl-4,6-dioxo-1-(3-phenylpropyl)-2H-thieno[2,3-d]pyrimidin-3-yl]acetic acid 2-[3-methylsulfanyl-4-(trifluoromethoxy)phenyl]propanedioic acid 1-[3-[(E)-2-bromoethenyl]phenyl]propan-1-one;ethane 4-methylsulfanyl-N-[[6-(2,2,3,3-tetrafluoropropoxy)pyridin-3-yl]methyl]cyclohexane-1-carboxamide N-[4-[(5,6-dimethylpyrimidin-4-yl)sulfamoyl]phenyl]acetamide 4-azidooxy-N,5,6-triphenylpyridazine-3-carboxamide 4-[(2-methyl-1,3-benzothiazol-5-yl)oxy]-N-[(E)-1H-pyrrol-2-ylmethylideneamino]benzamide 3-(3,4-dichlorophenyl)-N'-[2-hydroxy-2-(5-thiophen-2-ylfuran-2-yl)ethyl]propanimidamide N'-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-4-propan-2-ylbenzenecarboximidamide 4-[(3,4-dimethoxyphenyl)methylamino]-5-ethylsulfanyl-1H-pyrimidin-6-one 5-azido-N,N-dimethyl-1H-benzimidazole-2-sulfonamide N-[2-(4,5-dihydro-1H-imidazol-2-yl)phenyl]formamide;1-(7-fluoro-3-methylidene-2-oxo-1H-indol-6-yl)ethanone 6-[5-fluoro-2-(3,4,5-trimethylphenyl)pyridin-4-yl]imidazo[1,2-a]pyrazine 2-(6,8-dichloroimidazo[1,2-a]pyridin-2-yl)-3H-quinazolin-4-one 5-(azidomethyl)-2-[2,6-difluoro-4-(4-octoxyphenyl)phenoxy]aniline N-methyl-3-[(3S)-oxolan-3-yl]oxybenzenesulfonamide (3S,4R)-3-[3-[6-[1-[2-methoxyethyl(oxan-4-yl)amino]piperidin-4-yl]pyridin-3-yl]phenyl]-5-(trifluoromethyl)pyrrolidine-3,4-diol 4-methyl-2-(N-[1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl]anilino)-1,6-dihydropyrimidine-5-carboxylic acid 7-(3,4,6,7,8,9-hexahydropyrido[1,2-a]pyrazine-2-carbonyl)-N-methylnaphthalene-2-sulfonamide;hydrochloride 1-(2,4-dimethylphenyl)-3-[(E)-(3-ethoxy-4-hydroxyphenyl)methylideneamino]thiourea 7-(cyclopropylmethoxy)-2-(4,5-dihydropyrimidin-6-yl)quinoline N-[4-methyl-3-(morpholine-4-carbonyl)phenyl]-2-sulfanylidene-1H-pyridine-3-carboxamide 4-[2-(azidomethyl)phenoxy]-1,2-bis(fluoromethoxy)benzene N-methyl-2-phenylhexanamide 3-[1-(2,2-difluoroethyl)-5-methoxyindol-4-yl]-1-[4-[(5-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl)amino]phenyl]propan-1-one N-[(2S)-3-amino-1-oxobutan-2-yl]-1H-indazole-6-carboxamide 2-[[4-(difluoromethoxy)phenyl]sulfanylmethyl]furan;6-methoxy-1,2-benzoxazol-3-amine 5-[3-amino-4-(2,6-difluorophenyl)butanoyl]spiro[1H-indole-3,2'-thiolane]-2-one;(5Z,7E)-9-methoxy-8-methylidene-10-azatricyclo[6.4.0.02,7]dodeca-1(12),2(7),3,5,11-pentaene 1-(2,5-dimethylphenyl)sulfanyloxycyclopentane 1-[3,5-difluoro-2-(propan-2-ylamino)phenyl]ethenol 2-(2,4-dioxopyrrolidin-1-yl)-N-[5-(oxan-3-yloxy)pyridin-2-yl]acetamide N-[(1R)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-ylidene]pyridine-4-carboxamide N-[3-[(5Z)-4,7-dimethylocta-1,6-dienyl]iminobutyl]-2-(2-ethenylphenyl)acetamide 4-hydroxy-6,9,10,11-tetramethoxyphenanthrene-2-carboxylic acid N-[(1R)-4,5-diaminocyclohex-2-en-1-yl]-3-pyridin-4-ylsulfanylpropanamide;ethane (4-methoxyphenyl)-[5-(6,7,8-trichloroquinolin-2-yl)sulfanylthiophen-3-yl]diazene N-(3-bromo-2,5-dimethylphenyl)-4-nitro-N-(6-nitro-1,3-benzothiazol-2-yl)benzamide N-[(Z)-2,3-dihydroinden-1-ylideneamino]-4-pyridin-3-ylpiperazine-1-carbothioamide 2,6-bis(methyliminomethyl)-4-phenylphenol 4-chloro-3,5-dinitrobenzoic acid 4-N-butyl-1-N,4-N-dibutylbenzene-1,4-diamine 5-(4-ethenylphenyl)benzene-1,2,3,4-tetracarboxylic acid 3-[4-(3,5-dichloropyridin-2-yl)piperazin-1-yl]sulfonylthiophene-2-carboxylic acid 4-amino-N'-methoxypyridine-2-carboximidamide;4-(3,4-dihydro-1H-isoquinolin-2-yl)phenol 5-[3-chloro-4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidine-2,4,7-trithione 2-(N-butanoyl-3,5-dichloroanilino)decanoic acid (6Z)-6-[1,2,3,5,7,8-hexahydropyrrolo[2,3-e]indolizin-7-yl(methoxy)methylidene]cyclohexa-2,4-diene-1-thione (2S)-N-[(Z)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-2-(4-methylanilino)propanamide 1-(3-bromophenyl)sulfonyl-N-(2-cyanocyclohexyl)-N',N'-dimethylpyrrolidine-2-carbohydrazide N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3,4-dihydropyridine-2-carboxamide 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)azetidin-2-one N-[4-fluoro-3-(5-methyltetrazol-2-yl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide [4-amino-6,7-diethoxy-1-(4-fluoroanilino)isoquinolin-3-yl]-methylideneazanium 4-methoxy-2,6-dinitro-N-phenylaniline 1-[4,6-dichloro-2-(4-methoxyphenyl)sulfanylquinolin-3-yl]ethenol 2-[(3-fluorophenyl)sulfanylmethyl]-7H-purine 2-(3-aminopiperidine-1-carbonyl)-6-cyclohexyl-5-[1-(4-fluorophenyl)pyrazol-4-yl]pyridine-3-carboxylic acid N-[(2R)-3,4-dimethylpentan-2-yl]-6-fluoro-1H-indole-3-carboxamide (2S)-4,6-dichloro-N-[2-(4-cyano-3-fluorophenyl)ethyl]-5-[[(1R)-1-(4-methoxyphenyl)ethyl]amino]-2-methylpyridine-3-carboxamide [1-(5,6-dimethylpyrimidin-4-yl)piperidin-2-yl]-pyrrolidin-1-ylmethanone 4-[[(E)-[(Z)-4-aminobut-3-enylidene]amino]methyl]-2,5-dimethylthiophene-3-carboxylic acid 1-[4-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]phenyl]-N'-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-methoxypiperidine-4-carbohydrazide 2-azidooxy-6-(trifluoromethyl)pyridine 4-[2-(4-carboxylatobutyl)-3,5-dimethoxyphenyl]butanoate 1,4-dimethyl-2-phenylpiperazine;ethane N-[(1S)-2-hydroxycyclohexyl]-6-methoxypyridine-3-carboxamide N-azido-1-phenylmethoxy-2-(trifluoromethyl)imidazole-4-carboxamide N-[3-(dimethylamino)phenyl]cyclohexenecarboxamide 2-(2,3-difluorophenyl)-6-ethylbenzo[f]isoindole 2,3-dichloro-N'-hydroxypyrrolo[1,2-a]pyrazine-7-carboximidamide 5-(2,6-dimethylmorpholine-4-carbonyl)-N-ethyl-2-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]oxybenzamide 2-[(1Z)-3,4-diamino-5-chloropenta-1,3-dienyl]phenol 4-(5-amino-2,3-dihydropyrazin-6-yl)-N-[(Z)-1-aminoethylidenecarbamohydrazonoyl]benzamide 3-[1-(5-methylpyridin-2-yl)-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl]phenol 4-azido-1-[(3-methoxyphenyl)methyl]pyrazolo[3,4-d]pyrimidine 5-[(2,4-dihydroxyphenyl)methylideneamino]benzene-1,3-disulfonic acid N'-[4-(cyclopropanecarbonylamino)-3-hydroxyphenyl]oxamide [3-(1H-indol-2-yl)phenyl]-[4-(1,8a-dihydroisoquinolin-6-yl)piperazin-1-yl]methanone N-(diaminomethylidene)-4-[4-(trifluoromethoxy)phenoxy]butanamide 5-(2,3-dimethoxyphenyl)-4-ethyl-1H-pyrimidin-6-one 1-(2,3-dimethylphenyl)-N'-hydroxyimidazole-2-carboximidamide 3-bromo-2-ethyl-5,6-dihydrobenzo[h]cinnoline 3-azido-4,6-dibromoisoquinoline (2-fluorophenyl)methyl-[1-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)piperidin-4-yl]carbamic acid 6-(5-methoxy-2,3-dihydroindole-1-carbonyl)pyridine-3-carboxamide (3-cyanophenyl)imino-[4-(1,3,4-oxadiazol-2-yldiazenyl)anilino]-oxoazanium 5-(2,4-dimethylphenyl)sulfanyl-N'-hydroxypyrazine-2-carboximidamide 5-(1,2-benzodioxol-6-yl)-3-propan-2-ylidene-1H-indol-2-one 1-azido-4-(2-fluorophenyl)piperazine 3-chloro-6-(methoxymethyl)-5-methylsulfanylpyridine-2-carbonitrile 1,2-dichloro-5-methoxy-4-(trifluoromethyl)benzene 3-chloro-6,7-difluoroacridine 1-[3-azido-2,6-di(propan-2-yl)phenyl]ethanone 2-[(1S)-1-[[5-fluoro-4-methyl-6-[[(2R,3R)-3-methylpyrrolidin-2-yl]methoxy]pyridine-3-carbonyl]amino]ethyl]benzoic acid 2-[3-(1,4-diazepan-1-yl)-4-methoxyphenyl]-N-methylacetamide N-(1H-indazol-6-yl)-4-methoxynaphthalene-1-carboxamide 4-[(2R,6R)-4-[3-cyclobutyl-5-[(dimethylamino)methyl]benzoyl]-2,6-dimethylpiperazin-1-yl]-N-ethyl-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide N-(3-chloro-4-fluorophenyl)-5-methylpyrazine-2-carboxamide 1-[2,4-bis(trifluoromethyl)phenyl]-3-[3,5-di(propan-2-yloxy)phenoxy]benzene;ethane (3R)-4-[2-chloro-6-fluoro-N-methyl-5-(propanoylamino)anilino]-1,1-dioxothiane-4-carboxylic acid 1-[[1-(2-methoxyphenyl)cyclopropyl]methyl]piperidine;dihydrochloride 3-ethylsulfonyl-2-(trifluoromethyl)pyrimidin-4-one ethane;6-(4-methoxyphenyl)imidazo[1,2-b]pyridazine 2-(1-propanoylpiperidine-4-carbonyl)-9-oxa-2,12,14,15,17-pentazatetracyclo[8.7.0.03,8.011,16]heptadeca-1,3,5,7,10,12,15-heptaen-15-ol 2-amino-4-(2,6-dichloro-3,5-dimethoxyphenyl)-6-ethoxy-4H-pyran-3,5-dicarbonitrile 7-[4-(aminomethyl)phenyl]-5-ethynylfuro[3,2-c]pyridine-4-thione 1-cyclopropyl-N'-(dimethylaminosulfanyl)-4,5-difluoropyrazole-3-carboximidamide 1-(2,5-dimethylpyrazol-3-yl)oxy-3-[2-[(5-phenyltetrazol-2-yl)methyl]phenoxy]propan-2-one (E)-N'-[6-ethenyl-5-[2-(methoxymethyl)anilino]pyridin-3-yl]-N,N-dimethylhept-1-ene-1,7-diamine 7-(3,5-difluorophenyl)sulfanyl-1H-pyrido[2,3-b]pyrazine N-[2-[4-(5,6-dihydroquinolin-8-yl)piperazin-1-yl]ethyl]-3-methoxybenzamide 1-(2,3,6,7,8,9-hexahydrobenzo[g][1]benzofuran-4-yl)-N-methylethanamine 5-chloro-N-[(Z)-1H-indol-3-ylmethylideneamino]-2-propan-2-yloxybenzamide 1,3-dicyclohexyl-2-methoxybenzene;pentane 4-(2,3,3a,4,5,6,7,7a-octahydro-1H-indazole-6-carbonyl)-N-ethyl-3-methoxybenzamide 2-(4-methoxybutanoyl)-1H-pyridine-2,3-dicarboxylic acid 4-(4,8-dimethylquinolin-2-yl)morpholine 5-tert-butyl-3,8,11-triazatricyclo[7.4.0.02,6]trideca-1(9),2(6),3,7,10,12-hexaene;methanamine 6-[(2,3-dibromo-5-ethoxy-4-hydroxyphenyl)methyl]-2-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-(4-azidobutanoyl)chromen-2-one N'-[2,6-dimethyl-4-(1,3-oxazol-5-yl)anilino]-1-(oxan-3-yloxy)cyclopropane-1-carbohydrazide N-(2,5-dichlorophenyl)-3-propanoylbenzenesulfonamide 2-methylsulfanyl-5-[4-(2,3,4-trifluorophenyl)phenoxy]thiophene 3-[(Z)-but-2-enyl]-5-propan-2-ylsulfanylbenzonitrile 3-[3-(aminomethyl)phenyl]-1,1-difluoropropan-2-amine;hydrochloride 2-(3,4-dihydropyrazole-2-carbonyl)-5-methyl-1H-indole-3-carboxylic acid 2-(4-methylphenyl)-4-[4-(propan-2-ylamino)piperidin-1-yl]pyrimidine-5-carbonitrile N-(2-tert-butylimidazo[1,2-a]pyridin-6-yl)-4-cyclopropylidene-8-iodoquinazoline-6-carboxamide 6-fluoro-3-methyl-2-[(4Z)-4-propan-2-ylideneoxepan-5-ylidene]-1H-quinazolin-4-one 5-[2-azido-3-(trifluoromethoxy)phenyl]sulfonylpyrimidine 4-[4-(methylsulfonyloxycarbamoyl)phenyl]-2-(trifluoromethyl)benzoate 2-cyclohexyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide (3R)-4,5-dichloro-2,9,12-trimethyl-6H-indolo[1,2-d][1,4]benzoxazepine;5-fluoropyrimidine-2,4-diamine 4-[3,5-dimethyl-1-(2-piperidin-4-ylethyl)pyrazol-4-yl]pyrimidine (3E,5Z)-2-fluorohepta-1,3,5-triene;5-methoxy-4-(methylamino)pyrrolo[2,1-f][1,2,4]triazine-6-carbonitrile N-[1-(3,4-dichlorophenyl)sulfonylpiperidin-4-yl]-4-fluorobenzenesulfonamide 4-[5-(1H-indole-2-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-3-yl]-1-methyl-1,8-naphthyridin-2-one 3-[2,4-diamino-6-(cyclohexylamino)pyrimidin-5-yl]propanal N-[(6S)-2,3-dimethoxy-5,6-dihydrobenzo[b][1]benzazepin-11-yl]propanamide 2-hydroxy-5-(4-nitrophenyl)benzenesulfonic acid 3-[6,7-dimethoxy-1-(2-phenylethyl)isoquinolin-4-yl]sulfanyl-N-hydroxypropanamide 2-(2,4-dihydroxyphenyl)-N-[(Z)-2-methylbut-1-enyl]pentanamide 5-chloro-1,3-diiodoindazole 4-[5,6-di(propan-2-yl)pyridin-3-yl]-N-[4-(pyrrolidine-1-carbonyl)phenyl]-3H-pyrrole-2-carboxamide 5-(4,5-didehydroimidazol-1-yl)-N-[2-oxo-3-[4-(piperidine-1-carbonyl)phenyl]propyl]pyrazine-2-carboxamide 4-(7-hydroxy-5,6,8,9-tetrahydropyrido[2,3-d]azepin-3-yl)phenol 5-(1,3-benzodioxol-4-yl)-N-[6-(2,5-dihydropyrrole-1-carbonyl)pyridin-3-yl]pentanamide (E)-N'-[2-chloro-5-methylsulfonyl-4-(trifluoromethoxy)phenyl]but-1-ene-1,4-diamine 2-[(1-butylpyrazole-3-carbonyl)amino]-6,7-dihydro-5H-cyclopenta[b]pyridine-4-carboxamide 2-[5-(methylamino)-6,7-dihydro-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-N-phenyl-4H-chromene-8-carboxamide 4-[(3S)-1-[(2S)-2-benzylbutanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one N'-[5-bromo-2,4-bis(2,3,6-trifluorophenyl)benzoyl]-4-methylcyclohexanecarbohydrazide N-[2,3-dichloro-5-(1,3-thiazol-4-ylsulfonylamino)phenyl]-1H-pyrrolo[2,3-b]pyridine-6-carboxamide N-[(2S,3R)-6-azido-5-hydroxyhexan-2-yl]-4-benzamidobutanamide 1-methyl-2-(2,3,5-trichlorophenyl)imidazole 6-methyl-3-phenylquinoxaline 3-azidooxy-1H-benzimidazole-2-thione N-(4-azido-2,6-dichlorophenyl)-5-bromopyrimidin-2-amine (4S)-5-methoxycarbonyl-2,6-dimethyl-1-[(2R)-2-nitrobutanoyl]-3,4-dihydro-1H-isoquinoline-4-carboxylic acid N-[1-(2-methoxyethyl)pyrazol-4-yl]pyridine-3-carboxamide N-[5-(4,6-dimethylpyridin-2-yl)-1H-pyrazol-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carboxamide 3-azidooxy-6-[5,6-difluoro-1-(2-methylpyridin-4-yl)indazol-3-yl]pyrazolo[1,5-a]pyrimidine 3-[(5S,7R)-2-bromo-9-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a][1,3]diazepin-5-yl]phenol 2-(1H-benzimidazol-2-yl)-N-[2-cyclohexa-2,4-dien-1-yl-6-(4-fluorophenyl)pyrimidin-4-yl]ethanimine 3-benzyl-8,9-dimethoxybenzo[f]chromene 4-chloro-3-[5,6-diethyl-2-methoxy-3-(5-nitrosopyridin-2-yl)sulfanylphenyl]benzonitrile 1-(3,6-dihydro-2H-pyran-4-yl)-5-methoxy-N-methyl-N-[6-(piperidin-4-ylamino)pyridin-3-yl]pyrazole-4-carboxamide;hydrochloride 1-[6-(4-methoxyphenyl)pyridazin-3-yl]-N,N-dipropylpiperidin-4-amine 6-cyclobutyl-N-[[(2R,3S)-1-methyl-5-oxo-2-phenylpyrrolidin-3-yl]methyl]pyridazine-4-carboxamide [4-(2-phenylethyl)cyclohexa-1,3-dien-5-yn-1-yl]boronic acid 2-[4-(7,8-dihydroquinolin-5-yl)phenyl]aniline 1-(azidomethyl)-5-chloronaphthalene N-(4-chlorophenyl)-2-hydroxy-3,5-dinitrobenzenesulfonamide 3-azido-1,5-diethyl-4-methoxypyrazole 7-[3-(5,8-dihydroxynaphthalen-1-yl)propanoyl]naphthalene-2-carboxylic acid 2-[4-[(1R,3S)-3-aminocyclopentyl]pyridin-2-yl]-N-[5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]acetamide;dihydrochloride 2-[6-(oxolan-3-yl)indazol-1-yl]benzoic acid 3-cyclopentylsulfonylthiophene 2-[(1,4-dimethylpyrazol-3-yl)amino]-5-propan-2-ylbenzaldehyde 3-[(2,4-dihydroxyphenyl)methyl]-7-[1-methyl-5-[(Z)-prop-1-enoxy]cyclohexa-2,4-diene-1-carbonyl]heptanoic acid 1-methyl-2-(9H-thioxanthen-9-id-3-yl)pyridin-1-ium;rhodium 2-[4-(3,5-dimethoxyphenyl)-1H-pyrazol-5-yl]-6,7-dihydro-1H-indole 4-hydroxy-3,7-dimethyl-3H-1,8-phenanthroline-2-carboxylic acid 1-(4-phenylpyrimidin-2-yl)-6,7-dihydroindazole N-[2,4-difluoro-5-(2-methoxypyridine-3-carbonyl)phenyl]methanesulfonamide N-(4-anilinophenyl)sulfonyl-2,6-dichlorobenzamide 5-(2,5-dichlorophenyl)-3-methyloxolan-2-one N-[3,5-bis(4-chlorophenyl)phenyl]acetamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-7-methoxy-4-oxochromene-2-carboxamide 2-(5,6-difluorobenzimidazol-1-yl)-3H-pyrido[3,4-d]pyrimidin-4-one 4-chloro-2-(4,4-dimethylpiperidin-1-yl)pyridine;ethane 2-ethoxy-4-(methylsulfanylamino)benzonitrile;N-(6-oxohexyl)formamide 3-[5-ethylsulfanyl-6-(1,4,7-triazaspiro[3.5]nonan-7-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridine 7-chloro-5-(4-methylsulfanylphenyl)pyrido[3,2-b]indole 5-[2-(4-chlorophenyl)hydrazinyl]sulfanyl-3H-1,3,4-oxadiazole-2-thione N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]imidazo[1,5-a]pyridine-1-carboxamide N-[(E)-(2,3-dihydroxyphenyl)methylideneamino]pyridine-4-carboxamide;hydrate 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-3-(oxan-4-ylmethoxy)urea 4-(dimethylamino)-N-[3-(1H-pyrrol-2-ylamino)quinoxalin-6-yl]benzenesulfonamide 6-methyl-N'-[(3Z,5Z)-4-methylidenehepta-1,3,5-trien-2-yl]benzenecarboximidamide 2-chloro-3-(4-methoxyphenyl)-6-methylimidazo[1,2-a]pyrazine 3-(2-bromophenoxy)-N'-hydroxypyrazine-2-carboximidamide 1-[(5R)-8-benzoyl-2,8-diazaspiro[5.5]undecan-2-yl]pentane-1,4-dione 7-hydroxy-3-methylnaphthalene-1,2-disulfonic acid;2-[(4Z)-hepta-1,4-dien-6-ynyl]thiophene (E)-2-(3-formylphenyl)-N,6-dimethylidenehex-3-enamide 1-(benzenesulfonyl)-N-phenylmethoxyindol-5-amine N-[(5E)-1,4-dimethyl-6-oxo-3-bicyclo[3.2.0]hepta-2,4,7-trienyl]formamide;ethane 2-(1,5-dimethylpyrazol-4-yl)oxy-N'-[6-[4-[(4R)-4-methylazepane-1-carbonyl]phenyl]pyridin-3-yl]ethanimidamide 4-azido-3,5-dichloro-2-[1-(4-propan-2-ylphenyl)sulfonylpiperidin-4-yl]oxypyridine 2-[N-(2-carboxyethyl)-4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]anilino]octanoic acid 5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-sulfonamide (1S,3R)-N-[[5-chloro-2-fluoro-4-[[4-(1H-indole-3-carbonylamino)cyclohexyl]methyl]phenyl]methyl]-3-methoxycyclopentane-1-carboxamide 2-(3,4-difluorophenyl)-1-[2-methoxy-5-(trifluoromethyl)phenyl]piperidine 4-[(3,5-ditert-butyl-2-hydroxyphenyl)methylideneamino]-N-(2-phenylpyrazol-3-yl)benzamide (3-cyclopentyloxy-4-methylphenyl)-[2-(1,5-dimethylpyrazole-3-carbonyl)-6-azaspiro[2.5]octan-6-yl]methanone 3-[[3,5-bis(trifluoromethyl)phenyl]sulfonylamino]benzoic acid ethane;N-[2-methoxy-6-methyl-3-(trifluoromethyl)phenyl]acetamide 2-N-azido-6-N,8-N-dimethylquinoline-2,6,13-triamine 4-[3-chloro-4-(cyclopentylmethoxy)anilino]-7-nitro-1H-quinazoline-2,4-dione N-[(3S,4R)-1-methylsulfonyl-3,4-dihydro-2H-chromen-4-yl]-5-(5-phenyl-1,2,4-oxadiazol-3-yl)pyridine-3-carboxamide 6-[(1-methylpyrazol-4-yl)methoxy]pyridine-2-carboxylic acid 5-chloro-3,6-bis[(2S)-butan-2-yl]pyrimidine-4-thione ethane;5-[(2E,4Z)-3-(ethylaminomethylidene)hexa-2,4-dien-2-yl]-N'-hydroxypyridine-3-carboximidamide [6-methoxy-2-(2-methyl-1,3-dioxolan-2-yl)benzimidazol-1-yl]-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]methanone 1-(6-chloropyridine-3-carbonyl)-5-methoxy-2,3-dihydroindole-7-carbonitrile 2,2-diamino-3-[(3E,5Z)-octa-1,3,5-trien-4-yl]sulfonylcyclopropane-1,1-dicarbonitrile (3S)-N'-hydroxy-1-methyl-2,5-dioxo-N'-[4-[6-phenylhexanoyl(propyl)amino]butyl]pyrrolidine-3-carboximidamide (2S)-N'-hydroxy-3-phenylbutanediamide (7S)-5,7-dimethyl-N-[2-methylsulfanyl-3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide N-azido-2,2-dimethyl-5-phenylpentan-1-amine 1-(2,5-dimethylphenyl)sulfonyl-3-[6-(4-fluorophenyl)pyridin-3-yl]thiourea 1-butoxy-2,5-diethyl-4-[(3E)-penta-1,3-dien-3-yl]benzene N-(azidomethyl)-1-[2,3-bis(trifluoromethyl)phenyl]ethanamine (6R)-2-amino-6-methyl-5,6,7,8-tetrahydro-3H-pteridin-4-one (E)-3-[4-(2,6-dichlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]prop-2-enal 1-aminoethylidene(7H-pyrrolo[2,3-d]pyrimidin-4-yl)azanium 2-(3,4-dihydropyridin-5-yl)-6-[9-(2-hydroxyethylsulfanylmethyl)fluoren-9-yl]oxane-3,4-diol 2-(4-chlorophenyl)-N-[2,4-difluoro-3-[4-(1H-pyrazolo[3,4-b]pyridin-5-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-6-carbonyl]phenyl]acetamide 1-[(2R)-3,4-dihydroxy-5-propan-2-yloxolan-2-yl]pyrimidine-2,4-dione 3-[4-(furan-2-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-5-pyridin-3-yl-1H-pyrazolo[3,4-b]pyridine 4-(benzylamino)-2,3-dihydropyrimido[1,2-b]indazole-6-carboxylic acid 2,3-dichloro-6-(9H-fluoren-1-yl)pyridine 4-[4-[(dimethylamino)methyl]pyrazol-1-yl]-N',2,5-trimethylbenzenecarboximidamide [4-(3,5-dimethyl-1H-pyrazol-4-yl)sulfonylpiperazin-1-yl]-(4-phenylphenyl)methanone N-azido-3-[[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfonylamino]-1-benzofuran-2-carboxamide 2-(1,3-benzodioxol-5-yl)-N-[[2-(trifluoromethoxy)phenyl]methyl]propanamide 2-[(3Z)-5-phenylhepta-1,3-dien-4-yl]oxirane 2-(5-azidopyrazin-2-yl)-3,5-dimethoxyaniline N-[(2R)-1,4-dioxan-2-yl]-3-fluoro-5-methoxy-2-(pyridine-4-carboximidoyl)aniline 4-[1,2-dihydroacenaphthylene-1-carbonyl(methyl)amino]-3-hydroxybutanoic acid 2-chloro-4,4-difluoro-3-hydroxysulfanyl-5,6-bis(trifluoromethoxy)benzoic acid (5S)-4,7-dioxo-2-piperidin-1-yl-N-[3-(trifluoromethoxy)phenyl]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-[1-(benzenesulfinyl)piperidin-3-yl]oxy-5-cyclopropyl-2-fluorobenzoic acid 2-azido-5,7-dimethyl-1H-pyrrolo[3,2-c]pyridine 2-[azido(pyrrolidin-1-yl)methyl]-3,4-dihydro-1H-isoquinoline 3-[2,5-dimethyl-4-(2-sulfanylpropan-2-yl)phenyl]-N'-ethyl-1H-pyrazole-5-carboximidamide 7-amino-5-(3,4-dihydroxyphenyl)pyrazolo[1,5-a]pyrimidine-2-carboxylic acid;ethane N-[[4-chloro-3-(trifluoromethyl)phenyl]carbamothioyl]thiophene-2-carboxamide 1-(9-methylcarbazol-3-yl)-9,9a-dihydrocarbazole (2S)-5-N,3-dimethyl-7-phenylheptan-2-amine N-[2,2-dimethyl-3-(3-pyrrolidin-1-ylpropylamino)butanimidoyl]benzamide 4-(4-bromo-N-hexadecanoyl-2,5-dimethylanilino)benzenesulfonic acid 2-[(6R)-4,7-dioxo-6,8-bis(trichloromethyl)-3,5-dihydropyrrolo[3,2-g]quinazolin-6-yl]acetamide 2-[6-(difluoromethoxy)imidazo[1,2-a]pyridin-3-yl]-N-phenylpyrimidine-5-carboxamide 1-(2-azidoethyl)-4,6-bis[5-methyl-1-phenyl-3-(trifluoromethyl)pyrazol-4-yl]pyrazolo[3,4-d]pyrimidine 4-bromo-5-chloro-1-(4,4,4-trifluorobutyl)pyrrolo[2,3-b]pyridine 1-N,3-N,7-N-trimethyl-5H-[2]benzoxepino[4,5-c]pyrazole-10,12-dicarboxamide 2-chloro-1,3-difluoro-5-[4-[(E)-4-prop-2-enoxybut-3-enyl]cyclohexyl]benzene 3-ethyl-2-fluorobenzoate 1-[2,4-difluoro-3-(pyridine-3-carbonyl)phenyl]-2-(4-ethylsulfanylphenyl)-5-methoxypenta-2,4-dien-1-one 2-[[4-amino-6,7-dimethoxy-3-(5-methylfuran-2-carbonyl)quinolin-2-yl]amino]ethanol 3-[[7-cyclopropylimino-5-(1,2-oxazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-ylidene]methyl]-1H-pyrrole-2,5-diol N-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-1,3,7-trimethylpyrazolo[4,3-b]pyridine-5-carboxamide 1-(2-azidopropan-2-ylsulfonyl)-4,6-dimethoxybenzimidazole 6-hydroxy-8-methyl-7,9-dihydroimidazo[1,2-a]quinoxaline-3-carboxylic acid 4-[2-(7H-purin-6-yl)phenyl]benzonitrile 2-[(7S)-3,5-dimethyl-6-oxo-8-[3-[4-(trifluoromethoxy)phenyl]propanoyl]-7H-pyrido[2,3-b]pyrazin-2-yl]acetonitrile N-(3,5-dichlorophenyl)sulfanyl-2-methylbutan-1-amine 2-bromo-6,8,10,10a-tetrahydro-5H-benzo[f]quinoline 1-ethylcyclopropane;[3-methanidylimino-4-(naphthalen-2-ylmethoxy)piperidin-1-yl]-[5-methylsulfonyl-6-(triazol-2-yl)pyridin-2-yl]methanone;uranium(2+) N-(2,6-dichlorophenyl)-7-[1-methylsulfonyl-3-(trifluoromethyl)pyrazol-4-yl]-5H-[1,3]thiazolo[3,2-a]pyridine-3-carboxamide 4-azidosulfonyloxybenzamide ethane;4-[(2E,6Z)-octa-2,5-dien-3-yl]sulfanylaniline 1-[3-(6,7-dihydro-4H-triazolo[5,1-c][1,4]oxazin-3-ylmethoxy)piperidine-1-carbonyl]pyrazole-4-carbonitrile 1-[2-amino-3,6-bis(4-fluorophenyl)pyridin-4-yl]propan-2-one (7S)-5-methyl-6-pyridin-2-yl-3-[2-(trifluoromethoxy)phenyl]-2,4,5,7-tetrahydropyrazolo[3,4-c]pyridine 1-[1-(2-fluorophenyl)ethyl]cyclohexa-3,5-diene-1,3-dicarboxylic acid N-(2,3-dihydroindole-1-carbonyl)-2-methoxybenzamide 2-chloro-4-ethynylpyridine-3,5-dicarboxylic acid N-[(1,3-dimethylimidazol-1-ium-2-yl)methylidene]hydroxylamine N-[4,5-dimethoxy-2-nitro-3-(trifluoromethyl)phenyl]benzamide 4-[2-[[(1S)-3-(6,7-dimethoxyquinolin-4-yl)oxycyclohexa-2,5-dien-1-ylidene]amino]ethyl]piperidine-1-carboxylic acid (Z)-1-[5-[4,6-bis(3-bromophenyl)-1,3,5-triazin-2-yl]cyclohexa-2,4-dien-1-yl]but-2-ene-1,4-diimine 5-fluoro-3,4-dihydro-1H-pyrano[2,3-c]pyridine-8-carboxylic acid 4-(1,4-diazepan-1-yl)-2-[2-[6-(6-fluoropyridin-3-yl)pyridine-2-carbonyl]cyclopropyl]benzonitrile N-[6-(2,4-dichlorophenyl)imidazo[1,2-a]pyridin-8-yl]cyclopropanecarboxamide 4-(3-cyclopentylpropoxy)-2,6-difluorobenzaldehyde (2R)-1-[5-(4,4-difluoropiperidine-1-carbonyl)-6-methylpyridin-3-yl]oxypropane-2,3-diol 3-[5-(difluoromethoxy)pyridine-3-carboximidoyl]-1H-pyridin-2-one 2-[4-[6-[2-(dimethylamino)ethoxy]-1H-indol-3-yl]phenoxy]-N,N-dipropylacetamide N-[5,8-dimethyl-6-(1-methylpyrazol-4-yl)isoquinolin-3-yl]piperidine-4-carboxamide N-[4,6-dimethyl-5-(3-phenylpropanoylamino)pyrimidin-2-yl]formamide;ethane;N,N,6-trimethylpyridin-3-amine 2-(4-methoxypiperidin-1-yl)-N',N'-dimethyl-N-[6-(naphthalen-1-ylsulfonylamino)pyridin-3-yl]ethanimidamide 2-(3,5-dihydroxyphenyl)ethylsulfanium;tetrakis[4-(2-methoxyethoxy)phenyl]boranuide 4-tert-butylbenzoic acid;1,3-difluoro-5-methoxybenzene 1-[(2S,3R)-2-methyl-4-[(6-pyridin-3-ylpyrimidin-4-yl)amino]pyrrolidin-3-yl]ethanol 1,7-dioxopyrido[2,3-d]pyrimidine-6-carboxamide 2-[(4-methylpiperidin-1-yl)methyl]-N-[6-[2-[5-[(E,3Z)-3-propoxyiminoprop-1-enyl]pyridin-2-yl]ethynyl]isoquinolin-3-yl]pyridine-4-carboxamide N-[[4-(dimethylamino)phenyl]methyl]cycloheptanecarboxamide;ethanol 3-(2,6-dimethylphenyl)-7-fluoro-1H-1,6-naphthyridin-4-one N-(4,6-dimethoxypyrimidin-2-yl)-4-[2-methylpropanoyl(phenacyl)amino]benzenesulfonamide [4-(3-bromo-2,5-difluorophenoxy)cyclohexyl]carbamic acid 4-azidosulfanyl-2-(3,5-difluorophenoxy)pyrimidine 5-[4-(3,3-difluoropiperidine-1-carbonyl)phenyl]imidazolidine-2,4-dione [6-(2,3-dichlorophenyl)pyrazin-2-yl]methanol;4-ethoxycarbonylpiperazine-1-carboxylic acid 1-[4-(2,3-dihydrothiophen-5-yloxymethyl)cyclohexa-1,3-dien-1-yl]pyridin-2-one 4-[5-(1,3-benzothiazol-6-ylamino)-6-methoxypyridin-2-yl]-N,N-diethylbenzamide 3-[2-(9H-fluoren-1-yl)ethynyl]cyclohexane-1,2-dicarbonitrile 4-(5,6-dihydroxynaphthalen-2-yl)oxybenzoic acid 2-amino-4,6-dichlorobenzenesulfonic acid 2-(3,5-dihydroxyanilino)-7H-purine-6-carboxylic acid 2-[5,6-difluoro-3-(1H-indol-7-yl)naphthalen-2-yl]acetic acid 2-[2-oxo-4-(trifluoromethyl)spiro[indole-3,1'-cycloheptane]-6-yl]oxy-N-[[5-(piperidin-1-ylmethyl)pyridin-3-yl]methyl]propanamide 1-[4-[3,5-bis(trifluoromethyl)phenyl]phenyl]sulfonyl-2-(diethoxyphosphorylmethylsulfanyl)pyrrolidine 2-methoxy-1,3-bis(2,4,6-trimethylphenyl)imidazolidine 4-[3-(5,6-dichlorobenzimidazol-1-yl)piperidin-1-ium-1-ylidene]butanoic acid 1-[(4-fluorophenyl)methyl]-3-[2-hydroxy-5-[6-[1-(1H-pyrrolo[3,2-b]pyridine-3-carbonyl)piperidin-4-yl]oxy-3,4-dihydro-1H-isoquinoline-2-carbonyl]phenyl]urea 4-[(5,6-dimethylpyrimidin-4-yl)amino]-2-methoxybenzoic acid 1,2-dimethyl-N'-[N'-(2-methylquinolin-5-yl)carbamimidoyl]guanidine 4-(azidooxymethyl)-2,6-dichloroaniline (5E)-5-[[3,4-bis(trifluoromethyl)phenyl]methylidene]-2-imino-1,3-thiazolidin-4-one 1-azidooxynaphthalene-2,6-diamine (5Z)-2-(4-bromophenyl)imino-5-[(3,5-dichlorophenyl)methylidene]-1,3-thiazolidin-4-one [4-[[3-[(E)-2-(7,11-dihydroindolo[2,1-c][1,4]benzodiazepin-5-yl)ethenyl]phenyl]methylideneamino]phenyl]urea [(4E,5Z)-5-ethylidene-1,2,3,6,7-pentamethyl-6H-inden-4-yl]boronic acid N-[(2S,3R)-5-(1H-imidazole-2-carbonylamino)-4-oxo-2-phenyl-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl]pyridine-3-carboxamide [2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]ethynyl]phosphane 4-[2-oxo-1-[(3R)-piperidin-3-yl]imidazo[4,5-b]pyridin-3-yl]cyclohexa-2,4-diene-1-carboxylic acid N-[3-(2,4-dimethyl-5H-1,3-thiazol-4-yl)phenyl]-2-hydroxycyclopentene-1-carboxamide 5-[3-(trifluoromethyl)phenyl]imidazolidine-2,4-dione ethane;6-methyl-N-propan-2-ylidenepyridine-3-carboxamide 2-(dimethylamino)-N-[5-[3-[4-(furan-3-yl)-1H-pyrrolo[3,2-c]pyridin-2-yl]-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]acetamide 2-[(7-chloroquinolin-4-yl)amino]-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxylic acid (2R)-4,5-difluoro-N-[[3-fluoro-4-(1H-pyrrolo[2,3-b]pyridine-4-carbonyl)phenyl]methyl]pyrrolidine-2-carboxamide 2-(2,4-dichlorophenyl)acetamide;4-[(E)-1-[5-ethoxycarbonyl-3,6-bis(trifluoromethyl)pyridin-2-yl]but-1-en-2-yl]-3-fluorobenzoic acid 5-[(1S,3R)-2,2-difluorocyclopropyl]-4H-pyrrolo[3,4-d]triazole 3-[(4,6-diaminopyrimidin-5-yl)oxymethylidene]azetidine-1-carboxylic acid;hydrochloride 2,4-dihydroxy-N'-(3-nitrophenyl)-N-oxo-5-propan-2-ylbenzenecarboximidamide 2-[4-(3,4,6,7,8,9-hexahydrobenzo[d][1]benzazepine-5-carbonyl)piperazin-1-yl]-N-oxoacetamide N-[3,5-dimethyl-4-(1,2,3,4-tetrahydronaphthalen-2-yl)thiophen-2-yl]formamide;6-fluoro-2-hydroxy-1H-indole 3-butyl-2,7-di(propan-2-yl)fluoren-9-one 3-[(4-hydroxyphenyl)methyl]pyridine-2,6-dicarboxamide 4-N,2-diamino-5-azidopyridine-3,4-dicarbonitrile 2,4-bis[(1R)-1-methoxyethyl]-6-propan-2-ylphenol N-(6,8-dichloro-4-hydroxy-3-methylquinolin-2-yl)acetamide 1-chloro-4-[(5,6-dimethyl-1-benzofuran-2-yl)-cyclopropylidenemethyl]cyclohexa-1,3-dien-5-yne 1-[(E)-3,5-dimethylhex-2-enoyl]-4-hydroxyquinoline-2-carboxylic acid 3-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]benzenethiol 3-(azidomethyl)-2,6-dichlorobenzoic acid 5-cyclopropyl-N,3-dimethoxy-2-(1H-pyrazole-4-carbonyl)benzamide 5-chloro-2-N,4-N-bis(1H-indol-3-yl)pyrimidine-2,4-diamine [4-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]-[3-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]methanesulfonic acid N-azido-1,5-dimethyl-4-phenylpyrazole-3-carboxamide 2-[N-(2,3-dihydroxypropyl)anilino]octanoic acid 3-(hydroxymethyl)-N-[1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-ylidene]benzamide 2-[5-(2,4-dichlorophenyl)-1H-pyrazol-4-yl]-N-[4-[1-[4-(trifluoromethoxy)phenyl]piperidin-3-yl]butyl]acetamide N-[5-(2,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-4-(4-methylpiperazin-1-yl)benzamide 4-[4-hydroxybutyl(2H-tetrazol-5-yl)amino]butan-1-ol 2-(4,5-dimethylthiophen-3-yl)oxyacetaldehyde 2-[(3S,4R)-4-hydroxy-1-methylpyrrolidin-3-yl]-N-(furan-2-ylmethyl)acetamide 2-fluoro-N-[5-(1,3,4-oxadiazol-2-yl)-2-piperidin-1-ylphenyl]pyridine-3-sulfonamide N-(diaminomethylidene)-2-[[4-(3,5-dichlorophenyl)-2,6-bis(trifluoromethyl)phenyl]sulfinylamino]acetamide 3-[1,3-dimethyl-5-(pyridin-2-ylamino)pyrazol-4-yl]cyclopropane-1,1,2,2-tetracarbonitrile 4-(7-cyanoimidazo[1,2-a]pyridin-3-yl)-N-cyclopropyl-2-(difluoromethoxy)-6-hydroxybenzamide (5S)-2-amino-3,3'-dimethylspiro[5H-pyrano[2,3-d]pyrimidine-6,1'-cyclohexane]-4-one N-benzylsulfonyl-1-chlorocyclohexa-2,4-diene-1-sulfonamide ethane;6-methoxy-4-[4-(2,3,5,6-tetrafluorophenyl)cyclohexyl]oxyquinoline (5S,7R)-N-[3-cyano-4-(trifluoromethyl)phenyl]-5-(4-ethoxyphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide 1-[2-(cyclopentylmethoxy)ethyl]-N,3-dimethylpyrazole-4-sulfonamide 2-[1,3-dimethyl-6-(1H-pyrazol-4-yl)pyrazolo[3,4-b]pyridin-5-yl]oxyethanamine;propane N-[1-(6,7-difluoroquinoxalin-2-yl)pyrrolidin-3-yl]benzamide 6-[(Z)-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]prop-1-enoxy]quinoline (4R,5S)-2-benzylsulfanyl-N'-hydroxy-4,5-bis(phenylmethoxy)pentanediamide (2E,4Z)-3-(3-benzylphenyl)sulfanylhepta-2,4-dienoic acid 2-[2-methylpropyl(propan-2-yl)amino]-3H-quinazolin-4-one N-[3-[2-(3,5-dimethoxyphenyl)ethyl]-4H-azepin-7-yl]formamide N-[(Z)-1H-indol-3-ylmethylideneamino]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide 1-[6-fluoro-3-(propan-2-ylsulfamoyl)quinolin-7-yl]oxy-4-methylidenepentane-2,3-dione 2-[1-azido-5,6-bis(4-chlorophenyl)hexyl]thiophene 2-(4-ethylphenyl)-7,9-difluoroquinolizin-5-ium 1-[(3-methoxyphenyl)methyl]-5-methylimidazole N-[5-[2-[(4-chlorophenyl)methylamino]acetyl]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-3-yl]-4-(2-sulfanylethoxy)benzamide ethane;2-[3-(3-methylphenyl)-4,5-dihydro-1H-pyrazol-5-yl]propanoic acid 4-[(4S,5S)-2-(4-bromophenyl)-3-pyridin-4-yl-4,5-dihydroimidazole-1,2-oxazolidin-4-carbonyl]benzaldehyde (4S)-5,6-dimethoxy-4,8-dihydrochromene-2,3-dicarboxylic acid 6-amino-N,N-diethylpyridine-3-carboxamide 3-[2-[4-(benzylidenecarbamoylamino)phenyl]ethylcarbamothioyloxymethyl]butanoic acid 1-(1-benzylindole-3-carbonyl)-N,N-dimethylpiperidine-4-carboxamide (4-aminophenyl)-[3-[2-chloro-5-fluoro-4-[(1-methylpiperidin-4-ylidene)methyl]phenyl]azetidin-1-yl]methanone 4-[(5-azidosulfonylthiophene-2-carbonyl)amino]thiophene-3-carboxylic acid 5-ethyl-4-N-(2-methoxyphenyl)pyrimidine-2,4-diamine 2-(4-bromophenoxy)-N-[(Z)-(3,5-dichloro-2-hydroxyphenyl)methylideneamino]acetamide N-[4-[3-(1,1-difluoroethyl)phenyl]-2H-pyrazolo[3,4-b]pyridin-6-yl]propanamide 3-(2,6-dioxopiperidin-3-yl)-N-[5-methyl-4-[1-[2-(propan-2-ylideneamino)ethyl]piperidin-4-yl]sulfanyl-1H-pyrrolo[2,3-b]pyridin-3-yl]benzamide 2-bromo-1-fluoro-4-[(E)-3-nitroprop-1-enyl]benzene 2-[2-chloro-4-(hydroxymethyl)phenyl]sulfanyl-4-propyl-1H-pyrimidin-6-one (4R)-2-amino-3,8-dihydroxy-N-[(2S)-1,1,1-trifluorobutan-2-yl]-4H-pyrimido[5,4-c]quinoline-6-carboxamide 5-methyl-N-[(1S)-2-[4-(2,3,6-trifluorophenyl)piperazin-1-yl]cyclohexyl]-1H-imidazole-2-carboxamide 6-amino-4-methyl-2-sulfanylidene-4-(3,4,5-trimethoxyphenyl)-1,3-dihydropyrimidine-5-carbonitrile 6-(4,5-dihydro-1H-imidazol-2-yl)-3,5-bis(trifluoromethyl)imidazo[4,5-b]pyridine 5-[3-(4-methylsulfonylpiperazine-1-carbonyl)anilino]pyridazine-3-carboxamide 4-[(E)-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-ylhydrazinylidene)methyl]benzene-1,3-diol N-[(2,4-dihydroxyphenyl)methyl]pyridine-3-carboxamide;dihydrochloride 2-[[4-(3-cyanophenyl)pyridin-3-yl]methylideneamino]-N,N-diethyl-2-sulfanylacetamide 1-(3-tert-butyl-2,4,6-trimethoxyphenyl)hexane-1,1,5-triol 3-[1-methylsulfanylprop-2-enyl(5,6,7,8-tetrahydronaphthalene-2-carbonyl)amino]propanoic acid 1-[2,5-bis(trifluoromethyl)phenyl]-3-tert-butyliminoprop-1-en-1-amine N-(1,3-benzodioxol-5-ylmethyl)-N'-[1-[4-(2H-tetrazol-5-yl)phenyl]propan-2-yl]ethane-1,2-diamine 2-[2-(2,3-dihydroindol-1-yl)ethylimino]imidazolidine-4,5-dione 2-[N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)anilino]decanoic acid N-[2-(dimethylamino)ethyl]-3-naphthalen-1-yloxybenzamide [2-(6-methoxypyridin-3-yl)oxyphenyl]methanol 1-benzyl-N',2,5-trimethylpyrrole-3-carboximidamide 3-(cyclobutylmethoxy)-N-[2-(4-methylphenyl)ethyl]thiophene-2-carboxamide;2,2,2-trifluoroacetic acid 3-[8-amino-1-(4,6-dimethylpyridin-2-yl)imidazo[1,5-a]pyrazin-3-yl]cyclohexa-2,4-dien-1-one 4-[(Z)-[[2,6-dihydroxy-3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]methylidenehydrazinylidene]methyl]benzoic acid N-methyl-1-[2-(4-methyl-6-oxo-1H-pyrimidin-2-yl)-5-phenylpyrazol-3-yl]-5,6-dihydro-4H-cyclopenta[c]pyrazole-3-carboxamide 4-[5-chloro-1-(2,6-dimethylphenyl)pyrazole-3-carbonyl]piperazine-1-carboxylic acid [4-amino-2,5-di(propan-2-yl)phenyl]urea N'-(4-chlorophenyl)-3,6,7-trimethyl-5-piperidin-1-yl-2H-furo[2,3-e]benzimidazole-2-carboximidamide 2-(6,8-dimethylimidazo[1,2-a]pyrazin-3-yl)ethanamine 2-[(1,3-benzodioxol-5-ylamino)methyl]benzenecarboximidamide N-(4,4-difluoropiperidin-3-yl)-5-[[6-[2-(dimethylamino)ethoxy]quinoline-7-carbonyl]amino]pyrazolo[1,5-a]pyridine-7-carboxamide [4-(2,5-dimethylphenyl)piperazin-1-yl]-(3-nitropyridin-2-yl)methanone N-[4,5-difluoro-2-(1-hydroxypyridin-1-ium-3-yl)phenyl]methanesulfonamide 3-(4-methylcyclohexanecarbonyl)-1,2,4,5-tetrahydropyrrolo[2,3-d]azepine-7-carbonitrile 3-[4-(2-methylimidazol-1-yl)phenyl]-5-piperidin-4-yl-1,2,4-oxadiazole 4-[1-(3,5-dimethylphenyl)ethenoxy]-2,6-difluorophenol 2-[[2-(4,5-diphenyl-1H-imidazol-2-yl)indol-6-ylidene]amino]benzoic acid 1-cyclohexyloxy-3-(trichloromethyl)benzene (2R)-1-[3-(6-fluoroquinolin-4-yl)propanoyl]piperidine-2-carboxamide 5-[1-(4-chlorophenyl)ethyl]-2,3,6,7-tetrahydrocyclohepta[d]triazol-4-one 4-(3,5-dichlorophenyl)-1-methyliodanuidylpiperazine (4-azidopiperidin-1-yl)-[2-fluoro-6-methoxy-3-[[2-[(4-nitropyrazol-1-yl)methyl]benzoyl]amino]phenyl]methanone 2-[4-(cyclopentylamino)piperidin-1-yl]-N,N-dimethylpyrimidine-5-carboxamide N-[(Z)-1-aminoethylidenecarbamothioyl]-4-[3,5-bis(trifluoromethyl)phenyl]butanamide (5R)-2-benzylsulfanyl-8,8-dimethyl-5-phenyl-5,7,9,10-tetrahydro-3H-pyrimido[4,5-b]quinoline-4,6-dione 2-[N-(3,5-dichlorophenyl)-4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]anilino]ethanol 2-[3,5-difluoro-N-(oxan-4-yl)anilino]prop-2-enal 7-chloro-1-[(2S)-3,3-dimethylbutan-2-yl]oxyisoquinoline 1-[2-azido-6-(2,3-dimethoxyphenyl)-5-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]ethanone [2-(aminomethyl)morpholin-4-yl]-(1H-pyrazol-5-yl)methanone 1-(4-chlorobenzoyl)-3-(2,6-dimethylphenyl)imidazolidin-2-one N-methyl-5,6-bis(2,3,4,5,6-pentafluorophenyl)-1H-pyridine-2-thione 7-[2-(3-fluoroazetidin-1-yl)ethoxy]-6-methoxy-4H-1,4-benzoxazin-3-one 2-azido-1-(trifluoromethoxy)naphthalene 6-[(2,5-difluorophenyl)methyl]-2-methyl-1H-benzimidazole 5-[(4S)-1-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]-2-nitrobenzenesulfonamide 1-benzyl-N-(2,6-difluorophenyl)-5,8-bis(ethenyl)-7H-purin-6-imine 2-[5-carbamoyl-9-(furan-3-ylmethyl)carbazol-4-yl]-2-hydroxyacetic acid N'-(2-aminoethyl)-4-[[4-[N'-[6-chloro-3-(trifluoromethyl)carbazol-9-yl]carbamimidoyl]benzoyl]amino]butanimidamide 4-bromo-1-ethylsulfonylindazole 7-(4-methylphenyl)sulfanylheptanenitrile N-[5-bromo-2-(4,5-dihydrotriazolo[1,5-a]quinoline-7-carbonylamino)phenyl]carbamate N'-(3-amino-4,4-difluoropentyl)-2,5-bis[(6-methoxypyridine-3-carbonyl)amino]pyrazole-3-carboximidamide N-[(2R)-3-hydroxy-1-(4-morpholin-4-ylanilino)-1-oxobutan-2-yl]-4-methoxybenzamide 3-[2-(butoxycarbonylamino)ethyl]-6,8-dichloro-4H-chromene-2-carboxylic acid N-[4-[2-(3,5-dimethylanilino)thieno[3,2-d]pyrimidin-6-yl]phenyl]-1,2-oxazole-4-sulfonamide N-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]-3-methoxybenzamide N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-methoxy-6-methyl-N-phenyl-1,3,5-triazin-2-amine 4-(1,3-dioxan-2-yl)benzonitrile 1-[3-(2-aminoethylamino)phenyl]pyrimidine-2,4-dione 4-(2,5-dimethoxyphenyl)sulfonyl-1H-pyrrole-3-carboxylic acid 1-[5-[(3R)-2,6-dioxopiperidin-3-yl]oxy-7-methylspiro[1H-indole-3,4'-thiane]-2-yl]-3-ethylurea (6S)-2,8-bis[5-bromo-2-(dimethylamino)phenyl]-3-oxooctanoic acid 3-(2,5-diphenylfuran-3-yl)-1-azaspiro[4.4]nonane 3-butyl-4-oxothieno[2,3-d]pyrimidine-5-carbonitrile 4-ethyl-N-[1-(2-methoxyethyl)benzimidazol-2-yl]piperazine-1-carboxamide N-[3,5-dichloro-4-(trifluoromethyl)phenyl]-2-[6-[4-methoxy-7-(3-methylsulfonylpropoxy)quinazolin-6-yl]oxyquinolin-3-yl]acetamide N-[4-(methylamino)phenyl]-1,2-dihydronaphthalene-1-carboxamide 5-fluoro-3,7,9-trimethoxyanthracene 1-[(2R,5S)-2-(3,4-difluorophenyl)-5-(2-methylpropanoylamino)piperidin-1-yl]butan-2-ylideneazanium 4-ethoxycarbonyl-2,3,5,6-tetrafluorobenzoic acid 6-[(E)-2-carboxyethenyl]-7-hydroxy-1-methoxyquinolin-4-one;(6S,11R)-8-[(2-chlorophenyl)methoxy]-6-methyl-1,4-dioxa-8-azaspiro[4.5]decan-3-one 4-(1,1-dideuterioethyl)-2-methyl-5-[2-methyl-4-(trideuteriomethyl)phenyl]pyridine 4-(2,5-dioxoimidazolidin-1-yl)-N'-hydroxybenzenecarboximidamide 1-[4-[2-(methylideneamino)phenyl]sulfanylpiperazin-1-yl]ethanone N-[(2,3-dihydroxyphenyl)methylideneamino]benzamide (E)-3-phenyl-N-[5-[1-(2,4,6-trimethylbenzoyl)piperidin-2-yl]-1H-pyrazol-4-yl]prop-2-enamide (2R)-N-[(2S,3R)-1-amino-3-hydroxybutan-2-yl]-2-(4-hydroxyphenyl)propanamide;hydrochloride (2S)-3-[[1-[4-cyano-2-(trifluoromethyl)phenyl]piperidine-3-carbonyl]amino]-2-hydroxypropanoic acid 2-[2-(4-chlorophenyl)propyl]cyclobutan-1-one;ethane N-[2-(4-phenylmethoxyphenyl)propan-2-yl]hexanamide 4-[6-[5-[4,4-bis(4-methoxyphenyl)butanoyl]thiophen-3-yl]naphthalen-2-yl]benzonitrile (E)-N-[[4-(3,5-dimethylpyrazol-1-yl)phenyl]methoxy]butan-2-imine [3-(3,5-dimethylpyrazol-1-yl)piperidin-1-yl]-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)methanone 2-[3,5-difluoro-4-(1H-pyrazol-5-ylmethoxy)phenyl]-6-[2-[4-[[1-(cyclopropylmethyl)piperidin-4-yl]amino]phenoxy]ethyl]oxan-4-ol;formic acid 1-[(2,6-dichlorophenyl)methyl]-7-hydroxy-3,4-dihydroquinoxaline-2,3-dione 2-amino-9-[(3R,4S,5R)-3,4-dihydroxy-5-methyloxolan-2-yl]-1H-purin-6-one;trihydrochloride N-[2,6-difluoro-3-(iodoamino)phenyl]hydroxylamine 5-[1-(4-methylpiperidine-1-carbonyl)cyclopentyl]-2-phenyl-4H-1,2,4-triazol-3-one (7S)-2-(trifluoromethylsulfanyloxy)-3,4,6,7,8,9-hexahydropyrido[1,2-a]pyrazine (4Z)-1-cyclopentyl-4-[(2-methoxyphenyl)methylidene]-5,6-dihydroquinazoline (2S)-N,4-dimethyl-1-[(E)-3-naphthalen-2-ylprop-2-enoyl]pyrrolidine-2-carboxamide 5-[(3S)-6-(1H-indole-2-carbonylamino)-7-methoxy-4,9-dioxo-3a,6a-dihydrobenzo[f]isoindol-1-yl]pentanoic acid 3-[2-[(4-chlorophenyl)methyl]-6-oxo-1H-pyrimidin-5-yl]propanamide (1-azidopiperidin-4-yl)-(3,5-dimethoxyphenyl)methanone 1-N,4-N-dimethyl-6,7-dihydro-5H-pyrazolo[3,4-c]pyridine-1,4-dicarboxamide 2-[4-[2,2-diethoxyethyl(hexyl)amino]phenyl]acetonitrile N-(3,5-dimethoxyphenyl)-4-ethylbenzamide;2,3-dihydroxypropanoic acid 2-[4-hydroxy-3,5-di(propan-2-yl)phenyl]acetic acid 2-[1-carboxyheptyl(2,2-diethoxyethyl)amino]benzoic acid 2,3-bis(ethenyl)-1-[4-methoxy-6-(trifluoromethoxy)-3,4-dihydro-2H-chromen-8-yl]-9H-fluorene 6-chloro-N-cyclohexyl-2,4-dimethoxypyrimidine-5-sulfonamide 2-[3-(5,6-diaminopyridin-2-yl)piperidine-1-carbonyl]benzoic acid [2-chloro-4-(fluoromethyl)phenyl]-[7,7-dimethyl-5-(1H-pyrrolo[3,2-b]pyridin-6-ylmethoxy)-5,6-dihydropyrrolo[1,2-d][1,2,4]triazol-2-ium-3-yl]methanone (2R)-2-[[4-(6-fluoroquinolin-4-yl)piperidine-1-carbonyl]amino]-3-phenylpropanoic acid N-[(Z)-2-amino-3-[amino(methyl)amino]prop-1-enyl]-5-bromopyridine-3-carboxamide (2Z,3R)-1-[4-chloro-5-[(E)-1,2-difluoroprop-1-enyl]thiophen-2-yl]-N'-hydroxy-6,7-dimethylocta-2,6-dienediamide 4-[2,6-dichloro-3-(propanoylamino)phenyl]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide 4-methoxybenzenecarboximidate;tetraphenylphosphanium N-[4-(2,3-dimethylphenyl)-6-(2-hydroxypropan-2-yl)pyrimidin-2-yl]-7-ethoxy-1H-indole-4-carboxamide 7-azido-1,8-diphenylimidazo[4,5-f]quinoline (3S)-N-[6-(2,5-dioxopyrrolidin-1-yl)oxypyridin-2-yl]oxolane-3-carboxamide 1-[4-(2-methylpyridin-3-yl)phenyl]ethanone 3-[1-(2,4,6-trimethylphenyl)azepan-4-yl]-1H-benzimidazol-2-one 4-[5-chloro-2-(trifluoromethoxy)phenyl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione N-[3-[[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]methyl]cyclobutyl]formamide 2-[3,5-dichloro-4-[(6-cyclopropylimidazo[1,2-a]pyridin-7-yl)methoxy]phenyl]-3,5-dioxo-1,2,4-triazine-6-carbonitrile 2-azido-1,3-diethoxy-4-methylbenzene 7-methylsulfanyl-1,6,8,10,11-pentazatricyclo[7.3.0.02,4]dodeca-2(7),3,5,8,11-pentaene 1-cyclohexyl-3-[2,6-di(propan-2-yl)phenyl]urea 2-methyl-N-[4-(1-methylindole-3-carbonyl)phenyl]furan-3-carboxamide (2S)-5-amino-2-[(6-chloropyrazine-2-carbonyl)amino]-N-[(1R)-2,3-dihydro-1H-inden-1-yl]pentanimidate N-cyclopropyl-1-(3-ethyl-2H-benzimidazole-1-carbonyl)pyrrolidine-3-carboxamide 2-[(1E)-1-aminobuta-1,3-dienyl]aniline;6-methoxy-2,4-bis(pyridin-3-ylmethyl)benzaldehyde 2-[(1R)-1-carboxyethyl]-6-hydroxybenzoic acid 3,5-difluoro-N-[[4-methyl-2-(1H-pyrrol-3-yl)pyridin-3-yl]methyl]aniline 2-[4-[7-chloro-5-(2,3-dimethoxyquinoxalin-6-yl)-1H-indol-2-yl]-1-ethylsulfonylpiperidin-4-yl]acetonitrile [5-bromo-2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)phenyl]azanium [6-(2,3-dihydro-1H-inden-5-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-pyrrolidin-1-ylmethanone 3-chloro-N-[(2R)-1-hydroxy-4-methylpentan-2-yl]benzenesulfonamide 2-[1-cyclopropyl-5-(3,7-dimethyloctoxy)indole-3-carbonyl]benzoic acid (E)-3-(2,4-dinitrophenyl)-N-[4-methylsulfanyl-6-(trifluoromethyl)pyridin-3-yl]prop-2-enamide 6-methoxy-4-[3-(pyridin-2-yldisulfanyl)propylamino]pyridazine-3-carboxamide (6S)-2,6-dimethyl-3-[4-(trifluoromethoxy)phenyl]-5H-cyclopenta[b]pyran (1-azidocyclohexyl)methoxybenzene 6-[3-[2-[[1-(benzenesulfonyl)piperidin-4-yl]amino]ethoxy]phenyl]pyridine-3-carboxamide 5-(4,4-diphenylpiperidin-1-yl)sulfonyl-2-(2-phenylethoxymethyl)benzoic acid N-[(2E,4Z)-1,3,6-trimethyl-5-[(Z)-propylideneamino]octa-2,4-dien-2-yl]benzamide 5-[(6-fluoroquinolin-7-yl)methylidene]-1,3-thiazolidine N-ethyl-6-methoxy-7-(2,3,4-trifluorophenyl)quinazolin-4-amine 1-[(3-bromo-5-chlorophenyl)methyl]pyrrolidine 2-[(4,6-dimethylpyrimidin-2-yl)amino]-N-[1-[2-(6-morpholin-4-ylpyridin-3-yl)oxyethyl]cyclohexyl]acetamide 1-(1-hydroxycyclopentyl)sulfonyl-3-[6-methoxy-2,5-di(propan-2-yl)pyridin-3-yl]urea 5-[(4-methylphenyl)sulfonylamino]-N,2-dipropylbenzamide 2,7-dibromo-9H-fluorene;hydrochloride N-(1H-indol-5-ylmethyl)-1-[(2S,3R,4S,5S)-3,4,5,6-tetrahydroxyoxan-2-yl]methanesulfonamide 2-[(3R,4S)-1-[(3-fluorophenyl)methyl]-3-hydroxypiperidin-4-yl]-N-pyrrolidin-1-ylacetamide;2,2,2-trifluoroacetic acid 2-(1H-pyrrolo[3,2-c]pyridin-4-yl)spiro[3a,5,6,7a-tetrahydropyrrolo[1,2-b][1,2]oxazole-3,4'-piperidine];dihydrochloride N-(6,7,8,9-tetrahydrodibenzofuran-2-ylmethylideneamino)aniline 4-[1-(2-hydroxyethyl)indol-3-yl]butanamide (2S)-3-[1-[(3,5-difluorophenyl)methyl]indol-3-yl]-3-(methanesulfonamido)propanoic acid N-ethyl-2-(3H-imidazo[4,5-c]pyridin-2-yl)quinoline-8-carboxamide 5-[(E)-1-methoxybut-2-en-2-yl]-3-phenyl-1,2-dihydrotriazolo[4,5-b]pyrazine 5-azido-2-(4-fluorophenyl)imidazo[1,2-a]pyridine (3-fluorophenyl)-[4-[(1Z,3E,5E)-4-iodo-6-methoxycycloocta-1,3,5-trien-1-yl]piperazin-1-yl]methanone N-[2-[5-(1,3-dioxoisoindol-2-yl)pyridin-3-yl]ethyl]-4-methylpentanamide N'-hydroxy-3-[(6-methylpyridin-2-yl)oxymethyl]benzenecarboximidamide 5-methyl-N-[4-(2-methylidenepentanoyl)phenyl]pyridine-3-carboxamide N'-[2,4,6-trichloro-3-(2-methylpropyl)phenyl]ethane-1,2-diamine 7-N,8-bis[(4-methoxyphenyl)methyl]-1-N,2-dimethylbicyclo[3.2.0]heptane-1,7-diamine N-[4-cyano-2-fluoro-5-(2H-tetrazol-5-yl)phenyl]cyclopropanecarboxamide N-ethyl-N,3-dimethyl-6-(4-phenylpyridin-2-yl)imidazo[1,2-a]pyrazin-8-amine (1R,5S)-3-[2-[6-amino-8-oxo-7-[4-(2-pyrrolidin-1-ylethoxy)phenyl]purin-9-yl]acetyl]-N-methylbicyclo[3.1.0]hexane-2-carboxamide 2-[4-(dimethylamino)butyl]-1,3-benzothiazol-6-amine [5-(3,4-dimethylcyclohepta-1,3-dien-1-yl)-2-fluorophenyl]methanamine N-azido-2,5-dimethoxynaphthalene-1-carboxamide 4-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-N-phenylpiperazine-1-carboxamide 1-[(3,4-difluorophenyl)methyl]piperidine;3-(4-oxoquinazolin-3-yl)azetidine-1-carboxylic acid 6-[(3,5-dimethylpyrazol-1-yl)methyl]-2-phenyl-3H-thieno[3,2-d]pyrimidin-4-one 2-[3-(5-bromopyridin-2-yl)oxypropyl]pyridine (2S)-3,3,7,7-tetramethyl-1-[4-[4-(2H-tetrazol-5-yl)phenyl]phenyl]heptan-2-amine (2R)-N-[3-(1-benzylpiperidin-4-ylidene)propyl]-2,7-dimethoxy-5,8-dihydroquinoline-3-carboxamide;hydrochloride 2-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]-7-(2,6-dimethylphenyl)-8H-pyrido[2,3-d]pyrimidin-5-one 2-chloro-6-(5-methoxy-1H-indol-3-yl)-4,5,7,8-tetrahydro-[1]benzothiolo[3,2-d]pyrimidine 4-[3,5-dimethyl-1-(2-piperidin-4-ylethyl)pyrrol-2-yl]morpholine;hydrochloride N-(6,7-dihydro-5H-cyclopenta[c]pyridazin-3-ylmethyl)-1-methylpyrazole-4-carboxamide 1-[3-(2-methylpropoxy)phenyl]ethanone 2-(1,3-benzodioxol-5-yl)propanedioic acid 1-[2,6-di(propan-2-yl)phenyl]-3-[[5-oxo-1-(4-propan-2-yloxyphenyl)-4H-1,2,4-triazol-3-yl]amino]thiourea 1-(5,6-dichloro-2H-pyrimidin-1-yl)propan-2-one 2-[2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)ethynyl]quinoline 3,6-dichloro-7-(2,4-dimethoxypyrimidine-5-carbonyl)-8H-quinolin-4-one N-[(4-chlorophenyl)methyl]-1,3-dimethanimidoyl-5-pyridin-4-yloxyindol-2-amine N-(2-nitrophenyl)-N-(4-phenyl-1,3-thiazol-2-yl)ethenesulfonamide 1-[(E)-2-[4-(furan-2-ylmethoxy)phenyl]ethenyl]-3,4-dihydronaphthalen-2-ol 6-methoxy-N,2-dimethyl-4-[(E)-1-(methylideneamino)prop-1-en-2-yl]-7H-imidazo[4,5-c]pyridine-3-carboxamide N-[3-fluoro-4-(1,5,7,10,11-pentazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-12-ylcarbamoylsulfamoyl)phenyl]-4-methoxypyridine-2-carboxamide 4-(3,5-dimethylpyrazol-1-yl)-1H-pyrimidine-4,6-diamine 3-(6-hydroxynaphthalen-2-yl)sulfanyloxypropane-1,2-diol 4-[5,6-dimethyl-4-(methylamino)pyridine-2-carbonyl]piperazine-1-carboxylic acid 4-[(1E,3Z)-2-[1-(5-tert-butylcyclohexa-1,5-dien-1-yl)ethylideneamino]penta-1,3-dienyl]benzenethiol 5-(4,6-dimethylpyridin-2-yl)oxypyrimidine-2,4-diamine 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-(4-sulfamoylphenyl)benzenesulfonamide 1-[3,5-bis(trifluoromethyl)phenyl]-4-(1H-pyrrole-2-carbonyl)piperazin-2-one 5-[5-(methylamino)pyridin-3-yl]-N-[6-(4-propan-2-ylpiperazin-1-yl)pyridin-3-yl]-1H-indazole-3-carboxamide 3-bromo-1,6-dimethylquinoxalin-2-one 3-(2-bromo-5,6-difluoropyrimidin-4-yl)-1H-indole 2-(6,7-dimethoxyquinazolin-4-yl)sulfanylethanethiol 3-(6,7-dihydro-4H-pyrano[4,3-d][1,2]oxazol-3-yl)-1-ethyl-5,8-dimethoxyquinolin-2-one 3-[2-(6-methyl-2,3-dihydro-1H-inden-5-yl)ethyl]pyrrolidine 1-[(E)-3,4-dimethylpent-2-en-2-yl]sulfanyloxy-2-fluorobenzene (3R,4S)-1-[4-cyano-3-(trifluoromethyl)phenyl]-4-[1-(1-methylindole-5-carbonyl)piperidin-4-yl]pyrrolidine-3-carboxamide N-[4-[5-amino-6-(pyridin-3-ylmethoxy)pyrimidin-4-yl]sulfanylphenyl]pyridine-3-carboxamide 2-(4-aminophenyl)-6,7-dihydroquinoline-3,5-diol;hydrobromide ethane;1-[(4R)-2,8,10-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-1,3,5(16),9,11,13-hexaen-12-yl]ethanone N-(1,1a,6b-dihydrocyclopropa[b][1]benzofuran-1-yl)-3-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)benzamide 2,4-difluoro-5-[6-(2-methyltetrazol-5-yl)pyridin-3-yl]aniline 1-(4-chlorophenyl)-3-ethyl-7H-purine-2,6-dione (4-chlorophenyl)-(2,3-dihydro-1H-isoindol-1-yl)methanone 3-(1-bicyclo[2.2.1]heptanyl)-5-methyltriazolo[4,5-d]pyrimidine (Z)-2,5-diaminopenta-1,3-diene;4-[(5-methoxypyridine-2-carbonyl)amino]benzoic acid 4-azido-2,6-difluoro-N-(1H-pyrrol-3-ylmethylideneamino)aniline (1R,5S)-6-[3-fluoro-4-(trifluoromethyl)phenyl]-2-prop-2-enoyl-9-oxa-2,17-diazatricyclo[8.7.0.011,16]heptadeca-10,12,14,18-tetraene-5,15-dione 2-(1,3-dimethoxybutan-2-yl)isoindole-1,3-dione 2-(difluoromethoxy)-N-[1,6-dihydroxy-4-(3-nitrosopropanoylamino)naphthalen-2-yl]benzamide N'-[(1S)-2,3-dihydro-1H-inden-1-yl]ethane-1,2-diimine (6Z)-1-chloro-4',8'-diphenylspiro[3H-pyrrolo[2,3-h]quinazoline]-2',7'-dione 2-(3,6-dioxocyclohexa-1,4-dien-1-yl)chromene-4-thione 1-(4-methoxyphenyl)sulfanylpiperidine;uranium(2+) (E)-5,6-dimethylnon-4-en-3-one;N-ethyl-2,2,2-trifluoro-N-[[4-[[6-(1H-indole-4-carbonylamino)pyridine-3-carbonyl]amino]phenyl]methyl]heptanamide 1-azidooxy-3,5-dichloro-2-(4-methylphenoxy)benzene 2-[3,5-dimethyl-1-(5-propan-2-ylpyridine-3-carbonyl)pyrazol-4-yl]-N-ethylidene-N'-(oxolan-3-yl)propanediamide 5-N,6,8-trimethylquinazoline-2,4,5-triamine N-[5-(azepane-1-carbonyl)pyridin-2-yl]-N'-phenylethanimidamide N'-(6-bromopyridin-2-yl)-N,N-dimethylpropane-1,3-diamine 2-chloro-N-[[4-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]phenyl]methyl]-N-ethyl-6-methoxy-5-nitropyrimidine-4-carboxamide 2-methyl-N-[4-[(2Z,5E)-2,3,6,7-tetrahydroazocin-4-yl]phenyl]furan-3-carboxamide 2-[4-(4,6-dimethylpyrimidin-5-yl)oxycyclohexa-1,3-dien-1-yl]-N-phenylacetamide 2-[(1S)-3-(3,5-dichloropyridin-4-yl)oxycyclohex-2-en-1-yl]acetic acid 1-[3-cyclobutyl-7-(trifluoromethoxy)quinolin-4-yl]piperidine-2,6-dione;N'-propan-2-ylbenzenecarboximidamide N-methoxy-1,2-diphenylethenamine 3-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiophen-3-yl]-5,6-bis(trifluoromethyl)imidazo[4,5-b]pyridine 2-[4-(difluoromethyl)cyclohexyl]oxy-N-ethylsulfanylaniline [(2R,4S)-4-azidopyrrolidin-1-yl]-(3-chlorophenyl)methanone 4-[5,8-bis(ethenyl)naphthalen-1-yl]-2H-tetrazole 3-[6-(1,3-benzodioxol-5-yl)-2-morpholin-4-ylpyridine-3-carbonyl]benzoic acid N-(4,5-difluoro-2-hydroxyphenyl)pyridine-2-carboxamide 4-[2-(cyclopropylmethoxy)ethylamino]-1H-pyrimidin-6-one 2-[4-(N-butanoyl-2-nitroanilino)phenyl]sulfonylbenzenesulfonic acid 5-[7-(2,6-difluorophenyl)-2-methyl-3H-benzimidazole-4-carbonyl]thiophene-2-carboxylic acid (2S)-4,8-dimethoxy-1,7-dimethyl-5,10b-dihydro-2H-isochromeno[3,4-h]quinoline 4-(2,5-dioxopyrrol-1-yl)-6-(6-ethoxypyridin-3-yl)benzene-1,3-disulfonic acid 4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)morpholine-4-carbonyl]-2-(methoxymethyl)pyrrolidine-1-carboxylic acid 2-(benzenesulfonamido)-3-[4-(cyclopenten-1-yl)phenyl]propanoic acid 2-[(3,5-dimethoxyphenyl)methyl]propane-1,4-diol 5-[2,4-difluoro-N-(3-methylbutyl)anilino]pentan-1-ol 2-[2-methyl-N-[(3-nitrophenyl)methoxycarbonyl]anilino]decanoic acid ethane;N-[4-[5-[[2-hydroxy-3,6-dimethyl-5-(oxiran-2-yl)phenyl]methylideneamino]naphthalen-1-yl]oxybutyl]formamide N-[2-[4-(1H-benzimidazole-2-carbonyl)piperazin-1-yl]ethyl]acetamide;6,7-dimethoxy-2-methyl-3,4-dihydroisoquinolin-1-one 3-[(Z)-[(E)-2,3-diaminoprop-2-enylidene]amino]sulfanyl-N-[1-(4-ethoxyphenyl)ethyl]aniline N-[5-[1,2-diamino-6-(2,3-dihydrothiophen-2-yl)indol-3-yl]-2-hydroxyphenyl]acetamide 1-(4-propan-2-ylphenyl)sulfonylindole 4-[8,14-bis(2-hydroxyphenyl)-11-thia-3,5,13,15-tetrazatetracyclo[7.6.0.02,6.010,12]pentadeca-1(9),2,4,6,10(15),11-hexaen-4-yl]phenol ethane;N-[[4-fluoro-3-[5-(trifluoromethyl)pyridin-2-yl]phenyl]methyl]-2,3,4,5,6-pentafluorobenzamide 1-N,2-N-bis[(4-amino-5-oxotetrazol-1-yl)methoxy]benzene-1,2-disulfonamide;3-methylpyridine (1-phenylcyclopropyl)-[2-[[4-(trifluoromethyl)pyridin-3-yl]oxymethyl]pyrrolidin-1-yl]methanone (Z)-4-[3,5-bis(4-chlorophenyl)phenyl]but-2-enal;propane 3-[(5-fluoropyridin-2-yl)methylamino]cyclopentane-1-carboxylic acid N-[(3,4-dimethoxyphenyl)methyl]-5-fluoro-2-hydroxybenzamide 4-(2,3-difluorophenyl)pyridine;3-[[(3R)-piperidin-3-yl]methoxy]-1H-pyrazolo[3,4-b]pyridine 2-[(1R,5S)-3-azidooxy-6-azabicyclo[3.1.0]hexan-6-yl]-1,4,7-trimethylbenzimidazole 6-chloro-3-(2,2-difluoroethyl)pyrido[1,2-a]pyrimidin-4-one 1-cyclopentyl-N-[(3,4-difluorophenyl)methoxy]-4-[4-(hydroxymethyl)piperidin-1-yl]sulfonylpiperidine-4-carboxamide 4-(5,6,7,8-tetrahydroquinazoline-2-carbonylamino)benzoic acid 5-[3,5-difluoro-4-(trifluoromethyl)phenyl]-1-ethanimidoyl-7H-2,6-naphthyridin-8-imine [2-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-piperazin-1-ylmethanone 1-cyclopropyl-4-fluorobenzene;methanamine;4-[1-(methylamino)pentan-3-yl]benzaldehyde 2-benzylsulfanyl-6-[(4-chlorophenyl)methoxy]-N-[(E)-1,3-dihydroxypropan-2-ylideneamino]quinoline-4-carboxamide 4-[3-(difluoromethoxy)phenyl]-2-ethylsulfanyl-1H-pyrimidin-6-one 3-[6-(3,3-difluorocyclobutyl)oxypyridazin-3-yl]azetidine-1-carboxylic acid (2-aminophenyl)-[4-[2-(1,3,5-trimethylpyrazol-4-yl)ethoxy]piperidin-1-yl]methanone 5-[2-(4-bromo-3,5-dimethoxyphenyl)ethyl]-1,2,3-trifluorobenzene 6-[[3-amino-2,2-difluoro-4-(methylamino)butylidene]amino]-3H-1,3-benzoxazol-2-one 4-[[3,5-diamino-2-(1H-indole-4-carbonyl)phenyl]methyl]piperazine-1-carboxylic acid 3-[3-fluoro-4-[5-[(1E,3Z)-penta-1,3-dienyl]furan-2-carbonyl]phenyl]propanoic acid 2-(6,7-dichloro-1H-benzimidazol-4-yl)propanamide 5-hydroxy-3,4,6-trimethylpyridine-2-carboximidamide 2-methylsulfanyl-6-[(4-propan-2-ylphenyl)sulfonylamino]quinoline-3-carboxylic acid;trihydrochloride (4-azidocyclohexyl)benzene 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(4-hydroxyphenyl)propyl]acetamide N-(4-iodopyridin-2-yl)-5,6-dihydroquinoline-3-carboxamide 6-[(4aS,9aR)-8-methylsulfonyl-1,2,3,4a,5,7,8,9,9a-decahydropyrido[3,2-e][1,4]diazepine-3-carbonyl]pyridine-3-carbonitrile 3,4-dihydro-2H-quinoline;N,3-dimethyl-N-[(5Z)-7-methylidene-5-propan-2-ylidenedeca-1,9-dien-2-yl]aniline 2-[3-(hydroxymethyl)piperazine-1-carbonyl]benzonitrile 2-(4-chlorophenyl)-6-N,8a-dihydroimidazo[1,2-a]pyridine-3,6-diamine N-[2-[(1-methylpyrazole-4-carbonyl)amino]ethyl]-6-azaspiro[3.5]nonane-8-carboxamide 3-hydroxy-N-methyl-4-[(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)oxy]benzamide [4-methyl-3-(methylamino)phenyl]imino-oxoazanium 4-[(Z)-2-hydrazinylethenoxy]-3,5-dimethoxybenzoic acid (5Z)-3-(2,5-dimethoxyphenyl)-4-imino-5-[[1-[2-oxo-2-[[5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]amino]ethyl]piperidin-4-yl]methylidene]-1,3-thiazolidin-2-one 7-chloro-2-[(2R,6S)-2-ethyl-6-methylmorpholin-4-yl]-N-[(1R)-3,3,3-trifluorocyclohexyl]-1,3-benzoxazol-5-amine 2,3-dichloro-1-[(4-methoxyphenyl)methyl]indole 2-(3,4-dichloroanilino)-N-[(Z)-(2-hydroxynaphthalen-1-yl)methylideneamino]acetamide 1-(2,5-dichlorothiophen-3-yl)sulfonyl-N-[4-methoxy-6-(pyrazol-1-ylmethyl)pyrimidin-2-yl]azetidine-3-sulfonamide 1-(2,6-diaminopyrimidin-4-yl)-3-[5-(trifluoromethoxy)indol-1-yl]propan-2-ol 2,3-dihydroindole;2-[1,4-oxazepan-6-ylmethyl(pentyl)amino]-1H-pyridin-4-one 5-chloro-4-fluoro-1,3-dimethylindole (2E)-2-[3-chloro-4-(3,5-dimethylpyridin-2-yl)sulfanyl-1H-pyridin-2-ylidene]propanenitrile 1-[4-(4-fluorophenyl)sulfonyl-2,3-dihydropyrido[3,2-b][1,4]oxazin-6-yl]prop-2-en-1-one N-benzyl-2,3-bis(methylideneamino)cyclopent-2-en-1-imine 2-[3,5-dibromo-4-(hydroxymethyl)-1H-pyrrol-2-yl]acetic acid 3-[[4-(2,2-dichloropropanoyl)phenyl]methoxycarbonylamino]-6-(phenylcarbamoyl)hexaneperoxoic acid 2-hydroxy-N-(1H-pyrazole-5-carbonyl)butanamide 2-[(5R,10bS)-7-methoxy-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol N-[(2S)-5-amino-1-[6-(4-aminopiperidine-1-carbonyl)-7,8-dihydroimidazo[1,2-a]pyridin-3-yl]-1-oxopentan-2-yl]-1H-indazole-3-carboxamide N-[1-(2,3-dihydro-1H-inden-5-yl)ethyl]-4-methylthiadiazole-5-carboxamide 2-[[3-(trifluoromethyl)phenyl]carbamoylamino]cyclohexane-1-carboxylic acid 2-(4-aminopyridin-3-yl)-N-[[4,6-difluoro-5-(1H-indol-2-yloxy)-2-methylcyclohexa-1,3-dien-1-yl]methyl]ethanamine 2-(4,6-dichloro-N-ethenylsulfonyl-1,3,5-triazin-2-yl)acetamide N-(3,4-dimethoxyphenyl)-2-(4-ethylpiperidin-1-yl)-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide 1-N',4-N'-bis[(3E)-hexa-1,3,5-trien-3-yl]benzene-1,4-dicarboximidamide 3-[(2E)-2,4-dimethylhepta-2,6-dienyl]benzamide 5-[2,4-bis(trifluoromethyl)phenyl]-2H-tetrazole 3-(azidomethyl)-5-nitro-6-(trifluoromethoxy)-1H-indole 5-[(2,6-dichlorophenyl)methoxy]pyrazine 2-(6-bromoimidazo[1,2-a]pyridin-3-yl)ethylcarbamic acid 3-cyclopentyl-2-[5-(3,5-dimethoxyphenyl)spiro[2H-1-benzofuran-3,4'-piperidine]-1'-yl]acetic acid 3-(azidomethyl)-2-tert-butylpyridine N-[5-(2,4-difluorophenyl)sulfonyl-6-methoxypyridin-3-yl]-1,3-dimethylpyrazolo[3,4-b]pyrazin-6-amine 2-[(E)-1-amino-3-methyliminoprop-1-en-2-yl]-N-[6-[4-(cyclohexanecarbonyl)piperazine-1-carbonyl]pyridin-2-yl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 1-[(4Z,5E)-2-amino-5-ethylidene-6-iminopyridine-3-carbonyl]-N-(1H-indol-7-ylmethyl)pyrrolidine-3-carboxamide;N'-(4-cyanobenzoyl)benzohydrazide (2S)-3,4-dihydroxy-2-[[2-(methylamino)ethyl-(4-phenylphenyl)sulfonylamino]methyl]-N-[1-[(2R,3R)-4-methyl-2,6-bis(sulfanyl)-3,5-dioxopiperazin-2-yl]-1-oxopropan-2-yl]butanamide (4R)-6-[5-[3,3-difluoropropyl(methyl)carbamoyl]pyridin-2-yl]oxy-N-[[3-fluoro-4-[3-[(3S)-oxolan-3-yl]pyrazin-2-yl]phenyl]methyl]oxepane-4-carboxamide 3-[(2R)-4,6-dichloro-1H-indole-2-carbonyl]oxy-3-oxopropanoate [(1R)-2-[2-benzylsulfanylethyl(methyl)amino]cyclopentyl]-phenylmethoxyphosphinic acid (1S)-N,N-dimethyl-2-[(3R)-4-phenylpyrrolidin-3-yl]oxycyclohexan-1-amine 6-[3,5-difluoro-2-(4-methylphenyl)pyridine-4-carbonyl]-N'-methanimidoylnaphthalene-1-carboximidamide 2-[(3S)-6-fluoro-1,3,4,9b-tetrahydrodibenzothiophen-3-yl]-1H-benzimidazole 2-hydroxy-4-methoxy-5,7-dihydroindolo[3,2-d][1]benzazepine 3-[1-(2,4-dimethoxyphenyl)ethenyl]quinoline;uranium(2+) 5-chloro-N-(2,4-difluorophenyl)sulfonyl-6-[1-oxo-7-(trideuteriomethoxy)-3H-isoindol-2-yl]pyridine-3-carboxamide 3-[2-(6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepin-2-yl)-1H-indol-3-yl]propanamide 2-(4-chlorophenyl)-N-[[3,5-difluoro-2-[hydroxymethyl(propan-2-yloxy)amino]phenyl]methyl]azetidine-1-carboxamide 4-[4,4-dimethyl-2-(4-oxo-3H-quinazolin-2-yl)pyrrolidin-1-yl]benzoic acid (3R)-4-[[6-chloro-2-(5-phenylpyrazol-1-yl)quinoline-4-carbonyl]amino]-2,3-dimethylpentanoic acid 2-[(4-hydroxy-3,5-dimethylphenyl)methylidene]-7-iminooctanoic acid 3,5-difluoro-N-[(2R)-1-hydroxypropan-2-yl]benzamide 1-[1-(3,5-dimethoxybenzoyl)piperidin-4-yl]-2H-pyrimidine-5-carboxylic acid 2-[6,7-dichloro-1-(4-methyl-2-oxopyridin-1-yl)isoquinolin-3-yl]acetamide N-[3-(2,4-difluorophenyl)-1H-indazol-5-yl]furan-2-carboxamide 2-[[5,6-difluoro-1-(4-methylpyridin-3-yl)benzimidazol-2-yl]oxymethyl]-N,N-bis(propan-2-ylsulfanyl)cyclopenten-1-amine 1-[(3,5-dichlorophenyl)methyl]-3-[1-(4-fluorophenyl)cyclobutanecarbonyl]quinolin-4-one N-[(5,6-dimethyl-2-oxo-4H-1,3-oxazin-4-yl)methyl]-3,5-difluoropyridine-2-carboxamide N-[2-(1,3-dimethyl-7-oxopyrrolo[2,3-c]pyridin-6-yl)ethyl]formamide 2-(N-(4,5-dimethylpyrimidin-2-yl)-3-nitroanilino)acetamide 2-[(E)-3-[4,5-bis(ethenyl)furan-2-yl]-1-(4-methoxyphenyl)prop-1-enyl]benzenesulfonic acid;ethane 4-[2-(6-methylpyridin-3-yl)ethynyl]cyclohexan-1-ol 2-hydroxy-5,6-dimethyl-3-[1-(3,4,5-trifluorophenyl)ethenoxy]benzoic acid (1R,2R)-N-[8-amino-6-[3-(trifluoromethyl)phenyl]isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 4-[2-[(2,6-difluorophenyl)methoxy]-3-methylphenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-[3-(hydroxymethyl)-4-(pyridin-3-ylsulfonylamino)phenyl]acetic acid 5-[2,4-dinitro-6-(trifluoromethyl)phenyl]-1,3,4-thiadiazol-2-amine 5-chloro-N-(5-cyclohexylpentan-3-yl)-2,4-difluoroaniline 2,2-dichloro-N'-[5-(4-hydroxyphenyl)thiophene-3-carbonyl]propanehydrazide 3-amino-2,6-dichloro-N'-(4-nitrophenyl)benzenecarboximidamide N-(2,4-dichlorophenyl)-1-(3-methylbutanoyl)pyrrolidine-2-carboxamide [(3S)-1-(4,5-difluorobenzoyl)pyrrolidin-3-yl]carbamic acid N-[3-chloro-4-(2,5-dioxopyrrolidin-1-yl)phenyl]-N-ethylcarbamate 1-(2,3-dimethylphenyl)-N,3-dimethyl-4-propan-2-ylimidazolidin-2-imine 2-[1-(4-chlorophenyl)sulfonylpiperidin-3-yl]acetic acid 2-methoxyimino-5-[(E)-pyridin-4-ylmethylideneamino]oxy-N'-tritylpentanimidamide (E)-4,7-dimethylnon-5-en-3-one;N'-[6-(4-fluoro-2-methoxyphenyl)imidazo[1,2-a]pyridin-2-yl]-N-(2-hydroxyethylamino)methanimidamide 1-(4-fluorophenyl)-5-oxo-N,6-diphenylmethoxytriazole-4-carboxamide 1-(2,4-dimethoxyphenyl)pentan-1-one (3Z)-N,2-dimethylpenta-1,3-dien-4-amine;6-(5-fluoropyridin-3-yl)-8-N,12-N,13-trimethyl-2-(4-phenoxyphenyl)pyrazolo[5,1-c][1,2,4]benzoxadiazole-3,8-dicarboxamide 6-ethylsulfinyl-1,3-benzothiazol-2-amine N-[[4-(methoxymethyl)thiophen-2-yl]methyl]-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamide 2-[1,4-dimethyl-3-(2-oxoethyl)cyclohexyl]isoindole-1,3-dione 1-[5-fluoro-2,3-di(propan-2-yloxy)phenyl]-N'-methylmethanesulfonohydrazide (2E)-N',2-diamino-N-[(Z)-5-methoxyhexan-3-ylidene]-5-methylbenzenecarboximidamide 5-bromo-3-fluoroacridine 2-(N-(1,3-diethoxy-1,3-dioxopropan-2-yl)-4-methoxycarbonylanilino)decanoic acid 2-(N,3-dimethylanilino)-4-[(Z)-(5-phenylfuran-2-yl)methylideneamino]-1H-pyrimidin-6-one 5-tert-butyl-2-[1-(4,6-dimethylpyrimidin-2-yl)ethyl]-3H-isoindol-1-one 2-(4-chlorophenyl)-N-[1-(2,3-dihydro-1H-inden-5-ylmethyl)pyrrolidin-3-yl]acetamide 2-(difluoromethoxy)-4-hydroxy-3,7-dimethyl-1H-naphthalene-2-carboxylic acid 7-[(5S)-4,6-diamino-3-azabicyclo[3.2.0]heptan-3-yl]-1,3-benzoxazol-2-amine 3-[8-fluoro-2-(4-methylphenyl)sulfonyl-4-oxochromen-6-yl]oxypropanoic acid 2-[1,3-benzodioxol-5-ylmethyl-(4-fluorophenyl)sulfonylamino]-N-[(Z)-(4-hydroxyphenyl)methylideneamino]acetamide 2,6-dichloro-1-ethylsulfinylbenzimidazole 2-[[2,5-difluoro-4-(1H-pyrazol-5-yl)phenyl]methylamino]-9-propan-2-ylpyrido[1,2-a]pyrimidin-4-one 5-[2,3-difluoro-4-[(1Z)-1-[6-methyl-3-propan-2-ylidene-2-(trifluoromethyl)-4H-pyridin-2-yl]buta-1,3-dienoxy]phenyl]thiophene-2-carboxylic acid;methane 2-[3-azido-1-(9H-fluoren-1-yl)cyclohexa-2,4-dien-1-yl]-1H-indole 4-[2-(1,3-benzothiazol-6-yloxy)ethyl]pyridine-2-carbonitrile 4-[(3Z)-4-aminohexa-1,3,5-trien-2-yl]phenol 6-[5-(3,4-dihydropyridin-2-yl)furan-2-yl]-7H-pyrrolo[2,3-d]pyrimidine 2-[2-amino-4-(diethylamino)pyrimidin-5-yl]propanedioic acid 6-[4-(dimethylamino)phenyl]-9,9-dimethyl-3,8-dihydro-2H-pyrimido[1,2-a]pyrimidin-7-one 2-(1,3-dioxoinden-4-yl)naphthalene-1,6-dione 2-[(4S)-1-tert-butyl-3,4-dimethylazepan-4-yl]oxyaniline [(3S)-4,5-diamino-1-oxopentan-3-yl]azanide;vanadium 5-[3-[(Z)-but-1-enyl]-4,7,8-trimethylbenzo[g]indol-2-yl]-N,3-dimethylfuran-2-carbothioamide 2-[2,3-dimethyl-4-(trifluoromethyl)phenyl]propanamide 7-methoxy-N,2-dimethyl-9-(1H-pyrazol-4-yl)purin-8-imine 2-amino-8-(4-hydroxyphenyl)sulfanyl-1,7-dihydropurin-6-one 3-[(E)-3,5-dimethylhex-2-en-4-ynoxy]-6-methoxy-1H-quinolin-4-one 1-[4-(2,3-dihydroindole-1-carbonyl)-5,6,7,8-tetrahydronaphthalen-1-yl]-3-methoxypropan-2-one 5-azidosulfanyl-4-(3,4,5-trifluorophenyl)pyrimidine 5-(3,4-dimethoxyphenyl)-2H-1,3,4-thiadiazol-5-amine 2-amino-N'-(1H-indole-3-carbonyl)pyridine-4-carboximidamide;ethane 4-[3-[1,3-bis(2-methylpropyl)imidazol-1-ium-2-carbonyl]oxyphenyl]sulfanylbenzoate 1-[(Z)-[5-hydroxy-3,4-bis(phenylmethoxy)oxolan-2-yl]methylideneamino]-4-phenylpiperazine-2,5-dione N-[4-(4,6-dimethylcyclohepta-1,3,5-trien-1-yl)phenyl]aniline 2-bromo-1,3-dibromo-4-cyclopropylbenzene N-(4-bromophenyl)-7,9-dimethyl-1,2,3,4-tetrahydropyrido[3,4-b]indole-8-carboxamide 2-(4-chlorophenyl)-1-[2-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylamino)pyrrolidin-1-yl]butan-1-one 3-[7,8-dimethyl-2-(oxan-4-yl)imidazo[1,5-a]pyrazin-6-yl]aniline 2-[6,7,8,9-tetrahydrodibenzofuran-3-yl(thiophen-2-yl)methyl]propanedinitrile 6-(4,5-diethyl-1H-pyrazole-3-carbonyl)-N-pyridin-2-yl-6-azaspiro[3.4]octane-8-carboxamide N-[5-(6,7-dihydro-1H-indole-2-carbonyl)-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-3-yl]pyridine-3-carboxamide 3-[(3S)-5-[2-(4-carbamoylanilino)-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-4-yl]-3-methylpentan-2-yl]benzoic acid (2R,3S,4R,5R)-1-[bis(deuteriomethyl)amino]-3-hydroxy-5-[(2R,4R)-4-phenylpentan-2-yl]oxyhexane-2,4-diol 4-[2-(2,3-dimethylphenoxy)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 1-(4,5,6,7-tetrahydroindazol-2-ylmethyl)piperidine 4-(6,7-dihydronaphthalen-2-yl)-5-(trifluoromethoxycarbonylamino)pyrazole-1-carboxylate 3-(2,4-dimethoxyphenyl)-1-ethylpyrrolidine 3-(1,6-dimethyl-2,4-dihydropyrrolo[3,4-d]imidazole-5-carbonyl)-N,N-diethylbenzenesulfonamide 4-(6-bromopyridazin-3-yl)oxy-N,N-dimethylbutanamide N-(1,3-benzodioxol-5-ylmethyl)-4-[(2S)-6-[2-(5-hydroxypyridin-3-yl)ethynyl]spiro[2H-1-benzofuran-3,3'-pyrrolidine]-2-yl]benzamide 3-bromo-5-phenyl-1,4-diazepane 2-(N-[2,5-difluoro-4-(1-oxo-3H-pyrrolo[3,4-c]pyridin-2-yl)phenyl]anilino)-N-methylideneethanimidamide 2-(4-chlorophenoxy)-N-[(1S,3R)-3-(5-methylimidazol-1-yl)cyclopentyl]acetamide 3-bromo-1,2,3,4-tetrahydroacridine 2-[1,3-benzodioxol-5-ylmethyl-[(Z)-4-hydroxybutylideneamino]amino]acetic acid 5-methyl-3-[(Z)-3-(2,3,4,5-tetrafluorophenyl)but-1-enyl]-N-[(2,4,6-trifluorophenyl)methyl]pyrazole-1-carboxamide N-(7,8-dihydronaphthalen-2-yl)-3,5-dimethylhexanamide 3-[(1R)-2-oxo-1H-naphthalen-1-yl]-N-pyridin-4-ylpropanamide N-[5-methyl-6-(2,3,4,9-tetrahydropyrido[3,4-b]indole-1-carbonyl)cycloocta-1,4,6-trien-1-yl]-4-(trifluoromethoxy)benzenesulfonamide 3-(5,8-dimethylimidazo[1,2-a]pyrazin-6-yl)piperidine-2,6-dione 1-azido-3,5-dichloro-2-nitrobenzene 5-chloro-2,6-difluorobenzenesulfinic acid (3S,4R)-3-hydroxy-1-[5-methyl-2-(pyridine-3-carbonylamino)benzoyl]piperidine-4-carboxylic acid 1-[4-[3-(cyclohexylcarbamoylamino)phenyl]benzoyl]-N-(2,6-diethoxypyrimidin-4-yl)pyrrolidine-2-carboxamide N-[2-(4-acetamidophenyl)ethyl]-3-[5-[1-(hydroxymethyl)cyclopropyl]-1,2,4-oxadiazol-3-yl]azetidine-1-carboxamide 2-chloro-1,3,6,7-tetranitroanthracene 2-[(1R)-3-ethylcyclohexen-1-yl]quinoline 1-[(4-methoxyphenyl)methyl]-3-[3-[5-methanimidoyl-6-[2-(methylamino)ethylamino]pyrimidin-4-yl]-1H-indol-6-yl]urea N-[(2R,3S)-1,4-dibenzyl-5-oxo-3-phenylmethoxypyrrolidin-2-yl]acetamide 4-[2,3-bis(dimethylamino)phenyl]-6-imino-1,3,5-triazinane-2,7-dione (Z)-N-methoxy-3,4-diphenylpentanamide 7-(3,4-dihydroquinoxalin-2-yl)-1H-indole N-[(2S)-1-[5-chloro-4-oxo-3-[2-(trifluoromethoxy)anilino]quinazolin-2-yl]propan-2-yl]-3,5-dimethoxybenzamide 6-[(1E,3Z)-1-(methylideneamino)hexa-1,3,5-trien-2-yl]-N-[4-(oxan-4-yloxy)phenyl]quinazolin-4-amine 2-cyclopropyl-6-oxo-N-[(4-phenyloxolan-3-yl)methyl]-1H-pyrimidine-4-carboxamide N-methyl-4-[(1R)-6-oxo-2,3-dihydro-1H-pyrazin-5-yl]benzamide 3-[3-[(E)-2-[3,5-difluoro-4-(trifluoromethyl)phenyl]ethenyl]cyclobutyl]oxypropanal 4-[2-azido-6-(trifluoromethyl)pyridin-3-yl]-1,3-thiazole 3-methoxy-5-[6-(trifluoromethyl)pyrazin-2-yl]pyridine-2-carboxamide 5-(2,6-difluorophenyl)-N-methyl-3-[2-[[1-(methylsulfamoylamino)cyclopropanecarbonyl]amino]pyridin-4-yl]-1H-pyrrole-2-carboxamide 1-(1-methylpyrrol-3-yl)-5,6-dihydroindole (5R)-2-[3,5-difluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)anilino]-8-ethyl-N,N-dimethyl-9-oxo-6,7-dihydropyrimido[5,4-h][1,5]benzoxazepine-5-carboxamide 2-[3,4,5-triethoxy-N-(sulfanylamino)anilino]acetic acid 4-cyclopropyl-N-[2-(dimethylamino)-2-phenylethyl]oxane-4-carboxamide 1-methyl-N-[2,3,5-trifluoro-4-[(2S)-6-[(Z)-prop-1-enyl]nona-5,8-diyn-2-yl]oxyphenyl]benzimidazole-5-sulfonamide 2-[6-chloro-7-(1-methylpiperidine-4-carbonyl)oxyquinazolin-4-yl]oxyacetic acid ethane;(Z,3E)-2-ethylidene-N-methylhept-3-enethioamide;7-(6-fluoropyridin-3-yl)oxy-8-nitro-1H-quinolin-4-one 1-azidooxy-4-bromo-2,3,5-trimethylbenzene 1-[(4R,5S)-2,2-dimethyl-1,3-dioxolan-4-yl]-N-(1H-imidazol-2-ylmethylideneamino)methanamine 7-(cyclopropanecarbonyl)-2,5,6,8-tetrahydro-1H-4,7-naphthyridine-3-carboxylic acid;ethane 2-[4-[2-amino-3,6-bis(trifluoromethyl)pyridin-1-ium-1-yl]pyrazole-1-carbonyl]cyclopentan-1-one N-[[3-chloro-4-(methoxymethyl)phenyl]methyl]-1,2-oxazole-5-carboxamide N-[5-(1,3-dioxan-2-yl)-1-(4-phenylbutoxymethyl)pyrimidin-1-ium-2-ylidene]hydroxylamine N-[(4S)-4-[(2-aminoacetyl)amino]pentyl]-6-[1,3-dimethyl-7-oxo-5-[4-(trifluoromethyl)phenyl]-6H-pyrazolo[4,3-d]pyrimidin-7-ium-2-yl]pyridine-3-carboxamide 5-methoxy-1,3-dimethyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide 1-[(2,5-dimethylphenyl)methylamino]-3-propan-2-ylthiourea 6-azido-3-(2,5-dimethylphenyl)sulfonylquinoline N-[1-(2-azidoethyl)-2,3-dihydroindol-6-yl]cyclopentanesulfonamide 6-[3-(diethylamino)propyl]-4H-furo[2,3-b]pyrrole-5-carboxylic acid 4-[5,7-dimethyl-6-(2,3,5-trifluorophenyl)pyrazolo[1,5-a]pyrimidin-3-yl]aniline 2-ethyl-5-[4-(methylamino)phenyl]pentanamide N-[2,2,3,3,5,5,6,7,8,8a-decadeuterio-4-(trifluoromethyl)cyclohexen-1-yl]-2-thiophen-3-ylsulfanylacetamide 1-methyl-2-(5-pyridin-4-ylpentanoyl)pyrrolidine-3-carboxylic acid 2-[6-methyl-1-(oxolan-3-yl)pyrazolo[4,3-b]pyridin-7-yl]phenol 5-fluoro-3,4,9-trimethyl-1H-pyrano[2,3-g]indole [4-(azidomethyl)piperidin-1-yl]-(5-phenoxypyridin-2-yl)methanone 3-(difluoromethoxy)-2-(4,6-diphenyl-1,3,5-triazin-2-yl)benzenethiol [(2-hydroxybenzoyl)amino]carbamodithioic acid (NE)-N-[[3-ethyl-6-(3-pyridin-2-yloxyphenyl)imino-4H-1,3,5-thiadiazin-2-ylidene]hydrazinylidene]hydroxylamine 1-[5,6-dimethyl-2-(4,5,6-trifluorocyclohexa-1,3-dien-1-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid 1-[6,8-dimethyl-2-(trifluoromethyl)imidazo[1,2-a]pyridine-3-carbonyl]-3-(hydroxymethyl)piperidine-3-carboxylic acid 4-(2,3-difluorophenyl)-5-[6-ethyl-5-[1-methoxy-2-(oxan-2-yloxy)propan-2-yl]pyridin-2-yl]-N'-hydroxypyridine-2-carboximidamide 5-cyclohexa-1,3-dien-1-yl-2-(4-phenylpyridin-2-yl)benzonitrile 2-(4,5-dichloro-2-methylphenyl)-3H-pyrido[3,4-d]pyrimidin-4-one 1-(2,3-dihydro-1H-inden-5-yl)-3-[[4-[2-(ethylamino)pyridin-3-yl]phenyl]methylsulfonyl]urea N-[1-amino-2-(4,5-dihydroxycyclohepta-1,3,6-trien-1-yl)ethylidene]furan-2-carboxamide 2-[1-(2,6-dichlorocyclohexa-2,4-dien-1-yl)-3-methoxyazetidin-3-yl]oxy-5-(trifluoromethyl)pyridine 1-[2-[(dimethylamino)methyl]phenoxy]-3-[4-[4-[2-(trifluoromethoxy)phenyl]piperazine-1-carbonyl]piperidin-1-yl]propan-2-one 4-azido-3-iodopyridine 2-[4-(cyclobutylmethoxy)-3-fluorophenyl]benzo[g][1,3]benzothiazole 4-[[2-[1-(2,3,3a,4,5,6-hexahydro-1H-phenalen-2-yl)ethoxy]acetyl]amino]-N'-hydroxybenzenecarboximidamide ethane;8-N-[(Z)-1H-indol-3-ylmethylideneamino]naphthalene-2,7-diamine 2-(1H-benzo[g]indol-3-yl)-N-[(E)-(5-nitrothiophen-2-yl)methylideneamino]acetamide N-[(3S,4R)-1-[6-fluoro-8-(methylaminomethyl)quinazolin-2-yl]-4-propan-2-ylpyrrolidin-3-yl]pyrazine-2-carboxamide 2-[N-methylsulfonyl-4-(pyridin-2-ylsulfamoyl)anilino]decanoic acid 4-azido-N-(2,3-difluorophenyl)pyridine-3-carboxamide 2-[[2,5-dimethyl-4-(4-nitrophenyl)pyrazol-3-yl]amino]ethanol 4-bromo-5-[(E)-[(3R,6S)-6-methylpiperidin-3-ylidene]oxymethyl]thiophene-2-carboxylate N-[1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)piperidin-4-yl]butanamide (2E,3Z)-1-methyl-2-(2-methylidenebut-3-enoxyimino)-N-[[2-oxo-5-phenyl-1-propan-2-ylpyrrolidin-3-yl]methyl]hexa-3,5-diene-1-sulfonamide 4-[3-(N-formylanilino)-2,5-dioxopyrrolidin-1-yl]benzamide N-[6-(2-fluorophenyl)pyridazin-3-yl]spiro[1,4-dihydroquinoxaline-3,4'-oxane]-2-imine N-[3-(2-aminoethynyl)phenyl]-4,6,7-trimethoxy-2-(4-methylsulfonylphenoxy)quinazoline-8-carboxamide 4-chloro-2,6-dimethylquinoline;methoxyethane 4-[2-amino-5-(2-cyclopropyl-6-oxo-1H-pyrimidin-4-yl)phenyl]-7,8-dihydroimidazo[1,5-a]quinazoline-3-carboxamide [(3R,4R)-4-hydroxy-1-(2-morpholin-4-ylacetyl)piperidin-3-yl]-(4-methoxy-3,5-dimethylphenyl)methanone 3-[[2-[1-(dimethylamino)propan-2-yl]-6-oxo-1H-pyrimidine-4-carbonyl]amino]benzoic acid (3S)-2,7-dioxooctanedioic acid;N-[(1R)-2-hydroxycyclohexyl]-6-phenylbenzo[b][1,4]benzoxazepine-3-carboxamide 4-[5-(4-phenylphenyl)thiophen-3-yl]phenol 2-(4-azidobutyl)naphthalene 3-[6-(5-chlorothiophen-2-yl)pyridin-3-yl]hexanoic acid 4-[(2R)-1-azidopropan-2-yl]-N-methoxybenzamide [(3S,4R)-1-benzyl-3-hydroxypiperidin-4-yl]azanium 4-[5-bromo-2,6-di(propan-2-yl)pyrimidin-4-yl]-3H-1,3-thiazol-2-one 1,3-bis(4-nitrophenyl)propan-2-one N-[4-[2-amino-6-(2,5-difluorophenyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl]formamide 3-bromo-2-[4-(difluoromethoxy)phenyl]-5H-pyrido[2,3-b]pyrazin-8-one (4-methylphenyl)-(2-morpholin-4-ylspiro[5,6-dihydrocyclopenta[d]pyrimidine-7,3'-piperidine]-1'-yl)methanone 4-[5-fluoro-2-(methylsulfamoyl)phenyl]piperazine-1-carboxylic acid 4-[[(4aR,5R)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]methyl]benzenesulfonamide 1-(3,4,5-trimethylphenyl)imidazo[4,5-c]pyridine N-[(2R)-3,3-dimethylbutan-2-yl]-5-[1-[[1-(difluoromethyl)cyclopropyl]amino]ethenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine N-methylsulfonyl-4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]benzamide 4-(3,5-difluorophenyl)-1-hydroxy-2H-phthalazine 1-[4-[2-(3,5-diethoxyphenyl)cyclopenten-1-yl]phenyl]ethanone 1-ethenylsulfonyl-2,4-dimethoxybenzene 3-(2,3-dichlorophenyl)sulfonylpiperidine 1-[3-(aminomethyl)azetidin-1-yl]-2,2,2-trifluoroethanone;2,2,2-trifluoroacetic acid 2-(cyclohexylamino)-6,7-dimethoxyquinoline-3-carboxylic acid 1-methoxycarbonyl-3,4-dihydroisoquinoline-2-carboxylic acid N-azido-5,6,7,8-tetrahydroquinazoline-2-carboxamide N-[2-[1-(3,5-dimethoxyphenyl)ethylideneamino]pyrimidin-4-yl]propanamide 5-(4-hydroxypiperidine-1-carbonyl)-2H-isoquinolin-1-one 3-(1H-pyrazol-5-yl)imidazo[1,2-a]pyridine-6-carboxylic acid ethane;1-[4-[7-(6-methylnaphthalen-2-yl)heptoxy]phenyl]sulfonylpiperidine 2-[6-azido-4-[3,5-bis(trifluoromethyl)phenyl]pyridin-2-yl]oxyethanol 1,2-diamino-4-[3-ethoxy-4-(trifluoromethyl)phenyl]-6-oxopyridine-3,5-dicarbonitrile 3-(1,3-benzothiazol-6-yl)-4-[2,5-dimethyl-1-(1H-pyrrol-2-yl)pyrrol-3-yl]pyrrole-2,5-dione 6-methyl-5-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole 2-[(2-chloroacetyl)-(6-sulfonaphthalen-1-yl)amino]octanoic acid (Z)-2,3-dichloroprop-1-en-1-amine;ethane;2-(methylamino)-1-[4-(4-methyl-6-morpholin-4-ylpyrimidin-2-yl)phenyl]guanidine N-methylmethanamine;3-[5-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)pyridin-2-yl]butanal 4-(1H-imidazo[4,5-b]pyridin-2-ylmethoxy)piperidine-1-carboxylate 2-(1,3-benzoxazol-6-yl)-4H-benzo[g][1,3]benzothiazol-7-amine 2-[1-(4,5,6,7-tetrahydro-3H-benzimidazole-5-carbonyl)piperidin-3-yl]-3H-quinazolin-4-one (E)-N'-[2,4-difluoro-5-[[4-[(1Z)-2-methylbuta-1,3-dienyl]pyrimidin-2-yl]amino]phenyl]prop-1-ene-1,3-diamine N-[(2,3,4,5,6-pentafluorophenyl)methyl]acetamide 7-(1H-benzimidazole-2-carbonyl)-4a-hydroxy-3,5,6,8-tetrahydro-1H-pyrido[3,4-d]pyrimidine-2,4-dione 4-(2-methoxyphenyl)-N,N-bis[(3R)-piperidin-3-yl]butanamide;hydrochloride 4-amino-2-[(1S)-1-[5-[3-(difluoromethyl)phenyl]pyridin-3-yl]ethoxy]pyrido[3,4-d]pyrimidine-8-carbonitrile 2-[(4-fluorophenyl)methylsulfanyl]-5-iodo-4-propan-2-yl-1H-pyrimidin-6-one (5Z)-5-[[3,4-bis(2-chloroethoxy)phenyl]methylidene]imidazolidine-2,4-dione 3-[2,3-bis(ethenyl)pyrrol-1-yl]propane-1-thiol 4-(2,4-dichlorophenyl)sulfonyloxypentanoic acid 2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]acetamide N-[(4R)-4-benzylpiperidin-3-ylidene]nitramide 3-methyl-N-(5-methylsulfanylpyridin-2-yl)pyrazolo[1,5-a]pyrimidine-5-carboxamide 2-bromo-N-(1,3-diethoxy-1,3-dioxopropan-2-yl)-N-(4-hydroxyphenyl)benzamide 1-(6,8-difluoro-4-hydroxy-3,4-dihydronaphthalen-2-yl)ethanone 2-[1-(3,4-dichlorophenyl)-5-oxopyrrolidin-2-yl]acetic acid (4-hydroxy-2,3,5-trimethylphenyl)-[4-(2-methoxyethyl)piperazin-1-yl]methanone 3-azido-6-chloroquinoline 3-(7,7a-dihydro-1,5-naphthyridin-4-yloxy)-6-methyl-4H-pyran-2-one 1-[4-[(2R)-3,5-dimethylcyclohexanecarbonyl]-6-phenyl-2,3-dihydroquinoxalin-1-yl]ethanone 3-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N'-[(1R,2S)-2-hydroxycyclohexyl]benzenecarboximidamide 2,6-dichloro-4-methylquinoline;ethane 1-benzyl-2,5-dimethoxy-3,4,6-trimethyl-9H-pyrido[3,2-h]quinazolin-1-ium (3S)-N'-[3-cyano-4-(trifluoromethylsulfanyl)phenyl]-3-(1,3-dioxoisoindol-2-yl)pyrrolidine-1-carboximidamide N-[(4,5-dichlorocyclohexa-2,4-dien-1-yl)methyl]-6-nitro-7H-purine-8-carboxamide 2-[1-(4-butanoylphenyl)-4-[2-(3,5-difluorophenyl)ethyl]piperazin-2-yl]-N-hydroxy-2-[4-(trifluoromethoxy)phenyl]acetamide 5-[2,3-dimethyl-4-(4-methylphenyl)cyclobutyl]pentanoic acid 1-N-[3-(4,6-dimethylpyridin-2-yl)phenyl]ethene-1,1-diamine 4-[[(2S,3R)-2-methyl-1,1-dioxothiolan-3-yl]amino]benzamide 3-azido-6,8-dimethoxyquinoline 2-[4-chlorobutyl(pyridin-3-yl)amino]acetonitrile 4-(N-ethenylsulfonyl-2,4-dinitroanilino)benzenesulfonic acid N-[[(3R)-2,5-dioxooxolan-3-yl]methyl]-4-phenylbenzamide N-[4,5-dichloro-2-(1H-indole-2-carbonyl)phenyl]-3-methylbutanamide N-[(Z)-1-[2-methyl-4-[2-oxo-3-(phenylcarbamoylamino)pyridin-1-yl]anilino]-3-piperidin-1-ylprop-1-enyl]hexanamide 2-[(3S,4R)-3-fluoro-1-[(5-methylpyridin-2-yl)methyl]piperidin-4-yl]-N'-pyridin-2-ylethanimidamide ethane;5-[2-(4-methoxyphenyl)quinolin-4-yl]pyrazolidin-3-one [2-amino-3,6-bis(trifluoromethyl)phenyl]boronic acid N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-methoxy-6-methyl-N-octyl-1,3,5-triazin-2-amine N-(cyclohexylmethyl)-2-oxospiro[1H-indole-3,3'-oxetane]-4-carboxamide 4-[(2,3-dioxo-1H-pyrrolo[1,2-c]imidazole-5-carbonyl)amino]benzoic acid 6-[5-[5-[2-(1-methylpiperidin-4-yl)ethoxy]pyridin-3-yl]-1H-pyrazol-4-yl]imidazo[1,2-a]pyrimidine 2-[N'-(2,6-dichlorophenyl)carbamimidoyl]benzenecarboximidamide;hydrochloride 1-[2-(4-methoxyphenyl)ethyl]pyrazolo[3,4-c]pyridine 6-amino-4-(3,4-dihydroxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 2-[4-chloro-3-(cyclopropylmethoxy)phenyl]-6-(oxan-4-ylmethylsulfonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine 2-benzyl-3,4-dinitrobutanenitrile 4-[2-(7-methylnaphthalen-1-yl)oxyethyl]morpholine 4-[1,5-dimethyl-3-(trifluoromethyl)pyrazol-4-yl]-6-N-methylquinazoline-2,6-diamine;dihydrochloride N-[3-[3-(4-aminocyclohexyl)oxyphenyl]sulfanylpropyl]-2-methylbenzenesulfinamide N-[6-amino-5-(methylideneamino)pyridin-2-yl]-2,6-difluorobenzamide (4E)-3-ethylsulfanyl-N-methyl-2,3-dihydro-1H-1,6-naphthyridine-4-carboxamide 1-(azidomethyl)-4,5-bis(3-fluorophenyl)-2-propoxybenzene 4-(6-methylpyridazin-3-yl)piperidine-1,5-dicarboxamide (2E,4Z)-5-amino-N-ethyl-2-[3-fluoro-6-methoxy-5-[4-(4-oxopentanoyl)piperazine-1-carbonyl]pyridin-2-yl]hepta-2,4-dienamide ethane;6-ethyl-1,2-dimethyl-7-(4-methylphenyl)naphthalene 1-[(2S,4R)-2-(fluoromethyl)-1-[[2-(1H-indazole-3-carbonylamino)acetyl]amino]piperidin-4-yl]indole-3-carboxamide N-(2,6-dichlorophenyl)-4H-pyrazolo[1,5-a]quinazoline-3-carboxamide 5-[(3,4-dimethylphenyl)iminomethyl]-6-hydroxy-2-sulfanylidene-1H-pyrimidin-4-one N-(2,3-dihydro-1H-inden-4-yl)-5-piperidin-4-ylthiophene-2-carboxamide;hydrochloride ethane;1-[2-(3-methoxyphenyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4-yl]pyrrolidin-3-ol (3-azidophenyl)-[3,4-bis[(1S)-2-hydroxycyclohexyl]-6H-cyclopenta[b]pyrrol-5-yl]methanone [6-chloro-2-[(6R)-1,4-oxazepane-6-carbonyl]indol-1-yl]carbamic acid N'-[(E)-3-chloro-2-methylprop-1-enyl]-2,6-difluorobenzenecarboximidamide N-[(Z)-[5-bromo-2-hydroxy-3-[(4-nitrophenyl)methyl]phenyl]methylideneamino]pyridine-3-carboxamide 4-amino-2,6-ditert-butylphenol N-[(3,5-dimethoxyphenyl)carbamothioyl]benzamide N'-hydroxy-3-(4-methylsulfonylphenoxy)pyrazine-2-carboximidamide (2-benzylcyclohexyl)-cyclopentylmethanone 2-(azidomethyl)-5-fluoropyridine-3-carboxamide 4-(2-iodopropan-2-yl)benzoate 4-(4-methoxyphenyl)-3,9-dithiabicyclo[6.1.0]nonan-2-one 1-(2,3-dihydro-1H-indene-5-carbonyl)piperidine-4-carboxylic acid 5-[3-chloro-4-(difluoromethoxy)phenyl]sulfonyl-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carboxylic acid 2-[N'-(3,5-dichlorophenyl)carbamimidoyl]sulfanyl-2-methylpropanoic acid 1-[4-(2,5-dioxopyrrol-1-yl)oxy-3,6-bis(dimethylaminosulfanyl)naphthalen-2-yl]pyrrole-2,5-disulfonic acid 1-[4-[6-(3,5-dimethylpyrazol-1-yl)pyrimidin-4-yl]oxypiperidin-1-yl]ethanone 3-methyl-1-(4-propan-2-ylphenyl)piperidine (2R)-N-[3-[[4-amino-5-[1-(5-methylpyridin-2-yl)propanoyl]oxy-6H-quinazolin-7-ylidene]methyl]phenyl]-2,5-difluoropyrrolidine-1-carboxamide 1-(8-azidonaphthalen-2-yl)-3,5-difluoropiperidine 5-methyl-3-[4-(trifluoromethoxy)phenyl]-N'-(2,4,6-trichlorophenyl)-1H-pyrazole-4-carbohydrazide (7S)-6-N-(4-fluorophenyl)-5,7-dimethyl-3-N-pyridin-2-yl-4,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide 3-[2-(2,4-dimethylphenyl)ethyl]-6-fluoro-7-propanoyloxynaphthalene-1,5-disulfonic acid N-[2-(5-ethyl-4-methyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]-2,3-dihydro-1-benzofuran-7-carboxamide 1,7-diphenylheptane-2,4,6-triamine 1-[4-[(2,5-difluorophenyl)methylamino]-8-oxa-6,11-diazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-12-yl]ethanone;dihydrochloride 4-N,6-N-di(cyclopropylmethyl)-8-(1H-indole-5-carbonyl)-3,7-dihydro-2H-[1,4]dioxino[2,3-f]isoindole-4,6-dicarboxamide;oxolane 3-amino-N-[4-(4-morpholin-2-ylanilino)phenyl]benzamide 1-[(E)-4,4-dimethylpent-2-en-3-yl]-2-ethenylnaphthalene;ethane 2-[(6R)-2-amino-5-oxo-3,6-dihydro-1H-[1,4]oxazino[4,3-a]quinolin-9-yl]acetic acid;hydrochloride 1-[2-(2-ethylhexoxy)phenyl]-4-prop-2-enylphthalazine 1-(4-chlorophenyl)-3-[2-(oxan-4-ylsulfamoyl)phenyl]urea [3-hydroxy-2-(2H-tetrazol-5-yl)phenyl]urea 2-[4,5-diamino-6-(2,6-difluoroanilino)pyrimidin-2-yl]oxybutan-1-ol ethane;1-[6-(3-methylphenyl)pyridin-2-yl]piperazine 2-[4-[(4-methylpiperazine-1-carbonyl)amino]naphthalen-1-yl]oxyacetic acid 3-methyl-6-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]imidazo[1,2-b]pyridazine [(1-tert-butylpyrazol-4-yl)amino]methanol 2-(azidomethyl)-6,7-dichloro-3H-quinazolin-4-one 7-fluoro-6-methoxy-4-[(3R)-1-(pyridine-2-carbonyl)piperidin-3-yl]oxyquinazolin-8-ol N-[(3S,4S)-1-cyclohexyl-3-methoxypiperidin-4-yl]quinoxaline-2-carboxamide;dihydrochloride (6-chloropyrazin-2-yl)-pyridin-3-ylmethanol 2-[4,6-dimethoxy-1-(thiophene-3-carbonyl)indol-3-yl]acetamide 5-[(3,4,5-trifluorophenyl)methoxy]quinazoline 5-benzyl-2,6-bis(furan-2-ylmethoxy)pyridine 3-(4,5-dichloropyrimidin-2-yl)oxycyclobutane-1-carboxylate 1-[4-bromo-2,6-di(propan-2-yl)phenyl]-3-[5-tert-butyl-2-(2,2,2-trifluoroethoxy)pyridin-3-yl]urea 2-(furan-3-yl)pyrazolo[1,5-a]pyrimidine 1-[2-(4-cyclopentylpiperazin-1-yl)ethoxy]isoquinoline 2-[3-(1,3-dioxoisoindol-2-yl)propanoylamino]benzoic acid 2-[4-(bromomethyl)phenyl]quinoline 5-tert-butyl-1-[2-(3,4-dichlorophenyl)ethyl]imidazole [4-(2,3-dimethylphenyl)piperazin-1-yl]-(5-methoxy-4-methylfuran-2-yl)methanone 2-[(Z)-3-ethylsulfanylprop-1-enyl]chromen-4-one (1R)-6,7-difluoro-2-methyl-N'-[5-[3-methyl-5-[(Z)-propylideneamino]cyclohepta-1,4,6-trien-1-yl]pyridin-2-yl]-3,4-dihydro-1H-isoquinoline-1-carboximidamide (E)-3-[4-amino-2-(trifluoromethyl)phenyl]prop-2-enal 1-azidosulfanyl-3-propoxybenzene 6,7-dimethoxy-2,3,4,9-tetrahydro-1H-carbazole;ethane 3-[2-amino-4,7-dimethyl-5-(propan-2-ylsulfanylmethyl)pyrrolo[2,3-d]pyrimidine-6-carbonyl]benzoic acid 7-methoxycarbonylspiro[2,3,4,5-tetrahydro-1H-naphthalene-6,2'-furan]-2'-carboxylic acid 2-[(1S)-1-azidoethyl]-4,5-dihydrothieno[3,2-d][1]benzoxepine 5-[(3E)-3-hydroxyiminoindol-2-yl]-3,4-dihydropyridine-3-carbonitrile N-[(4Z,6E)-5-[(Z)-but-2-enoxy]octa-2,4,6-trienyl]-1-cyclopropyl-7H-pyrazolo[3,4-b]pyridine-4-carboxamide 1-[4-(2-chlorophenyl)sulfonylpiperazin-1-yl]-6,7-dimethoxy-N-propan-2-yl-3,4-dihydro-1H-isoquinoline-2-carboxamide [5-(2,4-dimethylphenoxy)-3-(hydroxymethyl)oxolan-2-yl]methanol (2Z)-3,7-dimethyl-6-[4-[(3E,5E)-5-(1,10,16,16-tetrazatetracyclo[16.7.0.02,7.08,14]henicosa-2,4,6,8,10,12,14,18,20-nonaen-17-yloxy)hepta-1,3,5-trien-3-yl]phenyl]hepta-2,6-dienenitrile 6-[4-(6,7-difluoroquinolin-2-yl)oxyphenyl]hexanamide (2S)-N-[4-[2,5-difluoro-3-methoxy-6-(2-oxa-8-azatricyclo[7.3.1.05,13]trideca-1(13),5,7,9,11-pentaen-10-ylmethoxymethyl)phenyl]pyridin-2-yl]pyrrolidine-2-carboxamide [6-fluoro-3-(2-propan-2-ylpyrimidine-5-carbonyl)indolizin-1-yl]urea 4-methyl-2-[3-(trifluoromethyl)phenyl]cyclohexa-1,5-dien-1-amine N-(4,5-diphenyl-1H-imidazol-2-yl)acetamide (3R,4S)-4-azido-1-[2-methyl-6-(5-methyltetrazol-2-yl)pyridine-3-carbonyl]pyrrolidin-3-ol 4-[[1-(5-chloro-6-methyl-2,3-dihydro-1H-inden-1-yl)pyrrolidin-3-yl]amino]pyridine-3-carbonitrile;hydrochloride N'-benzyl-2,3-difluorobenzenecarboximidamide 2-amino-4,6-bis(sulfanyl)naphthalene-1,7-disulfonic acid 2-(dimethylamino)-1,5-diphenylpentan-3-one 2-azidooxy-3-bromothiophene 3-[3-(4-hydroxyphenyl)butanoylamino]propylphosphonic acid 1-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-2-methyl-1,8-naphthyridine-2,3-diol 6-[2,2-diethoxyethyl(methylsulfonyl)amino]pyridine-3-sulfonamide (2R)-1-[5-[3-azido-4-(trifluoromethyl)phenyl]pyrazin-2-yl]piperidine-2-carboxylic acid (E)-3-[1H-benzimidazol-2-yl(butanoyloxymethyl)amino]prop-2-enoic acid 2-fluoro-4-(trifluoromethylsulfanyloxy)phenol 2-(azidomethyl)-N,4,5,6-tetraphenylpyrimidin-4-amine 2-(2,3-dimethylphenyl)-4-[ethoxycarbonyl(methyl)amino]thiophene-3-carboxylic acid 1-azido-2,3,4,5,6-pentafluorobenzene 5-chloro-4-[methyl(2,2,6,6-tetramethylpiperidin-4-ylidene)amino]oxynaphthalene-1-carboxamide 1-(3-azido-5,6-dimethylpyrazin-2-yl)-N-[(4,6-dichloropyridin-3-yl)methoxy]propan-2-imine 5-[[4-(trifluoromethyl)phenoxy]methyl]pyridine-3,6-diamine [3-(tert-butylamino)-2,4,6-trimethoxyphenyl]thiourea 3-(2,6-dichlorophenyl)-5-[4-[(1-pyridin-2-ylcyclopropanecarbonyl)amino]benzoyl]oxy-1H-pyrazole-4-carboxylic acid N-(4,7-dimethoxy-2-phenyl-1H-indol-3-yl)formamide;4-heptylcyclohexan-1-amine 2-azidosulfanyl-1-nitronaphthalene 2-(4-chlorophenyl)-7-methyl-N,3,8a-triphenylpyrazolo[1,5-a][1,3]benzodiazepine-9-carboxamide 2-[3,5-dimethyl-1-(4-oxo-7,8-dihydro-6H-pyrido[2,3-d]pyrimidin-3-yl)pyrazol-4-yl]-N-(4-phenoxyphenyl)acetamide 5-(1H-pyrazol-4-yl)-3-[(2E,4Z,6E)-nona-2,4,6-trien-2-yl]-2H-indazole (E)-3-[4-[2-[5-methyl-6-(1-phenylethoxy)pyridin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]phenyl]prop-2-enoic acid (7S)-N-(2,5-dimethoxyphenyl)-3-methyl-4-oxo-6,7,8,9-tetrahydro-5H-pyrazolo[1,5-a]quinazoline-7-carboxamide 1-(4-azidobutyl)anthracene N-(2,4-dimethylphenyl)formamide;6-[1,3-dioxo-8-(5,5,5-trifluoropentoxy)isoindol-2-yl]-5-ethoxyhexanal (Z)-3,3,5,5-tetrafluoro-6-quinolin-8-yloxyhex-4-enoic acid 1-chloro-2,3-difluorobenzene;2-[3-(dimethylamino)propoxy]-5-ethylaniline N-[(E)-3,3-dimethylbut-1-enoxy]-6,7-bis[(2-methylpropan-2-yl)oxycarbonylamino]phenazine-5-carboxamide;ethane N-[5-[4-fluoro-3-(7-pyridin-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]cyclopentanecarboxamide 3-(6,8-dimethylimidazo[1,2-a]pyrazin-2-yl)benzoic acid 2-[5-carbamoyl-9-[(3,4-difluorophenyl)methyl]-2-ethylcarbazol-4-yl]peroxyacetic acid 5-[3-(4-cyclopropylimidazol-1-yl)-2,6-difluorophenyl]-7-methylpyrrolo[2,3-d]pyrimidin-4-amine 2-(1,3-benzodioxol-5-yl)-4,6-bis[[2-chloro-6-fluoro-3-(trifluoromethoxy)phenyl]methylideneamino]phenol 5-[4-amino-1-[(3S,5R)-1-benzyl-5-methylpyrrolidin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenol (3S)-4-[1-hydroxy-1-phenyl-2-(1,3-thiazol-2-ylamino)ethyl]sulfonyl-2,2,6,7-tetramethylheptanoic acid 1-[5-tert-butyl-3-(cyclopropanecarboximidoyl)-2-methoxyphenyl]-3-[4-(6-morpholin-4-ylpyridine-3-carbonyl)naphthalen-1-yl]urea 1-(3-amino-4-phenylpyrazol-1-yl)-2-phenoxyethanone N-(5-acetylthiophen-2-yl)-2,2,3,3a,4,5,6,7,8,8a-decahydrobenzo[b]thiophene-1-carboxamide 2,3-diphenyl-2-pyridin-1-ium-1-ylpropanoic acid;bromide [(Z)-4-anilinobut-2-enyl]sulfanium 2-[1-(6,7-dimethoxyquinazolin-4-yl)piperidin-3-yl]propanamide;hydrochloride 7-(3,4-dihydronaphthalene-2-carbonyl)-1H-quinoxalin-2-one 1-azido-3,5-dichlorobenzene 4-[1,2,3,5]tetradeuterio-6-[9-(dimethylamino)-10H-acridin-10-id-10-yl]benzene-1,3-disulfonic acid 7-(3-methoxyphenyl)heptan-2-one 6-(3-butoxyphenyl)-4-oxo-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 4-cyclopropyl-3,5,6-trimethoxycyclohexa-2,4-diene-1-sulfonic acid 3-(3,4-dimethoxyphenyl)-N'-hydroxy-2-(6-methyl-1H-benzimidazol-2-yl)benzenecarboximidamide N-[4,5-bis(ethenyl)-2-(2-methoxyphenyl)imidazol-1-yl]acetamide 5-chloro-N'-hydroxy-3-methylsulfanylpyridine-2-carboximidamide 2-(1,4,5,6-tetrahydropyrimidin-2-yl)benzonitrile 3-(3,4-dihydropyridin-6-yl)-1H-indole (2R)-2-[N-[2-(5,6-dimethylbenzimidazol-1-yl)ethyl]-4-(trifluoromethoxy)anilino]propanamide 1-[4-(azidomethyl)phenyl]ethanesulfonic acid 3-[(1R)-2,6-dichloro-4-fluorocyclohexa-2,4-dien-1-yl]-1,2,5,6-tetrahydroindole 1-[3-(azetidin-1-ylsulfonyl)phenyl]-4,5-dimethoxyindole 4-[2-azidooxy-5-(trifluoromethyl)pyrimidin-4-yl]morpholine 1-[4-(N,2-dimethylanilino)-3,5-bis(trifluoromethyl)phenyl]ethanone 2-(3,5-dichloro-N-octylanilino)propanoic acid N-benzyl-4-(2,6-dimethoxyphenyl)-5-(furan-2-yl)-1,2,4-triazol-3-amine;ethane 6-[(2R,3S)-2-ethyl-1-methylpiperidine-3-carbonyl]-N,N-dimethyl-5,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide 4-N-[2,6-dichloro-3-(4-chlorobenzoyl)phenyl]-5H-pyrrolo[3,2-d]pyrimidine-4,7-diamine (2R)-3,3-dimethyl-N'-[3-[(6S)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-6-carbonyl]phenyl]pentanehydrazide 1-(2,4-diethylphenyl)-N-[3-(methylideneamino)prop-1-en-2-yl]ethanimine N-[2,6-dimethyl-4-(5-methylcyclohexen-1-yl)phenyl]formamide;ethane 2-methoxy-4-[(Z)-[[4,6,7-trihydroxy-1-oxo-3-phenylisochromene-5-carbonyl]hydrazinylidene]methyl]benzoic acid 4-azidooxy-7-chlorochromen-2-one 4-[azidooxy(phenyl)methyl]benzoic acid 2-(3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl)pyridine-3-carbonitrile 7-[(2,4-dimethoxyphenyl)methyl]-9H-carbazole-3-carboxamide N-cyclopropyl-5-hydroxy-3-methyl-2,4-dioxopyrimidine-1-carboxamide 4-[(3S)-1,2,3,5,6,7,8-heptahydropyrrolizine-3a-carbonyl]-3,3a,10,10a-tetrahydro-2H-cyclopenta[b][1,4]benzoxazepine-7-carbonitrile N'-hydroxy-1-(4-hydroxy-3,5-dimethoxyphenyl)-5-(trifluoromethylsulfanylamino)pyrazole-4-carboximidamide 3-[(4-methylphenyl)methoxy]-2-methylsulfanyl-5H-pyrido[1,2-b]pyridazine 3,5-dichloro-2-(2H-pyridin-1-yl)aniline N-[2-(3,4-dimethylpiperidin-1-yl)ethyl]-N-propan-2-ylpyridine-2-carboxamide 1-[(Z)-1-cyclohexa-2,4-dien-1-ylideneethyl]-7-fluoronaphthalene;ethane 7-methylsulfanyl-2-[(3R)-3-[4-(trifluoromethoxy)phenoxy]piperidin-1-yl]quinoline 6-amino-N-[3-[(2,4-dimethylphenoxy)methyl]phenyl]-9-ethyl-8-oxo-5H-pyrido[2,3-b]azepine-7-carboxamide N-(4,5-dihydroimidazol-1-yl)-1H-indazole-6-carboxamide (3Z)-1-amino-4,7-dimethyl-5-sulfanylidene-6H-hepta-3,8-dien-2-one;1-[(E)-2-(3-hydroxyphenyl)ethenyl]-N-methylcyclohexane-1-carboxamide 4-amino-2-(3-bromophenyl)-5-methyl-1H-pyrimidin-6-one 1-(4,6-dimethylpyridine-3-carbonyl)-N'-[2-[5-(4-hydroxyphenyl)-4-methylimidazol-1-yl]ethyl]piperidine-4-carboximidamide (2R)-3,4-dimethoxy-1-[(6-oxo-1H-pyrimidine-4-carbonyl)amino]propane-2-sulfonic acid 2-(1-bromobutyl)chromen-4-one 1-[[2-(1H-indol-3-yl)ethylamino]methylsulfanyl]propane-2,3-diol;2,2,2-trifluoroacetic acid 6-[3-(4,7-dimethylcyclohepta-1,5-dien-1-yl)azetidin-1-yl]-N-(3-pyridin-3-ylpropyl)pyridazine-3-carboxamide N-(2,5-dimethylphenyl)-2,4-dihydroxybenzamide (4S)-1,2-dimethyl-3,5-bis[2-(4-methylphenyl)ethynyl]imidazolidine 2-[(3R,5S)-1-benzyl-2-oxopiperidin-3-yl]-N-[[4-(trifluoromethoxy)phenyl]methyl]acetamide 4-(3-fluoropyrrolidine-1-carbonyl)-2-phenylmethoxycyclohexa-1,5-diene-1-carboxamide 4-[3-[2-(aminomethyl)phenyl]piperazine-1-carbonyl]benzamide;2,2,2-trifluoroacetic acid 1-[2-(3-methylphenyl)ethynyl]-4-(1H-pyrrolo[2,3-b]pyridin-6-ium-5-yloxy)pyrazolo[3,4-d]pyrimidine 1-ethyl-3-[2-(5-hydroxypentan-2-ylideneamino)propanoyl]benzotriazol-2-one 3-(7-chloro-2,3-dihydro-1H-indol-6-yl)propanoic acid 4-azidooxy-2,3-dibutylphenol 5-[[6-amino-3-(2-fluorophenyl)pyridin-2-yl]methoxy]pyridine-2,4-dicarboxylic acid (2-methylpyrazol-3-yl)-[4-[1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidine-4-carbonyl]piperazin-1-yl]methanone 2-N-(4,5-dihydrothieno[3,2-b]indol-1-yl)benzene-1,2-disulfonamide N-[5-[(4R)-1,3-dimethylpiperidin-4-yl]pyridin-2-yl]-5-fluoro-6-[4-hydroxy-3,3-bis(trifluoromethyl)butoxy]-7-methylimidazo[1,2-a]pyrimidine-2-carboxamide 2-[8-(1-benzothiophen-3-yl)-5,6-dihydropyrazolo[5,1-c][1,2,4]triazin-2-ium-2-yl]ethanol 6-[2,4-dichloro-5-(2-oxobutyl)phenyl]-7-ethoxy-3H-quinazolin-4-one (5S)-2-[(4-chlorophenyl)methylsulfanyl]-N-(3,5-dichlorophenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-[2-(5-tert-butyl-1,3,4-oxadiazol-2-yl)ethoxy]-N-(1H-pyrazol-4-ylsulfonylmethyl)cyclohexane-1-carboxamide (2S)-N-[1-cyclohexyl-6-oxo-4-[2-oxoethoxy(propanoyl)amino]pyrimidin-5-yl]pyrrolidine-2-carboxamide 5-azido-3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-1H-pyrazole 2-(3,5-dimethylphenyl)-N-[4-hydroxy-1-(methoxymethylamino)-1,1-dioxothian-3-ylidene]acetamide 3-[(2-phenylacetyl)amino]-N-(thiophen-2-ylmethyl)bicyclo[1.1.0]butane-1-carboxamide 5-(4-hydroxy-6,7-dihydronaphthalene-2-carbonyl)-N-[1-[methyl(3-phenylpropanoyl)amino]pentan-2-yl]-1H-pyrrole-3-carboxamide N-(4,6-dimethyl-2H-pyrazolo[3,4-c]pyrazol-3-yl)-2,6-difluorobenzamide N-(6,7-dihydroquinolin-5-ylmethyl)-2,3-difluoroaniline (6E)-4-amino-8-[2-fluoro-6-(trifluoromethyl)phenyl]-2,3-dihydrochromen-2-ol 4-[3-(azidomethyl)-2,6-dichlorophenyl]morpholine ethane;1-[4-(4-methylphenyl)piperazin-1-yl]-3-(1H-pyrrol-2-yl)propan-1-one 2-(3,5-difluorophenyl)-N-[1-[(4S)-6-oxooxepane-4-carbonyl]piperidin-4-yl]acetamide N-(6-chloropyridin-3-yl)-1,2,4-triazin-5-amine 2-methyl-6-[4-[2-(1H-pyrazol-5-yl)ethynyl]piperidine-1-carbonyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one [2-[3,5-difluoro-4-(trifluoromethyl)phenyl]cyclopropyl]carbamic acid 2-(5,6-dimethylpyridin-3-yl)-1H-indole N-butyl-4-(3,5-dimethoxyphenyl)-1H-imidazole-5-carboxamide 4-(benzenesulfonamido)-2,6-dichlorobenzoic acid 4-(2,1,3-benzothiadiazol-5-yloxy)piperidine 2-(4-ethylsulfanylphenyl)propane-1,1,3,3-tetracarbonitrile 3-[4-(3,5-dimethylphenyl)piperazine-1-carbonyl]-2-hydroxybenzonitrile 6-(3,5-difluoropyridin-4-yl)-7-methoxy-N-[2-methanimidoyl-5-(1-piperidin-1-ylethylsulfanyl)phenyl]quinazolin-2-amine 2-(5-bromothiophen-3-yl)-2,4-dimethoxycyclobutan-1-one N-[4,5,6,7-tetramethyl-2-(3-phenylmethoxypropyl)-1H-indol-3-yl]thiophene-2-sulfonamide 4-(2,3-dihydro-1H-indazole-5-carbonylamino)-N-[2-hydroxy-1-phenyl-2-(propan-2-ylamino)ethyl]pyridine-2-carboxamide N-(2-methylpropanoyl)-4-nitro-N-(oxolan-2-ylmethyl)benzamide (2R)-3,3,3-trifluoro-2-[[(1S)-2,2,5,8-tetramethyl-4H-[1,3]dioxino[4,5-f]isoindole-9-carbonyl]amino]propanoic acid 1-(azidomethyl)-3,4-dihydroquinolin-2-one 6-chloro-3-phenyl-4H-1,2,3-benzotriazin-8-amine (3R)-3-[(2S)-2-aminopentanoyl]-N-methoxy-N',2-dimethyl-5-(4-methylanilino)-6-[methyl(sulfamoyl)amino]-1,2-dihydroindole-3-carboximidamide [2,4-dichloro-3-(4-fluorophenyl)sulfanyl-5-(trifluoromethylsulfonyloxy)phenyl]azanium 3-methyl-1-(2-methylphenyl)pyrrolo[3,4-b]pyridine N-[1-(3-chlorophenyl)-2-ethyl-5-methoxybenzimidazol-4-yl]sulfanyl-1,3-thiazol-2-amine (E)-1-[4-(ethoxymethyl)-3,5-difluorophenyl]pent-1-en-3-one 4-[3-(2,6-difluorophenyl)phenyl]pyridine 4-chloro-5-phenyl-2,6-disulfobenzene-1,3-dicarboxylic acid [4-(azidooxymethyl)phenyl]-piperidin-1-ylmethanone [(3aR,7aS)-2-pyrimidin-2-yl-1,3,4,6,7,7a-hexahydropyrano[3,4-c]pyrrol-3a-yl]methanol;2,2,2-trifluoroacetic acid 5-(9H-fluoren-1-yl)-3,4-dimethoxy-2-[1-(pyridine-3-carbonyloxy)ethyl]benzoic acid N-[4-(carbamoylsulfamoyl)phenyl]-2,4,6-trimethyl-N-octylbenzenesulfonamide 1-[5-(3,5-difluoro-4-hydroxyphenyl)sulfanyl-2-(ethoxymethylamino)phenyl]ethanone N-(3,4-dimethoxyphenyl)-1-[5-methyl-2-oxo-7-(trifluoromethyl)-1H-quinolin-4-yl]piperidine-4-carboxamide (3R)-1,3-bis[2-(difluoromethoxy)phenyl]-4-[4-(trifluoromethyl)phenyl]butan-2-one 6-[[2-(dimethylamino)ethyl-methylamino]methyl]pyridine-3-carboxylic acid 3-methyl-6,9b-dihydro-7aH-naphtho[2,1-b]oxirene 2-[4-(2,3-dihydro-1H-inden-5-yl)phenyl]-1H-imidazole N-(5,6-dihydroquinolin-8-yl)-3,4,7,8-tetrahydro-2H-cyclopenta[b]indole-1-carboxamide 4-N-[(1S)-2-azido-1-(3,5-dimethylphenyl)ethyl]pyridine-3,4-diamine 4-[(5E)-2,3,6-trimethylocta-1,5,7-trien-4-yl]aniline (3Z)-1-butyl-4-methoxy-3-[[4-oxo-2-(trifluoromethyl)chromen-8-yl]methylidene]pyridine-2,6-dione 2-fluoro-6-[3-(trifluoromethyl)phenyl]aniline 3-(1-methylsulfanylcyclopropyl)oxy-5-[4-(trifluoromethoxy)phenoxy]benzonitrile 3-[1-[(2R)-5,8-dichloro-4-oxo-2-[4-(trifluoromethyl)phenyl]-6H-quinazolin-7-ylidene]ethylamino]propanoic acid 4-[5-(trifluoromethyl)pyridin-3-yl]aniline 1-[3,5-bis(4-methoxyphenyl)sulfonylphenoxy]-3-cyclohexylbenzene 2-[6-(ethylamino)pyridine-3-carbonyl]propanediamide 4-[[3,5-dioxo-2-(3-phenylpropyl)pyrazolidine-1-carbonyl]amino]benzoic acid 5-[(Z)-1-amino-3-iminoprop-1-en-2-yl]-N'-(3,4-dimethoxyphenyl)-6-ethoxypyridine-2-carboximidamide 5-amino-2-[3-[(4S)-2-(1H-imidazol-5-ylmethyl)-8-methoxy-2,3,4,6-tetrahydroquinolin-4-id-4-yl]propanoyl]isoindole-1,3-dione 6-methoxy-N,N-dimethyl-2-phenylquinazoline-4-carboxamide 2-(4-azidophenyl)-1,3-oxazolidine N-(1,3-benzodioxol-5-ylmethoxy)benzenecarboximidate 4-[2,6-bis(ethenyl)-3-methylidenecyclohexa-1,5-dien-1-yl]sulfanylbenzenethiol N-[1-(2,4-dichlorophenyl)ethyl]-7-methoxy-2,3-dihydrobenzotriazole-5-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxy-4-oxo-4a,8a-dihydrochromene-3-carboxamide (2-aminopyrimidin-4-yl)-[(1S,6R)-3-(pyridine-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-9-yl]methanone;hydrochloride [(3S,4R)-1-[6-(2-aminopyrimidin-5-yl)pyridin-3-yl]-3-fluoropiperidin-4-yl]methylcarbamic acid;hydrochloride ethane;2-[3-(hydroxymethyl)phenoxy]ethanol (5E)-2-imino-5-[(4-iodophenyl)methylidene]-1,3-thiazolidin-4-one N-[[3-(4,5-dimethyl-1H-imidazol-2-yl)phenyl]methyl]-N,4-diethyl-6-oxo-1H-pyridine-2-carboxamide 3-bromo-2-[(E)-3-hydroxy-5-phenylpent-1-enyl]phenol 4-(3,5-difluorophenoxy)-2-methylbutane-1,3-diol 3-methyl-1-phenyl-1,2-dihydroindene (2S)-1,2-diethoxy-3-(4-fluorophenyl)propan-2-ol 1-[2,5-bis(4-methylphenyl)furan-3-yl]ethanone 2-[(4-chloro-3,5-dimethylpyrazol-1-yl)methyl]-N-[[6-(cyclopropylmethoxy)pyridin-3-yl]methyl]pyrrolidine-1-carboxamide (2Z)-2-[5-cyano-4-ethyl-3,8-difluoro-7-[(2S)-pyrrolidine-2-carbonyl]oxycyclohepta-1,6-dien-1-ylidene]-N-methyl-2-phenylacetamide 3-[(3S)-1-(2,6-difluorophenyl)piperidin-3-yl]oxy-5-[4-methanimidoyl-5-[1-[[4-(trifluoromethyl)pyridine-2-carbonyl]amino]ethyl]-1H-pyrazol-3-yl]thiophene-2-carboxylic acid 4-chloro-5-(4,5-dihydro-1H-imidazol-2-yl)thiophene-3-carboxamide;ethane 1-[(3R)-2-methoxy-6,8,13,15,16-pentazatetracyclo[9.7.0.02,7.012,17]octadeca-1(18),10,14,17-tetraen-12-yl]propan-1-one 4-[(E)-2-[3-ethyl-5-methoxy-1-[3-methoxy-4-(4-oxo-1,3-diazaspiro[4.4]nonan-3-yl)phenyl]sulfinylindol-6-yl]ethenyl]benzonitrile 2-[1-(4-methylpiperidine-1-carbonyl)cyclohexyl]-3H-thieno[3,2-d]pyrimidin-4-one N-benzyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-2-amine;dihydrochloride 3-[(1R)-4,6-dichloro-2,3-dihydro-1H-inden-1-yl]-5-ethylsulfonylpyridine 2-(N-benzylsulfonyl-4-phenylanilino)acetamide 2-azidooxy-7H-1,7-phenanthroline 2-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1]benzazepin-11-yl)-N'-methylidene-1,3-thiazole-4-carboximidamide 2-[4-bromo-5,6-dimethoxy-8-[(3R)-1-(2-pyridin-4-ylacetyl)piperidin-3-yl]oxy-1H-isoquinolin-2-ium-2-yl]-N'-methanimidoyl-3,4-bis(sulfanylidene)cyclobut-2-en-1-one N-(2-amino-2-oxoethyl)-4-[[4-cyclopropylidene-5-methyl-3-(oxan-4-ylamino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanylmethyl]benzamide 3,4,5-trimethoxy-N-(2,6,6-trifluorocyclohexa-1,3-dien-1-yl)benzamide 5-[3,4-difluoro-5-(2-pyrrolidin-1-ylethoxy)phenyl]-N-[6-methanimidoyl-5-(prop-2-enylamino)pyridin-3-yl]-6-methoxypyridine-3-carboxamide 7-tert-butyl-3-(methoxymethoxy)-1,2-dihydropyrido[2,3-b]pyrazine 3-[3,4-dihydroxy-5-(6-methylcyclohexa-1,3-dien-1-yl)phenyl]-N-[4-(trifluoromethylsulfanyl)phenyl]-1H-pyrazole-5-carboxamide 3-(2,6-dichlorophenyl)-7-[4-[[4-[methyl-(5-methyl-1H-pyrrole-2-carbonyl)amino]piperidin-1-yl]methyl]anilino]-2H-pyrimido[5,4-e]thiazine-5-carboxylic acid 1-methyl-3-[(4-nitrosophenyl)carbamoylamino]thiourea N-[(2R,3S)-2-methyl-1,5-dioxohexan-3-yl]pyridine-4-carboxamide (2Z)-3,5,7-trimethyl-N-[1-(2H-tetrazol-5-yl)ethyl]-4-(2,4,5-trifluorophenyl)octa-2,6-dienamide N-ethylsulfonyl-2,4,6-trimethylbenzenesulfonamide (2E)-5,6-dibromo-2-[1-methyl-4,5-dioxo-3-propanoyl-3H-pyrido[2,3-e][1,2,4]thiadiazin-7-ylidene]indole-3-carboxylic acid 4-azidooxy-3,5-di(propan-2-yl)aniline [3-(2,5-difluorophenyl)-3-azabicyclo[3.1.0]hexan-6-yl]methanol 4-(dimethylamino)-3-fluorophenol;4-[(3E,5Z)-5-fluorohepta-1,3,5-trien-4-yl]oxybenzaldehyde 2-methyl-4-[4-[(3S)-3-methyl-1,1-dioxothiazinan-2-yl]piperidin-1-yl]benzonitrile 4-[2-(5,6-dimethylcyclohexa-1,3-dien-1-yl)phenyl]morpholine 2-[1-(cyclopropanecarbonyl)piperidine-4-carbonyl]pyridine-3-carboxamide 1-[5-[3,5-dichloro-4-(2-methoxyethylsulfonyl)phenyl]pyridin-2-yl]-N-iodopropan-2-amine 5-(5-ethylfuran-2-yl)-2-[4-(pyridine-3-carbonyloxymethyl)phenyl]benzoic acid 2-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)phenol N-[1-(2,5-dimethoxyphenyl)ethyl]-3H-pyrrole-4-carboxamide 1-(3-aminopropyl)-6,7,8-trimethoxyquinoline-2,4-dione 1-(3,5-dimethylphenyl)sulfanyl-2,4-difluorobenzene;1-[3-ethoxypropyl(methyl)amino]propan-2-one 5-[(2S,4R)-4-azido-1-benzylpyrrolidin-2-yl]pentanoic acid N-[2-(3,4-dimethoxyphenyl)ethyl]-5-iodo-1-methylpyrazole-3-carboxamide 1-[3-fluoro-4-[(E)-2-[(Z)-1H-indol-3-ylmethylideneamino]oxyethyliminomethyl]phenyl]-5,6-dihydro-4H-pyrimidin-2-amine 4-[[2,3-bis(trifluoromethyl)phenyl]methoxymethylidene]-1-(7H-purin-6-yl)pyrrolidine-2,5-dione 3-methylsulfanyl-2,4-dihydropyrrolo[3,2-c]pyrazole-6-carboxylic acid 1-[(5-methyl-4,6-dihydropyrrolo[3,4-d]imidazol-2-yl)sulfanyl]propan-2-ol 5-[1,6-difluoro-4-(hydroxymethyl)cyclohexa-2,4-dien-1-yl]oxy-N'-hydroxypyridine-2-carboximidamide (E)-N,3-dimethylbut-2-enamide;ethane;5-(4-ethoxyphenyl)-3H-1,3,4-oxadiazol-2-one N-[5-(3,4-dichlorophenyl)sulfanyltriazolo[1,5-a]pyridin-7-yl]-2-methoxyacetamide (2S)-5,7-dimethoxy-N-[4-[1-(2-pyridin-2-ylethylamino)ethenyl]phenyl]-2H-chromene-3-carboxamide 5-chloro-2,4,6-triphenylpyrimidine 1-[(5S,8aR)-7-[3-fluoro-4-(trifluoromethyl)phenyl]-5-(2-hydroxyethoxy)-3,6-dioxo-5,8,8a-tetrahydro-1H-imidazo[1,5-a]pyrazine-2-carbonyl]-N-(2-thiophen-2-ylethyl)piperidine-3-carboxamide N-[4,5-difluoro-2-(propanoylamino)phenyl]-6-methylpyridine-3-carboxamide N-[4-(hydroxycarbamoyl)-5,6,7,8-tetrahydronaphthalen-1-yl]thiophene-2-carboxamide 3-amino-N'-methyl-6-(2-pyridin-4-ylethynyl)pyridazine-4-carboximidamide N-[4-(2,3-difluorophenyl)butanoyl]-1,5,6,7-tetrahydropyrazolo[4,3-c]pyridine-4-carboxamide 2-(4-anilino-N-(1,3-diethoxy-1,3-dioxopropan-2-yl)anilino)acetic acid 3-cyclopropyloxy-N-(4,6-dimethylpyrimidin-2-yl)benzenesulfonamide 2-[4-(5-chloro-1H-indol-3-yl)piperidin-1-yl]-N-(oxan-3-ylmethyl)acetamide 2-[5-chloro-4-[(2R,4S)-4-methoxyoxolan-2-yl]pyridin-3-yl]-4,6-diphenylpyrimidine (3R,4S)-1-[2-[4-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]phenyl]cyclopropyl]sulfonyl-N-hydroxy-4-methoxypyrrolidine-3-carboxamide [4-(aminomethyl)-2,3-dichlorophenyl]-[4-[(1E,3Z,5E)-3-ethenyl-6-methylideneocta-1,3,5-trienyl]piperazin-1-yl]methanone [(2R,5S)-5-(3-cyclohexyloxyphenyl)pyrrolidin-2-yl]methanamine 2,3-dimethyl-7-propan-2-ylbenzimidazole-5-carbonitrile 2,3-bis(2-methylpropyl)-7-phenylquinoxaline (2S,3R)-N-[[6-(4-chlorophenyl)pyridin-2-yl]methoxy]-2-ethyloxolane-3-carboxamide N-[4-[(4,5-dimethyl-1H-pyrazol-3-yl)amino]cyclohexa-2,4-dien-1-yl]-6-methoxypyridine-3-carboxamide 6-chloro-3-(2-ethylsulfanylpropanoylamino)thieno[2,3-b]pyridine-2-carboxylic acid 5-(2,3-difluorophenyl)-4H-1,2,4-triazol-3-one 1-(benzenecarbonothioylamino)-3-[2-methyl-4-[3-methylbutyl(propanoyl)amino]phenyl]urea [5-(4,4-dimethylcyclohexen-1-yl)pyrimidin-2-yl]-[6-(hydroxymethyl)-3,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-8-yl]-methylideneazanium 2-[1-[4-(3,5-dichloropyridine-4-carbonyl)piperazin-1-yl]ethyl]-7-ethoxy-N'-hydroxyquinoline-4-carboximidamide 4-[7-(2,3-dimethylphenyl)imidazo[1,5-a]pyridin-8-yl]-3,6-dihydro-2H-pyridine-1-carboxylate N-benzylsulfanyl-1-(4-chlorophenyl)-N',3-dimethylcyclobutane-1-carbohydrazide 1-[2-(4-ethylsulfonylphenyl)pyrimidin-5-yl]ethanone 4-[5-(1H-indol-5-yl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-yl]piperazine-1-carboxylic acid 3-[2,4-bis(methoxycarbonyl)phenyl]propanoic acid 1-[(3R,4S)-1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-ol;dihydrochloride 3-(5-cyclopropyl-1H-pyrazol-4-yl)-6-fluoro-7-[4-[2-hydroxyethyl(methyl)carbamoyl]-3,5-dihydro-2H-pyrazine-6-carbonyl]-1-(thiophen-2-ylmethyl)quinolin-4-one 5-(2,6-dimethylphenyl)-7-methylidene-N-(4-piperidin-1-ylphenyl)pyrrolo[3,4-d]pyridazin-8-amine 1-[1-(4,5-diphenylimidazol-2-ylidene)ethyl]pyrrolidine 3,3-difluoropropoxybenzene;4-[(3S)-4-(4,6-dimethylpyrimidin-2-yl)-1-[(2E)-hexa-2,5-dien-2-yl]pyrrolidin-3-yl]morpholine 2-amino-6-hydroxy-N'-[2-methylsulfanyl-5-(trifluoromethoxy)phenyl]benzenecarboximidamide 1,2-bis(4-chlorophenyl)pentane-3,4-dione 5-(azidomethyl)-2,3-dimethoxybenzonitrile 2-(3,4-dihydropyridin-2-yl)-4,5,6,7-tetrafluoroisoindole-1,3-dione 2-[4-methyl-1-[4-(2-phenylethynyl)benzoyl]piperidin-4-yl]oxyacetamide (E)-2,3-diamino-4-[4-methoxy-6-[1-[methyl(propan-2-yl)amino]cyclobutyl]pyridin-3-yl]but-2-enamide (2S)-N,N-dimethyl-1-[1-(1H-pyrazolo[3,4-d]pyrimidin-6-ylamino)ethyl]pyrrolidine-2-carboxamide 4-[[1-(3,5-dimethylpyrazole-1-carbonyl)azetidin-3-yl]methoxy]-2,2-dimethylbutanoic acid N-(4-phenylphenyl)formamide 4-methyl-1-N,3-N-diphenylbenzene-1,2,3-triamine 6-(2,4-difluorophenyl)pyrazolo[1,5-a]pyrazine 4-chloro-N-[2,3-dimethyl-2-(1-piperidin-4-ylethoxy)butylidene]benzenesulfonamide 3-[N'-[(E)-[(2Z,5Z)-4-hydroxy-2-phenylmethoxyhepta-2,5-dienylidene]amino]carbamimidoyl]-1-methylquinoxalin-1-ium-6-sulfonic acid 6-[6-fluoro-2-(5-methoxypyridin-3-yl)-1H-indol-4-yl]-8-methoxyimidazo[1,2-a]pyrazine 5-butyl-3-[4-[2-(1-methoxycyclopropyl)ethynyl]phenyl]-6H-triazolo[4,5-d]pyrimidin-7-one 3-(2,4-dimethylimidazol-1-yl)-N'-[(E)-(3-hydroxyphenyl)methylideneamino]propanehydrazide [2,4-bis(3-methylphenyl)phenyl]boronic acid 2-chloro-N-cyclohexyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-amine 7-ethenyl-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-2,8-dione N-[(3S,4R)-1-benzyl-4-methoxypyrrolidin-3-yl]-2-chloro-6-fluoropyrimidine-4-carboxamide 5-ethyl-1,4-dihydroisoquinoline;5-(4-propan-2-ylsulfonylphenyl)imidazolidine-2,4-dione 1-[1-(4-aminophenyl)ethyl]-3H-imidazo[4,5-b]pyridin-2-one 2-[3-fluoro-4-[2-methyl-5-(oxan-3-yl)pyrimidin-4-yl]phenyl]spiro[5,6-dihydropyrrolo[1,2-b]pyrazole-4,3'-pyrrolidine] (2S,4R)-1-[2-amino-3-(5-nitropyridin-3-yl)propanoyl]-N-[(1R,2R)-1-phenyl-2-thiophen-3-ylcyclopropyl]-4-[2-(tetrazol-1-yl)ethoxy]pyrrolidine-2-carboxamide 4-[(2-chloro-6-methylphenyl)methoxy]-3,5-diethoxy-N-(4-fluorophenyl)benzamide 2-[4-(3,5-dichlorophenyl)sulfinylmorpholin-1-ium-4-yl]-N-ethyl-N-[[3-(trifluoromethyl)phenyl]methyl]pyrimidine-4-carboxamide 2-(6,8-dichloro-3,4-dihydro-1H-pyrano[3,4-c]pyridin-9-yl)-N-methoxy-5-methylpyrazine-2-carboxamide 4-[5,6-bis(ethenyl)-2,3-dihydrofuro[3,2-b]pyridin-7-yl]-N,N-dimethylaniline N-[(3R,4S)-3-aminooxan-4-yl]-2-(4-propan-2-ylphenoxy)acetamide;hydrochloride 7-(1-azido-2,3-dihydrotetrazol-5-yl)-N-[(4-carbamimidoylphenyl)methyl]naphthalene-2-carboxamide [5-(3-methylbutyl)thiophen-2-yl]-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)methanone (6Z)-N'-[2,5-dimethyl-4-[2-oxo-2-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethoxy]phenyl]-6-propylidenepyridine-3-carboximidamide;2-hydroxyacetic acid 5-[4,8-diamino-2-(4-fluorophenyl)imidazo[1,2-a]pyrazin-6-yl]-3H-1,3,4-oxadiazol-2-one;hydrochloride 5-(6,7-dihydro-1H-indole-2-carbonyl)-N,4,6,10-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,11-tetraene-12-carboxamide 3-[(7Z)-9,11-dihydrocycloocta[b]indol-6-yl]-N-(furan-2-ylmethyl)aniline 4-[(3S)-2-oxooxolan-3-yl]-N-[(6S)-3,3,7-trimethyloct-5-en-2-yl]benzamide (3S,5R)-1-[4-(5-hydroxy-2-propan-2-ylphenyl)triazol-1-yl]-N,N-dimethyl-5-phenylpiperidine-3-carboxamide 1-(3,4-dimethylphenyl)-5,6-dimethoxy-2-methylpyrrolo[3,2-b]pyridine [4-(8-amino-1,6-naphthyridin-3-yl)phenyl]methanol 2-(1H-indazole-5-carbonyl)-N,N-dimethyl-3,4-dihydro-1H-isoquinoline-7-sulfonamide (E)-N,1-diphenylmethanimine;N-methylsulfanylcyclohexa-2,5-diene-1-carbothioamide 2-ethyl-5-[4-(5H-imidazo[5,1-a]isoindol-5-ylmethyl)phenyl]pyridine-3-carbonitrile 2-bromo-1-phenylcyclohepta-1,3,5-triene 1-methyl-2,4-bis(methylideneamino)benzene;3-methyl-6H-benzo[c]chromene 1-[2-(3,5-difluorophenyl)acetyl]piperidine-4-carboxylic acid 4-N-(3,5-dimethoxyphenyl)-2-N-[4-(1H-pyrazol-5-yl)cyclohexyl]-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine 2-[(3Z)-4,5-difluoro-6-methoxyhepta-1,3,5-trien-2-yl]-7H-purin-6-amine N-[5-(1H-imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl]-4-methoxy-3-(2-oxopyrrolidin-1-yl)benzamide 5-[(3S)-1-propylpiperidin-3-yl]-2,3-dihydrothieno[3,4-b][1,4]oxazine (E)-2-chloro-3-[2-methyl-4-(trifluoromethoxy)phenyl]prop-2-enenitrile 4-[2-(2-aminopropyl)-5-chlorophenyl]-3-bromoaniline 2-(azidomethyl)-1,3,5-trifluoro-4-phenylbenzene 5-(4-chlorophenyl)-2-[4-methoxy-3-(3-methylbutylsulfanyl)anilino]pentanenitrile 4-(3,5-dimethylpyrazol-1-yl)-N-[2-hydroxy-2-(4-thiophen-2-ylphenyl)ethyl]benzamide (2E,4Z)-4-[5-methoxy-2-(pyridine-4-carboximidoyl)anilino]hepta-2,4-dienal 3-[4-(5,6-difluorocyclohepta-1,2,4-trien-1-yl)oxyphenyl]sulfanyl-N-hydroxypropanamide 6-amino-1-[[3,5-difluoro-2-(methylsulfanylamino)phenyl]methyl]pyrazolo[4,3-c]pyridine-3-carbonitrile 1-[5-(4,7-diazaspiro[2.5]octan-7-yl)pyrazin-2-yl]-N'-methanimidoyl-3-pyridin-3-ylimidazole-2-carboximidamide 1-(4,6-dimethylpyrimidin-2-yl)-3-[5-ethoxy-2-(oxolan-2-yl)pyrazole-3-carbonyl]urea (5Z)-2-[[3,4-bis(phenylmethoxy)phenyl]methylhydrazinylidene]-5-[(4-ethyl-6-oxo-1H-pyrimidin-2-yl)methylidene]-3-methyl-1,3-thiazolidin-4-one N-(2,4-dioxo-1H-pyrimidin-5-yl)-N-(1-hydroxypropan-2-yl)methanesulfonamide (5R)-5-[4-chloro-3-(2,4-difluorophenoxy)phenyl]-1,5,7,11-tetrazatricyclo[6.4.0.02,6]dodeca-9,11-diene (6R)-1,3-dimethyl-8-oxo-7-[(2S)-2-(pyridine-4-carbonylamino)butanoyl]-5,6-dihydroimidazo[1,5-a]pyrazine-6-carboxamide 3-[(1E)-2,4-dimethylpenta-1,3-dienyl]-N'-hydroxybenzenecarboximidamide 1-(3,4,5-trimethoxyphenyl)dodecane-2,6-dione 4-[2,6-dimethoxyethyl(ethenylsulfonyl)amino]benzenesulfonic acid 4-chloro-3,5,7-trimethyl-1H-pyrrolo[2,3-f]benzimidazole N-(4-chlorophenyl)sulfonyl-N-[[2,3-dichloro-6-(1H-pyrazol-5-ylmethyl)-1H-indol-4-yl]oxy]carbamate 4-(1-ethylpiperidin-3-yl)oxypyrimidine (Z)-N'-[4-chloro-2-hydroxy-3,5-bis(trifluoromethyl)phenyl]but-2-enediamide (3Z)-N'-[2,4-bis(phenylmethoxy)phenyl]-N-(5-bromo-1,3-dimethylpyrazol-4-yl)penta-1,3-diene-1,6-disulfonamide 5-[2,6-difluoro-3-(propylsulfanylamino)phenyl]-N-methylidenepyridine-3-carboxamide 2-(5,6,7,8-tetrahydroquinazolin-4-yl)butanamide 4-cyclohexa-1,3-dien-1-yloxy-N'-[(1-methylindol-2-yl)methylideneamino]benzenecarboximidamide 4-[5,6-bis(1,3-benzodioxol-5-yl)pyrazin-2-yl]phenol 2-[(1R,5S)-3-[(2S)-butan-2-yl]sulfonyl-3-azabicyclo[3.1.0]hexan-6-yl]phenol N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethylideneamino]pyridine-2-carboxamide 1-[4-(dimethylamino)phenyl]-3-hydroxypropan-1-one;ethane 1-[2-(3,4-dichlorophenyl)ethylamino]propan-2-one;2-methyl-5H-pyrrolo[2,3-b]pyrazine N-[2-[1,5-dimethyl-3-(trifluoromethoxy)pyrazol-4-yl]ethylsulfanyl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine 4-tert-butyl-N-[2,3-dimethoxy-6-(1H-pyrrole-3-carbonyl)phenyl]benzamide 3,5-ditert-butylpyridine;2,6-dimethylpyridine;iridium(3+);trifluoromethanesulfonate;hexachloride 2-(4,6-dihydropyrrolo[3,4-c]pyrazol-1-ylsulfonylamino)-N-phenylpropanamide 2-chloro-3-ethyl-1,4,5,6,7,8-hexahydrocyclopenta[c]azepine N-[1-(2,6-difluorophenyl)ethyl]-5-(6-methoxypyridin-3-yl)furan-2-carboxamide 2-chloro-4-N,6-diethylpyrimidine-4,5-diamine 1-(3,4,5-trifluorophenyl)pentan-2-one 1-methyl-3-(6-methylidenecyclohexa-2,4-dien-1-ylidene)-5-phenyl-N-propan-2-ylindene-2-carboxamide 2-N-(5-cyclopropyl-1H-pyrazol-3-yl)-4-methanimidoyl-6-(4-pyrrolidin-1-ylbutyl)pyrimidine-2,5-diamine 6-[(4-chlorophenyl)methyl]-2-ethenoxy-5,8-dihydro-3H-pyrido[3,4-d]pyrimidine-4,7-dione 3-[[2,6-bis(2,4-dimethylphenoxy)-1H-pyridine-2-carbonyl]amino]cyclobutane-1-carboxylic acid 3-methyl-2-[2-(3,4,5-trifluorophenyl)ethynyl]phenol 1-[4-bromo-5,6-difluoro-2-(4-fluorophenyl)benzimidazol-1-yl]propan-2-one N-ethyl-2-methoxy-3-(1H-pyrrole-2-carbonyl)benzohydrazide 5-fluoro-2-hydroxy-N,4,6-trimethyl-3-nitrobenzamide 1-[4-[(2,4-dihydroxyphenyl)methyl]piperazin-1-yl]ethanone 2-[(3R)-6-cyclopentyliminospiro[1,4-dihydropyrido[2,3-d]pyrimidine-2,4'-piperidine]-3-yl]phenol 6-[(3,5-difluoro-2-methylphenyl)methoxy]-1H-indole 2-[1-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonylamino)ethyl]pyrazol-4-yl]benzoic acid N-(1,2-oxazol-5-ylmethoxy)-9H-fluorene-2-sulfonamide 3-[2-(aminomethyl)butoxy]-N'-hydroxypyridazine-4-carboximidamide 5-[[4-[3-cyano-2-(difluoromethoxy)phenyl]quinolin-7-yl]sulfamoyl]-6-ethylpyridine-2-carboxylic acid N-[2,3-dichloro-5-(trifluoromethyl)pyridin-4-yl]-2-methyl-3-(trifluoromethoxy)benzamide 1-methylsulfonyl-3,4-dihydro-2H-quinoline 3-[2-fluoro-4-(trifluoromethyl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 1-azidosulfanyl-4-bromobenzene [2-[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]acetyl]-(4-fluorophenyl)azanium;chloride ethane;2-[5-(3,4,5-trimethoxyphenyl)pyrimidin-2-yl]phenol 4-[(3S)-5,5-difluoropyrrolidin-3-yl]-N-[2-methoxy-5-(trifluoromethylsulfanyl)phenyl]benzamide 5-(2,6-difluoro-4-phenylmethoxyphenyl)imidazolidine-2,4-dione 1-[2-(azetidin-1-yl)acetyl]-4-(3,5-difluorophenyl)pyrrolidine-2-carbonitrile 2-(cyclopropanecarbonylamino)-N-[4-cyano-2-methyl-5-(5H-pyrido[3,4-b]indol-7-ylsulfanyl)phenyl]pyridine-4-carboxamide N-[3,5-dimethyl-1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]formamide N-[3-cyano-5-(1,2-dihydroxyethyl)phenyl]benzamide (1S)-5-methyl-3-propyl-2,3-dihydro-1H-inden-4-ol [3-(1,3-dimethylpyrazol-4-yl)morpholin-4-yl]-(5-propan-2-ylthiophen-2-yl)methanone 1-(5,7-dichloro-3,4-dihydro-2H-quinolin-1-yl)butan-1-one 3-[5-methyl-2-(3-piperidin-1-ylpropoxy)phenyl]oxirane-2,2-dicarbonitrile 2-[2-amino-4,6-bis(trifluoromethyl)phenyl]sulfanyl-3H-quinazolin-4-one 2,5-dimethylbenzenesulfonate;diethoxyphosphinic acid 5-[4-(4-hexylphenyl)-1,3-thiazol-2-yl]-6,7-dihydro-4H-thieno[3,2-c]pyridine (4-hydroxyphenyl)-[8-phenyl-2-(trifluoromethyl)quinolin-3-yl]methanone 4-[4-(2,6-dimethylphenyl)piperazin-1-yl]-N'-hydroxypyridine-2-carboximidamide (4Z)-2-methyl-4-[[5-nitro-2-[(4-nitrophenyl)methoxy]phenyl]methylidene]-1,3-oxazol-5-one 3-(2,6-dichlorophenyl)-7-[4-(2-hydroxyethyl)piperazin-1-yl]sulfonyl-1H-quinazoline-2,4-dione (Z)-2-[3,5-dimethyl-1-[4-[5-[3-methylbutyl(propyl)amino]pentoxy]phenyl]pyrazol-4-yl]-N-ethenyl-N-ethylbut-2-enimidamide (4S)-3,4-dihydroxy-1-(2-methylpropylsulfanyl)-6-thiophen-2-ylhexa-1,5-dien-3-one 1-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-3-(2-fluoroethyl)urea 4-[8-amino-5-methyl-3-(trideuteriomethoxy)imidazo[1,2-a]pyrazin-6-yl]benzaldehyde;5-[[deuterio-[2-fluoro-3-(trifluoromethoxy)phenyl]methyl]amino]pyridine-3-carbonitrile 2-[[5-[(3-chlorophenyl)methyl]furan-2-carbonyl]amino]-3-thiophen-2-ylpropanoic acid N-methylsulfonyl-5-propan-2-ylthiophene-3-carboxamide 2-azidosulfanyl-1-[3,5-difluoro-4-(trifluoromethoxy)phenyl]ethanol N-(3,4-difluorophenyl)-7,8-dimethylpyrido[4,3-d]pyrimidin-2-amine;ethane 4-chloro-N-[(1R,2S)-2-nitrocyclohexyl]aniline 2-(5,6-diethylpyrimidin-4-yl)oxy-1-(3-methylpiperidin-1-yl)ethanone 3-(N'-benzylcarbamimidoyl)sulfanyl-N,N-dibutylpropanamide;hydrobromide 5-N,7-dimethylspiro[5H-imidazo[1,2-a]quinoline-4,3'-oxetane]-6-amine 3-[1-(2,5-dimethylphenyl)ethenyl]-4-[4-(methoxymethyl)phenyl]piperidine 5-[(Z)-hydroxyiminomethyl]-4-(2,3,6-trifluorophenyl)-1H-imidazole-2-carboxamide 4-[2,3-bis(trifluoromethyl)phenyl]-1H-pyridazin-6-one 2-[(4E,5Z)-3,7,11,15,19-pentadeuterio-6,10-difluoro-2-methyl-9-oxa-7,14-diazatetracyclo[9.8.0.03,8.013,18]nonadeca-1,3(8),4,6,12(18),13,16-heptaen-5-yl]benzaldehyde [4-(methylamino)piperidin-1-yl]-(2H-quinolin-3-ylidene)methanolate (5E)-2-cyclohexylimino-5-[[3,4-dihydroxy-6-(4-nitrophenyl)pyridin-2-yl]methylidene]-1,3-thiazolidin-4-one 5-(3,5-difluorophenyl)-1,2-oxazole 4-methylbenzenesulfonate;pyridin-1-ium-3,7-diol (3-methyl-3,6-dihydro-2H-1,4-oxazin-5-yl)-[4-(4-phenylphenyl)thiophen-2-yl]methanone 2-(3,4-difluorophenyl)sulfanyl-1-[2-(1H-pyrazol-5-ylmethoxy)ethyl]-6-pyrrolidin-1-ylimidazo[4,5-c]pyridine 2-[[4-(diethylamino)phenyl]methyl]-7-phenylpyrazolo[3,4-d]pyrimidine-3-carboxylic acid N-[4-(dimethylamino)-2,6-dimethoxyphenyl]furan-3-carboxamide N-[(E)-(3,4-dihydroxyphenyl)methylideneamino]-6-fluoronaphthalene-2-carboxamide 4-[(2S)-butan-2-yl]sulfanyl-6,7-difluoro-1H-indole N-[4-(1,3-benzothiazol-2-ylamino)phenyl]formamide 1-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-N'-hydroxyimidazole-2-carboximidamide N-(4-acetamidobutyl)-2,3-dimethoxybenzamide 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-[2-[1H-imidazol-5-ylmethyl(phenacyl)amino]ethyl]amino]octanoic acid (4E,5Z)-3,5-diamino-N'-[(Z)-1-(1H-benzimidazol-2-yl)ethenoxymethyliminomethyl]-4-methylidenehepta-5,7-dienehydrazide 5-chloro-1-[4-(difluoromethoxy)phenyl]-2,3-dihydroisoindole 2-(9-acetyl-4,9-diazaspiro[5.5]undecan-4-yl)-N-methylpyridine-3-carboxamide;2,2,2-trifluoroacetic acid 4-[3-(diethylamino)-2,5-dimethoxyphenyl]-1H-pyrimidin-6-one (E)-N'-amino-3-[4-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxymethyl)phenyl]piperidin-1-yl]prop-2-enimidamide (2E)-5-ethenyl-N'-[1-[4-(trifluoromethoxy)phenyl]propyl]hexa-2,4-dienehydrazide 3-[4-[3-ethylsulfonyloxy-5-(methoxymethoxy)phenoxy]-2,6-difluorophenyl]azetidine 4-methyl-3,5-diphenyl-1H-pyrazole 2-methylprop-1-ene;9-[4-(3,7,11-trimethyldodeca-1,8-dien-2-yloxy)phenyl]fluoren-9-ol (2R)-1,2-bis(benzenesulfonamido)-5-chlorocyclohexa-3,5-diene-1,3-dicarboxylic acid 2-(9H-fluoren-1-yl)-3,5,6-trifluorophenol 3-methyl-N-[6-(6-methyl-1,4-oxazepane-4-carbonyl)pyridin-2-yl]benzamide 6-(methyliminomethyl)-2-phenylcyclohexa-1,3-dien-1-amine 2-[(Z)-[6-(azepan-1-ylmethyl)benzimidazol-2-ylidene]amino]guanidine 4-azido-2,6-dimethyl-1H-indole N-(5-chloropyridin-2-yl)-3,4,6-trihydroxynaphthalene-1-carboxamide (3R)-1-[6-azido-3-fluoro-2-(2,3,5-trichlorophenyl)phenoxy]-3-methylpyrrolidine 4-tert-butyl-2-(triazolo[1,5-a]pyridin-3-ylmethylamino)-1H-pyrimidin-6-one 3,5-dichloro-4-methoxycarbonylbenzoic acid 4-azidooxy-2,3-dichloroaniline (Z)-3-[4-(furan-2-ylmethoxy)phenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile 2-bromo-5,6,7,8-tetrahydroquinoline 2-[6-(6,8-dichloro-4-methylquinazolin-7-yl)oxyhexylamino]ethanol 4-[1-azidooxy-2-methyl-1-(1,3-thiazol-4-yl)propan-2-yl]aniline 1-cyclopropylsulfonyl-4-methylbenzene;N-ethanethioylformamide 1-[[6-(4-ethylsulfonylphenoxy)-7H-purin-2-yl]amino]ethanol [5-(1,3-benzodioxol-5-yl)-6-[2-[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]ethoxy]imidazo[1,2-a]pyridin-2-yl]methanimine 3-amino-N'-[6,7-dimethyl-2-oxo-1-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-yl]pyrrolidine-1-carboximidamide N-(2,3-difluorophenyl)-N'-hydroxy-1H-imidazo[4,5-b]pyridine-7-carboximidamide N-[(1S,2R)-3-(4-methylphenyl)-3-oxo-1-(1H-pyrazol-5-yl)propyl]cycloheptanecarboxamide 3-azidooxy-5,6-dimethylpyridine-2-carboxamide 2-(cyclohexylamino)-3-[4-[[4,5-dimethyl-N-propanoyl-2-(trifluoromethoxy)anilino]methyl]phenyl]propanenitrile 2-(N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-5-yl]phenyl]anilino)guanidine 4-[(1Z)-3-cyanobuta-1,3-dienyl]-N-cyclohexa-1,5-dien-1-yl-N'-phenylbenzohydrazide 3-[4-[5-chloro-2,7-bis(sulfanyl)cyclohepta-1,4,6-trien-1-yl]phenyl]-1,1-dimethylurea 2-[4-(trifluoromethyl)phenyl]-3H-quinazolin-4-one 1-(6-chloropyrazin-2-yl)azepan-3-amine 1-azido-4,4a,5,6,10b-hexahydroindeno[2,3-b]indole 1-ethylsulfanyl-4,5-dimethoxy-2-nitrobenzene 4-(3,5-dimethylphenyl)-2,7-bis(ethenyl)quinoline;ethane 4-chloro-3-[(3,5-diethoxyphenoxy)methyl]benzoic acid 4-[3-fluoro-5-(trifluoromethyl)phenyl]cyclohexan-1-amine 6-(2-bromo-N-butanoylanilino)-4-hydroxynaphthalene-2-sulfonic acid 1-[2-(4-fluorophenyl)ethyl]-3-[(3R,5S)-1,2,3,4-tetrahydroisoquinoline-3,6-diyl]urea 2-[3,5-difluoro-4-[(2S)-6-nitro-9H-pyrido[2,3-b]indole-2-carbonyl]phenyl]acetic acid 2-(4,6-dimethoxypyrimidin-5-yl)-7H-purine (2S,5R)-1-[(3-bromophenyl)methyl]-2-ethynyl-4-(oxan-4-yl)piperazine 2-methyl-4-[(4-methylsulfanylanilino)methyl]phenol 4-[4,6-di(propan-2-yl)pyrimidin-2-yl]-5-methyl-1H-indazole (2R)-3-[6-[2-[4-hydroxy-5-(3,3,5,5-tetramethylcyclohexen-1-yl)pentyl]iminoethylamino]pyridin-3-yl]-N-methoxy-2-methylpropanamide 2-(5-amino-6-oxo-1H-pyrimidin-4-yl)isoindole-1,3-dione 1-(4-methylcyclohexyl)oxycarbonylpyridin-1-ium-3-carboxylic acid 4-[(6R)-7-acetamido-8,8-dimethyl-3-propanoyl-1,5-dioxonan-2-yl]oxybenzoic acid ethane;4-N-[1-(6-methoxypyridin-3-yl)ethenyl]-2-N-(3-morpholin-4-ylpropyl)pyrimidine-2,4-diamine 2-ethenylsulfanyl-3,4-difluoro-N'-hydroxybenzenecarboximidamide 1-[(4-chlorophenyl)methyl]-3-[2-(4,5-dihydro-1H-imidazol-2-ylamino)propanoylamino]thiourea (3E)-1-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-phenylpyrazol-3-yl]-3-[(3,4-dimethoxyphenyl)methylidenehydrazinylidene]propan-2-one 2-azido-1-(3,4-difluorophenyl)-N-(pyridin-2-ylmethyl)ethanamine 2-(3,4-dimethoxyphenyl)-N'-hydroxy-5-(2-hydroxyethylamino)pyridine-4-carboximidamide 6,9-dimethyl-2-pyridin-3-yl-5,6,7,8-tetrahydropyrimido[4,5-b]indole 2-[N-(3-methylbutyl)anilino]propanoic acid (E)-5,7-difluoro-N-[4-methoxy-2-(3-methylbutanoylamino)phenyl]-6,8-dioxooct-5-enamide;methane 6-[(6-cyclopropylpyridin-3-yl)methoxy]-2,3-dihydro-1H-pyrrolo[1,2-a]indole 2-[[6-(4,5-dimethylfuran-3-yl)pyridine-3-carbonyl]amino]-7-(3-methoxyazetidin-1-yl)thieno[3,2-b]pyridine-3-carboxylic acid N-ethyl-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a]quinoline-8-carboxamide;hydrochloride 2-(2,4-dichlorophenyl)ethyl-oxosulfanium 2-[3-(5,7-dimethyl-1H-indol-4-yl)phenyl]ethanol N-azido-N-methyl-5-phenylpentanamide 4-methoxy-2,3-dihydrobenzo[g]indazole N-[5-fluoro-4-(1,3-thiazol-2-ylmethoxy)pyrimidin-2-yl]-6-fluoro-2H-1,2,4-benzothiadiazine-8-carboxamide 2-azidooxy-3-chloro-5-(trifluoromethyl)benzonitrile 6-(1,1-dioxo-2H-thiopyran-3-yl)-N-methyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-amine 3-[5,6-difluoro-2-(4-propylphenyl)sulfanyl-1H-benzimidazol-4-yl]-N-(2-methoxyethyl)imidazo[1,2-b]pyridazin-6-amine 4-(2,3-dihydroindole-1-carbonyl)-N'-methylsulfanylbenzenecarboximidamide N-[[3,5-bis(trifluoromethyl)phenyl]methoxy]pyridine-2-carboxamide;ethane N-[2-chloro-5-(6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonyl)phenyl]-2-methylpropane-1-sulfonamide (3E)-1,4-dimethyl-3-[(2-methylpyrimidin-5-yl)methylidene]piperazine 5-(1,4-dimethylpiperazin-2-yl)-3-[1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfonyl)piperidin-4-yl]-1,2,4-oxadiazole N-[(2S,4R)-4-hydroxy-1-[3-methoxypropyl(2-pyridin-4-ylethyl)carbamoyl]pyrrolidin-2-yl]pyridine-3-carboxamide 1-azido-3,3,5-tributyl-2-methoxybenzene 5-[2-(7-chloroquinolin-4-yl)sulfanylphenyl]-6-(2,3,4-trifluorophenyl)-1H-pyrazolo[4,3-c]pyridin-7-one N-[4-(aminomethyl)-2-chlorophenyl]-6-[3,5-bis(trifluoromethyl)phenoxy]pyrimidin-4-amine 2-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]propanedioic acid 1-[2-(2,3-dihydrofuran-5-yl)ethyl]-3-[(4-fluorophenyl)methylamino]thiourea 2,4-dichloro-N-[(Z)-2-methyl-1-phenylbut-1-enyl]aniline 1-[(3,5-dichloropyridin-4-yl)methyl]-2-[5-ethenoxy-1-(propan-2-ylsulfamoylamino)isoquinolin-7-yl]imidazole 1-[(3,4-difluorophenyl)methyl]-2-[1-[(6-methoxypyridin-3-yl)methyl]piperidin-3-yl]benzimidazole N-[1-(4-ethylanilino)-3,4-dimethylpentan-2-yl]-4-(hydroxymethyl)-1H-pyrrole-2-carboxamide 2-[4-[(1S)-6-[3,5-difluoro-4-[(2-fluorophenyl)methoxy]phenyl]naphthalen-2-yl]cyclohexyl]propan-2-ol 2-[2-(methoxymethyl)azetidine-1-carbonyl]-6H-pyrrolo[3,4-c]pyrazol-4-one 6-chloro-2-(2,3,5-trimethoxyphenyl)quinoxaline 1-(3,4-dihydro-2H-quinolin-1-yl)butan-2-ol 2-amino-4,5-dichloro-N-cyclopropylbenzenecarboximidate 7-chloro-2,3-dihydro-1H-pyrrolo[2,3-c]pyridine;(4S)-2-ethyl-4-methoxy-3,4-dihydro-1H-isoquinoline 4-amino-6-[(3-bromo-5-methoxy-4-prop-2-enoxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-azidooxy-2,3-di(pentanoyl)benzenesulfonic acid N'-(1,3-thiazol-4-ylmethyl)spiro[1H-2-benzofuran-3,9'-xanthene]-5'-amine 2-[[(1S,3R)-4-[(2,6-dichloropyridine-3-carbonyl)amino]-3-hydroxycyclohexyl]-methylcarbamoyl]propanoic acid 1-(4-methoxyphenyl)-3-[2-[2-(trifluoromethyl)phenyl]-2H-pyridin-1-yl]propan-2-one 4-[4-(2,6-dimethylpyridin-3-yl)phenyl]-6-fluoro-3,8a-dihydro-1H-quinolin-2-one N-[3-(dimethylamino)phenyl]-5-propan-2-ylfuran-2-carboxamide 1-azido-4-fluoro-2-[(4-methoxyphenyl)sulfanylmethoxy]benzene 2-chloro-5-(trifluoromethylsulfanyl)-4H-pyrrolo[3,2-b]pyrrole N-[1-(2,5-dimethoxyphenyl)sulfonylpiperidin-4-yl]-N-pyrazin-2-ylacetamide N-(3,4-dimethoxyphenyl)-2-[3-fluoro-5-[2-[5-[(E)-1-iminobut-2-en-2-yl]pyridin-2-yl]pyridin-4-yl]phenyl]acetamide 1-(4-acetylpiperidin-1-yl)-2-[4-[3-[3-(6-chloropyridin-2-yl)propanoyl]-5-fluorophenoxy]-3,7-dihydro-2H-inden-1-ylidene]ethane-1,1-dione 2-methyl-N-[5,6,7-trichloro-3-(1H-indol-2-yl)quinolin-4-yl]propanamide [2-amino-5-(3,4-dimethoxyphenyl)pyridine-3-carbonyl]azanium 2-(3,4-dimethoxyphenyl)quinoline;ethane 2-[3-(4,6-dimethylpyrimidin-5-yl)-1-phenylpyrazol-4-yl]-N-ethylethanamine;propane 2,3-bis[(4-hydroxyphenyl)methylidene]imidazolidine-4,5-dione 3-(8,9-dimethoxy-3H-pyrazolo[4,3-c]quinolin-2-yl)propanamide 1-azidooxy-4-methylsulfanylnaphthalene 2-azido-4,6-ditert-butyl-N,N-bis[(2,3,5,6-tetrafluorophenyl)methyl]aniline 4-[4-[2-(4-cyclopropylpyridine-3-carbonyl)-1,3-thiazol-5-yl]phenyl]cyclohexane-1-carboxylic acid 5-[2,6-dichloro-4-(2-methoxyethyl)phenoxy]-1H-indazole 4-[(Z)-2-[5-[(E)-2-carboxyethenyl]thiophen-2-yl]ethenyl]pyridine-2,3-dicarboxylic acid 6-tert-butylsulfonyl-8,9,10,11,12-pentazatetracyclo[7.7.0.02,6.010,15]hexadeca-1(16),2,4,11,13-pentaene N-[1-(3,4-difluorophenyl)ethyl]-2-hydroxy-2-[3-[methyl-[[5-(trifluoromethyl)furan-2-yl]methyl]amino]pyrrolidin-1-yl]propanamide N-[4-fluoro-5-[2-(3-hydroxypiperidin-1-yl)pyrimidin-5-yl]-2-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-2-yl)phenyl]-6-oxo-4-(trideuteriomethyl)-1H-pyridine-3-carboxamide 1-(2,4-dimethoxy-6-methylphenyl)-3-[[2-(trifluoromethyl)cyclohepta-2,5-dien-1-ylidene]amino]urea 4-chloro-1-[2,6-di(propan-2-yl)phenyl]sulfonylindole 4-[(2S,3R)-1-butylsulfanyl-5-oxoheptan-2-yl]benzoic acid 2-amino-4-(3,5-dimethoxyphenyl)imino-5-(quinolin-6-ylmethylidene)imidazol-1-ium-1-ol 1-ethenylsulfonyl-3-propylbenzene [(2R)-3-hydroxy-2-[4-(trifluoromethyl)phenyl]propoxy]-oxido-oxophosphanium 2-[4-(3,6-dimethylpyrazine-2-carbonyl)piperazin-1-yl]-1-pyrrolidin-1-ylethanone 2-[5-methyl-4-[(1R)-1-[3-methyl-5-(2-phenylethynyl)pyridine-2-carbonyl]oxyethyl]-6-oxopyridazin-1-yl]acetic acid 2-methyl-2-[2-[4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)piperidin-1-yl]propanoylamino]propanoic acid 5-[3-[(2-propylpyrazol-3-yl)methoxy]phenyl]imidazolidine-2,4-dione 3-methyl-5-(4-propoxynaphthalen-1-yl)-2H-pyrazolo[3,4-b]pyridine N-cyclopentyl-2,5-dimethylpyrimidine-4-carboxamide 2-(2,3-dioxo-1,4-benzoxazine-7-carbonyl)benzoic acid [3-(4-hydroxyphenyl)thiophene-2-carbonyl]azanium 1-[1-(3,4-difluorophenyl)ethyl]-4-(triazol-1-ylmethyl)piperidine;formic acid 1-[4,6-bis(3-propanoylphenyl)-1H-inden-2-yl]ethenol 1-N',4-N'-bis(3,5-dimethylphenyl)butanedihydrazide 4-[2-(3,5-diamino-1H-pyrazol-4-yl)ethenyl]benzene-1,3-diol N-(3,4-difluorophenyl)-7H-purin-2-amine 5-(2,4-dihydroxyphenyl)-1H-pyrazole-3-carboxylate (2R,3R)-1-[3-methyl-7-oxo-6-(pyridin-4-ylmethoxy)-5H-pyrazolo[5,1-b][1,3]oxazepine-2-carbonyl]-N-[[3-(trifluoromethoxy)phenyl]methyl]pyrrolidine-2-carboxamide 2-tert-butyl-4-methyl-N-[5-(trifluoromethyl)pyridin-3-yl]morpholine-3-carboxamide 4-[(4,5-dimethyl-1H-pyrazol-3-yl)amino]benzoic acid (3E,5Z)-4,8-dimethylideneundeca-1,3,5,10-tetraene;5-methylcyclopenta-1,3-diene 3-[4,5-bis(2,2-dimethylpropanoyl)pyridin-2-yl]-1,3-oxazolidin-2-one 1-azidooxy-2-methylsulfanylnaphthalene [1-(5-cyanopyridin-2-yl)azetidine-3-carbonyl]azanium 1-[4-(2,3-dihydro-1H-pyrrole-5-carbonylamino)phenyl]-5-oxopyrrolidine-3-carboxylic acid 3-(benzenecarboximidoyl)benzonitrile;4,9-dihydrocarbazol-1-ylbenzene 1-[(4aS,7aS)-6-methyl-1,2,3,4,4a,5,7,7a-octahydropyrrolo[3,4-b]pyridin-8-yl]-2-(3H-benzimidazol-5-yl)ethanone 1-azidooxy-3,4,5,6-tetrafluoronaphthalene 3-amino-2-[[2,5-difluoro-4-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)phenyl]methyl]butanamide 4-(2,6-ditert-butylpyrimidin-4-yl)cyclohexa-1,3-diene-1-carbonitrile 3-amino-N-[(5E)-5-[(2,4-dichlorophenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]benzamide 2-[[7-(3,5-dichlorophenyl)-1,6-naphthyridin-5-yl]amino]-N-[(2R)-4-[4-(1-methylpiperidine-3-carbonyl)piperazin-1-yl]oxolan-2-yl]acetamide 4-[1-[2,6-dichloro-3-[1-(dimethylamino)ethenyl]phenyl]ethoxy]piperidine-1-carboxylic acid 2,4-dichloro-3-N,3-N-bis(ethylamino)benzene-1,3-dicarboxamide ethane;4-[1-methylsulfonyloxy-3,3-di(propanoyloxy)butyl]benzoic acid 2-(1,3-benzodioxol-5-ylmethoxy)-6-chloronaphthalene N-[(Z)-1-(4-hydroxyphenyl)ethylideneamino]quinoline-3-carboxamide 5-[2-hydroxyethyl(1,3-thiazol-5-yl)amino]naphthalene-2-sulfonic acid ethane;2-[(2E,5Z)-hepta-2,5-dien-3-yl]oxy-1,4-bis(sulfanyl)benzene 2-[4-chloro-2-(4,5-dihydro-1H-imidazol-2-yl)phenoxy]acetic acid 1-[3-(2,4-difluorophenyl)-5-methylpyridin-4-yl]ethanone;methane 2-(4,6-diphenylpyridin-3-yl)-7H-[1]benzofuro[3,2-b]quinoline 2,4-dichloro-N-ethyl-N-(4-propylphenyl)pyrimidin-5-amine 6-[(2,4-dimethoxyphenyl)methyl]-3-pentan-3-ylcyclohexene-1-carboxylic acid 2-(9H-fluoren-1-yl)ethenoxybenzene N-[4-(1H-benzimidazol-2-ylmethylamino)-3,4-dioxobutyl]-5-chloropyridine-2-carboxamide;hydrochloride N-[2-chloro-5-(trifluoromethyl)phenyl]-1-[(4-oxo-3H-quinazolin-2-yl)sulfanyl]cyclopentane-1-carboxamide (4-ethylphenyl)-[4-(2H-tetrazol-5-ylmethoxy)piperidin-1-yl]methanone 5-azidosulfanyl-2H-pyrazolo[3,4-b]pyridine 3-[2-(aminomethyl)-3-fluoropropoxy]-2-(1,1-difluoroethyl)-5-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonylamino)benzamide N-[(1R)-2-amino-2,3-dihydro-1H-inden-1-yl]-1-methylpyrazole-4-carboxamide N-(4-azidophenyl)-6-[[methyl-[(3R)-pyrrolidin-3-yl]amino]methyl]pyridine-3-carboxamide 3,5-dibromobenzoic acid;2-methylpropane 1-[4-[3-(trifluoromethoxy)phenyl]butanoyl]azetidine-2-carbonitrile N-[6-[2-(cyclopropanecarbonylamino)imidazo[1,2-b]pyridazin-6-yl]oxynaphthalen-1-yl]-4-hydroxypyrrolidine-3-carboxamide;prop-1-ene [6-hydroxy-3-(iodomethyl)-2H-indazole-5-carbonyl]oxidanium 1-(5-chlorofuran-2-yl)sulfonyl-N-[(2R,3S)-2-pyrazol-1-yloxolan-3-yl]pyrrolidine-3-carboxamide N-[(2,6-dichlorophenyl)methyl]-3-(2H-indazol-3-yl)thiophene-2-carboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-amine 2-(dimethylsulfamoylamino)-N-(5-propan-2-ylpyridin-2-yl)propanamide 1-(azidomethyl)-2,4,5-trifluoro-3-propan-2-yloxybenzene ethane;3-[(Z)-2-hydroxyethenyl]-N',5-dimethanimidoyl-1H-indole-6-carboximidamide 5-[5-(methoxymethyl)-1,3,4-oxadiazol-2-yl]-6-phenyl-7H-pyrrolo[3,4-b]pyridin-7-ol 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-1,3-benzothiazole (7S)-N-(4-ethoxyphenyl)-5-methyl-7-[2-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 1-N'-[2,3-difluoro-4-[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]-1-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide N-[(3R)-1-cyanopyrrolidin-3-yl]-2-(4-fluorophenyl)acetamide N-[(Z)-2-aminoethenyl]-N'-tert-butylbenzenecarboximidamide 6-[[5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]piperidin-2-one N'-[3-ethynyl-4-(5-methoxypyridin-2-yl)phenyl]-2,2,2-trifluoroethanimidamide (NZ)-N-[2-[3,5-dimethyl-4-(2H-tetrazol-5-yl)phenoxy]ethylidene]hydroxylamine N-[3-amino-1-(3,4-dihydroquinolin-2-yl)propyl]formamide 3-(N-pyridin-2-ylanilino)propane-1,2-diol N-(3,4-dihydroxyphenyl)-2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxoisoquinoline-5-sulfonamide 3,5-diethyl-2-methyl-1H-benzimidazole-4,6-dione N-[3-(azepan-1-ylmethyl)phenyl]-2-(4-methoxycarbonylpiperazin-1-yl)pyrimidine-5-carboxamide 3-(2,6-difluorophenyl)-5-[4-(trifluoromethylsulfonyloxy)phenyl]-1H-pyrrolo[2,3-b]pyridine 1-(7-chloro-5-methoxy-2,3-dihydroindol-1-yl)-2-[4-(trifluoromethyl)pyridin-3-yl]ethanone 2-(3,5-difluorophenyl)-N'-hydroxy-3-[4-(hydroxymethyl)cyclohexyl]propanehydrazide (2R,3R)-4,4,4-trifluoro-3-methoxy-N-[6-methyl-5-[2-[(2S)-oxolan-2-yl]acetyl]pyridin-2-yl]butanamide [3-(3,4-difluorophenyl)azetidine-1-carbonyl]iminoazanide;(2S,5R)-2-[(E)-but-1-enyl]-5-methoxyoxolane;5-chloro-3-methylimidazo[4,5-b]pyridin-2-one;yttrium ethane;6-[(2Z,4E)-hexa-2,4-dienyl]-1,3-benzothiazole 2-(4-anilinocyclohexyl)oxyethanol ethane;[4-(3-methylphenyl)-2H-1,2,5-oxadiazol-5-id-3-yl]-phenylmethanone 2-[(3-chlorophenyl)methyl]-3H-imidazo[4,5-c]quinoline 2-(5,6-dihydronaphthalen-1-yl)benzo[f]isoquinoline (5R,6S)-5-[3-[4-(2-hydroxyethylamino)-1-phenylbutan-2-yl]phenyl]-1-methyl-6-propylpiperidin-2-one 1-(4-azido-3,6-dihydro-2H-pyridine-1-carbonyl)pyrazole-4-carboxylic acid 6-[(5-fluoropyridin-2-yl)methoxy]-3,4,7-trihydroxy-1H-quinolin-2-one 3-(4-bromophenyl)-2,3-dihydroinden-1-one 3-amino-6-(4-methoxyphenyl)-5,6-dihydrobenzo[h]quinazolin-8-one 2-[[6-chloro-5-(3,4-dimethoxyphenyl)pyridine-2-carbonyl]amino]-3-(3-nitrophenyl)propanoic acid (E)-4,4-difluorobut-2-enoxy-[3-[6-[(1R)-1-hydroxyethyl]pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-5-yl]methanol 4-(2,5-dimethoxyphenyl)-2-[6-[3-(hydroxymethyl)pyrrolidin-1-yl]pyridin-2-yl]-N'-(2-propanoyl-6-azaspiro[3.3]heptan-6-yl)-5H-pyrrolo[3,2-d]pyrimidine-7-carboximidamide N-[2-(cyclohexylcarbamoylamino)phenyl]-N-(3,5-difluoro-1-methylpyrazol-4-yl)-N'-ethylethanimidamide 2-azido-4,5-dichloropyrimidine 2-(cyclohexen-1-yl)-5-[2-[6-[4-[difluoro(iodo)methoxy]-3,5-difluorophenyl]naphthalen-2-yl]ethynyl]pyrimidine 7-methyl-4-[4-(trifluoromethyl)phenyl]quinazoline 1-[(3S,7R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-N-cyclopentylpyrazole-4-sulfonamide (2S,3R)-4-[2-methyl-7-(1H-pyrazol-5-yl)quinolin-4-yl]oxypyrrolidine-3-carboxylic acid;hydrochloride 1-(3-ethylphenyl)-N,N'-dimethylpropane-2,3-diamine;hydrobromide 5-(1,3-benzodioxol-5-yl)-2,4-dimethoxy-N-methyl-N-[(Z)-pentylideneamino]benzamide 1,4-dimethylcyclohexa-2,4-diene;iridium(3+);8-(4-methoxybenzene-6-id-1-yl)quinoline N-[2,3-diamino-5-(trifluoromethyl)phenyl]acetamide [2-(3,5-difluorophenyl)pyrrolidin-1-yl]-(5-methoxypyrazin-2-yl)methanone;formic acid N-[(3,4-dimethoxyphenyl)methyl]-2-[(1S,4R)-4-hydroxy-3-(4-oxobutanoylamino)cycloheptyl]acetamide 5-(1H-indol-3-yl)thiophene-2-carboxylic acid 6-amino-4-(2,3-dichlorophenyl)-4-methyl-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile N-[(1S)-1-cyclohexylethoxy]-2-(1,3-dioxoisoindol-2-yl)benzamide 3-ethyl-1,2,3,4-tetrahydrophenanthrene 4-bromo-2,3-bis(ethenyl)pyridine 1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)propanoyl]piperidine-2-carboxylic acid;formic acid 1-[(3,4-dichlorophenyl)methyl]pyridine-2-thione 6-(4,5-dihydropyrimidin-2-yl)-5-methylidenecyclopenta[f][1]benzothiole 1-[(5-chloropyridin-2-yl)methoxy]-3,4-dihydro-2H-naphthalen-1-ol 5-bromo-6,8,9,10-tetrahydroindeno[1,2-b]pyridine-7,11,12-trione 3-[1,4-dimethyl-2-(4-methylphenyl)-5-methylidenepyrrol-3-yl]propanoic acid N-[4-(2,6-dimethoxyphenoxy)phenyl]propanamide;ethane 2-[6-(3,4-difluorophenyl)pyrazin-2-yl]-4-thiophen-2-ylbutanoic acid N-[4-[1-(2,3-dihydro-1H-indene-2-carbonyl)piperidin-4-yl]butyl]imidazo[1,5-a]pyridine-6-carboxamide 2-(4-ethylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 1-(3-ethyl-3,5-dimethoxycyclohexa-2,4-dien-1-yl)-7-hydroxy-6-methoxyquinolin-2-one 4-[3-(2,5-dimethylphenyl)buta-1,3-dien-2-yl]-2,6-bis(trichloromethyl)-1,3,5-triazine 1-[3-(dimethylsulfamoyl)phenyl]-7-[[6-methoxy-2-(4-methylbenzimidazol-1-yl)quinoline-3-carbonyl]amino]heptan-5-one 5-(2,3-dichlorophenyl)sulfanyl-N'-hydroxypyrazine-2-carboximidamide 6-methyl-3-(6-oxo-1H-pyridin-2-yl)pyridazine-4-carbonitrile N-[2,6-difluoro-3-(methoxyiminomethyl)phenyl]-1-methyl-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide 2-(1,3-benzodioxol-5-yl)-N-[4-methyl-6-[1-(oxetan-3-yl)piperidin-4-yl]oxypyridin-3-yl]acetamide 3-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[1-hydroxy-4-(1H-indol-3-yl)butan-2-yl]propanamide 4-(8,13,14-triazatetracyclo[7.6.0.02,7.010,15]pentadeca-1(9),2,4,6,11,14-hexaen-12-yl)piperidine-1-carboxylic acid ethane;4-methylpentanal;(E)-1,3,3-triphenylprop-2-en-1-one (Z)-2-[(Z)-1H-indol-3-ylmethylideneamino]oxy-N,N-dimethylethanamine 2-amino-4-[5-(1,3-benzodioxol-5-yl)-2-propan-2-yloxyphenyl]-6-methylbenzene-1,3-dicarbonitrile 3-[6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-yl)pyridazin-3-yl]benzonitrile 4-[2,3-dihydroxypropyl(phenacyl)amino]benzenesulfonic acid (4R)-3-[(2S,5R)-3,7-dimethyl-1-oxo-6-[2-(trifluoromethoxy)ethoxy]heptan-2-yl]-1,3-thiazolidine-4-carboxylic acid 6-[(3R)-3-methylpyrrolidin-1-yl]-N-propan-2-ylpyridazine-3-carboxamide N-[4-[1-(4-fluorophenyl)ethyl]cyclohexa-2,4-dien-1-yl]-4-hydroxy-3-methoxybenzamide 2-[(4-fluoro-3,5-dimethylphenoxy)-phenylmethoxy]-1H-pyridine 3-(4-hydroxybutyl)-2,3-dihydrochromen-4-one 1-[(2,6-dichlorophenyl)methyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one 2-chloro-N-(4,5-dimethyl-1H-pyrazol-3-yl)-4-(dimethylaminosulfanyl)aniline 5-[3-(azidomethyl)phenyl]-1,2,4-oxadiazole 4-(1-azidoethenyl)-2,3-dimethoxyphenol 5-(4,6-dimethylpyrimidin-2-yl)pyridine-3-sulfonamide 4-[1-[[2-methylsulfanyl-5-(trifluoromethyl)pyridine-3-carbonyl]amino]cyclobutyl]benzoic acid 2-[1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethyl]-3H-quinazolin-4-one 2-(4-fluorophenoxy)-N-[(1R,5S)-6-propanoyl-3,8-diazabicyclo[3.2.0]heptan-3-yl]acetamide N-[(1R)-4-oxo-5-[4-(3,4,5-trimethoxyphenyl)piperidine-1-carbonyl]cyclohexa-2,4-dien-1-yl]acetamide 2-[3-(4-cyanophenyl)-5-methoxyphenoxy]-N,N-diethylacetamide;ethane 3,5-dichlorobenzenethiol;N-(4,6-dimethylpyrimidin-2-yl)-1-phenylpropan-2-imine 1-[(2S,3S)-4-(cyclopentylamino)-3-hydroxy-1-phenylbutan-2-yl]pyrrolidine-2,5-dione 4-[(4-chlorophenyl)methyl]piperidine;ethane 3,5-dimethyl-4-[6-(trifluoromethoxy)-1,2,3,4-tetrahydronaphthalen-1-yl]aniline;2-(dipropylamino)acetaldehyde [2-amino-4,5-difluoro-6-(methylamino)-3-nitrosophenyl]methanol N-[2,4-dichloro-3-(4,6-difluoro-1H-benzimidazole-2-carbonyl)phenyl]-1-methylpyrazole-4-sulfonamide (2S)-1-[1-cyclohexa-1,5-dien-1-yl-3-phenyliminopropanoyl]pyrrolidine-2-carboxamide 7-[3-(4,5-dimethylcyclohexa-1,3-dien-1-yl)azetidine-1-carbonyl]-2-phenyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-one 1-[4-chloro-2,6-di(propan-2-yl)phenyl]-3-[5-ethoxypent-1-en-2-yl(methylsulfonyl)amino]urea 4-[[1-(2-methoxyethyl)pyrazol-3-yl]amino]-3,5,6,7,8,9-hexahydropyrimido[4,5-d]azepin-2-one 4-[5-(5-chloro-2,3-dihydrothiophen-2-yl)-1H-pyrazol-3-yl]-N-ethyl-N-[3-(2-methoxyethoxy)propyl]benzamide 1-(4-chlorophenyl)-3-[2-hydroxy-5-nitro-6-oxo-4-(trifluoromethyl)pyridin-1-yl]pyrrolidine-2,5-dione 1-[7-(3-aminophenoxy)naphthalen-2-yl]ethanone N-(4-hydroxyphenyl)-2,5-dimethoxybenzenecarbothioamide 3-(1,3-dioxoisoindol-2-yl)-4-hydroxybutanal N-[(6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl)methyl]-N'-ethyl-2-hydroxyethanimidamide (2-cyclopropylpyrimidin-5-yl)-[4-[6-methoxy-7-[3-(trifluoromethoxy)pyrrolidine-1-carbonyl]imidazo[1,2-a]pyridin-3-yl]-2-methylphenyl]methanone 6-[(5,7-dichloroquinoxalin-2-yl)amino]pyridine-3-carboxamide N-[(3R)-3-amino-5-cyclohexylpentanoyl]-1H-indole-2-carboxamide 5-[[6-[4-(dimethylamino)piperidin-1-yl]benzimidazol-2-ylidene]amino]-N'-hydroxythiophene-3-carboximidamide 5-(4,6-dibromopyridin-2-yl)-1H-pyrazole-3-carboxylic acid 5-amino-3-(2,4-dichlorophenyl)-N-propyl-6-[5-(pyrrolidine-1-carbonyl)pyridin-3-yl]pyrazine-2-carboxamide 1-azido-4,4-dimethyl-2-pentan-3-ylindeno[2,1-b]thiophen-9-one 1-[4-(2-aminopyrimidin-5-yl)phenyl]sulfonylpyrrolidine-3-carboxylic acid (4S)-1'-benzyl-6-chloro-2-fluoro-5,8-dimethoxyspiro[1H-quinoline-4,3'-indole]-2'-one N-[(2S)-4-amino-3,4-dioxo-1-phenylbutan-2-yl]-2-methyl-6-pyrimidin-5-ylpyrazole-3-carboxamide 4-(2,6-difluorophenyl)-6-(2-methoxyphenyl)-1H-pyrido[2,3-d]pyridazin-5-ium 2-(3-butoxyphenyl)-N,4-diphenyl-1,4,5,6-tetrahydropyrimidin-5-amine 2-amino-N-(3,5-difluorophenyl)-6H-pyrrolo[3,4-d]pyrimidine-7-carboxamide 1-(3,4-dimethylphenyl)-4-fluoropyrrolidine;1-(2,5-dimethoxyphenyl)piperidine [4-[[(3S)-1-azabicyclo[2.2.2]octan-3-yl]methoxy]phenyl]azanide 2-[4-amino-5-methoxy-3-methyl-2-(trifluoromethoxy)phenyl]propanoic acid 2-[4-(4-chlorophenyl)cyclohexyl]acetic acid (2E)-6-[3,5-bis(trifluoromethyl)phenyl]-N-[[4-(4-oxoquinazolin-1-yl)phenyl]methoxy]-2-prop-2-enylideneheptanamide N'-[3-(2,6-dichlorophenyl)-4-(hydroxymethyl)pyrazolo[3,4-d]pyrimidin-1-yl]benzenesulfonohydrazide 4-[[(2S)-1,5-dihydroxypentan-2-yl]amino]-3-(6-morpholin-4-ylpyridin-3-yl)-N-piperidin-4-ylbenzenesulfonamide 5-azidooxy-2,4-dichloropyrimidine 4-[2-(4-methoxyphenyl)ethynyl]benzaldehyde 3-azido-5-cyclopropylsulfonylpyridine (1S)-2-[4-[4-(3,5-dichloropyridin-4-yl)piperazine-1-carbonyl]-2-ethylpiperidin-1-yl]cyclopentan-1-ol N-[[5-(2-aminopyrimidin-4-yl)-7-fluoroimidazo[1,2-c]quinazolin-2-yl]methoxy]-2-pyridin-3-ylacetamide 3-[4-(2-bromophenyl)-1H-imidazol-5-yl]propanenitrile N-methyl-1-(4-propan-2-ylphenyl)sulfonylpiperidin-3-amine 5-[(2R,6S)-4-[4-chloro-3-(trifluoromethyl)phenyl]sulfonyl-2,6-diethylpiperazin-1-yl]-2-(oxan-4-ylamino)benzonitrile 7-[3-(4-methylphenyl)propoxy]-2,4,5,6-tetrahydro-1H-azepino[4,5-b]indole 5-cyclohexylsulfonylnaphthalene-2,3,7-triamine 1-[2-ethenyl-6-(3,4,5-trimethoxyphenyl)naphthalen-1-yl]-N-methylnaphthalene-2-carboxamide N-[(E)-3-(1H-indol-6-yl)prop-2-enoyl]formamide 1-(4,6-dimethoxypyrimidin-2-yl)pyrazole-3-carboxylic acid 1-methyl-2,3,5,6,7,8-hexahydro-s-indacene-4-carboxylic acid 4-[1-(2,4-dihydroxyphenyl)-3,5-dimethylpyrrol-2-yl]butanoic acid ethane;2-(1H-indol-6-yloxy)pyrimidine 4-(azidomethyl)-1,3-bis(2-fluorophenyl)-2H-benzimidazole (2R)-3-cyclohexyloxy-2-hydroxy-1-[4-[(5S,7S)-7-methyl-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-5-carbonyl]piperazin-1-yl]propan-1-one 5-N-[(1S)-3,4-dihydro-2H-chromen-7-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine (2R)-4,6-difluoro-1-[2-(3-hexyl-2-methoxyphenyl)ethynyl]-2,3-dihydro-1H-indene 3-[1-(2,4-dichlorophenyl)-7-hydroxyheptyl]sulfonylphenol N-[2,4-difluoro-3-(1H-pyrrolo[2,3-c]pyridine-2-carbonyl)phenyl]-2-phenylbenzenesulfonamide 2-[5-ethylsulfonyl-6-[8-oxo-1-(trifluoromethyl)-9H-pyrido[3,4-b]indol-3-yl]pyridin-3-yl]acetonitrile 3-[6-[3-(2,4-diaminopteridin-6-yl)oxypropoxy]pyridin-3-yl]benzaldehyde;methanamine 4-(1,2-dimethylimidazol-4-yl)-N,5-dimethoxypyridine-2-carboxamide N-[5-chloro-2-[3-(3,6-dihydro-2H-pyran-4-yl)-1H-indazol-5-yl]phenyl]acetamide (5S)-5-[4-fluoro-2-(1H-indazol-6-ylamino)pyrimidin-5-yl]-3-methylimidazolidine-2,4-dione (2E)-2-[(3Z,5Z)-hepta-1,3,5-trien-4-ylidene]-7-methyl-3H-inden-1-one (2R)-5-[3-cyclobutyl-4-(methanesulfonamido)phenyl]-N-(1H-indazol-6-ylmethyl)pyrrolidine-2-carboxamide 4-fluoro-6,7-dimethoxyquinoline 1-(1,3-benzodioxol-5-yl)-2-hydroxyisoquinolin-2-ium 2-cyclobutyl-4,5,6-triiodobenzene-1,3-dicarboxylic acid 2-[[2,5-dimethyl-1-(3-methylphenyl)pyrrole-3-carbonyl]amino]acetic acid 7-[5-[1-[(E)-2-phenylethenyl]piperidin-4-ylidene]pyrrol-3-yl]-5,6,8,9-tetrahydroimidazo[1,5-a]azepine N-[1-(3,5-dimethylphenyl)ethenyl]-2-propan-2-ylidene-3H-pyrrole-5-carboxamide 3,8-dinitrobenzo[f]chromene N-(2,3-dimethylphenyl)-3,3,4,5-tetradeuterio-1-[[4-(trifluoromethyl)phenyl]methyl]piperidine-4-carboxamide (4R,7S)-N-[3-(2,4-dichlorophenyl)propyl]-8-ethyl-1,6-dimethyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[4,3-c]azepine-4-carboxamide 3-(furan-2-yl)-N-[[4-methoxy-6-(pyrazol-1-ylmethyl)pyridin-2-yl]methyl]propanamide 2-[(4R)-6-amino-7-oxo-3,4-dihydrothieno[3,2-b]pyridin-2-yl]acetamide 2-[1-hydroxy-4-(1H-indol-6-yl)butan-2-ylidene]propanedinitrile 2-[(2E,5S)-2-[(Z)-furan-2-ylmethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]-N-phenylacetamide (5R)-3,4,7,8-tetramethyl-N-[2-(methylideneamino)ethyl]-5-naphthalen-1-yl-9-oxo-6,10-dihydropyridazino[1,2-a]indazole-2-carboxamide N-(2,3-dihydroindole-1-carbonyl)-N'-phenylmethanimidamide 2-chloro-1-(4-cyclopentylpiperazin-1-yl)ethanone;1-N',1-N'-dimethyl-1-N-[3-(3-phenylpropoxy)pyrazin-2-yl]ethene-1,1-diamine N-(4-anilinophenyl)-4,5-dimethylfuran-3-carboxamide N-[(4S,5R)-3,4-dihydroxy-1,6-dimethylpiperidin-2-yl]-2-fluorobenzamide;hydrochloride 1-(2-fluorophenyl)-5,7-dihydro-4H-pyrazolo[3,4-d]pyrimidine-6-thione (3R,4S)-1-[2-(6-methylpyridin-3-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid [(3aR,4R)-4-hydroxy-6-phenylmethoxyiminospiro[2,3,3a,4,5,7a-hexahydropyrrolo[2,3-c]pyridine-1,1'-cyclohexane]-5-yl]-pyridazin-3-ylmethanone 1-(1,3-dimethylpyrazol-4-yl)sulfonyl-2,3,6,7,8,9,10-heptahydropyridazino[4,5-b]azocine 2-[(1S,6R)-3-(5-methylimidazo[4,5-c]pyridine-7-carbonyl)-3,8-diazabicyclo[4.2.0]octan-8-yl]-N-[4-(trifluoromethyl)phenyl]acetamide (3E)-4,8-bis(benzenesulfonyl)-2-methyl-1H-1,5-benzodiazepine 1,5-dichloropyrene 4-(9,10-dihydroanthracen-1-yl)-6-(4-methoxyphenyl)sulfanyl-2-phenoxypyrimidine N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-5-(4-fluorophenyl)-6-oxo-1H-pyridazine-3-carboxamide N-[4,5-bis(ethenyl)thiophen-2-yl]acetamide 2-ethyl-1,3-dimethylpyrrolo[3,4-c]pyridine;propane N-(2,3-dihydro-1H-inden-5-yl)-2-[(2E)-2-[(4-methoxyphenyl)methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetamide N-[(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-3-naphthalen-1-yloxypropanamide N-[1-(2-methoxyethyl)piperidin-4-yl]-5-propan-2-ylfuran-3-carboxamide 4-tert-butyl-1,5,6-trimethoxyisoquinoline (1S,2R)-3-(butyliminomethyl)-N'-hydrazinylidene-1-phenylpropane-1,3-diamine 2-methyl-1,3-bis[2-(4-sulfanylidenecyclohexa-2,5-dien-1-yl)phenyl]propane-1,2-dione 6-methyl-4a-(3,3,5-trimethoxyphenyl)-1,2-dihydroquinoline 2-(4-methylpyrazol-1-yl)-7,8-dihydro-5H-1,6-naphthyridine;trihydrochloride 5-tert-butyl-2,3-bis(4-chlorophenyl)pyrazine [6-hydroxy-3-(1-phenylethyl)-2H-indazole-5-carbonyl]oxidanium 2-[5-(6-azaspiro[3.4]octan-7-yl)pyridine-2-carbonyl]-1,3-dihydroisoindole-5-carboxylic acid (3,5-dimethoxyphenyl)-(5-methyl-2,6-diazaspiro[3.4]octan-2-yl)methanone (2R,3S)-2,5-diamino-N'-[2-amino-4-(cyclopropylmethoxy)phenyl]pentanimidamide [5-hydroxy-3-(4-nitrophenyl)sulfonylpentyl]carbamic acid 4-[(2Z,5R)-2-[[1-(cyclohexylmethoxymethyl)cyclopentyl]methylidene]-3-oxo-1H-pyridin-6-yl]benzonitrile 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-propylamino]benzenesulfonic acid 2-[[6-(4-bromophenyl)-5-ethoxycarbonylpyridin-3-yl]methylcarbamoylamino]pentanedioic acid 4-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]quinolin-8-ol;propane 3-[(2R)-1-ethenylsulfonylpyrrolidin-2-yl]-5-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridine 4-ethyl-2,3-difluoro-N-methylaniline;1-[4-(3-ethynylazetidin-1-yl)cyclohexa-1,5-dien-1-yl]-N-phenylsulfanylmethanamine 1,2-bis(5-pyridin-3-ylthiophen-2-yl)imidazole;dioxidoazanium N-[2-amino-5-(1,3-dioxol-4-yl)phenyl]-6-[3-[(dimethylamino)methyl]piperidine-1-carbonyl]pyridine-3-carboxamide;cyclohexane N-(1,3-benzothiazol-5-yl)-4-[[6-(2-fluorophenoxy)pyridine-3-carbonyl]amino]piperidine-1-carboxamide 4-amino-2,6-dichloro-N-[(2R)-1-hydroxybutan-2-yl]benzamide 3-[4,7-bis(2,6-dimethylphenyl)-1,5-diazocane-1-carbonyl]benzoic acid N-[3-(3,4-dihydropyridin-2-yl)phenyl]-N'-methanimidoylpropane-1,3-diamine 4-[2-(4-oxopiperidin-1-yl)ethyl]benzamide 1-(3,5-dimethoxyphenyl)-4-[2-(hydroxyiminomethyl)pyridin-1-ium-1-yl]butan-2-one 5-amino-3-[2,4-dichloro-5-(1,1,2,2,2-pentafluoroethyl)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile ethane;1-(6-methoxy-5-pyridin-4-ylpyrazin-2-yl)azepan-4-amine 4-[5-(3,5-dichlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-2-yl]pyridine (2E,3Z)-2-[1-(5-carboxypyridine-2-carbonyl)piperidin-4-ylidene]-3-ethylidenehepta-4,6-dienoic acid 5-cyclopropyl-1'-[2-(3,4-dichlorophenyl)acetyl]spiro[6H-pyrazolo[4,3-c]pyridine-7,4'-piperidine]-4-one 2-[(3E)-2,6-dimethylhepta-1,3,5-trien-4-yl]-7-ethyl-5-methyl-1H-indole;hexane 6,7-dichloro-5-hydroxy-1H-quinazoline-2,4-dione 2-(6,11-dihydrobenzo[c][1]benzoxepin-4-ylamino)ethanol N-methyl-4,6-diphenyl-2H-azepin-7-imine ethane;N-[3-(4,5,7-trimethyl-1H-benzimidazol-2-yl)propyl]acetamide N-[(2S)-1-[(6-chloronaphthalen-2-yl)sulfonylamino]-3-cyclohexylpropan-2-yl]isoquinoline-7-sulfonamide N-(3-bromophenyl)-2,5-dimethoxy-6H-pyrimidin-4-amine 4-(aminomethyl)-6-[3-(2,5-difluorophenyl)-1,2-oxazol-5-yl]-2H-phthalazin-1-one 1-[4-(3,5-difluorophenoxy)phenyl]propane-2-sulfonate (2S,3R)-N-[4-(4-hydroxypiperidine-1-carbonyl)phenyl]oxolane-2-carboxamide 6-[(1S)-2,3-dihydro-1H-inden-1-yl]-1-methyl-4-pyrimidin-5-ylpyrrolo[3,2-c]pyridine 4-(2,3,5-trichlorophenyl)triazolo[1,5-a]pyridine 1-[4-(azidomethyl)-3-fluorophenyl]pyrrolidine 2-[(3R,4S)-3-fluoro-1-(pyrimidin-2-ylmethyl)piperidin-4-yl]oxyethanol;hydrochloride (2S)-5-[3,5-dichloro-2-hydroxy-4-(trifluoromethoxy)phenoxy]-1-phenylpentan-2-amine 1-[2-(2,4-dimethoxyphenyl)ethylamino]-3-(4-hydroxybutan-2-yl)thiourea 3-(2,4-difluorophenyl)-N'-hydroxy-5-oxo-8H-[1,2]thiazolo[5,4-b]quinoline-7-carboximidamide N-(1,3-benzothiazol-2-yl)-6-(4-hydroxyphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-2-carboxamide 5-(trifluoromethyl)-1-benzothiophene-3-carboxamide 2-[(6S)-8,10-dimethoxy-1,4-dioxa-7-azaspiro[4.5]decan-7-yl]benzoic acid 1-ethoxycarbonylnaphthalene-2,3,4-tricarboxylic acid N-[4-[2-(dimethylamino)ethyl]-5,6,7,8-tetrahydronaphthalen-1-yl]-3-nitrobenzenesulfonamide 4-(4-ethylphenyl)sulfonylcyclohexan-1-ol N-[(2S,3R)-1,1-dioxothiolan-3-yl]-4-hydroxy-3-methoxybenzamide 6-[(2,4-dimethylphenyl)sulfanylamino]-N-hydroxy-3-methoxy-5-propan-2-ylpyridazine-4-carboxamide 2-(6-phenylhexylamino)benzoic acid 2,6-dichloro-5-hydroxy-4-[(4R)-2-methyl-7,7-diphenylocta-1,3-dien-4-yl]benzenesulfonic acid N-benzyl-5-[2,3-dichloro-4-(cyclobutylamino)phenyl]pentanamide 4-[1-azido-2,3-dimethyl-3-(trifluoromethyl)pentan-2-yl]-N,N-diethylaniline 6-bromo-N-[2,4-dichloro-3-(cyclobutylmethoxy)phenyl]pyrimidine-4-carboxamide (1Z,3E)-2-[[4-[4-chloro-3-(trifluoromethyl)phenyl]piperazin-1-yl]sulfonylamino]penta-1,3-diene-1-sulfonic acid 5-methylsulfanylimidazo[1,2-c]pyrimidine;5-methylheptanenitrile 3-methyl-2-[4-(4,5,6-tricyclohexylpyrimidin-2-yl)phenyl]pyrazine [(2S,4R)-1-benzylsulfonyl-3,4-dimethoxypyrrolidine-2-carbonyl]azanium N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-4-[6-(4-fluorophenyl)pyridazin-3-yl]piperazine-1-carboxamide 4-[2-(2,6-dimethylphenyl)-5-(4-fluorophenyl)pyrido[2,3-d]pyrimidin-8-yl]benzenethiol (E)-1-[(6S,8R)-7,8-dichloro-2-cyclopropyl-3-(4-methoxyphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-N'-methylethene-1,2-diamine 4-(1,3-benzodioxol-5-yl)-2-(1-hydroxyethylamino)pyridine-3,5-dicarbonitrile 1-[4-(cyclopropylmethoxy)phenyl]-2,2,3-trifluoropropan-1-ol N-(2,3-dihydropyridin-5-ylmethyl)-3-methoxyaniline 1-(2,5-dimethylphenyl)-7-methoxy-3,5-dihydro-1H-imidazo[1,2-a]quinazoline-2,4-dione 1-[5-(azidomethyl)thiophen-3-yl]sulfonyl-2,4-dichlorobenzene N-[2,4-dimethyl-5-(2-phenylpropanoyl)phenyl]benzamide 2-[(2E)-2-[[4-[(3,5-dimethylphenyl)methoxy]-3-iodo-5-methoxyphenyl]methylidene]hydrazinyl]benzoic acid (NE)-N-[5-[2-[3,4-dimethoxy-5-(2-phenylethynyl)anilino]pyridin-3-yl]-1H-pyrimidin-2-ylidene]hydroxylamine 6-[3,5-bis(trifluoromethyl)phenyl]-N-(2,5-diethoxyphenyl)benzo[b][1,4]benzoxazepine-9-carboxamide 1-[2-(dimethylamino)ethyl]-4-(4,5-dihydro-3H-cyclopenta[c]pyrazol-2-ylmethoxymethyl)-5,6,7,8-tetrahydronaphthalen-2-ol 4-[(2Z)-3,7-dimethylocta-2,6-dienoxy]-7-hydroxychromen-2-one 2-[(5R)-2-[3,4-bis(difluoromethoxy)phenyl]imino-4-oxo-1,3-thiazolidin-5-yl]acetic acid 2-(diethylamino)-1,3,10,12-tetrazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13),11-pentaen-9-one N-[(3S,4S)-1-benzyl-4-cyanopyrrolidin-3-yl]-4-(2-methoxyethoxy)pyridine-2-carboxamide 3-[(2,4-difluorophenyl)sulfonylmethyl]-5-[4-(1-hydroxycyclopropanecarbonyl)piperazin-1-yl]-1,6-dihydropyrazolo[4,3-d]pyrimidin-7-one 3-[[6-(3-chlorophenyl)pyridazin-4-yl]amino]benzenesulfonamide 3-amino-4,5-dimethylbenzaldehyde;N-[2-(cyclopropylmethoxy)-7a-methyl-1,7-dihydroindole-6-carboximidoyl]-1-phenylmethanamine (2S)-3-[5-amino-6-[(E,4R)-4-methyloct-1-enyl]pyridin-2-yl]oxypropane-1,2-diol N-[(3S,4R)-1-cyclopropyl-2-oxo-4-phenylpyrrolidin-3-yl]-7-methoxyquinoline-6-carboxamide N-(3,4,5-trifluorophenyl)sulfonylacetamide N-ethylsulfanyl-1-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methanamine 4-(3,5-dimethoxyphenyl)-6-pyridin-2-yl-1H-pyrimidine-2-thione 3-[(2,4-diaminopteridin-6-yl)methylamino]-5,8-difluoro-7-methoxyquinazolin-4-one (3E,5Z)-6-amino-1-[4-fluoro-2-[3-methylbutyl(propanoyl)amino]phenyl]-3-hydroxyhepta-3,5-dien-2-one 2-(ethylsulfanylamino)-4-methylpyridine-3,5-dicarboxylic acid 3-[(2Z)-2-[1-[3-(dimethylamino)propyl]pyrazol-4-yl]oxyiminobutanoyl]-N,4-dimethyl-5-oxopiperazine-1-carboxamide (1R,2R)-N-[[(5S)-3-(cyclopropylmethyl)-5-[(2-ethoxy-6-oxo-1H-pyridine-4-carbonyl)amino]piperidin-1-yl]methyl]-2-phenylcyclopropane-1-carboxamide 3-bromo-2,7a-dimethyl-5-naphthalen-1-yl-4aH-[1,3]thiazolo[5,4-b]pyridine (1S)-4-bromo-2,7-dimethyl-9-(4-methylphenyl)sulfanylfluorene 2-[4-[[1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]amino]piperidin-1-yl]quinoline-8-carboxylic acid;dihydrochloride [4-[1-hydroxy-3-(trifluoromethyl)propyl]phenyl]boronic acid (4-bromo-3-methoxypyridin-2-yl)hydrazine N-[5-[3,5-bis(ethenyl)pyrazol-1-yl]pyridin-2-yl]-2-methoxyacetamide 1-(5,5-dimethyl-3H-1,2,4-oxadiazol-2-yl)naphthalene-2,7-disulfonic acid 2-(1,1-difluoroethyl)-4-[3-[(2-fluorophenyl)methoxy]piperidin-1-yl]pyrimidine [(4R,6S)-6-ethoxycarbonyl-5-hydroxy-2-phenyl-1,3-dioxan-2-yl]oxidanium (E)-3,4-dimethyl-N-[3-methyl-1-[3-(1H-pyrrol-2-yl)phenyl]butyl]pent-2-enamide;ethane 2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-4H-pyrazolo[1,5-a]quinazolin-5-one 2-[4-(6,8-dimethoxyquinazolin-4-yl)oxyphenyl]acetaldehyde;N-methyl-1-piperidin-3-ylethanamine 6-chloro-7-[(2R)-4-[3-(4-chlorophenyl)propanoyl]-2,5-dimethylpiperazin-1-yl]-1-cyclopropyl-8-fluoro-4-oxoquinoline-3-carboxylic acid 4-chloro-2,6-dimethyl-7H-[1]benzothiolo[3,2-d]pyrimidine ethane;4-[7-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]pyrimidine N-(2,6-dimethylphenyl)-4-(1H-imidazol-5-yl)butanamide;hydrochloride N-[(2S)-1-hydroxy-4-methylpentan-2-yl]oxy-3,5-dimethylbenzamide N-[1-(2-fluorophenyl)ethyl]-3-propan-2-ylidene-1,2-dihydroinden-5-amine 5-chloro-3,3-diethyl-2H-indole 5-[3-[(2S,4R)-5-azido-4-methylpentan-2-yl]phenyl]-N-methoxypyridine-2-carboxamide (4-azido-3,5-dimethylpyridin-2-yl)-[5-fluoro-6-hydroxy-1-(oxetan-2-ylmethyl)indol-3-yl]methanone N-butyl-4-methoxy-3,5-dimethylaniline N-[4-amino-3-(1,2-oxazole-5-carboximidoyl)phenyl]-5-cyano-3-methoxypyridine-2-carboxamide 2-[[4-(3-ethoxyphenyl)-6-oxo-1H-pyrimidin-2-yl]sulfanyl]acetic acid 7-(4-chlorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine N-[[3-(4,6-dimethoxy-1H-indole-2-carbonyl)phenyl]methyl]-5-oxopyrrolidine-3-carboxamide 4-[(5S)-3-benzyl-7-(ethoxymethyl)-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,7,9,11-pentaen-12-yl]phenol 1-(2,5-dimethylcyclohexa-2,4-dien-1-ylidene)-3-phenylpropan-2-one 3-(6-chloropyridin-2-yl)sulfanyl-5,7-dimethoxy-1H-indole 1-[4-[2-(5,7-dimethoxyquinolin-6-yl)ethynyl]piperidin-1-yl]-2-[3-methanimidoyl-1-(oxetan-3-yl)azetidin-3-yl]oxyethanone 1-[(2R,4S)-4-fluoro-5-hydroxy-2-methylpiperidin-1-yl]-3-quinolin-8-ylsulfonylpropan-1-one 5-chloro-2-fluoro-4-[1-(3-hydroxyphenyl)cyclopentyl]oxybenzoic acid 3-(1,4-dihydropyrido[2,3-d]pyrimidine-7-carbonyl)-5H-pyrrolo[3,4-b]pyrazin-6-one N-[2-(4,5-dihydrobenzo[g][1]benzazepine-9-carbonylamino)phenyl]formamide (2Z)-N-[3-(3,4-dichlorophenyl)sulfanylbutyl]-N-ethyl-2-(oxolan-1-ium-2-ylidene)acetamide 2-[4-hydroxy-N-(3-methylbut-2-enyl)anilino]propanoic acid 2-(2,3-dihydroindol-1-yl)-N'-hydrazinylidenepyrimidine-4-carboximidamide 5-(3,5-dimethylimidazol-4-yl)-3-[4-[4-fluoro-2-(trifluoromethyl)phenoxy]phenyl]-1H-indole N-[3,5-bis(trifluoromethyl)phenyl]-1-cyclopropylidenesulfanylpiperidine-4-carboxamide 4-amino-6-(cyclohexylmethylsulfanyl)-3-ethyl-1H-pyrimidin-2-one N-[2,4-difluoro-3-(2-methoxypyridine-3-carbonyl)phenyl]propane-1-sulfinamide (E)-2-[4-ethoxy-5-methoxy-6-[(3,4,5-trimethoxyphenyl)methyl]pyrimidin-2-yl]ethenol 6-(2,4-diaminopteridin-6-yl)hexanenitrile 2-[[1-[4-(3-chlorophenyl)piperazine-1-carbonyl]cyclobutyl]methoxy]-6,7-dihydroquinoline-5,8-dione 2-(4,6-dimethylpyrimidin-2-yl)sulfanylbenzene-1,3-dicarboxamide 4-[(4-aminophenyl)diazenyl]naphthalen-1-ol (2R)-3-[5-(4-hydroxyphenyl)pentoxy]propane-1,2-diol 3-(4-chlorophenyl)-1-ethyl-6,8-difluoro-7H-quinoline-2,5-dione 2-[5-(1H-benzimidazol-2-ylsulfanyl)furan-3-carbonyl]-4-benzamidopentanoic acid N-[3,5-bis(trifluoromethyl)phenyl]-2,4,6-trichloro-N'-methylcyclohexa-1,3-diene-1-carboximidamide 4-[2-(6,7-difluoroquinoxalin-2-yl)oxycyclopentyl]-1,3-oxazolidine 2-(4-azidophenoxy)-1,3,5-trichlorobenzene 1-[4-[[5-fluoro-2-methoxyethyl(3,3,3-trifluoropropyl)amino]methyl]phenyl]-N'-methanimidoyl-3-pyridin-3-ylimidazole-1,2-diium-5-carboximidamide 2-chloro-4-(4,6-dihydro-1H-pyridazin-5-yl)aniline N-[(4,6-dimethylpyridin-3-yl)methoxy]benzamide;hydrochloride [1-[(2S)-3,3-dimethylbutan-2-yl]-2H-pyridin-4-yl]-(6-phenylpyrazin-2-yl)methanone N-[1,3-bis(4-aminophenyl)butan-2-yl]propanamide (2S)-1-(4-bromophenyl)sulfanylpyrrolidine-2,5-dicarboxylic acid 3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dihydroxyisoindol-4-yl]-3-phenylmethoxypropanamide 4-[1-(cyclohexen-1-yl)pentan-3-yl]aniline 6-[[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl]-3H-quinazolin-4-one (5R)-1'-[2-chloro-6-fluoro-3-(propanoylamino)benzoyl]-N,N-dimethylspiro[7,8-dihydro-5H-naphthalene-6,4'-piperidine]-2-carboxamide 7-amino-5,6-bis(4-methylphenyl)pyrrolo[2,3-d]pyrimidine-2,4-diamine 2-[4-[3,5-diamino-6-(4-fluorophenyl)pyrazine-2-carbonyl]piperazin-1-yl]-N'-hydroxyethanimidamide 5-cyclohexa-2,4-dien-1-ylfuran-3-carbonitrile (3E)-5,6-dimethyl-N'-[2-(4-methylpiperazin-1-yl)ethyl]-4-oxo-3-propylidenequinazoline-8-carbohydrazide 3-[(3R)-1-(cyclobutanecarbonyl)pyrrolidin-3-yl]-2H-pyrazolo[4,3-d]pyrimidine-7-carboxamide 1-(1,3-benzodioxol-5-ylmethyl)-4-chloro-2-(1H-indol-2-ylsulfinylamino)pyrrole-3-carboxylic acid N-[5-chloro-2,4-difluoro-3-(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)phenyl]propane-1-sulfonamide 2-azido-5,8-dichloroquinoline (5Z)-2-imino-5-[[4-methoxy-3-(quinolin-6-ylmethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one N-[(E)-4,5-difluorohept-3-enyl]-1-ethylindole-2-carboxamide 2-(3-phenylphenyl)propanedinitrile 4-[6-[(E)-1-methyliminobut-2-en-2-yl]quinoline-3-carboximidoyl]phenol 4-(cyclohexylamino)-6-(3,5-dimethylanilino)pyridine-2-carboxylic acid ethane;2-ethoxy-4-(4-fluorophenyl)-N,6-dimethylthieno[3,2-d]pyrimidine-7-carboxamide N-(diethoxyphosphorylmethylidene)-2,6-dimethoxybenzamide 5-chloro-3-[4-(1H-indol-2-yl)phenyl]-N,N-dimethylpentan-1-amine 5-methyl-N-[(2-piperidin-1-ylpyridin-4-yl)methyl]-3,4-dihydronaphthalene-1-carboxamide 5-(4-methylphenyl)-N'-[[4-(trifluoromethoxy)phenyl]sulfonylamino]furan-2-carboximidamide 2-N,3-bis(3,5-diethyl-4-hydroxyphenyl)benzene-1,2,3,4,6-pentol 2-[4-(4,4-dimethylcyclohexen-1-yl)phenyl]ethanol 1-(2-cyclopropylpyrrolidin-1-yl)-2-[4-methoxy-3-(5,7,8,10,11-pentazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,9,11-hexaen-12-ylmethoxy)phenyl]ethanone N-[2,6-difluoro-4-(1-methylpyrazol-3-yl)phenyl]spiro[5H-tetrazole-7,4'-pyrrolo[1,2-a]quinoxaline]-8'-carboxamide 5-chloro-4-fluoro-6-[2-(3-iodopyrazolo[1,5-a]pyridin-2-yl)ethoxy]benzene-1,3-diol 3-(1H-indole-2-carbonyl)-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-1-carboxylic acid 7-[(6-chloropyridin-3-yl)methoxy]quinoline N-ethyl-2-[1'-(pyridine-3-carbonyl)spiro[4,7-dihydrotriazolo[5,1-c][1,4]oxazine-6,3'-pyrrolidine]-3-yl]acetamide 2,7-bis(2H-tetrazol-5-yl)-1,3-benzothiazole 2-(N-(4-bromo-2,5-dimethylphenyl)-3-nitroanilino)octanoic acid 1-[2,5-bis(trifluoromethyl)phenyl]-3-diazourea 4-bromo-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine 3-methyl-N-[(1S)-2-phenylcyclopropyl]-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carboxamide N-[[(5S)-3,4-dimethyl-1,2-oxazol-5-yl]methyl]-1-(5-fluoropyrimidin-2-yl)piperidine-4-carboxamide [4-[(E)-2-(1,3-benzothiazol-6-yloxymethyl)-3-fluoroprop-2-enoxy]phenyl]phosphane 4-(5-chloropyridin-3-yl)oxy-2,7-dimethyloctanal 4-[3-[[2,2-difluoro-2-(1-hydroxypyridin-1-ium-2-yl)ethyl]amino]-6-methoxypyridazin-4-yl]-N'-hydroxybenzenecarboximidamide N-(5,6-dimethylpyridin-2-yl)-1,3-thiazolidine-4-carboxamide N-cyclohexyl-2,3-bis[4-(trifluoromethoxy)phenyl]propanamide (2S,5R)-N-[(Z)-(4-hydroxy-3-iodophenyl)methylideneamino]-2,6-dioxopiperidine-1-carboxamide 2,6-bis[(Z)-1,3-dioxobutan-2-ylideneamino]-4-ethenylbenzenesulfonate N-butylformamide;3,4,5-trihydroxy-6-[2-[4-(2-piperidin-1-ylethoxy)phenyl]ethenyl]oxane-2-carboxylic acid (5R,7S)-5-[4-chloro-3-(trifluoromethyl)phenyl]-N-(1-hydroxypropan-2-yl)-7-(trifluoromethoxy)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide 2-[2,4-dichloro-N-(2-oxopropyl)anilino]acetamide 1-[3,5-bis(trifluoromethyl)phenyl]pyrrole 4-methoxycarbonyl-2,5-diphenoxybenzoate 2-[3-[(E)-1-methylsulfonylprop-1-enyl]phenyl]pyridine 2-(3,4-difluorophenyl)-5-methyl-6-[2-(1-propan-2-ylpiperidin-2-yl)ethoxy]-1H-pyrrolo[3,2-b]pyridine 4-methylsulfanyl-1-(2-propan-2-ylphenyl)piperazine N-(3,5-dichlorophenyl)-2-[7-(4-methoxyphenyl)-6-methyl-2-oxo-1,3-dihydroimidazo[1,2-b]pyrazol-3-yl]acetamide N-cyclohexyl-4,7-dimethoxy-2-[(Z)-prop-1-enyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-5-amine N-cyclopentyl-1,5-dimethylpyrazole-3-sulfonamide N-[5-(2,3-dichlorophenoxy)-1H-indazol-3-yl]-4-methoxybenzamide 3,4-dimethoxy-1-(2-phenylimidazo[5,1-b][1,3]thiazol-3-yl)butan-2-one [4-(1-benzylpyrazole-3-carbonyl)piperazin-1-yl]-(6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-ylmethylamino)methanol 5-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)indole 4-[N-(2,3-dihydroxypropyl)-4-methoxyanilino]butan-1-ol 1-[5-(4-chlorophenyl)-1H-pyrazole-3-carbonyl]piperidine-2-carboxylic acid 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]decanoic acid N-[1-(2-chlorophenyl)ethyl]pentan-3-amine 2,4-dichloro-3-iodothieno[3,4-b]pyrazine N-azido-2,6-dimethyl-3-nitrobenzenesulfonamide 2-(4,6-dioxocyclopenta[d][1]benzoxepine-3-carbonyl)oxyethylphosphonic acid 3-[(4-aminophenyl)methyl]hexanoic acid N-[2-(4,5-diphenyl-1H-imidazol-2-yl)cyclohexa-2,4-dien-1-ylidene]hydroxylamine 6-[5,7-difluoro-2-(4-fluorophenyl)-1H-indole-3-carbonyl]-N-propylpiperidine-3-carboxamide 1-[4-(4-butylcyclohexyl)phenyl]-2,3-difluoro-4-(trifluoromethoxy)benzene 1-[2,6-di(propan-2-yl)phenyl]-3-methoxy-7-(trifluoromethoxy)indazole N-[4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]oxyphenyl]prop-2-ynamide 2-[4-(azidomethyl)cyclohexyl]oxy-1,3,5-triazine 3-(7-cyanoimidazo[1,2-a]pyridin-5-yl)sulfanylbenzenesulfonamide (2S,3R)-1-azido-N'-[4-bromo-5-methyl-3-(trifluoromethyl)pyrazol-1-yl]-3-hydroxypiperidine-2-carboximidamide ethane;methoxymethane;1-[4-[2-(4-phenylbut-3-ynyl)-1H-indol-5-yl]piperidin-1-yl]propan-2-one N'-(5-methylisoquinolin-8-yl)methanimidamide 4-methyl-6,12-dithiatetracyclo[9.7.0.03,8.013,17]octadeca-1(11),3(8),4,6,9,14,16-heptaene 3-(2-fluorophenoxy)-1-[3-(4-methylphenoxy)azetidin-1-yl]propan-1-one [(2Z,4E)-5-[3-[(E)-(ethylideneamino)diazenyl]phenyl]penta-2,4-dienoyl]oxymethanesulfonate 2-[[1-(methylamino)isoquinoline-3-carbonyl]amino]acetic acid 2-[(Z)-5-chloro-4-methylimino-3,3a-dihydroimidazo[1,2-a]pyridin-7-ylidene]propanedinitrile 5-[6-(2,4-dichlorophenoxy)-8-methylsulfanylimidazo[1,2-a]pyridine-3-carbonyl]-1H-pyridin-2-one [2-(2,4-difluorophenyl)morpholin-4-yl]-[1-(pyridine-3-carbonyl)piperidin-3-yl]methanone 2-[2-[(4-chlorophenoxy)methyl]-1,3-thiazol-5-yl]acetamide 4-[3,6-bis(methylsulfanyl)-1-phenyl-2H-benzimidazole-5-carbonyl]piperazin-2-one (1R,2S)-N'-[5-chloro-4-[(4-fluorophenyl)methyl]-2,3-dihydropyrido[3,2-b][1,4]oxazepin-7-yl]-2-hydroxycyclopropane-1-carboximidamide;dihydrochloride 5-chloro-1-(4,6-dimethoxypyrimidin-2-yl)indole 1-[(2R,4S)-5-methyl-3,4-dihydro-2H-chromen-2-yl]ethanone 1-azidooxy-5,7-dihydroxy-2,8-bis(4-methylphenyl)octan-3-one N'-[5,6-dimethoxy-2-(4-phenylpyridin-3-yl)sulfanylpyrimidin-4-yl]-N-(4-fluorophenyl)ethane-1,2-diamine 1-[[4-[1-(dimethylamino)ethenyl]phenyl]methyl]cyclopentan-1-ol 1-(4-fluorophenyl)-6,8-dimethoxy-2H-quinoline 4-[8-amino-3-[(1R)-1-(5-chloro-6H-cyclohepta[d]pyrimidine-2-carbonyl)-3,4-dihydro-1H-isoquinolin-2-yl]imidazo[1,5-a]pyrazin-1-yl]-N'-[2-(dimethylamino)ethyl]benzohydrazide 2-(4-chloro-3,5-difluorophenyl)-N'-hydroxy-2-[1-(3-pyrrolidin-1-ylpropylsulfonyl)piperidin-3-yl]ethanimidamide [1-azido-5-(2,6-dichlorophenyl)penta-2,4-dienyl]benzene 6,7-dimethoxy-3-phenyl-2H-quinazoline 5-amino-2-(3-hydroxyphenyl)-7H-pyrrolo[2,3-b]pyrazine-6-carboxamide 4-(2,4-dichlorophenyl)-1H-pyrimidine-2,4-diamine 3-[(5R,7S)-5,7-dimethyl-1,4-oxazepane-6-carbonyl]pyridine-2-carbonitrile 1-[5-chloro-3,4-bis(ethenyl)pyridin-2-yl]ethenol;[4-ethenyl-3-(methylideneamino)phenyl]-pyrrolidin-1-ylmethanone 2-(4-hydroxybutyl)-N,N'-bis[(Z)-1H-indol-3-ylmethylideneamino]octanediamide 4-(2-hydroxyphenyl)-1,7-dihydropyrazolo[3,4-b]pyridin-6-one N-[(E)-3-(furan-2-yl)propylideneamino]formamide N-[(1S,2R)-1-[4-[benzyl(tert-butyl)amino]phenyl]-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]oxynaphthalene-2-sulfonamide 1-[(E)-3,4-dimethylpent-2-enyl]-9H-fluorene;(Z,2Z)-2-ethylidene-5-fluorooct-6-enal 2-methyl-3-[(2R)-1-phenylbutan-2-yl]oxypropanoic acid 4-azidooxy-5,6-diphenyltriazine 1-(3,5-dichloropyridin-4-yl)-N'-hydroxyimidazole-2-carboximidamide 3-(4,6-dimethoxypyrimidin-2-yl)-2-[(3Z)-penta-1,3-dien-2-ylamino]benzoic acid N-(2-chloro-6-fluorophenyl)-3-methyl-4-[2-oxo-2-(pyridin-3-ylamino)acetyl]piperazine-1-carboxamide N-[5,7-dichloro-2-(2-hydroxyacetyl)imidazo[1,2-a]pyridin-6-yl]-4-methoxybenzamide 2-methyl-3,4-bis(methylsulfanyl)-5-phenylbutanal 2-[4-(2,2-dimethylmorpholin-4-yl)sulfonylanilino]-6-methanimidoylbenzenecarboximidamide 1-(3,4-diethoxyphenyl)piperazine;2,2,2-trifluoroacetic acid 4-(2,3-dimethyl-3H-pyrazol-1-yl)-6-fluoropyridine-3-carbonitrile 1-[(2,3-dimethoxyphenyl)methylamino]-3-(1-ethylsulfonylpiperidin-4-yl)urea (3S)-N'-[2-[N-[(4-chlorophenyl)methyl]anilino]ethyl]pyrrolidine-1,3-dicarboximidamide (2R)-2-[3-[5-chloro-6-fluoro-1-(4-fluorophenyl)sulfonylindol-3-yl]propanoylamino]-N-hydroxy-4-methylpentanamide 4-[2-(2,3-dimethylbutanoyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl]piperazine-2-carboxamide N-azido-4,5-bis(ethenyl)pyridin-2-amine N-[[2,4-dichloro-3-[[6-cyano-5-(trifluoromethyl)pyridin-3-yl]carbamoylamino]phenyl]methyl]-N-ethoxy-4-(4-methylpiperidine-1-carbonyl)cyclohexane-1-carboxamide 5-fluoro-2-(5,6,7,8-tetrahydroisoquinolin-1-yl)-3H-quinazolin-4-one 4-[4-[3,5-difluoro-6-(2-methyl-1H-pyrazol-2-ium-4-yl)pyridin-2-yl]-3,6-dihydro-2H-pyridine-1-carbonyl]benzoic acid 1-phenylmethoxy-5-propylsulfonylindole 2-bromo-N-[(Z)-1H-indol-3-ylmethylideneamino]benzamide 5-[3-(2,2,2-trifluoroethoxy)phenyl]pentanoate (E)-3-[4-[(5-chlorothiophene-2-carbonyl)amino]phenyl]prop-2-enoic acid 2-[4-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]phenyl]sulfonylethanol 2-[[4-(trifluoromethyl)phenyl]methoxymethyl]-5,6,7,8-tetrahydroquinoline 7-methyl-2,4-dioxochromene-3-carboxylic acid N'-[amino(2,3-dimethoxypropyl)amino]-5-bromo-1H-pyrrolo[2,3-b]pyridine-3-carboximidamide N'-[(Z)-3-aminoprop-2-enimidoyl]-3-[6-methoxy-4-morpholin-4-yl-7-(piperidine-1-carbonyl)quinazolin-2-yl]benzenecarboximidamide [5-(6,7-dihydro-1H-indole-2-carbonyl)-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-3-yl]-pyrrolidin-1-ylmethanone 3-(2,6-dichlorophenyl)-7-[4-(3-hydroxypropyl)piperazine-1-carbonyl]-2H-isoquinolin-1-one 2-N-[2-(1,3-dimethylpyrazol-4-yl)-6-methoxypyridin-4-yl]-5-ethanimidoylpyrimidine-2,4-diamine N-[4-(1,3-benzothiazol-2-ylsulfanylmethyl)pyridin-2-yl]acetamide 5-chloro-N-(3,3-difluorocyclobutyl)-1H-indazole-6-carboxamide N-[(1R)-4,5,6-trimethoxy-2-methyl-3-oxo-7-phenylmethoxy-1H-isoindol-1-yl]acetamide 2-[4-(1,1-dioxothiolan-3-yl)piperazine-1-carbonyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one 2-[5-ethenyl-3-(methylamino)pyridin-4-yl]-1,5,6,7-tetrahydrocyclohepta[f]benzimidazol-4-one 4-[4-[2-(1H-indazol-5-ylamino)pyrimidin-4-yl]pyrazol-1-yl]cyclohexane-1-carbonitrile 2-amino-N-[1-(3-cyclobutyl-4,5-dimethoxyphenyl)ethenyl]benzenecarboximidate N-[1-[4-(2,5-dimethoxyphenyl)piperazine-1-carbonyl]pyrazol-3-yl]cyclopropanecarboxamide 2-(3,5-dichlorophenyl)-4-methylsulfanylbutanoic acid 3-[6-(azidomethyl)pyridin-2-yl]quinoline (7S)-2-[4-(3-fluoroazetidin-1-yl)anilino]-N,N,5,7-tetramethyl-8-oxopteridine-6-carboxamide 2-[(1R)-1-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-6-yl)ethyl]isoindole 5-(7H-cyclopenta[b]pyridin-3-yl)pyrazine-2-carboxylic acid (2R,3S)-2-[5-(2,6-dimethoxyphenyl)-1-(oxan-4-yl)pyrazole-3-carbonyl]piperidine-3-carboxylic acid 1-(4,5-dimethoxy-2-phenylphenyl)sulfonylpiperazine 1,3-bis[(Z)-(2-hydroxynaphthalen-1-yl)methylideneamino]thiourea 4-(methylamino)-3-propan-2-yloxycarbonylbenzenesulfonic acid [3-(3,4-dimethoxyphenyl)-5-(2-ethylbutanoylamino)penta-1,3-dienyl]azanium N-azido-1-[4-[5-(3,3-dichloroprop-2-enoxy)pyridine-2-carbonyl]phenyl]-N'-methylmethanediamine 2,5-bis(ethenyl)-1-methanimidoylnaphthalen-4-amine N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5-[(3,3-dimethylbutanoylamino)methyl]-2-fluorobenzamide 3-bromo-5-methoxybenzaldehyde 4-chloro-2,6-di(propan-2-yl)benzoic acid 5-[(Z)-(3-ethyl-1,4-dimethoxynaphthalen-2-ylidene)methyl]benzene-1,3-diol 2-[(Z)-hydroxyiminomethyl]-6,7-dihydrothieno[3,2-c]pyridin-5-one 1-[4,5-dihydroxy-7,8-dimethoxy-3-(5-nitro-2H-benzotriazol-4-yl)naphthalen-1-yl]ethanone 2-azido-5,6-dihydropyrido[3,2-h]quinazoline N-(4-chlorophenyl)-3-(1,3-dihydroisoindole-2-carbonyl)thiophene-2-carboxamide 1-(2,6-difluorophenyl)-5-hydroxy-4-(4-methoxyphenyl)-2H-pyrrol-3-one 1-(azidomethyl)-4-[(3,5-dichlorophenyl)methoxy]benzene 1-[(4-tert-butylphenyl)methylamino]-3-cyclohexa-2,4-dien-1-ylurea 1,3-dichloro-2-(4-methoxyphenyl)-5-phenylbenzene 4-[(3R,5S)-3-methyl-5-[2-[2-(trifluoromethoxy)anilino]acetyl]piperidin-1-yl]benzonitrile 1-[3-(2,4-dimethylphenyl)sulfonylpyrrolidin-1-yl]-2-ethoxybutan-1-one 3-[5-(azidooxymethyl)thiophen-2-yl]propanoic acid 3-[N-[(Z)-1H-indol-3-ylmethylideneamino]-4-propoxyanilino]butanoic acid N-[4-chloro-2-(3,5-dimethylpyrazole-1-carbonyl)phenyl]-N'-(2,6-difluorobenzoyl)-4-propan-2-ylpiperazine-1-carboximidamide 6-chloro-2,3-dihydropyrido[4,3-b][1,4]oxazine-1,4-bis(sulfanyl)indol-5-carbonitrile N-[2-(1H-indol-3-yl)ethyl]-4-oxopyrido[1,2-a]pyrimidine-2-carboxamide 6-[4-(2,3-dihydro-1-benzofuran-7-ylsulfonyl)piperazin-1-yl]-N-propan-2-ylpyridazine-3-carboxamide 3-[[(2S)-6-fluoro-4,4-dimethyl-5-oxo-1,3-thiazin-2-yl]amino]-N-[4-methyl-3-(trifluoromethoxy)phenyl]thiophene-2-sulfonamide N-[3,5-bis(ethoxycarbonyl)phenyl]acetamide ethane;4-methyl-2-(N-methylideneamino)benzenesulfonamide 3-[1,2-dihydropyrimidin-6-ylmethyl(propan-2-yl)amino]-5-phenylsulfanylpyrazine-2-carboxamide 7-N,8-N-bis[(2,6-dimethylphenyl)imino]-9H-fluoren-4-amine 1,4-dimethoxybenzene;N'-(2,5-dimethylphenyl)ethane-1,2-diamine 2-fluoro-3-[5-methyl-4-(1H-pyrazol-5-yl)pyridin-2-yl]oxyaniline N-[3-(2,5-dihydropyrrole-1-carbonyl)-4-fluorophenyl]-6-oxo-1H-pyrimidine-4-carboxamide 2-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]-3H-thieno[3,2-d]pyrimidin-4-one 2-N,5,7-trimethyl-6-[(1R)-1-phenylethyl]pyrido[3,4-d]pyrimidine-2,4-diamine 1-[4-fluoro-2,6-di(propan-2-yl)phenyl]-3-[(5R)-2-methyl-4-(oxetan-3-ylsulfonyl)piperazine-1-carbonyl]urea [3,4-difluoro-2-(2-fluoro-4-methylanilino)phenyl]-[3-hydroxy-4-imino-4-(propan-2-ylamino)butanoyl]azanium (2S)-4-hydroxy-3,8-dimethyl-N-([1,3]oxazolo[5,4-b]pyridin-2-yl)nonanamide N-[1-[4-[5-(2,3-dihydro-1H-indazol-5-ylamino)-1,3,4-thiadiazol-2-yl]phenyl]azetidin-3-yl]acetamide 2-[(E)-2-(3,4,5-trimethoxyphenyl)ethenyl]-1H-indole 2-[3-cyano-4-(2,5-dimethylphenyl)-6-fluoro-8-fluoronaphthalen-1-yl]oxyacetic acid 1-cyclobutyl-3-[2,6-di(propan-2-yl)phenyl]imidazolidine 3-[4-[[2-(1H-benzimidazol-2-ylsulfanyl)acetyl]amino]phenyl]propanamide 1-methyl-2-(3-methyliodanuidylpentan-3-yl)benzene ethane;1,2-xylene 2-(dimethylamino)-1-(2,4-dimorpholin-4-ylthieno[3,2-d]pyrimidin-6-yl)propan-1-one;ethane 4-(2,3-dichlorophenyl)sulfanyl-5-isocyano-6-(1H-imidazol-5-ylmethoxy)pyrimidine [2-amino-6-(4,4-dimethylazepan-1-yl)pyrimidin-4-yl]hydrazine N-[5-chloro-2-(4,6-dimethylpyrimidine-5-carbonyl)phenyl]-1-ethylpyrazole-3-sulfonamide 2-[6-(3,4-difluorophenyl)-8-ethyl-1,4-dioxonaphthalen-2-yl]acetic acid;2-methylpropan-2-ol 5-[2,3-dihydroxypropyl(phenacyl)amino]naphthalene-2-sulfonic acid 7-[3,5-bis(trifluoromethyl)phenyl]-1-hydroxy-2H-benzo[f]chromene [(3S,4R)-1-[2,6-difluoro-4-(3-methylpyridin-2-yl)phenyl]sulfonyl-4-hydroxypyrrolidin-3-yl]carbamic acid N-[3-[1-hydroxy-2,4-dioxo-6-(trifluoromethyl)quinazolin-3-yl]phenyl]propanamide 3-[4-(5-acetamidopyridin-2-yl)phenyl]butanoic acid 1-[3-(4-azidophenoxy)propyl]piperidine 2-(1,5-dihydroxycyclohexa-2,4-dien-1-yl)benzotriazol-2-ium-4-sulfonamide ethane;1-[2-(3-methoxyphenyl)sulfanylethyl]pyrrolidine N-ethyl-2,4-difluoro-6-[3-(1H-imidazol-5-yl)propanoylamino]benzamide 4-(3,4-dichlorophenyl)-1-(3,3,5-trimethylhexan-2-ylsulfonyl)butan-2-one 4-amino-1-[(3R)-3-hydroxypyrrolidine-1-carbonyl]pyridin-2-one (1Z,3E)-2,5-dibromo-6-[(1R)-3-methylcyclohepta-2,4-dien-1-yl]oxyhexa-1,3,5-triene-1,4-disulfonic acid 3-[2-methyl-4-[(Z)-prop-1-enyl]phenyl]cyclohepta-1,4,6-triene 4-[3-(3,5-dimethylphenyl)-7-(6-fluoroquinolin-4-yl)-5-sulfanylideneimidazo[1,2-c]imidazol-1-yl]butanenitrile;ethane 3-[(5R)-8,11,14-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-1(10),2,4,6,8,12(17)-hexaen-9-yl]propanoic acid 5-methyl-6,11b-dihydro-[1]benzofuro[2,3-a]carbazole 2-(N-hexyl-4,5-dimethyl-2-phenyldiazenylanilino)acetamide 2-methyl-5,6-dioxo-8-(1,3-thiazol-4-ylmethylamino)pyrimido[4,5-b]azepine-9-carboxylic acid 4-(benzenesulfonyl)-1H-inden-2-amine 4-cyclopropyl-N-[1-(5-methoxy-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carbonyl)azetidin-3-yl]benzamide 2-bromo-N,N-bis(oxiran-2-ylmethyl)benzamide (3-aminophenyl)-[4-[[4-(4,5-dihydro-1H-imidazol-2-yl)piperidin-1-yl]methyl]piperidin-1-yl]methanone 4-[3-(azidomethyl)phenyl]thiadiazole 2-[4-[(3S,5R)-3,5-dimethylpiperazine-1-carbonyl]-5-ethoxy-2-methylanilino]-8H-pyrido[2,3-d]pyrimidin-7-one 2-[4,7-bis(ethenyl)-1H-imidazo[4,5-c]pyridin-6-yl]aniline N-[2-amino-5-[methyl(methylamino)phosphanyl]phenyl]formamide;6-fluoro-4-methyl-1,3-dihydrobenzimidazol-2-one 2-methyl-1,3-bis(phenylmethoxy)propan-2-ol 6-[2-fluoro-3-(trifluoromethyl)phenyl]-5,8-dihydroxy-1H-quinolin-4-one N-[1-(3,5-difluorophenyl)sulfonylpiperidin-4-yl]thieno[2,3-c]pyridine-2-carboxamide 2-[4-amino-6-(dimethylamino)pyrimidine-5-carboximidoyl]oxyethanol 1-(3-aminopyrrolidine-1-carbonyl)-4,5-dichloropyrrole-2-carbonitrile (3Z)-4-[6-[[1-(5,6-dihydronaphthalen-2-ylmethyl)piperidin-3-yl]amino]pyrazin-2-yl]penta-1,3-dien-2-amine;1-ethylpyrrolidine 5-[6-[6-(4-azidopiperazine-1-carbonyl)naphthalen-2-yl]oxypyridin-3-yl]-1,2-thiazol-3-one (6R,11S)-8-[2-cyclopropyloxy-3-(hydroxymethyl)pyridine-4-carbonyl]-2-oxa-5,8,12-triazatricyclo[boratricyclo[12.4.0.06,10]octadeca-1(18),14,16-trien-4-one (2Z)-1-[4-(trifluoromethoxy)phenyl]octa-2,6-dien-3-ol 3-(4-methoxybenzoyl)-5-oxo-1,2-oxazole-4-carbonitrile 4-chloro-2,6-dimethoxy-3-nitrosobenzaldehyde 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N-[(E)-(6-methyl-4-oxopyran-2-ylidene)amino]acetamide 4-[4-[(2,6-dichlorobenzoyl)amino]phenoxy]-N-methylpyridine-3-carboxamide 2-[6,7,10a-trimethyl-4-(4-methylphenyl)sulfanyl-5-oxo-3,4,8,9-tetrahydro-1H-pyrido[1,2-a]pyrazin-2-yl]-N-[2,6-di(propan-2-yl)phenyl]acetamide 4-(1-amino-3,6-dihydro-2H-pyridin-5-yl)-N-[2-[[[2-(4-chlorophenoxy)acetyl]amino]methoxymethyl]phenyl]benzamide 7-(2,5-dimethylphenyl)-8-hydroxychromene-2,4-dione 4-hydroxy-2-oxochromene-3,7-dicarboxylic acid 3-[(2E)-3,7-dimethylocta-2,6-dienoxy]-4-pentylisochromen-1-one 5-(2,3-dihydroindole-1-carbonyl)-N-methylfuran-3-sulfonamide 3-benzyliminobutanal;2,2,2-trifluoroacetic acid 1-[4-(1,3-benzodioxol-5-yl)-4-ethoxypiperidin-1-yl]ethanone (4-aminophenyl)-(7,7-difluoroheptyl)azanide (2R)-4,6-dimethoxy-3-[[4-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-3-carbonyl]amino]-1H-indole-2-carboxylic acid 1-(4-methoxyphenyl)sulfinylpyrrolidine-2,5-dione 1-[3-(2,5-dioxopyrrolidin-1-yl)oxy-2-methylbenzoyl]pyrrolidine-3-carboxylic acid (5R)-3-[4,5-difluoro-2-[(7H-purin-6-ylamino)methyl]phenyl]-5-[1-hydroxypropyl-[2-methoxy-6-[[1-[(2-methylpropan-2-yl)oxycarbonyl]piperidine-4-carbonyl]amino]pyridin-3-yl]amino]-5-oxopentanoic acid 5-[(5-cyclopropyl-1H-pyrazol-4-yl)methylidene]-2-methylidenethiolan-3-one 2-[(E)-1-(4-chlorophenyl)ethenylsulfanyl]-N-ethyl-6-fluoroquinolin-3-amine N-[1-(2,6-dimethyloxan-4-yl)ethyl]pyrazine-2-carboxamide 2-[1-(4,5-dimethyl-1H-imidazole-2-carbonyl)piperidin-3-yl]-N-pyridin-4-ylacetamide 5-ethylsulfanyl-N'-hydroxypyrazine-2-carboximidamide N-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-2-(4-methoxyphenyl)triazole-4-carboxamide 3-[4-[bis(2-bromoethyl)amino]butanoyloxycarbonyl]benzoic acid 5-chloro-N,2-dimethylbenzenesulfonamide 7-[5-(3,4-dihydroxyphenyl)pentyl]-2,3-dihydrochromen-4-one (3S,4S)-3-[4-(trifluoromethylsulfanyloxy)phenyl]hex-1-en-2-amine N-(2,3-dihydro-1H-inden-5-yl)-5-fluorospiro[6H-pyrrolo[3,4-b]pyridine-7,1'-cyclobutane]-2-carboxamide 2-[3-[(4-aminophenyl)methyl]-5-[2-[1-cyclohexa-1,5-dien-1-yl-2-hydroxyethoxy]ethylamino]pyrazin-2-yl]phenol 2-(cyclopropylmethyl)-7-(trifluoromethoxy)quinoline-3,4-diamine (2S)-3-(5-cyanopyridin-2-yl)oxy-N-[2,6-dimethyl-4-(5-oxopyrrolidin-3-yl)phenyl]-1-(methanesulfonamido)pyrrolidine-2-carboxamide 1-(2-methoxypyridine-4-carbonyl)-2,3,6,7-tetrahydroazepino[3,2-b]indole-5-carboxylic acid 4-[(2,5-difluorophenyl)methyl]-3-[(4-methoxyphenyl)methylsulfanyl]azepane 3-[5-(3-chlorophenyl)hexanoylamino]propylcarbamic acid 2,3-dimethyl-1,4-bis(trichloromethoxy)benzene N-[(1S)-3-methoxy-2-oxocyclopentyl]-5-[2-(trifluoromethyl)pyridin-4-yl]-7,8-dihydro-6H-thieno[3,2-b]azepine-2-carboxamide 5-chloro-2-[1-(3,4-difluorophenyl)ethyl]-7-methylsulfonyl-1H-indole 4-[3-methyl-2,6-dioxo-1-(pyridin-4-ylmethyl)pyrimidin-4-yl]oxypiperidine-1-carboxylate 5-(1-azido-2,3,4,9-tetrahydro-1H-fluoren-3-yl)-2-methylpyridine [3-azidooxy-5-(trifluoromethyl)phenyl]methanol 6-(4-chlorophenyl)-5-pyridin-2-yl-1H-pyrazolo[3,4-d]pyrimidin-7-one 1-[6-[[(Z,2E)-2-ethylidenepent-3-enyl]amino]pyridine-3-carbonyl]piperidine-4-carboxylic acid 2-[(4,7-dimethylthieno[3,2-d]pyrimidine-6-carbonyl)amino]acetic acid (3Z)-2-[[1-(4-methoxyphenyl)pyrazol-4-yl]iminomethyl]hexa-1,3,5-trien-3-amine 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-N-methyl-N-(1,2-oxazol-3-yl)-1,2-oxazole-5-carboxamide (E)-N',3-dimethyl-2-[(Z)-prop-1-enyl]pent-2-enehydrazide;ethane;(2E,4Z,6Z)-2-methylocta-2,4,6-triene;N-[3-[methyl-(5-phenyl-1H-imidazol-2-yl)amino]propyl]formamide N-(4,5-dichlorothiophen-2-yl)sulfanyl-1,1-difluoromethanesulfinamide 2-[2-hydroxy-5-(2-methoxypyridin-3-yl)phenyl]-N-methyl-N-(1,2-oxazol-4-ylmethyl)-3H-benzimidazole-5-carboxamide 1-bromo-5-fluoro-2,4-di(propan-2-yl)benzene N-[1-(1,3-benzodioxol-5-yl)butan-2-yl]-5-ethoxy-6-fluoropyridine-3-carboxamide N-cyclopropyl-2-methoxy-4-[7-[(5-oxopyrrolidin-3-yl)methyl]imidazo[1,2-a]pyridin-3-yl]benzamide 2-(1H-pyrazol-5-yl)-N'-[[5-(trifluoromethyl)pyridin-3-yl]methoxy]benzenecarboximidamide 3-(4-methylpiperazin-1-yl)isoquinoline 6-(3,4-dichlorophenyl)-2H-1,3-oxazine-5-carboxylic acid [4-[[2-(5-bromo-2,6-dimethylpyrimidin-4-yl)sulfanylacetyl]amino]phenyl]urea 1-[4-methyl-3-(trifluoromethyl)phenyl]ethanethiol 2-[1,1,1,3,3,3-hexafluoro-2-(4-phenylmethoxyphenyl)propan-2-yl]benzaldehyde 3-[(1R,5S)-3-benzyl-9-azabicyclo[4.2.0]octan-8-yl]-2-(6-methylpyridin-3-yl)propanamide 5-(2,4-dihydroxyphenyl)-4-[1-(4-hydroxyphenyl)butyl]-3-methyl-1H-imidazole-2-thione 4-(3,5-dimethylphenyl)sulfonyl-N-[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]piperazine-1-carboxamide N-[2,6-difluoro-3-(methylamino)phenyl]acetamide N-[(1S)-1-cyclohexylethyl]-5-[[4-hydroxybutyl(methyl)amino]methyl]pyridine-3-carboxamide 7-(1,5-dimethylpyrazol-3-yl)-2-(furan-2-ylmethylamino)-6H-[1,3]thiazolo[4,5-d]pyrimidin-5-one 3-cyclohexyl-2-(trifluoromethyl)pyridine;ethanol [[5-fluoro-2-methyl-3-(methylamino)phenyl]-(6-pyridin-4-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl)methylidene]azanium 2-[(4-chlorophenyl)methyl]-N-[2-(diethylamino)ethyl]-5-propan-2-ylthiophene-3-carboxamide 1-[(3R)-5-[4-[2-(difluoromethoxy)phenyl]phenoxy]pentan-3-yl]pyrrolidine 2-(ethylamino)-6,8-dimethoxyquinazolin-4-amine;hydrochloride 4-(difluoromethoxy)-3-[5-fluoro-2-(oxolan-3-ylamino)pyridin-4-yl]sulfanylbenzoic acid 3-[(3S)-1,2,3,4-tetrahydroisoquinolin-3-yl]-5H-[1,2]oxazolo[5,4-d]pyrimidin-4-one 5-[3-(2,4-difluorophenoxy)pyrrolidine-1-carbonyl]-2-methylbenzamide 2-[4-chloro-3-(trifluoromethyl)phenoxy]-N-[2-[2,6-dichloro-4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]ethyl]acetamide 2-(4-benzoylphenoxy)-N-[5-cyano-6-[2-hydroxyethyl(propanoyl)amino]pyridin-3-yl]acetamide [4-[4-(difluoromethoxy)phenyl]sulfonylpiperidin-1-yl]-(2,3-dihydropyrrolo[2,3-b]pyridin-1-yl)methanone [(E)-4-[3,5-bis(trifluoromethyl)phenyl]-3-hydroxybut-1-enyl]azanium (3R)-4-(2,6-difluorophenyl)-3-[5-methoxy-6-methyl-1-(3-methyl-3-morpholin-4-ylbutanoyl)-2H-pyrrolo[2,3-b]pyridine-3-carbonyl]piperazin-2-one 4-[(3,5-difluorophenyl)methylamino]-2-[(1,1-dioxothian-4-yl)amino]pyrimidine-5-carboxamide;ethane 3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]benzene-1,2-diol N-[4-(cyclopropylamino)-3-hydroxybutyl]pyrimidine-5-carboxamide (3Z,6E)-3-[(5-chloro-2-hydroxyphenyl)methylidene]octa-1,7-dien-4-one 2,6-bis(tert-butylsulfanylamino)-9H-fluoren-4-ol (2S)-1-[4-(2,6-difluorophenoxy)benzoyl]pyrrolidine-2-carboxamide 7-(3,4-dichlorophenyl)-N-[3-methoxy-4-(6-methylpyridin-2-yl)sulfanylbutyl]-1H-indole-3-carboxamide N-(4-chlorobutyl)-2,6-difluoro-N-[4-[(2-phenylpyrazol-3-yl)sulfamoyl]phenyl]aniline N'-hydroxy-6-methyl-3-[(2,4,5-trimethoxyphenyl)methoxy]pyridazine-4-carboximidamide N-(5-chloropyridin-2-yl)-2,4,6-trimethyl-N-[(3R)-1-propanoylpiperidin-3-yl]benzenesulfonamide N-[2,4-dioxo-3-(phenylmethoxymethyl)piperidin-1-yl]acetamide 2-(4-tert-butylphenyl)-1,3,10-triazatricyclo[6.3.0.02,6]undeca-9,11-diene 6-[4-(1,4-diazepan-1-yl)-3-(trifluoromethyl)anilino]-2H-pyridine-3-carboxylic acid;ethane 4-chloro-2,6-dimethylpyrimidine-5-carbonitrile;ethane 2-(4-azido-1H-indole-7-carbonyl)cyclopentane-1,3-dione 4-chloro-N-[(2S)-1-[3,5-dihydroxy-7-methyl-3-(trifluoromethyl)azepan-1-yl]butan-2-yl]-3-ethoxybenzamide (2R,3S)-2-[[5-chloro-4-(3-methylanilino)pyrimidin-2-yl]amino]butanamide N-[3-(tert-butylamino)sulfanylphenyl]-2,4,6-trimethylbenzenesulfinamide 3-amino-1-(3,5-dichlorophenyl)pentan-2-one;hydrochloride 6-(3-morpholin-4-ylpropylamino)-2,4-dioxo-1H-pyrimidine-5-carboxamide 3-cyclohexyloxy-4-methoxyaniline N-[(4-methoxypyridin-2-yl)methyl]-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide 2-(3,5-dimethylpyrazol-1-yl)benzonitrile;ethane 6-(2,4-difluorophenyl)-5-ethyl-N-[4-(1H-imidazol-2-yl)cyclohexyl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine 3-[2-(4-hydroxyphenyl)ethynyl]phenol 3-[4-(difluoromethoxy)phenyl]-5,6-bis(trichloromethyl)-1H-imidazo[4,5-b]pyrazine 2-cyclohexyl-6-[(3,5-ditert-butyl-4-hydroxyphenyl)methyl]phenol N-(6,7-dihydro-1H-indazole-3-carbonyl)-2-methoxyacetamide 1,3-diamino-1-[2-(4-phenoxyphenyl)sulfanyl-3-propylphenyl]urea 2-[2,6-di(propan-2-yl)phenyl]-4-[3-(1H-inden-1-yl)phenyl]pyridine 2-[5-(3-bromophenyl)-1H-imidazol-2-yl]-6-tert-butylphenol N-[2-(1H-indole-3-carbonylamino)ethyl]imidazo[1,5-a]pyridine-6-carboxamide 2-(4-bromonaphthalen-1-yl)oxy-N-(2-hydroxyethyl)benzamide 5-[(E)-[6-bromo-2-oxo-3-[4-(trifluoromethoxy)phenyl]-1,3-dihydroindol-7-yl]methylideneamino]-1,3-thiazolidine-2,4-dione ethane;N-[5-methyl-2-(4-oxo-1,3-benzothiazin-2-yl)phenyl]acetamide 4-[(5Z,7Z)-7-ethoxynona-1,3,5-trienyl]phenol N-(4-chlorophenyl)-2,3-dihydroindole-1-carboxamide 2-[(3S)-4,4-difluoro-1-propanoylpyrrolidin-3-yl]oxy-5-[4-[1-[6-(methylsulfonylcarbamoylamino)pyridin-3-yl]cyclopropyl]phenyl]benzonitrile N-methyl-3-[4-(4-morpholin-4-ylanilino)thieno[3,2-d]pyrimidin-6-yl]propanamide 2-methoxyethyl(9H-xanthene-1-carbonyl)azanium (4R,5S)-1-methyl-6-[3-oxo-4-[[6-(trifluoromethoxy)pyridin-2-yl]amino]butanoyl]-3-phenyl-4,5,7,8-tetrahydropyrazolo[3,4-b]azepine-4a-carboxylic acid 2-[[4-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]methylamino]quinoline-5,8-dione N-[3,5-difluoro-4-(trideuteriomethyl)phenyl]-2-[2-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]ethynyl]pyrido[3,4-d]pyrimidin-8-amine 5-(4,6-difluorocyclohexa-1,3-dien-1-yl)-N'-[2-[4-(pyridine-4-carbonyl)piperidin-1-yl]acetyl]furan-2-carbohydrazide 5-chloro-N,4-dimethyl-6-(2,3,4-trifluorophenyl)pyrimidin-2-amine 5-(4-chlorophenyl)spiro[1,2-dihydropyrazolo[3,4-b]pyrazine-6,3'-pyrrolidine] N-[4-fluoro-6-[(3S)-1,2,3,5,6,7-hexahydropyrrolizin-8-yl]pyridin-2-yl]-1-methanimidoylpyrrolo[2,3-b]pyridine-5-carboxamide 4-[6-bromo-13-chloro-10-(dimethylamino)-2-oxo-3,4,9-triazatricyclo[7.5.0.03,7]tetradeca-1(11),5,13-tetraen-12-yl]-N-[[5-fluoro-2-(trideuteriomethoxy)phenyl]methyl]piperidine-1-carboxamide 3-[1-(3,5-diethylphenyl)-2-propan-2-yloxyethoxy]-4,6-dimethylpyridazine (Z)-1,3-diphenyl-2-sulfanylprop-1-en-1-amine ethane;4-[[6-methoxy-2-[1-(trifluoromethyl)cyclopropyl]quinoline-3-carbonyl]amino]pyridine-2-carboxylic acid N-[(E)-2-(3,4-dihydroxyphenyl)ethylideneamino]cyclohexanecarboxamide (3S)-N-[4-(dimethylamino)pyrimidin-2-yl]-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxamide 2-[(E)-but-1-enyl]benzenesulfonamide (5S)-3-[4-fluoro-3-[7-(6-methylpyridin-2-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl]-5-hydroxyhexanamide 2-[(3Z,5E)-4-ethylhepta-1,3,5-trien-3-yl]-1H-indole [(2S,3R)-4-ethyl-1-(2-methoxyphenyl)-2,5-dimethylhexan-3-yl]benzene 4-[5-(2,5-dimethylphenyl)furan-2-carbonyl]morpholine-3-carbonitrile 2-ethyl-3-fluoro-4-[1-(4-hydroxyphenyl)cyclohexyl]phenol 2-(5-cyanonaphthalen-1-yl)oxypropanoate 4-[1-azido-2-(3,5-dimethoxyphenyl)-6-methylsulfonylheptan-3-yl]pyridine N-[(4R)-1-azido-5-methylsulfonyl-3,6-dihydro-2H-pyridin-4-yl]benzamide 3-(2,6-dimethylmorpholine-4-carbonyl)benzoic acid 4-methyl-2-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-1-yl)pentan-3-one 2-[4-[2-(3-methylbutanoyloxy)phenyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxylic acid 1-(3,4-dichlorophenyl)-2-[6-fluoro-2-methyl-7-[methyl-(2,2,6,6-tetramethylpiperidin-4-yl)amino]quinazolin-5-yl]ethanone 3-[2-oxopropyl(phenacyl)amino]propanoic acid 3-(7,8-difluoro-2-methylimidazo[1,2-a]pyridin-6-yl)-4-ethoxybenzaldehyde;4-fluoro-N-methylcyclohexane-1-carboxamide 1-azidooxy-2,3,4-trichlorobenzene 4-[1,3-dioxo-2-(4-phenylmethoxycyclohexyl)isoindol-5-yl]butanoic acid (4-diphenylphosphoryl-2,6-difluorophenyl)methanamine (3Z,5E)-4-[5-chloro-2-fluoro-6-[5-fluoro-1-[2-[1-(methylamino)cyclopropyl]ethoxy]-7-(trifluoromethyl)indole-2-carbonyl]pyridin-3-yl]-5-methyl-3,5-di(piperidin-4-ylidene)pentan-2-one 6-(4-methoxybutanoyl)pyridine-3,4-dicarboxylic acid N-methyl-N-[4-[4-(2-phenylacetyl)piperazine-1-carbonyl]phenyl]-1H-imidazole-5-carboxamide N-[2-(3,4-dimethoxyphenyl)ethyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide 5-[3,5-bis(trifluoromethyl)phenyl]-N-methoxypent-4-enamide (2R)-1-[4-(5,6-dimethylpyrazine-2-carbonyl)piperidin-1-yl]propan-2-ol [4-methyl-3-(trifluoromethoxy)phenyl]-(2,3,4,6-tetrahydropyrano[2,3-b]pyrrol-5-yl)methanone 2-[(3S)-1-cyclohexylpyrrolidin-3-yl]oxy-6-fluoropyridine 1-[(3aR,6aS)-2-benzyl-5-hydroxy-3a-methyl-1,3,4,6,6a-hexahydrocyclopenta[c]pyrrol-5-yl]butan-1-one [5-chloro-1-(cyclopropylmethyl)indol-2-yl]-(4-prop-2-enoxyphenyl)methanone 4-[(3R)-1-[5-chloro-2-(3,4-dimethoxyphenoxy)phenyl]-5-oxopyrrolidin-3-yl]benzaldehyde 3-[3-(1,6-dihydrocyclohepta[b]pyrrol-2-yl)propyl]-7,8-dimethoxychromen-2-one 2-[4-chlorobutyl(pyridin-3-yl)amino]acetic acid N-(2-methoxyethyl)-4-[1-[4-(tetrazol-1-yl)phenyl]imidazo[1,5-a]pyrazin-3-yl]benzamide 4-[(4-chlorophenyl)diazenyl]-2H-benzotriazole-5-thiol N-[(3-bromophenyl)methyl]-2-[[4-(pyridine-3-carbonylamino)benzoyl]amino]benzamide (3-fluoropyridin-2-yl)-[2-hydroxy-4-methoxy-5-[3-methyl-7-[[[5-[(3R)-oxolan-3-yl]oxypyrimidin-2-yl]amino]methyl]-1,2-benzoxazol-6-yl]phenyl]methanone [2-[5-(cyclohexen-1-ylmethylamino)imidazo[1,2-c]pyrimidin-8-yl]phenyl]sulfanium N'-cyclohexyl-2,6-dimethoxybenzimidazole-1-carboximidamide 2-ethenylsulfanyl-5,6-dimethylnaphthalene 3-(6-azidohexyl)pyridine 2-[6-(3-chlorophenoxy)pyridin-3-yl]acetic acid 4-[(5,6-diethyl-2,3-dihydro-1H-inden-1-yl)methoxy]-N,N'-dimethylbenzenecarboximidamide;hydrochloride 3-(3,5-difluorophenoxy)propanamide;2,6-diethylpyridine 2-(2,6-dioxopiperidin-3-yl)-4-[[1-[1-[1-(4-methylsulfonylphenyl)ethenyl]piperidin-4-yl]pyrazol-4-yl]methylamino]isoindole-1,3-dione 6-[2-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-yl)ethoxymethyl]pyridine-3-carboxylic acid N-[(1Z)-3,4-dimethylpenta-1,3-dienyl]methanimine;ethane;2-methoxybut-2-ene N-(3,4-dihydro-2H-chromen-8-ylsulfanyl)pyrimidine-5-carboxamide 4-(2-bromoanilino)-N'-hydroxypyridine-2-carboximidamide (E)-N-[4-(1H-indole-3-carbonyl)phenyl]-2,4-dimethylpent-2-enamide 2-amino-4,5,6,7,8,9-hexahydro-1H-cycloocta[c]pyrazole-3-carboxamide;N-[[4-(1H-imidazol-5-yl)phenyl]methyl]-N-propylpropanamide N-[2-(1-methylpyrazol-4-yl)ethyl]-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-3-carboxamide 2-[4-amino-3,5-dicyano-6-(N'-methylcarbamimidoyl)pyridin-2-yl]sulfanyl-N-tert-butylacetamide N-(4,6-dimethylpyrimidin-2-yl)-4-[3-nitro-N-phenacylanilino]benzenesulfonamide [(3R)-1,4-dihydroxypentan-3-yl]oxy-phenylborinic acid N'-hydroxy-2-[(3R)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]ethanimidamide 1-[(3,4-difluorophenyl)methyl]pyrazolo[4,3-c]pyridine N-[[6,7-dichloro-2-methyl-4-oxo-1-(trifluoromethyl)isoquinolin-3-ylidene]amino]pyridine-4-carboxamide 4-amino-5-iodo-1H-pyrimidin-6-one 4-N,6-dimethyl-5-(4-methylphenyl)pyrimidine-2,4-diamine N-[(2R,3S)-2-butylsulfanylnonyl]-4-methoxybenzenesulfonamide 1-(4-aminophenyl)-6,8-dibromochromen-4-one 3-butoxy-5,6,7,8-tetrahydronaphthalene-2-carbonitrile 5-(1,2,3,6-tetrahydropyridin-4-yl)-3-[5-(pyrrolidine-1-carbonyl)-1H-indol-2-yl]-N-[[(Z)-2,4,4-trimethylpent-2-enoyl]amino]thiophene-2-carboxamide 4-[2,5-bis(trifluoromethyl)phenyl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione (1S,4R)-4-methyl-2-(1,3-thiazol-5-yl)cyclopentane-1-carboxylic acid 2-[4-[1,1-difluoro-2-(3,4,5-trifluorophenyl)ethyl]cyclohexyl]-6-propoxynaphthalene 1-[5-(2-ethoxypyridin-3-yl)sulfanylpyrazin-2-yl]-N,3-dimethylbutan-2-amine 2-tert-butyl-4-fluoro-1-[4-(trifluoromethyl)phenyl]benzene N-[3,6-difluoro-2-(triazol-2-yl)phenyl]-4-methoxybutanamide 2-(4-aminophenyl)-1-[8-hydroxy-3,7-dimethyl-6-[3-(trifluoromethoxy)phenyl]quinolin-5-yl]ethanone 1-[2-(1H-benzimidazole-2-carbonyl)phenyl]-3-propylurea 5-methylsulfinylpyridine-2,3-diamine 3,6-dicyclohexyl-5-(5-methylfuran-2-yl)pyridine-2,4-dicarbonitrile 2-(1,3-benzothiazol-2-yl)-5-chloro-4-fluorophenol (2S)-1-[4-(N'-hydroxycarbamimidoyl)phenyl]sulfonylpyrrolidine-2-carboxylic acid 2-[[(3aR,6aS)-5-methylsulfonyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole;2,2,2-trifluoroacetyl]amino]benzamide (3R,4S)-5-methyl-1-[2-phenyl-6-(trifluoromethyl)pyrimidin-4-yl]piperidine-3,4-diol N'-(3,4-dihydropyridin-5-yl)-2-methylidene-5,6-bis[(E)-3-phenylprop-1-enyl]-1H-pyrimidine-4-carboximidamide 2-azidooxy-5-bromopyridine 2-[4-(N-(2,5-dichlorophenyl)-4-propylanilino)phenoxy]acetic acid 5-(4-azidobutyl)-2-methoxypyridine 2-[4-(4-butylcyclohexyl)phenyl]-5-heptoxypyrimidine N-[4,5-bis(ethenyl)-2-methylphenyl]-6-methoxy-1H-indole-3-carboxamide 4-(2,6-dimethyl-3H-pyridine-5-carbonyl)-1-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)piperazin-2-one 3-amino-6-(2,5-dichlorophenyl)-N'-[4-(trifluoromethylsulfanyl)anilino]pyridine-2-carboximidamide 2-[(2R)-4,5-dimethyl-1-(thiophen-2-ylmethoxycarbonylamino)heptan-2-yl]-2-oxoacetic acid 1-(9H-fluoren-9-ylmethoxycarbonyl)piperidine-4-carboxylic acid 2-(1-azido-1,2-diphenoxyethyl)naphthalene 5-methyl-7-oxo-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-naphthalen-2-ylamino]propanoic acid (2S)-1-[[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]amino]propane-1,2-diol 4-(5,6-dimethylpyrimidin-4-yl)-N-[1-[5-fluoro-2-(triazol-2-yl)benzoyl]azetidin-3-yl]piperazine-1-carboxamide 2-[4-[(Z)-2-(aminomethyl)-3-fluoroprop-2-enoxy]phenyl]-N,N-diethylacetamide 7-methyl-4,7-diphenyloctanenitrile 2-(5-hydroxy-1H-indol-3-yl)butanoic acid 1-(2,6-dimethylphenyl)-3-[2-ethyl-4-methanimidoyl-5-[2-(trifluoromethyl)anilino]phenyl]urea 2-[(1S)-1-[6-[cyclopropylmethoxy(difluoro)methoxy]pyridin-3-yl]ethyl]-4,5-dihydrofuro[3,2-g]chromen-7-one 3-(N-hexyl-4-methoxyanilino)phenol 2-[3-[1-(3,5-dimethoxyanilino)ethenyl]thiophen-2-yl]benzoic acid [4-(3-chlorophenyl)piperazin-1-yl]-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]methanone 4-[(2Z,4E)-hepta-2,4-dien-4-yl]-5,8-dihydronaphthalene N-[4-(aminomethyl)phenyl]quinolin-5-amine 4-[(2,6-dichlorobenzoyl)amino]butanoate 6-methylsulfonyl-5,7-dihydropyrrolo[3,4-d]pyrimidine N-(8-bromoquinoxalin-5-yl)-2-methoxy-N-pyridin-2-ylacetamide 3-[1-(3,5-difluorophenyl)ethyl]-2H-pyrimido[4,5-b]quinoline 5-[4-(4-chlorophenyl)butyl]-2H-1,2,4-triazine 3-bromo-N-[(1R,2S)-2-methylcyclopropyl]thiophene-2-carboxamide 1,2-diamino-4-(5-cyano-6-methylpyridin-3-yl)-6-oxopyridine-3,5-dicarbonitrile 4-(2,6-difluorophenyl)-1,3-thiazol-5-amine;ethane 3-[5-(2,4,6-trimethylphenyl)pyrazin-2-yl]pyridine 4-(2,6-dichlorophenyl)sulfanyl-3-hydroxy-3H-pyridine-2-carboxylic acid 3,7-dichloro-4-fluoroquinoline [4-amino-2,3,5,6-tetrafluoro-N-methyl-4-(5-phenylbenzotriazol-1-yl)anilino]sulfanium 2-methoxycarbonyl-5,7-dihydroquinolino[1,6-c]quinazoline-9-carboxylic acid N-cyclopropylformamide;4,5-dimethoxy-2-methyl-3-(3-pentan-2-ylphenyl)aniline 1-methyliodanuidylcarbonyloxycyclohexa-2,4-diene-1-carboxylic acid 3-[8-methoxycarbonyl-7-(trifluoromethyl)naphthalen-2-yl]propanoic acid 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-N,N-dimethylmethanamine 2-(6-aminopyridin-3-yl)-N'-hydroxybenzenecarboximidamide 2-[5-methyl-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)naphthalen-1-yl]pyridine 1-[3,5-bis(trifluoromethyl)phenyl]-N,4-dipropylcycloheptan-1-amine 3-[[3-[2,6-dimethyl-4-(pyrrolidine-1-carbonyl)phenoxy]azetidin-1-yl]sulfonylmethylideneamino]benzoic acid 2-[3,5-difluoro-4-(trifluoromethylsulfanyl)phenyl]-4-oxobutanamide 2-[3-(1,4-diazepan-1-yl)propyl]isoindole-1,3-dione 1,2-bis(4-chlorobutyl)-9H-fluorene 2-(N,4-dimethylanilino)-7-fluoroquinoline-3-carbonitrile 1,3-dichlorocyclobutane;N-[4-methoxy-2-[(Z)-3-oxopent-1-enyl]phenyl]acetamide 7,8-difluoro-2-[(4E)-4-methoxyiminopiperidin-1-yl]-1H-quinolin-4-one 2-amino-4-(1H-indol-3-yl)butanoic acid 5-[(3,4-dichlorophenyl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine [(3S,4R)-3-[5-(difluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]-4-methoxypyrrolidin-1-yl]-[5-methyl-6-(methylideneamino)pyridin-3-yl]methanone 1-(4,7-diazaspiro[2.5]octan-7-yl)-3-(7-methoxy-1H-indol-3-yl)propan-1-one 2-(3,4-dimethoxyphenyl)iminocyclohexane-1,3,5-trione 4-N-[4,5-bis(ethenyl)pyrimidin-2-yl]benzene-1,4-diamine 1-[3,4-bis(ethenyl)benzoyl]pyrrolidine-2-carboxylic acid N-cyclohexyl-2,4,5-trifluoro-3-hydroxybenzamide 3,4-dichloro-N-[(2S)-1-(1H-indole-5-carbonylamino)propan-2-yl]benzamide 3-[3-[2,4-bis(phenylmethoxy)phenyl]pyrazolo[3,4-b]pyridin-1-yl]propan-1-ol N-[(3S,4R)-1-cyclobutyl-6-oxopiperidin-3-yl]pyrazine-2-carboxamide;hydrochloride 1-[3,4-bis(trifluoromethyl)phenyl]-3-[2-[[1,3,5-trimethyl-6-oxo-8-[3-(trifluoromethoxy)phenoxy]imidazo[1,2-a]pyridine-7-carbonyl]amino]ethyl]urea 4-[(1E,4Z)-5-[3,5-bis(trifluoromethyl)phenyl]penta-1,4-dienyl]phenol N-[1-(2,3-dihydro-1H-inden-5-yl)cyclopropyl]-4,6-dioxo-7-phenyl-2,3,8,9,10,11-hexahydro-1H-pyridazino[1,2-a]indazole-8-carboxamide 2-[1-cyclohexyl-4-(4-methoxyphenyl)piperazin-2-yl]ethanol;(2,5-difluorophenyl)thiourea 2-(1,3-benzothiazol-2-yl)-4,5-dimethoxybenzenethiol 6-methoxy-3,4-bis(phenylmethoxy)hexan-1-ol 4-[5-azido-2,3-dimethyl-6-(1H-pyrrolo[3,2-b]pyridin-2-yl)phenyl]morpholine (2S)-2-[(7R)-3,4,6,10b-tetrahydro-1H-pyrazino[2,1-a]isoindol-2-yl]-N-(cyanomethyl)-3-methoxypropanamide 6-[(2R)-1-propanoylpiperidin-2-yl]-3-pyrimidin-4-yl-4H-1,2,4-triazin-5-one 4-[1-carboxynonyl(ethenylsulfonyl)amino]benzoic acid 2,7-dimethyl-4-(1H-pyrazol-5-yl)quinoline 5-(N-[2,4-dichloro-3-[(4-chlorophenyl)sulfonylamino]benzoyl]anilino)pyridine-3-carboxylic acid 1-[4-(2,4,6-trichlorophenoxy)pyridine-3-carbonyl]azetidine-3-carboxamide (3S,4R)-3-benzyl-1-ethenylpiperidine-4-carbonitrile 3-[1-(3,4-dihydronaphthalen-1-ylsulfonyl)piperidine-3-carbonyl]-6,7-dimethoxyquinazolin-4-one (5E)-2-(3-chlorophenyl)imino-5-[(4-piperidin-1-ylnaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one 2-[2,4-bis(trifluoromethyl)phenoxy]-6-phenyl-3,5-dihydropyrimidine-4-thione ethane;3-(4-methoxyphenyl)bicyclo[1.1.0]butan-2-one 2,2-difluoropropane;1-[6-fluoro-4-methyl-5-(4-morpholin-4-ylphenyl)pyridine-3-carbonyl]azetidine-3-carboxylic acid N-(2,6-dibromopyridin-4-yl)-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]benzenesulfonamide 6-bromo-2-(4-ethoxybutyl)imidazo[1,2-a]pyridine 2-methylsulfanyl-N'-[1,3]thiazolo[5,4-f]quinazoline-9-carbohydrazide 5-(3,4-dichlorophenyl)-6-ethyl-3-[4-(4-pyrrolidin-1-ylpiperidine-1-carbonyl)anilino]pyridine-2-carboxamide 4-[6-(1H-indazol-3-yl)-2,7-dihydroindazol-3-yl]benzenesulfonamide 3-(3,5-difluorophenoxy)-1-phenylcyclobutane-1-carboxylic acid 1-methyl-N-(pyridin-4-ylmethylidene)piperidine-3-carboxamide 4-[2,6-difluoro-4-(methylamino)anilino]-3-fluorophenol ethane;5-[1,1,2,3,3,3-hexafluoropropan-2-yl(methyl)amino]sulfanylpyridine-2-carbonitrile 2-tert-butyl-4-propan-2-yl-5,6,7,8-tetrahydroquinoline 2-[4-amino-5-(2,6-difluorophenyl)pyridin-3-yl]-N-(4-chloro-1H-indazol-7-yl)acetamide 4-chloro-2,3,5-trideuterio-6-methylsulfanylphenol 4-[(4-hydroxyphenyl)methyl]-3,5-dimethylpiperazine-1-carboxylate 4-(6,7-dimethoxy-1H-indol-2-yl)piperidine 2-(3,4-dimethyl-6-oxo-1H-pyridazine-5-carbonyl)cyclopentan-1-one 5-[1-(6,8-dichloronaphthalen-2-yl)sulfonylpyrrolidin-3-yl]-2H-triazole-4-carboxylic acid 2-(azidomethyl)-5-(3,5-dimethoxyphenyl)sulfonylpyridine 6-[(4-ethoxyphenyl)methyl]-5-hydroxy-2,3-dimethyl-1H-pyridin-4-one N-[(E)-(3,4-dichlorophenyl)methylideneamino]-2-methylquinoline-6-carboxamide;ethane N-methyl-1,2,3,4-tetrahydrothieno[3,4-d]pyrimidine-8-carboxamide;hydrochloride 5-bromo-N,4-ditert-butyl-3-chloro-2-fluoroaniline 2-(1,5,7a-trimethyl-3,4,4a,8b-tetrahydro-2H-indeno[1,2-b]pyrrole-6-carbonyl)benzoic acid 5-[[1,3-bis(ethenyl)cyclohexa-2,4-dien-1-yl]methyl]-2-(6-chloropyridin-3-yl)oxypyrimidine N-[[(1R,3aR,7aS)-5-benzylsulfonyl-3,3a,4,6,7,7a-hexahydro-1H-furo[3,4-c]pyridin-1-yl]methyl]benzamide;2,2,2-trifluoroacetic acid N-(4,5-dichlorothiophen-2-yl)sulfanyl-2-fluoro-4-[5-methoxy-6-[(1R,2S)-2-phenylcyclopropanecarbonyl]pyridin-3-yl]benzamide N-benzyl-3,4,5-trimethoxy-N-propanoylbenzamide (1R)-4,7-dichloro-2-methyl-6-[4-[2-[2-methyl-5-[3-(trifluoromethoxy)phenyl]-1H-imidazol-4-yl]ethynyl]phenyl]-1,4,5,9-tetrahydropyrido[3,4-b]indole 2-[[4,5-bis(ethenyl)pyridine-2-carbonyl]amino]acetic acid;formaldehyde 1-(2,4-dichlorophenyl)-N-[(E)-(3-ethoxy-5-nitrophenyl)methylideneamino]pyrazolo[3,4-d]pyrimidin-6-amine (E)-3-[2-methyl-4-[(E)-3-pyridin-2-ylprop-2-enoxy]phenyl]-1-morpholin-4-ylprop-2-en-1-one 2-[1,3-bis(methylsulfamoyl)propan-2-ylideneamino]benzoic acid N-(1-cyclopropylethenyl)-5-[3-(4-pyridin-2-yl-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-amine N-[(2S)-1,4-dimethylpiperidin-3-yl]-7H-purine-6-carboxamide 5-[(6-methoxypyridin-3-yl)amino]-1,2-dihydroindazole-3-thione 2-chloro-1-[4-[(2,6-dichlorophenyl)methoxy]cyclohexyl]indole 2-(2,4-difluorophenyl)-2-[3-(5H-pyrrolo[1,2-a]quinoxaline-6-carbonyl)anilino]acetic acid 2-[azido(diphenyl)methyl]-1H-benzimidazole 5-[8-[4,6-di(carbazol-9-yl)pyrimidin-2-yl]-9H-xanthen-1-yl]benzonitrile 4-(ethoxymethyl)-1-[4-[4-(2-fluorophenoxy)phenyl]cyclohexa-2,4-dien-1-ylidene]piperidine 7-ethylsulfonyl-2,5-dimethylpyrrolo[2,3-d]pyrimidine N-[4-[3,5-bis(trifluoromethyl)phenyl]sulfanylphenyl]acetamide;ethane N-methyl-4-(6-methylpyridin-3-yl)aniline 3-(1,4-diazepane-1-carbonyl)benzaldehyde [4-(2,3-dimethylpropoxy)phenoxy]-(2-phenylethylsulfonylamino)phosphinic acid 1-N-[2,3-difluoro-6-(5-methylpyridin-2-yl)phenyl]-4-N-fluorobenzene-1,4-diamine;3-propanoyl-1H-pyrrolo[2,3-b]pyridine N-[(2S)-2-aminobutyl]-N',4,5-trimethoxy-2-nitrobenzohydrazide 2-[(2E,5S)-4-oxo-2-[(Z)-[3-[(4-piperidin-1-ylphenyl)methoxy]phenyl]methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 2,4-dichloro-1-(2,3-dimethylpentoxy)benzene 4-[(Z)-3-cyano-2-methylprop-2-enoyl]oxybenzoic acid (5R)-2,7,9-trimethyl-3-phenylspiro[4H-pyrido[1,2-a]pyrazine-1,4'-cyclohexane] [3-fluoro-2,6-di(propan-2-yl)phenyl]urea (4aS)-1,2,3,9b-tetrahydrochromeno[3,4-c]pyrrole;ethane 4-(1,3-benzodioxol-5-yl)-6-hydroxypiperidine-2-carboxylic acid [6-carboxy-5-(N,3-dimethylanilino)pyridin-2-yl]azanide;cyclopropanethiolate;oxolane;platinum(2+) N-[1-(3,5-difluorophenyl)pyrrolidin-3-yl]-4-ethylthiadiazole-5-carboxamide N-[3-[(5Z)-5-methoxyiminocyclohepta-1,3,6-trien-1-yl]phenyl]formamide 2-chloro-4-[(2,5-dimethylpyridine-3-carbonyl)amino]benzoic acid 2-(N-(4,6-dimethylpyrimidin-2-yl)-2-nitroanilino)acetamide 5-[4-(2,6-diphenylpyrimidin-4-yl)-3,9,10-triazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),4,8,10-pentaen-11-yl]-N,N-dimethylpyridine-2-carboxamide N-[3-(4-acetylpiperazine-1-carbonyl)phenyl]-5-fluoro-7a-methyl-2,3a-dihydropyrrolo[2,3-b][1,4]benzothiazine-6-carboxamide 2-ethylsulfinyl-N-[3-fluoro-4-(7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)phenyl]benzamide 6-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]-2-[(2R)-oxolan-2-yl]-3H-isoindol-1-one 5-azidooxy-2-methylquinoline 6-azidooxy-3H-quinazolin-4-one 4-[2,3-difluoro-4-(trifluoromethoxy)phenyl]-N-methylaniline 3-methyl-5-[[(2S)-piperidin-2-yl]amino]-1,4-dihydroquinazolin-2-one 6-fluoro-5,7-dihydrobenzo[d][2]benzoxepine [1-[4-(hydroxyamino)-6,7-dihydroquinazolin-2-yl]pyrazole-3-carbonyl]urea 2-[5-tert-butyl-3-(4,7-dioxo-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-2-hydroxyphenyl]-N-(2-ethoxy-6-methylphenyl)acetamide 3-[2-amino-5-(1H-pyrrole-2-carbonyl)phenyl]-2,2-dimethylpropanoic acid 4-[5-amino-6-(quinolin-6-ylmethylamino)pyrazin-2-yl]sulfanyl-N-cyclopentylbenzamide (1S,6R)-N-[8-amino-6-(4-propanoylcyclohexyl)isoquinolin-3-yl]-2-cyanocyclopentane-1-carboxamide 4-azido-2-benzylsulfonylquinoline [(3S)-1,2,3,5,6,7-hexahydro-s-indacen-4-yl]urea N-[2,6-difluoro-4-(1H-pyrazolo[3,4-b]pyridin-5-yl)phenyl]formamide;ethane 5-(1,3-benzodioxol-5-yl)-2,4,6-trimethoxypyridine 2-N,6-N-dihexylnaphthalene-1,2,5,6-tetramine 3-[3-[(4S)-2-amino-4-methyl-5,6-dihydro-1,3-thiazin-4-yl]-4-fluorophenyl]-1-(oxetan-3-yl)-1-azaspiro[4.5]decan-2-one 4-N-methyl-6-[(Z)-prop-1-enyl]-2H-pyrazolo[3,4-d]pyrimidine-3,4-diamine 3-(2,4-difluorophenyl)-1-ethylpyrrolidine;methoxymethane 2-[(4R)-7-chloro-10-oxo-4-propan-2-yl-9,12-diazatricyclo[6.5.0.03,5]trideca-1,3(11),4,7,12-pentaen-5-yl]-N-(5-methylpyrazin-2-yl)acetamide 2-[4,5,7-trimethyl-3-(7H-purin-6-ylsulfanylmethyl)pyrazolo[1,5-a]pyrimidin-6-yl]phenol 5-[7-amino-2,4-bis(sulfanylidene)-1H-pyrimido[4,5-d]pyrimidin-3-yl]pentanehydrazide 2-[2-ethoxypropyl(methyl)amino]-N'-hydroxypyridine-4-carboximidamide 2-[4-methyl-1-oxo-3-(propanoylamino)pentan-2-yl]-1H-indole-7-carboxamide 2-[(2,4-dichloropyrimidin-5-yl)-phenacylamino]benzenesulfonic acid 1-(4-fluorophenyl)-3-[2-(1H-indazol-5-ylcarbamoylamino)ethoxymethyl]urea 2-ethenyl-1-[(Z)-pent-3-ynoxy]naphthalene 2-[4-(1,3-diazetidin-1-ium-1-yl)-2,6-difluorophenyl]sulfanyl-5,6,7,8-tetrahydroisoquinolin-2-ium [2-fluoro-4-(3-methylpyridin-2-yl)phenyl]boronic acid 4-[[(2R)-3,3,6-trimethyl-1-oxoisoquinolin-2-yl]methoxycarbonylamino]butanoic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-bromoacetamide 2,4-dichloro-6-(1-methylpyrazol-3-yl)pyrimidine (5-bromopyridine-2-carbonyl)-dimethyl-[2-(3-nitrophenoxy)acetyl]azanium ethane;6-[4-(1-methylcyclopropanecarbonyl)piperazin-1-yl]pyridine-3-carbonitrile 2-[(4-fluorophenyl)methyl]-5-(pyridin-3-ylamino)pyridazin-3-one 4-azido-2,5-dibromopyrimidine 5-[[(6R)-5,8-dioxo-6,7,9,10-tetrahydrobenzo[g]pteridin-2-yl]sulfanylmethyl]furan-3-carbonitrile 3-(2,4,6-trimethylphenyl)pyridine;1,10-phenanthroline N-[1-[4-(hydroxycarbamoyl)cyclohexa-2,4-dien-1-yl]oxyisoquinolin-6-yl]pyridine-3-carboxamide 4-[(3R,4S)-1-azidopiperidin-3-yl]oxybenzoic acid 7-(2,6-difluorophenyl)-12-[4-(dimethylamino)phenyl]-N-(3-hydroxypropoxy)-13-methyl-8-thia-5,10,11,14-tetrazatricyclo[7.4.0.02,7]trideca-1(13),2,4,9,11-pentaene-6-carboxamide 6-[(Z)-but-1-enyl]-3,4-diethylpyridine-2-carboxylic acid 1-[4-hydroxy-3,5-bis(4-methoxyphenyl)cyclohexa-1,3-dien-1-yl]ethanone 4-(methylamino)-3-(4,6,7-triamino-1H-indole-2-carboximidoyl)phenol (3Z,5E)-6-[2-aminoethyl(propan-2-ylidene)azaniumyl]-4-methylidene-3-[1-(2-oxo-1H-quinolin-7-yl)ethenoxy]hepta-5,7-dienoate [(2S)-4,4-difluorobutan-2-yl]oxymethylbenzene N-(2,3-dihydroxypropyl)-N-[4-(pyridin-2-ylsulfamoyl)phenyl]nonanamide 2-methyl-4-[3-(1-methylbenzimidazol-2-yl)propanoylamino]thiophene-3-carboxylic acid (2R)-N',3-dihydroxy-2-[4-hydroxy-5-methyl-6-oxo-1-[3-(trifluoromethyl)phenyl]pyridin-3-yl]butanediamide 5-chloro-N-(2,6-difluorophenyl)-4-oxothiochromene-3-carboxamide N-[1-methyl-5-(1,2,4-triazol-1-yl)pyrazol-3-yl]-2H-triazolo[4,5-b]pyridine-6-carboxamide 4-[2-(3,5-dimethylphenoxy)ethyl]piperidine;N'-hydroxy-4-[(3R)-pyrrolidin-3-yl]oxypyridine-2-carboximidamide 3-methoxy-N,5,6-trimethyl-2-[(5S)-5H-pyrrolo[2,1-a]isoindol-5-ium-5-yl]thieno[2,3-b]pyridine-4-carboxamide [1-(4-ethylphenyl)sulfonylazetidin-3-yl]methanol 3-[2-fluoro-4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)phenoxy]propanenitrile 4-N,4-N-diethyl-1-N-methyl-3-(trifluoromethyl)benzene-1,2,4-triamine 2-azido-3,5-dichloro-6-(1H-indol-4-yl)phenol 1-(2,4-dichlorophenyl)-N-[6-fluoro-3-methylsulfanyl-2-[2-(trifluoromethoxy)phenoxy]pyridin-4-yl]-5-(trifluoromethyl)pyrazole-4-carboxamide 6-ethylsulfonyl-2,2,4-trifluoro-5-(1H-pyrazolo[3,4-b]pyridin-7-yl)-1,3-benzodioxole 2-[5-(4-chlorophenyl)-7,8-dihydro-6H-naphthalen-1-yl]ethanamine (3-tert-butylphenyl)methanesulfonic acid;ethane N-(2,5-dimethylphenyl)-3-[4-(4-methoxyphenyl)-1H-benzimidazol-2-yl]benzenesulfonamide 1-(1H-benzimidazol-2-yl)pyrazole-3-carboxamide;ethane 1-[5-(4-hydroxyphenyl)triazolo[4,5-b]pyridin-3-yl]ethanone 3-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]propanoic acid 2-[1,2-bis(4-methoxyphenyl)imidazol-4-yl]pyridine 2-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(naphthalen-1-yl)amino]acetonitrile 7-bromo-1H-indole-4,5-dicarbonitrile 3-[4,5-dimethyl-6-[(5R)-5-[6-(4-piperidin-1-ylbutoxy)pyridin-3-yl]cyclohexa-1,3-dien-1-yl]pyrimidin-2-yl]propanoic acid 5-[[3-(ethylamino)-1,2,4-triazin-6-yl]oxy]-N,N-dipropylpentanamide 5-methyl-4,9b-dihydro-1H-indeno[2,3-b]pyridine 1-(2,5-dichlorophenyl)-7-(4-methylpiperazin-1-yl)-3-nitrosoquinoxalin-2-one N-[2,6-di(propan-2-yl)phenyl]-1,3,5-triazinane-2-carboxamide (5Z)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[[4-methoxy-3,5-dimethyl-1-(4-nitrophenyl)pyrazol-4-yl]methylidene]-1,3-thiazolidin-4-one 1-methyl-4-[(2E)-5,8,10-trimethyldeca-2,9-dienyl]pyrazole 4-[2-(3,3,3-trifluoropropoxy)pyridin-4-yl]-1H-pyridazin-6-one 2-[4-(5,6-difluoro-1H-benzimidazol-2-yl)-3-fluorophenoxy]-N-methoxyacetamide;1-propylpyrrolidine [5-cyclopropyl-6-(2,4-difluorophenyl)pyridin-3-yl]methanol [2-(dimethylamino)-1,3-thiazol-4-yl]-[5-(oxan-4-yl)-1H-pyrazol-3-yl]methanone (3R)-5-[3,6-bis(dimethylamino)pyridin-2-yl]oxypentan-1-amine [(3S,4R)-1-[4-(6-fluoroquinolin-4-yl)cyclohexyl]-3-hydroxypiperidin-4-yl]carbamic acid [2-(3,5-ditert-butylphenyl)-1H-pyridazine 2-(3,5-dimethylpyridin-4-yl)-N'-[(Z)-2-ethoxy-1-[[3-fluoro-4-(2-oxopyridin-1-yl)phenyl]methoxy]ethenyl]-3H-benzimidazole-5-carboximidamide 2-(2,3-dihydro-1H-inden-5-yl)-N-methylethanamine 6-amino-2-[(1,4-dimethyl-5-nitropyrazole-3-carbonyl)amino]hexanoic acid (1R,3S)-3-[[5-fluoro-2-[5-methylsulfonyl-2-(propan-2-ylamino)anilino]pyrimidin-4-yl]amino]cyclopentane-1-carboxylic acid (5S)-2-benzylsulfanyl-N-(3,4-dimethylphenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-amino-6-[(6-cyclopentyloxynaphthalen-2-yl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-azido-5-fluoro-6,7-dihydroquinoline 4-[2,3-dibromo-5-(1H-indole-2-carbonyl)phenyl]benzenesulfonamide 1-[5,8-bis(4-fluorophenyl)imidazo[1,2-c]pyrimidin-7-yl]piperidine-3-carboxylic acid 1-[[2-amino-4,5-dichloro-N-ethylsulfinyl-3-(trifluoromethyl)anilino]methoxy-ethylsulfanylmethylidene]cyclohexane-1-carboxylic acid (5R)-3-chloro-5-[4,4-difluoro-2-methylidene-5-[6-(trifluoromethyl)pyridin-3-yl]pentanoyl]-N-[1-hydroxy-7-(trifluoromethoxy)heptan-3-yl]cyclohexa-1,3-diene-1-carboxamide 2-[(3S)-1,1-dioxothiolan-3-yl]oxy-4-(7-pyridin-2-ylimidazo[1,2-a]pyridin-3-yl)benzamide [5-fluoro-2-(hydroxymethyl)phenyl]-(7-fluorospiro[3,4-dihydroisochromene-1,4'-piperidine]-1'-yl)methanone N-[3-[2-(methanesulfinamido)ethyl]phenyl]methanesulfonamide 2-[[5-(5,6-dimethyl-1H-benzimidazol-2-yl)thiophene-3-carbonyl]amino]pentanedioic acid 6-[3,4-bis(phenylmethoxy)phenyl]-2-[methyl(pyridin-2-ylsulfonyl)amino]hexanoic acid 1-[2,5-dichloro-4-(trifluoromethoxy)phenyl]ethanol 3-[4-amino-6-(trifluoromethyl)pyrimidine-5-carbonyl]-1,2-oxazol-4-olate N-[3-chloro-4-(2-diazenyl-5H-pyrrolo[3,4-b]pyridine-1-carbonyl)phenyl]formamide 2-chloro-5,6-dihydroxynaphthalene-1-carboxylic acid 4-(azidomethoxy)-N-ethyl-3-nitrobenzamide [4-(aminomethyl)phenyl]sulfonylimino-oxidoazanium 1-[(3R,4S)-4-hydroxy-3-methylpiperidine-1-carbonyl]-N'-(4-propan-2-ylphenyl)piperidine-3-carbohydrazide 5-[(Z)-2-chloroprop-1-enyl]-6,7-dimethoxy-3H-quinazolin-4-one;N'-[[5-ethynyl-2-(trifluoromethyl)phenyl]iminomethyl]-N-(6-ethylidenecyclohexa-2,4-dien-1-ylidene)hydroxylamine (3S)-N-[(Z,4R)-4,6-dimethylhept-1-enyl]-7-fluoro-3,4-bis(phenylmethoxy)-2,3-dihydrochromene-8-sulfonamide 5-amino-4-(2,4,5-trichlorophenyl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione N-[5-[3-(4,6-dimethylpyridin-2-yl)propanoyl]-1H-pyrazol-4-yl]pyrazine-2-carboxamide 4-[2,6-dinitro-N-(1,3-thiazol-5-yl)anilino]butan-1-ol 2-(7,8-dihydro-5H-pyrido[3,4-d]pyrimidin-6-ylmethyl)-3,6-diethoxyphenol (2S,3R)-5-phenyl-1-[4-(propan-2-ylamino)piperidine-1-carbonyl]piperidine-2-carboxylic acid 3-[2-(dimethylamino)phenyl]-1H-quinolin-4-one 2,5-dimethyl-4-[2,3,6-trimethyl-1-(phenylcarbamoyl)cyclohexa-2,4-dien-1-yl]benzenesulfonic acid N'-(6,7-dimethoxyquinazolin-4-yl)pyridine-3-carbohydrazide 1-[4-[(3,5-difluorophenyl)methylamino]-1H-pyrazolo[3,4-b]pyridine-3-carbonyl]-N-hexan-2-ylpiperidine-4-carboxamide [1-(4-chlorophenyl)sulfonylpiperidin-3-yl]-[2-methoxy-6-methyl-5-(triazol-2-yl)pyridin-3-yl]methanone 6-(1,2,3,4,5,6,7,8,8a-octahydroisoquinolin-9-yl)-N,N-dimethylnaphthalene-2-carboxamide 1-[3-chloro-4-(trifluoromethoxy)phenyl]-N-[2,5-difluoro-4-[5-(hydroxymethyl)pyridin-3-yl]phenyl]methanesulfonamide 4-chloro-7-(4-chlorophenyl)-3,6-dimethoxy-8-methylchromene-2,5-dione N-(2,4-dinitrophenyl)-2-methoxy-N-pyridin-3-ylacetamide 2-[2-methoxy-4-(trifluoromethyl)phenyl]-7H-purin-6-amine (3S,4R)-1-methyl-4-[2-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyridin-4-yl]pyrrolidine-3-sulfonamide 1-(3,4,5-trichlorophenyl)propan-2-one 3-bromo-7,10-dihydro-6H-benzo[a]quinolizine [(3R)-1-azabicyclo[2.2.2]octan-3-yl]-[4-[5-chloro-6-(trifluoromethoxy)pyridin-3-yl]oxypiperidin-1-yl]methanone 1,3-bis[(2E)-penta-2,4-dienyl]benzene;propane 2-[[4,5-bis(ethenyl)-1H-imidazole-2-carbonyl]amino]-3-phenylpropanoic acid 1,3-dichloro-5-[(2S)-2-methylbutanoyl]-2-propoxybenzene N-[4-methyl-5-(1-pentan-3-ylpiperidine-2-carbonyl)thiophen-2-yl]sulfonylacetamide 2-(3-methyl-1,2-oxazol-5-yl)-6-[4-(trifluoromethoxy)anilino]-1H-benzimidazole-5-carbonitrile 1,2-bis[2-(2-methoxyethoxy)ethyl]imidazole (NE)-N-[3-fluoro-2-(6-piperazin-1-ylpyridine-3-carboximidoyl)inden-1-ylidene]hydroxylamine N-(4-hydroxyphenyl)-N',N',3-trimethylbenzohydrazide 4-methoxy-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide N-methyl-3-[(4-phenylquinazolin-2-yl)amino]benzamide 1-[4-(4-propyl-N-propylanilino)phenyl]ethanone 5-[2-(trifluoromethyl)phenyl]pyrazole-1-carboxamide 3-[2,6-dimethoxy-4-(methylamino)phenyl]-7-piperidin-4-yloxyheptanal;ethane 1-[4-(6-methylnaphthalen-2-yl)sulfonylphenyl]butan-2-ol (5E)-2-(4,7-dimethyl-1,3-benzothiazol-2-yl)imino-5-[[4-[3-[2-[(Z)-hydroxyiminomethyl]pyridin-1-ium-1-yl]propanoylamino]phenyl]methylidene]-1,3-thiazolidine-4-carboxylic acid;bromide 2-methyl-N-[(4-morpholin-4-ylthian-4-yl)methyl]pyridine-3-carboxamide N-(furan-2-ylmethylideneamino)-1,3-benzothiazol-6-amine N-[(4,5-dimethylcyclohexa-1,3-dien-1-yl)methyl]-1-[2-fluoro-5-methyl-4-[(E)-2-[3-(trifluoromethoxy)phenyl]ethenyl]phenyl]ethenamine 3-[1-(5,6-diethylthieno[2,3-d]pyrimidine-4-carbonyl)piperidin-3-yl]propanoic acid 4-amino-N-methyl-6-[(1R)-2,2,2-trifluoro-1-phenylethoxy]pyridine-3-carboxamide;ethane 5-bromo-2-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-2-yl)phenol 1-methoxyspiro[3,4-dihydroisochromene-1,4'-piperidine] 3-azido-2,5,6-trimethylbenzenesulfonic acid N-[3,4-dihydroxy-1-(hydroxyamino)-1,1-dioxobutan-2-yl]-5-(2-methoxyphenoxy)pentanamide 3,3-dimethyl-1-[2-[[(Z)-pent-3-enylidene]amino]acetyl]indol-2-one 3-[6-chloro-4-(trifluoromethyl)pyridin-2-yl]-4H-1,2,4-oxadiazol-5-one 2-amino-6-[2-(4-chlorophenyl)ethynyl]-4,5-dihydropyrimidine-1-carboxylic acid 3-[(E)-[5-ethenylsulfanyl-1-methylidene-6-(methylideneamino)benzimidazol-2-ylidene]methyl]-4-hydroxycyclobutane-1,2-dione 7-benzylsulfanyl-2-[(4-chlorophenyl)methylsulfanyl]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione N-(4-chlorophenyl)-2-[[6-oxo-9-[(4-propan-2-ylphenyl)methyl]-1H-purin-8-yl]sulfanyl]acetamide [(4-methoxyphenyl)methylamino]thiourea 2-(8-phenylnaphthalen-1-yl)pyridine 7-[(2R,5S)-1,3,4-oxadiazol-2-yl]-1,3,8-triazaspiro[4.5]decan-2-one 2-N,3,6-triphenylcyclohexa-1,3-diene-1,2,4-triamine 5-[1,3-bis(2,6-dimethylphenyl)imidazol-1-ium-2-yl]-2-tert-butyl-4H-pyridin-2-ide 2,3-dimethyl-N-(4-oxo-1H-pyridin-2-yl)-1,5,6,7-tetrahydroindole-4-carboxamide 6-(5-chloropyridin-3-yl)-2H-1,3-benzoxazine 1-(4,5,6a,9a-tetrahydrodibenzofuran-3-yl)but-2-en-1-one [3-azido-2-(4-chlorophenyl)propyl]carbamic acid 1-[(4S)-4-hydroxy-5-methyl-3,4-dihydro-2H-quinolin-1-yl]propan-2-one 3-[(4S)-2,2-dimethyl-1,3-bis(trifluoromethyl)cyclopropyl]benzenecarboximidamide N-[3-(3,4-dihydro-2H-quinolin-1-yl)propyl]-5-oxo-4H-pyrazolo[1,5-a]quinazoline-3-carboxamide 6-chloro-3-ethyl-1H-pyrrolo[2,3-b]pyridine (4-bromo-2,5-dimethylphenyl)-bis[(3,5-difluorophenyl)sulfanyl]phosphane 4-[1-(2,3-dimethylcyclopenta-1,4-dien-1-yl)propan-2-ylideneamino]aniline N-[5-(methylamino)pentyl]formamide;(3E,5Z)-4-(2H-tetrazol-5-yl)hepta-1,3,5-triene 4-azidooxy-2,5-diethylaniline 4-(1,3-benzothiazol-2-yl)-5-imino-1-(pyridin-4-ylmethyl)-2H-pyrrol-3-ol 1-azido-2-[4-(chloromethyl)phenyl]benzene 2-[3-[1-[(E)-3-chlorobut-2-enyl]sulfonylpiperidin-4-yl]oxyphenyl]-6-(1H-pyrrol-2-yl)imidazo[1,2-a]pyridine 4-(2,3-dihydrofuran-5-yl)benzoic acid;hydrochloride 2-[(1R)-4,6-difluorocyclohexa-2,4-dien-1-yl]benzoic acid 2-azido-4-(2,5-dimethylpyrrolidin-1-yl)thieno[3,2-d]pyrimidine 3-[5-cyano-2-(cyclopropylamino)phenyl]-5-[1-(4,6-dimethylpyrimidin-2-yl)piperidine-4-carbonyl]benzamide [4-[2-(5-fluoropyridin-3-yl)ethynyl]phenyl]methanol 2-azido-1H-indole-3-carboximidamide 3-(4-hydroxyphenyl)-5H-thieno[2,3-d]pyrimidine-4,6-dione N-[(1,5-dimethylpyrazol-4-yl)methyl]-2-[4-[2-[ethyl-[(2R,3S)-3-hydroxybutan-2-yl]amino]prop-2-enoyl]phenoxy]acetamide 4-[2,5-bis(trifluoromethyl)phenyl]-3-chlorobenzonitrile 5-fluoro-2-(4-fluorophenyl)-6-[2-methylsulfonyl-3-[[1-(trifluoromethyl)cyclopropanecarbonyl]amino]benzimidazol-5-ylidene]-4H-pyridine-3-carboxylic acid N-(2,5-dimethylphenyl)-1-ethyl-6-hydroxy-4-methyl-3-[3-(1-phenyl-3,6-dihydro-2H-pyridin-4-yl)propyl]pyrazolo[3,4-b]pyridine-5-carboxamide 4-[(3S)-1-ethylpiperidine-3-carbonyl]-6,8-dimethylpyrido[2,3-d]pyrimidin-7-one 3-[6-chloro-2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)benzimidazol-1-yl]piperidine-2,6-dione (5Z)-2-(3,4-dichlorophenyl)imino-5-[(1-methyl-2-pyridin-3-ylindol-3-yl)methylidene]-1,3-thiazolidin-4-one 1-[(4aS,7aR)-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazin-6-yl]-2-(5-tert-butylthiophen-2-yl)ethanone 2-[4,5-bis(ethenyl)-1H-pyrrol-3-yl]-2-imino-N',N,N'-trimethylpropanediamide 3-[(3-phenylphenyl)methoxy]pyridine N-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]-2-fluoro-5-(2-methylpyridin-4-yl)benzamide (5-azidooxypyridin-3-yl)-[4-(trifluoromethoxy)phenyl]diazene 5-[2-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)ethoxy]-2H-benzotriazole 2-[3,5-dibromo-4-hydroxy-N-(5-methyldodecanoyl)anilino]-1-[(2-methylphenyl)methoxy]ethanone 2-(4-bromo-3,5-dimethylphenyl)-1,3,10-triazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-9-one 4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-(1H-pyrazol-5-yl)benzonitrile (2S)-3-[4-[[6-chloro-5-fluoro-4-[[1-[(4-methoxyphenyl)carbamoyl]cyclopropanecarbonyl]amino]pyridine-3-carbonyl]amino]phenyl]sulfanyl-2-fluoropropanoic acid 4-(4-methylphenyl)-1,7a-dihydro-5aH-isoindole 2-chloro-5,10b-dihydro-1H-isochromeno[3,4-c]pyrrole (2S,3R)-N-[2-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]cyclopentyl]-2-(difluoromethoxy)oxolane-3-carboxamide 3-[(4-azidophenyl)methyl]-5-propan-2-yl-1,2-dihydrotriazolo[4,5-d]pyrimidin-7-amine 1-(1,3-benzodioxol-5-yl)-N'-[2-(4-chlorophenyl)ethyl]butane-1,4-diamine [(3S)-2,5-dihydroxy-3-methyl-4-oxo-2,3-dihydropyrido[3,2-b][1,4]oxazepin-7-yl]-methylidene-[(E)-[3-[(Z)-4-ethynimidoylhept-3-enoxy]phenyl]methylideneamino]azanium 2-[5,5-dimethyl-4-oxo-3-(1,3-thiazol-2-yl)-6H-2,1-benzoxazin-7-yl]acetic acid (4S)-3-[2-oxo-1-phenyl-2-[(Z)-prop-1-enyl]azetidin-3-yl]sulfanyl-1,3-oxazolidine-4-carboxylic acid 4-tert-butyl-N-[(2S)-1-[5-fluoro-8-methoxy-3,7-dimethyl-2,9-bis(phenylsulfanyl)-6H-benzo[c]chromen-10-yl]pyrrolidin-2-yl]benzamide N-[3-cyclobutyl-5,6-dimethoxy-1-(2-piperidin-4-ylethynyl)indol-2-yl]methanesulfonamide;3-methylideneoxolan-2-one 1-[(4aS,5R)-5-amino-3,4a,5,6,7,8,9,10,10a-decahydro-2H-benzo[g]quinazolin-4-yl]-1-phenylbutan-1-ol 4-ethoxy-2,3-difluoro-N'-(6-fluoropyridin-3-yl)sulfanylbenzohydrazide 2-amino-N'-(dimethylaminosulfanyl)benzenecarboximidamide;5-chloro-4-[[2-hydroxyethyl(methylsulfonyl)amino]methyl]thiophene-3-carboxylic acid [(3R,4R)-3-(2,6-difluoro-4-hydroxyphenyl)-2-(2H-triazol-4-ylmethyl)-1,3,9-triazatricyclo[8.4.0.02,7]tetradeca-2(7),10,12-trien-11-yl]-(1-pyrimidin-5-ylpiperidin-4-yl)methanone (2S)-3,3-dihydroxy-N'-[(1R)-5-(2-methoxyethylcarbamoylamino)-2,3-dihydro-1H-inden-1-yl]butanehydrazide (3R)-N-[(E,1S)-4-(dimethylamino)-2,5-bis(hydroxysulfanylmethyl)cyclohex-3-en-1-yl]-7-oxo-6-phenylmethoxyheptanamide 3,5-dibutyl-1H-pyrrole-2-carboxylic acid 1-benzyl-3,7a-dihydro-2H-indazole N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]-4-(3-hydroxypropylsulfanylamino)butane-1-sulfonamide [3-[4-(3-chlorophenoxy)piperidin-1-yl]sulfonylazetidin-1-yl]-naphthalen-2-ylmethanone 1-azido-2,5-dimethyl-3-phenylmethoxybenzene (3aR,7aS)-2-[4-chloro-2-methyl-5-(2-pyrrolidin-1-ylpropan-2-ylsulfonyl)phenyl]sulfonyl-1,3,3a,4,6,7-hexahydropyrano[3,4-c]pyrrole 3-azido-1-(2-chloroethyl)pyrrolo[2,3-b]pyridine N-[3-(dimethylamino)propyl]-5-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-3-yl)furan-2-carboxamide;2,2,2-trifluoroacetic acid 2-[3-[2-(3,5-dihydroxyphenyl)ethynyl]pyrido[2,3-b]pyrazin-6-yl]oxy-N-methylacetamide 6-chloro-7-fluoro-N-[(3R)-1-[(2R,5S)-2,4,5-trimethylpiperazine-1-carbonyl]piperidin-3-yl]quinoline-8-sulfonamide (2S)-6-methyl-4,11-dioxo-5H-benzo[b][1,4]benzothiazepine-3-carboxylic acid (E)-1,2-diphenylethenol 4-cyclohexa-1,5-dien-1-yl-N-[(3Z)-hexa-1,3,5-trien-2-yl]aniline N-[(3S)-4,5-dimethyl-7-(naphthalene-1-carbonyl)-2,3-dihydro-1H-inden-3-yl]acetamide 2-[(3,5-ditert-butylphenoxy)methyl]oxirane 2-(N-carbamimidoylanilino)benzenecarboximidamide 5-[(5-bromopyrimidin-2-yl)amino]-1,3-dimethoxycyclohepta-1,4,6-triene-1,2-disulfonic acid 7-amino-N',6-dihydroxynaphthalene-2-carboximidamide 2-[4-[1,3-benzothiazol-2-yl-(5-chloropyridin-2-yl)amino]phenyl]sulfonylacetic acid 5-azidonaphthalene-2,7-diol 1-phenyl-2,3-dihydro-1H-indene 1,3-di(pentan-2-yl)benzene;ethane 4-azidooxy-3,5,6-trichloropyridine-2-carbonitrile 1-[2,6-dichloro-4-(4-fluorophenyl)sulfanylphenyl]piperidine 2-azido-5,6-dimethylbenzenesulfonamide 3-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)cyclohexan-1-one 1-[3-[(5-chloropyrimidin-2-yl)amino]pyrrolidin-1-yl]-N,N-dimethylcyclopentane-1-carboxamide 4-[[(1R)-3-methoxycyclopentyl]amino]-5-nitro-1H-pyrimidin-6-one (3-fluorophenyl)methanesulfonothioylcarbamic acid 5-tert-butyl-2-methyl-4-(3-propanoyloxy-4-pyridin-4-ylbutyl)benzoate 4-N-butyl-2-N-cyclohexylpyrimidine-2,4-diamine 1-[5-(4,4-difluorocyclohexyl)oxypyrimidin-2-yl]-N'-hydroxypyrrole-3-carboximidamide;ethane 3-[[5-(2,6-dimethoxyphenyl)furan-2-yl]methyl]quinazolin-4-one 6-[1-(cyclopropylmethoxy)isoquinolin-7-yl]quinazolin-4-amine 1-amino-3-[2-[(2R)-3,4-dihydroxybutan-2-yl]pyrazol-3-yl]sulfonylurea 2-[(1Z,3E)-1-amino-4-[4-chloro-5-[(Z)-(4-oxoquinazolin-3-yl)methylideneamino]oxy-2-(trifluoromethyl)phenyl]buta-1,3-dienyl]guanidine N-[(2R,3S)-1-amino-5-(1H-pyrazol-4-ylsulfonylmethylamino)-6-azido-3-phenylhexan-2-yl]propanamide 1-[4-[[5-[2,6-dimethyl-4-(trifluoromethoxy)phenyl]-4-ethyl-1,3-thiazol-2-yl]carbamoyl]cyclohexyl]-N,N-dimethylindazole-5-carboxamide 2-bromo-5-methyliodanuidylfuran ethane;1-(1-phenylethenyl)dibenzothiophene 3-[(2S)-6-amino-4,5-dimethyl-1-phenylhexan-2-yl]oxyaniline 2-[3,5-bis(trifluoromethyl)phenyl]-N-[3-chloro-4-(1,2,4-triazol-1-yl)phenyl]acetamide N-[2-chloro-6-(trifluoromethyl)pyridin-3-yl]-1-[2-(3,4,5-trifluorophenyl)pyridin-3-yl]cyclopropane-1-carboxamide N-(4-butylcyclohexen-1-yl)benzamide 4-[2,3-dihydroxypropyl(1,3-thiazol-5-yl)amino]-N-thiophen-2-ylbenzenesulfonamide 3-(2,4-difluorophenyl)-N'-hydroxypyridine-4-carboximidamide 5-ethyl-1,4-bis[(2-methoxyphenyl)methylideneamino]octan-3-one 3,5-dichloro-4-methoxybenzamide 4-[2-(4-tert-butylpiperidin-1-yl)ethyl]-6-phenylbenzene-1,3-diamine;dihydrochloride 5-ethyl-4-methoxy-7,8-dihydronaphthalen-2-ol 3-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]propanamide 1-(5,6-dimethoxypyridin-3-yl)-3-[5-[2-(5,6,7,8-tetrahydroquinolin-4-yloxy)ethoxy]spiro[1,2-dihydroindene-3,1'-cyclopropane]-1-yl]urea (2R)-5,8-dioxo-6-phenyloctane-2,3-dicarbonitrile 7-(cyclohexa-1,3-dien-5-yn-1-ylmethoxy)-2-(trifluoromethylsulfonyl)-3H-quinazolin-4-one N-cyclopropyl-2,6-dimethoxy-4-[(5Z)-1-pyridin-3-ylocta-5,7-dien-5-yl]aniline 2-(6-chloropyridine-3-carbonyl)piperazine-1-carboxylic acid 2-(4,5-dimethyl-1H-pyrrole-2-carbonyl)-8-fluoro-3,4-dihydro-1H-isoquinoline-6-carboxylic acid 4-[(E)-2-(2,4-dimethoxyphenyl)ethenyl]benzene-1,3-diol 4-[3-(2,4,6-trimethylphenyl)triazolo[1,5-a]pyridin-8-yl]benzene-1,3-diol 2-[5-carbamoyl-2-(4-chlorophenyl)-9-[(2,6-difluorophenyl)methyl]carbazol-4-yl]oxyacetic acid 1-(2,4-diphenylbutan-2-yl)piperidine;formic acid N-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(6R)-2-(trifluoromethyl)-6H-furo[2,3-f][1]benzofuran-6-yl]benzenesulfonamide 2-[2-ethyl-6-oxo-1-(pyridin-3-ylmethyl)pyrimidin-4-yl]-N,N'-dimethylbenzohydrazide [(2S,4R)-4-amino-1-benzylsulfonylpyrrolidin-2-yl]methanol 5-[4-(3,5-dichlorophenyl)sulfanyl-2-methoxyphenyl]-1H-imidazole;dihydrochloride 2-(3-ethylanilino)-4,7-dioxo-N-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 1-ethyl-2,5-dimethyl-3H-cyclopenta[b]naphthalene 5-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxy-N-[2-(5-thiophen-2-ylfuran-2-yl)ethyl]benzamide 4-amino-5-methyl-2-[3-(propylsulfonylamino)cyclobutyl]oxybenzoate 3-[5-(1H-azepin-4-yl)pyridin-2-yl]-N,2,6-trimethylaniline 1-(2-iodophenyl)-N-methylpiperidin-4-amine N-[3,5-bis(trifluoromethyl)phenyl]-6-chloronaphthalene-2-carboxamide N-(2,5-dichlorophenyl)-N-hexyl-2H-tetrazol-5-amine [(4-aminophenyl)sulfonyl-methoxyphosphoryl]-oxoazanium 2-[5-(2,4-dihydroxyphenyl)-1H-pyrazole-3-carbonyl]benzenesulfonic acid N-[2-(4-chlorophenyl)ethyl]-4-pyridin-3-yloxan-4-amine (3S)-N,4-dimethyl-1-[5-oxo-1-[4-(trifluoromethoxy)phenyl]pyrrolidine-3-carbonyl]piperidine-3-carboxamide 5-(N,4-dimethylanilino)isoindole-1,3-dione 1-[(2R)-4,7-dichloro-6-fluoro-5-hydroxyspiro[2.4]heptan-2-yl]-3-[5-methoxy-4-(1H-pyrrolo[2,3-b]pyridin-3-ylsulfonyl)thiophen-2-yl]urea 2,4-diphenyl-6-[4-(5,9,10,11-tetrahydrobenzo[b][1]benzazepin-7-yl)butylcarbamoyl]benzoic acid N-[1-cyclopropyl-5-(furan-3-yl)pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide ethane;4-N,4-N-dimethylbenzene-1,4-disulfonamide (2Z,3S)-1-(4-fluorophenyl)-2-[1-(4-methoxyphenyl)ethylidenehydrazinylidene]hexan-1-one (3R)-4,5,6-trihydroxy-1',2-dioxospiro[2,3-dihydrochromene-5,4'-pyrrolidine]-3'-carbonitrile N-[2,6-difluoro-4-(1H-1,2,4-triazol-5-yl)phenyl]-3-(4-methoxyphenyl)sulfanylazetidine-1-carboxamide [1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidin-2-yl]methanesulfonamide 5-ethyl-N-[(E)-(3-ethynylphenyl)methylideneamino]pyridine-2-carboxamide N-(3,5-dimethylcyclohexa-1,5-dien-1-yl)-2-ethoxy-4-fluoroaniline 2-[5-bromo-3-(4,6-dichloro-1H-benzimidazol-2-yl)indol-1-yl]-N-diazoethanimidamide 2-(azidomethyl)-6-bromopyridine 3-[2,6-difluoro-4-(oxan-4-ylmethoxy)phenyl]-5-[3-(fluoromethyl)azetidine-1-carbonyl]pyrazolo[1,5-a]pyrimidine-7-carboxamide [4-(3-chlorophenyl)piperazin-1-yl]-[6-[2,5-difluoro-4-hydroxy-N-methylsulfonyl-3-(propan-2-ylcarbamoylamino)anilino]pyrimidin-4-yl]oxyborinic acid 3-[(4aR,6S)-6-morpholin-4-yl-1,2,3,4a,5,6,7,8,8a-decahydroisoquinolin-9-yl]aniline 2-N-[1-(3,4,5-trimethoxyphenyl)ethyl]quinazoline-2,4-diamine (4-ethylpiperidin-1-yl)-[6-methoxy-2-(3,5,5-trimethylcyclohexa-1,3-dien-1-yl)quinolin-3-yl]methanone 2-(N-cyclohexyl-4-hydroxyanilino)acetamide 4-[3-amino-1-(2-methylpyrrolidin-1-yl)propan-2-yl]-N-benzylaniline;ethane (4S,9aR)-8-[[2-[6-(2-chloro-3-methoxyphenoxy)pyridin-3-yl]pyrimidin-5-yl]methyl]-1-fluoro-4-propan-2-yl-3,4,6,7,9,9a-hexahydro-2H-pyrazino[1,2-a]pyrazine 2-chloro-N-[3-[1-(diethylamino)propan-2-yl]phenyl]propanamide 1-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]-3-(2-methyl-6,7-dihydroquinolin-8-yl)urea N'-[4-[2,3-bis(ethenyl)phenyl]butanoyl]-3-methoxybenzohydrazide 4-chloro-6,7-dihydroxyquinoline-2-carboxylic acid 3-(4,7-difluorobenzoyl)benzenesulfonamide 2-chloro-3-ethyl-5,6-dimethoxy-4-piperazin-1-ylpyridine 1-(6-chloro-3,4-dihydropyridin-2-yl)-2-[[5-(2-fluorophenyl)thiophen-2-yl]methylideneamino]guanidine;2,2,2-trifluoroacetic acid 2-(cyclopropylamino)-4,5,6,7-tetrahydro-3H-azepine-8-carboxamide;3-methylsulfanyl-N-[(1R,5S)-8-oxo-3-azabicyclo[3.2.0]heptan-9-yl]benzamide 1-(2,3-difluorophenyl)-7H-imidazo[4,5-c]quinoline 3-[3-(4,4,5,5-tetramethyloxaborolan-2-yl)phenyl]benzonitrile 1-cyclopentyl-3-methyl-4,6-dioxopyrazolo[3,4-d]pyrimidine-5-carbonitrile 4-chloro-2-methoxy-5-(1,3,4-oxadiazol-2-yl)benzenesulfonamide 3-[3,5-dimethyl-1-(4-oxo-2-pyridin-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6-carbonyl)pyrazol-4-yl]-N-(furan-2-ylmethyl)propanamide 6-hydroxy-2,2-dimethyl-7-(pyrrolidine-1-carbonyl)-3H-inden-5-one 3-[1-amino-2-(3,5-difluorophenyl)ethyl]aniline (2R)-N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-1-[6-(3-hydroxypropoxy)hexanoyl]piperidine-2-carboxamide 4-[3-(dimethylamino)phenyl]-N',2,5-trihydroxybenzenecarboximidamide 4-[[5-methyl-3-(6-morpholin-4-ylpyridazin-3-yl)-1,2,4-triazol-1-yl]methoxymethyl]benzonitrile [4-[4-amino-2-(3,3-difluoropyrrolidine-1-carbonyl)phenoxy]pyridine-2-carboximidoyl]carbamic acid 4-[(2S)-3-[methyl(pyridin-2-ylsulfonyl)amino]pyrrolidine-1-carbonyl]benzoic acid N-[5-(4-chlorophenyl)sulfonyl-2-methylpyrazol-3-yl]-3,4-difluorobenzamide (3S)-1-[4,5-bis(ethenyl)-6-[3-(trifluoromethoxy)phenyl]pyrimidin-2-yl]piperidine-3,4-diol N-[1-(2,4-difluorophenyl)ethyl]-3-(furan-2-yl)morpholine-4-carboxamide 3-(ethylamino)-N,N-bis[1-methyl-6-oxo-5-([1,2]thiazolo[4,3-b]pyridin-7-yloxy)pyrimidin-2-yl]propanamide 2-chloro-1,3,4-tris(phenylmethoxy)benzene 2-[3,5-dichloro-4-[(6-oxo-5-propanoyl-1H-pyridazin-3-yl)oxy]phenyl]-6-isocyano-1H-benzimidazole-4-carbonitrile [4-(4,5-diphenyltriazol-1-yl)piperidin-1-yl]-[2-(pyrrolidine-1-carbonyloxy)phenyl]methanone (2R)-3-methyl-1,1,1-triphenylbutane-2,4-diamine N-[1-(3-methoxyphenyl)-2,2,4-trimethylpiperidin-3-ylidene]acetamide 2-(2,4-difluorophenyl)-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one 4-cyclohexyl-1-phenylmethoxypentane-2,3-dione 2-[6-(4-chlorophenyl)-7-methyl-2-oxo-1,3-dihydroimidazo[1,2-b]pyrazol-3-yl]-N-(4-ethoxyphenyl)acetamide 3-amino-N-[1-(6-chloro-5-fluoropyridin-2-yl)cyclobutyl]-2,2-dimethylpropanamide (1E,3E)-N'-[4-[(1Z,3Z)-2-aminopenta-1,3-dienyl]-5-methylcyclohex-3-en-1-ylidene]-4-(4-methylphenyl)-6-phenylhepta-1,3,5-triene-1,8-diamine (2S,4R)-2-[(3-cyanophenyl)methyl]-4-fluoropyrrolidine-1-carboxylic acid 2-(1-azido-9H-fluoren-3-yl)-5-methoxy-4-phenylmethoxypyrimidine (E)-3-[4-methoxy-3-[(2,3,5,6-tetrafluorophenoxy)methyl]phenyl]-2-sulfanylprop-2-enoic acid N-[5-chloro-2,4-dimethyl-3-(2-morpholin-4-ylethoxy)phenyl]-6-(trifluoromethyl)pyridine-3-carboxamide N-[(5S)-5-(acetamidomethyl)piperidin-3-yl]-2-propan-2-ylidene-1H-pyrimidine-6-carboxamide (7Z)-7-ethylidene-1,2-dimethylacridine 2-(9,10-dihydroacridin-1-yl)-N'-hydroxyethanimidamide N-cyclobutylformamide;7,10-dimethyltriazolo[4,5-b]anthracene;6-[(2S)-1-methoxypropan-2-yl]oxy-7-methylsulfonyl-3H-quinazolin-4-one N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-methyl-3-[(6-pyridin-4-yloxy-2,3-didehydro-1H-isoindol-5-yl)oxy]benzamide (3S)-4'-chlorospiro[1,2-dihydroindene-3,5'-imidazolidine]-2'-one 2-[3,5-dichloro-4-(6-propoxynaphthalen-2-yl)phenyl]acetic acid;2-methylpropanal 5-[[4-[4-[(4E)-2,3,6-trimethylhepta-1,4,6-trien-2-yl]phenyl]butylamino]methoxy]pentanal N-(4-chlorophenyl)-6,7-dimethyl-2-oxochromene-3-carboxamide 5-(2,4-dimethoxyphenyl)-1,3-oxazole N-[4-[(3S)-3-[[amino-[(Z)-2-aminoethenyl]amino]methylideneamino]pyrrolidine-1-carbonyl]phenyl]cyclopropanecarboxamide 2,4-dichloro-1-[5-chloro-6-[(3S)-oxolan-3-yl]oxypyridin-2-yl]-N-cyclopropylsulfonylbenzimidazole-5-carboxamide (3S)-1-[(6R)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl]pyrrolidine-3-carboxylic acid (2S,3R)-4-[(1R)-1-hydroxyethyl]-N-[[4-methoxy-6-(pyrazol-1-ylmethyl)pyridin-2-yl]methyl]-3-methylmorpholine-2-carboxamide 2-[1-[3-(4-chloroanilino)-4-oxo-5H-pyrazolo[4,3-c]pyridin-1-yl]ethylideneamino]oxyethylphosphonic acid 5-(4-cyclopropylphenyl)-3,6-dimethyl-2H-pyrazolo[4,3-c]pyridine (1S)-2,2-dibromo-N-[4-chloro-3-[5-cyano-6-(oxan-4-yloxymethyl)pyrimidin-4-yl]phenyl]cyclopropane-1-carboxamide 6-ethylsulfonyl-2-(2,3,4,5-tetramethoxyphenyl)-1H-indole (5R)-2-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-5-pyridin-4-ylcyclohexan-1-amine 2-[5-(trifluoromethyl)pyrimidin-4-yl]piperidine-1-carboxylate 1-[4-(4-phenylbutanoyl)phenoxy]propan-2-one (Z)-1-[2,6-diethyl-4-(3-phenylpropoxy)phenyl]prop-1-en-1-amine (3S)-4-[2-fluoro-3-[2-[5-(piperidin-1-ylmethyl)pyridin-2-yl]thieno[3,2-b]pyridin-7-yl]oxyphenyl]-3-hydroxybutanoic acid 1-(5-aminopyridin-2-yl)pyrrolidine-3-carboxylic acid 3-[(E)-1,2-diphenylethenyl]phenol;propane 1-(2,3-dimethylphenyl)-4H-pyrazolo[3,4-d]pyrimidine 3-[1-(5,6-difluoro-2H-indazole-3-carbonyl)piperidin-4-yl]oxybenzamide 2-(benzenesulfinyl)-N,4-dibutylaniline 4-[[6-(diethylamino)-2-hydroxy-1H-indol-3-yl]methylideneamino]benzoic acid N-[3-(4,6-dimethylpyrimidin-2-yl)phenyl]acetamide;1-ethoxy-2,4-difluorobenzene 2-(4-amino-3-methoxybenzoyl)-1,4,5,6-tetrahydropyrimidine-6-carboxylic acid [4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]-phenylmethanone N-(cyclohexylmethyl)-2,2-difluoro-3-[4-[2-oxoethanimidoyl(propan-2-ylamino)amino]naphthalen-1-yl]oxypropanamide 3-(3,4,6,7,8,9-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-9a-yl)-N'-hydroxypyrazine-2-carboximidamide 2-(2,5-dibromobenzoyl)oxyethanesulfonate 7-[4-(1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]heptanamide 1-cyclopentyl-3,4,5-trimethoxy-2-nitrobenzene 2-ethoxypropane;3-(6-oxo-1H-pyridine-2-carboximidoyl)benzenecarboximidamide N-(2-chlorophenyl)-3-methyl-5,6,7,8-tetrahydrothieno[3,4-c]oxepin-9-amine (3Z)-4-chloro-2,5-difluorohexa-1,3,5-triene;4-[2-[cyclopropylmethyl(methyl)amino]ethoxy]pyridine-2-carbonitrile 5-fluoro-2,6-dimethyl-4-(trifluoromethoxy)pyridine 1-[(2S,4R)-5-amino-2-azidooxan-4-yl]pyrimidine-2,4-dione 6-amino-4-methyl-2,4-diphenylpyridine-3-carbonitrile 4-(2,6-difluorophenyl)-5-methoxycarbonyl-3,6-dihydro-2H-pyridine-1-carboxylate [1-(4-fluorophenyl)triazol-4-yl]carbamic acid 6-[[[1-(cyclopropylmethyl)triazol-4-yl]-deuterio-phenylmethoxy]methyl]-2,3-dihydrochromen-4-one N-(3,5-dichlorophenyl)-4-[6-(oxolan-2-ylmethoxy)pyridine-3-carboximidoyl]piperazine-1-carboxamide N-[6,8-dichloro-2-(2-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]-4-methoxybenzamide N-(3,5-dichloropyridin-4-yl)-3-[1-[1-[(E)-4-[ethenyl(methoxy)amino]but-2-en-2-yl]pyrazole-3-carbonyl]piperidin-4-ylidene]propanamide;N-methylmethanesulfonamide 4-(7,8-diazabicyclo[4.2.0]octa-1,3,5-trien-7-yl)benzoic acid N-[4-(2,3-dihydro-1H-inden-2-ylamino)butan-2-yl]formamide;N-methylpropan-1-amine;[6-(2-methylpropoxy)-2,3-dihydropyridin-5-yl]methanol 4-[(3S,4R)-1-[2-methoxyethyl(methyl)amino]-3,4-dimethylpyrrolidine-3-carbonyl]benzonitrile;hydrochloride 3-[3-hydroxy-5-(2-methylpentan-2-yl)phenyl]propanenitrile 2,3-dihydro-1H-pyrrolo[2,3-b]pyridin-5-yl-(4-imidazol-1-ylphenyl)methanone (4S)-1,3,3-trimethyl-N-[4-methyl-2-(6-oxo-1H-pyridin-3-yl)phenyl]-7-(3,4,5-trimethoxyphenyl)-4,8-dihydropyrazolo[3,4-e][1,4]thiazepine-4-carboxamide 6-(5-ethenylpyridin-3-yl)pyrido[2,3-b]pyrazine 2-amino-N-(4,5-dimethoxypyrimidin-2-yl)-6-methylpyrimidine-4-carboxamide 3-methyl-1'-(pyridine-4-carbonyl)spiro[6,7-dihydroimidazo[2,1-c][1,2,4]triazine-8,3'-pyrrolidine]-5-one;2,2,2-trifluoroacetic acid N-(6-butyl-4,5,7,8-tetrahydrothieno[2,3-d]azepin-2-yl)-3-methoxy-2-(4-methylphenyl)propanamide 1-[5-(3,4,6,7,8,8a-hexahydro-2H-pyrrolo[1,2-a]pyrazin-1-yl)-3-fluoropyridin-2-yl]ethanone;dihydrochloride 3-(hydroxymethyl)oxolane-2,4-dione;1-[[(E)-4-methoxybut-2-en-2-yl]amino]anthracene-9,10-diol [(3S,4R)-4-hydroxy-1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-yl]-thiomorpholin-4-ylmethanone (3S,4R)-1-[4-cyano-3-(trifluoromethyl)phenyl]-4-(2-phenylethynyl)pyrrolidine-3-carboxamide (5S)-1-[4,6-bis(ethenyl)pyridin-2-yl]-4,7-dimethyl-8-oxatricyclo[10.3.0.03,9]pentadeca-1(12),3(9),4,6,13-pentaene 2-[(1S,3R)-3-aminocyclopentyl]-4-methoxybenzamide 1-cyclopropyl-3-ethenyl-2-methoxy-4-(4-methylphenyl)benzene N-cyclohexylsulfanyl-2,4,6-trimethoxyaniline 2-[[(1,3-dioxoisoindol-2-yl)methoxycarbonylamino]methyl]piperidine-4-carboxylic acid 4-methyl-2-[1,3]thiazolo[5,4-c]pyridine-6-sulfonamide 5-(2-diazohydrazinyl)-2,3-dihydrochromene-4-thione N-[2,3-difluoro-4-[6-methoxy-7-(piperidine-1-carbonyl)quinolin-4-yl]phenyl]benzenesulfonamide 3-(4-fluorophenyl)-5,6-dimethyl-1H-pyrimidine-2,4-dione N-(3,4-dimethoxyphenyl)-5-ethyl-7-oxo-2-propan-2-ylsulfanyl-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide (NE)-N-[[1-(4-cyclopropylphenyl)cyclopentyl]methylidene]hydroxylamine 2-(3-chloropyridin-4-yl)benzoic acid 2-[4-[(6R)-1-azido-3,6-dimethyl-5,6-dihydro-4H-pyrano[2,3-c]pyrazol-4a-yl]phenyl]-N-ethylacetamide 6,8-dibromo-9-ethylnaphtho[2,1-b]oxirene (2R)-3-[1-(2,3-dihydropyridine-4-carbonyl)piperidin-2-yl]oxy-N-hydroxypropanamide 6-[5-(3,4-dichlorophenyl)furan-2-yl]-N-ethylsulfanylhexanamide N-[3-[(6-oxo-4-propyl-1H-pyrimidin-2-yl)sulfanyl]propyl]imidazo[1,2-b]pyridazine-2-carboxamide 5-fluoro-2,4-diiodophenol 5-chloro-4-[3-[(2,2-difluoroethylamino)methyl]phenyl]pyridine-2-carboxylic acid 3-(3,4-dihydronaphthalene-2-carbonylamino)propanoic acid 4-azidooxy-1,2,5-tris(methylsulfonyl)benzene 3-(1H-indole-2-carbonyl)benzohydrazide 1-cyclopropylsulfinyl-4-nitrobenzene (5R,6S)-4-bromo-1-(2-methylpropyl)-3-azabicyclo[3.1.0]hexane;1-(7-chloroimidazo[1,2-a]pyridin-2-yl)ethanone (2S,4R)-1-[(2S)-2-[[(2R)-2-aminopropanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide;hydrochloride 1-azidooxy-3,5-dimethyl-2-phenoxybenzene 1-[2-(2,5-difluorophenoxy)-5-methylsulfonylphenyl]pyrrolidine 2-[[4-(pyridin-3-ylamino)thieno[3,2-d]pyrimidin-6-yl]methyl]benzoic acid 1-(3,5-dichlorophenyl)ethanethiol;ethane [2-(hydroxymethyl)piperidin-1-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)methanone 2-[(5R)-3-methyl-1,4-diphenyl-6,7-dihydropyrazolo[3,4-e][1,4]thiazepin-5-yl]phenol 4-azidooxy-N,3-dimethylnaphthalene-2-carboxamide 3,4-dichloro-N-[2-(1H-pyrrolo[2,3-b]pyridin-5-yl)ethyl]benzenesulfonamide 4-bromo-2,6-dichloro-N-[(E)-(2,3-dihydroinden-1-ylidenehydrazinylidene)methyl]benzamide 1-(4,6-dimethylpyridin-3-yl)-3-[1-[(2R)-1-hydroxybutan-2-yl]-7-(1H-pyrazol-5-yl)benzimidazol-2-yl]urea 2-N,4-N,6-tributyl-1H-pyridine-2,4-dicarboxamide 5-[(2,3-dihydro-1H-inden-5-ylamino)methyl]-N'-hydroxypyridine-2-carboximidamide 4-[2-(dimethylamino)ethyl]spiro[8H-1,6-naphthyridine-5,1'-cyclopropane]-7-one (NZ)-N-[4-(2,2-dimethylpropanoyl)-6-phenyl-1H-pyridin-2-ylidene]benzenesulfonamide 7-methyl-5-phenyl-3H-pyrido[4,3-d]pyrimidin-2-one 1-(2,3-dihydro-1H-inden-5-ylsulfonyl)-N'-hydroxy-2,3-dihydroindole-6-carboximidamide 3-(1,4-diaminobutyl)-8-fluoro-2H-isoquinolin-1-one 5-(2-fluoro-3,4-dimethoxyphenyl)imidazolidine-2,4-dione 6-amino-4-[2,5-dimethyl-3-nitro-4-(trifluoromethoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 3-(2,6-dimethoxyphenyl)-4-[2,5-dimethyl-1-[(Z)-prop-1-enyl]indol-3-yl]pyrrole-2,5-dione;ethane 4-[2,6-bis(trifluoromethyl)phenyl]-N-[5-cyano-6-(1H-tetrazol-5-yl)pyridin-3-yl]butanamide 5-(4-tert-butyl-2,6-dimethoxyphenyl)-5-methyl-7H-imidazo[1,2-a]imidazole 4-amino-2-[(1S)-1-cyanoethyl]phthalazin-1-one 4-(3,5-difluorophenyl)-1-[2-(hydroxymethyl)prop-2-enoyl]piperidine-4-carbonitrile 5-(3-bromophenyl)-1,2-dimethyl-4-[(6-pyrrolidin-3-yloxypyridin-3-yl)methylidene]pyrazol-3-one 4-[N'-[2,6-dichloro-4-(trifluoromethyl)phenyl]carbamimidoyl]benzamide 1-[4-(2-methoxypyridine-3-carbonyl)piperazin-1-yl]-2-morpholin-4-ylethane-1,2-dione 2-[3-ethenyl-4,5-bis(sulfanylidene)imidazolidin-1-yl]-6-propan-2-yloxypyridine-3-carboxylic acid N-[3-methoxy-4-(oxolan-2-yl)phenyl]-1,5-dihydrotetrazolo[1,5-a]quinazolin-7-imine (Z)-3,7,7-trimethyl-6-[2-[(5-phenylpyridin-2-yl)amino]ethoxy]oct-4-enoic acid (2S)-3-[4-amino-1'-[(E,2R)-2,4-dimethylpent-4-enoyl]spiro[indole-3,4'-piperidine]-5-yl]-2-methoxypropanoic acid;hydrochloride 4-[[4-hydroxy-5-[(2-oxo-1,3-dihydroindol-6-yl)iminomethyl]-1,3-thiazol-2-yl]amino]benzenesulfonamide N-ethyl-4-(trifluoromethoxy)benzamide;3-fluoroaniline 4-[2-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]-N-octylanilino]benzenesulfonic acid 4-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-methoxy-N-[6-(4-propan-2-ylpiperazin-1-yl)pyridin-3-yl]thiophene-2-carboxamide N-[1-(5-ethylthiophene-3-carbonyl)piperidin-4-yl]-N,2-dimethyloxane-4-carboxamide 4-N-azido-5,6-dihydropyrrolo[2,3-d]pyrimidine-2,4-diamine 3-azido-2-(1H-benzimidazole-2-carbonyloxy)propanoic acid N-(4-fluorophenyl)-3-methoxy-2-[2-oxo-2-[1-(trifluoromethylsulfonyl)piperazin-2-yl]ethyl]sulfanylbenzamide 4-(7,8,10,11-tetrahydropyrido[3,2-b]xanthen-11-yl)phenol 3-hydroxy-N'-[(E)-(2-hydroxyphenyl)methylideneamino]pyridine-4-carboximidamide N-[(2S)-3-methylbutan-2-yl]isoquinoline-7-carboxamide 3-(4-methylpiperazin-1-ium-2-ylidene)-7,10-dihydroanthracene-9,10-dione;bromide 4-[3,5-bis(4-fluorophenyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile N-[4-(2,3-dihydro-1H-indazol-6-ylamino)phenyl]-6-[(E)-1-pyridin-2-ylprop-1-en-2-yl]pyridine-3-carboxamide N-(3,4-dimethoxyphenyl)cyclopropanecarboxamide 4-[2-fluoro-5-(5-methoxy-1,2,3,4-tetrahydroisoquinolin-6-yl)phenyl]-6-methoxyquinoline-3-carbonitrile 2-bromo-4,5,6,7-tetrahydrothieno[3,2-c]pyridine N-[(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylamino)methyl]-1H-pyrazole-5-carboxamide;dihydrochloride 1-N'-(3,4-dimethylphenyl)-1-N',1-N'-diethylethene-1,1-diamine 4-fluoro-N-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]-1H-pyrrole-2-carboxamide [4-(4-chlorobenzoyl)phenyl]methoxy-cyclopropylphosphinic acid N-ethenylsulfonyl-2,4,6-trimethyl-N-(5-nitro-1,3-thiazol-2-yl)benzenesulfonamide 1-N,4-N,5-N,4-N-tetrakis(3-chlorophenyl)benzene-1,4-diamine N-[4-(3,5-difluorophenyl)sulfanyl-2-nitrophenyl]acetamide [2-[4-(6,7-dihydrothieno[3,2-c]pyridin-4-yl)piperidine-1-carbonyl]pyrrolidin-1-yl]-phenylmethanone [(3R)-2,6-dihydroxypiperidin-3-yl]methylidene-[(E)-7H-pyrrolo[2,3-d]pyrimidin-4-yl(thieno[3,2-b]pyridin-5-yl)methylidene]azanium ethane;N-[4-[3-(morpholine-4-carbonyl)phenoxy]phenyl]quinoxaline-6-sulfinamide 4-N-[2,3-bis(ethenyl)phenyl]benzene-1,4-dicarboxamide;ethane N-(2,5-dichlorophenyl)-2-ethoxy-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]acetamide 6-[(2S,4R)-4-hydroxy-2-propan-2-ylcyclopentyl]-5-methoxypyridine-3-carboxylic acid N-(3,4-dihydropyridin-6-yl)-5-[1-hydroxy-2-methyl-3-[1-(2-phenoxyethylamino)ethenyl]phenyl]furan-2-carboxamide N-[(3R,4S)-1-benzyl-3-hydroxypiperidin-4-yl]-2-(1H-indole-5-carbonylamino)pyridine-4-carboxamide;hydrochloride 5-[2-azido-1-(3,4-dimethoxyphenyl)ethyl]-N'-pentan-3-yl-7H-pyrrolo[2,3-d]pyrimidine-2-carbohydrazide 5-[1-(azidomethyl)cyclohexyl]oxybenzene-1,3-dicarboxylic acid (5Z)-2-cyclohexylimino-5-[[4,6-dioxo-1-propan-2-yl-2-[(Z)-(4-propoxyphenyl)methylidenehydrazinylidene]-1,3-thiazinan-5-yl]methylidene]-1,3-thiazolidin-4-one [4-(5-bromopyrimidin-2-yl)oxypiperidin-1-yl]-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)methanone N-[2-amino-5-(3,3-difluoropyrrolidine-1-carbonyl)phenyl]-4-fluorobenzamide 2-[1,3-benzodioxol-5-yloxy(methyl)amino]ethanol (3-ethoxyphenyl)-[4-(2-methylsulfonylethylamino)phenyl]methanone 1-[5-(trifluoromethyl)pyrazin-2-yl]piperidine-4-carboxylic acid 1-[[3,5-bis(trifluoromethyl)phenyl]methoxy]cycloheptan-4-one N-[3-(dimethylamino)phenyl]-2,3,4,5-tetrahydropyridin-6-amine 3-amino-2-[1-[(2,4,5-trifluorophenyl)methyl]pyrazolo[3,4-b]pyridin-3-yl]prop-2-enenitrile;ethane N-methyl-N-[(2Z)-2-prop-1-en-2-ylpenta-2,4-dienyl]quinoline-3-carboxamide (5Z)-2-(4-bromophenyl)imino-5-[[3,5-diiodo-4-[(4-nitrophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one N-[(1S,2R)-3-oxocyclopentyl]-5-(6-oxohexanoylamino)thiophene-3-carboxamide 3-amino-N-(2-fluorophenyl)-4-hydroxybenzamide;propane (E,2S)-1-[(4aS,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-4-[3-chloro-5-(trifluoromethoxy)phenyl]but-3-en-2-ol 2-[5-[(E)-3-[(4R)-4-[hydroxy-(6-iodonaphthalen-2-yl)amino]piperidin-1-yl]prop-1-enyl]pyridin-2-yl]benzonitrile N-(5-azido-4-fluoro-2-methylphenyl)-1,2,3,6-tetrahydropyridine-5-sulfonamide 1-(4-tert-butylphenyl)-2,3,3a,4,5,6,7,7a-octahydropyrrolo[2,3-b]pyridine 4-(azidomethyl)-2-chloro-1-[(4-fluorophenyl)methoxy]benzene 2,4-dimethyl-3-[(5-methyl-1H-pyrazol-4-yl)sulfonylamino]benzoic acid 3-chloro-5-(ethylamino)benzoic acid 3-azidooxypropylsulfinylbenzene 4-(cyclohexylmethoxy)benzoate N-[(1R,2S)-2-hydroxycyclohexyl]-7-methoxy-6-pyrrolidin-1-ylquinoline-4-carboxamide 3-N,4-N-bis[2,6-di(propan-2-yl)phenyl]pyrazine-1,3,5-triamine N-(5-methyl-2-nitrophenyl)-N-pyridin-3-ylethenesulfonamide 4-N-[2,4-difluoro-5-(3-morpholin-4-ylazetidine-1-carbonyl)phenyl]-7-methoxythieno[3,2-d]pyrimidine-6-carboxamide;ethane 6-N-[2-(dimethylamino)ethyl]-5,7-dihydroxy-3-[1-[4-(2-phenylquinolin-5-yl)piperidin-1-yl]ethenyl]chromene-4,6-dione 5-[4-fluoro-3-[7-(1-methylpyrazol-4-yl)-3H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl]-N,N-dimethylpyridin-3-amine (2S)-1,2-dibutylpyrrolidine;N-[4-(5-methoxypyridin-3-yl)phenyl]cycloheptanesulfonamide N-[(Z)-3,4-dichlorohex-2-enyl]sulfanylpropanamide;ethane 4-[3-(2-bromophenyl)phenyl]-6-chloro-2-sulfanylidene-1H-pyrimidine-5-carbonitrile N-[3-[4-amino-5-(1,5-dimethylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]phenyl]-4-fluorocyclohexa-1,5-diene-1-carboxamide (7S)-6,8-diphenyl-N-(1-methylpyrazol-4-yl)-5H-imidazo[1,2-a]pyrimidine-7-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]formamide;5-chloro-2-hydroxy-4-phenylbenzonitrile 5-butoxy-2-[3,4-dichloro-6-(difluoromethylsulfanyl)-9H-pyrido[2,3-b]indol-8-yl]benzonitrile 5-(4,6-diphenylpyridin-2-yl)-3-methyl-1,8a-dihydroquinoxaline N-[5-chloro-2-(5-propanoylthiophen-3-yl)phenyl]formamide;methoxyethane 5-amino-4-(2,6-difluoro-3-methoxyphenyl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione (5-ethyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)hydrazine 3-[(5-chloropyridin-2-yl)methoxy]-1H-indole 2-[[4-(2,6-dimethylanilino)-1,3,5-triazin-2-yl]sulfanyl]-N-phenylacetamide 2-(4-methoxyphenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxylic acid 2-amino-N'-[4-cyano-3-(trifluoromethyl)phenyl]-1H-imidazole-5-carboximidamide 3-[2,4-bis(trifluoromethyl)phenyl]-5-[[2-ethoxy-6-(trifluoromethoxy)benzoyl]amino]benzoic acid N-[2-(diethylamino)ethyl]-1,3-benzothiazole-6-carboxamide (E)-1,3-bis[4-(hydroxymethyl)-2,6-dimethoxyphenyl]prop-2-en-1-one 2,4-dimethyl-6-[3-(5-pyridin-2-yl-1H-pyrrol-3-yl)-1,2,4-oxadiazol-5-yl]phenol (2S,3R)-N-[6-cyano-4-(trifluoromethyl)pyridin-2-yl]-1-[(2,5-difluorophenyl)methyl]-2-(1H-pyrazol-4-yl)pyrrolidine-3-carboxamide N-[(2-phenylphenyl)carbamoyl]propanamide N-[5-[6-fluoro-3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclopentanecarboxamide 2-[4,5-dimethyl-N-(3-nitrophenyl)-2-phenyldiazenylanilino]acetic acid 5-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]imidazolidine-2,4-dione 3-azidooxy-N'-[2-(trifluoromethyl)phenyl]propanehydrazide 2-[[4,5-dimethyl-3-(4-piperidin-1-ylsulfonylphenyl)pyrazole-1-carbonyl]amino]acetic acid (3-benzylsulfanylphenyl)methanimine 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-3,3-bis(fluoromethylsulfanyloxy)-4H-indole N-(5-fluoropyrimidin-2-yl)-1,3-benzothiazol-6-amine 2-[(4,6-dimethylpyridin-3-yl)amino]-N'-hydroxypyrimidine-5-carboximidamide 5-[2,6-difluoro-4-(methoxysulfanylamino)phenyl]-1H-pyrrole-3-carboxamide;N-propan-2-ylformamide 4-[1-(2-methylpropyl)pyrazole-3-carbonyl]piperidine-2,6-dione 1-[(4aS,7aS)-6-methyl-4a-(pyridine-2-carbonyl)-3,4,5,7,7a-hexahydro-2H-pyrrolo[2,3-c]pyridin-1-yl]propan-1-one N-(4,5-dichloropyridin-2-yl)-2-[3-methoxy-4-[1-oxo-6-(trifluoromethyl)-3H-isoindol-2-yl]phenyl]acetamide 5-[(2,6-difluorophenyl)methyl]-N-[[4-(propan-2-ylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-a]pyridine-3-carboxamide 3-fluoropyridine;1,2,4,5-tetrafluoro-6-(5-fluoropentoxy)-3-phenylbenzene 5-(4-tert-butylphenyl)-3-methoxy-1-(2-methoxyethoxy)-2H-pyridine (4aS,8aR)-N-[2-(3,5-dichlorophenoxy)ethyl]-6-methylsulfonyl-2,3,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridine-4-carboxamide 2-methyl-4-[[(1S)-3-methyl-1-[6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)pyridine-3-carbonyl]oxybutyl]amino]pentanoic acid;dihydrochloride 3-chloro-2-methyl-6-(trifluoromethoxy)phenol 3,4-dimethyl-1-(3,4,5-trimethoxyphenyl)-4H-pyridazine 6-(4-fluorophenyl)-N-[4-(2-hydroxyethylamino)sulfanylphenyl]pyridine-3-carboxamide (2R,4S)-1-[3-chloro-4-(pyridin-4-ylmethoxy)phenyl]sulfonyl-N-hydroxy-4-morpholin-4-ylpyrrolidine-2-carboxamide [2-(4-aminophenoxy)pyridin-3-yl]methanol 2-[(2,3,6,7-tetramethoxynaphthalene-1-carbonyl)amino]acetate 2-aminopyrazolo[1,5-a]pyridine-3-carboxamide;N-cyclohexyl-4-propan-2-ylbenzamide 4-bromo-2,5-dimethyl-N-[(4Z)-3-(4-methylphenyl)hepta-1,4,6-trien-2-yl]aniline;ethane 7-[3-(aminomethyl)-1,2,4-oxadiazol-5-yl]isoquinoline-1-carboxamide 2-amino-6,7-dihydrobenzo[d][1]benzoxepine-3-carboxylic acid;hydrochloride N-[4-amino-1-(2-phenylethyl)piperidin-3-yl]-2-ethynoxybenzamide 2-[2-chloro-4-(3,7-dimethylocta-2,6-dienoxy)phenyl]-N-(4-ethylsulfanylphenyl)ethanethioamide [2,6-di(butan-2-yl)phenyl]-[[2,6-di(propan-2-yl)phenyl]iminomethyl]azanide;molybdenum(2+) N'-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carbohydrazide (3R,4S)-1-benzyl-N-[3-(diethylaminomethyl)phenyl]-4-propan-2-ylpyrrolidine-3-carboxamide;hydrochloride (3R)-1'-[6-cyano-5-fluoro-4-[2-methylpropyl(methylsulfonyl)amino]pyridin-2-yl]-7,10-dioxospiro[4H-pyrido[1,2-a]quinoxaline-3,4'-piperidine]-2-carboxamide 5-(4,6-dimethyl-3,5-disulfophthalyl)oxycarbonylbenzene-1,3,3-tricarboxylic acid N-[(2S)-1-(1H-indol-3-yl)-1-oxopentan-2-yl]propane-1-sulfonamide 3-[(E)-5-ethylsulfanylpent-4-enoxy]-1H-quinolin-2-one [3-hydroxy-4-methyl-2,6-di(propan-2-yl)phenyl]carbamic acid 5-(1,3-benzodioxol-4-yl)-N-[2-methoxy-6-(trifluoromethyl)pyridin-3-yl]-6-methyl-1H-pyrrole-3-carboxamide 2-[4-[1-(2-methoxyethyl)indole-3-carbonyl]piperidin-1-yl]acetamide 2-[[4,7-dibromo-5-(3-hydroxyphenyl)iminopyrazolo[1,5-a]pyrimidin-6-ylidene]methyl]-5-hydroxypyran-4-one [2-amino-1-(4-hydroxyphenyl)-2-oxoethyl]phosphonic acid N-[[2,4-difluoro-3-(methylamino)phenyl]methyl]-N'-methanimidoyl-3H-pyrrole-5-carboximidamide 1-chloro-3,5-bis(2-chlorophenyl)benzene;ethane N-[1-methoxy-5,6,7-trimethyl-4-oxo-8-(2,3,6-trifluorophenyl)naphthalen-2-yl]propanamide N-[1-cyclohexyl-2-oxo-2-[4-[(2,3,6,7,8,9-hexahydroimidazo[4,5-h]isoquinolin-5-ylamino)methyl]phenyl]ethyl]-3H-benzimidazole-5-carboxamide 2-azido-1,3,5-tris(chloromethyl)benzene (1S,3R)-2,2-dichloro-N-[4-chloro-3-[2-[5-methyl-6-(3,3,3-trifluoropropoxy)pyridin-3-yl]acetyl]phenyl]-3-(3,4,5-trichlorophenyl)cyclopropane-1-carboxamide N-[5-(4-methoxyphenyl)sulfanyltetrazolo[1,5-a]quinolin-7-yl]formamide 2-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonylamino)-1-cyclopentyl-5,6,7,8-tetrahydroimidazo[4,5-c]azepine-8-carboxylic acid;dihydrochloride N-[[(3S,4R)-1-(benzenesulfonylmethyl)-3-fluoropiperidin-4-yl]methyl]ethenesulfonamide (4R)-2-[6-oxo-1-[1-phenylpropan-2-yl([1,3]thiazolo[5,4-b]pyridin-5-yl)amino]pyrimidin-5-yl]oxy-4-[2-[4-(trifluoromethyl)pyrazol-1-yl]ethyl]cyclopentane-1-carboxylic acid (2S,3R)-4-[2-(5-amino-1H-imidazol-2-yl)piperidin-1-yl]-N-[2-methoxy-5-(1-propan-2-ylpyrazol-4-yl)pyridin-3-yl]-2,3-dihydroxybutanamide;ethane 2-[4-(1H-indol-3-ylmethyl)piperazin-1-yl]-6,7-dihydro-5H-cyclopenta[d]pyrimidine 5-chloro-1'-[(2,4-difluorophenyl)methyl]spiro[3H-indole-2,4'-piperidine] 2,4-dichloro-1-[(3Z)-penta-1,3-dien-2-yl]benzene;ethane 1-(6-chloro-3,4-dihydro-2H-quinolin-1-yl)pentan-1-one 3-N,4,8-trihydroxynaphthalene-2,3-dicarboxamide 2-[4-(1,3-benzodioxol-5-ylmethoxy)phenyl]acetamide N-[4-(2,6-dimethoxyphenyl)-5-(2-hydroxypropan-2-yl)-1,3-thiazol-2-yl]-6-formamidopyrazine-2-carboxamide 6-(2,5-dichlorophenyl)-4-oxopyran-3-carbonitrile N-[4-chloro-5-(2,3-dimethylbutanoylamino)pyridin-2-yl]pyrrolidine-1-carboxamide 7-[3,5-dichloro-4-(2,2,2-trifluoroethoxy)phenyl]-N-(1,3-dihydroinden-2-ylmethyl)-6-oxo-2-thia-5,7,11-triazatricyclo[6.3.1.04,12]dodeca-1(11),8(12),9-triene-3-carboxamide N-[(3,5-dimethyl-1H-pyrazol-4-yl)methylidene]hydroxylamine (2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-phenylcyclopropane-1-carboxamide 4-cyclopropylimino-5-(2,3-dichlorophenyl)imidazolidin-2-one 5-[(2,3-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-one N-cyclohexyl-4-(3,5-dimethylphenyl)aniline N-[4-[(Z)-[2-(4-ethylphenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]-1,3-thiazol-2-yl]-6-hydroxy-2,3,4,9-tetrahydro-1H-carbazole-3-carboxamide 4-azidooxy-1,3-dichloro-2-(trifluoromethylsulfonyl)benzene 2-(2,4-dimethylphenoxy)-N-[(Z)-1H-indol-3-ylmethylideneamino]acetamide 1,4-ditert-butyl-2-(3-chlorophenyl)benzene N-[1-(furan-2-yl)ethenyl]-6-methyl-3,4-dihydroisoquinoline-1-carboxamide 4-(benzylamino)-N,6-bis(pyridine-3-carbonylamino)pyrimidine-5-carboxamide 1-[3,5-difluoro-2-(triazol-2-yl)phenyl]-4-methoxypiperidine (5R,6R)-3-[[3-fluoro-4-[4-hydroxy-2-methyl-4-(trifluoromethoxy)piperidine-1-carbonyl]phenyl]methyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraene-12-carboxylic acid 4-methyl-6,8-dipyridin-2-yl-1H-imidazo[4,5-f]purine (Z)-N',2-bis[3,5-difluoro-4-(trifluoromethyl)phenyl]ethenedithioamide N-[4-(2,6-dimethylmorpholin-4-yl)-3-fluorophenyl]-5-[2-[(1S)-1-methoxyethyl]pyrrolo[1,2-b]pyridazin-7-yl]-2-methylpyridine-3-carboxamide 1-N,5-N-bis(4-methylphenyl)-9H-fluorene-1,5-disulfonamide 1-[(2,3-difluorophenyl)methyl]-5-ethoxy-4-iminoimidazolidin-2-one 2-[4-[2-(8-methylimidazo[1,5-a]pyridin-3-yl)acetyl]piperazin-1-yl]benzamide 1-ethylsulfanyl-2,3-bis(4-fluorophenyl)-1H-indene [1-[2-(2,6-difluorophenyl)ethyl]pyrazol-3-yl]-(4-methoxypiperidin-1-yl)methanone (Z)-3-[3-(dimethylamino)phenyl]but-2-enal 2-ethenyl-N,5-dimethyl-1H-imidazole-4-carboxamide;3-(2-formamido-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl)-N-[3-fluoro-4-[(2E,4Z)-3-(hydroxycarbamoylamino)penta-2,4-dienimidoyl]phenyl]benzamide 2-[3,5-bis(trifluoromethyl)phenyl]-N-[(E)-(4-nitropyridin-1-ium-1-ylidene)amino]sulfonylacetamide 2-(2-methyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl)-1H-benzimidazole 5-methyl-N-[(2S,3R)-1-oxo-6-phenyl-4-(3,3,3-trifluoropropylamino)-1-(2,2,2-trifluoroethylamino)hexan-2-yl]-1H-indole-2-carboxamide (E)-2-cyano-3-[4-[(2R,6S)-1-ethyl-2,6-dimethylmorpholin-4-ium-4-carbonyl]phenyl]prop-2-enoic acid 3-cyclohexyl-N'-[5-(difluoromethoxy)pyridin-2-yl]-3-hydroxypropanimidamide 2-[4-azidooxy-1-(2,6-difluorophenyl)butyl]-1,3,5-trimethoxybenzene 2-[2,4-bis(ethenyl)phenyl]sulfonylpropanoate 5-[(2,5-dimethylpyrrol-1-yl)methyl]-3H-1,3,4-oxadiazol-2-one 1-ethenyl-2,3-bis(ethenoxy)-4-[(Z)-prop-1-enyl]naphthalene 3-methyl-5-[(E)-2-thiophen-2-ylethenyl]benzamide 2-amino-3-[4-[(6R)-6-(3,5-dichlorophenyl)-1,4-oxazepan-7-yl]pyrimidin-5-yl]propanoic acid 3-bromo-N'-hydroxy-5,6-dimethylpyridazine-4-carboximidamide 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(6,7-dihydropyrrolo[1,2-a]imidazole-2-carbonyl)-2,3,3a,4-tetrahydroindol-1-yl]acetamide (Z)-N'-[2-amino-5-fluoro-4-(methylaminosulfanyl)phenyl]-1,3-diphenylprop-2-enimidamide 1-(3,5-difluorophenyl)-N-[2-fluoro-6-methyl-4-[4-(trifluoromethoxy)anilino]phenoxy]cyclobutane-1-carboxamide;ethane 3-(3,4-dimethylpiperazin-1-yl)-N'-hydroxypyridazine-4-carboximidamide 2-[4-(2,5-difluorophenyl)-1H-imidazole-5-carbonyl]-N-[3-[(dimethylamino)methyl]oxan-4-yl]pyrrolidine-1-carboxamide (1R,2R)-2-[4-[(E)-3-cyclobutyl-1-hydroxyprop-1-enoxy]phenyl]-N-[2-fluoro-5-(trifluoromethoxy)phenyl]sulfonyl-1-methanehydrazonoyl-3-oxo-N-propan-2-ylazetidine-2-carboxamide N-(1,3-benzodioxol-5-ylmethyl)-N-ethanimidoylthieno[2,3-b]quinoline-7-carboximidamide 7-[6-(4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]quinoline N-[5-[2-amino-4-(hydroxymethyl)-5,6-dihydro-1,3-thiazin-4-yl]-4-chloropyridin-2-yl]formamide 5-[(E)-2-ethenylhex-1-enyl]-3-methoxyquinoxalin-6-amine ethane;N-[2-(hydroxymethyl)cyclohexyl]-2-pyridin-3-ylacetamide 2-[2-(dipropylamino)ethoxy]-1,5-dimethylpyrazole-3-carboxylic acid 1-(2,6-difluorophenyl)-5-methylhexane-1,3-dione;ethene 5-azido-1,3,4-trimethylindole 2-(3,4-dichlorophenyl)-N-[4-[5-ethyl-1-(prop-2-ynylaminomethyl)pyrazol-4-yl]pyridin-2-yl]acetamide 5-[(1S,2R)-2-aminocyclohexyl]oxy-2-benzyl-3-methanimidoylphenol 1-(4,5-dihydro-1H-imidazol-2-ylmethoxy)indole 5-[2-(3,4-dimethoxyphenyl)pyridine-4-carbonyl]-2-hydroxybenzaldehyde N-[2-(3,5-dimethylphenyl)ethynyl]-1,4-oxathiepane-7-carboxamide N-[2-(dimethylamino)ethyl]-4-[1-[3-methanimidoyl-5-(trifluoromethoxy)phenyl]ethylamino]-6-oxo-2,3-bis(sulfanylidene)-1H-pyrazine-5-carboxamide 4-ethoxy-2,3-bis(methylsulfanyl)benzenethiol 3-(N-(2,4-dichloropyrimidin-5-yl)-4-ethoxyanilino)propane-1,2-diol (4S)-5-methyl-1,3-bis[2,6,7-tris(trifluoromethoxy)benzoyl]piperidin-4-one 2-methoxy-4-[(1E,3Z)-penta-1,3-dienyl]naphthalene (NE)-N-[2-(4,5-dimethoxycyclohepta-1,3,6-trien-1-yl)-5,6-dihydroimidazo[2,1-b][1,3]thiazin-7-ylidene]hydroxylamine (2S)-1-[3-[[4-chloro-2-(7-chloro-6-methoxyquinolin-4-yl)phenoxy]methyl]-5-fluorophenyl]propan-2-amine 2-chloro-3,4,5,6-tetrafluoro-N-methylbenzenesulfonamide [2-(2,6-dichloropyridin-4-yl)phenyl]methanamine 3-[4-(1,2-benzoxazol-3-yl)piperazine-1-carbonyl]-7H-pyrrolo[2,3-d]pyrimidin-6-one 1-[4-(5,7-dimethylthieno[3,2-d]pyrimidin-2-yl)oxyphenyl]-3-methylbutan-2-ol 6-(4-acetylpiperazin-1-yl)-3-[1-methyl-5-(propanoylamino)pyrazol-3-yl]-N-[2-oxo-3-[4-(trifluoromethoxy)phenyl]imidazolidin-1-yl]pyridine-2-carboxamide N-[3-(2,5-dioxoimidazolidin-1-yl)phenyl]-2,3-dihydrothieno[3,4-b][1,4]oxazine-6-carboxamide 1-(4-methylsulfanylphenyl)heptane-2,6-dione 1-(4-methoxyphenyl)sulfonylpiperidine;2,2,2-trifluoroacetic acid (E)-3-[4-[9-[3,5-bis(trifluoromethyl)phenyl]fluoren-9-yl]oxyphenyl]prop-2-enoic acid 4-(2,6-difluorophenyl)-6-ethylcyclohexa-1,3-diene-1-carboxamide 5-[3-(2,6-dimethoxyphenyl)-1H-pyrazol-5-yl]-4-methylthiadiazole 4-[3-(2,5-dimethylphenyl)propanoyl]morpholine-3-carboxylic acid 4-azido-N-(5-propylnonan-3-yl)benzamide 3-[2,4-bis(phenylmethoxy)phenyl]-N-[5-(diethylamino)pentanoyl]-6-methylimidazo[1,2-a]pyrazine-2-carboxamide N-(2,2-dimethylcyclohexyl)-6-ethoxy-7H-purin-8-amine 3-[5-(1,3-benzothiazol-2-yl)-6-methoxy-9-oxoxanthen-4-yl]piperidine-1-carboxylic acid 2-tert-butyl-4-[[7-cyclopropylimino-5-(3,4,5-trimethoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-ylidene]methyl]-6-iodophenol N-butyl-1-methoxy-N,2-diphenylcyclohexa-2,4-dien-1-amine 2-[(3E)-2,4-dimethylhexa-1,3,5-trien-3-yl]oxy-6-oxo-N-[4-(pyrazol-1-ylmethyl)phenyl]-1H-pyrimidine-4-carboxamide 2-(1H-imidazol-5-yl)-N,4-dimethoxy-7-nitrocyclohepta-1,3-dien-1-amine 5-(2,4-difluorophenyl)-7-hydroxy-3H-imidazo[1,2-a]pyrimidine-6-carboxylic acid 2-(3,4-dichlorophenyl)sulfonyl-N'-[1-(3,4-dihydro-1H-isoquinolin-2-yl)ethenyl]-N'-methylidenebenzenecarboximidamide 6-amino-9-(furan-2-ylmethyl)-2-propan-2-ylsulfanyl-7H-purin-8-one 4-[3-cyclopropyl-1-(difluoromethoxy)pyrazole-4-carbonyl]piperazine-2-carboxylic acid 5-(2,4,6-trichlorophenyl)-1H-tetrazolo[1,5-a]quinazoline (E)-3-[2-[6-fluoro-4-(trifluoromethyl)quinolin-7-yl]oxyphenyl]-1-pyrrolidin-1-ylprop-2-en-1-one 3-(3,4-difluorophenyl)-N-(1-methylcyclopropyl)azetidine-1-carboxamide 1-amino-2,4-dichloro-5-(trifluoromethyl)anthracene-9,10-dione 2-[3-aminobutyl(propyl)amino]-N-[(1,7-dimethylbenzimidazol-2-yl)methyl]acetamide 3-[5-(cyclobutylmethoxy)pyridin-3-yl]propanenitrile 3-[2-azido-5-methyl-6-(oxolan-3-yl)pyridin-4-yl]oxy-1,2-dihydropyrazine 2-hydroxy-4,7-dimethyl-N'-(methylideneamino)-6H-cyclohepta[b]indole-3-carboximidamide 2-[(3E)-5-(2,3-dihydro-1H-inden-4-yloxymethyl)hexa-3,5-dien-3-yl]-3H-isoindol-1-one 5-chloro-N-(3,4-dihydro-2H-chromen-4-yl)-6-methoxypyridine-3-carboxamide 1-azidooxy-2,3,4-trichlorobenzene N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-fluoro-8-methoxy-2-oxochromene-6-sulfonamide (2S)-4-[[1-(dimethylamino)cyclohexyl]amino]-N-(3-fluoropyridin-2-yl)pyrrolidine-2-carboxamide;formic acid (7-methyl-2,3-dihydroimidazo[1,2-a]pyridin-3-yl)-(4-pyrimidin-5-ylpiperazin-1-yl)methanone (2R)-6-chloro-N-[(5-chloro-3-methylpyrazolo[1,5-a]pyrimidin-7-yl)methyl]-4-oxo-2,3-dihydrochromene-2-carboxamide 5-[(2,6-dichlorophenyl)methoxy]-2-[(3,4,5-triethoxy-1H-indole-7-carbonyl)amino]benzoic acid N-[(4S)-2-oxopiperidin-4-yl]benzamide [6-(3,4-dichlorophenyl)-5-methyl-2-propan-2-ylpyrimidin-4-yl]hydrazine 4-[1-[6-(7,8-dihydroquinolin-5-yl)pyridin-2-yl]cyclobutyl]aniline 4-[5-(1H-imidazol-2-yl)tetrazol-2-yl]butanoic acid 3-cyclobutyloxy-2-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butyl]propanoic acid 2-azido-3,5,7-trihydroxynaphthalene-1,4-dione N-(2-methyl-1,3-benzothiazol-6-yl)-5-[(Z)-prop-1-enyl]thiophene-2-sulfonamide ethane;N-methyl-4-[5-(trifluoromethyl)pyridin-2-yl]aniline 2-[(6-chloropyridin-3-yl)methoxy]pyrimidine (2Z,4E)-7-[(1R)-1-hydroxyethyl]-3-methylocta-2,4-dienenitrile;N'-hydrazinylidene-9-oxophenalene-1-carboximidamide 2-amino-5,6-bis[(3-methylphenyl)diazenyl]benzenesulfonic acid 7-[(2-amino-5,6,8,9-tetrahydrooxepino[4,5-b]pyridin-3-yl)methoxy]-N-[3-[1-(cyclopropanecarbonylamino)propan-2-yl-methylamino]propylsulfanyl]quinoline-2-carboxamide (2E)-N',3,7-trimethyl-4-[3-[2-(methylideneamino)ethoxy]phenyl]octa-2,6-dienimidamide 2-(3,5-dimethylphenyl)imino-5-[[5-(4-fluorophenyl)furan-2-yl]methylidene]-1,3-thiazolidin-4-one N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-4-[3-(1H-indol-2-yl)piperidine-1-carbonyl]cyclohexane-1-carboxamide 5-ethyl-1H-carbazole;4,4,5,5-tetramethyl-2-(3-phenylphenyl)-1,3,2-dioxaborolane (5R,6S)-5-[4-fluoro-3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydropyran-6-ol;hydrochloride 4-[[5-(2,6-dichlorophenyl)furan-2-yl]methylideneamino]pyridine-3-carboxylic acid 1,2-difluorobenzene;ethane;N-(4-methylbutan-2-yl)-3-phenoxyaniline 2,3-dichloro-5-methylpyridine;ethane 5-azido-2-fluoro-4,6-dimethylbenzimidazole 4-cyclohexyloxycarbonylbenzoic acid 1-[2,5-diamino-6-(4-nitrophenyl)hexyl]pyrrolidine-2,5-dione N-(2,6-dimethoxypyrimidin-4-yl)-4-[N-(3-nitrophenyl)anilino]benzenesulfonamide N-(3,4-dimethylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 3-[(2R)-6,7-dihydro-5H-cyclopenta[b]pyridine-2-carbonyl]-4H-1,2,4-oxadiazol-5-one (1R,2S)-N-[2,6-di(propan-2-yl)phenyl]-3-(3-methoxyphenyl)-2,3-dihydro-1H-inden-1-amine N-[4,5-dichloro-2-hydroxy-3-(6-methoxypyridin-3-yl)phenyl]-3-fluorobenzamide 2-[1-(8,9-dihydro-7H-purin-6-yl)piperidine-4-carbonyl]-N'-methylidenebenzenecarboximidamide N-(6,7,8,9,10,11-hexahydropyrazolo[3,4-a]acridin-5-yl)cyclopropanecarboxamide 2-chloro-1-(3,4-dihydro-2H-pyrano[2,3-b]pyridin-6-yl)ethanone (4S)-N'-[2,6-difluoro-4-[2-[5-[(E)-hydroxyiminomethyl]pyridin-3-yl]ethynyl]phenyl]-3-(oxolan-3-yloxy)-1,2-oxazolidine-4-carboximidamide 1-methyl-3-(methylamino)pyrido[2,3-b]pyrazin-4-one;propane N-[4-(2,6-dimethoxyphenyl)-5-(6-methylpyridin-3-yl)imidazol-1-id-2-yl]-3-phenylpropanamide;platinum(2+) N-[6-[4-(3,5-dimethoxybenzoyl)piperazin-1-yl]pyridin-3-yl]azetidine-2-carboxamide ethane;N-[4-(hydroxymethyl)phenyl]-2-oxo-1,3-dihydroindole-5-carboxamide N-[[4-(1,2,3,6-tetrahydropyridin-4-yl)phenyl]methyl]-1H-pyrrolo[3,2-c]pyridine-2-carboxamide N-(3-chlorophenyl)sulfonyl-4,5,6,7,8,9-hexahydrothieno[2,3-b]quinoline-2-carboxamide 1-ethenyl-4-(2,5,8-triphenyldecoxy)benzene (2S)-1-methyl-2-(4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridine-2-carbonylamino)piperidine-4-carboxylic acid 1-ethyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperidine-4-carboxamide 6-bromo-3-methyl-1,4-dihydroquinazolin-2-one N-(1,2-dihydropyridin-5-ylmethyl)-N'-phenylethane-1,2-diamine N-[5-(furan-2-yl)-1H-pyrazol-3-yl]-4-methylpyridine-3-carboxamide 3-[(4R)-7,10,11-trimethyl-3-thia-8,11-diazatetracyclo[8.6.0.02,7.012,16]hexadeca-1(16),2(7),5,10,14-pentaen-4-yl]propanoic acid 2-amino-6-[(6S)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl]phenol N-(6-benzylsulfonyl-1,2,3,4-tetrahydropyrido[3,4-b]indol-8-ylidene)hydroxylamine (3S,5R)-1-[2-methyl-4-(3,4,5-trifluorophenyl)benzoyl]-5-phenylpyrrolidine-3-carboxylic acid 1-[(3R)-5-(2,4-difluorophenyl)-7-methyl-4-phenylsulfanylspiro[1H-indole-3,4'-oxane]-6-yl]-N-methylmethanamine 3-[(2E)-3,7-dimethylocta-2,6-dienoxy]-4-hydroxy-5-propanoylpyran-2-one N-[1,4-dimethyl-2-(oxan-4-yl)-3,5,6,7-tetrahydropyrazolo[4,3-c]pyridin-4-ium-3-yl]thiophene-2-carboxamide N-[1-(2-chlorophenyl)-2,2,2-trifluoroethyl]-3-oxopiperazine-1-carboxamide 4-[[5,6-dichloro-1-[2-methoxy-3-(oxan-4-ylamino)phenyl]benzimidazol-2-yl]methyl]cyclohexane-1-carboxylic acid N-[2-(1H-indol-3-yl)ethenyl]-N'-pyridin-3-yl-1,4-diazepane-1-carboximidamide 5-N-[2-(1H-indol-3-yl)ethyl]-3-phenyl-6,7-dihydropyrazolo[1,5-a]pyrimidine-5,6-diamine 1,2-dimethyl-4-(1-methylpyridin-1-ium-2-yl)-6,7-dihydrobenzimidazole;chloride 1-(3,6-dihydro-2H-pyran-4-yl)-2-[6-[6-hydroxy-1-methoxy-5-[4-(trifluoromethyl)phenyl]pyridin-1-ium-3-yl]cinnolin-3-yl]ethanone 4-[(2S)-1-azidopropan-2-yl]oxy-1,2-dimethoxybenzene 5-amino-6-[(2,4,5-trimethylphenyl)methoxy]naphthalene-1-sulfonic acid N-(2,5-dichlorophenyl)-4-nitro-N-octylbenzamide 1-(3-chloro-2,5-dimethylphenyl)-6-hydroxy-5-[[(5Z)-4-oxohepta-5,7-dien-3-ylidene]amino]pyrimidine-2,4-dione [2-amino-3-(4-bromophenyl)-1,2-dihydrobenzo[e]indol-5-yl]-phenylmethanone 3-amino-N-[2-(1,4-diazepan-1-yl)ethoxy]benzenecarboximidate 1-(2,3-dimethylphenyl)-5-imino-4-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-2H-pyrrol-3-ol 3,3,7-trimethyl-2-[4-(6-methylcyclohexa-1,5-dien-1-yl)phenyl]indene N-[2-(4-methylphenyl)ethyl]-N',3-dihydro-1H-pyrazole-5-carbohydrazide 1-benzyl-N-[(2S)-1,3-dihydroxybutan-2-yl]piperidine-4-carboxamide N-[3,5-dimethyl-4-(4-piperazin-1-ylbutoxy)phenyl]hydroxylamine;ethane (1S)-2,3,5-trimethyl-8-[4-(tetrazolo[1,5-a]quinoline-7-carbonylamino)butanoyl]cyclopentane-1-carboxylic acid 2-[5-[3-methyl-4-(4-pentoxyphenyl)buta-1,3-dienyl]pyridin-2-yl]sulfanylethanethiol [(3R)-3,4-dihydroxypyrrolidin-1-yl]-(6-ethynylindol-1-yl)methanone 3-(1H-imidazol-2-yl)-6,7-dimethoxyisoquinoline 5-[(1S)-2,2,4-trimethylcyclopentyl]benzene-1,3-diol 1-methyl-4-[2-(3-thiophen-3-ylphenyl)ethynyl]piperidine 2-[2,3-difluoro-4-(4-methylphenyl)phenyl]-6-propylnaphthalene N-[3-chloro-5-(methylamino)phenyl]-4-(dipropylamino)benzamide 1-azidosulfanyl-N',5-dibenzyl-2-methoxy-6-(4-methylphenyl)sulfonyl-9H-fluorene-3-carboximidamide N-[(2R)-2,6-dimethylmorpholin-4-yl]-1-(5-fluoropyrimidin-2-yl)pyrrolidine-3-carboxamide 1-[3-(5-chlorobenzotriazol-2-yl)-4-hydroxyphenyl]-N,N-dimethylpyrrolidine-2-carboxamide 2-N,5-dicyclopropyl-4-N-(1,3-thiazol-4-ylmethyl)pyrimidine-2,4-diamine 4-[5,6-dichloro-2-(methylideneamino)pyridin-3-yl]-N'-hydroxybenzenecarboximidamide 5-amino-3,3-difluoro-4-(2-fluoroethoxy)-N'-hydroxy-2-oxo-1H-indole-7-carboximidamide 2,6-difluoro-N'-(3-oxopiperazine-1-carbonyl)benzenecarboximidamide 2,6-dichloro-4-[3-[5-(1H-pyrrole-2-carbonyl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]-3,4-dihydroquinolin-8-yl]benzamide 2-[(2Z)-3,7-dimethylocta-2,6-dienoxy]-1,4-dimethylbenzene 1-[2,3-difluoro-6-(2-fluoro-4-methylphenyl)phenoxy]-3-nitropropan-2-amine 7-(4,6-diphenylpyrimidin-2-yl)-5a,8a-dihydroindolo[3,2-b]carbazole 1-azidooxysulfanylanthracene 3-azido-7-bromocinnoline 1-butyl-3,4-difluoro-2-(2-fluoro-4-iodoanilino)-5-methoxyoxybenzene N-[(2,3-dichloro-4-hydroxy-5-methoxyphenyl)methylideneamino]-4-methylbenzenesulfonamide 1-[(2Z,4Z)-6-diphenylphosphanylhepta-2,4-dien-3-yl]-N,2-dimethylnaphthalen-1-amine 2-(3-morpholin-4-ylphenyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-4,7,9(13)-trien-11-one 4-[3-fluoro-5-methoxy-2-(trifluoromethyl)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile 3-bromo-2,5-difluoro-N,4-dimethylbenzenesulfinamide 4-[4-[3,5-dimethyl-2-(trifluoromethoxy)phenyl]sulfonylpiperazine-1-carbonyl]benzenesulfonamide N-methyl-2,4-dioxo-N-[3-(1H-pyrrole-2-carbonyl)oxolan-3-yl]pyrimidine-1-carboxamide 2-ethylsulfanyl-N'-[(E)-3-(furan-3-yl)prop-1-enyl]benzenecarboximidamide 4-[2,6-difluoro-4-(4-methylcyclohexyl)phenyl]-1,3-thiazol-2-amine N-[4-amino-3,5-bis(ethenyl)phenyl]-2-methoxypropanamide;ethane 2-[(4R)-6,7-dichloro-1,3-dioxospiro[2H-isoquinoline-4,3'-piperidine]-1'-yl]acetic acid;ethane N-(4-bromobutan-2-yl)-N-tert-butylpyridin-3-amine (6S,9aS)-8-(2,3-dimethoxyphenyl)sulfanyl-6-[3-methyl-4-[[(1R,2S)-2-phenylcyclopropanecarbonyl]amino]butyl]-N-pentan-3-yl-5,6,7,9-tetrahydroimidazo[1,5-a][1,4]diazepine-9a-carboxamide (E)-3-[4,5-bis(4-chlorophenyl)-1H-imidazol-2-yl]-1-[5-ethylsulfonyl-6-[3-methyl-6-(trifluoromethyl)imidazo[4,5-b]pyridin-2-yl]pyridin-3-yl]prop-2-en-1-one 3-azidooxy-N-butyl-2,4,5,6-tetrachloroaniline (5E)-2-imino-5-[[4-[3-methoxy-5-nitro-4-(propylaminomethyl)phenyl]furan-2-yl]methylidene]-1,3-thiazolidin-4-one 2-(N,4-dimethylanilino)-N'-[(Z)-(2-hydroxyphenyl)methylideneamino]benzenecarboximidamide 2-(3-ethylphenyl)-6-[4-(trifluoromethoxy)phenyl]pyridine 5-[3-(dimethylamino)pyrrolidin-1-yl]quinoline-8-carbonitrile 2-azidooxy-4-cyclohexyloxypyrimidine N-[(4-chlorophenyl)methyl]-2-ethyl-3,5-dihydroxyheptanamide N-(2,3-dichlorophenyl)-5-[1-(trifluoromethyl)cyclopropanecarbonyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 3-cyclobutyl-2,6-diphenyl-1H-imidazo[4,5-b]pyridine 2-tert-butylsulfinyl-1H-indole 4-[[4-methylsulfanyl-5,8-bis(prop-2-enoxy)naphthalen-1-yl]diazenyl]phenol N-[6,7-dichloro-2-[(3R)-oxolan-3-yl]imidazo[1,2-a]pyridin-5-yl]acetamide 3-(4-bromophenyl)bicyclo[1.1.1]pentane N-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-1H-pyrazole-5-carboxamide N-(5,6-didehydropyridin-3-yl)-1-[[4-(trifluoromethoxy)phenyl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine 1-(5-bromo-2,4-dinitrophenyl)azetidine 2-(2-chlorobenzoyl)piperidine-1-carboxylate (2R)-N-[4-fluoro-3-[(3S,5R)-5-[(methoxycarbonylamino)methyl]-1-propan-2-ylpyrrolidin-3-yl]phenyl]piperidine-2-carboxamide N-[3-(4-chloropyrazol-1-yl)propyl]-N,2,3-trimethylpentanamide 4-(aminomethyl)-5-[4-chloro-2-methoxy-6-(1,2,3,6-tetrahydropyridin-4-yl)phenoxy]-N-cyclopropylsulfonyl-3-fluoro-2-hydroxybenzamide 1-[3-(4-cyano-3-methylphenyl)-5,6-dimethoxypyridazin-4-yl]-N-[2-(1H-indol-3-yl)ethyl]pyrrolidine-2-carboxamide (4Z)-2,3-dihydro-1H-azepino[7,6-b]indole (3S)-1-azido-N'-hydroxy-N,2,5-trimethylimidazole-4-carboximidamide N-(4,6-dimethylpyrimidin-2-yl)sulfanyl-N',N'-dimethylethane-1,2-diamine 4-ethyl-2-iodo-6-methoxyaniline (2R)-N'-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-3-chloropropane-1,2-diamine;(E,5Z)-5-ethylidene-4,6-dihydroxyhept-2-enenitrile 2-[1-[[4-(furan-3-yl)phenyl]methyl]piperidin-4-yl]acetonitrile 1-azido-2,3-bis(phenylmethoxy)benzene ethane;1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]sulfanylnaphthalene 2-(4-bromophenyl)-6,7,8-trimethoxynaphthalene 1-[4-(7-tert-butyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-2-yl)piperazin-1-yl]prop-2-en-1-one 4-(2,6-dichlorophenyl)sulfanylpyridine 3-(4-fluorophenyl)-N-[2,6-dimethyl-1-(methylideneamino)benzimidazol-5-yl]propanamide (2R,3S)-N-[4-(3-azidoanilino)phenyl]pyrrolidine-2-carboxamide 1-(4,5-dimethylpyrazole-1-carbonyl)-3,4-dihydro-2H-quinoline-6-carboxylic acid 1-[2,6-di(propan-2-yl)phenyl]-2-nitroethenethiol N-[(3R,4S)-1-cyclohexyl-2-oxopiperidin-3-yl]-7-fluoro-1H-indole-6-carboxamide N-(8H-cyclohepta[b]pyridin-4-yl)-2,3,4-trimethoxybenzenesulfonamide 4-(3-pyridin-2-ylpropyl)-2-[5-(trifluoromethoxy)pyridin-2-yl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine N-[4-(3,5-dimethylpyridin-2-yl)oxy-3-fluorophenyl]sulfanyl-1-phenylethanamine 1-azidooxy-3-(4-chlorophenoxy)benzene 5-[(1R,3S)-3-hydroxycyclopentyl]oxycarbonylpyridine-2-carboxylic acid 2-hydroxy-5-[(Z)-indol-3-ylidenemethyl]-1,3-thiazol-4-olate 1-[[6,8-bis(hydroxymethyl)naphthalen-2-yl]oxymethyl]cyclohexan-1-ol 2-[4-(cyclohexylmethoxy)phenyl]ethanamine (5Z)-5-[[4-bromo-3,5-dimethoxy-2-[(3R)-3-(4-nitrophenyl)sulfanylpyrrolidin-1-yl]phenyl]methylidene]-4-hydroxy-6,7-dihydro-1H-indazole 4-bromo-3-chloro-1-fluoro-2-[(2R)-2,3,3,5,6,7-hexafluoroheptyl]benzene 2-(2,6-dioxopiperidin-3-yl)-4-[4-(morpholine-4-carbonyl)piperidin-1-yl]isoindole-1,3-dione N-(2,3-dihydropyridin-5-yl)-6-[4-[4-[(E)-prop-1-enyl]cyclohex-2-yn-1-ylidene]piperidin-1-yl]pyrimidin-4-amine [7-chloro-2-(5-methyl-1,3,4-thiadiazol-2-yl)-1H-indol-5-yl]-(azetidin-1-yl)methanone 2-[(Z)-1H-indol-3-ylmethylidenehydrazinylidene]-5-propan-2-yl-1,3-thiazolidin-4-one 3-[4-(5,6-dichlorobenzimidazol-2-ylidene)piperidin-1-yl]sulfonylbenzonitrile 2-[1,3-benzodioxol-5-yl(methyl)amino]-N-(cyclopropanecarbonyl)-7-methoxy-6-sulfanylidene-1H-quinoline-4-carboxamide 2-[4-[(E)-1,3-diaminobut-2-enylidene]pyrimidin-5-yl]pyridine-4-carbonitrile 2-chloro-5-[5-(4,4,5,5-tetramethyloxaborolan-2-yl)pyridin-3-yl]phenol N-[(2S)-1-hydroxypropan-2-yl]-4-oxo-6,7-dihydro-5H-1-benzofuran-3-carboxamide 2-[5-(4,6-diphenyl-1,3,5-triazin-2-yl)pyridin-2-yl]pyridine-4-carbonitrile (3S)-3-cyclohexylsulfanyl-N'-hydroxy-2-[[4-(trifluoromethoxy)benzoyl]amino]butanediamide 4-methoxy-1-[6-(2-phenylethynyl)-2,3-dihydro-1H-inden-5-yl]piperidine;1-phenylsulfanylpyrrolidine 1-amino-3-[6-oxo-2,3-bis(prop-2-enyl)pyrimidin-4-ylidene]thiourea N-[(3R)-5,6-dimethoxy-2,3-dihydroinden-1-ylidene]hydroxylamine 2-(7-oxo-3,8-diazabicyclo[3.2.1]octan-3-yl)-N-(2-phenylethyl)acetamide 3-[2,5-dichloro-N-(2,4-dinitroanilino)anilino]butanoic acid 5-(3,4-dimethoxy-2-nitrophenyl)-4-iminopentanoic acid 2-tert-butylsulfinylpyridine;5-[3-(1,4-dimethoxyisoquinolin-7-yl)propoxy]-6-phenyl-N-[4-[2-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]pyrazine-2-carboxamide 4-[(5Z)-5-[[1,2,5]oxadiazolo[3,4-b]pyridin-7-yl(phenylsulfanyl)methylidene]cyclohexa-1,3-dien-1-yl]morpholine [2-(6,7-dimethoxyquinazolin-4-yl)spiro[5,6-dihydropyrrolo[1,2-a]imidazole-8,3'-pyrrolidine]-1'-yl]-phenylmethanone 3-bromo-1-cyclopropylpyrazolo[3,4-d]pyrimidine 2,4-ditert-butyl-6-(ethylideneamino)phenol 2-[(E)-1-(4,5-dihydro-1H-imidazol-2-ylamino)prop-1-enyl]-6-[4-[ethoxy(oxido)phosphoryl]oxyphenyl]naphthalene-1-carbonitrile 1-[(4-hydroxyphenyl)methyl]-3-(3,5,6-trifluoropyridin-2-yl)urea N-[2-(dimethylamino)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxamide;hydrochloride 2-[3,4-bis(ethenyl)thiophen-2-yl]ethanol N-(4,5-dimethyl-1H-pyrazol-3-yl)-2-[(6R)-3-methoxy-6-prop-2-enoyl-6,7-dihydro-4H-pyrano[4,3-c]pyrazol-1-yl]acetamide 2-[6-(dimethylamino)naphthalen-1-yl]benzenesulfonamide N-[4-(4-ethylpiperazin-1-yl)cyclohexyl]-2,3-dihydro-1H-indene-5-carboxamide (2R,3S)-3-azido-4-phenylsulfanylbutane-1,2,3-triol N'-[3,5-bis(trifluoromethyl)phenyl]ethane-1,2-diamine 5-cyclopentyloxy-1,2,3,4-tetrahydronaphthalene 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(6R)-2-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl]acetamide 2-[5-(difluoromethyl)pyrazin-2-yl]sulfanylacetamide (Z)-2-methylidene-3-(6-phenylmethoxypyridin-3-yl)hex-4-enal [1-azidooxy-4-(3-ethylphenoxy)-9H-fluoren-2-yl]-diphenylphosphane 6-bromo-4,5-bis[(2Z)-2-(pyridin-3-ylmethylidene)hydrazinyl]pyrrolo[3,4-b]pyrazine-7,8-dione 2-[(E)-2-[3,5-bis(trifluoromethyl)phenyl]ethenyl]-N,4-dimethoxyaniline 4-[5-(aminomethyl)thiophen-2-yl]sulfonyl-6,7,8,9-tetrahydropyrimido[5,4-b]indolizine-1,3-diamine N-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide 4-tert-butyl-2-(1,3-dihydropyrrolo[3,4-c]pyridine-2-carbonyl)-1H-pyrimidin-6-one 6-amino-4-[3-(6-cyanopyridin-2-yl)phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide ethane;2-ethoxy-N,3-dimethylaniline 2-amino-4-[3-fluoro-2-(trifluoromethyl)phenyl]-6-methylbenzene-1,3-dicarbonitrile N-methyl-3-oxo-2,4-diphenyl-4H-thieno[3,4-b]pyrrole-5-carboxamide 5-bromo-N,N-dimethylpyridine-3-carboxamide 1-[4-(2,3-dihydro-1H-inden-1-ylamino)phenyl]sulfonylpiperidine-2-carboxylic acid N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxymethyl]cyclohexyl]-2,6-difluorobenzamide 4-amino-1-[4-(diethylamino)phenyl]-2,2,3,5,6,7,8,9,10-octadeuterioanthracene-9,10-diol 5-(2-methoxypyridin-3-yl)-N-[1-(2,4,6-trimethylphenyl)imidazol-4-yl]-1H-pyrrole-3-carboxamide 5-(4,7-dimethoxy-1H-pyrrolo[3,2-c]pyridine-6-carbonyl)cyclohepta-1,4,6-triene-1-carboxamide 1,3-bis(4-fluorophenyl)-5-methylimidazole (4R)-4-[4-chloro-3-(trifluoromethyl)phenyl]-1-propan-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 3-[(2,6-difluorophenyl)methyl]-N-propan-2-yl-1,5,7,10,11-pentazatricyclo[7.3.0.02,6]dodeca-2(6),4,8,11-tetraen-12-amine [4-(dimethylamino)phenyl]-(4-hydrazinylidenephenyl)methanone 1-butyl-3,4-dimethoxypyrazole 3,5-bis(trifluoromethyl)aniline;hydrochloride 2-[(3,5-dimethoxyphenyl)sulfonylamino]-N-hydroxyacetamide 3-azidooxy-1-[(4-cyclohexylphenyl)methyl]-2-(oxan-2-ylmethoxy)piperidine 5-[6,7-dimethyl-2-(4-methylpiperidin-1-yl)imidazo[4,5-b]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidine 5-[[6-(3,4-difluorophenyl)imidazo[1,2-a]pyridin-8-yl]amino]-2-methoxyphenol 5-bromo-1,3-diethyl-6-(2,4,5-trimethoxyphenyl)pyrazolo[3,4-b]pyridine 2-[(3R,4R)-1-(4-aminophenyl)sulfonyl-4-hydroxypiperidin-3-yl]acetamide 4-[[5-(3,4-dihydroxyphenyl)-1,3,4-oxadiazol-2-yl]amino]benzenesulfonamide 1-[(4R)-6-chlorospiro[2H-1-benzofuran-3,5'-imidazolidine]-4'-yl]-N,N-dimethylmethanamine;formic acid 3-N,5-N-dimethyl-3-[2-oxo-2-(propanoylamino)ethoxy]benzene-1,2,4,5-tetramine;propane 1-[5-(4-fluorophenyl)-1H-pyrrole-3-carbonyl]piperidine-4-carbonitrile 4-[4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]-5-nitro-2H-triazole 4-azidooxy-1,3,5-trimethylquinolin-2-one 3,5-dibromo-N-[2-(2-tert-butylphenoxy)ethyl]benzamide 2,4-dimethyl-N-(6-methylsulfanylpyridin-3-yl)piperidine-1-carboxamide 6-[[5-chloro-2-(1H-indol-4-ylamino)pyrimidin-4-yl]amino]hexanenitrile N-methyl-2-[1-(2,4,5-trifluorophenyl)cyclopenta-2,4-dien-1-yl]oxyethanamine 2-[3,5-dichloro-4-(3-nitronaphthalen-1-yl)oxyphenyl]acetamide 2-[(3R,4S)-3-methoxy-1-[2-(oxan-4-yl)ethyl]piperidin-4-yl]oxypyridine (1S,3R)-2,2-dimethyl-3-[1-(2-oxopropyl)naphthalen-2-yl]cyclopropane-1-carbonitrile 3-(azidomethyl)-6,8-difluoroquinoline 1-(5,7-dimethylfuro[3,2-c]pyridin-3-yl)ethanone N-[2-[(E)-1-[3-[(5-methyl-1H-pyrazol-4-yl)amino]phenyl]prop-1-enoxy]ethyl]formamide [2-chloro-6-(3,4-dihydro-1H-isoquinolin-2-yl)pyrimidin-4-yl]methanamine;2-ethenyliminopropanimidamide 4-methyl-2-[5-(3-oxocyclobutyl)tetrazol-1-yl]benzoic acid N-(3-bromophenyl)-2,4-dichloropyrimidine-5-carboxamide N'-hydroxy-5,7-dimethyl-3-(2-phenylethoxy)quinoline-2-carboximidamide (5Z)-2-(3,4-dimethylphenyl)imino-5-[(1,2,2,4,7-pentamethylquinolin-6-yl)methylidene]-1,3-thiazolidin-4-one 2-[7,8-dideuterio-4-(trifluoromethyl)indeno[1,2-b]pyridin-5-ylidene]propanedinitrile 4-(2,3-dichlorophenyl)pyridine N-(5,7-dichloroquinazolin-4-yl)-2-[3-(trifluoromethoxy)phenoxy]acetamide 3-[4-(2,4-dichlorophenyl)phenyl]-1H-imidazole-5-carboxylic acid (1R)-3,3-difluoro-5-[6-(5-methoxypyridin-2-yl)-7H-purin-8-yl]cyclopentan-1-ol [(2R,3S)-4-benzoyl-3-methoxy-5-oxopyrrolidin-2-yl]phosphonic acid N-[(1R,5S)-3,6-diazabicyclo[3.2.0]heptan-6-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide;hydrochloride N-[1-(2,4-dihydroxyphenyl)ethylideneamino]pyridine-3-carboxamide N-[(1R)-3,4,17,19,20-pentazahexacyclo[15.7.0.02,10.04,9.011,16.018,23]tetracosa-2(10),5,8,11,13,15,18(23),19-octaen-14-yl]methanesulfonamide 7-amino-3,5,10,16,19-pentazapentacyclo[11.8.0.02,10.04,9.014,18]henicosa-1(13),2,4(9),5,7,11,14(19),15,17,20-decaen-6-one 2-methyl-4-(4-morpholin-4-ylsulfonylpiperidine-1-carbonyl)pyrazolo[3,4-c]pyridine-6-carboxylic acid N-[(6E,9R)-10H-acridin-9-yl]-4-cyano-2-[(4-hydroxyphenyl)methylsulfanyl]benzamide N-[2-(4-chlorocyclohexa-1,3-dien-5-yn-1-yl)ethyl]-4-[6-fluoro-7-(trifluoromethoxy)-9H-pyrimido[4,5-b]indol-8-yl]aniline 3-methoxy-5-[(3-methylcyclobutylidene)methyl]benzaldehyde ethane;1-[3-(methylamino)propyl]triazole-4,5-dicarboxamide 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidin-2-ide;manganese(2+) 4-N,6-N-diethyl-2-[(4-methoxyphenyl)sulfanylmethyl]-1H-pyrimidine-4,6-diamine 5-chloro-4-[2-(3-methylbutoxy)ethoxy]-2H-thieno[2,3-d]pyrimidine 1-ethenylsulfonyl-N'-phenyl-5-sulfamoylpyrrole-2-carbohydrazide 4-(2,4-difluorobenzoyl)-1H-quinoxaline-2,3-dione [2-hydroxy-6-(2,4,5,6-tetrafluorophenoxy)phenyl]-trimethylazanium;dichloride N-(4-chlorophenyl)-2-[[4-cyclopropyl-5-(1H-indol-3-yl)-1,2,4-triazol-3-yl]sulfanyl]acetamide 2-[4-(6-amino-1,3,5-triazin-4-yl)-1,4-oxazepan-7-yl]acetic acid 5-[2-acetamidoethyl(methylsulfonyl)amino]naphthalene-2-sulfonic acid 2-(1,5,7,10-tetrazatricyclo[6.4.0.02,6]dodeca-2(6),3,7,9,11-pentaen-12-ylmethoxycarbonylamino)benzoic acid ethane;1-phenylmethoxycarbonylpiperidine-2,6-dicarboxylic acid 1-chloroethane;2-methylbutan-1-amine;(Z)-4-[(3E,5E)-5-methylocta-3,5-dien-7-yn-3-yl]oxypent-3-enal (E)-1,3-bis(4-fluorophenyl)-2-[4-(5H-indeno[1,2-b]pyridin-9-yl)phenyl]prop-1-en-1-amine 1-(2,6-diethyl-4-methylphenyl)-3-[(Z)-[4-[1-(4-ethoxyphenyl)propan-2-ylideneamino]oxy-3-fluorophenyl]methylideneamino]thiourea N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-octylbenzamide 2-(2,4-dichlorophenoxy)-N-[4-oxo-1-phenyl-5-[[(E)-3-piperidin-4-ylprop-2-enoyl]amino]pentan-2-yl]acetamide 2-[6-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-1-benzothiophen-2-yl]pyridine 4-[(Z)-3-amino-2-methylprop-1-enyl]-N-[2-[4-(difluoromethoxy)phenyl]ethyl]-6,7-dihydro-5H-cyclopenta[d]pyrimidine-2-carboxamide (NE)-N-[2,4-bis(phenylmethoxy)cyclopenta-1,3-dien-1-yl]-4-methylpiperazine-1-carbothioamide (3S)-4,7-dibenzyl-1-methylsulfonyl-2,3-dihydropyrido[3,2-b][1,4]oxazine;(6Z)-1,1-dichloro-6-ethylidenecyclohexa-1,3-diene 3,5-diamino-6-chloro-N-cyclopropylpyrazine-2-carboxamide 1-[2-(3,5-dichlorophenyl)ethyl]piperidine 2-amino-6-ethoxy-4-[5-(1,3-oxazol-4-yl)thiophen-2-yl]-4H-pyran-3,5-dicarbonitrile N-(5-phenylpentanoyl)octanamide N-methyl-6-[4-(3,3,8-trimethyl-1,2-dihydroindole-5-carbonyl)piperazin-1-yl]pyridazine-3-carboxamide N-[2-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-cyanocyclohexa-1,3-dien-1-yl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-2-sulfonamide 1-N,3-N-dibutylbenzene-1,3-dicarboxamide;ethane 3-(2,6-dichlorophenyl)-7-[4-[5-methyl-2-(2H-tetrazol-5-yl)phenyl]piperazin-1-yl]-8H-pyrido[3,4-d]pyrimidine 3-(4-tert-butylphenyl)sulfanyl-2-[6-[(5-chlorocyclohepta-1,4,6-trien-1-yl)methoxy]spiro[3.3]heptan-2-ylidene]propanenitrile 6-[4-(5-chloro-3,4-dihydro-1H-isoquinoline-2-carbonyl)-2-methylphenoxy]hexanamide 1-[3-(hydroxymethyl)cyclobutyl]pyridin-2-one 2-[4,7-dimethyl-1-(naphthalene-2-carbonyl)-3-oxo-5,6-dihydro-2H-1,8-naphthyridin-2-yl]acetic acid 7-[2,4-dichloro-6-(difluoromethoxy)phenyl]-N-(3-hydroxycyclobutyl)-3-oxo-1H-pyrazolo[1,5-a]pyrimidine-2-carboxamide 4-(6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl)-6-ethyl-3,4a,5,7,8,8a-hexahydro-1H-1,6-naphthyridin-2-one 6-chloro-4-(5-cyclopropyloxy-2,3-difluorophenyl)-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 3,5-difluoro-4-[(2E)-penta-2,4-dienyl]-6-phenyl-9H-xanthene (E)-4-(dimethylamino)but-2-enal;1-[4-[(5S,7R)-9,11,15-triazatetracyclo[8.6.0.03,8.012,16]hexadeca-1,3,6,10,13,16-hexaen-5-yl]piperidin-1-yl]ethanone (3S,4R)-N-(4-fluorophenyl)-3-methyl-1-oxo-2-pyridin-3-yl-3,4-dihydroisoquinoline-4-carboxamide 1-[(2,5-difluorophenyl)methyl]-4,7-dioxofuro[3,4-b]pyridine-5-carboxylic acid 2-[(3S)-1,1-dioxothiolan-3-yl]oxy-N'-hydroxypyrimidine-4-carboximidamide 5-(azidomethyl)-2-[3,4-difluoro-2-(trifluoromethoxy)phenyl]pyridine N-[2-(4-bromophenoxy)ethyl]-1H-pyrazole-5-carboxamide N-[[4,6-bis(methoxymethyl)pyrimidin-2-yl]methylideneamino]methanamine 2-[N-[(3,5-difluorophenyl)methyl]-4-methoxyanilino]ethanol 3-ethylsulfanyl-N',2-dimethoxybenzenecarboximidamide 4-(4-chlorophenyl)sulfanylpyrimidine 2-(2,3-dihydro-1H-inden-5-yl)-6-[4-(trifluoromethoxy)phenoxy]benzonitrile;ethane 4-[[2,6-dichloro-3-(ethylamino)phenyl]methylamino]benzoic acid (2S)-3-cyclopropyl-N-[4-[5-(1H-imidazol-5-ylmethyl)thiophen-2-yl]phenyl]-N-[(Z)-(3-methoxyphenyl)methylideneamino]butanamide N-(1,3-dimethylpyrazol-4-yl)-2-[7-methoxy-3-methyl-1'-(thiophen-3-ylmethyl)spiro[chromeno[2,3-c]pyrrole-9,3'-pyrrolidine]-1-ylidene]acetamide 3-[6-chloro-2-(2,3-dihydrofuran-4-yloxy)-8-fluoro-7H-purin-9-ium-9-yl]pentane-1,5-diol 2-[4-[7-(8,9-dihydrodibenzofuran-3-yl)imidazo[1,2-c]pyrimidin-5-yl]phenyl]-6-phenylpyridine 1-[5,6-bis(ethenyl)pyrimidine-4-carbonyl]pyrrolidine-2,3-dione N-(2,3-dihydroimidazo[1,5-a]pyridin-6-ylmethylideneamino)-4-phenylbenzamide 4-methyl-3,6-dinitro-2H-pyrazolo[4,3-c]quinoline 6-[1-(4-fluorophenyl)cyclopropyl]-3H-pyrido[2,3-d]pyrimidine-4,7-dione N-[3-[(1R,5S)-1-hydroxy-2-oxabicyclo[4.2.0]octan-7-yl]phenyl]propane-2-sulfonamide 2-[5-(difluoromethyl)-1,3-thiazol-4-yl]-6-(oxolan-3-ylsulfonylamino)pyridine-4-carboxylic acid 5-tert-butyl-N-[1-(5,7-dichloroisoquinolin-4-yl)ethyl]-2-methylpyrazole-3-carboxamide 6-fluoro-2-(4-propylcyclohexyl)-1,4-dihydronaphthalene 3-(6,7,8a,9a-tetrahydro-5H-imidazo[1,2-a]quinoxaline-1-carbonyl)benzonitrile 1-(3-bromophenyl)-2-chloroethanone;1,3-dimethylbenzene 4-(2,3,6-trifluoroanilino)benzonitrile 5-chloro-N-(3,3-dimethylcyclohexyl)-1-benzofuran-2-carboxamide N-[2-(dimethylamino)ethyl]-N'-(6-oxo-1H-pyridin-3-yl)oxamide 5-[[2-(3,4-dichlorophenyl)-1H-imidazol-5-yl]amino]-3-(2-methoxypyridin-4-yl)-1-piperidin-4-ylpyrazolo[4,3-d]pyrimidin-7-one 3-methoxy-6-[2-(pyridin-3-yloxymethyl)morpholin-4-yl]pyrimidin-4-one N-[(2E,4Z)-3,6-dimethylhepta-2,4,6-trien-2-yl]-5-[3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-amine 4-[3-(methyliodanuidylamino)phenyl]benzaldehyde 2-[4-(6-methoxy-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]ethanol (4-fluorophenyl)-[2-(1,3-thiazol-5-ylmethoxy)phenyl]methanone 3-(4-chlorophenyl)-N-[1-(4-ethylsulfanylphenyl)-2-hydroxyethyl]prop-2-ynamide 1-N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-5-methanimidoyl-3-N,3-N,2-trimethylbenzene-1,3-diamine [2-(1,3-benzodioxol-5-ylmethoxy)phenyl]-[4-(1H-pyrazole-5-carbonyl)piperazin-1-yl]methanone N-[2-(diethylamino)-1,3-benzothiazol-6-yl]pyridine-4-carboxamide;hydrochloride 1-[2-[(5-azidopyridin-3-yl)methylsulfonyl]ethyl]piperidine-4-carbonitrile (5Z,6Z)-5-(3-methoxy-2-phenylpropylidene)-1,4-diazepane (3S,5R)-5-azido-1-benzylpyrrolidin-3-ol 4-[3-(5,6-diamino-2H-pyrimidin-1-yl)phenyl]benzoic acid N-(1,3-benzodioxol-5-yl)-2-[8-methoxy-6-(oxolan-3-yloxy)quinolin-2-yl]acetamide 3-methylsulfanyl-1,2-diphenylprop-2-en-1-one 4-(6-bromo-3,7-dimethyl-3a,4,5,10b-tetrahydrobenzo[e]benzimidazol-2-yl)phenol (Z)-2-ethylsulfanyl-4,4-dimethoxybut-1-en-1-amine;3-[[2-(trifluoromethyl)quinolin-6-yl]amino]cyclohexa-2,5-diene-1,4-dione (2E,4Z)-N-cyclobutyloxy-6-morpholin-4-yl-5-piperidin-3-yloxyhepta-2,4,6-trienamide (2S)-2,4-diamino-N'-[5-bromo-4-chloro-2-[(Z)-3-iminoprop-1-enyl]phenyl]butanimidamide 4-(2-methyl-1,3-dioxolan-2-yl)aniline (5Z)-2-methyl-5-[(2-propan-2-yloxyphenyl)methylidene]imidazolidin-4-one (3E)-3-[[5-bromo-2-(trifluoromethyl)phenyl]carbamoylhydrazinylidene]propanoic acid (4-azidophenyl)sulfonyl-(trifluoromethylsulfonylamino)azanide 2-[(Z)-1-amino-3-iminoprop-1-enyl]-4-pyridin-4-ylbenzonitrile 3,5-difluoro-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]benzamide (5S,7R)-N-[3-[4-amino-6-[2-(azetidin-1-yl)ethoxy]pyrrolo[2,1-f][1,2,4]triazin-5-yl]phenyl]-5-chloro-7-fluoro-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine 2-[[6-chloro-3,4-dihydropyridin-5-yl(cyclopropylmethoxy)amino]methyl]pyrimidin-5-ol 1-[2-(aziridin-2-yl)-3,5,7-trimethoxynaphthalen-1-yl]-2,4-dichlorobenzimidazole 2-(5-ethoxycarbonyl-3-iodo-1H-indol-2-yl)acetic acid 1-(cyclopropylmethylamino)-3-[(4,6-dimethylquinazolin-2-yl)amino]thiourea 4-(8,14-diphenyltetracyclo[10.2.1.05,15.08,13]pentadeca-3,5(15),6,8,9,11,13-heptaenyl)pyridine (2E)-3,4-dihydroxy-5-oxo-N-[1-[4-(trifluoromethylsulfanyl)phenyl]ethyl]hexa-2,6-dienamide 2-azidooxy-4-[(1R)-1-cyclopentylpropyl]benzenesulfonic acid 2-(4-fluorophenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidine 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]hexanoic acid 2-[(5S,10bR)-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-methoxyphenol 2-bromo-6,7-dichloro-N-[(4R)-1,3,2-dioxazepan-4-yl]pyrido[3,4-b]pyrazin-8-amine 2-[6,6-dimethyl-4-[(1E)-1-phenylbuta-1,3-dien-2-yl]heptyl]-1H-indole (4R)-1-[4,5-bis(ethenyl)pyridin-2-yl]oxy-3-N,3-N-dimethylpentane-3,4-diamine N-[1-[2-(3,4-dimethylphenyl)ethyl]piperidin-4-yl]-1,6-naphthyridine-5-carboxamide N-azido-3,5-dichloroaniline 2-[(5Z)-4-oxo-5-[[3,5,6-trimethyl-1-(3-nitrophenyl)pyrazol-4-yl]methylidene]-1,3-thiazolidin-2-ylidene]butanoic acid 4-[2-(1H-indol-2-yl)hydrazinyl]phenol N-[5,7-dimethyl-6-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]piperidine-1-carboxamide 5-[2-(methoxymethyl)thiophene-3-carbonyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide (2R)-1,3-bis(2-methylphenyl)-5-[[4-nitro-3-(trifluoromethyl)anilino]methylideneamino]oxypentan-2-ol 4-[7-fluoro-5-(4-fluorophenyl)-2,3-dimethyl-4H-azepin-6-ium-1-yl]benzoic acid 2-[2-(azidomethyl)phenyl]-5-propan-2-ylfuran 5-[5-(cyclopropylmethoxy)pyridin-3-yl]-N,4-dimethylsulfanyl-1H-indazole-3-carboxamide 2,4-dichloro-6-(2-ethyl-3H-benzimidazol-5-yl)phenol 1-cyclohexyl-4-(9H-xanthene-9-carbonyl)piperazin-2-one;ethane 6-[2-(trifluoromethyl)pyrimidin-5-yl]oxynaphthalen-1-ol 1-[(E)-2-nitroethenyl]anthracene 4-[(E)-3-methoxy-2,3-dimethylprop-1-enyl]-5,7-dihydropyrrolo[3,4-b]pyridine 5-(2,4-dihydroxyphenyl)-2-methyl-1H-imidazo[4,5-b]pyridine-7-carboxylic acid 1-phenyl-2H-thieno[2,3-d]imidazole 4-azidooxy-1H-indole-2,3-dione 1-methyl-5-(2,4,5-trifluorophenyl)-N-[6-(triazol-2-yl)pyridin-3-yl]pyrazole-3-carboxamide N-[5-fluoro-4-(1H-indol-2-yl)pyridin-3-yl]acetamide 5-amino-2-(4,4-dimethylcyclohexen-1-yl)pyridine-3-carboxylic acid 1-[(3Z)-penta-1,3-dien-2-yl]-4-propan-2-yl-2-[4-(trifluoromethoxy)phenyl]benzene 3-(5-tert-butylpyridin-2-yl)cyclohexan-1-imine 6-[4-methyl-5-(6-piperidin-1-yl-3H-imidazo[4,5-c]pyridine-2-carbonyl)thiophen-3-yl]pyridine-3-carbonitrile 5-[2-[4,6-bis(trifluoromethyl)pyridin-3-yl]phenyl]sulfanylpentanoic acid 3-(4-azidophenyl)-1H-pyrazolo[4,3-d]pyrimidine [3-(4,5-dihydrobenzotriazol-1-yl)phenyl]-phenylmethanone (3S)-N-benzyl-5,7-dimethyl-1-[(2R)-2-methyloxiran-2-yl]-4-oxo-2,3-dihydropyrrolo[3,2-c]quinoline-3-carboxamide 3-[2,6-dimethyl-4-(1H-pyrazol-5-yl)phenoxy]propanoic acid 3-bromo-1-[5-[4-(4-methoxyphenyl)phenyl]pyridin-2-yl]indole 6-fluoro-3-[2-(4-pentanoylpiperazine-1-carbonyl)phenyl]quinazolin-4-one 2-[4,6-di(propan-2-yl)cyclohexa-1,3-dien-1-yl]ethynamine;dichloromethane 1-ethylsulfonyl-3,3,7-trimethyl-2H-indole (2S)-2-[2,3-bis(4-chlorophenyl)-5,6-difluoro-4-oxoquinazolin-1-yl]-N-(4,5-dimethoxy-2-nitrophenyl)butanamide 5-methoxy-1-(4-methylphenyl)sulfinylindole 1,2-diamino-6-oxo-4-(5-phenoxy-3H-1,3-oxazol-2-ylidene)pyridine-3,5-dicarbonitrile [4-methylsulfonyl-2-(trifluoromethoxy)phenyl]urea 3-(4-chlorophenyl)-N'-[5-methyl-1-[2-oxo-2-[6-[4-(trifluoromethoxy)phenoxy]pyridin-2-yl]ethyl]triazol-4-yl]prop-2-enimidamide N-[5-[3-[7-(2,6-difluorophenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-indazol-5-yl]pyridin-3-yl]cyclopropanecarboxamide N-[(3R)-1-azabicyclo[2.2.2]octan-4-yl]-5,6-difluoro-2-methoxypyridine-3-carboxamide [(3R)-1,3-dimethylpyrrolidin-2-ylidene]-[[4-ethoxy-5-(6-fluoropyridine-3-carbonyl)pyridin-2-yl]carbamoyl]azanium 1,3-bis(2-fluoroethyl)-7H-purine-2,6-dione N-[1-(3,5-ditert-butylphenyl)ethylidene]hydroxylamine 6-azidooxy-3,4-di(propan-2-yl)benzo[c]chromene 3-(5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carbonyl)cyclohexane-1-carbonitrile 2-[(2Z)-2-[(Z)-[3-bromo-5-methoxy-4-(naphthalene-1-carbonyloxy)phenyl]methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 4-[(3S)-1-[3-[2,6-dichloro-4-(2-methylphenyl)sulfanylphenoxy]propyl]pyrrolidin-3-yl]oxybenzoic acid 2-(4-ethylphenyl)ethanamine;3-[[3-fluoro-5-(trifluoromethoxy)benzoyl]amino]propanoic acid 2,2-dichloro-3-(4-ethyl-5-iodothiophen-2-yl)cyclopropane-1,1-dicarbonitrile 4-(3,5-difluorophenyl)-N'-hydroxybutanimidamide [4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)cyclohexyl]carbamic acid 2-bromo-1-(6-methoxy-4-phenylnaphthalen-1-yl)ethanone 2-[(3R)-5-oxopyrrolidin-3-yl]oxypyridine-3-sulfonamide (E)-4-[(3S,5R)-2-(4-methoxyphenyl)-1-oxaspiro[4.5]decan-8-yl]but-3-en-2-one 1-[2-(5-methylpyrazol-1-yl)acetyl]-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide 2-(1,4-benzodioxin-3-ylmethoxy)-N'-hydroxypyridine-4-carboximidamide 1-[(E)-2-methyl-3,3-diphenylprop-1-enoxy]-4-propan-2-ylbenzene 2-azido-4-bromo-5,7-difluoroquinoline 6-methyl-2-(3,3,5-trimethyloxetan-2-yl)imidazo[1,2-a]pyridine 4-[[2-(4-chloroanilino)-5-fluoropyrimidin-4-yl]amino]piperidine-1-carboxamide 2-[3-[1-(3,5-dimethylbenzoyl)piperidin-4-ylidene]-6-fluoro-1H-isoindol-2-yl]acetaldehyde N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-phenyl-5-sulfanylidene-1,2,4-oxadiazolidine-2-carboxamide 2-[(6,8-dichloroquinazolin-4-yl)amino]-3-methoxyphenol N-[2-(4-methylphenyl)ethyl]-5,6,7,8-tetrahydroquinazolin-2-amine 1-benzyl-2-ethenoxy-4-[(Z)-3-methylhept-3-en-2-yl]benzene 3-[(2Z)-3,5-dimethylhepta-2,6-dienoxy]propanal;methanamine;4-methylbenzenethiol;N-[1-(methylamino)-1-oxobutan-2-yl]-N'-(2-pyrrolidin-1-ylethyl)heptanediamide (2S,5R)-2-azido-5-[4-cyclobutyloxy-3-[(4-fluorophenyl)methoxy]phenyl]pyrrolidine 5-chloro-4,6-bis[difluoro(iodo)methyl]-1H-indazole (3S)-N'-[4-cyano-2,6-dimethyl-1-[3-methyl-5-(trifluoromethoxy)phenyl]sulfonylpiperidin-4-yl]-2,3-bis[[deuterio(deuterio)methoxy]carbonylamino]butanediamide 5-(4-chlorophenyl)-2-(1-hydroxyethylamino)-3-methoxychromen-4-one 2-[[methyl(phenyl)hydrazinylidene]methyl]cyclohexa-1,3-dien-5-yne-1,4-diamine 1-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridin-8-yl)-N-(6-methoxypyridin-3-yl)pyrazole-4-sulfonamide 3-[4-[3,3-difluoropropyl(pyrimidin-2-yl)amino]phenyl]-5-methylimidazolidine-1,2-thiazol-thione 3,5-dimethyl-4-(6-oxa-2-azaspiro[3.4]octan-2-ylsulfonyl)phenol 1-[(1Z)-buta-1,3-dienyl]-2-methylcyclopentane;ethene;6-(4-fluorophenyl)-N-(1-formamidopropan-2-ylideneamino)imidazo[1,5-a]pyridine-1-carboxamide N-methyl-2-(4-methylsulfinylphenyl)-6-oxo-1H-pyrimidine-5-carboxamide 3-(cyclobutylmethyl)-6-(4,5-dichloropyridine-2-carbonyl)-1-(1H-pyrrolo[3,2-c]pyridin-2-ylmethyl)imidazo[4,5-b]pyridin-2-one (3R)-1,4'-dihydroxyspiro[indole-3,5'-7H-furo[2,3-f][2]benzofuran] 4-benzyl-1-(methoxymethoxycarbonyl)piperidine-2-carboxylic acid 3-[(5E)-7-hydroxyhepta-1,4,6-trien-2-yl]oxy-5-[5-methyl-6-(3-methylpentylamino)-3-[(Z)-prop-1-enyl]pyridin-2-yl]benzonitrile 4-(N-tert-butyl-3-nitroanilino)benzenesulfonamide 2-[5-(cyclopropylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]-N,N-dimethylacetamide;2,2,2-trifluoroacetic acid 2-[3-(5-nitro-1H-indazol-3-yl)phenyl]ethanamine 3-[3-azido-1-(2,4,6-trimethylphenyl)sulfonylindol-5-yl]propanoic acid 5-[(Z)-(3,4-dichlorobenzoyl)-[2-methoxy-5-oxo-8-(2-phenylethynylamino)-9H-naphtho[1,2-b][1]benzofuran-6-ylidene]methyl]-2-hydroxybenzoic acid 3-[1-(1,2,4-thiadiazol-5-yl)azepan-3-yl]-6,7-dihydro-5H-pyrrolo[3,4-b]pyridine 5-ethyl-2-(4-methoxyphenyl)-4H-pyrazol-3-one 1-(2,4-dibromophenyl)-5-methylhexane-1,3-dione (4S)-3,7,7-trimethyl-4-pyridin-3-yl-4,6,8,9-tetrahydro-[1,2]oxazolo[5,4-b]quinolin-5-one 2-bromo-1,3,4-trimethylindazole 6-[3-methylbuta-1,3-dien-2-yl(pyridine-4-carbonyl)amino]pyridine-3-carboxylic acid 2-[5,6-dichloro-4-(1H-pyrazol-4-ylamino)pyrimidin-2-yl]sulfanylethane-1,1-diol [3-aminooxy-2,4,6-tri(propanoyl)phenyl]methylphosphonic acid 1-[(3R)-4-azido-2,3-dihydroindole-1-carbonyl]azetidin-3-one 6-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]pyridin-2-amine 5-(4,7-dichlorobenzo[c]xanthen-3-ylidene)-2-hydroxyimino-1,3-thiazolidin-4-one N-[(4S)-6,8-difluoro-4-phenylmethoxyspiro[2H-naphthalene-3,1'-cyclohexane]-1-yl]acetamide 1-(3-chlorophenyl)-7,8-dimethoxy-N-[(3S)-piperidin-3-yl]-5H-chromeno[4,3-c]pyrazole-3-carboxamide;hydrochloride N-[(1R,2S)-4,6-difluoro-2-phenylmethoxycyclohexyl]-5,6-dimethylpyrimidine-4-carboxamide 6-(2,4-dimethoxyphenyl)-3H-pyrido[2,3-d]pyrimidin-4-one 6-hydroxy-2,3-bis(propan-2-ylsulfanyl)pyridine-4-carbonitrile N-[3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]-1H-indole-7-carboxamide 5-azido-2,3-dibromo-4-hydroxybenzonitrile N'-[2-aminoethyl(1,3-thiazol-5-yl)amino]-4-methoxybenzenecarboximidamide 2-[4-hydroxy-N-(3-methylbutyl)anilino]acetamide (3,4-difluorophenyl)methylazanide;1-ethyl-5-(4-fluorophenyl)-N'-methylidenepyrrole-2-carbohydrazide 2-[4-(1-ethylpiperidin-4-yl)oxy-3,5-difluorophenyl]-1-methylideneguanidine (3-aminophenyl)-[5-[2-(4-methylpiperazin-1-yl)ethoxy]-1,3-dihydroisoindol-2-yl]methanone 2-(7-chloro-1H-indazol-5-yl)spiro[5,6-dihydropyrrolo[1,2-b]pyrazole-4,3'-pyrrolidine] 3-(6-cyclohexa-1,5-dien-1-ylhexanoyl)-6,7-difluoroquinazolin-4-one N-[6-(2,5-dimethylpyrazol-3-yl)pyridazin-3-yl]-2-[3-fluoro-4-[(3-methoxyphenyl)carbamoylamino]phenoxy]acetamide N-[4,5-dichloro-2-methyl-3-(4-propan-2-ylphenyl)indol-1-yl]sulfonylacetamide 1-(4-azidobutyl)-3-[(2,5-dimethoxyphenyl)sulfonylamino]thiourea N-[(2,5-difluorophenyl)methyl]-6-iodopyrimidine-4-carboxamide N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-methanimidoyl-3-[[1-methyl-2-(oxan-4-ylamino)propylidene]amino]-5-[(E)-pent-3-en-1-ynyl]benzamide N-[5-(azidomethyl)thiophen-2-yl]ethenesulfonamide 1-(3-azidophenyl)-2,4,5-trimethylbenzene 2-(3,5-dimethylbenzene-6-id-1-yl)oxyquinoline;8,9,10,11-tetrahydrobenzo[a]azulen-7-ol;zirconium N-(2,4,6-trimethylphenyl)acetamide 4-methyl-3,5,6,7,8,9-hexahydrocyclohepta[c]pyridazine;[1-(5-methoxypyridin-2-yl)-2H-pyridin-5-yl]methanimine 4-(2,3-dihydro-1H-inden-5-yl)-2,6-dioxo-1,3-diazinane-5-carbonitrile (3R,5S)-5-benzyl-6-(hydroxymethylidene)-4-methylpiperazin-2-one 1-(3,3a,5,6a-tetrahydro-2H-furo[3,2-b]pyrrole-4-carbonyl)-N-benzylcyclohexane-1-carboxamide (Z)-3,4-dimethylpent-1-en-2-ol;ethane;N'-[5-[[2-fluoro-5-(trifluoromethoxy)phenyl]methoxy]pyrimidin-4-yl]methanimidamide 2-tert-butyl-4-[(E)-(4,5-dimethoxycyclohexa-1,3-dien-1-ylidene)methyl]phenol 2-[4-(8-acetyl-3-oxo-1,5,6,7-tetrahydroimidazo[1,5-a]pyridin-6-yl)-N-propan-2-ylanilino]-4-methoxybenzenecarboximidamide 3-amino-5-(4-bromophenyl)pentanoate 1-(3,5-diphenyl-4H-pyrazol-1-yl)ethanone 6-methyl-2-[5-[4-(trifluoromethoxy)phenyl]thiophen-3-yl]-1,8-naphthyridine 4-(2,3-dihydrothiophen-5-yl)-2,6-bis[(1R)-3-fluorocyclopentyl]pyridine 5-chloro-6-methyl-N-[(1S)-2,3,4,9-tetrahydro-1H-carbazol-1-yl]pyrimidine-4-carboxamide 3-(2,6-difluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine 4-[1-[2,3-difluoro-5-(trifluoromethyl)phenyl]ethoxy]benzamide N-[[4-(4-hydroxyoxan-3-yl)phenyl]methoxy]-1H-pyrazole-5-carboxamide 2-[3-(1H-imidazol-5-yl)-1,2,4-oxadiazol-5-yl]benzenesulfonamide 6-(5-acetyl-2-chloroanilino)-N,4-dimethoxypyridine-3-carboxamide N-[5-(1,6-dimethylpyrazolo[3,4-b]pyridin-4-yl)pentyl]carbamate 2-[3,5-dimethyl-4-[1-(thiophen-3-ylsulfonylamino)ethyl]pyrazol-1-yl]acetic acid N-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]-5,6-dihydronaphthalene-1-carboxamide 3-[(E)-2-[3,5-difluoro-4-[1-(methylamino)ethenoxy]phenyl]ethenyl]phenol (6S)-7-acetyl-3-hexylsulfanyl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 4-(6-bromo-2,4-dioxoquinazolin-1-yl)benzamide N-[5-(aminomethyl)-2-[2-chloro-3-[[6-methoxy-5-(4-methylimidazol-1-yl)pyridine-2-carbonyl]amino]phenyl]imidazo[4,5-b]pyrazin-6-yl]carbamate 4-[2-(4-methoxyphenyl)acetyl]morpholine-3-carboxamide 5-[6-(2-chlorophenyl)imidazo[1,2-b]pyridazin-3-yl]-1H-pyrrole-2-carbonitrile N-[(3S)-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]benzamide 1-(1,3-benzodioxol-5-yl)cyclohexa-2,4-dien-1-ol (E)-N'-[(2,6-difluorophenyl)methyl]-3-methylidenepent-4-enehydrazide 4-[[5-(5-chloro-2-fluorophenyl)spiro[1,3-dihydropyrido[2,3-e][1,4]diazepine-2,4'-piperidine]-1'-yl]sulfonylmethyl]-N-cyclobutylidenebenzenecarboximidamide (1R,2R)-4-[2-chloro-6-fluoro-5-(trifluoromethoxy)phenyl]-N-[8-[3-[5-(difluoromethyl)pyridin-3-yl]propyl]quinolin-5-yl]-2-methylcyclopentane-1-carboxamide 2-methyl-5,6,7,8-tetrahydronaphthalene-1-carboxylic acid 3-(6-fluoro-2,4-dihydroxy-1H-indole-5-carbonyl)benzoic acid (E)-4-[2,6-dichloro-4-(trifluoromethyl)phenyl]-N-(1H-imidazol-5-yl)but-3-enamide N-[(5E)-4-methylhepta-1,3,5-trien-2-yl]sulfanylpyrimidin-4-amine N-(1,3-benzodioxol-5-yl)-2-[methyl(4-phenylbutanoyl)amino]-2-piperidin-1-ylacetamide 3-[4-(aminomethyl)cyclohexyl]imino-1,2-diphenylpropan-1-one N-[(4-chlorophenyl)methyl]-2,6,8-trifluoro-3,4-dihydronaphthalene-1-carboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]-1,2-benzothiazol-6-amine 2-[(2,3,6-trichlorophenyl)methyl]propanedinitrile 4-(2,3-dichlorophenyl)-N-[(4S)-7-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]piperazine-1-carboxamide 2-(4-chlorophenoxy)acetamide;3,3-difluoro-4-hydroxypentanal 5-(5,6-difluoro-1H-indole-2-carbonyl)-N-[3-hydroxy-4-(methylamino)cyclohexyl]-N-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 1-(6-oxocyclohexa-2,4-dien-1-yl)pyridin-2-one (3R,4S)-1-[4-cyano-3-(trifluoromethyl)phenyl]-N,2-dimethyl-3-propan-2-ylpiperidine-4-carboxamide 6-(cyclopropylmethoxy)-2-[5-(cyclopentylamino)pyridin-3-yl]pyrazolo[1,5-a]pyridine-4-carboxylate 2,7-bis(4-tert-butylpyridin-2-yl)-1,9-dihydrofluoren-1-ide;zirconium(4+) (2S)-5-[3,5-bis(trifluoromethyl)phenyl]-N-[2-chloro-4-nitro-6-(pyridine-4-carbonylamino)phenyl]-1-(2-cyclopropylacetyl)pyrrolidine-2-carboxamide [6-(2,3,5-trihydroxyphenyl)hexylphosphanyl]-(2,4,6-trimethylphenyl)methanone 4-[(E)-2-aminoethenyl]-N-[3-chloro-4-[1-(dimethylamino)ethenyl]phenyl]pyridine-2-carboxamide 2-[[(3S)-1-(2-fluorophenyl)pyrrolidin-3-yl]methylamino]-5,6,7,8-tetrahydro-3H-quinazolin-4-one 2-tert-butyl-4,5-dinitro-1H-imidazole N'-[[5-(4,6-dimethylpyrimidine-2-carbonyl)pyridin-3-yl]methoxy]pyridine-2-carboximidamide 2-(1,3-dithiolan-2-yl)-5,6-bis[(4-fluorophenyl)methoxy]phenol 3-(5-acetamidopyrazin-2-yl)sulfonylbutanoic acid 4-chloro-1-[1-(3,5-dichlorophenyl)ethyl]-3-methylpyrazolo[3,4-d]pyrimidine N'-(2,3-dimethoxyphenyl)-4-[(E)-3-hydroxyprop-1-enyl]benzohydrazide (3S)-2-[4-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]phenyl]-6-cyclohexyloxy-5-methylidene-1-propanoylpiperidine-3-carboxylic acid 2,5-difluoro-N-[(E)-(3,4,5-trimethoxyphenyl)methylideneamino]aniline N-(1-azabicyclo[2.2.2]octan-3-ylmethyl)-4-cyclopropylbenzamide 2-amino-4,6-dimethylpyridine-3-carbonitrile;N,N-dibutylformamide;ethane N-[4-amino-1-[(2R)-3,3-difluoropropanoyl]piperidin-4-yl]-5-cyclopentyl-6-(dimethylamino)pyridine-3-carboxamide 2-azido-1,3-dihydropyrido[3,4-b]indole 2-[5-(3-oxoisoindol-1-ylidene)benzimidazol-1-ium-2-yl]oxyacetic acid 5-methyl-4-oxo-N'-[(3S)-1,2,3,4-tetrahydronaphthalene-1-carbothioyl]-1H-quinoline-3-carbohydrazide N-(2,3-dioxoindol-1-yl)butanamide 4-(3-fluorophenyl)-5-[(1S,2R)-2-propan-2-ylcyclobutyl]oxy-1H-pyridazin-6-one N-[4-methyl-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxamide;hydrochloride 3-[5-amino-2-(4-bromophenyl)-1,3-thiazol-4-yl]propanoic acid (5S)-7-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide (5R)-6,13-bis(ethenyl)-2,3,4,5,14-pentazatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),3,8,10,12,15,17-heptaene 2-[1-(3-aminopropyl)indol-5-yl]-N',N'-diethylbutane-1,4-diamine (E)-1,4-diphenylbut-3-en-2-one N-[6-(2-hydroxyethoxy)pyridin-3-yl]-2-[4-[(E)-[(5-methyl-1,3-thiazol-2-yl)hydrazinylidene]methyl]phenyl]acetamide 1-[3-[2-(difluoromethoxy)phenyl]propylamino]-N-hydroxypentan-2-imine 4-[2-chloro-3-(trifluoromethyl)phenyl]-1H-pyrrole-2-carboxylate 5-[6-(2,4-difluorophenoxy)pyridine-3-carbonyl]-N-methylsulfonyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 1-chloro-N,3-diethyl-4-methoxyindole-2-carboxamide 5-ethyl-2,4-dimethoxy-3-(1-propan-2-ylpyrazol-4-yl)benzaldehyde N-[1-(dimethylamino)pentan-3-yl]-2,6-difluorobenzenesulfonamide 2-[[4-ethylsulfanyl-5-[(2Z,3E)-2-hydrazinylidenepenta-1,3-dienyl]pyridin-2-yl]amino]acetic acid (7S)-2-[[1-[4-fluoro-3-(trifluoromethyl)phenyl]pyrazol-4-yl]methoxy]bicyclo[4.2.0]octa-1(6),2,4,7-tetraene [1-[4-(3-fluorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]cyclohexyl]methanamine;hydrochloride 2-[4-chloro-5,8-dioxo-9-(2,4,6-trifluorophenyl)imidazo[1,2-a]quinoxalin-7-yl]sulfanyl-N-methylacetamide;ethane ethane;6-[[1-[3-(methylamino)-2,4-dioxo-1H-pyrimidine-5-carbonyl]piperidin-3-yl]amino]pyridine-3-carboxamide 4-[[5-(5-chlorothiophen-2-yl)sulfonyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl]methoxy]benzamide 6-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-2,7-dimethylfuro[3,2-c]pyridine 2-[3-(4,6-dimethylpyridine-3-carbonyl)-1,3-oxazolidin-5-yl]acetic acid N-[3-[(2-fluorobenzoyl)amino]phenyl]sulfonylthiophene-2-carboxamide 3-[4-amino-5-fluoro-6-(N'-methylcarbamimidoyl)pyridine-2-carboximidoyl]-N,7-dimethoxy-1H-pyrrolo[3,4-c]pyridine-2-carboxamide 2-[(7S)-3,4-dimethyl-1-oxo-5,6,7,8-tetrahydroisoquinolin-2-yl]-N-[(4R)-4-phenylcyclohexen-1-yl]acetamide 6-[[3-amino-2-[(3R)-3,4-difluoropyrrolidine-1-carbonyl]-5-fluorophenyl]methyl]-8a-ethyl-7-hydroxy-1,5,9,10-tetrahydroimidazo[1,5-b]isoquinolin-2-one 4-(cyclohexyloxymethyl)-1-[2,6-dichloro-3-(2,2-difluoropropanoyl)phenyl]pyrazole-3-carbonitrile N-(2,4-dimethylpentan-3-ylidene)-N'-[1-[(E)-ethylideneamino]piperidin-4-yl]-2-[4-(trifluoromethyl)phenyl]benzenecarboximidamide 1-[3-chloro-4-(2,4-dimethylphenyl)sulfanylphenyl]-5-(trifluoromethyl)pyrazole [5-amino-2-[(3,4-dimethoxyphenyl)methylsulfanyl]pyridine-3-carbonyl]azanium 5-amino-3-(4-fluorophenyl)-6-[2-methyl-6-morpholin-4-yl-4-[(Z)-prop-1-enoxy]pyridine-3-carboximidoyl]pyrazine-2,7-diamine N-[5-tert-butyl-3-(2,4-dioxoimidazolidine-1-carbonyl)cyclohexa-2,4-dien-1-ylidene]benzamide (2S)-3-[4-(4-chlorophenyl)phenyl]-2-methylpropanoate 4-[2-(2,6-dimethylphenyl)imidazo[1,2-a]pyridin-7-yl]-N'-methanimidoylpiperazine-1-carboximidamide 5-[[3,4-bis(hydroxymethyl)phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one 2-(4,5-dihydro-1H-imidazol-2-yl)-3-hydroxy-N'-[N'-[1-(4-methylbenzoyl)piperidin-4-yl]carbamimidoyl]prop-2-enimidamide ethane;N-ethenyl-4-methoxybutan-1-amine;3,6,7,11b-tetrahydro-2H-[1]benzofuro[2,3-a]quinolizine 2-[(2Z,5S)-2-[(Z)-1-phenylethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 5-tert-butyl-2-[[2,6-di(propan-2-yl)phenyl]iminomethyl]-4-isocyanophenol (2E,5R)-2-[(Z)-1-phenylpropylidenehydrazinylidene]-5-phenyl-1,3-thiazolidin-4-one 2-[4-[3,5-dichloro-N-(4-hydroxybutyl)anilino]phenyl]decanoic acid 1-bromo-4,4-dimethyl-7H-pyrazolo[3,4-b]pyridine-5-carboxylic acid N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-(3-ethoxypiperidin-1-yl)sulfonylbenzamide 3-(1,3,2-dioxaborolan-4-yl)-5-fluoro-8-methoxy-[1,2]oxazolo[5,4-c]quinoline N-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[2-[3-(trifluoromethyl)phenyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-5-carbonyl]benzamide 2-[(3S)-2-oxo-1,4-diazepane-3-carbonyl]isoquinolin-1-one 5-methylsulfonyloxypyrazine-2,3-dicarboxylic acid 2-amino-4-[3,5-dibromo-4-(5-phenylpentoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile (4-methylphenyl)-(2H-1,3,5-triazin-1-yl)diazene 2-(3,5-dimethylphenyl)sulfanyl-N'-hydroxy-6-methylpyrimidine-4-carboximidamide (E)-3-(2,4-dichlorophenyl)-N-[2-(2-fluoroethoxy)ethyl]-3-[4-methylsulfonyl-2-(trifluoromethyl)phenoxy]prop-2-enamide 4-[N-(2-phenylethyl)-4-propylanilino]benzenesulfonic acid 3-(2-aminoethyl)-N,5-dicyclopropylaniline 1-[2-(4-hydroxycyclohexyl)ethynyl]-3,7-dimethylpurine-2,6-dione (1R)-4-[(2R,3R)-3-cyclopentyloxy-2-hydroxy-3-methylbutanoyl]-1-prop-2-enyl-2,3-dihydro-1H-indene-5-carboxylic acid 1-(3,6-diaminopyrazin-2-yl)ethenethiol;3,7-dimethoxyquinoxalin-2-amine N-[2-[(3S,4R)-3-amino-4-fluoropiperidin-1-yl]pyridin-4-yl]-5-cyclopropyl-3-methoxypyridine-2-carboxamide 1-[3,4-dichloro-2-(trifluoromethyl)phenyl]pyrazole 2-[4,6-di(butanoyl)-1H-benzimidazol-2-yl]-3-methoxy-5-sulfamoylphenolate;rhodium(3+) 2-(4-methoxycarbonyl-N-methylsulfonylanilino)propanoic acid 3-amino-N-(2,6-dimethylphenyl)-5H-pyrrolo[2,1-c][1,4]benzoxazine-7-carboxamide 7-bromo-5,8-difluoro-3H-quinazolin-4-one 2-[5-(1H-pyrrol-3-yl)-1,2,4-oxadiazol-3-yl]thiophen-3-ol (1R)-2,3-dichloro-1-ethoxycarbonyl-1-[3-fluoro-5-(trifluoromethyl)pyridin-2-yl]cyclopropane-1-carboxylic acid N-methylsulfonyl-3-[4-(trifluoromethoxy)phenyl]propanamide 4-[[2-[[5-tert-butyl-3-(2,6-dichlorophenyl)pyrazol-1-yl]methyl]phenyl]carbamoylamino]benzoic acid (6R)-6-butyl-6H-benzo[c]chromene 3-[6-(dimethylamino)pyridin-2-yl]-2-phenyl-4H-chromene-5,7-diol (E)-N-[2-[5-[4-(3,5-dimethylpyrazol-1-yl)-2-methoxyphenyl]-6-fluoropyridin-3-yl]ethyl]-4-(dimethylamino)but-2-enamide N-[(4R)-1,3,4-oxadiazol-2-yl]-N'-pyridin-2-yl-N-(2,2,6,6-tetramethylpiperidin-4-ylidene)ethanimidamide (2R)-3,3-dimethyl-1-(2-phenylpyrrolidin-1-yl)butan-2-amine;formic acid 3-bromo-2-[3-chloro-4,5-bis(ethoxycarbonyl)pyridin-1-ium-1-yl]-6-methylbenzoate 2-(3,4-dimethylphenoxy)-N'-hydroxypyrimidine-4-carboximidamide 2-methoxy-5,8-dihydropyrimido[4,5-d]pyrimidine-7-carboxylic acid N-[2,4-dichloro-3-[(7-chloroquinolin-6-yl)methoxy]phenyl]benzenesulfonamide 2-[5-(4,4-difluoropiperidin-1-yl)-3-ethanimidoylpyrazolo[1,5-a]pyrimidin-7-yl]phenol 2-[(3S,7S,8aS)-7-hydroxy-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]-N-[(4,5-dimethylfuran-2-yl)methyl]acetamide [4-[5-[1-amino-6,7-dimethyl-2-(oxolan-3-yl)benzimidazole-5-carbonyl]pyrimidin-2-yl]piperazin-1-yl]-phenylmethanone 4-azido-1-(2,5-dichlorophenyl)imidazole 5-chloro-1'-[(2,3-difluorophenyl)methyl]spiro[2H-1-benzofuran-3,4'-piperidine] 2-(4-chloro-3,5-dimethylphenyl)benzenethiol 2-tert-butyl-6-[(3,5-diphenyl-1,2,4-triazol-1-yl)methyl]-4-phenylpyridine 4-[2,5-dimethoxy-3-(pyrrolidine-1-carbonyl)phenyl]oxane-4-carbonitrile 4-[3-(1H-imidazol-2-yl)-5-pyridin-4-yloxyindol-1-yl]phenol 4-[2,5-dimethyl-1-(oxan-4-yl)imidazol-4-yl]pyridine 4-[5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl]phenol 3-(4-chlorobenzoyl)-N,2-dimethyl-N-(1H-pyrazole-5-carbonyl)indolizine-8-carboxamide 3-azido-N,5-di(propan-2-yl)benzamide 6-chloro-1,3-dihydrobenzimidazol-2-one;2-[(2S)-2-cyclohexylpyrrolidin-1-yl]-5-ethylpyridine (3aR)-1-[2-(4,6-difluorocyclohexa-1,5-dien-1-yl)ethynyl]-7-phenylmethoxy-3a,9b-dihydroindeno[1,2-b]pyrrole 2-(N-ethyl-4-nitroanilino)benzoic acid 2-[4-chloro-3-fluoro-1-[[3,4,5-trifluoro-6-(2,2,2-trifluoroethoxy)pyridine-2-carbonyl]amino]cyclohexa-2,4-dien-1-yl]oxyacetic acid 2-benzyl-N'-(1,3-thiazol-4-yl)butanediamide 2-[(1,5-dimethylpyrrolidin-3-ylidene)amino]-5,7-difluoroquinolin-8-amine 4-(2-azidoethyl)-3-methoxybenzenesulfonamide 2-[N-(1,3-thiazol-5-yl)anilino]octanoic acid (5Z)-2-(4-methoxyphenyl)imino-5-[(3,4,5-trihydroxyphenyl)methylidene]-1,3-thiazolidin-4-one 1-[4-(6-methylpyridin-3-yl)cyclohexanecarbonyl]azetidine-2-carboxamide [3-[(4-tert-butylphenyl)methoxy]pyrazin-2-yl]carbamic acid (E)-3,7-diethyl-9-hydroxy-4-phenylnon-8-enal [4-[2-(3,5-difluorophenoxy)ethyl]piperazin-1-yl]-[4-(2-pyridin-4-ylethoxy)phenyl]methanone 4-[[(1S)-1-aminopropyl]-[3,5-bis(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carboxylic acid 1-(2,6-dimethylphenyl)-3-[1-(4-fluorophenyl)ethylideneamino]urea N-[(2R)-3-hydroxy-1-phenylpropan-2-yl]-4-(3-methylsulfanylphenyl)pyridine-2-carboxamide 4-[[6-(dimethylamino)pyridin-3-yl]amino]-2,5-difluorobenzoic acid (4S)-5-[4-bromobutyl-(4-methoxybenzoyl)amino]-2,6-dihydroxy-3,3-dimethylheptanoic acid 2-[(3R,4S)-4-[(8-amino-1-hydroxyquinolin-6-yl)methyl]-1-[3-(3-aminophenyl)propanoyl]piperidin-3-yl]acetamide;dihydrochloride N-methyl-4-(oxan-3-ylamino)-3,5-dinitrobenzenesulfonamide 2-(6-ethyliminocyclohexa-1,3-dien-1-yl)benzo[g][1]benzofuran-4,5-dione 1-[(5R)-1,3,4-trihydroxy-6-methylheptan-2-yl]pyridin-2-one [3-hydroxy-4,6-bis(phenyliminomethyl)cyclohexa-2,4-dien-1-ylidene]azanide (5Z)-2-imino-3-[2-[4-[2-(1H-indol-5-yloxy)ethyl]piperidin-1-yl]pyrimidin-4-yl]-7,8-dihydro-6H-quinoline-1-carboxamide 5-fluoro-2-[(2-nitrophenyl)methyl]pentanamide 3-[5-(aminomethyl)-4H-pyridin-1-yl]-1,2,6-triazin-5-amine N-[4-hydroxy-1-(2,3,5-trimethylphenyl)butan-2-yl]-2-propyl-6-pyridin-3-ylpyridine-4-carboxamide 5-[(3S)-3-methoxypyrrolidine-1-carbonyl]-2,4-dimethylpyridine-3-carboxamide N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-2-phenylacetamide N-[2-(3,4-dichlorophenyl)ethyl]-7-hydroxy-5H-pyrrolo[1,2-a]quinoxaline-4-carboxamide 3-chloro-5-(2,4-difluorophenyl)-6-ethylsulfonylimidazo[2,1-b][1,3]oxazole 3-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde 2-azidooxy-4-[3,5-difluoro-4-(trifluoromethyl)phenoxy]-1-nitrobenzene N-[(3E,5Z)-2,4,7-trichlorohepta-1,3,5-trien-3-yl]sulfanyl-1-thiophen-3-ylmethanamine 1-(5-tert-butyl-2,3-dimethoxyphenyl)hexan-1-one 1-[5-(2-aminophenyl)-7,8-dihydropyrido[4,3-d]pyrimidin-6-yl]propan-1-one;hydrochloride (Z)-but-2-ene;ethane;(E)-N-ethenyl-3,4-dimethylhept-1-en-3-amine;4-[6-fluoro-2-(2-hydroxyphenyl)quinoline-4-carboximidoyl]aniline 4-[5-[3-(2,2-dimethylpropyl)-5-[1-(fluoromethoxy)ethenyl]phenyl]-6-methylidenecyclohexa-2,4-dien-1-ylidene]-N,N-dimethylbutan-1-amine 2-[(3-tert-butylphenyl)methylidene]propanedinitrile N-[4-(2,3-dihydrofuran-2-yl)phenyl]-5-fluoronaphthalene-1-carboxamide (4-methylphenyl)sulfanylamino-[2-[[2,3,5-trifluoro-4-[6-fluoro-7-[4-(trifluoromethoxy)phenyl]quinazolin-8-yl]benzoyl]amino]ethoxy]azanium [3-[amino-[(E)-2-(5,7-dichloroquinolin-6-yl)ethenyl]sulfamoyl]phenyl]methylideneazanium 2-(1,3-benzothiazol-2-ylamino)-6-chloropyridine-4-carboxylic acid 1-[(2S)-5,7-dibromospiro[1H-indole-3,4'-piperidine]-2-yl]-N,N-bis(methoxymethyl)methanamine 2-bromo-N'-(5,6-dimethylpyridin-3-yl)-1,3,4-thiadiazole-5-carbohydrazide 2,4-dichloro-5-nitro-N-(3-phenylpropyl)benzenesulfonamide 3-fluoro-5-(2-fluoroethoxy)benzamide [5-(3,4-dimethoxyphenyl)tetrazol-2-yl]methanamine;3H-1,3,4-thiadiazole-2-thione (5S)-N-[3-cyano-6-(2,4-difluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-5-yl]-5-methyl-2-(4-oxo-3H-phthalazin-1-yl)hexanamide 2-ethenyl-1,3-difluoro-6-[4-(4-prop-2-enoxyphenyl)cyclohexa-2,4-dien-1-yl]naphthalene (5Z)-2-[3-chloro-4-methoxy-5-(trifluoromethyl)phenyl]imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one 1-(2,4-difluorophenyl)sulfinylindole-3-carboxylic acid N-[[4-(N'-hydroxycarbamimidoyl)phenyl]methyl]prop-2-enamide 4-amino-6-[(2,3-dimethoxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one N-[1-(3,5-difluoropyridin-2-yl)piperidin-4-yl]-5-methoxy-6H-azepine-7-carboxamide 1-(1,4-dioxan-2-yl)-3-[3-fluoro-5-(trifluoromethoxy)phenyl]urea 3-(2-aminophenyl)-1-[4-(2,5-difluorophenoxy)piperidin-1-yl]propan-1-one 2-(6,7-dimethoxyquinazolin-4-yl)-5-methylpyrazole-3-carboxylic acid 2-amino-3,4,5-tribromophenol [[1-(difluoromethoxy)-3,6,6-trihydroxy-7-methylocta-2,4,8-trienylidene]amino]sulfonylurea 2-methoxy-4-[1-(4-methylphenyl)-1,2,4-triazol-3-yl]aniline ethane;2-hydroxy-3-(phenylmethoxycarbonylamino)propanoic acid N-[(Z)-1-amino-3-hydroxy-4,4-dimethylpent-2-enylidene]-5-fluoropyridine-3-carboxamide 6-(3,4-dihydroxyphenyl)-N-[3-[ethyl(2-pyridin-2-ylethyl)amino]propyl]benzo[b][1,4]benzothiazepine-3-carboxamide (E)-2-[4-[(Z)-(3,7-dimethylquinolin-2-ylidene)amino]piperazine-1-carbonyl]pent-2-enal 1-(3,4-difluorophenyl)-2H-pyridine;hydrochloride 5-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]imidazolidine-2,4-dione 3-(8-phenylimidazo[1,2-a]pyrazin-6-yl)-7-propan-2-ylindolizine (2E)-3-[[4-(1,3-dioxolan-2-ylmethoxy)-3-ethoxyphenyl]methylidene]-6,6-bis(ethoxymethyl)morpholine 1-(2,4-difluorobenzene-6-id-1-yl)-N'-methanimidoyl-3-methyl-7-(trifluoromethyl)indole-5-carboximidamide;uranium(2+) 2-chloro-1,4-dimethylbenzene;ethane N-[4-[(2,4-dichloropyrimidin-5-yl)-octylamino]phenyl]sulfonylbenzamide 2-amino-4,7-dioxo-5-(3-propoxynaphthalen-1-yl)-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile 6-(cyclohexen-1-yl)isoquinoline 2-[5-[5-chloro-6-(cyclopropylsulfonylamino)pyridin-3-yl]-4-fluoropyrazol-1-yl]acetic acid 2-(4-aminophenyl)benzene-1,3-dicarboxamide;hydrochloride N'-[2,5-difluoro-4-(1H-imidazol-5-yl)phenyl]-N-ethylbutanediamide N-[6-(difluoromethoxy)-3,4-dihydro-2H-chromen-8-yl]prop-2-enamide 2-[3-(2-methoxyethylamino)azetidin-1-yl]sulfonylphenol 2,4-bis(2,3-dihydro-1H-inden-5-yl)quinazoline;ethane 1-[(2R)-1,4-dioxan-2-yl]-3-[6-(oxolan-3-yl)pyridin-2-yl]urea 2-[4-[(3S)-3-[[methyl(propan-2-yl)carbamoyl]amino]piperidine-1-carbonyl]phenoxy]acetic acid 1-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-en-1-one 4-N,5-N-bis(1H-indol-2-yl)-[1,3]thiazolo[5,4-d]pyrimidine-2,4,5,6-tetramine;dichloride 4-[(E)-2-(2,5-dimethylfuran-3-yl)ethenyl]-2-(thiophen-2-ylsulfanylamino)benzonitrile 4-[1,4-dimethyl-5-[(4-methylphenyl)sulfonylamino]pyrazol-3-yl]-2-fluorobenzoic acid 4-(aminomethyl)-2-[1-[6-[[[(3S)-3-hydroxypyrrolidin-1-yl]amino]methyl]pyridine-3-carbonyl]piperidin-4-yl]-1H-pyrimidin-6-one;dihydrochloride (4aR,6R)-1-(cyclopropylmethoxymethyl)-N'-[(2-fluorophenyl)methyl]-6-methoxy-3,4,4a,5,6,7,8,8a-octahydro-2H-isoquinoline-6-carboximidamide;dihydrochloride 2-[4-chloro-2-[5-methyl-2-[(1-propan-2-ylpyrazol-3-yl)amino]pyrimidin-4-yl]phenoxy]acetonitrile;ethane 2-methyl-4-[5-(1,2,4-triazol-1-yl)pyridin-3-yl]quinazoline 2-(2-bromophenyl)pentanedioic acid (3S)-7-[1-benzyl-4-hydroxy-5-(4-methoxyphenyl)imidazol-2-yl]-3,4-dimethyl-3H-1,4-benzothiazin-2-one 5-amino-4-[2-(3,5-difluorophenyl)ethyl]-1H-pyrimidin-6-one ethane;2-(5,6,7,8-tetrahydronaphthalen-1-yl)thiophene 1-[5-(4,6-diaminopyridine-3-carbonyl)-2-methylphenyl]propan-1-one 2-(3,5-dimethoxyphenyl)-4-methyl-6-oxo-1H-pyrimidine-5-carboxylic acid 2-cyclohexyloxy-3,6-bis(3-ethylcyclopenta-1,4-dien-1-yl)phenol N-[2-(4-methylphenyl)ethyl]-6,7-dihydrobenzo[d][1]benzazepine-11-carboxamide 4-chloro-3-[2,6-dimethyl-4-(trifluoromethyl)phenyl]-5-fluoropyridine 2-[4-(cyclohexylmethoxy)piperidin-1-yl]-6-methoxypyrazine N-[4-[(1R)-1,2-bis(5-methylthiophen-2-yl)ethyl]phenyl]acetamide 1-[2-(3-bromo-4-methylphenyl)morpholine-4-carbonyl]cyclobutane-1-carbonitrile 2-[(4Z,7Z)-5,8-dimethyldeca-1,4,7,9-tetraen-3-yl]-5-ethylsulfanyl-1H-imidazole 1-(3,4-dichlorophenyl)-2-[6-methyl-5-(methylideneamino)-1H-indazol-3-yl]ethanone 2-[(2Z,5R)-4-oxo-2-[(Z)-(3-propan-2-yloxyphenyl)methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 5-chloro-6,8-difluoro-4H-1,3-benzothiazin-2-amine 2-[4,5-bis(4-chlorophenyl)-3H-1,4-benzodiazepin-2-yl]-N-cyclohepta-1,3,6-trien-1-ylacetamide 1-[4-methylsulfanyl-3-(trifluoromethoxy)phenyl]pyrazole N-[4-chloro-2,6-di(propan-2-yl)phenyl]formamide 1-[(2R,4R)-2-methyloxolan-3-yl]pyrimidine-2,4-dione N-[4-[(3Z)-5,6-dimethoxyhepta-1,3,5-trien-2-yl]phenyl]-4-ethynylpyridine-3-carboxamide N-[(3S)-4-hydroxyoxolan-3-yl]-2,5,6,7-tetrahydro-1H-pyrrolizine-8-carboxamide 2-[4-(2-phenylethyl)piperidin-1-yl]ethanol 3-[[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]methoxy]cyclohexane-1-carboxylic acid N-(1,3-benzodioxol-5-ylmethoxy)-4-[(2Z,6E)-7-chloro-10-methoxy-3-methyl-2,3-bis(prop-2-enylidene)azocin-1-yl]aniline (7S)-N-(2,4-dimethylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 1-phenyl-4-[2-(10H-phenothiazin-5-yl)acetyl]piperazine-2,6-dione (6R)-3,4-dimethyl-7-[(2E,5Z)-6-propan-2-ylhepta-2,5-dienoyl]-10-sulfanylidene-6,8,9,11-tetrahydro-1H-pyrazolo[3,4-a]acridin-13-one 5-[4-(3,7-dioxa-11-azaspiro[5.6]dodecan-11-yl)phenyl]sulfonyl-N-ethoxypyridin-2-amine 4-(4-chlorophenyl)-2-[4-(3,5-dibromocyclohexa-1,3-dien-1-yl)oxyanilino]pyridine-3-carbonitrile 5-(1,3-dioxolan-2-yl)-3H-pyrano[4,3-d]pyrimidine 1-(2,4-dimethoxyphenyl)-N-[3-[6-(2-hydroxypropan-2-yl)pyridin-3-yl]imidazo[1,2-a]pyrazin-8-yl]ethenesulfonamide N-[(1S,3R)-2,2-dichloro-3-[4-fluoro-3-(trifluoromethyl)phenyl]cyclopropanecarbonyl]-N'-[4-fluoro-5-(methylideneamino)thiophen-2-yl]ethanimidamide 2-[4-methoxycarbonyl-N-(2-methylpropanoyl)anilino]-4-methylpentanoic acid 4-(2-fluoro-6-methylpyridin-3-yl)morpholine;dihydrochloride 1-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-8-(1H-imidazol-5-yl)-N,N-bis(3-morpholin-4-ylpropyl)quinoxalin-6-imine 2-(4-methoxyphenyl)-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]cyclopropane-1-carboxamide (1R)-2,2,4-trimethyl-8-(pyridine-3-carbonyloxy)-3,5-dihydro-1H-pyrido[1,2-e]thiazine-6-carboxylic acid 5-methyl-3-[(2-oxopiperidin-1-yl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-4-one 3-amino-2-[2,6-difluoro-4-(trifluoromethyl)phenoxy]-6H-furo[3,2-e]indole-7-carboxamide N-azido-2,3-dichloro-1H-inden-4-amine N-cyclopentyl-2-[3-(1-methylpyrazol-4-yl)indolizin-1-yl]acetamide;2,2,2-trifluoroacetic acid 5-[4-(trifluoromethyl)phenyl]-3H-pyrrole-2,4-dione 4-[5-(2,3-dihydrofuran-5-yl)thiophen-2-yl]-5-methylidene-1H-imidazol-2-amine 5-[3-(4-chlorophenyl)cyclobutyl]oxy-3H-quinazolin-4-one 4-[1-(pyridine-3-carbonyl)piperidin-4-yl]oxybenzonitrile;5,6,7,8-tetrahydronaphthalen-2-ol 4-amino-6-[(2,3,5,6-tetrafluorophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 6,7-dimethoxy-1-(4-methylphenyl)sulfonylisoquinoline 2-(3,4-dihydroxyphenyl)sulfanyl-5-[(4Z)-4-hydroxyiminobutoxy]benzonitrile N-azido-1-(2,3-dichlorophenyl)ethanamine 3-fluoro-2-[4-(1H-indol-2-yl)anilino]-N-methyl-N-oxobenzamide (2S)-3-(3-cyclopropylindol-1-yl)propane-1,2-diol;1-(4-fluorophenyl)-N'-[5-[methyl(sulfanyl)amino]pentyl]piperidine-4-carboximidamide 4-(diethylamino)-2,5-bis[(4-hydroxyphenyl)methyl]phenol ethane;4-[(E,3Z)-4-iminohex-1-enyl]benzaldehyde N-(3,5-dichlorophenyl)-N-(2,6-dibromopyridin-4-yl)butanamide 2-methyl-3,4-bis(2-methylphenyl)phenol N'-[(Z)-2-[3,5-dichloro-4-(hydroxymethyl)phenyl]ethenyl]ethanimidamide 1-[2-(3,4-dimethylphenyl)ethynyl]cyclohexan-1-ol 6-methoxy-2,4-dimethyl-N-phenylpyridine-3-carboxamide [4-methyl-6-(4-oxospiro[3,5-dihydrochromene-2,4'-piperidine]-1'-yl)pyrimidin-2-yl]methanesulfonate 1-[(6R)-3,6-difluorocyclohexen-1-yl]-N-[[4-(2,4-dimethylphenyl)sulfonyl-5-ethoxythiophen-2-yl]methyl]propan-2-amine 1-azidooxy-6,7-dihydroxyisoquinoline-4-carbonitrile (2S,3aS,7aR)-6-[(4-methylphenyl)sulfonylamino]-N-(thiophen-2-ylmethyl)-3,3a,5,6,7,7a-hexahydro-2H-furo[3,2-b]pyridine-2-carboxamide [1-(3,5-dichloropyridine-4-carbonyl)piperidin-2-yl]-thiomorpholin-4-ylmethanone (4R)-1,3-bis[2,6-dichloro-4-(1H-pyrazol-5-yloxymethyl)phenyl]-4-propan-2-ylimidazolidin-2-one 2-[(1R,6S)-3-azabicyclo[4.1.0]heptan-3-yl]-5-phenyl-1,3,4-oxadiazole (2S,3S)-4-cyclobutyl-N-[2-fluoro-5-(propanoylamino)phenyl]-1-methyl-3-sulfamoylpyrrolidine-2-carboxamide 2-[4-(3-acetylphenyl)cyclohexyl]-2-aminopentanoic acid 3,6-diamino-N'-propanoylpyrazine-2-carboximidamide 4-[[2,6-dichloro-3-(ethoxymethyl)phenoxy]methyl]benzonitrile 3-(2,5-dimethoxyphenyl)-N'-hydroxyprop-2-enimidamide N-[5-chloro-4-(3,5-dimethyl-1H-pyrazol-2-ium-4-yl)pyrimidin-2-yl]-6-fluoroquinoline-8-carboxamide (7R)-6,11-dihydroxy-9,10-dioxo-4-oxa-1,8-diazatricyclo[8.5.0.02,7]pentadeca-10,13-diene-16-carboxylic acid 2,3-bis(4-chlorophenyl)-1H-indole 1-(2,3,4a,5,6,7,8,9b-octahydrobenzo[e]indol-1-yl)-N-methylpentan-1-imine N-(cyclohexylmethyl)-N'-[2,6-di(propan-2-yl)phenyl]ethane-1,2-diamine 4-[4-(dimethylamino)butyl]benzenecarbothioamide (5E)-2-cyclopentylimino-5-[[4-(dibutylamino)phenyl]methylidene]-1,3-thiazolidin-4-one 4-[3-(cyclobutylmethoxy)azetidin-1-yl]sulfonylbenzoic acid N-methyl-1-[2-(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanylacetyl]piperidine-3-carboxamide (E)-3-[4-[[6-chloro-2-hydroxy-1-(methoxymethyl)indol-3-yl]diazenyl]phenyl]but-2-enoic acid 3-ethenyl-2,5-dimethoxybenzoic acid 6-(2,3-dihydro-1H-inden-5-yl)-4-N-[3-methoxy-4-(2-pyrrolidin-1-ylethylamino)phenyl]pyrimidine-2,4-diamine 1-[4-(2,3-dihydrothiophene-5-carbonylamino)phenyl]piperidine-4-carboxamide;dihydrochloride 3-[[1-(4,4-difluorocyclohexyl)sulfonylpiperidin-2-yl]methoxy]pyridine 1-[4-(2,4-difluorophenyl)piperazin-1-yl]ethanone;ethane 1-[2-(5,5-dimethylcyclohepta-1,3-dien-1-yl)ethyl]-2H-indazole 3,6-diamino-1-[3-(4-methoxyphenyl)propyl]indole-5-carboxylic acid (2S)-4-amino-2-[(3R)-1-ethylsulfonylpiperidine-3-carbonyl]-5-phenylmethoxypentanamide 4-methyl-2-[5-(trifluoromethyl)pyridin-3-yl]quinoline 1-[5-(2,4-difluorophenyl)sulfonylpyridin-3-yl]-6-methoxy-2H-quinazoline 1-[4-(dimethylamino)phenyl]pyrrolidine-2,5-dione 1-[1-(4-tert-butylphenyl)ethenyl]piperidine 4-tert-butyl-2,6-bis[(3-methoxyphenyl)iminomethyl]phenol 2-[6-chloro-1-methyl-4-oxo-7-(3,5,6-trimethylpyrazin-2-yl)quinolin-3-yl]acetaldehyde;ethane;N-ethylmethanamine 2-benzyl-7-chloro-4H-azepine N-[4,5-bis(phenylmethoxy)-2H-pyran-6-yl]pentanethioamide 1-(3-chlorophenyl)sulfonyl-4,5,6,7-tetrahydropyrazolo[3,4-c]pyridine 4-[2-(cyclobutylmethyl)piperidin-1-yl]-2,5-difluorobenzoic acid 3-[1-[2-(oxan-4-yloxy)ethyl]imidazol-2-yl]quinoline (2S)-1-[4-(3,5-dichlorophenyl)benzoyl]pyrrolidine-2-carboxylic acid 6-bromo-8-fluoro-1H-quinoline-2,4-dione 5-azido-6-methyl-1,3-diphenylpyrazolo[4,3-d]pyrimidine 3-[(E)-2-pyridin-4-ylethenyl]-1H-indazole 4-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-2-(methylamino)-5-[(Z)-prop-1-enyl]phenol N-(5,6-dichlorobenzimidazol-1-yl)hydroxylamine 6-[5-(2-pyrrolidin-1-ylethoxy)pyridin-3-yl]quinoline N-(2,6-dimethylphenyl)-N-[5-[1H-imidazol-5-ylsulfonyl(phenyl)methylidene]pyrrol-3-yl]hydroxylamine (5Z,7E)-6-amino-1-[4-methyl-2-[(4-phenoxyphenyl)methoxy]piperidin-1-yl]nona-3,5,7-trien-1-one N-(4-ethenyl-3,5-dimethoxyphenyl)hydroxylamine 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]-6-iodophthalazin-1-one 4-(3,5-dichlorophenyl)-2,6-dioxo-1,3-diazinane-5-carbonitrile 4-(2,6-dimethylphenyl)iodanuidylcarbonylbenzonitrile 2-[6-(4,5-dihydroimidazol-1-yl)imidazo[1,2-b]pyridazin-2-yl]acetamide N-(1,3-benzodioxol-5-yl)-1-methylpiperidine-4-carboxamide 3-[[5-(3,4-dichlorophenyl)pyridine-2-carbonyl]amino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid (3R)-1-[(2S,3R)-4-(3,5-difluorophenyl)-4-imino-1-methylpyrrolidine-2-carbonyl]piperidine-3-carboxylic acid (NE)-N-[(3-chloro-2,5-difluorophenyl)methylidene]-4-ethylbenzenesulfonamide 3-[4-(6,7-dihydroquinolin-5-yl)triazol-1-yl]-2-hydroxypropanoic acid N-(furan-2-ylmethyl)-6,7-dihydrodibenzothiophen-1-amine N-[2-bromo-4-chloro-6-(trifluoromethyl)phenyl]-3-cyclopentylpropanamide 5-chloro-1H-indole;3-[3-[4-(5,6-dihydro-2H-thieno[2,3-b]pyran-3-ylmethoxy)phenyl]propanoylamino]-N-hydroxypentanamide 3-[4-(2,6-diphenylpyrimidin-4-yl)dibenzofuran-1-carboximidoyl]aniline [4-(3-iodophenoxy)phenyl]-methyl-methylideneazanium [4-(3-methoxycarbonylphenyl)-1H-pyrrole-2-carbonyl]iodanium 2-methoxy-4-methylsulfonylbenzenethiol 1-(5-azidothiophen-2-yl)sulfonylpiperidine 2-methyl-3,4-dihydropyrido[1,2-a]pyrazine;5-[6-methyl-5-(trifluoromethoxy)pyridin-2-yl]imidazolidine-2,4-dione 5-[3,5-dichloro-4-(1,2,3,4-tetrahydronaphthalen-1-yloxy)phenyl]-1-methylpyrazole 2-(5-phenylmethoxy-1,3-dihydroisoindole-2-carbonyl)benzamide N-[5-fluoro-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]-2-fluoroacetamide N-[(3,4-dichlorophenyl)methyl]-3-[2-(1H-imidazol-5-ylmethylideneamino)ethoxymethyl]aniline 2-[1-(6,7-dimethoxyquinolin-4-yl)piperidin-3-yl]-N-ethylacetamide 5-hydroxy-4-[3-(1,2,4-triazol-1-yl)propanoylamino]pent-4-enoic acid 3-[3,5-difluoro-4-(trifluoromethyl)phenyl]azetidine 1-[2-cyclopropyl-4-(6,7-dihydropyrrolo[3,2-c]pyridine-5-carbonyl)phenyl]pyrrolidin-2-one 2-[(5,6-dimethoxypyridine-3-carbonyl)amino]acetic acid 3-[2,3-dihydroxypropyl(hexyl)amino]phenol (1S)-N,4-dimethyl-2-phenylcyclohexa-2,4-dien-1-amine 1-[4-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethoxy)phenyl]ethanone 5-methyl-4,6-diphenyl-2-(triazin-4-yl)pyridine-3-carbonitrile ethane;1-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-4-(phenylmethoxymethyl)imidazole 1-azidooxy-2,4,5-trimethyl-3H-fluorene 6-[(3R)-5-oxo-1-[(3S,4R)-4-phenylpyrrolidin-3-yl]pyrrolidin-3-yl]oxypyridine-2-carbonitrile 2-[(1R)-1-(4-fluorophenyl)ethyl]imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one 2-[(6S)-3,5-dimethyl-1H-inden-2-yl]propanal (1S,2R)-2-azido-N,4-dibenzylcyclopentan-1-amine 2-[4-chlorobutyl-(5-nitro-1,3-thiazol-2-yl)amino]acetic acid 3,4-dimethylpyridine;N,N-dimethylmethanamine;5-[4-(ethoxyiminomethyl)phenyl]pyrimidine 4-benzyl-2-(pyridin-3-ylmethylidene)morpholine (3R,5S)-1-[2,6-dimethyl-4-(methyliminomethyl)phenyl]piperidine-3,5-diamine 5-[2,6-dimethyl-4-(trifluoromethoxy)phenyl]-1,3-oxazole 6-chloro-1,3,4,5-tetrahydropyrido[3,2-h][1,7]naphthyridin-2-one N-[4-(2,4-dimethylphenyl)butyl]hexanamide N-[2-[(3R)-4,5-bis(4-chlorophenyl)morpholin-3-yl]ethyl]-5-[(4-methylpiperazine-1-carbonyl)amino]-2,3-dihydroindole-1-carboxamide 3-(2,6-dimethoxypyridin-4-yl)azepane;ethane 2-bromo-6-(1H-1,2,4-triazol-5-yl)aniline 4-(2,3,5,6-tetrafluorophenoxy)phenol 1-(6-fluoro-7-methyl-3,4-dihydro-2H-chromen-2-yl)pyrrolidine N-[2,4-dichloro-5-[(2E)-3,7-dimethylocta-2,6-dienoxy]phenyl]-5-oxo-1,4-dihydro-1,2,4-triazole-3-carboxamide 1-amino-5-(benzenesulfonyl)octan-2-ol [4-(2,3-diphenylpropyl)piperazin-1-yl]-(1H-pyrazol-5-yl)methanone N-[4-(3,4-dichlorophenyl)butanoyl]-2,6-dimethylbenzamide [2-[3,5-bis(trifluoromethyl)phenyl]ethoxymethyl-difluorophosphaniumyl]methyl-diethynylphosphinate 2-N-[3,4-bis(ethenyl)phenyl]quinoline-2,4-dicarboxamide 2-(azidomethylsulfanyl)-1,3,4-trifluorobenzene 2-chloro-N-diazo-4-(trifluoromethyl)benzenesulfonamide 2-amino-N'-[(2Z,4E)-6-chlorohepta-2,4,6-trien-3-yl]-5-(1,4,5-oxadiazepan-4-yl)benzenecarboximidamide;propane N-[4-(2,5-dimethylphenyl)-1,3-thiazol-2-yl]-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]sulfanylhydroxylamine;4-methoxybutan-2-one N-(4,5-dimethyloxolan-2-yl)-1-[(6R)-4,8,10-triazatricyclo[7.3.0.02,6]dodeca-1,9,11-trien-4-yl]benzimidazole-4-carboxamide 6-(4-tert-butylphenoxy)benzene-1,2,3,4,5-pentol 5-[(E)-2-amino-4,4-dimethylhex-3-enoxy]carbonylpyridine-3-carboxylic acid 1-(2,6-diethylphenyl)-3-[(E)-(3-hydroxyphenyl)methylideneamino]urea 4-[6,8a-dihydrobenzotriazolo[1,5-a]pyrazine-7-carbonyl(propyl)amino]butylcarbamic acid 5-[2-(4-methoxyphenyl)ethyl]-3,6,9,12-tetrazatricyclo[8.7.0.03,8]heptadeca-1(10),11,13,15-tetraen-4-one (2S)-3-[4-methyl-N-[(2R)-1,1,1-trifluoropropan-2-yl]anilino]-2-phenylpropanenitrile 6-[(2E,4Z)-hexa-2,4-dien-3-yl]-1-methylbenzimidazole 3-amino-1,4-bis[(2S)-4-methyl-2-propan-2-ylpiperazin-1-yl]butane-1,4-dione 7-[4-hydroxy-3,5-bis(prop-2-enyl)phenyl]-5-methoxyheptanenitrile (4Z)-2-methyl-3-pentan-3-ylidene-5-phenylcyclohexene [2-amino-5-[(6-ethoxypyridin-3-yl)methylcarbamoyl]phenyl]methylideneazanium N-[2,3-difluoro-5-(4-sulfanylpiperidin-1-yl)phenyl]-3-methoxyquinoxaline-6-carboxamide;5,7-dihydropyrrolo[3,4-b]pyridin-9-one (2R)-4,5-dihydroxy-2-[(3E)-5-hydroxyocta-1,3,7-trien-6-yn-3-yl]oxy-6-[(E)-2-methoxyethenyl]-8-(3-methoxyphenyl)-7-propan-2-yloxychromen-2-one 6-methyl-4-[3-(methylamino)-1H-pyrazole-5-carbonyl]piperazin-2-one 3,5-dimethoxy-4-[5-methyl-2-(2H-tetrazol-5-yl)phenyl]-1,2-oxazole 2-azido-1-(7-chloro-6-methoxynaphthalen-2-yl)ethanone 2-(2,6-difluorophenyl)-3-methyl-4H-pyrimido[1,2-a]pyrimidine 4-bromo-2-[(E)-2,3-dimethylbut-1-enyl]aniline N-[(1R)-3-methyl-1-(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)butyl]-2-thiophen-2-ylacetamide 3,4-dimethyl-5-(3-methylbutoxy)benzoic acid;ethane 2-[4-(dimethylamino)phenyl]-3,5-difluoro-6-methoxy-1H-quinolin-4-one N-azido-3,5-difluoro-4-[(1S)-1-methoxyethyl]benzamide (2S)-2-[4-(trifluoromethoxy)phenyl]piperidine 4-[2-chloroethyl(propyl)amino]-N'-hydroxypyridine-2-carboximidamide 1-(2,6-diethyl-4-fluorophenyl)sulfonyl-3-methoxypyrrolidine (3S)-3-amino-2-[4-(4-benzylpiperidine-1-carbonyl)phenoxy]-N'-butylbutanediamide (3E)-4,5-dimethylhepta-1,3,5-triene;1-[2-(4-propan-2-ylidenecyclohexa-1,5-dien-1-yl)oxyethyl]naphthalene 4-methyl-1-[2-oxo-3,6-bis(thiophen-3-yl)benzimidazol-1-yl]pentan-3-one 5-[(3,5-dimethylimidazol-4-yl)methoxy]quinazoline 3-(azidomethyl)-4-[(3-bromophenyl)sulfonylamino]benzoic acid 1-[3-(2,6-dimethoxyphenyl)sulfanylphenyl]-N-methylbutan-1-imine;pentane 5-chloro-4-[(1-methylcyclopropyl)amino]-1H-pyrimidin-6-one 5-(6-chloropyridin-3-yl)-1,2,4-oxadiazol-3-amine 3-[4,5-bis(ethenyl)imidazol-1-yl]phenol 1-[2,3-difluoro-5-(methylsulfanylamino)phenyl]-6-ethyl-8H-cyclohepta[d]imidazol-7-one 3-[2,3-bis(1H-indol-2-yl)quinoxalin-6-yl]-4H-1,2,4-oxadiazol-5-one N-[3-(2-aminoethyl)phenyl]thiophene-2-sulfonamide (3-aminopiperidin-1-yl)-[6-[4-methoxy-2-(trifluoromethyl)phenyl]-5,7-dihydropyrazolo[5,1-b][1,3]oxazin-3-yl]methanone 1-[(3S)-4-[2-amino-6-[4-[2-methoxyethyl(methyl)carbamoyl]cyclohexen-1-yl]pyrimidin-4-yl]-2,5-dioxopyrrolidin-3-yl]-3-phenylurea [6-amino-5-(4-morpholin-4-ylanilino)pyridin-3-yl]-[6-[[2,2-difluoroethylamino(hydroxy)methyl]amino]pyrimidin-4-yl]azanium 3-(5-fluoropyridin-2-yl)-4-[1-hydroxy-2-(methoxyamino)ethylidene]-N,N-dimethylcyclohexa-1,5-diene-1-carboxamide 3-bromo-2,4-ditert-butylpyridine 6-bromo-N-methyl-N-[(2R)-1-oxobutan-2-yl]-3,4-dihydroquinoline-8-sulfonamide 6-bromo-N-cyclobutyl-8-fluoro-1,2,3,4-tetrahydroquinoline-2-carboxamide N-[6-ethenyl-5-(ethylideneamino)-3H-imidazo[4,5-b]pyridin-2-yl]-1-[2-(methylamino)acetyl]pyrrolidine-2-carboxamide N-[4-(3,5-dichlorophenyl)sulfonylphenyl]propanamide 3-[4-(2,6-dimethoxyphenyl)phenoxy]propanoic acid 2-[2,3-bis(ethenyl)naphthalen-1-yl]ethanamine;ethene 3-chloro-N'-hydroxy-2-(2-methoxyphenyl)sulfanylpyridine-4-carboximidamide 5-(3,4-dichlorophenyl)sulfanyl-1-[4-methoxy-2-[(E)-prop-1-enoxy]pyridin-3-yl]pentan-3-one 1-(3,4-dichlorophenyl)sulfinyl-N-[2-(6-methylpyridin-2-yl)ethyl]piperidine-3-carboxamide 4-[3-[4-(1-adamantyl)phenyl]propoxymethyl]phenol 2-[2,5-dichloro-N-(3,4-dimethylphenyl)sulfonylanilino]propanoic acid 2-amino-6,7-dihydropyrimido[4,5-b]acridine-9-carboxylic acid 2-[5-azidooxy-6-(4,4-difluoropiperidin-1-yl)pyrimidin-4-yl]sulfanylpropanenitrile 2-[N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)anilino]ethanol 2-[(3aR,6aS)-2-(6-chloronaphthalene-2-carbonyl)-1,3,4,5,6,6a-hexahydrocyclopenta[c]pyrrol-3a-yl]-N-benzylacetamide N-[(2S)-1-[[4-cyano-3-(trifluoromethyl)phenyl]amino]-5,7-dioxoheptan-2-yl]-6-[(1R)-2-oxocyclopentyl]oxynaphthalene-2-carboxamide (1R,3S)-3-(azidomethyl)-5-[4-chloro-2-(trifluoromethyl)phenoxy]cyclohexan-1-amine 3-azido-1-propan-2-ylbenzimidazole-2-thione 4-[2,5-dimethyl-4-[5-oxo-3-(trifluoromethyl)-1H-pyrazole-4-carbonyl]piperazin-1-yl]sulfonyl-1-methylpyrrole-2-carbonitrile 2-hydroxy-N-(4-methylphenyl)-3-[[4-(trifluoromethoxy)phenyl]sulfonylamino]benzamide 1-(2-azidoethyl)-3,5-difluoro-4-propoxybenzene 1-[2,6-dimethyl-4-(5-methylpyrimidin-2-yl)piperazin-1-yl]ethanone [5-(2,6-dichlorophenyl)-4H-pyrazol-3-yl]-[[4-[1-(trifluoromethyl)cyclopropyl]phenyl]methylideneamino]azanium 3-hydroxy-N'-(2-imidazol-1-ylethyl)-5,6,7,8-tetrahydronaphthalene-2-carbohydrazide N-[(3,5-dichlorophenyl)methyl]-2,4-difluoro-N-methylaniline 3-fluoro-5-[2-(5-pyridin-4-yl-1H-pyrazolo[3,4-c]pyridin-3-yl)-1H-imidazo[4,5-b]pyridin-7-yl]phenol N-[(4,5-difluorocyclohexa-1,3-dien-1-yl)methyl]-2-[(E)-(2-phenylimino-4-pyrrolidin-1-yl-1,3-thiazol-3-ylidene)amino]acetamide 3-(2-bromophenyl)imino-N-tert-butylsulfanylpropanamide N-[2,4-difluoro-3-[5-(1H-pyrazolo[4,3-b]pyridin-6-yl)-2H-pyrazolo[3,4-b]pyridine-3-carbonyl]phenyl]propane-1-sulfonamide 1-methylsulfanyl-4-(2,3,5-trichlorophenyl)benzene 6-[2-[3,5-difluoro-4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]ethynyl]-N-[3-hydroxy-4-(2-methoxyethoxy)phenyl]naphthalene-2-carboxamide 1-methylsulfonyl-7H-cyclohepta[c]pyridine 4-amino-6-[(2,3-dimethoxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one N-[5-(4,7-diazaspiro[2.5]octane-7-carbonyl)-2-methylphenyl]-3-fluorobenzamide 4-N,4-N-diethyl-1-methoxybenzene-2,4-diamine (2R)-N-[4-[3-chloro-5-cyano-4-(trifluoromethyl)pyridin-2-yl]oxyphenyl]-1-[5-oxo-5-[4-(trifluoromethyl)phenyl]pentanoyl]pyrrolidine-2-carboxamide (3,4-difluorophenyl)-[1-ethyl-6-hydroxy-2-(methoxymethyl)indol-3-yl]iminomethanolate 1-(2,4-dichlorophenyl)-3-[4-[4-(2-hydroxyethylamino)anilino]-7-methoxyquinazolin-6-yl]urea 5-(2-aminophenyl)-4-N-ethyl-6-methoxypyrimidine-2,4-diamine 6-(4,5,6a,7,8,9-hexahydropyrazolo[1,5-a]quinoxaline-5-carbonyl)-3H-quinazolin-4-one 1-[4-(4-aminophenyl)piperidin-4-yl]-N,N-bis(pyridin-3-ylmethylideneamino)-2H-pyrazin-5-amine N-[2-(3,4-dihydronaphthalen-1-yl)-5-hydroxyphenyl]benzamide 2-tert-butyl-4-[4-[5-[5-[3-(1,1,1,3,3,3-hexafluoropropan-2-ylideneamino)phenyl]pyridin-3-yl]benzimidazolo[1,2-a]benzimidazol-7-yl]oxypyrimidin-2-yl]isoindole-1,3-dione N-[6-amino-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]-3-chlorobenzamide N-[4,5-difluoro-1-(3-methoxyphenyl)sulfonyl-2-nitrosoindol-6-yl]-2-(trifluoromethyl)benzenesulfonamide 5-(4-methoxyphenyl)-6H-pyrazolo[1,5-a]pyridin-7-one 4-(benzenesulfonamido)-N,N-dimethylbenzamide [5-[(6,8-dibromo-3-pentylimidazo[1,2-a]pyridin-2-yl)methoxy]spiro[1H-indene-3,4'-piperidine]-1'-yl]carbamic acid 3-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxybenzaldehyde 4-(2-hydroxyethyl)-3,5-diphenylcyclohexan-1-one 5-[(2R)-2-[1-(4,6-dimethoxypyrimidin-2-yl)piperidin-3-yl]butyl]quinoline 6-(1-benzylpyrazol-4-yl)-3-methoxypyrazine-2-carboxamide 1-[2,4,6-trifluoro-3-(propan-2-ylamino)phenyl]piperazine-2,5-dione 4-N-[2-(2,5-dimethylphenyl)ethyl]-1-N-(2-fluorophenyl)benzene-1,4-disulfonamide 4-methylbenzonitrile;2-[(4-methylpiperazin-1-yl)methyl]quinoline 1-azidooxy-N,N',2,3-tetramethylbenzenecarboximidamide 5-azidosulfonylquinoline (5S)-5,8-dimethyl-1-[(2R)-oxiran-2-yl]-5,7,8,9-tetrahydropyrido[3,4-b]indole N-[3,5-bis(trifluoromethyl)phenyl]sulfonylcyclopropanecarboxamide;ethane (6R)-7,11b-difluoro-1-(4-methoxyphenyl)sulfanyl-2,3,5,6-tetrahydro-[1]benzofuro[2,3-a]quinolizine 1-[4-[1-(4-fluoro-2,6-dimethylphenyl)azetidin-3-yl]piperazine-1-carbonyl]pyrrolidin-2-one N-(5,6,7,8-tetrahydronaphthalen-2-yl)quinoline-4-carboxamide 2-[1-azido-5-chloro-3,6-bis(2-methylpropoxy)naphthalen-2-yl]-N,N-diethylethanamine 5-(3-chlorophenyl)-2-methyl-4,6-bis(2-phenylethynyl)pyrimidine;N-(6-fluoropyridin-3-yl)-N'-propanoylheptanediamide [(5S)-2-benzylimino-4,6-dimethoxyspiro[1H-indole-3,4'-thiane]-5-yl]-cyclopentylmethanone (E)-3-[2,4-bis(phenylmethoxy)phenyl]prop-2-enoic acid 3-(2,6-dimethoxyphenyl)-5-[2-oxo-1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carbonyl)piperidin-4-yl]-N-(1H-pyrazol-5-yl)-1H-pyrrole-2-carboxamide 4-[[3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(2-hydroxyethyl)-2H-pyrido[2,3-d]pyrimidin-7-yl]amino]-N-[4-(pyrrolidine-1-carbonyl)cyclohexylidene]benzamide 2-[2-ethenyl-6-(2-methoxyethoxy)naphthalen-1-yl]-7-fluoro-3H-pyrido[4,3-d]pyrimidin-4-one 2-azido-5,6-diethylnaphthalene N-[[4-(cyclohexa-2,5-dien-1-ylmethyl)phenyl]methyl]-N'-[(E)-1H-pyrrol-2-ylmethylideneamino]ethane-1,2-diamine 1-[(5R,7S)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]butan-1-one (5E)-2-imino-5-[[1,4-dimethyl-7-(2-oxoazepan-1-yl)-[1]benzofuro[3,2-c]pyridin-9-yl]methylidene]-1,3-thiazolidin-4-one 1-(4,5-difluorocyclohexa-2,4-dien-1-yl)-N-[(4-methoxyphenyl)methyl]sulfanyl-N'-propan-2-ylethane-1,2-diamine N-(2,5-difluorophenyl)sulfonyl-1-methyl-6-oxopyridine-3-carboxamide (5Z)-2-cyclopropylimino-5-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-1,3-thiazolidin-4-one N-[3-fluoro-4-(triazol-1-yl)phenyl]-6,7-dimethoxyquinazoline-2-carboxamide N-[(2R)-1-(1H-imidazol-5-ylmethylideneamino)-3-methylbutan-2-yl]-4-methoxynaphthalene-2-carboxamide 2-chloro-1,3-diphenylpropane-1,3-dione (3-fluorophenyl)-[2-[methyl(propanoyl)amino]-1,3-thiazol-4-yl]methanesulfinic acid 3-[3-(4,5-dichloroimidazol-1-yl)propoxy]butanal N-[2-(3,4-dihydronaphthalen-1-yl)phenyl]-2-fluoroacetamide;ethane N-[1-(3,5-difluorophenyl)ethyl]-2-[methanethioyl-[[4-[4-(trifluoromethoxy)phenoxy]phenyl]carbamothioyl]amino]acetamide N-(2-aminocyclohexa-1,3-dien-5-yn-1-yl)benzamide N-[1-(3,4-dimethylphenyl)-2-oxopiperidin-3-yl]propanamide N-(2,5-diethylphenyl)-2-[[4-methoxy-6-(propan-2-ylamino)pyrimidin-2-yl]sulfamoyl]acetamide 2-(4,5-dimethylthieno[2,3-d]pyrimidin-6-yl)propanedioic acid 3-(hydroxymethyl)-1-[2-oxo-2-[4-(2-phenylethynyl)anilino]ethyl]piperidine-2,6-dione 2-[3-(1-methylpyrrol-2-yl)azepan-1-yl]ethanol 3-[7-(8,8-difluorooctyl)-6,8-difluoronaphthalen-2-yl]-1,4-difluoroisoquinoline 2,4-ditert-butyl-6-[(5-methoxypyrazin-2-yl)iminomethyl]phenol 2,4-dibromo-1H-[1]benzofuro[3,2-d]pyrimidin-2-amine 4-amino-5-[(1E)-buta-1,3-dienyl]-2-fluorophenol;ethane 1-[2,3-bis(hydroxymethyl)-4,5-dihydro-1-benzothiophen-6-yl]-3-diazourea 4-[1-[4-(4-hydroxyphenyl)phenoxy]ethyl]phenol N-(4-ethoxyphenyl)-2-[(1,3,5-trimethylpyrazol-4-yl)sulfonylamino]acetamide 2-(1,4-dimethylcyclohexanecarbonyl)-N-[2-methyl-5-nitro-3-(trifluoromethoxy)phenyl]butanamide 7-amino-5-[3-(oxolan-2-ylmethoxy)phenyl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 1-N,3-N-bis(2-butyl-4-methoxyphenyl)-2,6-difluorobenzene-1,3-dicarboxamide 5-methyl-2-pyridin-3-ylpyrimidine;4-pyrrolidin-1-ylbenzonitrile 2-(2-ethoxyphenyl)benzo[g][1,3]benzothiazole 7-[2,3,4,5-tetrafluoro-6-(trifluoromethyl)phenyl]quinazoline 1-(2-methoxyphenyl)-6-oxopyridine-3-carbohydrazide 5-bromo-N-(2-methoxyethyl)thiophene-3-sulfonamide 1-[3-methylsulfonyl-4,5-di(propan-2-yl)phenyl]ethanone 1-[(3R)-1-(4,5-dimethylbenzoyl)piperidin-3-yl]triazole-4-carboxamide N-[(3-chlorophenyl)methyl]-2-[2-(cyclohexa-1,5-dien-1-ylamino)-6-oxo-1H-pyrimidin-4-yl]acetamide 3-azidooxy-1-N,2-N-diethylbenzene-1,2-diamine 2-methyl-6,7,8,9,10,11-hexahydrobenzo[c][1]benzoxepine N-[4-amino-3-(1,2,4-triazol-1-yl)phenyl]-2,6-dichloro-5-methylpyridine-3-carboxamide 2-methyl-N-[1-[(3S)-pyrrolidin-3-yl]ethenoxy]aniline 6-methoxy-1',3'-dimethylspiro[1H-indole-2,4'-thiane] 2-[4-(4-chlorobenzoyl)phenoxy]acetamide 2-[(4R,5S)-2-(2,3-dihydroindole-1-carbonyl)-5-(4-fluorophenyl)-4-methyl-4H-imidazol-5-yl]benzenesulfonamide N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]hydroxylamine;hydrochloride 5-bromo-4-methyl-1H-indole;hydrochloride 4-chloro-3,6-dimethylbenzene-1,2-disulfonic acid N'-azido-2,2-dichloroacetohydrazide 4-[(3R)-3-ethyl-4-hydroxypyrrolidin-1-yl]-N,2,5-trimethylpyridine-3-carboxamide 4-[(2,4-dimethoxyphenyl)sulfonylamino]-N'-hydroxybenzenecarboximidamide 2-(3,4-dimethoxyphenyl)sulfanylbenzoic acid 5-[2-acetamidoethyl(ethenylsulfonyl)amino]naphthalene-2-sulfonic acid N-[5-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)carbazol-9-yl]pyridin-3-yl]methanesulfonamide 2-methyl-2,3-bis[2-methyl-6-(trifluoromethyl)phenyl]butan-1-amine 4-[1,3-dioxo-2-[5-(trifluoromethyl)furan-2-yl]isoindol-5-yl]-N-[[2-hydroxy-3-(2H-tetrazol-5-yl)phenyl]methylideneamino]piperazine-1-carboxamide 2-fluoro-4-[4-(1-methoxyethenyl)phenyl]phenol 1-[4-chlorobutyl(2,3-dihydroxypropyl)amino]-5a,6-dihydropyrido[2,3-b]quinoxaline-8,9-dione [2-(cyclopropylmethyl)phenyl]-(9,10-dihydrothieno[3,4-b][1,5]benzodiazepin-5-yl)methanone N-(3-methylbut-1-en-2-yl)-5-[3-(4-pyridin-3-yl-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-amine (1R,2S)-N-[(4-fluorophenyl)methyl]-5-(oxolan-3-ylsulfonyl)cyclohexane-1-carboxamide 1-[3-[(2S,4R)-1-benzyl-2-methylpiperidine-4-carbonyl]piperidin-1-yl]ethanone 1-[4-chlorobutyl(pyridin-2-yl)amino]propan-2-one (3S)-2-[(E,1R)-4-phenylsulfanylbut-2-enoxy]oxane 2-azido-3,4-dihydro-1H-pyrido[4,3-b]indole (2R)-2-[4-chloro-3-[[4-[(E)-3,4-dihydroxybut-1-enyl]-7-methylquinolin-8-yl]oxymethyl]phenoxy]propanoic acid N-[5-(2,3-dichlorophenyl)sulfonylpyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-4-carboxamide 6-[4-(2,3-dimethyl-1H-pyridazine-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile N-(2,6-dichloro-3,5-dimethoxyphenyl)thieno[3,4-d]pyrimidine-7-carboxamide 5-[(3,4-dihydroxyphenyl)methylidene]-3-(2-ethylpentanoylamino)thiophene-2-carboxylic acid (5Z)-2-[4-chloro-3-[[(4S,6R)-7-cyano-1,8-diazatricyclo[8.4.0.02,6]tetradeca-9,11,13-triene-14-carbonyl]amino]phenyl]imino-4-oxo-1,3-thiazolidine-5-carboxylic acid (5-bromofuran-2-yl)-[(7S)-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-yl]methanone 4-N-cyclopropyl-2-N,4-N-dimethoxyquinazoline-2,4-diamine 4-[2-(4-fluorophenyl)azetidin-1-yl]-6-methylpyrimidine 3-methylsulfonyl-5,8-dioxatricyclo[7.4.0.02,6]trideca-1(9),2(6),3,10,12-pentaene N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-N-(4-hydroxybutyl)-3-methylbenzamide N-[2-chloro-5-(3,5-dimethylpyrazol-1-yl)pyridin-4-yl]-1H-indole-7-carboxamide 2-(4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl)benzoic acid 1-azidooxy-2,3-dichloro-4-methylsulfonylbenzene ethane;N-[5-methyl-3-[(4-pyridin-2-ylpiperazin-1-yl)methyl]thiophen-2-yl]pentanamide [2-(4,6-dimethylcyclohexa-1,3-dien-1-yl)-5-methoxyphenyl]methanamine 6-[(2S,4R)-2-methyloxan-4-yl]oxypyridine-3-carbonitrile 6-[6-(2,6-difluorophenyl)-7H-purin-8-yl]-5-methylpyridine-3-carboxylic acid 2-methoxy-5-[2-(4-methylsulfanylphenyl)ethynyl]pyridine ethane;1-ethyl-3,4-difluoro-2-[(E)-6-(propoxymethoxy)hept-1-enyl]benzene 1-[(4aR,7aS)-2-hydroxy-6-[3-[methyl-[2-oxo-2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-ylamino)ethyl]amino]propoxy]-5-propanoyl-3,4,4a,7,7a-hexahydropyrrolo[3,4-b]pyridin-1-yl]-3-phenylpropan-1-one N-[(Z)-2,6-dimethylhept-3-enoxy]-1-[4-[[4-[[(E)-2-pyridin-4-ylethenyl]sulfonylamino]phenyl]methyl]phenyl]methanesulfonamide 1-[3-(dimethylamino)propyl]-5-phenylcyclohexane-1,3-dicarboxamide [1-[4-(N'-diazenylcarbamimidoyl)anilino]-2,3,3-trimethylbutan-2-yl]carbamic acid 2-bromo-N-tert-butyl-4,5-dimethoxybenzenesulfonamide [1-[5-fluoro-2,4-dimethyl-3-(2-pyridin-3-ylethoxy)phenyl]azetidin-3-yl]carbamic acid N-(2-aminophenyl)-3,4,5,6,7,8,9,10,11,12b-decahydro-1H-pyrrolo[1,2-a]azocine-13-carboxamide 2-[3,5-dichloro-N-(2-phenylethyl)anilino]decanoic acid 4-[3-(1-aminoethylidene)-4-methyliminopyrrolidin-1-yl]-6-chloro-N-(6-fluoropyridin-2-yl)-8-[[(3S,5R)-5-fluoropiperidin-3-yl]amino]cinnoline-3-carboxamide (3S)-1-[[2,4-dimethyl-6-(5-oxopentan-2-ylcarbamoylamino)pyridin-3-yl]methylsulfonyl]piperidine-3-carboxamide 6-azidooxyhexyl-(3,4-dimethoxyphenyl)-hydroxyphosphanium N-(4,5-dihydro-1H-imidazol-2-yl)-9-ethylcarbazol-3-amine 6,7-bis(4-methoxyphenyl)pyrazolo[5,1-b]quinazoline 3-amino-N-[(2R)-1,4-dioxan-2-yl]-5-(trifluoromethoxy)benzamide (3R,4S)-1-[2,6-dimethyl-5-[(3E,5Z)-hepta-1,3,5-trien-3-yl]pyrimidin-4-yl]-4-fluoropyrrolidine-3-carboxamide 4-[2,6-dichloro-4-(trifluoromethyl)phenoxy]-N'-hydroxybenzenecarboximidamide N-[6-(4,5,6,7-tetrahydro-1H-indazole-5-carbonyl)spiro[3.3]heptan-2-yl]cyclopropanecarboxamide 2-(1H-imidazol-5-yl)-N'-[4-(4-phenylmethoxypiperidin-1-yl)phenyl]propanehydrazide (2E,4Z)-6-amino-3-[3-(4-azidophenyl)propyl]hepta-2,4-dienoic acid [(3S)-1-azabicyclo[2.2.2]octan-3-yl]-[4-(4-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]methanone;hydrochloride 3-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]benzonitrile 2-[4-(3,3-dimethylbutanoyl)piperazin-1-yl]-6-pent-4-yn-2-yloxypyridine-3-carboxamide 3-[4-(2,3-dihydro-1H-indol-6-yl)piperazine-1-carbonyl]benzoic acid 4-[(2R)-4-carboxybutan-2-yl]-7-fluoro-5-hydroxynaphthalene-1-carboxylic acid 5-ethyl-N,2-dimethyl-4-oxo-N-(2-pyridin-3-ylpropan-2-yl)-1H-quinoline-3-carboxamide [2-oxo-2-(3,4,5-trimethoxyphenyl)ethyl]phosphonic acid 2-(8-chloro-3,4-dihydro-1H-pyrazino[1,2-a]indol-2-yl)-5-ethoxy-N-hydroxypyrimidine-4-carboxamide 2-[6-methylsulfanyl-4-(3,5,7,11,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,8,10-hexaen-13-ylamino)pyridin-3-yl]acetamide (E)-4,6-dimethyl-N-[2-(trifluoromethyl)phenyl]heptanamide (1R,2S)-4-azido-N-[3-chloro-5-(2-methoxyphenoxy)pyridin-2-yl]-2-fluorocyclohexane-1-carboxamide 4-[2-(2,3-dihydrothieno[2,3-c]pyridin-7-yl)ethyl]-N-hydroxyoxane-4-carboxamide 5-[6-(3-methyl-5-piperidin-4-yltriazolo[4,5-c]pyridin-2-yl)-1H-benzimidazol-2-yl]-N-propan-2-ylpyridin-3-amine 4-amino-6-[(2-bromophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-[1,1-bis(3-hydroxyphenyl)ethyl]phenol 3-[[4,5-dimethyl-1-(4-nitrophenyl)imidazol-2-yl]sulfanylmethyl]-5-fluoropyridine 6-(4-butylcyclohexyl)-2,3-difluoronaphthalene 6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carbonylamino)hexanoic acid 1-azido-5-fluoro-3,4-dimethylnaphthalene 2-(4,5-dihydropyrimidin-6-ylmethyl)-1-oxoisoquinoline-3-carboxamide 1-[7-[3-[4-(dimethylamino)quinazolin-2-yl]propyl]-5,6-dihydrocyclopenta[c]pyridin-4-yl]ethanone 4-[3-(1H-indol-2-yl)imidazo[1,5-a]pyridin-8-yl]cyclohexa-1,3-diene-1-carboxamide 4-amino-2-[3,5-dimethyl-1-(3-nitrophenyl)pyrazol-4-yl]sulfanyl-1H-pyrimidin-6-one N-(1,3-benzoxazol-2-yl)-2-[6-(4-chlorophenyl)-2-[(E)-3-hydroxyprop-1-enyl]pyrimidin-4-yl]acetamide 6-methoxy-4-[3-(1-propan-2-ylpiperidine-4-carbonyl)anilino]pyridazine-3-carboxamide 4-amino-2-(4-methoxyphenyl)-5,6,7,8-tetrahydroquinazoline-3-carbonitrile N-[2-(1H-indol-3-yl)ethyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 4-amino-2-[3,5-bis(trifluoromethyl)phenyl]butanoic acid 4-[3-(2,6-dioxopiperidin-3-yl)-1-propan-2-yl-2H-benzimidazol-5-yl]-N'-methylmorpholine-2-carboximidamide 2-amino-8-hydroxy-3-methoxy-5,6-dihydrobenzo[b][1]benzoxepine-4,11-dione 4-cyclopropyl-5-iodo-2-(1,3-thiazol-4-yl)-1H-pyrimidin-6-one 3-[5-(2,6-dichlorophenyl)pyridin-1-ium-2-yl]propanenitrile 2-(4-methylphenyl)sulfanyl-4-[(E)-3-phenylprop-1-enyl]phenol (2R,3S)-3-hydroxy-N-[2-[2-oxo-5-phenyl-1-propyl-4-(pyridin-4-ylmethyl)pyrazin-3-yl]ethyl]oxolane-2-carboxamide N-cyclopropyl-2,4-difluoro-5-[5-(1H-indazol-6-ylamino)-1,3,4-oxadiazol-2-yl]benzenesulfonamide 2-(2-hydroxypropylamino)acetic acid;1-[3-[4-(methoxymethyl)phenyl]sulfanylpyrrolidin-1-yl]ethanone N-(6,7-dihydrobenzo[d][1]benzoxepin-11-yl)-2-oxopiperidine-3-carboxamide N-methyl-1-[3-(trifluoromethoxy)phenyl]ethanamine 4-[5,7-difluoro-2-(3-methoxyphenyl)-1H-indol-3-yl]benzoic acid 2,4-dibromo-1-methylimidazo[1,5-a]quinazolin-9-one 1-[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]ethanone 1-[(3-azidophenoxy)methyl]-2,4-dichlorobenzene N-[6-(1H-indol-2-yl)pyridin-3-yl]benzenesulfonamide 4-[3-(methylamino)pyridin-2-yl]sulfanylbenzaldehyde 5-[(4-hydroxyphenyl)diazenyl]benzene-1,3-diol 1-azido-4-chloro-2,3,5,6-tetrafluorobenzene 1-(4-methyliodanuidyloxyphenyl)-2,3,4,9-tetrahydropyrimido[1,2-a]benzimidazole N-[(3R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-3-yl]-1,3-benzothiazole-5-carboxamide 3-[1,2-bis(4-chlorophenyl)ethylideneamino]aniline 2-[4-(1,3-thiazol-2-yl)pyridin-1-ium-1-yl]acetic acid [4-(3,5-difluorophenyl)sulfanylphenyl]methanol;formic acid [(2R,3S)-1-(cyclopropanecarbonyl)-6,7-dimethoxy-4-oxo-2,3-dihydro-1H-naphthalen-2-yl]azanide (2S)-1-[(3R,4R)-4-acetamido-1-benzylpyrrolidine-3-carbonyl]pyrrolidine-2-carboxamide N-[2-bromo-5-(methylcarbamoyl)phenyl]-3,4-dihydropyridazine-6-carboxamide 3-[(2Z)-2-[(6Z,8E)-1-methyl-4,5-dihydroazonin-8-ylidene]propyl]pyrazin-2-amine 1-[6-bromo-2-fluoro-3-(methoxymethyl)phenyl]ethanamine N-(3,4-dimethylphenyl)-2-methoxy-5-[(6-oxo-1,7-dihydropurin-2-yl)amino]benzamide N-[(E)-2-[5-chloro-1-methyl-3-[4-(trifluoromethoxy)phenyl]pyrazol-4-yl]prop-1-enyl]methanimine 6-(2,3-dihydropyrrole-1-carbonyl)naphthalene-2-carboxamide 6-fluoro-7-(2-methylphenyl)pyrido[3,4-b]pyrazine 5-chloro-N'-[(2R,3S)-1-[2-chloro-4-(4,5-difluoro-2-methylphenyl)benzoyl]-3-hydroxypiperidin-2-yl]benzohydrazide 3,4-dichloro-N'-(2-hydroxynaphthalen-1-yl)-N-phenylbenzohydrazide (5R)-3,3-difluoro-5-[(2S)-1-hydroxypropan-2-yl]oxycarbonyl-4-oxo-7-(3-phenoxyphenyl)heptanedioic acid (Z)-3-ethoxycarbonyl-4,7-dihydroxy-8-oxonon-5-enoate;cobalt(2+);methanol 3-(N-[4-bromo-2,5-dimethyl-N-propanoylanilino)phenyl]-2,6-dichloropyridine-4-carboxylic acid 3-[2,4-dihydroxy-5-[(6-oxo-1H-pyrimidin-4-yl)methyl]phenyl]-N-ethylbenzamide 3-N,4-dimethyl-7-(1-methylpiperidin-4-yl)oxypyrido[2,3-d]pyrimidine-2,7-diamine 2-(3-azido-5-methylpyrazol-1-yl)ethanol 3-bromo-6,7-dimethoxyquinoline 1-[2-fluoro-5-(propan-2-ylcarbamoyl)phenyl]pyrazole-3-carboxamide 3-[4-(pyridin-2-ylmethoxy)phenyl]-6-(trifluoromethoxy)quinazolin-4-one 4-(3,4-difluorophenoxy)butylcarbamic acid 3-(azidomethyl)-1-(5-butoxynaphthalen-2-yl)sulfonylazetidine (2S)-1-benzylsulfonyl-5,8-difluoro-N-[1-methoxy-4-(trideuteriomethoxy)isoquinolin-7-yl]pyrrolidine-2-carboxamide 5-methyl-4,5-diphenyl-2H-tetrazole 7-(3,4-dichlorobenzoyl)-2-(1H-pyrazol-5-ylmethoxymethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-one N-[2-(6,7-dimethoxyquinazolin-4-yl)oxyethyl]-5-fluoropyridine-3-carboxamide 4-N-[2,6-difluoro-3-(2-methyl-4H-imidazol-5-yl)phenyl]pyrimidine-4,5,7-triamine 3-(4-chlorophenyl)imino-2,6,7,8-tetrahydroindolizine-1,5-dione 5-chloro-2-cyclopropyl-4,7-difluoroquinoline 5-[4-(2,2,3,6-tetramethylpiperidin-1-ium-1-ylidene)butylamino]pyrazine-2-carbonitrile 2-chloro-N,4-dimethylaniline;3-(4-methoxyphenyl)-1-propan-2-ylpyrrolidine 4-amino-2-[(4-methoxyphenyl)methylsulfanyl]-6-[5-(2,3,4,6-tetrafluorophenyl)pyridin-2-yl]pyrimidine-5-carbonitrile 6-amino-2,3-dichlorobenzenesulfonic acid 2,6-difluoro-3-[3-(trifluoromethyl)phenoxy]aniline N-[(2R)-3-methylbutan-2-yl]-7-(2H-tetrazol-5-yl)pyrazolo[1,5-a]pyrimidine-2-carboxamide 2-(4-fluorophenyl)-3,4-dihydro-1H-isoquinoline-5-sulfonic acid 5-ethyl-2-[3-(oxan-4-yl)-1,2,4-oxadiazol-5-yl]phenol 1-(7-hydroxyquinolin-8-yl)propan-1-one 5-(3,4-dimethoxyphenyl)sulfanyl-2,4-bis(4-fluorophenyl)-1H-pyrimidin-6-one N-[(2,3-difluorophenyl)methyl]-2,4-bis(hydroxymethyl)pentanamide [4-(6-fluoroquinolin-2-yl)morpholin-3-yl]-piperazin-1-ylmethanone [4-hydroxy-3,5-bis(3-methylbut-2-enoxy)phenyl]-(1-hydroxycyclopentyl)methanone 3-[(2R,4S)-4-hydroxy-1-(6-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5-phenyl-1H-pyrazole-4-carbonitrile 2-(3-chloro-5-methylphenyl)-7-[4-(2,6-difluorophenyl)butanoyl]-N-ethyl-3-oxo-1,4-dihydropyrido[1,2-a]pyrazine-8-carboxamide 4-[2-(3,5-dimethylphenyl)-6H-1,3,4-oxadiazin-5-yl]-N,N-dimethylaniline (5Z)-1-[(Z)-1,2-diaminoethenyl]-7-ethoxy-8-methyl-3,4-dihydroquinolin-2-one 1-(4-chlorophenyl)-6,7-dimethylindazole N-[3-(dimethylamino)phenyl]-2-[(5R)-2-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-6-(furan-2-yl)-4-oxothieno[2,3-d]pyrimidin-5-yl]acetamide 2-(1,3-dihydroisoindol-2-yl)-N'-hydroxypyrimidine-4-carboximidamide (2Z,5E)-5-[(3-methylphenyl)methylidene]-4-oxohexa-2,5-dienal 1-methyl-2,3,4,9b-tetrahydrodibenzofuran 1-[2-(4-hydroxyphenyl)ethyl]-3-methoxy-2,3,5,6,7,8-hexahydro-[1,4]diazepino[1,7-a]indole-9-carboxylic acid 2-[1-(4-oxobutyl)-3,6-dihydro-2H-pyridine-5-carbonyl]benzoic acid 1-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl)-2-[3-(2-methoxyethylamino)phenoxy]ethanone N-[4-(3-aminophenoxy)pyridin-2-yl]-2-pyridin-3-ylacetamide 2-azido-5-[2-[4-(2-chlorophenyl)piperazin-1-yl]ethoxy]imidazo[1,2-a]pyridine [(4aS,7R)-1-methyl-7-phenyl-5,6,8,9,10,11b-hexahydro-4bH-naphtho[2,3-d]imidazol-7a-yl]hydrazine 2-[6-chloro-3-(4,4-dimethylcyclohexyl)imidazo[1,5-a]pyridin-8-yl]acetonitrile 1-(2-hydroxybenzoyl)-3-(2,4,6-trimethylphenyl)urea 7-(3-chlorophenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidine 3-[4-(3,5-difluoropyridin-2-yl)piperazine-1-carbonyl]benzonitrile N-(4,4-difluorocyclohexyl)-5-[2-methoxyethyl(propyl)sulfamoyl]thiophene-3-carboxamide (2R)-2-(benzylsulfanylamino)-3-hydroxybutanoic acid 2-amino-5-[6-(hydroxymethyl)pyridin-3-yl]-N'-[3-[[4-(trifluoromethoxy)phenyl]carbamoylamino]cyclopenta-1,3-dien-1-yl]benzenecarboximidamide N-[(4-azidocyclohexyl)methyl]-1,3,5-triazin-2-amine N-[4-(aminomethyl)phenyl]-5,6-dichloro-3-hydroxy-1H-isoindole-2-carboxamide 4-[(E)-6-ethenyl-7-methoxyhept-2-en-3-yl]phenol N'-[(3,4,5-trimethoxyphenyl)methyl]butanediamide (1R)-N'-hydroxy-3-[4-methyl-2-[[5-(trifluoromethoxy)pyridin-2-yl]amino]pentanoyl]-1,2-dihydroisoquinoline-7-carboximidamide 6,8-dimethyl-5-(3-propanoyloxybutanoyl)naphthalene-2-carboxylic acid 4-methyl-2-phenyl-1,3,5-triazine 2-[azido(methyl)amino]-3,5,6-trifluorobenzonitrile 2-azidooxy-5-(2,4-dichlorophenyl)pyrimidine 2-[5-amino-1-(4,5-difluorocyclohexa-1,3-dien-1-yl)pyrazole-4-carbonyl]-1H-indol-6-one (Z)-4,6-dihydroxy-3,5-bis[(1E)-3-(4-methylphenyl)buta-1,3-dienyl]hept-2-enedioic acid N-[5-[4-fluoro-3-(7-piperidin-1-yl-3H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]propanamide 1-[4-(2,3-dihydroindole-1-carbonyl)phenyl]propan-2-one N-[3-cyano-5-(2,5-dimethoxyphenyl)pyrazolo[1,5-a]pyrimidin-7-yl]butanamide N-azido-2,5-diethyl-7-methoxypyrazolo[1,5-a]pyrimidine-3-carboxamide 2-amino-3-(1H-indol-3-yl)-N-[4-oxo-5-(2,2,2-trifluoroethoxy)-7H-pyrrolo[2,3-d]pyrimidin-3-yl]propanamide 3-[2-(1H-indol-5-yl)ethenyl]-1,4,6,7,8,9-hexahydro-1,10-phenanthroline 2-[(1S,3R)-4-amino-3-methoxycyclohexyl]-N-butanoylbenzamide 4-[3-(1,2-dimethylindol-5-yl)oxyprop-1-ynyl]aniline 4-(diaminomethylideneamino)benzenesulfonamide (Z)-3-[2-amino-5-(methylamino)phenyl]-N'-[6-(4,4-difluoropiperidine-1-carboximidoyl)pyridin-2-yl]prop-2-enimidamide 1-[4-(azidomethoxy)phenyl]piperazine N-[4,4-bis(hydroxymethyl)cyclohexyl]thiophene-2-carboxamide;methanamine 1-methyl-3,3-diphenylazetidine N-[1-(2,4-difluorophenyl)cyclopropyl]-2-[3-(cyclobutanecarbonyl)phenoxy]acetamide 1-cyclohexyl-4-[4-(3,5-difluorophenyl)-2,6-bis(methoxymethoxy)benzoyl]piperidine-4-carbonitrile 4-(2-acetamidoimidazo[1,2-b]pyridazin-6-yl)-N-[4-cyano-3-(trifluoromethyl)phenyl]-5-fluoro-2-(1,1,1,2,3,3-hexadeuteriopropan-2-yloxy)benzamide [2-amino-5-(3-morpholin-4-ylazetidine-1-carbonyl)phenyl]-[6-fluoro-7-[(1S,2R)-2-methoxycyclopentyl]oxynaphthalen-2-yl]methanone [(1R,2S)-3-phenylmethoxycyclopentanecarbonyl]azanide (2-hydroxyphenyl)methoxyimino-oxidoazanium N-(5,6-dimethylcyclohexa-1,3-dien-1-yl)-4-methylbenzenesulfonamide 6-(4-methoxyphenyl)-4-pyridin-3-ylthieno[2,3-d]pyrimidine 4-[2-[(3S)-6,8-dichloro-1-methyl-3,4-dihydro-2H-quinolin-5-yl]phenoxy]-N,N-dimethylbutan-1-amine 3-[[5-(2,6-dimethoxyphenyl)-1H-pyrazole-4-carbonyl]amino]azetidine-1-carboxylate 4-azido-5-butyl-2,3-dimethoxyphenol 2-cyclopropyl-N-[3-(2,2-dimethylmorpholin-4-yl)phenyl]-5-oxo-1H-pyrazole-4-carboxamide 5-(4-bromophenyl)-2,3-dihydrothieno[3,4-b][1,4]dioxine 5-phenyl-1,2,3,4,7,8,8a-hexahydropyrido[1,2-a]pyrazin-6-one 5-methyl-1-[2-(5-methylpyridin-3-yl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyrrolidin-2-one 4-[(2Z,3E)-2-ethylidenehexa-3,5-dienyl]-7-fluoro-1H-benzimidazole 4-azidooxy-1,2-dimethyl-3,5-bis(phenylmethoxy)benzene 6-methoxy-N-(4,5,6,7-tetrahydro-1H-indazol-3-yl)spiro[2.5]octane-2-carboxamide 4-[2-(4,6-dimethylpyrimidin-5-yl)oxyethyl-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butyl]amino]-2-(quinazolin-4-ylamino)butanoic acid (3S)-2-[[4-ethyl-6-[1-methyl-5-[[(2R)-oxetan-2-yl]methoxy]triazol-4-yl]pyridine-2-carbonyl]amino]butanoic acid 1-azido-4-(3,5-dimethylphenoxy)benzene N-cyclohexyl-2-(3,4,5-trimethoxyphenyl)benzamide [3-(2,4-dioxopyrrolidine-1-carbonyl)phenyl]-methylidene-(oxan-4-yl)azanium 6-(cyclopentylamino)-1,3-dimethylpyrimidine-2,4-dione [2-(4-methylphenyl)-3H-benzimidazol-5-yl]methanamine 4-[1-(2,5-dihydroxyphenyl)ethylideneamino]benzoic acid 2,6-dimethyl-4-(3-pyridin-3-yl-1H-indazol-5-yl)phenol (2S)-N-[1-(1H-imidazol-5-ylmethyl)-7-(trifluoromethyl)indol-3-yl]oxolane-2-carboxamide 2-bromo-6-butyl-4,7-dihydroxyfluoren-1-one N-[1,2-dimethyl-3-(trifluoromethoxy)-5H-pyrazolo[4,3-c]quinolin-8-yl]-3-morpholin-4-ylpropanamide 4-bromobutyl(1,2-diphenylpropan-2-yl)carbamic acid 4-[5,6-dimethyl-2-(5-phenylpentoxy)pyridine-3-carbonyl]piperazine-1-carboxylic acid 4-[(E)-2,5-dimethylidenehex-3-enyl]sulfanyl-1H-pyridin-2-one 6-N-(4-propylphenyl)naphthalene-1,6-dicarboxamide 4-[2-(4-chlorophenyl)sulfanylethyl]-3,5,8,10,12-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,6,11-pentaene 2-[4-(5-fluoro-6-methylpyridin-3-yl)phenyl]acetaldehyde 2-[N-(carboxymethyl)-4,5-dimethoxy-2-nitroanilino]propanoic acid (3-chloropyrazin-2-yl)methanesulfonate 2-(1,3-benzodioxol-5-yl)-N-[4-cyano-2-methoxy-6-(morpholine-4-carbonyl)phenyl]acetamide 4-(5-chlorothiophen-2-yl)-1H-pyrrole-3-carbonitrile 5-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-2-carbonylamino)thiophene-2-carboxylic acid N-azido-5,6,7,8-tetrahydroquinoline-2-carboxamide 2-[3-(1,4-dioxan-2-yl)phenyl]-N-[6-methoxy-5-[2-[(4-methylpiperazin-1-yl)amino]pyrimidin-4-yl]pyridin-2-yl]acetamide N-(3-ethynylphenyl)-2,4-dioxo-6-[4-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]-1H-pyrimidine-5-carboxamide 5-chloro-2-[1'-(cyclopropanecarbonyl)spiro[3,4-dihydrochromene-2,4'-piperidine]-4-yl]benzonitrile 4-methyl-1,3-diphenylpentane-2,4-dione 4-amino-5-chloro-6-(2,3-difluorophenyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile 1-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-N-[[4-(trifluoromethoxy)phenyl]methyl]cyclopentane-1-carboxamide 1-[4-(methoxyamino)butyl]-6-[3-(trifluoromethyl)phenyl]imidazo[4,5-c]pyridin-2-amine N-[6-(4-chlorophenoxy)pyridin-3-yl]-N'-(2,2-dimethoxyethyl)ethane-1,2-diamine 5-[2,6-difluoro-4-(4-methylcyclohexyl)phenyl]-1,3-difluoro-2-propylbenzene 4-N,5-N-dimethyl-2-N-(3,4,7,8-tetrahydro-1H-isoquinolin-2-id-6-yl)pyrimidine-2,4,5-triamine;tungsten 1-[(2S)-6,8,9-trimethoxy-4a,9b-dihydro-3H-chromeno[3,4-b]pyrrole-2-carbonyl]pyrazole-3-carboxylic acid 3-methyl-N-[2-(2,4,5-trifluorophenyl)cyclohexa-1,3-dien-1-yl]sulfonyloxetan-3-amine N-azido-3-chloro-1-(2,4-dimethoxyphenyl)prop-2-en-1-imine 2-[6-(4-azidooxybutyl)-7,8-dimethoxynaphthalen-2-yl]oxyethanol 2-(3,5-difluoropyridin-2-yl)benzene-1,4-dicarboxamide 2-[4-fluoro-3-(trifluoromethyl)phenyl]butanoate 1-(2,5-dimethoxyphenyl)-N'-ethyl-3-hydroxybutane-1,4-diimine 5-(2,3-dihydro-1,4-benzodioxin-6-ylmethylidene)-1H-pyrimidine-2,4-dione (3-chloropyridin-4-yl)-[4-(1,2,6-thiadiazinan-2-ylamino)piperidin-1-yl]methanone [7-fluoro-6-(triazol-2-yl)-1,4,5,7-tetrahydropyrazolo[3,4-c]pyridin-3-yl]-pyrrolidin-1-ylmethanone 2-azido-3-[5-(2,5-dimethylpyrrol-1-yl)pentanoyl]imidazolidin-4-one 5-chloro-4-[(E)-1-cyanobut-2-enyl]sulfanyl-3-nitrobenzenesulfinic acid N-(2,6-dimethoxypyrimidin-4-yl)-4-[(3-fluorophenyl)methyl-(3-nitropropanoyl)amino]benzenesulfonamide 2-[4-(2,3-difluorophenyl)-1,3-thiazol-2-yl]piperidine-1-carboxamide (3S,4S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-(3,4-dichlorophenyl)-1-oxo-6-azaspiro[2.5]octane-8-carboxamide (3R,4R)-4-[1-[4-cyano-3-(trifluoromethyl)phenyl]piperidin-4-yl]-1-[(2S)-2-hydroxypropanoyl]pyrrolidine-3-carboxamide N-methyl-4-[5-(2-pyridin-3-ylethynyl)pyridin-1-ium-2-yl]pyrimidin-2-amine 1-[2,3-bis(ethenyl)-6-methylidenecyclohexa-2,4-dien-1-ylidene]ethanol;ethane 2-[(3-chlorophenyl)methylsulfanyl]-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-4-one 5-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(2-methoxyphenyl)cyclopropyl]pyrimidin-2-amine (E)-1-[2-(4,5-dihydro-1H-imidazol-2-ylamino)-7-methoxy-1,3-benzothiazol-6-yl]prop-1-en-1-one 5-[3-fluoro-5-[2,4,6-trimethyl-5-(1H-pyrazol-4-yl)pyridine-3-carbonyl]phenyl]-N-phenylpentanehydrazide (5Z)-5-[[2,6-dichloro-4-(trifluoromethylsulfanyloxy)phenyl]methylidene]-4-prop-2-ynyliminoimidazolidine-2-thione 1-[4-(aminomethyl)phenyl]-5-chloro-6-ethoxy-2H-pyridine-3,4-diamine 2-ethyl-3,3-dimethyl-6-[(4E)-5-methylidene-4-prop-2-enylidene-1H-pyrrol-2-yl]-1,8-naphthyridine 2-[4-methoxy-3,5-bis(trifluoromethyl)phenyl]benzoic acid 3-azidooxysulfonylbenzenesulfonic acid N-[2-(6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl)phenyl]propanamide;hydrochloride 5-chloro-3-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)amino]thiophen-2-ol 2-[(3Z)-3,4-dimethylpenta-1,3-dien-2-yl]-1H-imidazole;ethane;hexane 3-[(4-tert-butylphenyl)methyl]-1-ethyl-2-iminoimidazolidine-4,5-dione 4-methyl-2-[6-(piperidine-1-carbonyl)-3H-imidazo[1,5-a]pyridin-3-yl]-1,3-thiazole-5-carboxamide 2-(3,5-dichloropyridin-4-yl)sulfanyl-N'-hydrazinylacetohydrazide 1-[(1R)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]pyrrole-2,5-dione N-[3-(4,6-dimethoxypyrimidin-2-yl)propanoyl]-N'-methylcyclobutanecarbohydrazide 3-[1-[2,4-bis(trifluoromethyl)phenyl]ethylamino]-5-propan-2-ylidenecyclopentene-1,2-diolate N-[(Z)-[5-bromo-2-hydroxy-3-methyl-4-[[4-nitro-2-(trifluoromethyl)phenyl]diazenyl]phenyl]methylideneamino]benzamide 1-[2,6-di(propan-2-yl)phenyl]-3-(3,4,5-trimethoxycyclohexa-1,3-dien-1-yl)imidazolidine-2,4-dione [1-(5-bromopyridin-2-yl)azetidin-3-yl]carbamic acid 1-(4,6-dimethoxypyrimidin-2-yl)-3-[2-[(3Z,5E)-6-hydroxyhepta-1,3,5-trien-2-yl]pyridin-3-yl]urea 2-(4,5,6,7-tetrahydrobenzimidazol-1-yl)cyclopropane-1-carboxylic acid 2-[(4,5-dimethylfuran-2-carbonyl)amino]butanoic acid 6-N,6-N-dimethyl-5-nitroquinoline-2,3,6-triamine 2-[4-chloro-5-(2,3-dihydroindole-1-carbonyl)thiophen-2-yl]-N-methoxy-1,3-thiazole-5-carboxamide N-[(4R)-1-[2-methoxy-4-[(E,3S)-3-methyloct-5-enyl]phenyl]-6-oxopiperidin-4-yl]acetamide 4-[3,5-bis(4-aminophenyl)thiophene-2-carbonyl]-1,4-diazepan-6-one (2R)-1,3-dimethyl-N-[6-(4-propanoyl-2H-pyrrol-5-yl)pyridin-2-yl]pyrrolidine-2-carboxamide 5-[(2,3-difluorophenyl)methyl]-1,4-dihydropyrimidine (3S)-N-[2,5-bis(trifluoromethyl)phenyl]piperidin-3-amine 4-amino-N'-[(2S,3R)-1-methyl-5-oxo-2-propan-2-ylpyrrolidin-3-yl]pyrimidine-5-carboximidamide 2-[(4E,5Z)-3-ethylhepta-1,5-dien-2-yl]-4,6-diphenylphenol 6-bromo-2,3,4,9-tetrahydrocarbazole 2-methyl-6-[1-(oxan-4-yl)pyrazol-4-yl]benzoic acid 2,4-ditert-butyl-6-[[5-(cyclopropylmethoxy)furan-3-yl]iminomethyl]phenol (4-fluorophenyl)-[2-[3-methoxy-3-[2-oxo-5-(trifluoromethyl)pyrrolidin-1-yl]propyl]-6,7-dihydro-5H-pyrrolizin-1-yl]methanone 3-[2,6-dimethyl-4-(4-phenylbutoxy)phenoxy]propan-1-ol (Z)-N'-[2-amino-4-(2-ethoxypyridine-3-carbonyl)phenyl]prop-1-ene-1,3-diamine 3-amino-2-(4-phenoxyphenyl)propanoic acid;hydrochloride N-[2-(dimethylamino)ethyl]-4-[3,5,6-trifluoro-4-(morpholine-4-carbonyl)indol-1-yl]benzamide 3-[4-(2,5-dioxopyrrol-1-yl)phenyl]propanehydrazide 2-[1-(4-methoxyphenyl)azetidin-3-yl]ethanol 4-(6,7-dihydro-5H-cyclopenta[c]pyridine-1-carbonyl)-N-[3-fluoro-2-(propylcarbamoylamino)phenyl]piperidine-1-carboxamide N-cyclohexyl-N,1-dimethylimidazole-4-sulfonamide 2-tert-butyl-6-[4,5-bis(ethenyl)-1H-imidazol-2-yl]phenol [5-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethylsulfanyl)triazin-4-yl]hydrazine 5-[2,6-difluoro-3-[(4-methylcyclohexa-1,5-dien-1-yl)sulfanylamino]phenyl]pyrimidine-2-carbonitrile [3-(4-fluorophenyl)pyrrolidin-1-yl]-[(5R,7S)-2-methyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazol-7-yl]methanone 2-[(3S)-1-[4,5-bis(ethenyl)-1H-pyrrole-2-carbonyl]piperidin-3-yl]acetamide N-[(4-hydroxyphenyl)methyl]-1,1-dioxospiro[2H-pyrrolo[1,2-c]quinazoline-3,3'-oxetane]-6-carboxamide 3-N-(1,3-benzothiazol-2-yl)-5-tert-butyl-2-methoxy-4-methylbenzene-1,3-diamine 1-methyl-2,4-dioxo-6-[3-(trifluoromethyl)phenyl]-1,6-naphthyridine-3-carboxamide 3-(1,3-benzothiazol-5-yl)-5-[4-(4-chlorophenyl)-5-methoxycarbonylfuran-2-yl]-6-oxo-1H-pyridine-2-carboxylic acid 3-(2,4-dihydroxyphenyl)oxirane-2,2-dicarbonitrile (2R,5R)-6-(3-chlorophenyl)-2-[4-(cyclopropylmethoxy)phenyl]-1,7-dihydroxyheptan-4-one 2-N,7-N-bis[3-(diethylamino)propyl]-6-phenylpteridine-2,4,7,8-tetramine 1-[3-fluoro-4-(trifluoromethyl)phenyl]pyrazole 2-(ethylamino)-6-(5,8,11-triazatricyclo[7.4.0.02,7]trideca-1(13),2,4,6,9,11-hexaen-12-yl)phenol 1-[4-(2,6-dichlorophenyl)-5-methoxy-7H-pyrrolo[3,4-b]pyridin-6-yl]ethanone 2-[(E)-2-aminoethenyl]-6-N,7-N,3-trimethylimidazo[1,2-a]pyridine-6,7-diamine [(4-bromophenyl)methylamino]thiourea 6-(1,3-dimethylpyrazole-4-carbonyl)-N'-methyl-5-oxa-9-azaspiro[3.8]decane-10-carbohydrazide (6R)-7,8-bis(3-chloropropoxy)-4-ethyl-6-phenylmethoxyoxocane N'-(4,5-dimethylpyrimidin-2-yl)-6-[4-methoxy-3-(trifluoromethyl)phenyl]pyridine-2-carbohydrazide 2-[3-(4-fluorophenyl)sulfanylquinolin-6-yl]acetic acid N-[3-(ethylsulfonylamino)phenyl]benzenesulfonamide 3-(1,2-diphenylethyl)benzo[f]chromene 2-(4-aminocyclohexyl)-N,3-dimethylbenzamide 4-[[6-ethyl-2,3-bis(hydroxyimino)cyclohexen-1-yl]methylideneamino]phenol 1-(azidomethyl)-4-benzylsulfanylbenzene [(3-aminophenyl)methylamino]carbamic acid 3-azido-2-(4-fluorophenyl)-4,5-dihydroimidazole 1-[(3Z,5E)-6-cyclopropylnona-1,3,5-trien-2-yl]oxyethenamine;methanol;1-methyl-4-(1-phenylethyl)piperazine 4-[5,6-bis(4-chlorophenyl)pyridin-2-yl]piperazine-1-carboxylic acid;ethane 2-amino-6-(2,3-dihydrothiophene-5-carbonyl)-4-methylbenzenesulfonate 2-[1'-(5-chloro-4-fluorocyclohexa-2,4-dien-1-yl)spiro[4H-naphthalene-3,4'-piperidine]-1-yl]acetic acid 6-methyl-2,4-dioxo-3H-furo[3,2-d]pyrimidine-7-carboxylic acid 1-[4,5-dichloro-6-(pyridine-2-carbonyl)pyrimidin-2-yl]oxyethanone N-(5-chloropyridin-2-yl)-6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazole-3-carboxamide;ethane 3-bromo-4-[(2S)-5-ethyloxolan-2-yl]oxyaniline [3-(1,3-benzothiazol-2-yl)-4-hydroxyphenyl]carbamic acid 3-chloro-1,2-dihydroquinoxaline;4,6-dimethylbenzenesulfonic acid 3,5-ditert-butylbenzene-1,2-disulfonate 2-(3-aminocyclobutyl)-4-chloropyrrolo[1,2-a]pyrimidine-8-carboxamide 5-(2,4-difluorophenyl)-N-[1-[3-(trifluoromethyl)phenyl]cyclobutanecarboximidoyl]-1H-pyrazole-3-carboxamide 1-[4-(difluoromethoxy)phenyl]-5-oxopyrrolidine-2,3-dicarboxylic acid N-[2-(hydroxymethyl)-4,6-dihydrofuro[3,4-c]pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1H-benzazepine-7-carboxamide N-[2-(4-methylpiperidin-1-yl)ethyl]-2,5-dioxo-4H-thieno[3,2-b][1,6]naphthyridine-7-carboxamide 3-[(2S,6R)-2-tert-butyl-6-phenylmorpholine-4-carbonyl]benzamide 4-(2-hydroxyethylamino)-5-methoxy-1H-pyrimidin-6-one 1-(6-aminopyridin-3-yl)-5,5-dimethylimidazolidine-2,4-dione N-[(E)-[4-methoxy-3-[5-(trifluoromethyl)pyridin-2-yl]phenyl]methylideneamino]-N-(methylcarbamoyl)benzamide 4-[(1R)-1-azidoethyl]sulfonylbenzenecarboximidamide 2-(6,7-dichloro-4-fluoroisoquinolin-3-yl)-N-[2-(1H-indazol-5-ylamino)ethyl]acetamide 4-amino-2,6-dimethyl-8-(2,3,5-trimethylphenoxy)pyrrolo[1,2-a]pyrimidine-7-carboxylic acid 2-amino-N-[5-(3,6-dihydro-2H-pyran-4-yl)pyrimidin-2-yl]acetamide;hydrochloride [3-(2-propan-2-ylbenzimidazol-1-yl)azetidin-1-yl]-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-6-yl)methanone 2-[1-(azidomethyl)cyclopentanecarbonyl]oxybenzoic acid 1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-N-ethylpyrrolidine-2-carboxamide;formic acid 2-[(5-chloropyridin-2-yl)-[(3-fluorophenyl)methyl]amino]propanoic acid 1-[4-(azidomethoxy)phenyl]pyrrolidine 3-[4-(difluoromethoxy)phenyl]-7-ethyl-1,8-naphthyridine N-[5-[2-(4-hydroxyoxan-4-yl)acetyl]pyridin-2-yl]-3,6-dimethoxy-4-oxospiro[1H-quinoline-7,4'-piperidine]-2-carboxamide 4-(1-benzothiophen-2-yl)-3-[[[1-cyclohexyl-2-methyl-6-oxo-5-(4-pyrrolidin-1-ylanilino)pyrimidine-4-carbonyl]amino]methyl]benzoic acid 4-[(2,5-dimethyl-1H-pyrrole-3-carbonyl)amino]benzoic acid 1-ethyl-4-(2,3,5,6-tetrachlorophenyl)imidazole 2-[6-(2,4-dimethylphenyl)sulfanylpyridin-3-yl]acetonitrile 2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[3-(1H-imidazol-2-yl)oxetan-3-yl]acetamide (2S)-N'-hydroxy-4,4-dimethyl-1-[5-propan-2-yloxy-2-(trifluoromethyl)benzoyl]pyrrolidine-2-carboximidamide 2-amino-N-azido-1,3-benzothiazole-5-carboxamide 6-azido-1,3,4,9-tetrahydropyrido[3,4-b]indole 1-[(4R,5S)-5-benzyl-2,2-dimethoxy-4-methyl-3a,4,6,7-tetrahydrocyclopenta[d]pyrimidin-7a-yl]propan-1-one 1-ethyl-5,6-difluoroindole;5-hydroxy-N'-(2-oxo-3H-1,3-benzoxazol-6-yl)pyridine-2-carboximidamide 2-(cyclopropanecarbonylamino)-N-[6-(3,5-dimethylpyrazol-1-yl)pyridin-3-yl]pyridine-4-carboxamide 2-(1,3-benzothiazol-2-yl)phenol;chlorobenzene;ethane 5-(8,9,10,11-tetrahydronaphtho[1,2-h]quinazolin-6-yl)quinoline N-[(5-chlorothiophen-2-yl)methyl]-1-cyclopentylethanamine 4-(2,3-diethylphenyl)piperidine 2-ethoxycarbonylnaphthalene-1-carboxylic acid N-[1-cyclohexyl-2,4,5-trimethyl-3-(pyridine-3-carbonylamino)pyrrol-3-yl]-1H-imidazole-5-carboxamide 2-hydroxy-3,6-dimethylpyrrolo[3,4-b]pyridine-5,7-disulfonic acid (1S)-2,2-dimethylspiro[cyclopentane-3,4'-piperidine] N-(4,5-dimethyl-1H-pyrazol-3-yl)benzamide 1-(1-azidooxybutyl)-3,5-dimethoxybenzene 2-[2-ethyl-5-(4,4,5,5-tetramethyloxaborolan-2-yl)phenyl]pyrrolidine 1-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-yl)-N,N-bis[(3-fluorophenyl)methyl]piperidin-4-amine 2-[3,5-di(propan-2-yl)phenyl]pyridine 5-(4-phenylbutyl)-3a,6a-dihydrocyclohexa-1,3-diene-1-carboxylic acid 6-chloro-N-(2,5-difluorophenyl)sulfonyl-1H-indole-4-carboxamide 1-[[2,4-bis(methylsulfonyl)phenyl]methyl]-3-diazourea 4-[2-(2,5-dimethylphenoxy)ethylamino]-3-[6-fluoro-1-methyl-8-(propylamino)-7-(pyrrolidin-1-ylmethyl)-2H-isoquinolin-3-yl]butanal 2-[2-methyl-3-(3-phenylcyclohexa-1,3-dien-5-yn-1-yl)-5H-pyrido[2,3-b]indol-7-ium-9-yl]phenol 2-(4-cyclopropyl-1,3-thiazol-5-yl)-N-[5-[2-(1H-imidazol-5-yl)ethoxy]-1H-indazol-3-yl]-1H-benzimidazole-4-carboxamide 1-cyclopropyl-6,7-difluoro-3-methylidene-4H-quinoxalin-2-one (2S,4R)-N-[5-cyano-2-[(4,6-diaminopyridine-3-carbonyl)amino]phenyl]-4-methylpyrrolidine-2-carboxamide;hydrochloride 1-[(E)-[3,5-bis(trifluoromethyl)phenyl]methylideneamino]-1-(2-chloro-6-methoxypyridin-4-yl)thiourea 2-[[3,5-bis(trifluoromethyl)phenyl]sulfanylamino]-3-oxopropane-1-sulfonic acid 7-[5-[5-(diethylcarbamoyl)pyridin-2-yl]pyrazin-2-yl]-1,3,4,8,12b-hexahydroperylene-4a-carboxylic acid 4-cyclohexylsulfanylpyridine-3-carboxamide 2-chloro-N-ethyl-N-(1,3-thiazol-5-yl)acetamide 5-chloro-N'-hydroxy-1-(4-phenylbutanoyl)spiro[2H-indole-3,3'-pyrrolidine]-6-carboximidamide 2-[(3,4-dimethoxyphenyl)methyl]benzenecarboximidamide;ethane N-[2-hydroxy-3-(1H-pyrrolo[2,3-b]pyridin-5-ylmethoxy)propyl]-5-oxo-4H-pyrazolo[1,5-a]quinazoline-2-carboxamide 5-azidosulfanyl-7-ethynylisoquinoline 2-[1-(4,6-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-6-pyridin-2-ylpyridazin-3-one 4-(1,3-benzothiazol-5-yloxy)-6-methylcyclohexa-2,4-dien-1-one N-[(2S)-1,3-dihydroxypropan-2-yl]thiophene-2-carboxamide 2-(3,4-dimethoxyphenyl)-N,N,2-trimethylpropanamide;ethane;2-hydroxyethylazanium 1-[(5S)-4-amino-2,7,8-trimethyl-3-oxospiro[2H-pyrido[3,4-b]pyrazine-1,1'-cyclopropane]-6-yl]-3-ethylurea N-[5-[(Z)-1,3-diaminoprop-2-enyl]pyridin-3-yl]cyclopropanesulfonamide N-[4-[chloro(difluoro)methoxy]phenyl]-1-(3,5-dichloropyridin-2-yl)-6-oxopyrimidine-4-carboxamide N-(4,4-dimethyl-1,3-thiazolidin-2-ylidene)naphthalene-1-sulfonamide 4-chloro-2-[(3,5-dichloropyridin-4-yl)methoxy]-1-nitrocyclohexa-2,4-dien-1-ol 3-amino-4-[3,5-dimethyl-2-(propanoyloxymethyl)phenyl]butanoate N-(3,5-dimethoxyphenyl)-N-[4-ethylsulfanyl-2-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)phenyl]methanesulfonamide 3-[5-fluoro-6-(2,3,4,9-tetrahydro-1H-carbazol-3-yloxy)pyridin-3-yl]propanoic acid 1-[4-(4-azidooxybutoxy)butyl]naphthalene 2-fluoro-N-[1,4]benzodioxino[3,2-c]chromene-6-carboxamide N-[3-cyano-7-ethoxy-4-(7-methylpyrrolo[2,1-f][1,2,4]triazin-2-yl)chromen-2-ylidene]hydroxylamine 4-(dimethylamino)-3,5-bis[(2-oxo-1H-quinoline-3-carbonyl)amino]benzoic acid 2,4-ditert-butyl-6-[4-(5,8-dimethoxyimidazo[1,2-a]pyrazin-3-yl)phenyl]phenol 2-[5-(2,4-dimethylpiperazine-1-carbonyl)furan-3-yl]-N'-hydroxyethanimidamide 5-[(2E,4Z)-hexa-2,4-dien-3-yl]-1H-pyrrolo[2,3-b]pyridine 1-(4-methylphenyl)sulfonyl-N-[(Z)-thiophen-2-ylmethylideneamino]piperidine-3-carboxamide 6-(2,3-dimethoxyphenyl)-5-hydroxy-2-propan-2-yl-2H-pyran-4-carboxylic acid 2-methoxy-6-propanoyloxynaphthalene-1,4-dicarboxylic acid 4-(2-fluorophenyl)-1-[3-[5-methyl-6-[(E)-prop-1-enyl]pyridin-3-yl]sulfonylphenyl]butan-2-one 5-[3-[2-(diethylamino)phenyl]iminobutyl]-N,N-diethylpyridine-3-carboxamide N-(5,8-dimethoxy-4a,7a-dihydronaphthalen-1-yl)-N'-[6-(methylamino)-2-morpholin-4-ylpyrimidine-4-carboximidoyl]propane-1,3-diamine N-[[2,3-dichloro-4-(hydroxymethyl)phenyl]methyl]acetamide 6-(4-but-3-enylphenyl)-1,2,3-trifluoronaphthalene 4-[1-(4-butylsulfanylphenyl)sulfanylbutan-2-ylamino]-N-[3-cyano-5-(trifluoromethyl)phenyl]benzamide (7S)-N-[1-(2,3-dichlorophenyl)ethyl]-5-oxo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide (Z)-3-[2-methoxy-4-(trifluoromethyl)phenyl]prop-1-en-1-amine 4-ethenyl-N,2-dimethylbenzenecarbothioamide 1-(4-acetylphenyl)-2,2,3,3,5,6,7-heptafluoroheptane-1,4-dione (1S,2R)-2-[(5,6-diphenylpyrazin-2-yl)amino]cyclohexan-1-ol N-(2,3-dimethyl-5-oxo-4H-pyrazolo[1,5-a]pyrimidin-6-yl)-3-fluorobenzamide N-[5-tert-butyl-3-(difluoromethoxy)-2-hydroxyphenyl]butanamide [(2R)-4,7-difluoro-3,5-bis(methylsulfanyl)-1-benzofuran-2-yl]methanamine (6S)-3-[(2S,4R)-1-[2-[3-(dimethylamino)propoxy]benzoyl]-4-hydroxypyrrolidine-2-carbonyl]-8-oxo-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 7-(2,3-difluorophenyl)-9H-xanthene-1,2-disulfonic acid 2-chloro-4-[(4Z)-3,5-dimethylidenehepta-1,4-dien-2-yl]-6-(5-phenylpyrimidin-2-yl)phenol 5-azido-2,4-dimethoxy-1H-indole N-[(2R,3R)-4-methylsulfanyloxolan-3-yl]-2-pyridin-2-ylacetamide 2-[7-[[6-(2,3-dihydro-1,4-benzodioxin-5-ylmethoxy)pyridin-3-yl]methylamino]-3-oxo-1H-isoindol-2-yl]acetic acid 2-[(4R,6S)-1-methyl-3,6-diphenyl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridine-4-carbonyl]pentanoic acid 5-(4-ethylphenyl)-2-methoxy-6-N,6-N-dipropylpyrazine-3,6-diamine [4-(2,5-dimethylphenyl)piperazin-1-yl]-[4-hydroxy-3-(trifluoromethyl)phenyl]methanone 6-[[2-hydroxy-5-(trifluoromethyl)phenyl]diazenyl]-7,8-dihydronaphthalene-1,3,4,5-tetrone (2S)-N'-[(Z,1Z)-2-cyclopentyl-1-[4-[3,5-dimethoxy-6-(oxolan-3-ylmethoxy)pyridin-2-yl]pyrazol-1-yl]buta-1,3-dienyl]-2-fluorobutanediamide 4-[1-(5-fluoropyridin-2-yl)piperidin-4-yl]pyrimidine 2-[4,5-bis(4-methylphenyl)-1H-imidazol-2-yl]phenol 3-azidooxy-N,1-dimethyl-2-propan-2-ylidenebenzimidazole-5-carboxamide 1-(2,6-difluorophenyl)-7-[4-hydroxybutyl(methylsulfonyl)amino]-N-(3-morpholin-4-ylpropyl)pyrazolo[4,3-d]pyrimidine-5-carboxamide 2-(2,6-dichloroanilino)-3H-benzimidazole-5-carbohydrazide 1-(3-hydroxybutyl)-N',5-dimethylpyrazole-4-carboximidamide 3-(2,6-dichlorophenyl)sulfanylpropane-1-thiol 2-[N-(3-nitrophenyl)-4-[1,3,4-oxadiazol-2-yl-(2-oxo-propyl)amino]anilino]acetonitrile 1-[2-methoxy-5-(propan-2-ylamino)pyridin-3-yl]piperidine-4-carboxamide 4-(3,4-dimethoxyphenyl)-1H-benzimidazole 2-bromo-3,4-dihydroisoquinolin-1-one 4-[2-(cyclopropylmethoxy)-3,5-difluoropyridin-4-yl]benzamide 1-[4-(2,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-3-phenylprop-2-en-1-one 4-[(1,3,5-trimethylpyrazol-4-yl)sulfonylamino]-N-(1,4,6-trimethylpyrazolo[3,4-b]pyridin-5-yl)benzenesulfonamide (3R)-N-[2,4-dichloro-5-[1,5-dioxo-1,2,4-triazol-4-ylmethyl]phenyl]-2-imino-3-(methylideneamino)butanamide 1-(3,4-diethylphenyl)-2-pyrrolidin-1-id-4-ylbutan-1-one;yttrium 2,2,4-trifluoro-N-[(Z)-[1-[(3-propan-2-yloxyphenyl)methyl]-5H-pyrazolo[3,4-d]pyrimidin-4-ylidene]amino]-1,3-benzodioxol-5-amine ethane;1-[1',4'-dimethyl-3'-(2-phenoxyacetyl)spiro[1H-indole-2,4'-piperidine]-5-yl]butan-2-one 6-(3,5-dimethylphenyl)quinazoline (2R,3S)-4,4,4-trifluoro-N-[4-methyl-3-(trifluoromethoxy)phenyl]-3-propan-2-yl-3-(trifluoromethyl)butanamide 1-cyclopropyl-5-ethoxycarbonyl-3,6-dimethyl-2H-pyrazine-2-carboxylic acid 1-[5-amino-6-oxo-4-(2,2,3,3,3-pentafluoropropoxy)pyridazin-1-yl]pentane-2,4-dione 4-(7H-purin-6-ylmethylamino)benzenesulfonamide (2R,3S)-4-(2-phenylcyclopropyl)butane-1,2,3-triol 6-(2,2-difluoroethoxy)-3-methyl-1H-benzimidazol-2-one 2-N,6-N-bis(1H-indazol-5-yl)pyrazine-2,6-dicarboxamide 1-[3,5-bis(trifluoromethyl)phenyl]propane-2-sulfinamide 7-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-2-[(4-fluorocyclohexa-1,3-dien-1-yl)amino]pteridine-6-carbonitrile 6-(3,4-dichlorophenyl)-2-methyl-7H-[1]benzofuro[2,3-b]pyridine [(2R,4S)-4-(5-chloroindol-1-yl)pyrrolidine-2-carbonyl]azanium 2-(5,6-dihydrobenzo[b][1]benzoxepin-7-yl)acetonitrile (1Z)-4,6-dimethyl-1-propylidenebenzo[de]isoquinoline;ethane 2-(N-butanoyl-3-hydroxyanilino)-4-methylpentanoic acid N-[4-(2-diazohydrazinyl)phenyl]propane-1-sulfonamide ethane;1-ethylnaphthalene;5,9,10-trimethoxy-2,7-dimethyl-6H-benzo[a]quinolizin-4-one (6-ethylcyclohexa-1,3-dien-1-yl)-phenylphosphane 2-[4-(3-acetylphenyl)piperazin-1-yl]-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carboxylic acid 1-[4-(dimethylamino)phenyl]sulfonyl-3,4-dihydroquinolin-2-one 2-methyl-6,8,12,13,15-pentazatetracyclo[7.7.0.03,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaene 1-[(1-ethylpiperidin-4-ylidene)amino]-2,3-difluorobenzene 2-(3,5-ditert-butyl-2-hydroxyphenyl)ethanone 2-[7-(4-bromophenyl)-5-methyl-2-[3-(trifluoromethyl)pyridin-2-yl]-1,3-benzothiazol-6-yl]acetic acid 1-azido-2,3,4-triphenoxybenzimidazole (3-hydroxypiperidin-1-yl)-[2-[4-hydroxy-5-(indol-3-ylidenemethyl)-2-oxoimidazol-1-yl]phenyl]methanone N-[4,6-bis(4-chlorophenyl)-2H-1,4-oxazin-3-ylidene]hydroxylamine 3-chloro-N,2-dimethyl-1H-pyrrolo[3,4-c]pyridine-7-carboxamide 3-[1,2-bis(trifluoromethyl)indol-4-yl]oxy-5-ethanimidoyl-N'-methylpyridine-2-carboximidamide 6-[4-(3,4-dimethoxyanilino)pyrimidin-2-yl]sulfanyl-N-hydroxyhexanamide (E)-1-chloroprop-1-ene;N-[3-methylbuta-1,3-dien-2-yloxy(phenoxy)phosphoryl]propan-1-imine 1-(3,4,5-trifluorophenyl)propane-2,1-diol (2-methylpyrazol-3-yl)-(6-methylidenecyclohexa-2,4-dien-1-yl)methanone 2-amino-9,10-dioxoanthracene-1-sulfonic acid 3-[6-chloro-2-(4,7-diazaspiro[2.5]octan-7-ylmethyl)pyrimidin-4-yl]cyclopentane-1-carboxylic acid;ethane 4-ethyl-3,5,6-trifluoro-2-methoxybenzenesulfonic acid 3-[3-(2-ethylbutylamino)propyl]-5,6,7,8-tetrahydro-1H-quinoline-4-thione 4-(2-azidoethyl)-5,6,7,8-tetrahydropyrido[3,2-d]pyrimidine (5E)-2-(3-chlorophenyl)imino-5-[(2,7-dimethoxynaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one 1-(3,3-diphenylpropyl)pyrrolidin-2-one 1-[[4-(5,6,7,8-tetrahydronaphthalene-2-carbonyloxy)phenyl]methyl]piperidine-3-carboxylic acid N-[(4-acetylphenyl)methylideneamino]naphthalene-2-carboxamide;propanoic acid 3-bromo-1-(2,4-difluorophenyl)-6-methoxypyrazolo[4,3-c]pyridine N-(1,2-dimethylindol-5-yl)sulfanyl-6-[1-(3-fluorophenyl)cyclopropanecarbonyl]pyridine-3-carboxamide 6-(3,4-dimethoxyphenyl)hexane-1-thiol 4-amino-N'-(1,3-benzothiazol-2-yl)-5-nitropyridine-2-carboximidamide 7-tert-butyl-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine;(3Z,6E)-6-(3-ethoxyprop-1-ynyl)octa-3,6-diene 2-azido-5,7-dichloronaphthalene 2-[N-(2-bromophenyl)-4-methoxyanilino]decanoic acid (3S,5R)-3-phenylmethoxycarbonylbicyclo[4.2.0]octane-7-carboxylic acid [(3R,4S)-1-benzyl-4-fluoropyrrolidin-3-yl]-spiro[2H-furo[2,3-b]pyridine-5,3'-pyrrolidine]-1'-ylmethanone 1-[4-(2,2-difluoroethylsulfanyl)phenyl]ethanone 2-[[(3aR,7aS)-1-(4-fluorophenyl)-2,2-dimethyl-3,3a,4,6,7,7a-hexahydropyrrolo[3,2-c]pyridin-5-yl]methoxy]acetamide 1-[4-[2-amino-5-(4,5-dihydro-1,3-thiazol-2-yl)pyridin-3-yl]phenyl]-2-(6-chloronaphthalen-2-yl)ethanone 6-azidooxy-3-chloroquinoline 3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-7-methoxyquinoline-5-carbonitrile 7-(2,4-dichlorophenyl)-3H-quinazolin-4-one (2-bromo-5,6-diethoxy-3H-1-benzofuran-2-yl)methanol 6-chloro-5-(2,5-difluorophenyl)-1H-indazole 6,7-dimethoxy-2H-phthalazine-1,4-dione 1-chloro-3-(2,4,6-trimethylphenyl)butan-2-one 4-[6-[[(E)-1-[amino(methyl)amino]prop-1-en-2-yl]amino]pyrimidin-4-yl]oxypiperidine-1-carboxylic acid ethane;N-[2-(6-phenyl-1,3-benzodioxol-5-yl)cyclohexyl]propanamide 1-[(E)-2-nitroethenyl]spiro[2,3-dihydro-1H-naphthalene-4,5'-imidazolidine] 3-cyclopentyl-5,7-dimethoxy-1H-quinoxaline-2,6-dione 2,6-dichloro-N'-[1-(2-methoxyphenyl)ethyl]benzohydrazide (7S)-2-chloro-9-(4-fluorophenyl)-5,6,7,8-tetrahydropyrimido[4,5-d]azepin-7-ol;hydrochloride (2S,4R)-N-[(1R)-1-[5-(3-cyanoazetidine-1-carbonyl)thiophen-2-yl]ethyl]-4-fluoropyrrolidine-2-carboxamide 4-(8-amino-2,3-dihydroimidazo[1,5-a]pyrazin-1-yl)naphthalene-1-carboxamide (E)-3-[4-bromo-5-[2-[3,5-dichloro-1-(3,3-dimethylbutanoyl)indol-2-ylidene]hydrazinyl]-2-sulfophenyl]prop-2-enoic acid 2-[[2-(4-fluoroanilino)pyrimidine-5-carbonyl]amino]propanoic acid 4-[2,6-dimethyl-3-(3-nitrosophenyl)phenoxy]benzoic acid 4-(4-cyclopropylpyrimidine-5-carbonyl)-N,2,3-trimethoxybenzamide 2-(4-methoxyphenyl)-5,6-dihydro-1H-indole 2-chloro-4,5-diphenyltriazole 5-fluoro-4-[6-(5,7,8,10-tetrazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,9,11-hexaen-13-yl)spiro[3H-chromene-2,4'-piperidine]-4-yl]pyrimidin-2-amine 2-(methylideneamino)spiro[5H-thieno[3,4-d]pyrimidine-7,1'-cyclobutane]-6-amine 2-ethenyl-1-[(3Z)-2-ethenylhexa-3,5-dienoxy]benzene 1-[(2-methylpropan-2-yl)oxycarbonyl]-4-(phenylmethoxycarbonylamino)pyrrolidine-3-carboxylic acid 4-(2,4-difluorophenyl)-3-(4-methoxybenzoyl)chromen-2-one 3-(2,4-dichlorophenyl)-1-[2-[ethyl-[[2-methoxy-6-(trifluoromethyl)pyridin-3-yl]methyl]amino]ethyl]-6-[5-(2-morpholin-4-ylethoxy)pentanoyl]quinazoline-2,4-dione 3-(methoxymethyl)-4-[3-[2-[5-methyl-6-[(3R)-oxolan-3-yl]pyrazolo[1,5-a]pyrimidin-2-yl]piperidine-1-carbonyl]phenyl]benzonitrile 5-[[4-(4,6-diphenylpyridin-2-yl)-1H-diazet-2-ylidene]methyl]benzo[b][1]benzoxepine 2-[4-[[5-(2,3-difluorophenyl)spiro[3.3]heptan-2-yl]carbamoyloxymethyl]piperidin-1-yl]pyrimidine-5-carboxylic acid 2-(1H-benzimidazol-2-yl)-5-[2,6-dichloro-4-(trifluoromethoxy)phenyl]sulfonyl-4-(trifluoromethylsulfanyl)-1,3-thiazole 1-[4-(2,5-dihydroxypyrrol-1-yl)phenyl]ethanone 2-methyl-4,6-diphenylpyrimidine;1-[(2E)-3-methylpenta-2,4-dien-2-yl]sulfanylbenzene 3-(2,4-difluorophenyl)imino-7-pyridin-3-yl-1H-indol-2-one [5-amino-4-methoxy-2-[1-(3,6,6-trimethylcyclohexa-2,4-dien-1-yl)ethyl]phenyl]methanol 1-[4,5,6,7-tetramethyl-2-(4-methylphenyl)quinoline-3-carbonyl]piperidine-4-carboxylic acid 2-[1-(4-chlorophenyl)sulfonyl-3,6-dihydro-2H-pyridine-5-carbonyl]butanoic acid N-[2,4-dimethyl-5-(1-methylidenepyridin-1-ium-3-yl)phenyl]acetamide;ethane 1-[7-tert-butyl-5-(4,4-difluoropiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-3-yl]oxypyrrolidine-2-carboxylic acid 4-[4-chlorobutyl(propyl)amino]benzenesulfonamide 1-methyl-N-[(3S)-5-(2H-tetrazol-5-yl)-2,3-dihydro-1H-inden-4-yl]imidazole-4-carboxamide 2-(4-chlorophenyl)-1,3-thiazolidine N-[[(5S)-3-[4-[1-(2,6-dichlorocyclohexa-1,5-dien-3-yn-1-yl)pyrazol-4-yl]phenyl]-5-methyl-4,5-dihydro-1,2-oxazol-5-yl]methyl]ethanamine 5-(1H-imidazol-2-yl)thiophene-3-carboxamide 6-(1,3-dimethylindazole-6-carbonyl)-8-fluoro-2-[2-[4-(2H-pyrimidin-1-yl)phenyl]ethylamino]pyrido[2,3-d]pyridazin-5-one 3-[[5-chloro-2,4-bis(propoxymethyl)phenoxy]methyl]oxirane (6E,10Z)-5-benzylidene-3,4-dihydroxy-N'-[2-(1H-indol-3-yl)ethyl]octa-6,8-dienimidamide 4-fluoro-1-phenylpiperidine;N-(2,4,5-trichlorophenyl)acetamide 1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidine-4-carboxamide 2-[(3aR,6aS)-5-(cyclopropylmethoxy)-3,4,6,6a-tetrahydro-1H-furo[3,4-c]pyrrol-3a-yl]-N-(cyclohexanecarbonyl)benzamide 2-(difluoromethyl)-N-[(3S)-1-(7-fluorospiro[5H-1,4-benzothiazepine-10,1'-cyclopropane]-8-carbonyl)pyrrolidin-3-yl]pyridine-3-carboxamide 1,3-bis(chloromethoxy)-2-(difluoromethyl)benzene 1-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridin-6-ylmethyl)-5-methoxycarbonyl-4,6,7,8-tetrahydropyrazolo[4,3-c]azepine-3-carboxylic acid 5-[2-[1,4-bis(trifluoromethyl)cyclohexa-2,4-dien-1-yl]sulfanyl-3-phenylpropanoyl]oxypentanoic acid 4-chloro-N'-[(Z)-1H-pyrrol-2-ylmethylideneamino]benzenecarboximidamide N-ethyl-2,5,7-trimethyl-4H-pyrazolo[1,5-a]pyrimidine-6-carboxamide 2-amino-5-[4-(difluoromethoxy)phenyl]-1H-pyrrole-3-carbonitrile 2-[4-azido-3,6-dioxo-1-(phenylmethoxycarbonylamino)piperazin-2-yl]acetic acid 4-[5-(2,6-dimethylpyridine-3-carbonyl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]-N,N,5,6-tetramethylpyrimidine-2-carboxamide N-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-2,6-dimethoxy-N-propan-2-ylpyridine-3-carboxamide;methane 5-bromo-4-(methoxymethyl)-2-[2-(trifluoromethylsulfanyl)ethyl]-1H-pyrimidin-6-one 6-[2-(3,4-dimethoxyphenyl)-1H-indol-3-yl]hexanamide N-[(1R)-2,3-dihydro-1H-inden-1-yl]-6-oxo-2-pyrimidin-5-yl-1H-pyrimidine-4-carboxamide N-cyclopropyl-2-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzenesulfonamide 2-[2,6-dichloro-3-(6-methyldodecanoyl)anilino]acetic acid N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-(5-fluoropyridin-3-yl)-9-methylidene-4,5,6,7-tetrahydro-3H-pyrimido[1,2-d][1,4]oxazepine-8-carboxamide (3E,5Z)-4,6-dichlorohepta-1,3,5-triene;N-[1-[4-(4-fluorophenyl)-1-hydroxybutan-2-yl]piperidin-4-yl]-4-methoxybenzamide (2R,3S)-2-(1H-indol-3-ylmethylsulfanylamino)butane-1,3-diol N-[1-(5-bromopyridin-2-yl)propan-2-ylidene]-3,4-difluorobenzenecarboximidamide 3-azidooxy-1,2,4-trifluoro-5-methylsulfonylbenzene 1-[4-(2,6-dimethoxyphenyl)-5-pyridin-3-ylsulfonyl-1,2,4-triazol-3-yl]cyclopropane-1-carbonitrile (3S)-N-[5-[4-fluoro-3-(7-pyridin-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]-3-methylpentanamide 3-(2,5-dimethylphenyl)-7-fluoro-4-iminoquinazoline-6-carbonitrile N-[2-chloro-4-(trifluoromethoxy)phenyl]-6-[2-methyl-5-[(E)-4,4,4-trifluorobut-1-enyl]phenoxy]pyridine-3-carboxamide ethane;2-(4-hydroxy-3,5-dimethoxyphenyl)-7-methyl-6,8-bis(nitrosomethyl)chromen-4-one 4-(6,8-dihydrobenzo[c]chromen-1-yl)butan-2-ol N-[[(3R,6S)-2-cyclohexyl-6-(1H-pyrazol-4-ylmethyl)-4,5,6,7-tetrahydroindazol-3-yl]methyl]pyridine-2-carboxamide 4-(5,5-dimethylcyclohexa-1,3-dien-1-yl)oxyaniline 4-[(3E)-2,5-dimethylhexa-1,3,5-trien-3-yl]oxybenzamide [3-(aminomethyl)phenyl]sulfonylurea 2-(azidomethyl)-4-(1,3-dioxolan-2-yl)-5-methoxypyrimidine 2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)phenyl]-3H-pyrido[2,3-d]pyrimidin-4-one 2,7-diphenylspiro[4H-quinoxaline-3,1'-cyclohexane]-6-amine [2-(aminomethyl)-4,5-dichlorophenyl]-[3-[methoxy-(2-oxopiperidin-1-yl)methylidene]azetidin-1-yl]methanone 4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluoroaniline 5-[2-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]-1H-quinolin-4-one 3-(5-fluorothiophen-2-yl)piperidine 4-methyl-3,5-bis(phenylsulfanyl)pyridine 2-(3,4-dichlorophenyl)ethyliminomethanolate (3R)-3-[4-[[2,3-dihydro-1H-inden-2-ylcarbamoyl(pentan-2-yl)amino]methyl]phenyl]hex-5-enoic acid 1,4-dibromonaphthalene 5-[4-(1,3-benzodioxol-5-yloxy)phenyl]-2-ethyl-1,3-oxazole;ethane 1-cyclopropyl-2-[3-(1,3-oxazol-5-yl)pyrazolo[1,5-a]pyrimidin-7-yl]ethanone [3-(1H-indole-2-carbonylamino)azetidin-1-yl]carbamic acid 2-(5,6-dimethylpyridin-3-yl)-4-fluoroimidazo[1,2-a]quinoline (E)-3-[4-[2-(5,6-dichlorocyclohexa-1,5-dien-1-yl)ethynyl]phenyl]prop-2-enal (2S)-2-amino-3,4-dihydro-1H-acridine-9-carboxamide 1-azidooxy-3-cyclopropyl-5-propan-2-yloxybenzene 6-methyl-2-[(E)-[(4Z,7E)-9-methylideneundeca-1,4,7-trien-5-yl]iminomethyl]naphthalen-1-ol 1-methyl-4-[3-(2,2,6,6-tetrafluorocyclohexylidene)prop-1-enyl]benzene N-[(3S)-5,7-dimethyl-4-oxo-2,3-dihydropyrido[3,2-b][1,4]oxazepin-3-yl]-4-phenoxypyridine-2-carboxamide 5-azidooxy-2-(3,4-dichlorophenoxy)benzenethiol 3,4-dichloro-N'-[(2S)-1,1,1-trifluoropropan-2-yl]benzenecarboximidamide 3-amino-6-phenylsulfanylbenzene-1,2-diol 4-fluoro-7,9,10,11-tetrahydrobenzo[b]quinolizin-8-one N-[1,3-bis(4-nitrophenyl)propan-2-yl]acetamide 2-chloro-4,5-dicyclopropylaniline N-(1,4-dimethylpyrimidin-2-ylidene)nitramide (1-acetylcyclopropanecarbonyl)-[2-(4-methylphenyl)-3-phenyl-5,6-dihydroimidazo[1,2-a]pyridine-7-carbonyl]azanium (2S,6R)-4-[2-[1-(3-bromophenyl)ethenylamino]acetyl]-N-[(1S)-1-(4-methoxyphenyl)ethyl]-5-oxomorpholine-2-carboxamide 5-methylsulfanyl-7,8-dihydronaphthalene-2,6-disulfonic acid (5S,6R)-3-cyclopentylsulfanyl-6-(4-ethoxyphenyl)-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-1-one 1-[[(3R,4S)-4-[(6-ethoxypyridine-2-carbonyl)amino]oxolan-3-yl]methyl]triazole-4-carboxamide 1-(2,6-dimethylpyridin-4-yl)-3-[(E)-pent-2-en-2-yl]oxypyrazolo[3,4-d]pyrimidine 3-[8-[3-[(4R)-2-amino-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinoline-4-carbonyl]-2,5-dimethylpyrrol-1-yl]sulfonyloctylamino]benzamide 2-(9H-fluoren-1-yloxy)benzoic acid N-[1-(cyclopropanecarbonyl)piperidin-4-yl]-2-pyridin-3-ylacetamide 4-chloro-N,6-dimethyl-2-(propanoylamino)benzamide 3-amino-2,6-dimethylfuro[2,3-b]pyrazine-7-carboxylic acid;5-amino-4-fluoro-N-(1-hydroxybutan-2-ylidene)naphthalene-2-carboxamide;ethane 1-[3,5-bis(trifluoromethyl)phenyl]-2-butoxyethanol 1-(2,6-difluorophenyl)-7-[4-[3-hydroxypropyl-(2,2,2-trifluoroacetyl)amino]-2-methoxyanilino]-N-methyl-4H-[1,2,4]triazolo[4,3-a]quinoxaline-3-carboxamide 2-[4,5-bis(trifluoromethyl)pyrazol-1-yl]pyridine-3-carboxylic acid 6-chloro-2,3-dihydro-1H-benzo[e]indole-8-sulfonic acid 1-[(Z)-2-bromoethenyl]-3,7-dimethoxy-4H-quinoxaline 2-[3-fluoro-4-(methylamino)phenyl]-N-pyridin-2-ylquinoline-4-carboxamide N-[5-chloro-2-(1H-tetrazol-1-ium-5-yl)phenyl]pyridine-3-carboxamide 2-methylsulfinyl-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]acetamide 4-N,4-N-dimethyl-2-(5H-pyrrolo[3,4-b]pyridin-7-yl)-6H-1,3,5-triazine-4,6-diamine 2-[2-(5-methoxynaphthalen-1-yl)ethynyl]aniline (3R)-N-[(5R)-5H-imidazo[5,1-a]isoindol-5-yl]-3-methoxycyclohexane-1-carboxamide 3-[(2,4-dimethoxyphenyl)methyl]-1-(2-pyridin-2-ylethylcarbamoylamino)urea 6-[(3S)-oxolan-3-yl]oxy-4-oxo-1H-quinoline-2-carboxylic acid N-(4-aminophenyl)-5,6-dimethoxy-1H-benzimidazole-2-carboxamide 4-(1,3-benzodioxol-5-yl)-6-N-[(2S)-butan-2-yl]pyrimidine-2,6-diamine 4-[5-(2,6-dimethylpyridine-4-carbonyl)-3-(hydroxymethyl)-1H-pyrrol-2-yl]-N,N-diethylbenzenesulfonamide 4-[1-(2,5-dichlorophenyl)-3-methyl-6,7-dihydro-2H-pyrazolo[1,5-a]pyrazin-5-yl]-N-methylaniline (Z)-2,3-difluoro-N'-[4-[7-(1H-pyrazol-5-yl)quinolin-4-yl]oxyphenyl]pent-2-enimidamide 1-[4-chlorobutyl(2,3-dihydroxypropyl)amino]-N-phenylmethoxyformamide 2-[4-[[5-chloro-4-(2,3-dihydro-1H-inden-1-ylamino)pyrimidin-2-yl]amino]-7-methoxyindol-1-yl]ethanol N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-3,3-dimethylbutanamide;1-ethoxypropane 1-(cyclopropylmethoxy)-4-iodopyridin-2-one 1-cyclohexylbutylbenzene;ethane 5-methyl-N-[(1S)-2,2,3,3,4,4,5-heptafluorocyclohexyl]-1H-pyrrolo[2,3-b]pyridine-6-carboxamide N-[1-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)pyrrolidin-3-yl]prop-2-enamide [(E)-3-amino-2,2-difluoroprop-1-enyl]-[[4-amino-2-methyl-5-[4-(morpholine-4-carbonyl)phenyl]thiophen-3-yl]amino]azanium N-[(4S,5R)-1-ethyl-2-oxo-3,4-dihydropyrano[3,4-b]indol-8-yl]cyclopropanecarboxamide 6-[(1S,2R)-2-methylcyclohexyl]oxypyridine-3-carboxamide N-[6,7-dimethoxy-4-oxo-3-[(E)-2-phenylethenyl]chromen-5-yl]acetamide (3R)-4-[5-chloro-6-[2-(oxan-4-ylamino)ethoxy]pyridin-3-yl]-3-methylpiperazine-1,2-dione;2-methylpropane N-methyl-2,3-dinitroaniline 2-[2-(4-ethenylcyclohexen-1-yl)-6-methoxynaphthalen-1-yl]-5-pentoxypyrimidine N-[2,6-diamino-5-(3-aminophenyl)pyrimidin-4-yl]-2-methoxyacetamide [2-[(1S)-3,4-dihydro-1H-isochromen-1-yl]-2-oxoethylidene]cyanamide N'-[3,5-bis(trifluoromethyl)phenyl]propanediamide 3-[3,5-bis(trifluoromethyl)phenyl]propane-1-sulfonic acid (1S,2R)-N'-[5-chloro-4-[4-(3-fluorophenyl)piperazine-1-carbonyl]pyridin-2-yl]cyclopropanecarbohydrazide 4-(cyclobutylmethylamino)-2,6-diethoxypyridine-3-carbonitrile 1-butyl-3-[2-(4-cyclohexa-1,5-dien-1-yloxyphenyl)ethyl]imidazolidine-2,4-dione 2-(3,4-dihydronaphthalen-1-yl)-N-[6-[(2-oxopiperidin-1-yl)methyl]pyridin-2-yl]acetamide 1-[4-(3-oxopiperazine-1-carbonyl)phenyl]piperidine-2,6-dione 1-azido-3,5-dichloro-4-[1-(methoxymethyl)cyclopropyl]benzene N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)pyridine-2-carbohydrazide 2-[(2E)-2-[(2,4-diethoxyphenyl)methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid [1-(4-chlorophenyl)pyrrol-2-yl]sulfonylurea (7R)-5,9-dimethyl-6,7-dihydropyrimido[4,5-d]pyrimidine 4-[[1-(4-amino-2,3-difluorobenzoyl)-3-propan-2-ylazetidin-3-yl]methoxy]benzonitrile 4-amino-5-bromo-N-(2,6-difluorophenyl)pyridine-3-carboxamide 4-N,4-N-bis(2,5-dimethylphenyl)benzene-1,3,4-triamine 2,6-dimethyl-4-(2-methylpyrimidin-5-yl)benzonitrile 1-[4-(4-ethyl-5,7,12,14-tetrazapentacyclo[11.8.0.02,10.03,8.015,20]henicosa-1(13),2(10),3,5,7,11,15,17,19-nonaen-15-yl)phenyl]-N,N'-dimethylpyrrolidine-3-carbohydrazide N'-hydroxy-2-[4-(trifluoromethyl)phenoxy]pyrimidine-4-carboximidamide (2S)-N'-[4-cyano-3-(trifluoromethyl)phenyl]-2-ethylpentanediamide 2-chloro-7-methyl-N-[3,4,5-trimethoxy-6-(methylideneamino)cyclohexa-1,3-dien-1-yl]imidazo[1,2-a]pyridine-6-carboxamide (2R)-1,2,5-triphenylpentane-2,4-diol 3-methyl-N-[6-methyl-2-(1H-pyrazole-5-carbonylamino)cyclohexen-1-yl]thiophene-2-carboxamide 3-[4-[[5-[3,4-bis(fluoromethyl)phenyl]-1-(2,6-dichlorophenyl)pyrazole-3-carbonyl]amino]butyl]benzoic acid 7-benzyl-4-[(2E)-3,6-dimethylocta-2,6-dienyl]-8-hydroxy-1H-quinolin-2-one N-[6-(4-chlorophenyl)pyrimidin-4-yl]cyclopentanecarboxamide (3E)-1,5-dimethyl-3-[(2-methylphenyl)methylidene]indol-2-one 2-(6-chloro-4-oxochromen-3-yl)oxyacetic acid 4-(2,2-dimethylpropoxy)-5-iodopyrimidine N-[1-(oxolan-3-yl)piperidin-4-yl]-1H-indazole-5-carboxamide N-[2,6-di(propan-2-yl)phenyl]-4-(3-oxo-1H-isoindol-2-yl)butanamide;ethane 4-[(Z)-2-fluoroprop-1-enyl]-5-methoxycarbonylfuran-3-carboxylic acid 1-[4-(2,3-difluorophenyl)-5-methylpyrazol-1-yl]propan-2-one N-[2,6-di(propan-2-yl)phenyl]-3-oxobutanamide;ethane 2-[1,2-dihydroxyethyl(naphthalen-1-yl)amino]acetic acid 2-[1-azido-3,3,5-trimethyl-2,4-bis(phenylsulfanyl)piperidin-4-ylidene]acetonitrile 1-[4-(4-methoxyphenyl)piperazin-1-yl]-3-morpholin-4-ylpropan-2-ol 3,5-ditert-butyl-4-hydroxybenzenesulfonate 2-[4-(difluoromethoxy)phenyl]-N-[3-(hydroxymethyl)furan-2-yl]piperidine-1-carboxamide 2-(4-tert-butylphenoxy)sulfanylacetaldehyde;ethane (4R)-4-benzyl-3,3a,4,5,6,7-hexahydro-1H-pyrrolo[2,3-c]pyridine [(3Z,5E)-7-(4-aminophenyl)-2-methylhepta-1,3,5-trien-3-yl]-ethenyl-propan-2-ylhydrazine 5-amino-3-(4,6-dichloro-2-propylpyrimidine-5-carbonyl)oxy-2-(trifluoromethyl)benzoic acid 2-[(4-bromo-3-methoxyphenyl)sulfonylamino]propanoic acid 1-N,4-N-bis[(3,5-dichloropyridin-2-yl)methylideneamino]benzene-1,4-disulfonamide 5-[3-(3,4-dimethoxyphenyl)propylsulfanyl]-1,4-dihydronaphthalene 6-amino-5-(4-iodopyridine-2-carboximidoyl)-N,3-dimethylpyrimidin-3-ium-4-carboxamide N-[1-(2-chloro-4-methoxyphenyl)ethenyl]methanimine 4-[3-[(1R)-6,8-difluoro-7-hydroxy-2-oxo-1H-quinolin-3-yl]-5-(methoxymethyl)phenyl]piperidine-1-carboxylate N-[1-amino-3-imino-3-(4-phenylphenyl)prop-1-enyl]-3,5-dimethoxybenzamide 4-[(5,7-dimethyl-2-oxochromene-3-carbonyl)amino]butanoic acid 1-(4,5-diethylpyrimidin-2-yl)-N,N-diethylpiperidine-3-carboxamide 6,13-dimethyl-4-phenyl-5,7,11,12-tetrazatricyclo[8.3.0.02,6]trideca-1(10),2,4,7,11-pentaen-9-amine;N'-ethenyl-N'-ethyl-N-methylmethane-1,2-diamine N-ethyl-3,4-difluoro-N-methoxybenzamide 1-cyclohexyl-2,3,4,5-tetrafluorobenzene;ethane 3-[6-(2,4-difluorophenyl)pyrimidin-4-yl]-8-ethoxy-5H-[1,3]oxazolo[4,5-c]quinolin-4-one 1-(4-ethoxyphenyl)cyclohepta-2,4,6-trien-1-ol 4-(4,5,6a,7-tetrahydronaphtho[1,2-b]oxiren-10-yl)aniline [4-(3-ethynylanilino)piperidin-1-yl]-[(2S,6R)-2-phenyl-6-propan-2-ylmorpholin-4-yl]methanone N-[[5-methyl-3-(2,4,6-trifluorophenyl)imidazol-4-yl]methyl]piperidin-4-amine;dihydrochloride (Z)-3-amino-2-aminosulfanyl-1-[4-chloro-3-(1,2,5-thiadiazol-3-yl)phenyl]prop-2-en-1-one N-[(2S)-1-[[(4R,5R)-7-chloro-3-methyl-4,5-dihydro-2H-1,5-benzothiazepin-4-yl]amino]-3-ethyl-1-oxobutan-2-yl]oxolane-2-carboxamide 3-[(4,4-difluoropiperidine-1-carbonyl)amino]thiophene-2-carboxylic acid N-(3,4-dihydro-2H-quinolin-1-yl)-2-[(2E)-2-[2-(3,5-dimethoxyphenyl)ethylidene]hydrazinyl]-7,8-dihydro-6H-pyrano[3,2-d]pyrimidine-4-carboxamide (2S)-5,6-dimethoxy-7-oxo-3-phenylmethoxycarbonylnonanoate 1-[5-[4,6-bis(ethenyl)pyridin-2-yl]pentanoylamino]-2-(2,3-dihydro-1H-inden-2-yl)-1-methylideneguanidine 2-chloro-N,N'-dimethyl-4-[(3R)-1-[(6-methylpyridin-3-yl)amino]pentan-3-yl]benzenecarboximidamide 2-benzylimino-5,5,8a-trimethylspiro[1,3-dihydrothieno[2,3-d]pyrimidine-4,6'-piperidine] [4-methoxy-3,5-bis(2-phenylpropan-2-yl)thiophen-2-yl]boronic acid 6-methoxy-4-[(2,3,5-trichlorophenyl)diazenyl]naphthalene-1,2,3-triol 2-azido-5,7-difluoro-1H-pyrrolo[2,3-c]pyridine 5-butoxycarbonylbenzene-1,3-dicarboxylic acid [4-methyl-2,3-bis(phenylmethoxy)phenyl]boronic acid 5-azido-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfanylpyridine 1-[4-amino-6,7,8-trifluoro-3-(1H-indol-5-yl)quinolin-2-yl]oxy-3,3,3-trifluoropropan-2-ol 2-[2,4,6-tribromo-N-(2-phenylethyl)anilino]acetamide 1-azidooxy-5,6-dichloro-2-methyl-3,4-dihydroquinoline 3-chloro-6-(2-hydroxyethoxy)-1H-quinolin-4-one 5-[3-(difluoromethyl)-4,5,6,7-tetrahydroindazole-1-carbonyl]pyrazine-2-carboxylic acid N-[(Z)-1H-indol-3-ylmethylideneamino]-2,4-dioxo-7,8-dihydro-6H-quinoline-3-carboxamide 2-[3,5-ditert-butyl-4-(3-methylpentan-2-ylideneamino)phenyl]prop-2-enenitrile 4-[3-(azidomethyl)-5-pyridin-2-ylpyridin-2-yl]oxy-3,5-dichlorobenzonitrile 5-(3,4-diethoxyphenyl)-2,2-dimethylpentanal 4-[(1Z,3E)-1,4-bis(ethenyl)-6-methylhepta-1,3-dien-5-ynyl]pyridine (3-azidophenyl)methanesulfonic acid 5-[4-(trifluoromethyl)phenyl]-2,3-dihydropyridine (3E)-2-amino-4-[1-[3-[3,5-dichloro-4-(trifluoromethyl)phenoxy]propoxy]propan-2-ylidene]-6-oxo-3-[1-phenylethylidene]piperidine-1-carboxylic acid 2-azido-4-(4-methylsulfonylphenyl)pyrimidine 1,2-bis[(3,5-dibromophenyl)sulfonylmethyl]benzene (4S)-1-[3,5-bis(trifluoromethyl)phenyl]-2,2-difluoro-7-methoxy-4-methyloctan-4-amine 3-[6-ethyl-8-fluoro-9-(methylsulfanylamino)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carbonyl]cyclobutane-1-carboxylic acid 1-(6-azido-2,3-dihydroindol-1-yl)ethanone N-[(E)-1,3-diamino-2-(2,4,6-trimethylphenyl)prop-2-enylidene]-2-pyridin-3-ylacetamide 4-[5-(difluoromethyl)-3-methoxypyridin-2-yl]oxan-4-ol ethene;1-ethenyl-4-methoxybenzene;2-ethylpiperidine 1-(3,5-dimethylphenyl)-4-[2-hydroxyethyl(propyl)amino]-2-(trifluoromethylsulfanyl)butane-1,4-dione;1-methoxy-4-propan-2-ylbenzene 4-[(1R,2S)-1-hydroxy-1-pyridin-3-ylbutan-2-yl]piperazine-1-carboxylic acid [4-(6,7-dimethoxyquinazolin-2-yl)oxynaphthalene-1-carbonyl]carbamic acid ethane;N-[[4-(5-methyl-1H-pyrrole-2-carbonyl)phenyl]methyl]cyclopropanecarboxamide 1-butylnaphthalene;8-[2,3-dihydroxypropyl(methyl)amino]-6H-benzo[c]chromene-9-carboxylic acid 6-[2,6-difluoro-4-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydronaphthalene-2-carbonitrile 3-(2,6-dimethylphenoxy)-N'-hydroxypyrazine-2-carboximidamide 3-(2-cyclopenta-1,4-dien-1-ylethoxy)-5-[2-(2-propan-2-yl-1H-indol-3-yl)ethyl]benzoic acid 2-N,4-diamino-1-N-azidobenzene-1,2-disulfonamide 5-[4-[(1S,3R)-3-aminocyclopentyl]phenyl]-N-methylpyrimidin-2-amine (7S)-5-(4-methoxyphenyl)-7-[3-methyl-2,6-dioxo-1-(4-phenoxybutyl)pyrimidin-4-yl]-6,7-dihydro-5H-pyrazolo[1,5-a]pyridine-2-carboxylic acid 5-chloro-N-[[(3S,4R)-1-pyridin-2-yl-4-(pyrrolidine-1-carbonyl)pyrrolidin-3-yl]methyl]thiophene-2-carboxamide;2,2,2-trifluoroacetic acid N-(4-tert-butyl-3,4-dihydropyridin-6-yl)-5-[5-[2-[4-(1H-imidazol-2-ylsulfonyl)anilino]pyrimidin-4-yl]thiophen-2-yl]furan-2-carboxamide (6R)-3-[[4-(trifluoromethyl)phenyl]carbamoylamino]-7-[(1,2,4-thiadiazole-5-carbonylamino)methylsulfonyliminomethyl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2,4,6-tetraene-11-carboxylic acid N-[2-(1H-pyrazole-5-carbonylamino)ethyl]-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-3-carboxamide 2-(7,8-dihydroimidazo[1,5-a]pyrazin-3-yl)-N'-hydroxy-6-methoxypyridine-4-carboximidamide 7-[4-(6,8-dihydro-5H-pyrido[3,4-c]pyridazine-7-carbonyl)phenyl]-6,6-dimethyl-5H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile 2-(3,4-dimethoxyphenyl)-1-[3-fluoro-5-[(6-oxo-1H-pyridin-3-yl)methyl]piperidin-1-yl]ethanone 1-[4,5-diethoxy-2-(piperidin-4-ylamino)phenyl]ethanone 4-[1-[3-(2,5-dimethylfuran-3-carbonyl)azetidine-1-carbonyl]cyclopropyl]benzoic acid 5-[2,3-dimethyl-4-(trifluoromethoxy)phenyl]-2,3-dihydro-1H-indene N-[(3S)-1,1-dioxothiolan-3-yl]-3,4-dimethoxybenzamide 5-[4-amino-7-methyl-6-[1-(3-pyrrolidin-1-ylpropoxy)ethyl]pyrrolo[2,1-f][1,2,4]triazin-5-ium-5-yl]-N-(4-morpholin-4-ylphenyl)pyrazolidine-3-carboxamide (5S)-2-(4-acetamidoanilino)-N-(3,4-dichlorophenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 7-[2-(dimethylamino)ethyl]-5,6,8-trifluoronaphthalen-1-ol 4-[(6,7-dimethoxyquinazolin-4-yl)amino]-5-fluoro-2-[1-(3-hydroxypropanoyl)piperidin-4-yl]oxybenzamide 4-bromo-3,5-diethoxyphenol N-[(4-azidooxyphenyl)methyl]-1,3-thiazol-2-amine 4-(1H-benzimidazol-2-ylsulfanylmethyl)benzonitrile 2-[(3,4-difluorophenyl)methyl]-1,5-dihydroisochromeno[3,4-c]pyridine (5E)-2-cyclopentylimino-5-[(1,3-dimethoxynaphthalen-2-yl)methylidene]-1,3-thiazolidin-4-one (NZ)-4-methyl-N-[(6-pyrrolidin-1-ylquinolin-2-yl)methylidene]benzenesulfonamide 1-[3-(2,6-dichlorophenyl)propyl]-N-[1-(5,6-dimethoxypyridine-3-carbonyl)pyrrolidin-3-yl]triazole-4-carboxamide N-[(3S,4R)-1-cyclohexyl-3-[2-(4-hydroxyphenyl)ethynyl]piperidin-4-yl]pyridine-2-sulfonamide 2-[1-(2,4-difluorobenzoyl)-3-hydroxypiperidin-3-yl]oxypyridine-4-carbonitrile 1-[4-[5-[6-(2,3-dihydro-1H-inden-2-yl)pyridin-3-yl]pentoxy]phenyl]ethanone 3-(2-anilinoquinazolin-6-yl)-N-benzylcyclobutane-1-carboxamide 4-(2,5-dichloro-4-pyrrolidin-1-ylanilino)sulfanylbenzoic acid N-ethylsulfonyl-2,4,6-trimethylbenzenesulfonamide 2-[4-methyl-6-(oxan-2-yloxy)pyridin-3-yl]-1,3-thiazole 4-[2,3-difluoro-4-(2,3,5,6-tetrafluorophenoxy)phenyl]-7,8-dihydroisoquinoline N-[4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]-2-methoxy-N-(2-nitrophenyl)acetamide 4-fluoro-N-[1-[2-[(2R)-5-oxopyrrolidin-2-yl]ethyl]-6-propan-2-ylpiperidin-3-yl]benzamide 5-(3,4-dichlorophenoxy)-2,3-bis[ethoxy(ethylsulfanyloxy)phosphoryl]pyrazine N-[2,6-dimethyl-4-(methylideneamino)phenyl]-6-methoxypyridine-3-carboxamide 3-[1-methyl-4-oxo-7-(trifluoromethoxy)quinolin-3-yl]-N-propanoylpropanamide 6-(6,7-dihydro-5H-[1,3]dioxolo[4,5-f]benzimidazol-7-yl)pyridine-2-carbonitrile N-[5-chloro-4-(1,3-thiazol-2-yl)pyridin-2-yl]-6-oxopiperidine-2-carboxamide 3-[2,4-dichloro-6-(trifluoromethyl)phenyl]-5-cyclopropyl-1H-pyrazole 4-[3-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]prop-2-ynamide 1-phenyl-4-(1,2,3,6-tetrahydropyridine-5-carbonyl)piperazin-2-one 4-methyl-1,6-diphenylmethoxypyridazine-3-thione 4-hydroxy-1,3-diphenylbutan-2-one 1-(2-azidoethyl)-3-methoxynaphthalene 5-[4-(3,4-dimethoxyphenyl)-2H-1,3,5-triazin-6-yl]-1,3,8-thiadiazecane N-[(1R,2R)-2-methoxycyclohexyl]-4-(oxolan-3-yloxy)benzamide 1-[[4-[(2,6-dioxopiperidin-3-yl)carbamoyl]phenyl]methoxy]piperidine-4-carboxylic acid 5-[3,4-bis(phenylmethoxy)phenyl]imidazolidine-2,4-dione 4-(3-methylphenoxy)-2,6-bis[3-nitro-5-(trifluoromethoxy)anilino]quinoline-7-carbonitrile N-[4-fluoro-5-(2-pyrrolidin-1-ylethoxy)-2,3-dihydroinden-1-ylidene]hydroxylamine [4-(2,5-dimethoxyphenyl)piperazin-1-yl]-(3-propan-2-ylimidazo[4,5-b]pyridin-6-yl)methanone 2-[3-(2,4-difluorophenyl)propanoyl]cyclohexane-1,3-dione 3-[5-fluoro-2-(trifluoromethoxy)phenyl]oxirane-2,2-dicarbonitrile 4-[2-azido-6-(1,3-benzodioxol-5-yl)pyridin-3-yl]oxy-N,N-dimethylaniline 1-[4-(aminomethyl)phenyl]cyclopropane-1,3-dicarboxylic acid 3-[6-(4-tert-butylpiperazin-1-yl)pyrimidine-4-carboximidoyl]phenol N-[4-methylsulfanyl-2,6-di(propan-2-yl)phenyl]methanesulfonamide N-[4-(dimethylamino)phenyl]-2,5-dihydrotetrazol-1-amine 1-(2-butyl-4-methoxyphenyl)ethanone;7H-purin-6-amine [2-(aminomethyl)azetidin-1-yl]-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)phenyl]methanone 5-[(4,6-dimethoxypyrimidin-2-yl)carbamoyl]-1-phenylpyrazole-3-carboxylic acid 2-(3,5-difluoro-4-morpholin-4-ylanilino)-6-(oxan-3-ylmethoxy)-1H-quinoline-4-thione 4-[3-(azepan-1-yl)pyrrolidine-1-carbonyl]-2,6-dimethoxybenzonitrile 4-amino-2,6-dimethyl-1H-pyridine-3,5-dicarboxylic acid 1-(azidomethyl)-3-[3,5-bis(trifluoromethoxy)phenyl]-N-(4-pyridin-2-yloxan-4-yl)azetidine-2-carboxamide 2-[(5R,7S)-5-benzyl-7-ethynyl-6-methoxy-7H-imidazo[1,2-a]imidazol-3-yl]phenol 1-[(4S,5R)-2,2-dimethyl-3-phenyl-3-azabicyclo[3.1.0]hexan-6-yl]-N-isoquinolin-6-ylmethanesulfonamide [6-(dimethylamino)pyridine-3-carbonyl]-phenylazanium N-(4-hydroxynaphthalen-1-yl)-1H-benzimidazole-2-carboxamide 3-[5-(5-bromo-2,4-difluorophenyl)-1H-pyrazol-4-yl]-7-oxa-3,10-diazaspiro[5.6]dodecan-11-one 5-azido-2,3-dimethylquinoxaline N-[(Z)-1-amino-3-hydroxybut-2-enylidene]-2,4-dimethylbenzamide 1-(3,5-dichlorophenyl)-N-[2-[4-[3-(trifluoromethoxy)phenyl]piperazin-1-yl]ethyl]pyrrolidine-3-carboxamide 4-N,6-bis[2-(diethylamino)ethoxy]-5-N-[[6-(dimethylamino)pyridin-3-yl]methyl]pyrimidine-2,4,5-triamine 4-[3-(6,7-dimethylquinolin-2-yl)prop-1-enyl]morpholine 2-cyclohexyl-3,4-dimethylbenzoate 2-(4-cyclopropylphenyl)-1-[7-methoxy-5-(2-oxopyrrolidin-1-yl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]ethanone 5-(3,4-dihydro-2H-1,5-naphthyridine-1-carboximidoyl)-6-methyl-2,4-bis(2-methylphenyl)pyridin-3-amine N-[4-methyl-2-(trifluoromethoxy)phenyl]-4-phenoxypyrimidine-5-carboxamide 1-benzyl-4-methylcyclohexa-3,5-diene-1,2-disulfonic acid 1-azidooxy-3-(2-butylphenyl)benzene 6-chloro-2-N-(4,5-dihydropyren-1-yl)quinazoline-2,3-diamine 2-(2,3-dichlorophenyl)imino-5,6-bis[[1-(4-methoxyphenyl)triazol-4-yl]methylsulfanyl]-7H-[1,3]thiazolo[4,5-d]pyrimidin-8-one 2-[5-(3,5-dimethoxy-4-methylphenyl)pyrazin-2-yl]-1H-benzimidazole;ethane 2-[4-chlorobutyl(1,3-thiazol-5-yl)amino]benzenesulfonic acid 5-[6,7-dimethoxy-1-(pyridin-2-ylmethyl)quinazolin-4-ylidene]-2H-triazole-4,6-diamine (3S)-N-[3-fluoro-5-[[6-methoxy-7-(2-methylbutan-2-yloxy)quinazolin-4-yl]amino]phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide N-[2-amino-3-(1-methylcyclohexa-2,4-dien-1-yl)-1H-indol-5-yl]-4-chlorobenzamide 4-[5-[(Z)-1,2-diaminoethenyl]-3H-1,2-oxazol-2-yl]benzonitrile 1-(2-ethylphenyl)-4-methoxy-9H-pyrido[3,4-b]indole N-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide 2-(3,6-dihydroxyoctyl)benzenesulfonic acid (5S)-3-[3,5-difluoro-4-[6-methoxy-7-(piperidin-4-ylsulfanylmethyl)quinolin-4-yl]oxyphenyl]-2-oxo-1,3-oxazolidine-5-carboxylic acid 5-ethyl-3,4-difluoro-2-(4-methoxyphenyl)benzoic acid 1-[1-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperidin-3-yl]triazole-4-carboxylic acid 3-[[(2S)-1-(cyclopropanecarbonyl)pyrrolidin-2-yl]methoxy]pyridine-4-carboxamide 2-[2,6-dimethyl-4-(8-oxo-3-phenyl-5H-pyrido[2,3-b]pyrazine-7-carbonyl)phenoxy]acetic acid (5S)-N-(2,4-difluorophenyl)-2-methylsulfanyl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 1-[[4-(5,6-dimethylpyridin-3-yl)cyclohexanecarbonyl]amino]cyclopropane-1-carboxylic acid 5-amino-N-(2,3-dihydro-1H-inden-4-yl)-7-methoxy-8-[6-(2-piperidin-1-ylethoxy)naphthalene-2-carbonyl]-9H-carbazole-4-carboxamide 2-(N-hexadecanoylanilino)benzenesulfonic acid N-(4-aminophenyl)formamide;2,3-dichloro-6,7,11b-trihydroxy-9H-indeno[1,2-a]inden-5-one 1-(7,8-dihydronaphthalen-2-ylsulfonyl)-3-[4-fluoro-3-(trifluoromethyl)phenyl]-4-(pyridin-3-yloxyamino)pyrrolidine-2,5-dione 1-azido-2-ethoxy-3,4-difluorobenzene 5-[4-chloro-6-(trifluoromethyl)pyrimidin-2-yl]-1,3-dihydrobenzimidazole-2-thione 2-[4,5-dimethyl-3-(6-morpholin-4-ylpyridin-3-yl)-1H-pyrrol-2-yl]acetamide N-[3-(4-fluorophenyl)-1,2-oxazol-5-yl]-6-hydroxyhexanamide 5-[[4-chloro-2,6-di(propan-2-yl)phenyl]carbamoylamino]pyridine-2-carboxylic acid N-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2,3-difluorophenyl]-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxamide N-[4-fluoro-2-(6-fluoro-1H-indole-3-carbonyl)phenyl]acetamide 2-[1-[4,5-dimethyl-6-(propanoylamino)pyridin-3-yl]sulfonylpiperidin-2-yl]acetic acid 2-methyl-4-[3-[5-(2,4,6-trimethylphenyl)-1H-pyrrol-3-yl]propylamino]butan-2-ol N-[4-(3,3-difluoropiperidin-1-yl)phenyl]-6-hydroxyspiro[2H-1-benzofuran-3,4'-piperidine]-1'-carboxamide 4-cyclopropyl-2-[6-(1,1-dioxothietan-3-yl)pyridin-2-yl]oxybenzonitrile 1-(4-methylcyclohexyl)-3H-pyrido[2,3-d]pyrimidine-2,4-dione N-[(4-fluorophenyl)methyl]-1-[7-hydroxy-5-(pyridine-3-carbonylamino)-6H-naphthalen-2-yl]-6-oxopyrimidine-5-carboxamide 4-[(2S,3R)-1,5-dihydroxypentan-2-yl]oxycarbonylbenzoate 1-azidooxy-4-chloroisoquinoline (2R)-1,4,6-trimethyl-N-[(3R)-piperidin-3-yl]-2,3-dihydroquinoxaline-2-carboxamide;hydrochloride N-[5-[2-(4-azidooxycyclohexyl)ethynyl]-2-phenylpyrazol-3-yl]benzenesulfonamide N-[2-(1,5-dimethylpyrazol-4-yl)ethyl]-8-fluoro-6-methoxyquinoline-3-carboxamide 1-[4-fluoro-2,5-bis(trifluoromethyl)phenyl]-3-[5-methanimidoyl-6-(methoxyamino)pyridin-2-yl]urea (5R)-3,4,6,8-tetrahydroxy-7,8-dimethyl-N-[4-(trifluoromethyl)phenyl]octa-1,6-dien-2-yl]octanamide 3-(5,7-diethylquinolin-6-yl)-2-oxopropanoic acid N-(3,4-dichlorophenyl)-2-(3-methoxy-4-nitrosoanilino)acetamide 4-chloro-N,6-diethylthieno[2,3-d]pyrimidine-5-carboxamide;3,4-dihydro-1H-1,8-naphthyridin-2-one N-[3,5-bis(trifluoromethyl)phenyl]-2-(4-cyclopentylpiperazin-1-yl)-1H-pyrazine-2-carboxamide 3-(4-methoxyphenyl)-2H-indene-1,5-dione N-(2,4-dichloropyrimidin-5-yl)-1,2-oxazole-3-carboxamide (3S)-6-methoxy-N,2-dimethyl-4-oxo-2,3-dihydrochromene-3-carboxamide 4-N,4-dimethylbenzene-1,3,5-tricarboxamide 1-[2-(3,5-dimethoxyphenyl)ethynyl]cycloheptane 2-[6-chloro-1-(3,4-dimethoxyphenyl)-2H-pyridin-5-yl]-3-hydroxy-2,7a-dihydro-1H-azirino[2,1-b]quinazolin-8-one 2-methyl-N,3-bis(2-nitrophenyl)aniline N-[(2S)-5-amino-4,5-dioxopentan-2-yl]-6-hydroxynaphthalene-1-carboxamide 2-[7,8-difluoro-2-(4-methylcyclohexyl)-1,2,3,4-tetrahydronaphthalen-1-yl]-5-(2-methoxyethyl)pyrimidine 2-methyl-4-oxo-5-phenoxypentanoic acid 4-[[8-(2,6-difluorophenyl)-7H-purin-2-yl]amino]benzaldehyde 2-[(4E)-3,5-dimethylhepta-1,4,6-trien-2-yl]-1-fluoro-4-[(Z)-hept-1-enyl]benzene;propane (3R)-1-[2-[6-amino-5-(1,3-thiazol-2-ylmethoxy)pyridin-3-yl]phenyl]pyrrolidine-3-carboxamide 1-[3-(4,5-dihydrobenzotriazol-2-yl)phenyl]hexan-3-one (4Z)-3-methyl-4-[[3-nitro-6-propoxy-2-(trifluoromethyl)phenyl]methylidene]-1,2-oxazol-5-one [2-amino-6-(4-methylphenyl)pyrimidin-4-yl]-(5,6-dichlorocyclohexa-1,3-dien-1-yl)methanone [(E)-2-(4-chlorophenyl)ethenyl]-dimethyl-[3-[methyl(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)amino]propyl]azanium 4-[3-(diethylamino)propylcarbamoyl]benzoic acid 2-(N-butylanilino)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carbonitrile 1-cyclopentyloxy-4-[5,6-dichloro-1-(4-chloro-3-methylphenyl)sulfonyl-2-methylindol-3-yl]cyclohexa-2,4-diene-1-carboxylic acid 3-(2,6-difluorophenyl)sulfanyl-1H-indole 1-[3-(cyclohexylmethyl)phenyl]ethanol 3-cyclobutyloxy-7,8-dihydro-6H-quinoline (3S,4R)-4-(4-methoxy-1H-indazol-7-yl)pyrrolidine-3-carboxylic acid 1-[4-[2,6-bis(2-methylbutan-2-yl)phenoxy]-1-phenylbutyl]piperidine (3S,4R)-1-[[4-chloro-5-(cyclopropylmethoxy)-2-fluorophenyl]methyl]-4-(hydroxymethyl)pyrrolidine-3-carboxylic acid 4-[2,6-di(propan-2-yl)phenyl]-5-(4-hydroxyphenyl)triazole-1-carboxylic acid 1-[5-[(2E,4Z)-3-methylhepta-2,4,6-trienoxy]-4H-pyran-2-yl]ethanone 1-cyclohexyl-2-methyl-4-[(3S,5R)-2-methylideneheptanoyl]pyrrole-3-carboxylic acid [(2S)-1-amino-5-azido-4,4-dimethylpentan-2-yl]-phenylcarbamic acid (1R,2S)-1,2-bis[(6-chloropyridine-3-carbonyl)amino]guanidine 1-azido-2-(methoxymethyl)-3,4-dihydro-2H-quinoline N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-5-nitro-N-(2-nitrophenyl)-1,3-thiazol-2-amine (3S)-4-[6-amino-5-(3-propan-2-yloxyphenyl)pyrazin-2-yl]-1-[[5-chloro-2-(tetrazol-1-yl)phenyl]methyl]pyrrolidin-3-ol ethane;5-fluoro-4-N,6-dimethylpyrimidine-2,4-disulfonamide 1-[4-[5-(6-chlorocyclohexa-2,4-dien-1-yl)pyridin-3-yl]phenyl]-N-methylpropan-1-imine;4-ethoxybenzoic acid N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-4-(3,5-dimethoxyphenyl)benzamide [3-bromo-4-(5,5-dimethyl-1H-tetrazol-4-yl)phenyl]boronic acid 4-methyl-5-(2-nitrophenyl)-6-piperidin-1-ylpyrimidine N'-(3-nitrophenyl)sulfonylpiperidine-4-carbohydrazide 3-ethylhexanedioate;trimethyl(2-pyridin-2-ylethyl)azanium N-[5-cyano-2-(1-methoxyethenyl)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide 2-[4-chlorobutyl(hexanoyl)amino]benzenesulfonic acid 3-(1H-indazol-4-yl)butanamide N-[2,3-dihydrofuran-5-ylmethyl(1H-imidazol-5-yl)carbamoyl]benzamide 3-(4-butoxyphenyl)bicyclo[1.1.0]butan-1-ol 2-(4-hydroxyphenyl)acetamide;methane 3-[(1R,2R)-2-hydroxy-4-phenylcyclohexyl]propanoic acid [4-hydroxy-3,5-bis(phenylmethoxy)cyclohexa-1,5-dien-1-yl]-piperidin-2-ylmethanone 2-[[4-[[6-(3,4-difluorophenyl)imidazo[1,5-a]pyridin-8-yl]amino]-2-ethylbenzoyl]amino]acetic acid;methanol 3-[(2,6-dichlorobenzoyl)amino]-N-(3-piperidin-1-ylsulfonylphenyl)benzamide;2,2,2-trifluoroacetic acid 3-[4-(4-chlorophenoxy)-2,6-dimethoxyphenyl]cyclopropane-1,1,2,2-tetracarbonitrile 5-[2,6-dimethyl-4-[[5-(trifluoromethyl)pyrazin-2-yl]sulfamoyl]phenyl]-N-(2-hydroxyethyl)-1H-pyrrole-3-carboxamide (6S)-4,12-dibenzyl-9-oxa-3,5,15,17-tetrazatetracyclo[8.7.0.02,7.011,16]heptadeca-1(10),2(7),3,11(16),12,14-hexaene;methane N-cyclopropyl-2-[(1S,3R)-4-[2-(ethylideneamino)imidazol-1-yl]-3-hydroxycyclohexyl]acetamide N-[3-[1-(cyclopropylmethylamino)-4-methoxypiperidine-4-carbonyl]phenyl]-2,6-difluorobenzenesulfonamide 1-[(3R,4S)-4-aminopyrrolidin-3-yl]-N-(2-anilinoethyl)methanesulfonamide;dihydrochloride (3R)-N',2-dihydroxy-3-[[4-(4-nitroanilino)phenyl]sulfonylamino]butanediamide ethane;3-[[(2E,4Z)-5-methylhepta-2,4,6-trien-3-yl]amino]-4-(2-propan-2-ylimidazol-1-yl)benzoic acid 1-ethenyl-4-(2,3,5-tributylphenyl)benzene [[6-cyclopropyl-5-(2,2-dimethoxyethoxy)pyridin-3-yl]amino]phosphonic acid 1-[(E)-2-chlorobut-2-enyl]-4-(4-methoxyphenyl)-7H-pyrrolo[3,2-c]quinoline 3-(1-cyclopropylsulfanylpiperidine-4-carbonyl)-7,8-dimethoxy-5-methyl-2H-benzo[g]quinazolin-4-one (5Z,6E)-2-amino-4-[amino-(3-methoxyphenyl)methyl]-6-ethylidene-9H-pyrido[2,3-b]indol-7-one;1-[2-[6-(4-tert-butylcyclohexen-1-yl)oxypyridin-3-yl]morpholin-4-yl]-2-piperazin-1-ylethanone 4-(5-amino-6-sulfanylidene-1H-pyrimidin-4-yl)piperidine-1-carboxylic acid 6-[(3S,4R)-3-amino-4-methylpyrrolidin-1-yl]-5-chloropyrazine-2-carbonitrile;hydrochloride 2-methyl-3-(3,4,5-trifluorophenyl)benzenesulfinic acid 1-[(2S)-1-[3,5-bis(trifluoromethyl)phenyl]pyrrolidin-2-yl]propan-2-amine 4-chloro-1-iodopyrazolo[3,4-b]pyridine 2-(2-chlorophenyl)-2-ethoxypentanoic acid 2-[4-[3,5-bis(trifluoromethyl)phenyl]phenyl]-5-methylthiophene N-(2,4-dimethoxyphenyl)-1-[3-oxo-7-(quinolin-6-ylmethyl)imidazo[5,1-f][1,2,4]triazin-4-ium-4-yl]pyrrolidine-2-carboxamide;chloride 4-(azidomethyl)-2,5-dimethoxypyrimidine N-[4-(2-methoxyphenyl)-1,3-thiazol-2-yl]-5-oxo-6-azaspiro[3.4]octane-6-carboxamide N-[[1-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)cyclopropyl]methyl]furan-2-carboxamide 5-methoxy-2,2,4-trimethyl-1H-quinoline (2S)-3,4-dihydro-2H-chromene;4-[5-methyl-6-[(1Z,3E,5Z)-octa-1,3,5-trienoxy]pyridin-2-yl]-N'-propanoylpiperazine-1-carboximidamide 1-methyl-5-(2,3,5-trichlorophenyl)pyrazole (2S,3R)-1-benzyl-5-chloro-6-(methoxycarbonylamino)-2,3-dihydroindole-2-carboxylic acid [1-(6,7-dihydrothieno[3,2-c]pyridin-5-yl)-4-methoxybutan-2-yl]carbamic acid (3R,4S)-1-[2-(1H-benzimidazol-2-ylsulfanylmethoxy)ethyl]-4-hydroxypyrrolidine-3-carboxylic acid;dihydrochloride 2-(4-methylphenyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrimidine 4-bromo-N-[5-cyano-2-methyl-4-(trifluoromethoxy)phenyl]-1,3-thiazole-5-carboxamide N-[1-(2,3-dihydroindole-1-carbonyl)cyclohexyl]-3-(5H-imidazo[5,1-a]isoindol-5-yl)benzamide 4-[2,3-dihydroxypropyl(propyl)amino]benzenesulfonic acid 1-(4-cyclopropylpiperazin-1-yl)-2,2-difluoroethanone;4-[[3-(4-fluorophenyl)imidazo[1,2-a]pyrazin-8-yl]amino]-N'-methyl-2-oxo-1H-pyridine-3-carboximidamide 4-amino-5-benzylsulfanyl-N'-hydroxypyridine-2-carboximidamide 7-benzyl-1,3-dimethylidene-2,5-diphenyl-6,8-dihydrobenzo[f]isoindole;ethane 2-[N-(3-aminopropyl)-5-bromo-2-nitroanilino]ethanol 4-[1,3-diamino-2-carbamoyl-3-(methyliminomethyl)prop-2-enylidene]-N-[2-fluoro-6-(trifluoromethyl)phenyl]piperidine-1-carboxamide;3,5-dichloroaniline 3-[4-(6-aminopyridin-1-ium-3-yl)phenyl]hexanoic acid N-[3-[2-(3,4-difluorophenyl)pyrrolidin-1-yl]propyl]methanesulfonamide 5-[2,6-difluoro-4-(2-methylbutoxy)phenyl]imino-1-(2-hydroxyethyl)-3-propan-2-ylidenepyrrolidin-2-one N-[(2S)-6-fluorospiro[1,3-dihydroisochromene-4,1'-cyclopropane]-2-yl]-5-methoxypyrimidin-2-amine 2-[(2Z)-4-oxo-2-[(Z)-phenylmethoxyiminohydrazinylidene]-1,3-thiazolidin-5-yl]-N-(4-propan-2-ylphenyl)acetamide 3-azido-7,8-dimethoxy-2,6-bis(phenylsulfanyl)quinoxaline (6R)-1,3-dimethyl-2-[(E)-3-pyridin-4-ylprop-2-enimidoyl]-6-[4-[5-(trifluoromethyl)pyrimidin-2-yl]phenyl]-6,7-dihydro-5H-pyrrolizin-8-one 5-[8-(3,5-dimethyl-1,2-oxazol-4-yl)-7H-purin-6-yl]pyridin-2-amine 3-amino-N'-ethylthieno[2,3-b]pyridine-5-carboximidamide N-[(1R)-5,7-dihydroxy-2,3-dihydro-1H-inden-1-yl]-3-(4,6-dimethoxypyrimidin-2-yl)benzamide N-azido-2-(2,6-difluoroanilino)benzamide 1-(6-bromonaphthalen-2-yl)-5,7-dihydroxy-8-(4-methylcyclohexyl)oxyoctan-4-one 4-[(3,5-dimethoxyphenyl)methylamino]-2-(3-hydroxypropylamino)pyrimidine-5-carboxamide 2-[6,7-dihydro-5H-1,3-benzothiazol-4-ylidene(methoxy)amino]-N-ethylacetamide 6-[4-chlorobutyl(3-methylbutyl)amino]-5-nitronaphthalene-2-sulfonic acid 4-[2,2-dimethoxyethyl(phenacyl)amino]-N-(2-phenylpyrazol-3-yl)benzenesulfonamide 3-[5-(4-methoxyphenyl)-1H-pyrazol-3-yl]piperidine;3,3,3-trifluoroprop-2-enal 1-[(3R,4S)-4-(dimethylsulfamoylamino)oxolan-3-yl]sulfonyl-2-phenylpiperidine 3-[1,5-bis(trifluoromethyl)indol-2-yl]-N'-hydroxypyridazine-4-carboximidamide 3-[1-(2,4-dichlorophenyl)ethyl]-7H-purin-6-imine 2-[1,3-dihydrobenzo[f]chromen-2-yl(hydroxy)methoxy]benzamide 1-methyl-5-(4-pyridin-2-ylpiperazine-1-carbonyl)pyrazole-4-carboxylic acid 4-[5-[(4R)-7-chloro-10-(oxan-2-ylmethoxymethyl)-3,4-dihydro-1H-benzo[b][1,6]naphthyridine-2-carbonyl]pyridin-2-yl]oxycyclohexane-1-carbonitrile [2-(butylamino)phenyl]-methoxyphosphinic acid [(1R)-2,3-dihydro-1H-inden-1-yl]carbamic acid N-[(Z)-1-aminoethylidenecarbamothioyl]-4-[3,5-dichloro-4-(3,3,3-trifluoropropoxy)phenoxy]-2-fluorobenzamide 3-[(2,4-dichloropyrimidin-5-yl)-(6-nitro-1,3-benzothiazol-2-yl)amino]butanoic acid 3-bromo-6-chloro-5-hydroxy-1-methylbenzimidazol-2-one 4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxylic acid 4-[[7-[(2Z)-2,3-dimethylpenta-2,4-dienyl]quinolin-6-yl]methyl]-1,3-thiazole 1-methyl-3-phenyl-2,4-dihydrotriazolo[4,5-b]pyridine-4,6-dicarboxylic acid [4-(2,6-dimethylphenoxy)phenyl]-methoxyphosphane (Z,5E)-6-bromo-2-cyano-3,3,7-trimethyloct-5-enoic acid;(4R)-4-amino-6-phenylhexanal 2-chloro-N-[(1R)-1-(4-fluorophenyl)ethyl]-9H-fluoren-1-amine 6,8-ditert-butyl-4H-isoquinoline 5-methyl-4-(2-methylphenyl)-N-[1-(3,4,5-trimethoxyphenyl)imidazol-4-yl]pyrimidin-2-amine 1-[3,5-dimethyl-4-(2,2,2-trifluoroethoxy)pyridin-2-yl]-3-methoxy-4-[[4-methanimidoyl-5-(oxolan-3-ylamino)pyrimidin-2-yl]amino]butan-2-one 3-[(2R)-1-hydroxypropan-2-yl]oxy-5-[6-[(3S)-3,4,5-trimethylpiperazin-1-yl]pyridazin-3-yl]benzonitrile 4-(3-azidophenoxy)benzenesulfonic acid 2-[N'-(4,6-dimethylpyrimidin-2-yl)carbamimidoyl]sulfanyl-N,N-dimethylacetamide 4-benzyl-5,6-difluorocyclohex-2-en-1-one 2-[2,6-di(propan-2-yl)phenyl]imino-5-(quinolin-8-ylmethylidene)-1,3-thiazolidin-4-one 2-amino-N-[(5-tert-butylthiophene-3-carbonyl)amino]acetamide 3-[3,5-dichloro-4-[(4-hydroxy-2-oxochromen-6-yl)oxymethyl]phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 1-[(5E)-5-ethylidene-6,6-dimethylocta-2,7-dienoxy]-4-fluorobenzene 4-[4-(3-chloro-5-methoxyphenyl)piperazine-1-carbonyl]-2,2-dimethylchromene-6-sulfonamide 2-[(5Z)-4-oxo-2-sulfanylidene-5-[[1-[3-(trifluoromethyl)phenyl]imidazol-4-yl]methylidene]-1,3-thiazolidin-3-yl]acetic acid 4-(3-chlorophenyl)sulfinyl-N,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-2-chloro-4-[3-[(Z)-2-hydroxy-2-(1-methylbenzimidazol-2-yl)ethenyl]-1H-pyrazol-5-yl]benzamide N-[(2S)-1-hydroxypropan-2-yl]-1H-indole-4-carboxamide 4-(2,3-dihydroindol-1-yl)-6-hydroxycyclohepta-2,4,6-trien-1-one 2-[6-(3,4-dimethylphenyl)-5-(4-fluorocyclohepta-1,3,7-trien-1-ylamino)pyridin-3-yl]acetamide N-[4-chloro-2-(thiophene-3-carbonyl)phenyl]-4,5-dimethyl-1H-pyrazole-3-carboxamide [4-methyl-2-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)pyrazol-3-yl]-(2,4,6,7-tetrahydrotriazolo[4,5-c]pyridin-5-yl)methanone 5-(1,3-benzothiazol-6-yl)-N-[2-methoxy-4-(oxan-4-ylamino)phenyl]-1H-pyrrole-3-carboxamide 2,6-dichloro-N-(6-ethylpyridin-3-yl)benzamide;1H-imidazole N-[2-[4-(3,5-dimethylpyridin-4-yl)piperazine-1-carbonyl]phenyl]ethanesulfonamide 5-(3-aminopropyl)-2,4,6-triethoxybenzene-1,3-diamine 4-(2,6-dimethoxyphenyl)cyclohex-3-en-1-ol;ethane N-(3,5-dichlorophenyl)-N-ethyl-2H-tetrazol-5-amine 2,3-bis(ethenyl)-4-phenylpyridine;ethane 2-chloro-N'-(1-cyanopropan-2-yl)pyridine-4-carboximidamide (3-methylimidazo[4,5-b]pyridin-2-yl)-piperidin-1-ylmethanone 5-chloro-6,7,12-triazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(14),3,8(16),9,11,13-hexaen-2-one N-[[5-(3,4-difluorophenyl)-1H-pyrazol-4-yl]methyl]spiro[1,4-dihydroquinoline-3,1'-cyclohexane]-2-imine 6-ethenylsulfonylacridine 3-(1H-indazol-4-yl)pyrazine-2-carbonitrile 4-methylsulfonyl-1H-indole-6,7-dione N-[(2S,3R)-1-cyclobutyl-4,4-difluoro-2-phenylpyrrolidin-3-yl]-4-methoxyoxane-4-carboxamide 1-[2-(3,4-dimethylphenyl)ethynyl]-2-phenylbenzene N-(3,4-difluorophenyl)-1,2-dimethylimidazole-4-sulfonamide (E,2R)-1-[4-[[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]piperidin-1-yl]-2-cyano-3-(3-chloro-5-hydroxyphenyl)prop-3-en-1-one 3-[[4-(2,6-dioxopiperidin-3-yl)piperazin-1-yl]methyl]benzamide (3R)-N-methyl-4-[[1-[2-methyl-5-[[5-(trifluoromethyl)pyridin-2-yl]oxymethyl]phenyl]pyrazol-4-yl]methylamino]pentanamide (2S)-N,3-dihydroxy-2-[[(2R)-4-methyl-1-oxopentan-2-yl]amino]-3-thiophen-2-ylpropanamide (Z)-1-amino-N'-(2,6-dichlorophenyl)-1-phenylmethanimidamide [4-chloro-2,5-bis(phenylmethoxy)phenyl]methanol [3-[(4-chloropyrazol-1-yl)methyl]azetidin-1-yl]-[2-methoxy-5-(trifluoromethoxy)phenyl]methanone 1-[(2,5-dimethylphenyl)methylamino]-3-(4-fluorophenoxy)propan-2-ol 1-[4-amino-5-(3-methoxypropyl)-2,3-dihydroindole-1-carboximidoyl]-3-(3-fluorophenyl)urea N-[(5Z)-5-[amino(benzamidomethyl)carbamoyl]octa-1,5-dien-4-yl]benzamide 2-[(3S)-3-ethylcyclohexyl]acetaldehyde;N-[1-(4-fluorophenyl)ethenyl]methanimine 1-(2,4-dimethylphenyl)-5-hydroxy-N-[(Z)-(3-iodo-5-propan-2-ylidene-1H-pyrrol-2-ylidene)methyl]triazole-4-carboxamide 2-(1,5-dihydropyrazolo[4,3-c]pyridin-3-yl)imidazo[1,2-a]pyrimidine 2-[[7-(4-chlorophenyl)-3-oxoheptyl]-methylamino]acetamide N-[4,5-difluoro-2-(1H-indol-3-yl)phenyl]acetamide N-[3-(ethylamino)-2-methoxyphenyl]propanamide N-[5-(4-fluorophenoxy)pyridin-2-yl]formamide N'-(4-methoxyphenyl)sulfanyl-N,N'-dimethylethane-1,2-diamine N-ethenylsulfonyl-N-(4-phenoxyphenyl)benzenesulfonamide 3-(9H-fluoren-1-yl)pentanedioic acid 7-[(3,5-dichloropyridin-4-yl)methoxy]-N-[2-(dimethylamino)ethyl]quinazolin-4-amine 1-[(2E,4Z)-3-bromohepta-2,4-dienyl]-6-(2-methoxypyridin-4-yl)-2H-pyrimidine [7-chloro-6-(2,6-difluorophenyl)-4H-1,3-benzodioxin-5-yl]hydrazine 4-[(Z)-2-[(Z)-[methyl-[6-(trifluoromethyl)quinazolin-4-yl]hydrazinylidene]methyl]but-1-enyl]benzene-1,3-diol 2-azido-1,3-dichloropyrrolo[3,4-c]pyridine (Z)-3-N,5-dimethyl-4-N-[6-methyl-3-propan-2-yloxy-6-(trifluoromethyl)cyclohexa-1,3-dien-1-yl]hept-3-ene-2,4-diimine 2-[(E)-1,3-diamino-4-azidobut-2-enylidene]-3H-indene-1,3-dione [1-[2,3-dichloro-4-(3-methylcyclohexa-1,5-dien-1-yl)phenyl]ethylideneamino]thiourea 2-[[1-azido-5-methoxy-7-(pyrrolidin-3-ylamino)-9H-fluorene-4-carbonyl]amino]-N,N-diethylacetamide N-(4,6-dimethylpyrimidin-2-yl)-4-[2-nitro-N-(1,3-thiazol-5-yl)anilino]benzenesulfonamide 1-methylsulfanyl-3-[2-(2,4,5-trichlorophenyl)ethylamino]thiourea 2-[3,4-dihydro-1H-isoquinoline-2-carbonyl(1,2,3,6-tetrahydropyridin-4-yl)amino]benzoic acid 2-chloro-4-[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]benzonitrile (2R,4S)-1-[3-(5-chloronaphthalen-2-yl)sulfonylbutanoyl]-N'-hydroxy-4-methoxypyrrolidine-2-carbohydrazide 5-(4,6-difluorocyclohexa-2,4-dien-1-yl)-7-[(4-ethoxyphenyl)methyl]pyrrolo[2,3-d]pyrimidin-2-amine 1-[4-[3,5-bis(trifluoromethyl)phenyl]piperazin-1-yl]butan-2-one (4-chlorophenyl)methanamine;1',3',4',5'-tetrahydroxy-6'-nitrospiro[indene-2,9'-xanthene]-3-one (2S)-3-[5-[3-chloro-4-fluoro-2-methyl-5-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-3-yl]pyrrolidine-1-carboxylic acid 6-azido-1,2,4-trichloronaphthalene 1-[4-amino-3-(methoxyiminomethyl)phenyl]-2-[4-(2,5-difluorophenyl)phenyl]ethane-1,2-dione (NE)-4-chloro-N-[(3,4-dichlorophenyl)methylidene]benzenesulfonamide 4-methyl-2-[(3R)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]-1H-pyrimidin-6-one N-[[4-(1,3-benzothiazol-2-yl)phenyl]methylideneamino]acetamide 1-(azidomethyl)-4-bromopyrrolo[2,3-b]pyridine 1-(2,3,3a,4-tetrahydro-1H-inden-1-yl)-N-[5-fluoro-6-(triazol-2-yl)pyridin-3-yl]pyrazole-3-sulfonamide 3-[[(2S)-3,4-dihydro-2H-chromene-2-carbonyl]amino]-2-hydroxybenzoic acid 1-(4-ethylphenyl)-3,6-difluoro-2-[4-(3,4,5-trifluorophenyl)phenyl]indole 1-[(E)-2-(4-bromophenyl)ethenyl]sulfonyl-6,7-dimethoxyisoquinoline 3-[[6-(3,4-dimethylphenyl)iminocyclohexa-2,4-dien-1-ylidene]amino]butanoic acid 4-[2,3-dihydroxypropyl(hexadecanoyl)amino]benzenesulfonic acid 2,4-dimethyl-3-[(2Z)-1-phenylpenta-2,4-dienoxy]pyridine 4-tert-butyl-N-methylidenebenzenesulfonamide;5-(2,6-difluorophenyl)heptane 2-hydroxy-N'-[4-methoxy-3-(trifluoromethyl)phenyl]cyclopropane-1-carboximidamide [1-(6-aminopyrimidin-4-yl)piperidin-3-yl]-[3-[2-[(4-fluorophenyl)methoxy]ethyl]pyrrolidin-1-yl]methanone 2-chloro-5,6,7,8-tetrahydroacridine-1,4-dione;ethane (4S)-1-(3,5-dimethylphenyl)-3-[hydroxy(phenyl)methylidene]-2-imino-6-iminopiperidin-4-ol 2-[(4S)-2-methyl-1-phenyl-3,4-dihydro-2H-pyridin-5-yl]acetonitrile 2-(6,8-dichloro-4-oxochromen-3-yl)oxy-N-(7-hydroxynaphthalen-1-yl)acetamide 4-[3,3-dimethylbutanoyl(methyl)amino]-N-(2,6-naphthyridin-3-ylmethyl)benzamide N-ethenylsulfonyl-2,4,6-trimethyl-N-(4-nitrophenyl)benzenesulfonamide 6-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(oxan-2-yloxy)ethyl]pyridazin-3-amine 1-(5-butyl-2-methylphenyl)ethanone [3-(2,4-dichlorophenyl)sulfonylimino-5-methylheptan-2-ylidene]azanide 1-[3-(4-methoxyphenyl)propyl]piperidine;dihydrochloride (2R,4R)-N-[cyclopropyl-[3-fluoro-5-(trifluoromethoxy)phenyl]methyl]-1-[3-(2-hydroxyethoxy)benzoyl]-2-methylpiperidine-4-carboxamide N-[(3,4-dichlorophenyl)methyl]-1-ethyltriazole-4-carboxamide 7-hydroxy-N-(1H-indazol-5-yl)quinoline-3-carboxamide (5Z)-2-cyclopentylimino-5-[[3,4-dihydroxy-5-(pyridin-4-ylmethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one 4-(2,6-dimethylphenyl)-3-iodo-5-methoxycarbonylbenzoate N-azido-2,4-dichlorobenzenesulfonamide (2S)-N-[(2R,3S)-1-(3,5-difluorophenyl)-4-hydroxybutan-2-yl]-1-[(4-methoxyphenyl)sulfonylcarbamoylamino]pyrrolidine-2-carboxamide 1,3-bis(5-methylthiophen-2-yl)propane-1,3-dione 2-[5-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-3-[6-oxo-2-(trifluoromethyl)piperidine-3-carbonyl]pyrazin-2-yl]benzamide N-[2-(4-chlorophenyl)ethyl]-2-[4,5-dimethoxy-3-(trifluoromethyl)pyrazol-1-yl]acetamide 2-(3,4-dimethoxyphenyl)-1H-benzimidazole N-[(4S)-1,3-oxazolidin-4-yl]quinoline-6-carboxamide 2-methyl-6,11,12-trioxo-5-propan-2-yl-N-pyridin-3-yl-1,8,12,15-tetrazatetracyclo[7.6.0.02,7.010,14]pentadeca-9,13-diene-4-carboxamide (2-azido-4,5-difluorophenyl)-pyrrolidin-1-ylmethanone (1S,3R)-2,2-dimethyl-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethyl)-3-(2,2,2-trifluoroethoxy)cyclobutane-1-carboxamide;formic acid N-[[5-fluoro-2,3-bis(phenylmethoxy)phenyl]methyl]butanamide N-(4-nitrophenyl)-6,8-dihydro-5H-[1]benzothiolo[2,3-d]pyrimidin-7-amine 2-azido-7-chloro-5,6-diethoxy-3H-quinazolin-4-one 2-methoxy-5-[[4-(trifluoromethyl)pyridin-3-yl]methylidene]cyclohepta-1,6-dien-3-yne 2-cyclopropyl-N'-hydroxy-6-methoxypyrimidine-4-carboximidamide 3,6-ditert-butyl-1H-quinolin-4-one 1-[(E)-3,5-dimethylhex-2-en-2-yl]sulfanyl-4-phenylbenzene 5-azidooxy-N'-(6-chloropyridine-3-carbonyl)-2,4-difluorobenzohydrazide 2-[N-(1,3-thiazol-5-yl)anilino]acetonitrile 1-methyl-4-[(2E,5Z)-4-pentan-3-ylhepta-2,5-dien-3-yl]sulfanylbenzene N-[2,4-difluoro-3-(3-hydroxybutylsulfamoyl)phenyl]-3,4-dimethoxybenzamide 4-(methylamino)-2-[6-(1,3-thiazol-5-ylamino)pyridin-2-yl]-8H-pyrido[2,3-d]pyrimidin-7-one 6-bromo-2,3-dimethylbenzo[h]quinoline N-[4-(1-adamantyl)phenyl]-3,6-dihydroxy-2H-naphthalene-1-carboxamide N-(cyclohexylmethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 2,6-dibromo-3-[(1E)-1-(4-hydroxy-5-methoxycarbonylfuran-2-yl)buta-1,3-dien-2-yl]-5-propanoyloxybenzoic acid 1-[(2S)-4-[5-fluoro-6-[(4,4,7,7-tetramethyl-1,3,5-trioxonan-2-yl)amino]pyridin-3-yl]-2-propan-2-ylpiperazin-1-yl]ethanone 2-[4-(6,7-difluoroquinoxalin-2-yl)piperazine-1-carbonyl]pyrrolidine-3-carbonitrile 1-amino-N-[(1R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]cyclopropane-1-carboxamide 3-chloro-1-methyl-5-(4-pentoxyphenyl)pyrazole N-[[5-(difluoromethyl)-1,2,4-oxadiazol-3-yl]methyl]benzenesulfonamide 2,3-dichloro-5-[(6-oxo-4-propyl-1H-pyrimidin-2-yl)amino]benzonitrile 1-[(3S,4R)-1-methyl-4-(5-phenyltetrazol-2-yl)pyrrolidin-3-yl]-N-(pyridin-2-ylmethyl)methanamine 1-[2-(3,4-difluorophenyl)ethyl]-6-methoxy-7-propan-2-yloxyquinolin-2-one;hydrochloride 5-[8-(diethylamino)-2,3-dihydro-1H-imidazo[1,2-a]pyridin-4-ium-6-yl]-7-fluoro-N-(4-morpholin-4-ylphenyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide 5-methyl-6-(2,3,5-tribromophenyl)pyridine-2-carbonitrile N-[(4Z,5E)-2,3-dimethyl-1-phenyl-6-propan-2-ylidenenona-2,5,7-trien-4-yl]-4-ethenylaniline 3-[2,4,6-tris(4-methoxyphenyl)phenyl]propanamide 4-[2,5-dimethoxy-3-(pyridin-2-ylsulfinylamino)phenyl]piperidine-1-carboxylic acid 1-[3-fluoro-4-(3-methyl-4,5-dihydrobenzo[e]indol-2-yl)phenyl]pentan-2-one 1-[(2S)-4,6-dioxo-4-phenylpiperidine-2-carbonyl]piperidine-3-carboxylic acid 1-[4,6-bis(2H-triazol-4-yl)pyrimidin-5-yl]propan-2-one 4-(5-benzyl-1,3,4-oxadiazol-2-yl)-N-[4-cyano-2-methoxy-6-(pyrazol-1-ylmethyl)phenyl]piperidine-1-carboxamide N-[(1R,2S)-2-hydroxycyclohexyl]-7-methoxy-6-[3-[1-(oxetan-3-yl)piperidin-4-yl]propoxy]quinoline-5-carboxamide 3-(1-methylcyclopropyl)-N-[1-(5-pyridin-3-yl-1,2-dihydrotriazol-2-ium-3-yl)ethyl]quinoxalin-6-amine 5-[(3,4-dimethylphenyl)sulfonylamino]-2-[methyl-(1-propan-2-ylpiperidin-4-yl)amino]pyridine-3-carboxylic acid;2,2,2-trifluoroacetic acid 2-[4-chloro-5-(cyclopropylsulfonylamino)pyridin-2-yl]-N-methoxy-N,2-dimethylpropanamide 5-[(4R,10bS)-8,9-dimethoxy-3,4,6,10b-tetrahydro-1H-pyrazino[2,1-a]isoindole-2-carbonyl]thiophene-2-carboxylic acid 4-[5-bromo-1-(3,5-dichlorophenyl)sulfinylpyrrolo[2,3-b]pyridin-2-yl]morpholine (2S)-1-[(3R,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]piperidine-2-carboxylic acid N-(2,4-difluorophenyl)-5,6-dimethylpyridine-3-carboxamide 2-cyclohexylsulfanyl-4,6-dinitrophenol 2-[5-cyano-6-hydroxy-1-[(3-methylphenyl)methyl]-4-oxo-2,3-dihydroquinolin-7-yl]acetic acid 2-[4-(1-hydroxycyclohexyl)phenyl]acetic acid 2-[(2Z)-3,7-dimethylocta-2,6-dienoxy]-4-pentylnaphthalene 2-[(3,4-diethoxyphenyl)methyl]-8-ethylsulfonyl-1H-pyrrolo[2,3-e]benzimidazole 1-[7-(3,5-difluorophenyl)-3,4-dihydro-2H-chromen-4-yl]-N-methylsulfonylpiperidine-4-carboxamide 1-[(1Z,3E)-2,6-dimethylhepta-1,3-dienyl]-4-hydroxy-5-methoxypyridin-2-one 2,4-difluoro-1-methylbenzene;N-(2-oxoazetidin-3-yl)-5-(trifluoromethyl)pyridine-2-carboxamide (Z)-3-amino-N'-[4-[4,5-bis(ethoxymethyl)-1,2-oxazol-3-yl]phenyl]but-2-enimidamide 2-bromo-1H-benzo[f]chromene 1-(2,3-dihydro-[1]benzofuro[3,2-d]pyrimidin-4-yl)piperidin-3-ol 5-(4-azidophenyl)-2H-tetrazol-1-ium 2-[4-[(E)-3-oxo-3-phenylprop-1-enyl]pyridin-1-ium-1-yl]acetic acid 1,3-difluoro-5-(4-methylcyclohexen-1-yl)benzene N'-[2,6-dimethyl-4-[(E)-1-[[5-methylidenecyclohexa-1,3-dien-1-yl(phenyl)methylidene]amino]prop-1-en-2-yloxy]phenyl]-N-ethyl-N-methylmethanimidamide 2-(2,6-dioxopiperidin-3-yl)-5-[4-(piperidine-1-carbonyl)piperazin-1-yl]isoindole-1,3-dione 4-ethyl-1-[1,1,1-trifluoro-4-methoxy-3-(5-nitrothiophen-2-yl)butan-2-ylidene]piperazine 2-(2-methylpropyl)-4-[[5-(2-methylphenyl)sulfanylthiophen-2-yl]methylideneamino]phenol 5-bromo-4-chloro-N,N-bis(propan-2-ylsulfanyl)pyrimidin-2-amine 4-chloro-N'-methylbenzenecarboximidamide;6-[6-(2,3-dihydro-1H-inden-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]hexan-1-ol N-(3,4-dimethoxyphenyl)-6-hydroxy-N'-[(1E)-2-methylbuta-1,3-dienyl]heptanediamide 2-(3,4-dichlorophenyl)-1-[4-(dimethylamino)-2-fluorophenyl]ethanone;ethane 4-[[2,5-diamino-6-(quinoline-3-carbonyl)pyrimidin-4-yl]amino]benzaldehyde;ethane [4-(5,6-dichloro-3H-indole-2-carbonyl)piperazin-1-yl]-[2-methoxy-4-(propan-2-ylamino)phenyl]methanone 4-[3-(4,6-diphenylpyridin-2-yl)phenyl]benzonitrile 4-[5,5-dimethyl-3-(2-oxopropanoylamino)hexanimidoyl]benzoic acid 5-chloro-2-methylimidazo[1,2-a]pyridine-7-sulfonamide;ethane 2-benzamido-3-[4-(1H-indol-6-yl)phenyl]propanoic acid N-[4,5-dimethyl-2-(3,4,5-trifluorophenyl)pyrazol-3-yl]formamide;2-(ethoxymethyl)pyridine 1-butyl-2-phenylbenzimidazole;ethane N-cyclohexyl-3,5-dihydro-2H-1,4-benzoxazepine-7-sulfonamide 2-[6-(1H-indazole-3-carbonylamino)spiro[3.3]heptan-2-yl]oxypyridine-4-carboxamide (5Z)-5-[[3,6-dichloro-4-[(2E)-2-hydroxyiminobutanoyl]oxypyridin-1-ium-1-yl]methylidene]-4-ethyl-2,2-diphenylfuran-3-carboxylic acid (2S)-2-[(2-bromobenzoyl)amino]-3-hydroxypropanoic acid N-[6,8-bis(4-methoxyphenyl)pyrido[3,2-d]pyrimidin-4-yl]cyclopropanecarboxamide (3-cyclopropylmorpholin-4-yl)-[2-methoxy-5-(1,2-oxazol-3-yl)phenyl]methanone 3-(2,6-dichlorophenyl)-7-[4-[2-hydroxyethyl(methyl)amino]anilino]-2H-pyrimido[5,4-e][1,3]oxazin-4-one 2-[3-oxo-5,6-bis(4-phenylphenyl)-1H-isoindol-2-yl]acetamide 2-[3-(1,3-dioxolan-2-yl)prop-2-enoyl]benzoic acid 4-[2-oxopropyl(octyl)amino]benzenesulfonic acid N-[4-(aminomethyl)phenyl]sulfonylbenzamide N-[5-(diethoxyphosphorylmethylamino)naphthalen-1-yl]hydroxylamine 2-[2-(1,3-dioxolan-2-yl)ethoxy]-8-nitronaphthalene 2-[(E)-[1-methyl-5,6-dihydroisoquinolin-3-yl]methylideneamino]oxyacetic acid 2-(2,3-dihydro-1H-inden-5-yl)-N-[(E)-1H-indol-3-ylmethylideneamino]acetamide 2-(N-butyl-4-methoxycarbonylanilino)octanoic acid [(4S,7R)-2-phenylmethoxycarbonyl-5-oxa-8-azaspiro[3.5]nonan-8-yl]boronic acid 6-[(2S)-butan-2-yl]oxy-N-(5,6-dihydro-4H-cyclopenta[d][1,3]thiazol-2-ylmethyl)pyrazine-2-carboxamide 2-(3,5-dimethylpyridin-4-yl)acetamide 2-methyl-4-[3-[(6-oxo-5H-benzo[b][1,4]benzoxazepine-3-carbonyl)amino]phenoxy]butanoic acid N-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-(4-fluorophenyl)-2-oxopyrrolidine-3-carboxamide 4-[2-azido-5-(3,4-dichlorophenoxy)pentyl]morpholine 1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]phenyl]propan-1-one 4-[(5S)-3-cyclopropyl-8-methoxy-1-methylidene-2,6,7,9-tetrahydroquinolizin-5-ium-4-yl]phenol 2-[5,6-diamino-2-(2,4-dicyanophenoxy)pyrimidin-4-yl]oxyacetamide [6-(5-methylsulfonylcyclohexa-1,3-dien-1-yl)-3-(3H-pyrrole-2-carboximidoyl)pyridin-2-yl]urea 4-chloro-2-[(3S)-1-[(E,6R)-6-(4-chlorophenyl)hept-5-enyl]pyrrolidin-3-yl]oxypyridine N-(5-chloro-1H-indazol-3-yl)-2-[4-(4-ethoxyphenyl)piperazin-1-yl]acetamide 4-(6-bromonaphthalen-2-yl)-N,2,5-trimethylaniline 4-cyclopropyloxy-N-[(1R)-2,3-dihydro-1H-inden-1-yl]pyridine-2-carboxamide [(2-aminopyridine-3-carbonyl)amino]carbamodithioic acid N-benzyl-1-[4-hydroxy-3,5-bis(hydroxymethoxy)phenyl]-6-oxo-2-phenylpiperidine-3-carboxamide 4-[5-ethylsulfonyl-6-[8-oxo-2,7-di(propan-2-yl)-1H-pyrido[2,3-d]pyrimidin-4-yl]pyridin-3-yl]benzonitrile N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]-2,5-dimethylthiophene-3-sulfonamide N-(4,5-dichloro-2-hydroxyphenyl)-3-methylimidazo[1,2-b]pyridazine-6-carboxamide 4-amino-2-[(4-ethylphenyl)methoxy]-5-iodo-1H-pyrimidin-6-one 1-[3-methyl-5-[(2R,6S)-2,4,6-trimethylpiperazine-1-carbonyl]pyridin-2-yl]pyrazolo[3,4-d]pyrimidine-4-carbonitrile (2R)-1-[(2S,3aS,6aR)-2-ethyl-2,3,3a,4,5,6,7,8,8a-octahydroindole-1-carbonyl]-N-(1H-indazol-6-ylmethyl)pyrrolidine-2-carboxamide;hydrochloride 5-chloro-4-[4-(3,6-dihydro-2H-pyran-4-yl)phenyl]-N-phenylpyrimidin-2-amine N-[3,5-bis(trifluoromethyl)phenyl]-4-nitrobenzenesulfonamide 4-[2-(4-methoxyphenyl)-3-(5,6,7,8-tetrahydronaphthalen-1-yl)propanoyl]-5,6,7,8-tetrahydroquinoline-2-sulfonamide N-[4,6-dichloro-1-(3,4-dimethylphenyl)sulfonyl-2-oxoquinolin-5-yl]acetamide 3-[(2,4-dichlorophenyl)methyl]-6-(4-hydroxyphenyl)-2H-1,3-benzothiazole-2,5-diol (5Z)-2-(2,3-dichlorophenyl)imino-5-[(4-hydroxy-3-nitrophenyl)methylidene]-1,3-thiazolidin-4-one 1-cyclopenta[b]pyran-6-ylpyrrolidine-3-carboxylic acid 1,3-dicyclohexyl-1-methoxynaphthalen-2-one 2-(4,5-dimethyl-1H-imidazol-2-yl)-6-propan-2-ylidenecyclohexa-2,4-dien-1-one 1-(3,4-dimethoxyphenyl)sulfonyl-3-[2-fluoro-5-[3-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]piperazin-1-yl]pyridin-3-yl]urea N'-hydroxy-4-[(1,2,3,4-tetrahydroisoquinolin-8-ylmethylamino)methyl]pyridine-2-carboximidamide 1-[4-(2,6-dimethylphenoxy)phenyl]butan-1-one;N-methylpentanamide 1-[5-ethenyl-4-(1-pyridin-2-ylazetidine-3-carbonyl)-1,3-thiazol-2-yl]piperidine-4-carboxylic acid N-[5-[3-(4-pyridin-2-yl-1H-pyrrolo[2,3-b]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclopentanecarboxamide (2-chlorophenyl)methyl-dimethylazanium;chloride ethane;4-methylmorpholine;2,3,5,6-tetrafluoro-4-[(2-fluoro-1H-inden-5-yl)oxy]aniline 2-(3,4-dimethoxyphenyl)-2-hydroxybutanoic acid 1-[(2S)-2-aminopropanoyl]-N-[(3R,4S)-3-hydroxypiperidin-4-yl]-9H-carbazole-2-carboxamide;hydrochloride 1-[(2R,4R)-4-fluoro-5-nitro-3,6-bis(phenylmethoxy)oxan-2-yl]-N-propan-2-ylmethanamine N-[2-(1,3-benzothiazol-6-ylamino)-5H-pyrrolo[3,2-d]pyrimidin-4-yl]-N',3-dimethylazetidine-1-carboximidamide N-[2,6-difluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-2,4-dimethoxybenzamide 2-amino-6,7-dihydrobenzo[d][1]benzazepine-3-carboxamide 2-[7-methoxy-5,6-dimethyl-1-(4-methylphenyl)sulfonylindol-3-yl]-N-[2-oxo-2-(3-phenylpropanoylamino)ethyl]acetamide 5-bromo-2-(2,2-dimethylpropylamino)pyrimidine-4-carbonitrile 2-[3-[3-(4-methoxycarbonylpiperidin-1-yl)propanoylamino]-3,6-dihydro-2H-pyridin-1-yl]-N-phenylquinoline-8-carboxamide 7-(3-chloro-4-hydroxyphenyl)-6-fluoro-1-[2-hydroxy-2,2-dimethyl-4-(phenoxyamino)butanoyl]-8aH-naphthalene-2-carboxylic acid 1-[2-cyclopropylethoxy(phenyl)methyl]piperidine 6-[2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]ethynyl]-1-fluoro-2-pentan-2-ylnaphthalene 4-(2,1,3-benzoxadiazole-6-carbonyl)-5-methyl-3-phenyl-1H-imidazol-2-one 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]benzo[g][1,3]benzothiazole N-azido-N-(diphenylphosphorylamino)-1-pyridin-2-ylethanamine 2-(2-azidooxyethyl)-7-ethynyl-5,8-dimethoxy-[1,2,4]triazolo[1,5-c]quinazoline 1-(1-azabicyclo[2.2.2]octan-3-yl)ethanone;6,7-difluoro-4-methoxyquinazoline N-[(2R)-2,3-dihydroxypropyl]-6-methyl-N'-[1-methyl-5-[(E)-4-oxobut-2-enoyl]benzimidazol-2-yl]pyridine-3-carbohydrazide;methane 5-fluoro-1,2-dimethylbenzo[e]indole;(3Z)-hexa-1,3,5-triene 4-tert-butyl-2-(2,6-dimethylphenyl)pyridine 4-azido-1,7-ditert-butylquinazolin-2-one (E)-2,3-difluorobut-2-ene;3-methylbuta-1,3-dien-2-ol;(Z)-N'-[5-oxo-4-[6-oxo-1-[4-(trifluoromethoxy)phenyl]pyridazin-3-yl]-1,3-thiazol-2-yl]prop-1-ene-1,3-diamine 4-[(2,6-dimethylmorpholin-4-yl)methoxy]-3-fluoro-N'-hydroxybenzenecarboximidamide 1-[2,3-bis(phenylmethoxy)phenyl]propane-1,2,2-triamine N-[4-(8,9,10,11-tetrahydrobenzo[b][1]benzazepin-5-yl)butyl]-6-thiophen-2-ylhexanamide N-[4-[2-(3,4,5-trimethoxyphenyl)ethenyl]-1H-pyrazol-5-yl]furan-2-carboxamide 1-(5,6-dimethoxy-3a,4-dihydroindeno[2,1-b]furan-9b-yl)-N-methylethanimine ethane;1-[(3E)-hexa-1,3,5-trien-3-yl]-N-methoxy-2-pyridin-4-ylethanimine N-[[1,4-dimethyl-2-(5-methylthiophen-2-yl)pyrrolo[3,2-c]pyridin-7-yl]methylideneamino]acetamide (2S)-3-cyclobutyloxy-1-[4-[6-methoxy-7-(3,3,3-trifluoropropoxy)quinolin-4-yl]oxypiperidin-1-yl]propan-2-ol 5-chloro-2-[5-(cyclopropylmethoxy)pyridin-3-yl]-N-[(1R,6S)-3-propan-2-ylbicyclo[4.2.0]octa-2,4-dienyl]pyrimidine-4-carboxamide N-(2,4-dihydroxyphenyl)-3-[2-hydroxy-5-(2-methylpropanoylamino)phenyl]-1H-pyrazole-5-carboxamide 2-[(4-azidophenyl)methyl]pyrimidine 3-methyl-1,2,8-triphenylquinoline 5-[[5-(1H-indol-3-yl)-4-[[2-methoxyethyl(methyl)amino]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2,2,8,8-tetramethyloctanoic acid 5-ethyl-2-[1-(4-methoxyphenyl)-1H-inden-5-yl]-N,N-dimethylpyridine-3-carboxamide N-[3-(3,4-dihydropyridin-6-yl)phenyl]-N'-[7-(3-hydroxyazetidine-1-carbonyl)pyrido[2,3-d]pyrimidin-4-yl]-N'-methylpropanehydrazide 2-chloro-3-[4,5-dimethyl-6-oxo-1-(pyrimidin-4-ylmethyl)pyridazin-3-yl]benzonitrile;ethane 1-[(4-chlorophenyl)methyl]-5-methylidenetriazolo[4,5-d]pyrimidine N-[(Z)-3-aminoprop-2-enimidoyl]-4-(azetidine-1-carbonyl)benzamide 3-(6-methylpyridin-2-yl)oxy-1-[2,3,5,6-tetradeuterio-4-hydroxy-7-(trifluoromethyl)indol-1-yl]propan-1-one 2,3-diamino-4,5-bis(methylsulfonyl)benzenesulfonic acid 4-[(3-chloro-4,5-dimethoxyphenyl)methyl]quinazoline (5S)-N-(4-chlorophenyl)-2-[(3R,6S)-6-methylpiperidin-3-yl]imino-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide N-[2,5-difluoro-4-(1H-indol-3-yl)phenyl]acetamide 3-[(2Z,4E)-5-amino-6,7-dimethylocta-2,4-dien-4-yl]oxy-N-(1,2-oxazol-4-yl)pyridine-2-carboxamide 4-[3-[4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)phenyl]propylamino]quinazoline-2-carbonitrile 3-azidooxy-2-methylquinoline (3E,5Z)-7-[6-(dipropylamino)hexoxy]octa-1,3,5,7-tetraen-4-amine;ethane;5-fluoro-2-(2-methoxyphenyl)phenol [2-ethylsulfanyl-6-methoxy-5-(trifluoromethyl)pyrimidin-4-yl]-(3-fluoropyridin-2-yl)carbamic acid N-methyl-2-(7,8,10,11-tetrazatricyclo[7.4.0.02,6]trideca-1,3,5,8,10,12-hexaen-13-yl)ethanamine 3-methyl-N-[2-(4-pyridin-3-yloxyphenyl)ethynyl]benzamide ethane;2-methyl-4-(3-phenylthiophen-2-yl)butan-1-amine 4-[(3Z)-3-[2,5-dimethyl-4-oxo-6-(trifluoromethyl)chromen-7-ylidene]propoxy]benzoic acid 3-methyl-N'-(2,5,6-trichloropyridine-4-carbonyl)benzohydrazide 3-(1,4-dimethoxybutan-2-yl)-6-ethyl-7-fluoro-1H-quinazoline-2,4-dione (2S,4R)-5-[(3,4-dichlorophenyl)methyl]-2-(1H-imidazol-2-yl)-4-propanoyloxy-6-(trifluoromethyl)heptanoic acid N-[3-(dimethylamino)propyl]-2-methoxy-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-4-carboxamide 1-[(4aS,8aR)-3a-(hydroxymethyl)-5-methylidene-2-[[1-(oxolan-3-yl)pyrazol-4-yl]methyl]-4,4a,6,7,8-pentahydroquinazolin-4-yl]ethanone 4-amino-5-(2,6-dimethoxyphenyl)iminopenta-1,3-dienylazanium 2,4-dichloro-N-(2,6-diethylphenyl)benzenesulfonamide 2-N-[(2R)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]-5-fluoropyrimidine-2,4-diamine 3-[2-methoxy-4-(trifluoromethyl)phenoxy]-5-(3-phenylcyclobutyl)-1,2,4-oxadiazole 5-[4-(aminomethyl)phenyl]-1H-pyrimidine-2,4-dione 4-[2-(4-iodophenyl)pyrazol-3-yl]phenol 5-(azidomethyl)-4-chloropyridine-2-carbonitrile 4-N,6-N-bis(2-ethoxyphenyl)pyrimido[5,4-b]indole-3,6-diamine 2-[3-(dimethylamino)propylimino]-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one 1,2-dichloro-N-[(2S)-3-cyclohexylpropan-2-yl]benzimidazole-5-carboxamide 2-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]-4-dodecan-8-ylbenzenethiol 2-[(3,4-dichlorophenyl)methyl]propanedioate N-(4,5-dimethylthiophen-2-yl)sulfonylthiophene-3-sulfonamide 3-[1-(benzylamino)ethenyl]pyridine-2,6-dicarboxylic acid 5-(4-methylphenyl)-2,3-bis(2-morpholin-4-ylethoxy)benzoic acid N-[(E)-3-[(4-chlorophenyl)methyl]pent-2-enyl]aniline N-[5-methyl-2-(4-oxo-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-3-yl)pyrazol-3-yl]quinoxaline-5-carboxamide 1-chloro-3,5-bis(2,6-diethylphenyl)cyclohexa-1,3-diene 4-[2-(2,3-dihydroxypropoxy)phenyl]benzamide 3-azido-2-butyl-5,6-dimethoxy-1H-indole (3S)-4-amino-2,2-bis(methoxycarbonyl)-5-phenylpentanoic acid 7-(3,5-dimethylphenyl)-N-[4-[methyl(1-propan-2-ylpiperidin-4-yl)amino]cyclohexyl]pyrrolo[2,3-d]pyrimidin-2-amine 6-[2-(3,5-dimethylphenyl)pyridin-1-ium-4-yl]-2-methyl-7H-[1]benzofuro[2,3-b]pyridin-7-ide;iridium;trimethyl-[4-(1-methylpyridin-1-ium-2-yl)-6-phenylpyridin-3-yl]silane (E)-2-cyano-3-[4-(1,5-diphenylpentan-3-yloxy)phenyl]prop-2-enoic acid N-[(5-tert-butyl-1,3,4-thiadiazol-2-yl)sulfonyl]spiro[2H-indole-3,4'-oxane]-6-carboxamide N-methyl-1-[[3-(trifluoromethoxy)phenyl]methylideneamino]piperidine-4-carboxamide 4-bromo-2,6-difluoro-N-(furan-2-ylmethyl)benzenesulfonamide 2-(5-methyl-1,3,4-thiadiazol-2-yl)-N-[6-[(2S)-5-oxopyrrolidine-2-carbonyl]-7,8-dihydro-5H-1,6-naphthyridin-3-yl]acetamide 2-[(Z)-1-aminoethenyl]-3H-isoindol-1-imine;N-[4-methyl-3-(methylamino)phenyl]acetamide N-cyclopropylformamide;ethane;2-methoxy-4,6-dinitrophenol 3-(2,6-dimethylphenoxy)-N'-hydroxypyrazine-2-carboximidamide 3-[2-(4-chlorophenyl)ethenyl]-N'-hydroxypyridine-2-carboximidamide 5-(5-bromopyridin-3-yl)-4-methylideneimidazolidin-2-one (2R,4S)-N-[6-cyano-5-(4-methoxyphenyl)pyrazin-2-yl]-2-hydroxy-4-phenylpyrrolidine-1-carboxamide 5-[2,4-dihydroxy-3,6-bis(3-methylbut-1-en-2-yl)phenyl]benzene-1,2,3-triol 1-(2-pyridin-4-ylethoxy)propan-1-ol 5-[(2E)-6-ethylhepta-2,4,6-trien-3-yl]-N-(4-pyridin-3-ylpyrimidin-2-yl)-1H-indazole-3-carboxamide [4-methyl-1-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)azepan-4-yl]methanamine 4-[[6,7-dimethoxy-3-(2-morpholin-4-ylethoxy)quinolin-4-yl]amino]-N'-propan-2-ylbenzenecarboximidamide 2-[3-(2,4-difluorophenoxy)azetidine-1-carbonyl]-N-propan-2-ylbenzenesulfonamide ethane;N-[1-(3-fluorophenyl)propyl]butanamide 1,3-dichlorobenzene;N-(6-phenylpyridin-2-yl)-5-pyridin-4-ylsulfonyl-1H-pyrrole-2-carboxamide 1-(cyclohexylamino)-3,6,7-trimethyl-5H-pyrimido[5,4-c]carbazole-2,4-dione N-(3,4-dimethoxyphenyl)-2,6-dimethylpyridine-3-carboxamide 1-[(3,4-difluorophenyl)methyl]-5-[3-(dimethylamino)-5,6,7,8-tetrahydro-2H-quinoline-1-carbonyl]-N-pyridin-3-ylpyrazolo[4,3-d]pyrimidine-7-carboxamide (3E)-1-(cyclopropylmethyl)-3-ethylidene-6-[(Z)-prop-1-enyl]-2,5-dihydroindole (2S)-N-[(3R)-1,1-bis(2-fluorophenyl)-4-methylpyrrolidin-3-ylidene]piperidine-2-carboxamide (5R)-4,5-dibenzyl-1-hydroxyimidazolidin-2-one 1-[(E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]piperidine-3-carboxylic acid 2-[[(3R)-1-benzylpyrrolidin-3-yl]methyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine;dihydrochloride (5Z)-5-[[4-[3-chloro-4-(2-methylphenyl)sulfanylanilino]quinazolin-6-yl]methylidene]-1,3-thiazolidine-2,4-dione N-(4-azidophenyl)-6-chloro-1H-benzimidazole-2-carboxamide N-[(2S)-1-amino-1-oxopropan-2-yl]-5,6-dimethoxy-N'-(1,3-thiazol-2-yl)spiro[2H-indole-3,4'-oxane]-1-carboximidamide 3-[2,3-difluoro-4-[4-(4-propylphenyl)cyclohexyl]phenyl]-6-pentylpyridazine 1-[4-(azidomethyl)phenyl]benzimidazole 4-[[3,5-bis(trifluoromethyl)phenyl]methoxymethyl]-N-[(2S)-1-hydroxypropan-2-yl]pyridine-2-carboxamide 4-[[(Z)-3-amino-2-methylprop-1-enyl]-ethylamino]-N,3,5-trimethoxybenzamide 4-ethyl-N'-hydroxy-1H-imidazo[4,5-b]pyridine-6-carboximidamide 3-[1-methoxy-4-[2-(4-methylpiperazin-1-yl)pyridin-4-yl]pyrazolo[4,3-c]pyridin-6-yl]propanal 5-[(3S)-2,4,7-trioxo-1-phenyl-5,6-dihydroheptan-3-yl]thiophene-2-carboxylic acid 2-[[3-(azidomethyl)pyrrolidin-1-yl]methyl]quinoxaline 2-[4-(3,4,6,7,8,9,10,11,12b-octahydro-1H-pyrazino[2,1-d][2]benzazocine-5-carbonyl)-2-fluorophenyl]isoindole-1,3-dione N-(3,4-dimethylphenyl)-2-fluoro-6-iodoaniline N-[4-(9H-fluoren-1-ylsulfonyl)phenyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide 1-azido-2,3-dimethoxy-5-propylbenzene 2-[(3R)-3,4-dihydroxypyrrolidin-1-yl]-N'-(4-fluorophenyl)-6,7-dihydrothieno[3,2-d]pyrimidine-4-carbohydrazide 1-(3-azidophenyl)-2-cyclopropyl-N,N-dimethoxyethanamine 3-(2,6-difluorophenyl)-5-[4-(dimethylamino)phenyl]-7-(3,4-dimethoxycyclobutyl)pyrrolo[2,3-b]pyrazine-2-carboxamide 2-(5,6-dimethylimidazo[1,2-a]pyrazin-8-yl)butanoic acid 2-[3,4-bis(phenylmethoxy)phenyl]propanoic acid 1-[(2,6-difluorophenyl)methyl]-N,3-diethylimidazolidine-2-carboxamide N-[4-(benzylcarbamoylamino)but-1-en-2-yl]formamide 3-[[2,6-dichloro-4-(trifluoromethyl)phenyl]methoxy]pyridine 3-[1-(4-methoxyphenyl)cyclopropyl]-5-(2-phenoxyphenyl)-1,2,4-oxadiazole 1-N,4-dimethylbenzene-1,2-diamine;4-ethynoxybenzenesulfinic acid 3-(4,5-dimethylthiophene-2-carbonyl)morpholine-4-carboxylate 4-[3-methylbutyl(phenacyl)amino]benzenesulfonic acid 4-(5-benzyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl)-7H-pyrrolo[2,3-d]pyrimidine (2E)-1-(furan-2-yl)-2-[(Z)-2-hydroxy-2,3-dihydroinden-1-ylidene]ethanone 1-[4-methyl-5-(2H-tetrazol-5-yl)thiophen-3-yl]pyrrole (2S)-1-[3,4-bis(phenylmethoxycarbonylamino)benzoyl]azetidine-2-carboxylic acid 5-bromo-4-cyclopropyl-1-[(2,4,6-trifluorophenyl)methyl]pyridin-2-one N-(6-methoxycyclohexa-1,5-dien-3-yn-1-yl)-4-[2-(pyridin-2-ylamino)ethoxy]benzamide 4-[2,3-bis(methoxycarbonyl)naphthalene-1-carbothioyl]benzoic acid (2-amino-5,6-dimethylpyrimidin-4-yl)-(oxan-3-ylmethoxy)methanesulfonic acid 2-[3,5-dimethyl-1-(4-methylpyridin-2-yl)pyrazol-4-yl]-1H-benzimidazole 3-[1-(2-methoxyethyl)imidazol-4-yl]-5-(trifluoromethyl)pyridine 5-[(Z)-2-chloro-3-fluoroprop-1-enyl]-N',3,4-trimethylpyridine-2-carboximidamide 1-(2,6-dimethylphenyl)-3-[(Z)-4-hydroxy-2,3-dihydropyrano[3,2-c]chromen-4-ylidene]thiourea 1,3-dimethyl-N-(4-propanoylphenyl)sulfonylpyrazolo[4,3-b]pyridine-6-carboxamide 1-(2,4-dimethoxyphenyl)-N'-hydroxycyclopentane-1-carboximidamide (4S,5R)-5-[[(2Z)-2-hydrazinylideneethoxy]methyl]-1-methyl-3-(2-phenylethyl)imidazolidine-2-thione 4-[2-(2,5-dihydroxy-3,6-dimethylphenyl)cyclopropyl]-2-(4-methoxyphenyl)phenol 6-[[(1S,2R)-3-methylsulfonyloxycyclohexanecarbonyl]amino]quinoline-4-carboxylic acid 4-chloro-1-ethyl-5-[2-methoxy-6-(2,2,3,3-tetrafluoropropoxy)pyridin-3-yl]-N-[(4-methylsulfonylcyclohexylidene)methyl]pyrazole-3-carboxamide 7-[[1-(cyclopentylmethyl)triazol-4-yl]methoxy]-N,2-diethylimidazo[1,2-a]pyridine-3-carboxamide 5-bromo-3-(2,6-dimethoxyphenyl)triazolo[4,5-b]pyrazine 1-(4-methoxyphenyl)-2,3-dihydroindole N-cyclohexyl-2-[5-[(3,4-dimethoxyphenyl)carbamoyl]thiophen-2-yl]-1H-benzimidazole-4-carboxamide (2-benzylpyrazol-3-yl)-[4-[(2-methoxyphenyl)methyl]piperazin-1-yl]methanone;hydrochloride N-[3,5-bis(trifluoromethyl)phenyl]-1-methoxymethanimidate 1-[(3R)-piperidin-3-yl]pyrazolo[3,4-b]pyridine-6-carboxamide 4-[3-(1,3-benzothiazol-2-yl)phenyl]butanamide 2-(3,5-difluorophenyl)-4-[4-hydroxy-1-[1-(1H-pyrazole-4-carbonyl)azetidin-3-yl]piperidin-4-yl]benzonitrile 7-benzyl-2-[4-(trifluoromethoxy)phenyl]-1,8-dihydroimidazo[4,5-g]quinazoline 4-tert-butyl-N-[(3S)-1-methylpyrrolidin-3-yl]benzamide (3aR,7aS)-2-[[2-methoxy-6-(trifluoromethyl)pyridine-4-carbonyl]amino]-5-(oxan-4-ylmethylcarbamoyl)-1,3,4,6,7,7a-hexahydropyrrolo[3,4-c]pyridine-3a-carboxylic acid 1-[2,4-bis(ethenyl)phenyl]-N,2-dimethoxyethanimine 4-hydroxy-5-[(1Z)-1-indol-3-ylideneethyl]-3H-1,3-thiazol-2-one 3-[1,2-di(ethylamino)ethenyl]-5-methanimidoylphenol 4-[(5E)-5-(2,3-dihydro-1H-inden-2-yloxymethylidene)furan-2-yl]sulfonylbenzonitrile 5-[(E)-4,4-dimethylpent-2-enoyl]-N-methylpyridine-3-carboxamide;ethane (1R,2S)-N-[3-(5-methylfuran-2-yl)propyl]-2-phenylcyclopentan-1-amine 3-(4-azidophenyl)-N,N-dimethylpropanamide 5-[(1R)-3,3,7-trimethyloctoxy]naphthalene-2-carboxylic acid 4-[[1-(cyclohexylmethyl)piperidin-3-yl]amino]pyrimidine-5-carbonitrile (3-fluorophenyl)-[4-[6-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]pyrimidin-2-yl]azanium N-(4,5-dihydrooxepin-2-ylmethyl)-6-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrazin-8-amine 7-[4-(6-methoxypyridin-2-yl)piperazine-1-carbonyl]imidazo[1,2-a]pyrimidine-5-carboxamide (3R)-3-[2,6-difluoro-4-[1-methyl-4-oxo-8-(1H-pyrrole-3-carbonylamino)isoquinolin-3-yl]phenyl]-3-hydroxypropanoic acid 5-hydroxy-1-methyl-4-[(3-methylphenyl)diazenyl]-2-oxo-7,8-bis[[2-(trifluoromethyl)phenyl]diazenyl]quinoline-6-carbonitrile 3-[2,6-dimethyl-4-(2H-triazol-4-yl)phenyl]-5-[(2,2,6,6-tetrafluorocyclohexyl)oxymethyl]-1,2,4-oxadiazole [4-(benzylamino)phenyl]-[2-hydroxy-6-methyl-3-(3-pyrrolidin-1-ylpropoxy)phenyl]methanone 2-[(1-benzylpiperidin-4-ylidene)methyl]-5-bromophenol 1-(4-bromophenyl)-4-ethylhexan-2-one 3-[2-(3-hydroxyoxolan-3-yl)ethynyl]benzamide 1-[(4,6-dimethylpyridin-3-yl)methoxy]benzimidazole 5-[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]pyrimidine 1-chloro-3,5-dimethylbenzene;ethane N-[4-amino-2-fluoro-5-(2,3,6,7-tetrahydrofuro[2,3-f]benzimidazole-5-carboximidoyl)phenyl]propanamide 2-chloro-4,5-dihydropyrazolo[3,4-b]pyridine-7-carboxylic acid 3,5-dichloro-N-[4-(3-chlorophenyl)sulfanylphenyl]aniline N-[[1-(cyclopropanecarbonyl)piperidin-4-yl]methyl]benzenesulfonamide 3-[[6-(4,5-dihydro-1H-imidazol-2-yl)pyridin-2-yl]methylsulfanyl]propane-1-thiol (E)-5,8-dihydroxy-2,2-bis(4-propoxyphenyl)non-6-enoic acid 4-[[3,5-bis(trifluoromethyl)phenyl]carbamoyloxymethyl]cyclohexane-1-carboxylic acid N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-7H-purine-6-carboxamide (5Z)-2-(4-chlorophenyl)imino-5-[[3,5-diiodo-4-[(3-methylphenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one 3-N-(5-chloropyridin-2-yl)-1-N,4,6-trimethylbenzene-1,3-diamine N-[2,3,5,6-tetrafluoro-4-(trideuteriomethoxy)phenyl]benzenesulfonamide 2-[4-(trifluoromethyl)phenyl]-1H-1,3,5-triazine-2,4-diamine 1-[(2R)-2,3-dimethylcyclohexyl]oxy-4-fluorobenzene;formaldehyde 4-(3,3-dimethylbutanoyl)-2-pyridin-3-yl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidine-3-carboxamide 2-cyclopropyl-5-[3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-2,6-difluorophenyl]-1,3,7,8-tetrahydropyrazino[2,3-b]azepin-4-one 5-[1-(2-fluoroethyl)pyrazol-4-yl]oxy-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile 4-[[5,5,7,7-tetrafluoro-6-(3,4,5-trifluorophenyl)heptyl]amino]benzoic acid [3-[4-amino-2-(cyclohexylmethyl)butanoyl]-5,6-dihydroxy-2H-indazol-4-yl]urea 2-(4,5,6,7-tetrahydroindazol-1-yl)pyrazine 2-[(3,4-dimethoxyphenyl)sulfanyl-methylamino]-5-[(4S)-4-methylhex-5-enoyl]benzoic acid (2S)-N-[5-(1,3-benzothiazol-2-ylamino)-5-oxopentan-2-yl]pyrrolidine-2-carboxamide 2,6-difluoro-N-methyl-4-[(3R)-1-phenylpyrrolidin-3-yl]oxybenzamide [(3R,4S)-2-[2-chloro-6-(trifluoromethyl)benzoyl]-3-ethyl-4,5,7-trihydroxyheptyl]phosphonic acid 7-amino-5-[4-chloro-3-(trifluoromethyl)phenyl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 4-chloro-N-[(2,5-dimethoxyphenyl)-phenylphosphanyl]benzamide 2-[azido(diphenyl)methyl]oxolane 3-(4-chlorophenyl)-2,2-dimethylpentanamide ethane;1-[2,4,6-tri(propan-2-yl)phenyl]-3,4-dihydro-2H-quinoline 1-(5-tert-butyl-2-propan-2-ylideneoxolan-3-yl)-4-pyridin-3-ylbutane-1,4-dione (2S)-3-[4-ethoxy-2-(ethylaminomethyl)phenyl]-2-ethynylpropanoic acid 1-[3-(4-methylsulfonylphenyl)-5-propan-2-ylidenecyclohexen-1-yl]piperazine 1-[(4Z,6E)-2,5-bis(methoxycarbonyl)nona-2,4,6-trienyl]-3-[[4-[[[(4-chlorophenyl)-phenylmethyl]amino]methyl]benzoyl]amino]urea 2-[(Z)-but-1-enyl]-N-propan-2-ylideneaniline 6-methoxy-7,8-dihydro-2H-chromene-4-carboxylic acid N-[(4E)-2,3-dihydro-1H-azocin-6-yl]-1-phenylpropan-1-imine (5S,7R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-ethyl-5,7-dimethyl-1,4,5,6-tetrahydroindazole-3-carboxamide (Z)-N'-[4-(5,6-dihydronaphthalen-2-ylamino)benzoyl]octadec-9-enehydrazide (1-methylpyrazolo[4,3-d]pyrimidin-7-yl)-[8-(2-phenylethynyl)-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl]methanone 2-[(E)-2-[4-(dimethylamino)phenyl]ethenyl]-5-(1H-pyrrolo[3,2-b]pyridin-5-ylsulfonylamino)benzoic acid 2-[3-(difluoromethyl)phenyl]-N-methoxybutanamide 7-fluoro-8-(3-methylphenyl)-4H-1,4-benzoxazin-3-one 4-[3,3-bis(3-tert-butyl-5-cyanophenoxy)-2-methylidenepentanoyl]oxybenzoic acid 2-[6-oxo-5,7-di(propan-2-yl)benzo[d][1]benzazepine-11-carbonyl]oxyacetic acid 2-(6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl)phenol N-(4,5-dimethyl-2-phenyldiazenylphenyl)-4-nitro-N-(2-oxopropyl)benzamide N-[(E)-3,6-diphenylhept-4-enyl]acetamide 4-[6-(1,2,3,6-tetrahydropyridin-5-yl)imidazo[1,2-a]pyrazin-8-yl]benzamide N-(4,4,5,6,7,8-hexadeuterionaphthalen-1-yl)dibenzothiophen-2-amine 5-methyl-2,4-diphenyl-6-(1H-pyrrol-3-yl)pyridine-3-carboxylic acid (E,4S)-1-[2-ethoxy-5-(trifluoromethyl)phenyl]-4-(methylideneamino)hex-1-en-3-one 1-azidooxy-3-[4-(2,5-difluorophenoxy)butyl]piperidine 2-chloro-N'-methylbenzenecarbothiohydrazide N-(4,5-dimethoxy-2-nitrophenyl)pyrimidine-2-carboxamide 1-[4-[(E)-2-pyridin-3-ylethenyl]phenyl]-1,7,8-triazaspiro[4.4]nonane 2-(4,5-dimethylcyclohepta-1,3,6-trien-1-yl)-3,4,5,6-tetrahydrobenzo[h]quinoline 2-[2,6-dichloro-3-(1-hydroxyethyl)phenyl]-N-methoxyacetamide (4S)-3-[[2,6-difluoro-4-[5-(4-methoxyphenyl)-1,2,4-oxadiazol-3-yl]phenoxy]methyl]-4-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine N-[(1Z)-3-[2-[6-cyano-5-methoxy-2-methyl-7,8-dihydroquinoline-3-carbonyl]-4H-1,4-benzoxazin-6-yl]-1-[5-(trifluoromethyl)pyridin-2-yl]buta-1,3-dienyl]methanimidate [(1R)-2,2-difluoro-6-iodo-1-phenylcyclohexyl]carbamic acid 2-[4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]ethanol 5-[2,6-dichloro-4-(trifluoromethyl)phenyl]-3H-1,2,4-oxadiazol-2-amine 2-[1-(2,4-difluorophenyl)sulfonylpyrrolidin-3-yl]oxy-3H-pyrido[3,4-d]pyrimidin-4-one N-[(5,6-dimethylpyridin-2-yl)methoxy]benzamide N'-[(2Z,4E)-3-(dimethylamino)hexa-2,4-dienyl]-2-hydroxy-6-methoxybenzenecarboximidamide 2-(1H-benzimidazol-2-ylsulfanyl)-N'-[4-chloro-3-(trifluoromethoxy)phenyl]acetohydrazide N-[(E)-1H-indol-3-ylmethylideneamino]naphthalene-1-carboxamide 2-benzylsulfanyl-5-[(4-chlorophenyl)methyl]-1H-imidazole 1-(6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidine-3-sulfonamide 4-[1-(3,5-difluorophenyl)-3-oxobutan-2-yl]oxycarbonylpiperazine-1-carboxylic acid 3-[(4S,5R)-2,5-dimethyl-1,6-dioxaspiro[4.5]decan-4-yl]phenol 5-methyl-1H-imidazo[4,5-b]pyridine;2-(1,3,5-triazin-6-ylamino)ethanol 1-methoxy-7-[(Z)-pent-3-enyl]naphthalene 4-[2-(1,5-dimethylpyrazol-3-yl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-(3,4-diethylphenoxy)-N'-hydroxypyrimidine-4-carboximidamide 4-[1-(cyclopentylmethylamino)propan-2-ylamino]-5-methoxy-1H-pyrimidin-6-one 1,3-diamino-1-[3,5-bis(trifluoromethyl)phenyl]urea 2-amino-4,5-dimethylbenzenethiol;(3S)-3-aminooxane-2,6-dione;1-[2-(5-chlorothiophen-2-yl)ethynyl]piperidin-2-one 2-[1-hydroxy-2-(4-methylphenyl)ethoxy]-6-methoxybenzoic acid 5-(4-chlorophenyl)-2,3-dimethyl-1H-pyrazole;ethane N-[4-[(2R,4S)-2-amino-1,4-dimethylcyclohexanecarbonyl]phenyl]-2-methoxybenzenesulfonamide 4-bromo-N-(2,2,6,6-tetramethylpiperidin-4-ylidene)-1-[[3-(trifluoromethoxy)phenyl]methyl]indole-7-carboxamide (E)-1-[3-chloro-4-(2-methylpropoxy)phenyl]pent-1-en-3-one 3-[2,6-difluoro-4-[(E)-pent-1-enyl]phenyl]-7-ethenyl-8-fluoro-1,2-dihydronaphthalene 1-[5-ethylsulfonyl-6-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyridin-3-yl]cyclopropane-1-carboxylic acid 6-(2-cyclopropylpyrimidin-5-yl)-1-(4-fluorophenyl)-4,4-dimethyl-[1,3]oxazolo[4,5-c]pyridine 4-[7-(2,4-dimethylpyridin-3-yl)imidazo[1,2-a]pyridin-5-yl]benzonitrile 3-[2-(5,5-dioxo-4H-imidazo[1,2-c]quinazolin-1-yl)ethoxy]propanoic acid 2,5-diphenyl-1,3-oxazole N-(1,3-benzothiazol-2-yl)-6-methoxy-5H-isoquinoline-8-carboxamide N-[4-(3-amino-1,2,4-triazin-6-yl)-3,5-difluorophenyl]-2-chloro-5-fluorobenzenesulfonamide N-[(E)-3,3-dimethylbut-1-enyl]ethanimine;N'-[(4-fluorophenyl)methyl]-N-propylbutane-1,4-diamine;N-(2-hydroxy-2-methylpropyl)formamide (6R)-2-amino-3,4,5,6-tetrafluoro-9H-fluoren-1-amine 5-[4,5-bis(4-fluorophenyl)thiophene-2-carbonyl]imidazolidine-2,4-dione 3-[5-[(2,6-difluorophenyl)methoxy]-1H-indazol-3-yl]-N-[2-[di(propan-2-yl)amino]ethyl]-4-[4-(morpholin-4-ylmethyl)phenyl]benzamide 3,5-dimethyl-N-(2-morpholin-4-ylethyl)benzenesulfonamide 5-amino-3-[(4-butoxy-3-methoxyphenyl)methyl]-1-propan-2-ylpyrazole-4-carbonitrile 3-(4,5-dicyclopropyl-1H-imidazol-2-yl)phenol N-azido-2,3-bis(4-methoxyphenyl)propanamide 5-[3-(5-fluoro-2,3-dihydro-1H-inden-4-yl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-2-one 4-methyl-N-(1,3,5-triazin-2-yl)cyclohexane-1-sulfonamide 2-(3-azidosulfanylpropoxy)naphthalene 6-chloro-3-[2-(4-phenylpiperazin-1-yl)ethoxy]quinoxaline;dihydrochloride 1-[2,5-dimethyl-4-[[(3S)-pyrrolidine-3-carbonyl]amino]phenyl]pyrrolidine-2-carboxylic acid N'-[4-(3,5-dimethylpiperidine-1-carbonyl)-2,5-dimethoxyphenyl]ethanimidamide;ethane N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-fluoro-6-[1-[(4-formyl-2-methylphenyl)methylamino]ethenyl]-1-(4-hydroxycyclohexyl)indole-4-carboxamide 3-azido-5-(2,6-dichlorophenyl)-4H-1,2-oxazol-5-ol (E)-3-[4-[2-hydroxyethyl(methylsulfonyl)amino]phenyl]prop-2-enoic acid 5-(3,4-dimethoxyphenyl)sulfinyl-2-[4-ethyl-4-(hydroxymethyl)piperidin-1-yl]pyridine-3-carbonitrile 2-(1H-indol-3-yl)-N-methoxy-1-naphthalen-2-ylethanimine 2-[(3R)-4-methylpiperidin-3-yl]pyridine 5-methyl-N-[[4-(pyridine-2-carbonyl)phenyl]carbamothioyl]furan-3-carboxamide 3-(2,4-dihydroxyphenyl)-N'-ethylthieno[2,3-c]pyrazole-5-carbohydrazide (3-bromophenyl)-(2,6-dimethoxybenzoyl)phosphinic acid N-[(4R,5S)-6-amino-2-[4-(trifluoromethyl)phenyl]sulfonyl-3,4-dihydropyrazol-5-yl]-4-chlorobenzenesulfonamide N-[3-(difluoromethyl)phenyl]sulfanyl-1-[5-ethenyl-2,4-bis(ethenyl)-6-oxopyran-3-yl]methanesulfinamide N-(5-cyclobutylpyridin-2-yl)-3-(1H-pyrazol-4-yl)propanamide 6-[4-(dimethylamino)phenyl]imino-1,3,5-triazinane-2,4-dione N-cyclohexyl-2-[3-(trifluoromethoxy)phenyl]imidazo[1,2-b]pyridazine-6-carboxamide (5S,7R)-5-(4-hydroxyphenyl)-N-[3-(trifluoromethyl)phenyl]-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide (E)-N,2-dimethyl-4-phenylbut-3-enamide 3-amino-1-[4-(6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl)phenyl]piperidin-2-one;hydrochloride 4-[(1,3-dimethylpyrazol-4-yl)sulfonylamino]pyridine-2-carboxamide N-(1,3-diethyl-2H-quinolin-4-ylidene)hydroxylamine 5-[(3,4-dichlorophenyl)methylamino]-1-ethylpyrazole-4-carbonitrile N-(1,4-dimethylindol-5-yl)-2-(2-hydroxyethoxy)acetamide 1-[6-(4,5-dihydro-1,2-oxazol-3-yl)naphthalen-1-yl]-N'-methanimidoyl-N-methylethenamine;ethane 2-ethyl-1-[4-(5-iodopyridin-3-yl)phenyl]heptan-1-one 1-[2,4-difluoro-3-(propylsulfanylamino)phenyl]-3-(6-methoxyquinolin-5-yl)urea (2R)-N'-[(3Z,5E)-6-phenylhexa-1,3,5-trien-2-yl]sulfanyl-2-[4-(quinolin-8-ylamino)cycloheptyl]propanediamide 1-methyl-4-[5-(2-methylpropoxy)quinolin-8-yl]piperidine-3-carboxylic acid 3-amino-6-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]hexanoic acid 2-(3,4-diethoxyphenyl)-5-hexylpyrazine (E)-N-[4,5-dichloro-2-fluoro-3-(propanoylamino)phenyl]-3-(3-fluoro-6-oxopyridin-1-yl)but-2-enamide 4-[4-(2,6-diphenylpyrimidin-4-yl)phenyl]benzoic acid (1S,3R)-N-[3-cyano-4-[2-[(4R)-4-hydroxy-2-oxopyrrolidin-1-yl]pyridin-4-yl]phenyl]-3-(2,2,2-trifluoroethoxymethyl)cyclohexane-1-carboxamide 2-[6-(4-chlorophenyl)spiro[3,9a-dihydroindeno[1,2-b]pyrazine-8,4'-piperidine]-1'-yl]acetic acid N-azido-N,3-dimethylquinoxalin-2-amine N-(2-methoxyphenyl)sulfanylpyridine-4-carboxamide (E)-3-amino-2-hydrazinyl-3-[1-methyl-5-(3,4,5-trifluorophenyl)pyrazol-4-yl]prop-2-enoic acid 4-[6-[(2Z,7E)-11-ethyl-3,5-dimethylideneundeca-2,8,10-trien-1-ynoxy]pyridin-2-yl]morpholine N-(3,5-dimethylphenyl)-7H-purin-6-amine 2-[(3,5-dichloropyridine-4-carbonyl)amino]propanedioic acid (1R,2S)-2-[[8-bromo-4-(cyclopentylamino)-6,7-dihydro-5H-pyrido[3,4-d]pyrimidin-2-yl]methylcarbamoyl]cyclopropane-1-carboxylic acid;ethane [4-(2,5-dimethylfuran-3-carbonyl)piperazin-1-yl]-[6-(triazol-2-yl)pyridin-3-yl]methanone N-(2,6-dichlorophenyl)-8-(4-methyl-1H-pyrazole-5-carbonyl)quinoxaline-6-carboxamide 3-(1-benzylpiperidin-4-yl)oxycarbonylbenzoate 5-azido-4-(2,6-dichlorophenyl)-1H-pyrazole 2-[(2-chloropyrimidin-4-yl)amino]-N',3-dimethylbenzenecarboximidamide 2-methyl-4-[(3R)-3-methyl-5-oxooxolan-3-yl]oxypyridine-3,5-dicarbonitrile 1-benzyl-3,6-dimethoxy-2H-indole 2-bromo-3-(3,5-dichloropyridin-4-yl)sulfanylpropanamide 2-amino-7-[(2S,4R,5R)-5-acetyloxolane-2-carbonyl]-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 2-[5-ethoxy-6-(3,4,5-trifluorophenyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine 2-methoxyimino-3-(2-morpholin-4-ylsulfonylphenyl)propanoic acid 5-(3,4-dichlorophenyl)sulfanyl-1,2-dimethylbenzimidazole;ethane 1-(6-bromo-5-methylpyridine-2-carbonyl)-4-[(6,7-difluoroimidazo[1,2-a]pyrimidin-3-yl)methyl]pyrrolidine-2-carboxamide 1-[3-(1-azidoethyl)phenyl]-N,N-dimethylpyrrolidin-3-amine 5-[(E)-2-(6,8-difluoronaphthalen-2-yl)ethenyl]pyrimidine 6-[(2E)-2-[(3,5-dibromo-4-hydroxyphenyl)methylidene]hydrazinyl]-1H-pyrimidine-2,4-dione 1-[(E)-2-fluoro-3-methylsulfanylprop-1-enoxy]-4-(4-methylphenoxy)benzene;methanethiol N-[(E)-1-[4-(4,7-dimethyl-2,3-dihydroindol-1-yl)phenyl]ethylideneamino]-N'-methylmethanimidamide N-(2,6-dimethylphenyl)-4-[1-(1-ethanimidoylpiperidine-4-carbonyl)piperidin-3-yl]piperazine-1-carboxamide 5-[(2E)-3,7-dimethylocta-2,6-dienoxy]carbonyl-4-propan-2-ylthiophene-2-carboxylic acid 5-[(3R)-1-(2-phenylacetyl)piperidin-3-yl]-2H-triazole-4-carboxylic acid 4-(2-bromophenyl)-1-phenylcycloheptane N-benzyl-2-[1,3-dihydroisoindol-2-yl(methyl)amino]acetamide 3-[3-(1,5-dihydropyrrolo[2,3-b]pyridin-4-ylideneamino)propyliminomethyl]benzamide N-(6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-ylsulfonyl)formamide;3-(pyridin-4-ylmethoxy)cyclobutan-1-amine 1-benzylsulfonyl-3-methoxy-3,4-dihydro-2H-pyrrolo[2,1-c][1,4]benzothiazine 3-[(2,4-dichloropyrimidin-5-yl)-phenacylamino]propanoic acid 1-(3,5-dimethoxyphenyl)sulfonyl-N-[[4-fluoro-2-(trifluoromethyl)phenyl]methyl]pyrrolidine-2-carboxamide (3R)-6,7-dimethoxy-5-methyl-2,3,4,9a-tetrahydro-1H-indeno[2,1-c]pyran;ethane 1-methyl-4-(3,8,10-triazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-12-yl)piperazine 1-(2-methylpropyl)-4-[5-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]-6-(trifluoromethoxy)pyridin-2-yl]piperazine N-[6-[1-(2,3-dichlorophenyl)ethyl]pyridin-3-yl]methanesulfonamide 6-azidooxy-1H-phenanthro[9,10-d]imidazole N-[5-[(1R,3S)-3-[5-cyano-2-[4-(1H-pyrazol-5-ylamino)pyrrolo[2,1-f][1,2,4]triazin-7-yl]pyridin-3-yl]cyclohexyl]oxy-2-fluorophenyl]propanamide 6-[(4,7-dimethylindazol-2-yl)methyl]isoquinoline N-[(1R)-2,3-dihydro-1H-inden-1-yl]-1-piperidin-4-ylindole-5-carboxamide 1-[4-chloro-6-(trifluoromethyl)pyrimidin-2-yl]-3,3a,5,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrole 3-[4-(2,5-dimethylphenyl)piperazin-1-ium-1-ylidene]-4H-chromen-2-one 7-[2-(4-methylphenyl)ethylamino]bicyclo[3.2.0]hepta-1,3,5-triene-6-carboxylic acid 2-(5-chlorobenzimidazol-1-yl)-N-[2-(4-iodophenyl)ethyl]acetamide 4-amino-N-(3-methylbut-2-enyl)-1,2,5-oxadiazole-3-carboxamide 4-methylsulfanyl-6,7,8,9-tetrahydropyrido[2,1-c][1,3]benzodiazepine N-[(Z)-(2,3-dibromo-5-ethoxy-6-hydroxyphenyl)methylideneamino]-4-morpholin-4-ylbenzamide 6-[1-(4,5-dimethylthiophen-3-yl)sulfonylpyrrolidin-2-yl]pyridine-3-carboxamide N-[(3R)-1-amino-2-oxoheptan-3-yl]-6-methylpyridine-3-carboxamide;ethane (1S)-5-benzyl-4,7-ditert-butylspiro[2.5]octane 2-(2,3,5-triiodophenyl)propanedinitrile 6-chloro-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]pyridine-3-sulfonamide 2-[4-(1,3-dimethylimidazol-1-ium-2-carbonyl)piperazine-1-carbonyl]oxyimino-3-pyridin-3-ylpropanoic acid 2-[(4R,5S)-3,5-diphenyl-1,3-oxazolidin-4-yl]acetate 1-(7-fluorospiro[3,9-dihydro-2H-pyrano[2,3-h][1]benzoxepine-4,1'-cyclohexane]-1-yl)pyrrolidin-2-one (5S)-2-(4-carbamoylpiperidin-1-yl)-N-[3-chloro-4-(morpholin-4-ylmethyl)phenyl]-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 1-(2-cyclohexylacetyl)-N-[2-methyl-5-oxo-4-[3-[1-(pyridine-3-carbonyl)piperidin-4-yl]imidazolidin-1-yl]-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]pyrrolidine-2-carboxamide 3,5-dimethylbenzo[f]benzimidazole 2-[(2R)-3,3,4,4,5,5,6,7,8,9-nonadeuterio-1-(4-fluorophenyl)sulfonyloxyheptan-2-yl]decanoic acid 5-[1-[(3S)-4-[(2-fluorophenyl)methyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopentanecarbonyl]pyridine-2-carbonitrile 4-[4,6-dimethoxy-2-(3-phenylpropyl)pyrimidin-5-yl]oxybenzonitrile;ethane 2-(azidomethyl)-3-phenyl-4-propan-2-yloxypyridine N-(2,6-dichloro-4-nitrophenyl)-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]ethenesulfonamide 1-(4-bromophenyl)cyclopentane-1,2-dicarboxamide N-[3,5-bis(trifluoromethyl)phenyl]-5,6-difluorospiro[1H-indole-3,4'-thiane]-2-imine 3-(3,5-dimethylphenyl)-2H-benzo[e]benzimidazole 1-[4-(5-chloro-2H-pyrrolo[3,2-b]pyridine-1-carbonyl)phenyl]cyclopropane-1-carbonitrile 6-(5,7-difluoroquinolin-3-yl)-4H-pyrido[3,2-e]thiazin-8-one 6-[1-(6-aminopyridine-3-carbonyl)pyrrolidin-2-yl]-N,N-dimethylpyridazine-4-carboxamide 2,4-dichloro-N-(3-ethylphenyl)aniline (E)-3-[1,6-dimethyl-7-(4,8,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5,11-tetraen-12-yloxy)naphthalen-2-yl]-N-methylprop-2-enamide 7-cyclopropyl-N-[2,3-dihydro-1H-inden-1-yl(phenyl)methyl]pyrazolo[5,1-b][1,3]oxazole-6-carboxamide 1-[4-(dimethylamino)phenyl]-N'-[2-fluoro-6-methoxy-4-(5,5,8,8-tetradeuterio-6,7-dihydronaphthalen-2-yl)phenyl]cyclopropane-1-carboximidamide 3-[(4E,5Z)-4,6-dimethylhepta-1,4,5-trien-2-yl]pyridine N-[(4S,8aR)-3-phenyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-4-yl]-2-oxo-4H-1,4-benzoxazine-5-carboxamide 4-amino-3,5,6,8-tetrafluoro-9H-fluorene-2-carbonitrile 2-(4-azidocyclohexyl)phenol 4-[[1-(4-chlorophenyl)pyrrolidine-3-carbonyl]amino]benzenesulfonic acid 5-chloro-2-[3-methoxy-4-(2,2,2-trifluoroethylsulfonyl)phenyl]-7-(1,3,5-triaza-4-azanidacyclopenta-2,6-dien-2-yl)-1H-imidazo[4,5-b]pyridine 5-(1H-pyrazole-4-carbonyl)-2,3-dihydroindole-1-carboxamide 1-(4,5-dimethyl-6-phenylpyridin-2-yl)-2,3,3-trimethylbutan-1-one 2-[2-(5-fluoropyridine-3-carbonyl)-9H-fluoren-1-yl]acetic acid 5-azido-2,3-ditert-butylbenzamide 2-methyl-N'-[[4-(trifluoromethoxy)phenyl]diazenyl]propanediamide 4-[[2-(1H-indol-3-yl)ethyl-methoxycarbonylamino]methyl]piperidine-1-carboxylic acid 2-(2,3,5,6-tetrachlorophenyl)butanedioic acid N-[4-[2-ethyl-3-[2-(3,6,7-trimethoxyisoquinolin-1-yl)ethyl]phenyl]pyridin-2-yl]benzamide (5S)-5-[3,4-bis(phenylmethoxy)phenyl]-1,5,6,8-tetrahydropyrazolo[4,3-g]quinazoline N-(cyclobutylmethyl)-6-fluoroquinoline-3-carboxamide ethane;1-methyl-2-[[(2E,4Z)-penta-2,4-dien-2-yl]oxymethyl]benzene 2-(2-ethoxyphenyl)-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one 3,4-dimethoxy-N-[1-(pyridin-4-ylamino)propan-2-yl]benzamide N-(4-azidobutyl)benzenesulfonamide 1-[(4-ethylphenyl)methyl]pyrazole 4-[2-(6-iodo-5-methoxynaphthalen-1-yl)ethynyl]benzoic acid 4-cyclopropyl-6-(2,3,5-trifluorophenoxy)pyrimidine N-(5,6-dihydro-4H-cyclopenta[d][1,3]thiazol-2-yl)-3,5-dimethoxybenzamide [3-chloro-2-(cyclohexen-1-yl)phenoxy]boronic acid 1-[[3-[(3R)-7,12-dichloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),5,7,9,12,14-hexaen-2-yl]-4,5,6,8,13a-hexahydrobenzo[f]indazol-7-yl]methyl]pyrrolidine 1-[4-(1H-benzimidazol-2-yl)phenyl]pyrrolidine-2,5-dione 1-[5-[2-(cyclopropylmethylamino)pyrimidin-4-yl]-2,3-dihydroindole-1-carbonyl]piperidin-3-one 3-(2,5-difluorophenyl)-5-[3-[4-fluoro-3-(trifluoromethyl)phenoxy]propoxy]-1-(pyridin-2-ylmethyl)indole (3S)-4-acetyl-N,2-dibenzyl-1,5-dioxo-N-propan-2-ylpyrrolidine-3-carboxamide N-[2-(dimethylamino)ethyl]-4,5-dimethoxy-2-nitrobenzenesulfonamide 4-(5,6-dimethoxypyridin-3-yl)-N-[1-[2-ethyl-3-fluoro-4-(trifluoromethyl)phenyl]propan-2-ylsulfanyl]-5-(1H-pyrazol-4-yl)-1,2,4-triazol-3-amine 2-(2,3,6,7-tetrahydropyrrolo[1,2-a]imidazol-5-yl)propanamide 5-[4,6-bis(trifluoromethyl)pyrimidin-2-yl]-1,3-dihydroindol-2-one 2-ethylbutanoic acid;N'-(4-methoxyphenyl)heptanediamide N-azido-5-phenyl-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide 5-(3,4-dimethoxyphenyl)imidazolidine-2,4-dione 4-(1,3-thiazol-2-ylmethylamino)-N-[2-(trifluoromethoxy)phenyl]benzamide (4-pyridin-3-ylpiperazin-1-yl)-[5-(1H-pyrrol-2-ylmethylideneamino)furan-2-yl]methanone 4-azido-N,N-dibutylaniline 2-[4-(2,3-dihydrofuran-5-yl)cyclohexen-1-yl]aniline 2-[(3R)-1-(5,7-difluoroquinolin-6-yl)pyrrolidin-3-yl]-N-[(4S)-5-methoxy-6-phenylpiperidin-3-yl]acetamide N-[1-(5-cyclopropylpyrimidin-2-yl)ethoxy]-2,5-difluorobenzamide N-[(3,5-dimethylphenyl)methyl]-8-(2-ethoxypropylsulfonylamino)-4-oxo-3,7-dihydropyrido[2,1-b]quinazoline-6-carboxamide 6-[2-[[1-(2,4-difluorophenyl)ethyl-methylamino]methyl]pyridin-3-yl]-3-methylidenepyrido[2,3-e]thiazin-4-one 2-[(E)-1,2-dichloroethenyl]isoindole 4-(3,5-dimethylphenyl)-2,6-dimethylpyrimidine;ethane 4-[1-(6,7-dimethoxyquinazolin-2-yl)piperidin-3-yl]-1-oxidopyridin-1-ium N-(furan-2-ylmethyl)-5,6-dioxo-4H-imidazo[1,5-a][1,4]benzothiazepine-3-carboxamide 2-cyclobutyloxy-N-methyl-N-(2,4,6-trimethylphenyl)acetamide (2S)-5,7-dihydroxy-1'-methyl-3,7-dioxospiro[2H-pyrano[4,3-c]pyran-8,4'-piperidine]-6-carboxylic acid 2-ethyl-1-methoxy-3,4-dihydroisoquinoline-1-carboxylic acid [2-(3,5-dimethoxyphenyl)-1,3-benzothiazol-6-yl]-ethoxymethanamine 7-fluoro-6-(5-methylsulfonylpyridin-3-yl)oxyquinoline 5-azido-2-butyl-1,3,4-thiadiazole 1-[3,4-dimethoxy-5-(trifluoromethyl)phenyl]ethanamine;hydrochloride 2-[4,7-bis(carboxymethyl)-5-[(3-cyanophenyl)methoxy]-1,8-dioxonaphthalen-2-yl]acetic acid 2-[3,5-dihydroxy-4-[6-(4-methylpiperazin-1-yl)naphthalene-1-carbonyl]oxyphenyl]acetic acid 2-(2,5-dibromophenyl)acetamide;ethane 1-(4-chlorophenyl)sulfinyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrole 3-methyl-2-(N-[4-(pyrimidin-2-ylsulfamoyl)phenyl]anilino)butanoic acid 4-[(E)-but-2-enoxy]-N-methylsulfonylbenzamide 4-[2,3,5,6-tetradeuterio-4-(trideuteriomethyl)phenyl]-2H-benzotriazol-5-amine 3-[5-(1,3-benzodioxol-5-ylmethylidene)-2,4-dioxo-1,3-thiazolidin-3-yl]propanamide N'-(5-bromopyrimidin-2-yl)butanediamide 2-[azido(benzylsulfonyl)amino]acetamide 2-(4-bromophenyl)sulfinyl-N'-(4-hydroxybutylamino)propanediamide 1,2-diamino-4-[4-ethoxy-3-(trifluoromethyl)phenyl]-6-oxopyridine-3,5-dicarbonitrile 2-[(3R,4S)-1-acetyl-3-fluoropiperidin-4-yl]oxy-5-[4-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]phenyl]benzonitrile 1-[4-[2-(oxan-4-yl)benzimidazol-1-yl]phenyl]azetidin-3-ol 2-[4-[[(4R)-1-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-4-carbonyl]amino]pyrazol-1-yl]acetic acid (3-fluorophenyl)methyl-[5-[(3-hydroxy-6,7-dimethoxyquinolin-4-yl)amino]-2,4-bis(sulfanylidene)pentyl]oxidanium 3-bromo-N-[1-(cyclohexanecarbonyl)piperidin-4-yl]benzenesulfonamide 4-[3-[(2R)-2,5-dimethylmorpholine-4-carbonyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]cyclohexane-1-carboxamide 2-(4-ethylpiperazin-1-yl)-5-fluorobenzenecarboximidamide 1-[4,5-bis(ethenyl)-3H-pyrazole-2-carbonyl]-4-hydroxypyrrolidine-2-carboxylic acid 2-N,5-N-diethyl-1,4-dihydronaphthalene-1,2-disulfonamide 3-[1-(4,6-dichloro-1H-benzimidazol-2-yl)ethoxy]benzonitrile 2-[5-[(2S)-butan-2-yl]-4-methoxypyrimidin-2-yl]propanedioic acid 4-[2-amino-3-methyl-5-(trifluoromethoxy)phenyl]-6,7-dihydro-5H-1,3-benzothiazol-2-amine N-(1,3-benzodioxol-5-ylmethyl)spiro[1,4-dihydroquinoxaline-3,4'-oxane]-2-imine;hydrochloride (5Z)-2-(4-chlorophenyl)imino-5-[(2,3-dimethylindazol-6-yl)methylidene]-1,3-thiazolidin-4-one 3-[1-(2,6-dichlorophenyl)propan-2-yl]-5-pyrimidin-4-yl-1,2,4-oxadiazole 2-[N-(1,3-diethoxy-1,3-dioxopropan-2-yl)-4-nitroanilino]octanoic acid 4-fluoro-2,3-di(propan-2-yl)aniline (2S)-N,N-diethyl-3-[6-methoxy-1-[3-methoxy-4-(1H-pyrrolo[3,2-c]pyridin-7-yl)phenyl]hexyl]pyrrolidine-2-carboxamide 2-(2-azidoethoxy)benzenesulfonic acid ethane;N-[1-(3-nitrophenyl)ethenyl]-4-propan-2-ylidenecyclohexa-1,5-diene-1-sulfonamide 1-[(1R)-5,7-dimethoxy-3,4-dihydro-2H-naphthalen-1-yl]ethanol 2-cyclopropyloxy-N-[(3,4-dimethylphenyl)methyl]-5-fluorobenzamide 5-[(4-bromophenyl)methyl]-2,3-dihydro-1H-pyrrolizine;5-nitro-3,4-dioxo-2H-pyrrole-1-sulfonate 4-amino-3-bromobenzoate (1R,3S)-3-[6-[5-[[methoxycarbonyl(propyl)amino]methyl]pyridin-2-yl]-3-oxo-1H-isoindol-2-yl]cyclohexane-1-carboxylic acid 4-amino-3-(1,2,3,5,6,7-hexahydropyrrolizine-8-carbonyl)-N-[(1R)-1-phenylethyl]cyclohexane-1-carboxamide [3-methyl-2,6-di(propan-2-yl)phenyl]phosphane 4-azidooxy-5,6-diethylpyrimidine N-[4-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1]benzazepine-11-carbonyl)phenyl]-N-ethylacetamide 2,3-bis(4-methoxyphenyl)-5H-[1]benzofuro[3,2-c]azepine N-(4-aminophenyl)sulfanyl-1,3-thiazol-2-amine 7-(methylamino)-5,6,7,8-tetrahydronaphthalene-2-carbonitrile N-[2-[(5S)-3-(4-methoxyphenyl)-5-propanoylimidazolidin-1-yl]ethyl]acetamide 3-[5-(2,4-dimethoxyphenyl)pyridin-3-yl]oxyphenol 3,4-dichloro-N-[4-(difluoromethyl)phenyl]cyclohexa-1,5-diene-1-carboxamide 3-cyclohexyl-6,8-dihydroxy-4H-quinazoline-2-carboxamide 1-(2,3-dihydroindol-1-yl)pentan-3-one N-cyclohexyl-5,6-dimethoxy-2H-pyrazolo[1,5-a]pyrimidine-3-carboxamide (3S,5R)-1-[2-chloro-4-(trifluoromethyl)phenyl]sulfonyl-N-[[3-ethoxy-2-(1H-pyrrole-2-carbonylamino)pyridin-4-yl]methyl]-5-methylpiperidine-3-carboxamide 2-(4-butylphenyl)-1,3-difluorobenzene N-[2-(3,4-dimethoxyphenyl)ethyl]-5-methylpyrazine-2-carboxamide 4-[4-(3-cyano-6,7-dimethoxyquinolin-4-yl)pyrazol-1-yl]butanoic acid 2,6-dimethyl-7-[(3R)-pyrrolidine-3-carbonyl]-5,8-dihydro-4H-pyrazolo[1,5-d][1,4]diazepine-3-carboxamide 5-methyl-1-(4-pent-1-en-2-ylphenyl)pyrrolidine-3,4-diol 4-(5-bromopyridin-2-yl)-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione N-[2,4-difluoro-3-[7-(5-methyl-1H-indazol-4-yl)-2-oxo-4H-pyrimido[4,5-c]pyridazin-3-yl]phenyl]propane-1-sulfonamide 1-[5-(2,6-difluorophenyl)sulfonylpentyl]azetidine;ethane 2-(benzimidazol-1-yl)-N-[(4,5-dimethoxycyclohexa-1,3-dien-1-yl)methyl]ethanamine 3-[4-[2-(8-chloro-1,7-naphthyridin-2-yl)ethynyl]phenyl]pyrazine-2-carboxamide 4-(2,5-dimethoxyphenyl)imino-N-ethyl-5-[(4-hydroxy-3,5-dimethoxyphenyl)methylideneamino]-1,3,4-thiadiazol-2-amine 4-[[5-[(E)-1,2-bis(4-bromophenyl)ethenyl]tetrazol-2-yl]methoxy]benzoic acid 2-[[(4S)-1,3-dibenzylpiperidin-4-yl]methoxy]acetamide (2E,4Z)-N-[(3S,5R)-1-benzyl-5-methoxypiperidin-3-yl]-3-(hydroxyamino)hepta-2,4-dienamide N-(3,4-dimethoxyphenyl)-2-[2-ethylsulfanyl-6-[(2-iminopiperidin-1-yl)methyl]pyrimidin-4-yl]acetamide 4-[(2,3-dimethylphenyl)iminomethyl]benzene-1,3-diol 4-[[6-(3-aminopyrrolidine-1-carbonyl)-2,5-dimethylindol-1-yl]sulfonylmethyl]benzoate 1-(dimethylamino)-3,4-bis[2-(trifluoromethoxy)phenyl]butane-1-sulfonic acid 4-[(1,5-dimethylpyrazole-3-carbonyl)amino]-N-[1-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)propan-2-yl]benzamide (E)-N'-[1-[5-(2,4-dichlorophenyl)-3H-pyrrol-2-yl]ethenyl]ethene-1,2-diamine (4S)-3,7-dimethyl-1-phenylazecan-5-one N-[(E)-but-1-enyl]-5-chloro-4-(pyridin-2-ylmethoxy)cyclohexa-2,4-diene-1-sulfonamide N-[2-(4,5-dimethylthiophen-3-yl)ethyl]-2-oxocyclopentane-1-carboxamide N-azido-4,5-dimethyl-2-phenyldiazenylaniline 3-benzylsulfanyl-6,7-dichloro-4H-chromene 4-[(3S,5R)-3-methyl-5-(trifluoromethyl)piperidin-1-yl]pyridazine 2-[1-(6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl)piperidin-4-yl]acetic acid (E)-N,3-dimethyl-2-[1-[4-(methylideneamino)sulfanylphenyl]ethenylimino]but-1-en-1-amine 7-bromo-2-[(4R,5S)-5-chlorocyclohexa-1,3-dien-1-yl]sulfonyl-5H-pyrrolo[2,3-b]pyrazine (2R)-1-N,2-N-diethyl-4-methoxycarbonylbenzene-1,2-disulfonamide 2-[5-(4-chlorophenyl)-4-methyl-4-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenol N-[4-(2,6-dimethoxypyrimidin-4-yl)phenyl]-3-oxobutanamide N-[6-(2,4-dimethyl-1H-pyrrol-3-yl)pyridin-3-yl]formamide;N-ethyl-3-phenylpropanamide (3E)-5-chloro-3-[(5,6-dimethyl-1H-benzimidazol-2-yl)imino]indole-2,7-dione 1-azidosulfanyl-3,5-dimethoxybenzene 1,3-dichloropropylbenzene;ethane;N'-(3-methoxyphenyl)-2-methylidene-3H-1,4-benzothiazine-5-carbohydrazide (6R)-6-ethenyl-2,3,4,9,11-pentazatricyclo[8.5.0.02,7]pentadeca-1(10),11,13-triene 2-(4-methoxyphenyl)-1H-imidazo[4,5-b]pyridine (Z)-2-amino-4,4-dimethyl-N'-[N'-(1H-pyrrolo[3,2-c]pyridin-6-yl)carbamimidoyl]pent-2-enimidamide (3-benzylpyrrolidin-1-yl)-[4-hydroxy-5-(2,4,6-trimethylphenyl)sulfanylthiophen-2-yl]methanone 2,3-difluoro-N'-(2-hydroxy-1H-indol-5-yl)benzenecarboximidamide 3-N-[1-(3-fluorophenyl)propyl]pyrazine-2,3-diimine 2,5-dichloro-4-(3,3,3-trifluoropropyl)benzoate 3-[2-(1,3-benzodioxol-5-yl)ethyliminomethyl]-5-tert-butyl-1H-indol-2-ol (E)-2-cyano-N'-[1-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)ethoxy]-3-[2-[2-(trifluoromethoxy)phenyl]phenyl]prop-2-enimidamide N-[3,5-bis(trifluoromethyl)phenyl]acetamide;8-chloro-2-ethyl-3H-imidazo[4,5-c]quinoline 3-(2,6-dimethylpyrimidin-4-yl)piperidine-1-carboxylic acid ethane;N-[(Z)-3-hydroxyiminobutan-2-ylideneamino]quinoline-6-carboxamide 1-[3-(2,6-dichlorophenyl)propyl]-4-methoxypiperidine 2-[(4-ethylphenyl)methylamino]benzaldehyde 2-methylsulfinylspiro[1,3-dihydroisoquinoline-4,1'-cyclopropane] 6-(4-methylpiperazin-1-yl)pyridine-3-carboxamide 2-[5-(1H-pyrrol-3-yl)-1,3,4-oxadiazol-2-yl]naphthalen-1-ol 2-[4-(trifluoromethoxy)anilino]pyridine-3-carboxylic acid 2-(4-azidophenyl)sulfonylethanamine 2-cyclopropyl-5,6,7-trimethoxyimidazo[1,2-a]pyridine (4R)-4-[2,3-dihydro-1H-inden-5-ylsulfonyl(2,2-dimethoxyethyl)amino]pentanoic acid 3-[[4-[[(1R)-6,7-difluoro-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraen-12-yl]oxymethyl]phenyl]methyl]-1-propan-2-ylpyridine-2,6-dione 7-(4,4-dimethylpiperidine-1-carbonyl)-9-[3-(2H-tetrazol-5-yl)pyridin-4-yl]carbazole-3-carboxamide N-[(E)-1,3-diphenylprop-2-enylideneamino]-4-phenoxyaniline N-[4-(2,3,5-trifluorophenyl)phenyl]benzenesulfonamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-[[4-methoxy-5-(3-pyridin-2-ylpropylsulfanyl)-1,3-thiazol-2-yl]amino]benzenesulfonamide (2S)-3-phenyl-1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazole-2-carboxamide [(2S,3R)-6-(4-chlorophenyl)-1-methyl-3-propan-2-yloxycarbonylhexan-2-ylidene]oxidanium N-[(2R)-2,3-dihydroxypropyl]-2-methyl-4-oxo-6-pyrrolidin-1-ylpyran-3-carboxamide 2-amino-3-[1,4-dimethyl-6-(trifluoromethyl)indol-3-yl]propanoic acid 2-[3-(1H-indol-6-yl)-2,5-dimethylidenepyrrolidine-1-carbonyl]-3H-1,7-naphthyridin-4-one 4-hydroxy-N'-methyl-3-[(E)-2-methyl-3-oxo-1-phenylbut-1-enyl]benzenecarboximidamide 6-tert-butyl-5,7-dimethoxythieno[2,3-b]pyridine;5-(5,6-dihydronaphthalen-1-ylamino)quinoline-8-sulfonic acid 3-[3-[2,6-dichloro-4-(trifluoromethyl)phenoxy]-5-ethoxyphenyl]propanoic acid 2-[(3S)-piperidin-3-yl]oxy-5-(trifluoromethyl)pyrazine;hydrochloride N-[1-[1-(2,6-dimethylpyridin-4-yl)cyclopropanecarbonyl]piperidin-3-yl]-N-(2-morpholin-4-ylethyl)acetamide (2R)-5,6-dichloro-2-methyl-3-(3-methylidenepentanoylamino)-N-[1-oxo-4-phenyl-1-[4-(pyrrolidine-1-carbonyl)anilino]butan-2-yl]hexanamide 1-(4-chloro-2,3-dihydroxyphenyl)pentane-1,5-dione 4-(2,6-dimethylpyridin-3-yl)-1-[2-ethoxy-5-(2-pyrrolidin-1-ylethoxy)phenyl]pentan-2-one 4-[4,5-bis(ethenyl)-2-hydroxyphenyl]-3-hydroxybenzonitrile N-[3-amino-5-(furan-2-yl)phenyl]-4-[(1Z,3E)-penta-1,3-dienoxy]benzamide (2S)-1,3-bis[(4-methoxyphenyl)sulfanyl]propane-2,2-diamine 3-[(3S,4R)-1-benzyl-6-oxo-4-[2-(5-oxopyrrolidin-2-yl)ethoxy]-5H-pyrimidin-2-yl]benzoic acid 3-(methanesulfonamido)-1-[4-[2-[1-[(1S,5R)-3,3,6,6-tetramethyl-6,7-dihydro-4H-furo[3,2-c]pyridine-5-carbonyl]piperidin-4-yl]ethyl]phenyl]pyrrolidine-2-carboxylic acid 2,4-dimethyl-5-(5-morpholin-4-ylsulfonyl-3-propanoylbenzenecarboximidoyl)-N-[1-(1,3-thiazol-2-yl)cyclohexyl]oxypyrazole-3-carboxamide 3-chloro-N,5-dimethyl-4-[5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]benzenesulfonamide;ethane 2-[(1R)-1-[4-cyclobutyl-3-[methyl-(5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-4-yl)amino]phenyl]ethyl]isoindole-1,3-dione 2-cyclohexa-1,5-dien-1-yl-N'-(2-hydroxyphenyl)ethanimidamide 2-(4,5-diphenylpyrimidin-2-yl)cyclohexa-1,3-diene-1-thiol 7-(6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonyl)-4H-1,4-benzoxazin-3-one 4-(3,5-difluorophenyl)-6-[2-(methylamino)pyrimidin-4-yl]pyrazolo[1,5-a]pyridine-3-carbonitrile N-(4,5-dihydroxy-2-methylphenyl)acetamide 3-[3,5-bis(4-methylphenyl)-1,2,4-triazol-1-yl]-N-[4-cyano-3-(trifluoromethyl)phenyl]butanamide (6S)-7,8-difluoro-N-methoxy-1'-methylspiro[4H-quinoxaline-3,2'-piperidine]-2-imine;dihydrochloride 5-bromo-2,3-dimethyl-1-benzothiophene (2S)-3,4-difluoro-N-[6-(5-phenylmethoxy-1H-indazol-3-yl)pyrazin-2-yl]pyrrolidine-2-carboxamide (E)-3-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl-(3,4,5-trimethoxyphenyl)methanone 1-[4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]-3-[2-oxopropyl(3,4,5-trifluorophenyl)methyl]urea N-[2,4-difluoro-3-(furan-3-yl)phenyl]pentanamide;1,4-xylene 4-(3-azido-1H-pyrrolo[2,3-b]pyridin-5-yl)benzaldehyde 2-(3,6-dihydro-2H-pyridin-1-yl)-N'-hydroxypyrimidine-4-carboximidamide 2-(6-chlorocyclohexa-1,3-dien-5-yn-1-yl)-5H-indeno[1,2-b]pyridine 7-[3-hydroxy-3-methyl-5-(2,4,4-trimethylpentanoylamino)pentoxy]-1H-indole-2-carboxylic acid 5-(2,3-dichlorophenyl)-1H-imidazole;ethane 2-[(2S)-1-azidooxypropan-2-yl]-6-chlorobenzenesulfonamide 3-[7-[4-(2,2-dimethylpropoxy)benzoyl]-4a-hydroxy-1H-pyrrolo[2,3-b]pyridin-5-yl]benzoic acid 1-bromo-4-(3,7-dimethyloctoxy)benzene 3-[4-amino-3-(2,5-difluorophenyl)pyrazolo[3,4-d]pyrimidine-1,7-diium-1'-yl]phenol N-[(Z)-1-amino-3-iminoprop-1-enyl]-5,6-difluoro-1-methylindazole-7-carboxamide 2-[(Z)-1-bromoethenyl]-5,6,7-trimethoxy-3H-quinazolin-4-one 3-ethylsulfonyl-N,4-dimethylbenzamide 4-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-3-yl)-N-methylbenzamide 2-[3-(4-aminophenoxy)propoxy]aniline 4-[2-azido-1-(3,4-dimethoxyphenyl)ethyl]phenol (4R)-2-(1,3-benzoxazol-2-ylmethylidene)-5-methoxy-8-oxo-N-phenyl-4-propan-2-yloctanamide 1-[6-(difluoromethoxy)pyridin-3-yl]-7-fluoroimidazo[4,5-c]quinoline N-(3,3-diphenylpropanoyl)benzamide 4-benzyl-2,4-dimethoxycyclohexa-1,5-dien-1-ol 2-[(E)-2-ethenylbut-1-enyl]-5-pyridin-4-yl-3H-thieno[2,3-d]pyrimidin-4-one N-[(2R)-1,1-dihydroxypropan-2-yl]-4-(3-fluoroanilino)benzamide 4-(1H-imidazol-5-yl)-3,5-dimethyl-N-[2-oxo-2-(2-phenylethylamino)ethyl]thiophen-2-amine;2,2,2-trifluoroacetic acid 1-(4-methoxyphenyl)sulfonyl-2,3,6,7-tetrahydroazepine 2-(4-fluorophenyl)sulfanyl-N'-hydroxypyrimidine-4-carboximidamide 2-(4-acetylphenyl)imino-5-methylcyclohexane-1,3-dione 3-(1,2,4-triazol-4-ylmethoxy)piperidine-2,6-dione 1-(3,5-difluoro-4-methoxyphenyl)cyclopropane-1-carbonitrile;3-fluoro-4-hydroxybenzamide N-benzyl-6-[2,6-di(propan-2-yl)phenyl]-1-methylpyrazolo[3,4-d]pyrimidin-7-amine;ethane 5-(2,6-dimethylpyridin-4-yl)oxy-N-[1-(3-fluorophenyl)cyclobutanecarboximidoyl]pyridine-3-carboxamide 2-[6-(5-chloro-1H-indazol-7-yl)-4-oxoquinazolin-3-yl]-N-propanoylacetamide 3-[1-(2,4-dimethylphenyl)ethenyl]-5-ethoxycarbonylpyridine-2-carboxylic acid 1-[1,3-bis(3-methoxyphenyl)-2-methyl-2H-imidazol-5-yl]pyrazole N-[2,4,6-trimethyl-3-(4-methylsulfinylphenyl)sulfanylanilino]sulfanylhydroxylamine (2-azidopyrimidin-4-yl)-diphenylphosphane N-(2,4-dichloropyrimidin-5-yl)-3-methoxy-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]benzamide [5-chloro-2-(methylamino)phenyl]-piperidin-4-ylmethanone N-[4-amino-3-(1,2-oxazole-5-carboximidoyl)phenyl]-3-methoxybenzamide;methane ethane;N-[6-(2-ethylhexoxy)-1,3-benzothiazol-2-yl]cycloheptanecarboxamide [(1R,2R)-2-[4-(5-fluoropyridin-3-yl)-5H-pyrrolo[3,2-d]pyrimidine-7-carbonyl]cyclopentyl]-pyrrolidin-1-ylmethanone 4-(cyclohexylmethoxy)naphthalene N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-3-(1H-imidazol-5-ylmethylamino)benzamide N-[(2S)-1-[4-[ethyl(oxan-4-yl)amino]piperidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]quinoline-8-carboxamide 7-methyl-2-(4-pyridin-4-yl-1H-pyrazole-5-carbonyl)-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 3-chloro-N,6-dimethoxy-1H-indole-2-carboxamide 3-chloro-2-ethylbenzo[f]isoindole-1,4-dione 6-azido-N'-[4-[3-[(3S)-5,7-dichloro-2,3-dihydro-1-benzofuran-3-yl]propoxy]phenyl]pyridine-2-carboximidamide 2,7-ditert-butyl-4-(propanoylamino)benzo[e]indole-9-carboxylic acid [4-(azidomethyl)phenyl]-(6,8-dihydro-5H-imidazo[1,5-a]pyrazin-7-yl)methanone 6-[1-(6-chloronaphthalen-2-yl)sulfonylpiperidin-4-yl]oxy-5,8-difluoro-1H-quinolin-2-one 5-[3-[(2R)-5,7-difluoro-4-methoxy-1H-indol-2-yl]propyl]pyrimidine-2,4-diamine 4-cyclohexyloxyquinoline-7,8-diamine 2-[5,6-bis(ethenyl)pyridin-3-yl]-4-N-(4-cyclohexyloxyphenyl)pyrimidine-4,6-diamine 2-(1H-imidazole-5-carbonyl)-3-methylsulfanyl-4-phenylbutanenitrile 3-amino-6-chloro-4-phenylcyclohexa-1,5-diene-1-carboxylic acid N-(1,3-benzothiazol-2-yl)-2-[[4-methyl-6-oxo-2-(1,2,4-triazol-1-ylmethyl)-1H-pyrimidine-5-carbonyl]amino]acetamide (4-azidophenyl)sulfanylurea 2-[(E)-3-[5-amino-6,7-dihydroxy-8-[3-(trifluoromethyl)phenyl]naphthalen-2-yl]prop-1-enyl]cyclohexan-1-one 5-(4-butoxy-3,5-difluorophenyl)imidazolidine-2,4-dione 4-[2,4-diamino-6-(methylamino)pyrimidine-5-carboximidoyl]benzenesulfonamide 2-[[(E)-3-hydroxy-1,4-dioxobut-2-en-2-yl]-[(E)-2-nitroprop-1-enyl]amino]benzenesulfonic acid 6-methyl-2,4,5,7-tetrahydropyrazolo[3,4-b]pyridine-3-sulfonamide N-[2,6-dimethoxy-4-(3-methyl-1,3-benzothiazol-3-ium-5-carbonyl)phenyl]-2,4-dioxopentanamide 4-[1-(1,5-dimethylpyrazole-4-carbonyl)piperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one 2-(3-carbamimidoylanilino)propanoate 3-[5-tert-butyl-4-hydroxy-2-[(Z)-prop-1-enyl]phenyl]acetic acid [[2-aminoethyl(pentanoyl)hydrazinylidene]methylhydrazinylidene]azanide;rhenium;triphenylphosphane N-(6,7-dihydro-5H-cyclopenta[c]pyridazin-3-ylmethyl)-2-iodo-3,4-dihydropyrazole-5-carboxamide 6-(N'-benzylcarbamimidoyl)-2,3-dihydronaphthalene-1-carboxylic acid 1-[2,5-difluoro-3-(3-fluoro-4-hydroxyphenyl)sulfanyl-6-propylcyclohexa-1,3-dien-1-yl]ethanone 2-(2,4-dichlorophenoxy)-1-[3-[(E)-3-(hydroxyamino)prop-1-enyl]piperidin-1-yl]propan-1-one 3-[(1R)-3,3-dimethylcyclohexyl]-5-(4,6-dimethylpyridin-2-yl)-7H-pyrazino[2,3-b]pyrazin-6-one 7-cyclopentyl-2-[3-hydroxy-4-(pyrrolidine-1-carbonyl)anilino]pyrrolo[2,3-d]pyrimidine-6-carboxamide (2Z,4E)-N'-[1-[5-(2-ethylbutoxymethyl)thiophen-3-yl]ethenyl]-2-fluoro-3-methylidene-6-methyliminohexa-2,4-dienimidamide 6-[1,3-dimethyl-4-(2-phenylethoxy)pyrazolo[3,4-b]pyridin-5-yl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 4-[3-(2,6-dioxopiperidin-3-yl)-1H-pyrazol-5-yl]benzenesulfinamide 5-[4-chlorobutyl(ethenylsulfonyl)amino]naphthalene-2-sulfonic acid (E)-5-[2-azido-3,5-bis(trifluoromethyl)phenyl]pent-4-en-1-ol 7,9-bis(2-methylpropoxy)naphthalene-1,3,8-trithiol 6-(2,3,5,6-tetrafluorophenoxy)hexane-1,5-diol (3R)-3-[1-(1H-indol-2-yl)ethoxy]pyrrolidine 4-methyl-2-[(3S)-5-oxopyrrolidin-3-yl]sulfanyl-1H-pyrimidin-6-one 2-(2,6-difluorophenyl)acetonitrile;5-[3-methoxy-4-[(1-tritiopyrazol-3-yl)oxymethyl]thiophen-2-yl]-7H-pyrrolo[2,3-d]pyrimidine 2-(4-fluoro-3-pyridin-4-ylphenyl)-N,2-dimethylpropanamide 4-[5-(2,3-dichlorophenyl)furan-2-yl]-1-(4-hydroxyphenyl)azetidin-2-one 4-(3,6-dihydro-2H-pyridin-1-ylmethyl)-1H-indole 1-[4-[(3Z,5E)-2-chlorohepta-1,3,5-trien-3-yl]phenyl]-3-(trifluoromethyl)pentan-2-one N-methyl-3,9-diphenylfluoren-2-amine N-[(2R,3R)-4-cyano-1-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)piperidine-1-carbonyl]piperidin-3-yl]acetamide (E)-N-[3-bromo-5-(2,2-difluoroethoxy)phenyl]-3-thiophen-2-ylprop-2-enamide 1-[3-[2,6-diethyl-4-(hydroxymethoxy)phenyl]-6-hydroxyisoquinoline-8-carbonyl]azetidine-3-carboxylic acid 5-chloro-3,4-diethylpyridine-2-carboxylic acid 3-chloro-5-[1-(cyclohexylamino)ethenyl]benzenesulfonamide 7-(cyclohexylamino)-2,4-dioxo-1H-pyrimido[4,5-b]quinoline-3-carboxylic acid 6-(4-chlorophenyl)sulfanyl-N-[3,5-difluoro-4-(1H-pyrazol-4-yloxy)phenyl]pyrrolo[2,3-b]pyridine-1-carboxamide 4-[5-(3,5-dimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]cyclohexan-1-amine N-[3-(aminomethyl)phenyl]-6-[2-fluoro-5-(hydroxymethyl)phenoxy]-1H-benzimidazole-4-carboxamide 4-[4-(3,3a,5,6,7,7a-hexahydro-2H-pyrrolo[3,4-b]pyridine-1-carbonyl)phenyl]-6-(1,3-thiazol-2-ylamino)sulfanyl-1H-pyridin-2-one 1-ethylsulfanyloxy-2,3-bis(phenylmethoxy)benzene 1-(4-phenylmethoxyphenyl)-2H-thieno[3,2-d]pyrimidine 2-methyl-4-[6-(1H-pyrazolo[3,4-b]pyridin-5-yl)pyridazin-3-yl]quinoline 2-hydroxy-3,4-diphenylpentanenitrile 2-[N-(4-bromobutan-2-yl)-3,5-dichloroanilino]octanoic acid 4-[(5-methyl-1,2-oxazol-3-yl)diazenyl]-2,6-dinitrophenol N-(4,5-dimethylpyrimidin-2-yl)-4-[ethoxycarbonyl(2-hydroxyethyl)amino]benzenesulfonamide (1R)-3,4,5-trihydroxy-6-[(E)-nonylideneamino]-7-phenoxycyclohepta-2,4-dien-1-one 2-[5-bromo-4-(trifluoromethyl)pyrimidin-2-yl]sulfanylacetic acid 2-[5-bromo-3-(4-chlorophenoxy)-2-methylindol-1-yl]acetic acid 2-(2,3-dichlorophenyl)-3-oxobutanamide N-[5-(1,3-benzoxazol-6-yl)pyrazin-2-yl]cyclopropanecarboxamide 3-[(4-chlorophenyl)methyl]quinolin-7-ol 5-[2,6-bis(hydroxymethyl)phenyl]-1H-carbazole-3-carbonitrile 5-bromo-N-[(3R,4S)-3-hydroxypiperidin-4-yl]-1H-indole-7-carboxamide;hydrochloride 2-methyl-4-oxo-3-[(1,3,5-trimethylpyrazole-4-carbonyl)amino]chromene-8-carboxylic acid N-benzyl-3-[(4,4-difluorocyclohexen-1-yl)methylsulfanyl]-6-nitroquinolin-2-amine 1-(4-nitrophenoxy)-3,5-dihydro-2H-imidazo[1,2-b]pyrazole 3-(2,5-dimethylphenyl)-1H-pyrrole-2-carboxamide;hydrochloride 1-(2,6-dimethoxyphenyl)sulfonyl-3-piperazin-1-ylpyrrolo[2,3-b]pyridine 4-tert-butylbenzenesulfonate;(1R)-3-[(E)-2-pyridin-4-ylethenyl]cyclohexan-1-ol 2-N,3-diphenyl-1H-isoindole-2,4-diamine 3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]propanamide 6-[3-(3-hydroxypyrrolidine-1-carbonyl)phenyl]-4-oxo-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 3-[2-[(E)-(1,5-dimethylpyrazol-4-yl)iminomethyl]phenyl]propanoic acid 2-(5,6-dimethylpyridine-3-carbonyl)-N-[4-[2-hydroxyethyl(methyl)amino]phenyl]piperazine-1-carboxamide [4-[3-[2-methyl-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]-5,6-dihydroimidazo[1,2-b]pyrazole-1-carbonyl]cyclohexyl]-morpholin-4-ylmethanone 3-(5-chloropyridin-2-yl)-4-(2,6-difluorophenyl)-1H-imidazol-3-ium;methanesulfonate N-(dimethylaminosulfanyl)-2,4,6-trinitroaniline (2S)-2-[2,2-dimethyl-3-(5-methyl-1H-indol-2-yl)azetidine-1-carbonyl]pyrrolidine-1-carboxylic acid 1-[3,4-bis(phenylmethoxy)phenyl]-2-[(2-bromophenyl)sulfonylmethylamino]ethanone (2S)-3-(1H-indol-6-ylamino)propane-1,2-diol 5-(5,6-dimethyl-1H-benzimidazol-2-yl)-4-iminohexa-2,5-dienenitrile N-(4,5-dihydro-1H-pyrazol-3-yl)-2-oxo-6-pentan-2-ylchromene-3-carboxamide 2-(4,5,6,7,8,9-hexahydrocycloocta[b]furan-3-yl)-1H-imidazole 4-(1,3-benzodioxol-5-ylmethylidene)-1,2,6-tri(propan-2-yloxy)pyrimidine 2-[5,6-dimethyl-2-(oxan-4-yl)pyridin-3-yl]-N-methylacetamide 3-chloro-N'-[(Z)-1H-indol-3-ylmethylideneamino]benzenecarboximidamide N-[[(2S,4R)-1-tert-butyl-4-fluoropyrrolidin-2-yl]methoxy-hydroxyphosphoryl]benzenesulfonamide 4-[2,3-dihydroxypropyl(phenacyl)amino]benzenesulfonic acid [[2-[(3S)-1,5-dioxohexan-3-yl]oxyphenyl]-hydroxymethylidene]oxidanium 5-bromo-N-cyclopropyl-2,3-dimethoxyaniline (3R)-1-[(2R,6S)-4-hydroxy-7-methoxy-6-(5-methylfuran-2-yl)heptanoyl]piperidine-3-carboxamide 4-N-[(1S)-2-(dimethylamino)-3-(2,3-dimethylindazol-5-ylidene)cyclopenten-1-yl]-2-N-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]pyrimidine-2,4,6-triamine 2-[4-(2,6-difluorophenyl)pyrrolidin-3-yl]-7-methoxyimidazo[1,2-a]pyridine 2-amino-3,4-dihydronaphthalene-1,6-disulfonic acid (4-azidophenyl)-methoxycarbamic acid (2Z)-N',3-diethyl-2-[3-(methoxymethylidene)-4H-1,4-benzoxazin-7-yl]buta-2,4-dienimidamide 4-[7,9-dimethyl-8-(2-methylphenyl)-1,3,6,2-dioxadiazonine-2-carbonyl]-N-[4-(2H-tetrazol-5-ylmethoxy)phenyl]piperidine-1-carboxamide 2-[5-bromo-2,4-bis(phenylmethoxy)phenyl]-1-bromoethanone [7-[3,5-bis(trifluoromethyl)phenyl]-4-(methoxymethoxy)-3,9-dimethylidenexanthen-2-ylidene]cyanamide 1-methyl-3,7-dihydropyrrolo[2,3-f]indole-6-sulfonic acid 4-(2,3-dihydropyrrolo[1,2-a]indol-5-yl)-N'-hydrazinylidenethieno[3,2-b]pyridine-7-carboximidamide 4-[2-hydroxypropyl(phenylcarbamothioyl)amino]butanamide 6-[2,3-dihydroxypropyl(phenacyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 2-fluoro-1,8-dioxoanthracene-9-carboxylic acid 1-(4-fluorophenyl)sulfonyl-N,2,3,5,6,7-hexahydro-s-indacene-4-carboxamide [2-bromo-3,5-bis(trifluoromethyl)phenyl]boronic acid ethane;4-[(2S)-3,3,7-trimethylnonan-5-yl]-1,2-bis[(2-methylpropan-2-yl)oxy]benzene 6-N,2-dimethyl-4-N-[(2R)-1-naphthalen-2-ylbutan-2-yl]pyrimidine-4,6-diamine 5-(diethoxyphosphorylmethyl)-1,2,3-trimethoxybenzene 2-[4-(1,1-diphenylethyl)piperazin-1-yl]-N'-(3-methoxyphenyl)-2-oxoacetohydrazide 3-(2,4-dimethylphenyl)sulfanylpropanal 3-(5,6-diethylbenzimidazol-2-ylidene)-1H-indol-2-one 3-cyclopropylimino-1',4-dimethylspiro[1H-quinoxaline-2,3'-piperidine]-6-ol 3-methyl-2,6-bis(4-phenylpyridin-1-ium-1-yl)pyrimidine [3-(2-chlorophenyl)-1,5-dimethylpyrazol-4-yl]-[3-hydroxy-3-(triazol-1-ylmethyl)piperidin-1-yl]methanone 2-chloro-N-cyclopropylsulfonyl-6-fluorobenzamide 5-[1-(azidomethyl)cyclobutyl]oxypyridine-2,3-diamine 1-[1-(4-acetylphenyl)ethenylamino]-3-naphthalen-2-ylurea 2-[4,5-dichloro-1-[(3R)-pyrrolidin-3-yl]benzimidazol-2-yl]sulfanylacetic acid N-[4,5-dihydroxy-1-(2H-pyrimidin-5-yl)pentan-3-yl]formamide 2-(4-ethylphenyl)-6,7-dihydro-1H-[1,3]thiazolo[5,4-f]benzimidazole 1-[3,5-bis(trifluoromethyl)phenyl]sulfonyl-2-(3,4-dichlorophenoxy)-3-[(3-fluoropyridin-2-yl)oxymethyl]-3-hydroxypropane-1-sulfonic acid 1-[2-(2,3-dihydro-1H-inden-2-ylamino)pyrimidine-5-carboximidoyl]-6-pyridin-2-yl-7,8-dihydro-3H-imidazo[4,5-c]azepin-2-one 6-[4-(4-fluorophenyl)butanoylamino]pyridine-2-carboxamide (2S)-2,7-diamino-3-oxo-1,5-bis[(4-phenylbenzoyl)oxy]octanoic acid 1-[(4-methoxyphenyl)methyl]piperidine;2,3,5,6-tetrafluorobenzoic acid [4-fluoro-3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonyl)phenyl]methylcarbamic acid 1-butyl-2-chloro-3-[4-(trifluoromethoxy)phenyl]sulfonylbenzene 2-chloro-N-(5-hydroxy-9,10,11-trioxonaphtho[2,3-f][1]benzofuran-8-yl)acetamide 4-(4-aminophenoxy)-3,5-ditert-butylphenol 2-[(3S)-5-(4-chlorophenyl)-1,1-dioxothiolan-3-yl]guanidine 2-cyclobutylsulfanyl-4-methylpyrimidine (3S,5R)-N-[2-methoxy-4-(4-oxo-1H-pyridin-2-yl)phenyl]-7-(4-methoxyphenyl)-6-oxo-2-thia-7,11-diazatricyclo[6.3.1.04,12]dodeca-1(11),8(12),9-triene-3-carboxamide 1-[2-(2,5-dimethylpyrrol-1-yl)ethyl]-N'-hydroxy-1,2,4-triazole-3-carboximidamide ethane;3-(4-methoxyphenyl)sulfanylthiophene 2-(N-pyridin-3-ylanilino)octanoic acid [(4-fluorophenyl)methylamino]thiourea 5-[6-(1-ethoxyethenyl)pyridin-3-yl]oxy-N-methylsulfonyl-2,3-dihydroindole-1-carboxamide 3-(2,4-dihydroxyphenyl)-5-[1-(2,6-dihydroxybenzoyl)piperidin-4-yl]pyrazole-1-carboxamide (3R)-4-cyclopropyl-1'-methylspiro[2,7-dihydro-1H-imidazo[1,5-a]pyridine-3,4'-piperidine] 1-benzylsulfanyl-3-diazourea (7-methyl-2,3-dihydropyrido[4,3-b][1,4]oxazin-5-ium-6-yl)methanol 1-(8-phenylmethoxynaphthalen-2-yl)propan-2-one [3-(methylamino)phenyl]-morpholin-4-ylmethanone 4-[3-(3,5-dichlorophenyl)-1H-pyrazol-5-yl]-N'-[2-(3-ethoxyphenyl)ethyl]benzenecarboximidamide 5-(cyclopentylmethyl)-2-[4-(difluoromethoxy)-3-methoxyphenyl]-1,3-thiazole 6-[2,6-dichloro-4-(trifluoromethyl)phenyl]cyclohexa-1,5-diene-1-carboxylic acid 5-fluoro-1-methyl-3-[4-(trifluoromethoxy)phenoxy]pyrazole N-[(3-acetamidophenyl)methyl]-2,3-difluorobenzenesulfonamide 1-(3,4-dihydronaphthalen-2-yl)ethanone N-[3-(2,6-dimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]propanamide (3R)-N-[(4,6-dimethylpyridin-2-yl)methylidene]-1-[2-(2H-tetrazol-5-yl)phenyl]pyrrolidine-3-carboxamide 1-[2-(4-bromophenyl)pyrrolidin-1-yl]-3,3-dimethylbutan-1-one 1-[[2-(7-chloroquinolin-4-yl)-3,4-dihydro-1H-isoquinoline-6-carbonyl]amino]cyclohexa-2,4-diene-1-carboxylic acid N-[(E)-4,5-dimethylhept-1-enyl]methanimine;N-[3-fluoro-2-[3-(piperidine-1-carbonylamino)-6,7-dihydrocyclopenta[b]pyridin-5-yl]phenyl]formamide [1-[[2-ethyl-4-(6-fluoropyridin-3-yl)phenyl]methyl]pyrazol-4-yl]carbamic acid 3-[(4R)-1,6-dimethylpiperidin-2-yl]-5-fluoro-N'-hydroxybenzenecarboximidamide 7-[2-(3,4-dimethoxyphenyl)ethyl]-6,8-bis[3-hydroxy-2-(4-propylpiperazin-1-yl)propoxy]-5H-thieno[2,3-c]quinolin-9-one 4-(3,5-dibromophenyl)sulfinyloxane 2-(3,5-dichloropyridin-2-yl)-N-[[4-fluoro-3-methoxy-2-(1,1,2-trifluoroethylsulfanyl)phenyl]methyl]-5-methylsulfonylaniline 4-[[3,5-difluoro-2-(hydroxymethyl)phenyl]methyl]morpholine-3-carboxamide 5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-4-carboxylic acid (E)-3-[4-(4-aminophenyl)-2,3-dimethylpyridin-1-ium-1-yl]prop-1-en-1-amine N-[(2S)-1-aminopropan-2-yl]-4-[6,7-dimethoxy-2-(morpholine-4-carbonyl)quinolin-4-yl]benzamide (1S)-1-(2,4-dichlorophenyl)-3-ethylhexan-1-amine 1-[2-(methylamino)ethyl]-N'-[2-[4-[5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl]phenoxy]acetyl]piperidine-4-carbohydrazide;hydrochloride 3-[4-(2-hydroxypropoxy)cyclohexyl]-6H-benzo[c]chromen-1-ol [2-amino-5-(4,5-dimethylthiophen-2-yl)pyrimidin-1-ium-4-yl]-[3-(2H-tetrazol-5-yl)cyclohexa-2,4-dien-1-ylidene]azanium 4-cyclohexa-1,5-dien-1-yl-2-[2-(3-fluorophenyl)ethoxy]-6,7-dimethoxyquinazoline 1-cyclopentyl-7-[(3,4-dimethoxyphenyl)methylamino]-5,6,7,8-tetrahydronaphthalene-2,3-diol 4-[3-(2,6-difluorophenyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 5-fluoro-2-N-(6-fluoropyridin-3-yl)pyrimidine-2,4-diamine 1-[4-methyl-3-(trifluoromethyl)phenyl]-2,5-dihydrotetrazol-5-amine ethane;N-[(E)-1-[3-[ethyl(propanoyl)amino]phenyl]pentylideneamino]benzamide 2-[(E)-(4-chlorophenyl)methylideneamino]oxyacetic acid;4-methylbenzenesulfonic acid 6-(4-bromophenyl)-3-(2-hydroxyethylsulfanylmethyl)-7H-[1,2,4]triazolo[3,4-f][1,2,4]triazin-8-one 2-(4-iodophenyl)-3,6-dimethylpyrazine (Z,6S)-N'-benzyl-6,7,8-trimethoxy-2-oxo-4-phenyloctanediamide [2-fluoro-4-(6-fluoro-1H-indole-3-carbonyl)phenyl]carbamic acid 4-[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazol-3-amine 1-[2-(5-azido-6-chloropyridin-3-yl)-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl]-N,N-dimethylmethanamine 1,4-dimethyl-2-[(E)-pent-3-en-2-ylidene]-5-prop-1-ynylnaphthalene 2-[(E)-(4-fluorophenyl)methylideneamino]-N-[3-(1H-imidazol-5-yl)propyl]-3-oxo-[1,2,4]triazolo[4,3-a]pyridine-8-carboxamide 4-amino-1-[2,6-difluoro-3-(trifluoromethyl)phenyl]-8-ethoxy-7H-imidazo[4,5-f]quinazoline-9-carboxylic acid N-[2,5-dimethyl-4-(2-oxoimidazolidin-1-yl)phenyl]cyclopropanecarboxamide 1-[2-(2,4-difluorophenyl)acetyl]-N-methylpyrrolidine-3-sulfonamide 4-azido-2-(2,6-dichlorophenyl)phenol N-[4,5-bis(ethenyl)thiophen-2-yl]benzenecarboximidate 2-[5-(dimethoxymethyl)-1-benzofuran-3-yl]-N,N-diethylethanamine 3-[1-[1,2,4-triazol-1-yl(oxan-4-yl)amino]ethyl]benzonitrile 2-(3,5-dimethylphenyl)imino-1,4-dihydro-3,1-benzoxazin-6-amine 4-[1-(2-propan-2-ylsulfanylphenyl)benzimidazol-2-yl]phenol 3-(2-cyclopropylpyrimidin-5-yl)imidazo[1,2-a]pyrazine 1-[(2,3-difluoro-4-methoxyphenyl)methyl]-7-iodo-N-methylpyrrolo[3,2-b]pyridine-5-carboxamide 1-(5,6-diphenylpyridazin-3-yl)-2-(1-methoxybutan-2-ylideneamino)guanidine 2-[4,5-dichloro-N-(1-phenylethyl)anilino]acetamide 6-[2-(benzylamino)pyrimidin-5-yl]-1,3,4,5-tetrahydro-1,5-benzodiazepin-2-one 6-bromo-4,8-dimethyl-7H-carbazole 6-[1-[2,4-di(propan-2-yl)phenyl]tetrazol-5-yl]-N-methyl-1H-benzimidazol-2-amine (4-azidopyrimidin-5-yl)-[3,4,5-tris(trifluoromethoxy)phenyl]methanone [3-(methylamino)-5-thiophen-2-ylpyridin-4-yl]hydrazine (2S)-N'-[3,5-bis(trifluoromethyl)phenyl]-1-chlorobutanediamide 5-bromo-4-N-(3,6-dihydro-2H-pyran-5-yl)-2-methoxypyrimidine-4,6-diamine (1S,2R)-3-methylspiro[5-propan-2-ylsulfanyloxy-1,2,3,4-tetrahydronaphthalene-2'-piperidine]-1'-carboxylic acid 1-[2,6-di(propan-2-yl)phenyl]-3-[(E)-(5-methoxy-1H-indol-3-yl)methylideneamino]thiourea N-[4-amino-1-(6-hydroxy-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-2-yl)-3,4-dioxobutan-2-yl]-4-pyridin-4-ylsulfonylpiperazine-1-carboxamide 2-[(E)-but-1-enyl]-4,6-dimethyl-3-[4-(methylamino)phenyl]cyclohexa-2,4-diene-1-carboxamide;ethane 7-[(4-methoxyphenyl)methyl]-8-phenyl-9H-purine 6-(5-chlorothiophen-2-yl)-4-[4-(dimethylaminosulfanyl)phenyl]iminopyrido[3,2-c]pyridazine-1-carboxamide 2,4-dichloro-1-[(Z)-3-methylbut-1-enyl]benzene 3-[2,4-bis(trifluoromethyl)phenyl]-1-[2,6-dichloro-5-(1-iodoethylamino)pyridine-3-carbonyl]imidazolidin-4-one 5-(6-chloropyridin-3-yl)sulfanylpentanamide 3-[4-(cyclohexylmethoxy)phenyl]-5,7-diethynyl-2H-imidazo[4,5-f]benzimidazole N-(2,3-dihydro-1H-inden-5-yl)-2-methoxybenzamide;N-methylpentan-2-amine 4-(3-chloropyridin-2-yl)oxypiperidine-1-carboxylate N-[(2S)-2-aminopropyl]-2,4-difluoro-5-[6-[(1-phenylcyclopentanecarbonyl)amino]pyridazin-3-yl]benzamide 5-bromo-4-N-[(Z)-3,6-dimethylhept-2-en-4-ynyl]-2-N-[4-[3-methoxypropyl(methyl)amino]phenyl]pyrimidine-2,4-diamine 6-(2,4,5-trichlorophenyl)benzo[c]chromene 2,4-dihydroxy-6-methylbenzenesulfonate;tin(4+) 5-chloro-6-(2,4-difluorophenyl)-N-[4-(3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclohexyl]pyridine-3-carboxamide N-azido-2-hydroxy-5-[(5-methylfuran-3-carbonyl)amino]benzamide N-[(1S,2R)-2-hydroxycyclohexyl]-7-(methylamino)-5-[1-(2-oxo-2-piperidin-1-ylethyl)pyrrolo[3,2-b]pyridin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 2-[2-(3,5-dimethoxyphenyl)ethyl]-4,6-dimethylbenzenesulfonate [6-(difluoromethoxy)pyridin-3-yl]-[2-methyl-4-[[5-(trifluoromethyl)pyrazol-1-yl]methyl]phenyl]methanone 2-bromo-5-[(3-chlorophenyl)sulfonylamino]-N-hydroxybenzamide 5-[(E)-6-hydroxy-6-phenylhex-2-en-4-ynyl]benzene-1,3-diol ethane;3-[2,4,6-trichloro-N-(1,3-thiazol-5-ylmethyl)anilino]propanenitrile 3-amino-6-(1,3-benzothiazol-2-yl)pyrazine-2-carboxamide [4-(3,7-dimethyloctoxy)phenyl]boronic acid 6-[3-[4-(3,4-dimethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]pyridazine-3-carbonitrile N-[3-[(2R)-4,4-difluoro-2-methylpyrrolidine-1-carbonyl]-4-fluorophenyl]ethanesulfonamide 4-[6-(3,5-dimethylpyrazol-1-yl)pyrimidin-4-yl]morpholine 3-azido-2,6-diphenylphenol 3-(2,6-difluorophenyl)-5-[[(3R,4S,5R)-3,4,5-trihydroxy-4-methyloxan-2-yl]amino]cyclohexa-2,4-diene-1,2-dione N-(4,6-dimethylcyclohexa-2,4-dien-1-ylidene)benzenesulfonamide N-benzyl-2-[7-methoxy-5-(4-methoxyphenyl)sulfonyl-1,3-dihydroisoindol-2-yl]acetamide N-azidosulfonylpyrazolo[1,5-a]pyrimidine-3-carboxamide 4-(4-fluorophenyl)-2,5-dimethylfuran (Z)-3-[4-fluoro-2-methoxy-5-[(1-propan-2-ylpyrazole-4-carbonyl)amino]phenyl]-2-(2H-tetrazol-5-yl)prop-2-enoic acid N-[2-(4-phenylmethoxyphenoxy)propyl]butanamide (1E)-1-[3,5-dimethoxy-4-(6-piperidin-1-ylhexoxy)phenyl]propan-2-one 4-(7-azidonaphthalene-2-carbonyl)oxybenzenesulfonic acid 3-[6-[[(1S)-4,4-difluorocyclohexyl]amino]-2-methylpyrimidin-4-yl]-1H-indole-5-carboxamide 2-ethylsulfanyl-6,7-dihydrothieno[3,4-d]pyrimidin-5-one 3-methyl-1,4-diphenylbutane-2,2-diol 1-[4-[2,3-difluoro-6-methyl-5-(methylideneamino)phenyl]piperazin-1-yl]ethanone 3-(2,4-dichlorophenyl)-6-[(dimethylamino)methoxy]-1H-1,5-naphthyridin-4-one N-[(2R)-1-[4-[5-cyano-6-(difluoromethoxy)pyridin-3-yl]-2-fluorophenyl]propan-2-yl]-2-[3,4-dioxo-2-(propanoylamino)-7,8-dihydro-6H-cyclopenta[e]indol-1-yl]acetamide 5-(3,4-dimethoxyphenyl)-2-(5-ethylsulfonylpyridin-2-yl)-6H-1,3-thiazine N-[2,4-bis(2H-benzotriazol-5-yl)phenyl]naphthalene-1-carboxamide 2-hydroxy-4-[(1,3,5-trimethylpyrazol-4-yl)sulfonylamino]benzoic acid 5-[[4,7-dimethyl-9-(2-oxopropyl)-6H-pyrazino[1,2-a]quinoxalin-8-yl]oxy]pyridine-3-carbonitrile 6-[4,7-dimethyl-9-(3,4,5-trifluorophenyl)fluoren-2-yl]hexanoic acid 2-(4-chlorophenyl)imino-5-[(3,5-dimethylpyrrol-1-ium-2-ylidene)methyl]-3-ethoxy-6-hydroxypyrimidin-4-one 1-amino-3-[4-[(2E)-2-[6-(dimethylamino)pyridin-3-yl]oxyiminopropanoyl]anilino]propane-1-sulfonic acid;ethene N-(2,5-dichlorophenyl)-1H-indole-2-carboxamide 5-[2-(4,6-diphenylpyrimidin-2-yl)phenyl]quinoline N-(2,4-dimethylphenyl)-2-[6-(2-methoxyethoxy)pyridin-3-yl]ethanesulfonamide ethane;1-(2-propan-2-ylphenyl)-4,5-dihydroimidazole N-[(1S)-2,3-dihydro-1H-inden-1-yl]propanamide [(3aR,7aS)-2-[(3-methylphenyl)methyl]-1,3,4,6,7,7a-hexahydropyrano[3,4-c]pyrrol-3a-yl]methanol;2,2,2-trifluoroacetic acid 4-(5,6-dimethoxypyridin-3-yl)-2-[6-[(3R,5S)-3,5-dimethylpiperazin-1-yl]pyridazin-3-yl]-1H-benzimidazole 4-N,6-dimethyl-2-N-[(5R)-5-methylheptan-3-yl]pyrimidine-2,4-diamine (2S,6R)-4-[5-(difluoromethoxy)pyridin-2-yl]-N,2-dimethyl-6-(3-oxo-1H-isoindol-2-yl)piperidine-3-carboxamide 2-azidosulfanyl-3-(trifluoromethoxy)thiophene 4-(2,6-difluorophenyl)-5-hydroxy-3-propylthiophen-2-one 3-(3,4-dihydroxyphenyl)-N-ethylbenzamide 5-(4-aminophenyl)-3-bromo-2-methoxyaniline (2R)-1,4-dimethyl-2-[[2-[3-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]-2H-pyrazolo[3,4-b]pyridin-5-ylidene]acetyl]amino]piperazine-2-carboxylic acid 2-[(2E,4Z)-hexa-2,4-dien-3-yl]-4-methyl-5-phenylpyridine N-(2,6-dichlorophenyl)-4-[5-(3-hydroxyphenyl)thiophen-3-yl]-1,3-thiazol-2-amine;hydrochloride 4-(6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl)-N-[3-(trifluoromethoxy)phenyl]piperidine-1-carboxamide 2-[(4S)-7-(5,6-dichlorobenzimidazol-1-yl)-3,4-dihydro-2H-chromen-4-yl]-2-phenoxyacetonitrile 1-[3-(cyclopropylmethoxy)phenyl]-2,4-dioxopyrimidine-5-carbonitrile 1-[4-[bis(2-hydroxyethyl)amino]butylsulfonyl]-3-[(E)-1-[4-(trifluoromethoxy)phenyl]propan-2-ylideneamino]thiourea (2R)-1-[4-[[8-(methoxymethyl)-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]pyrazol-1-yl]propan-2-ol 1,5-dibutylnaphthalene (2Z,5Z)-1-ethyl-7-[1-(2-fluoroethoxymethyl)-3,6-dihydro-2H-pyridine-4-carbonyl]-4-hydroxy-2-(methylideneamino)-8-(5-propan-2-ylpyridin-2-yl)octa-2,5,7-trien-1-one (Z)-3-(2,6-dichlorophenyl)-2-methylprop-1-en-1-amine 4-[(2-aminopyridin-3-yl)methoxy]benzamide (2S)-N-[(1R,5S)-8-amino-3,6-dibicyclo[3.2.0]heptanyl]-4-[(2-ethoxyphenyl)methyl]-2-(methanesulfonamido)butanamide;hydrochloride 3-[2-(5-ethylpyridin-2-yl)ethynyl]-N-propan-2-ylaniline 6,7-dihydro-4H-[1,2]oxazolo[5,4-c]pyridine-5-carbonyl(3-hydroxypyrrolidin-1-yl)methanesulfonamide ethane;4-fluoro-3-methylpyridine;2,8,9,10-tetrahydropyrimido[5,4-h][1,6]naphthyridin-7-one 6-bromo-N-[1-[[4-(trifluoromethyl)phenyl]methoxy]naphthalen-2-yl]pyrimidin-4-amine 3-[(2-chloro-4-fluorophenyl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine;2,2,2-trifluoroacetic acid 4-(1,3-dioxoisoindol-2-yl)benzamide N-benzyl-1,3-dihydroxy-2-propan-2-ylisoindole-5-carboxamide 2-[4-azidooxy-1-(benzenesulfonyl)pyrrolo[3,2-b]indol-3-yl]acetamide N-(4-chlorophenyl)-2-[(6R)-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 2-(3-chloro-4-fluorophenyl)-N-methylsulfanyl-6-nitrobenzimidazole-1-carboxamide 3-[[4-[(2R,3R)-1-(2,6-dimethylphenyl)sulfonylpyrrolidin-2-yl]benzoyl]amino]propanoic acid 4-methyl-2,6-di(propan-2-ylidene)cyclohexa-1,3-diene;osmium(2+);tetraphenylboranuide 1-[3-chloro-4-(trifluoromethyl)phenyl]butan-2-one 4-amino-6-[[1-(3,5-dimethylphenyl)-2-hydroxyindol-3-yl]methylideneamino]quinoline-3-carboxylic acid 3-[7-bromo-4-[(4-hydroxycyclohexyl)amino]quinazolin-2-yl]-4,6-dihydro-1H-cyclohepta[b]pyrrole-5-carboxylic acid 3,5-dimethyl-N-[(2R)-1-phenylpropan-2-yl]aniline 2-(N-methylanilino)-5,6,7,8-tetrahydronaphthalene-1,4-dione 2-(5-chlorothiophen-2-yl)pyridine 2-benzamido-3-(4-bromophenyl)propanoic acid 1-azido-3-chloro-2,4-dimethoxybenzene 7-amino-3-azidoisoquinoline-4-carboxamide 4-methyl-N-[1-(6-methyl-2H-thiopyran-3-yl)ethyl]-5,6-dihydronaphthalene-2-carboxamide 4-[(5R)-7-(3,4-dichlorobenzoyl)-2-[(4S)-1-ethanimidoylazepan-4-yl]-6-fluoro-8-methoxy-4-oxo-3,5-dihydropyrrolo[2,1-f][1,2,4]triazin-5-yl]-N-methylbenzamide 2-[(3R,4S)-3-[4-amino-3-(trifluoromethyl)phenyl]-1-(cyanomethyl)piperidin-4-yl]oxy-5-isocyanobenzonitrile 6-chloro-3-methylsulfanyl-N-(2,4,6-trifluorophenyl)imidazo[1,5-a]pyrimidin-8-amine 1-[5-(2,4-dimethoxyphenyl)-3,6-dihydro-2H-pyridin-1-yl]ethanone 3-[[2-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)pyrrolidine-1-carbonyl]amino]propanoic acid 4-chloro-5-(2,3-dihydro-1H-indol-6-ylamino)sulfanyl-2-fluorobenzoic acid N-ethenylsulfonyl-N-(2H-tetrazol-5-yl)benzenesulfonamide 3-(4,6-dimethylpyridin-2-yl)pyridine;ethane N-(2,3-dihydro-1H-isoindol-5-yl)-4-methoxybenzenesulfonamide;ethane N-(3,4-dichlorophenyl)formamide;3-[1-hydroxy-5-methoxy-2-(2-sulfamoylethyl)-2H-pyridin-6-yl]benzoic acid 2-(4-azido-3,5-dichlorophenyl)propanal (Z)-N,2-bis[(E)-(3-bromophenyl)methylideneamino]oxy-4,4,5,5-tetrafluoropent-2-enamide 6-amino-4-methyl-4-[3-(3,4,5-trifluorophenyl)phenyl]-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile [2-amino-4-(cyclohexylmethylamino)phenyl]-dimethoxyphosphanium [4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]urea 5-chloro-2,4-dimethoxy-N-[2-oxo-2-(1-propyltriazol-4-yl)ethyl]benzamide (4-propan-2-ylsulfonylphenyl)methanethiol 4-bromo-1,2,3,5-tetraethylbenzene 4-amino-2-(3,5-difluorophenyl)butanal 2-amino-4,5-bis(3-bromophenyl)-4H-pyran-3,5-dicarbonitrile (5Z)-2-sulfanylidene-5-[[4-(4,4,7,7-tetramethylnonoxy)phenyl]methylidene]imidazolidin-4-one 1-methyl-3-[4-(2-methylphenyl)piperazin-1-yl]benzimidazol-2-one 1-azidooxy-2,4-bis(trifluoromethyl)benzene 4-chloro-1-[2,6-difluoro-3-(trifluoromethyl)phenyl]butan-1-one N-[(2S,3R)-4,6-dimethyl-7-oxo-1-phenyloctan-3-yl]-4-methoxypyridine-2-carboxamide 4-[4-[[2-(hydroxymethyl)pyridin-3-yl]amino]imidazo[1,5-a]pyrazin-8-yl]benzene-1,2-diol 3-[4-(methoxycarbonylamino)-1,2,5-thiadiazol-3-yl]propanoic acid 2-(4-chlorophenyl)-2-methoxy-N,N-dimethylethanamine N-[2-[[4-(benzimidazole-1-carboximidoyl)benzoyl]amino]ethyl]-4-phenylbenzamide 2-[2-azido-1-(benzenesulfonyl)ethyl]pyridine 2-(5,7-dimethyl-4-phenylquinolin-2-yl)acetic acid 2-(3,4-dichlorophenyl)-1-[6-fluoro-4-(2H-pyrimidin-1-ylmethoxy)-9H-pyrimido[4,5-b]indol-8-yl]ethanone 4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxyaniline 2-azido-7,8-dimethyl-3H-purino[9,8-a]pyridin-4-one 2-(2,4-dichloroanilino)-5-methylthiophene-3-carboxamide 4-[(2E,4Z)-5-amino-3-imino-6-methylideneocta-2,4-dienyl]-N-[(6-chloropyridin-3-yl)methyl]benzamide 4-[3-hydroxy-3-(triazol-1-ylmethyl)piperidine-1-carbonyl]-7,8-dihydro-6H-cyclohepta[b]furan-2-carboxamide 4-[1-(cyclopropylmethoxy)ethenyl]benzoic acid 4-[1-(3,5-difluorophenyl)imidazol-2-yl]piperidine;ethane 2-[(3S,4R)-1-acetyl-4-hydroxypiperidin-3-yl]-N-pyridin-3-ylacetamide 3-amino-1-[4-(4,5-dihydroimidazol-1-yl)piperidin-1-yl]-2-methoxy-2-methylpropan-1-one 5-chloro-1H-imidazo[4,5-b]pyridine;5-chloro-N-[(2R)-3-oxocyclopentyl]spiro[1H-indole-3,4'-piperidine]-2-carboxamide 1-azidosulfanylnaphthalene 3-[[4-[(E)-2-[6-fluoro-1'-[(4R)-4,5,5,5-tetrafluoropentanoyl]spiro[1H-indole-3,4'-piperidine]-2-yl]ethenyl]phenyl]methyl]imidazolidine-2,4-dione N-methylformamide;4-[2-[4-[(4-nitrophenoxy)carbamoyl]cyclohexyl]ethoxy]benzamide 2-[4-(8-bromoquinoxalin-5-yl)piperazin-1-yl]acetamide 2-chloro-4,5,6-triethoxy-3,4-difluoro-N-phenylaniline 1-azidooxy-2,3,4,5,6,7-hexamethylnaphthalene 1-[(2S,4R)-1-(1H-indole-3-carbonyl)-4-methoxypyrrolidin-2-yl]ethanone 2-(4-fluorophenyl)-3-[(Z)-(6-hydroxynaphthalen-2-yl)methylideneamino]quinazolin-4-one N-[4-[(3S)-1-(2,6-difluorophenyl)pyrrolidine-3-carbonyl]pyridin-2-yl]cyclopropanecarboxamide N-[4-[(3-cyanophenyl)sulfonylamino]phenyl]quinoline-2-carboxamide (6R,9S)-2-methylsulfanyl-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one N-(2-fluoropyridin-4-yl)-3-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)pyrrolidine-1-carboxamide N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-yl)propyl]isoquinoline-8-carboxamide 5-(6-azido-3,3-dimethylhexan-2-yl)pyridine-2,3-diamine 5-(2,6-dimethoxyphenyl)imino-3H-1,3,4-oxadiazole-2-thione 5-azidooxy-3-(2,4-difluorophenoxy)-1H-pyrazole 1-[5-(1,3-benzothiazol-2-yl)-6-methoxypyridin-3-yl]piperidine-4-carboxylic acid 3,4-difluoro-2-(2-fluoro-5-methylphenyl)aniline N-(1,3-benzothiazol-2-yl)-4-[N'-[4-(trifluoromethoxy)phenyl]carbamimidoyl]benzamide 1-(4-chlorophenyl)sulfonyl-6,7-dimethoxyquinolin-4-one 1-[(4Z)-3,5-dimethylidenehepta-1,4-dien-2-yl]-6,6-diphenylpiperazine;1H-indole 2-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butoxy]quinoline 2-(6-methoxynaphthalen-1-yl)furan;dihydrochloride 4-[2,6-dichloro-3-(methyliminomethyl)pyridin-4-yl]oxy-N,2-diethylaniline 4-[2-[(3R,5S)-3,5-dimethylpiperazin-1-yl]ethoxy]-N'-[3-[1-(5-ethoxy-6-fluoropyrimidin-4-yl)piperidin-3-yl]prop-1-ynyl]benzenecarboximidamide 3-(3-cyclopropyl-2H-pyridin-1-yl)-N,N-dimethylaniline [3-(hydroxymethyl)azetidin-1-yl]-[2-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)-1,3,4,5-tetrahydropyrido[4,3-b]indol-8-yl]methanone [3-[2-(methylamino)propanoylamino]phenyl]azanide (2S,3R)-N-(4-amino-1H-pyrazolo[3,4-b]pyridin-5-yl)-2-(2,4,6-trifluorophenyl)oxane-3-carboxamide (3-fluorophenyl)-[8-methyl-5-(6-methylpyrazin-2-yl)-3,4,6,7-tetrahydroimidazo[1,5-a]pyridin-1-yl]methanone 2-azido-6-fluoro-4,7-bis(trifluoromethyl)-1H-benzimidazole 2-[4-(3,6-dimethylpyrazin-2-yl)pyridazin-1-ium-1-yl]ethanesulfonic acid 7-hydroxy-1,2-dihydroimidazo[4,5-f]indazole-3-carboxylic acid 1-(2-methoxynaphthalen-1-yl)piperidine;hydrochloride 2-[[5-[4-(3,5-dichloroanilino)-7,8-dihydroquinazoline-6-carbonyl]thiophen-2-yl]methyl-methylamino]acetic acid (E)-5-[3-methoxy-4-(phenylcarbamoylsulfamoyl)phenyl]-2-methylpent-3-enoic acid 3-[(1R)-5-bromospiro[2H-indene-3,4'-piperidine]-1-yl]propan-1-ol 2-[(4,5-dimethoxycyclohexa-1,3-dien-1-yl)amino]-6-methyl-8-propan-2-ylpteridin-7-one 4-(1,3-benzodioxol-5-ylmethoxy)benzenecarboximidamide N-[(3R)-1,2,3,4-tetrahydroisoquinolin-3-yl]carbamate N-[(2,4-dichlorophenyl)methyl]-2-methoxy-4-(trifluoromethyl)benzamide 5-cyclohexylimino-4-[5-methoxy-6-(3,4,5-trifluorophenyl)pyridin-2-yl]thiophene-2-carboxylic acid 4-(3,6-dichlorocarbazol-9-yl)benzenecarboximidamide 6-chloro-N,3-dimethyl-4H-thiochromeno[4,3-d]pyrimidine 3-[(4S)-2,5-dioxopyrrolidin-1-yl]sulfonyl-N-(2-methoxyphenyl)benzamide N-[4-(2,6-difluorophenoxy)-3-methylphenyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine 5-[(2,4-dihydroxyphenyl)methyl]benzene-1,3-diol 5-fluoro-2-methoxy-4-[(3R,4S)-1-methyl-4-pyridin-3-ylpyrrolidine-3-carbonyl]benzonitrile N-(3,4-dimethylphenyl)-4-[4-fluoro-1-methyl-2-[6-(trifluoromethoxy)benzimidazol-1-yl]benzimidazol-5-yl]pyrimidin-2-amine 2-amino-5-(trifluoromethyl)benzenethiol;N-[3-chloro-1-[4-[(dimethylcarbamoylamino)methyl]phenyl]sulfonylindazol-6-yl]cyclopropanecarboxamide 4-[4,5-dimethyl-3-(1H-pyrrolo[2,3-b]pyridin-4-yl)furan-2-yl]morpholine 5-(methoxycarbonylamino)benzene-1,2,3,4-tetracarboxylic acid 2,3-diethoxyphenanthrene;1-[(4R)-4-methoxyoxolan-2-yl]-N-(2-phenylethyl)methanamine [2-hydroxy-3-methyl-5-(2,3,4-trihydroxy-6-methylphenyl)pentyl]phosphonic acid 6-[(2,4-dimethylphenyl)sulfanylamino]-N'-hydroxypyridine-2-carboximidamide 2-[4-(3-bromopropoxy)phenyl]benzotriazole (4R)-4-[4-fluoro-2,6-dimethyl-3-[(1S)-1-[(5Z)-7-methylidene-6-(trifluoromethoxy)cycloocta-2,5-dien-1-yl]ethoxy]phenyl]-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one 1-[7-(5-hydroxyquinolin-4-yl)oxyheptyl]pyrrolidine-2,5-dione 2-[(1Z,3E)-1-bromopenta-1,3-dienyl]naphthalene 4-[2,3-difluoro-6-(methylcarbamoyl)phenyl]-7-N-methyl-2-propan-2-ylindazole-3,7-dicarboxamide 1-[2,4-dichloro-3-(1H-indol-3-yl)quinolin-6-yl]-4-hydroxypiperidine-4-carboxylic acid 1-(2,4-dimethoxyphenyl)-N-[[1-[(3-ethyl-2H-indazol-5-yl)sulfonyl]piperidin-4-yl]methyl]pyrrolidine-2-carboxamide 2-[2,6-dimethyl-4-(trifluoromethyl)phenyl]-N'-hydroxyethanimidamide;ethane 2,3-bis(4-ethoxyphenyl)propanoic acid (3S,4R)-1-[(2R,3R)-5-cyano-3-fluoro-6-oxo-1-phenyl-2H-pyridin-2-yl]-4-(triazol-1-ylmethyl)pyrrolidine-3-carboxylic acid 1-[(3R,5S)-3-amino-7-methyl-4-oxa-6,14-diazatetracyclo[12.2.1.05,16.09,18]octadeca-1(17),10,12,15-tetraen-13-yl]ethanone 2-[N-(4-bromobutan-2-yl)-4,5-dimethyl-2-phenyldiazenylanilino]ethanol 2-[5,6-dichloro-4-(3,4,5-trimethoxyphenyl)pyridin-3-yl]-4H-1,3,4-oxadiazolidine;ethane;uranium(2+) (7R)-N-(2,4-dimethylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 1-[[3-(azidomethyl)phenoxy]methyl]naphthalene 3-(4-methoxyanilino)benzene-1,2-disulfonic acid N-[5-(azidomethyl)-2-nitrophenyl]-2,4-dimethoxybenzamide 2-[4-(2,6-dimethoxyphenyl)-5-(1H-indazol-5-yl)-1,2,4-triazol-3-yl]acetamide ethene;3-[4-[7-(2-methoxypyrimidin-5-yl)imidazo[1,2-c]pyrimidin-5-yl]pyrazol-1-yl]-N,N-dimethylcyclobutan-1-amine 5-[4-[2-(diethylamino)ethyl]piperazine-1-carbonyl]-3,7a-dihydroisoindol-1-one 4-(3-chlorophenyl)-1,6-dimethylcyclohexa-2,4-dien-1-amine 2-[(1S)-1-azidoethyl]-6,7-dimethoxy-3H-quinazolin-4-one 3-amino-5-(1-azidobutyl)benzaldehyde 2-[6-fluoro-3-methyl-1-(1H-pyrazol-4-yl)isoquinolin-7-yl]cyclopropane-1,1-dicarboxamide (NZ)-N-[1-(7,8-diethylquinolin-2-yl)-2,2,3-trimethylindol-6-ylidene]hydroxylamine 2-[1,2-diaminoethyl(3-methoxypropyl)amino]benzoate (2S,3R)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methoxy]-2-(1H-pyrazol-5-yl)oxane-3-carboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]-2-methoxybenzamide N-(2,4-dimethylphenyl)sulfonyl-1,3-thiazole-5-carboxamide 6-(4-cyclopropylphenyl)-N-[3-(difluoromethoxy)phenyl]-2H-pyrimidin-1-amine 3-[(3R,4S)-1-benzyl-3-hydroxypiperidin-4-yl]-N-methoxy-2H-indazole-5-carboxamide 5-(4,6-dicyclopropylpyrimidine-2-carbonyl)-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid;formic acid N-(6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)-1-methoxyisoquinoline-3-carboxamide (1R,3S)-1-[6-[4-ethyl-5-(trifluoromethyl)-1H-pyrazol-3-yl]pyridin-3-yl]-2,2,3-trimethylcyclopentan-1-amine 1-[5-(2-azidopropan-2-yl)pyridin-2-yl]ethanone 1-(4-azidocyclohexyl)oxy-3,5-dichlorobenzene (E)-3-(2,4-dichlorophenyl)-N-[(Z)-1-(4-hydroxy-6-oxocyclohexa-2,4-dien-1-yl)ethylideneamino]prop-2-enethioamide 6-[1-(4-azidooxycyclohexyl)oxyethenyl]-5,7,8-trimethoxyquinoxaline (1R)-2-[[5-chloro-2-hydroxy-4-methyl-3-(trifluoromethyl)phenyl]diazenyl]-N,N-dimethylacetamide 4-(1-benzylpiperidin-4-yl)phenol;ethane 5-[(1R)-1-azidoethyl]-3-methoxypyrazine (3E)-4-amino-3-[[4-fluoro-2,6-dimethyl-3-(trifluoromethoxy)phenyl]methylidene]azete-2-thione 1-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-ylmethyl)-4-(5-fluoro-2-methoxypyridine-4-carboximidoyl)piperidin-4-ol 5-(3,4-dihydro-2H-chromen-6-yl)-N'-hydroxypyridine-2-carboximidamide 1-[(2,6-dichlorophenyl)methyl]-3-(1H-indazole-5-carbonylamino)thiourea 2-[(3S)-1-[5-chloro-6-(3,3-difluoropyrrolidin-1-yl)pyridine-3-carbonyl]piperidin-3-yl]-7-(oxolan-3-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one (2E)-5,6-dihydroxy-1-phenylhepta-2,4-dien-3-one 6-chloro-N-ethyl-2,3-dimethoxyaniline;1-[4-(hydroxymethyl)piperidin-1-yl]propan-2-one N-[(3R,4S)-1-acetyl-4-methoxypyrrolidin-3-yl]-3-chlorobenzamide [4-(2,5-difluorophenyl)piperazin-1-yl]methanesulfonic acid 1-azido-2-(2-methylpropoxy)naphthalene 2-[[(3S)-1-(cyclopropanecarbonyl)pyrrolidine-3-carbonyl]amino]-9-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)nonanoic acid 4-amino-3,5-dimethylsulfonylpyridine-2-carboxylic acid N-methyl-3-(4-phenylpiperidine-1-carbonyl)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-2-carboxamide 2-[3-(4-aminophenoxy)phenyl]isoindole-1,3-dione (5S)-5-[2-hydroxy-3-[2-methyl-4-(oxan-2-yloxyamino)phenyl]sulfanylpropyl]imidazolidine-2,4-dione 4-[(7-azidooxy-9H-fluorene-2-carbonyl)amino]benzoic acid 1-(5-fluoro-2,4-dimethylphenyl)-3-[4-[4-[2-(methanesulfonamido)ethylsulfanyl]anilino]phenyl]urea 4-ethyl-2-(4-hydroxyphenyl)-6-oxo-1H-pyrimidine-5-carbonitrile 5-[(4-bromophenyl)methyl]-7-chloropyrrolo[2,1-f][1,2,4]triazin-4-amine 3-[1-(benzenesulfonyl)pyrrol-2-yl]sulfanylaniline 2-N,6-N-bis(3,4-dimethoxyphenyl)-9H-pyrimido[5,4-b]indole-2,6-diamine N-[3-[2,4-bis(phenylmethoxy)-5-propan-2-ylphenyl]propylidene]hydroxylamine (6-bromoimidazo[1,2-a]pyridin-2-yl)-(oxan-4-yl)methanone 2-(3,5-difluorophenyl)-7-methyl-6-[4-[2-[1-(oxetan-3-ylamino)propan-2-ylideneamino]ethoxy]benzoyl]-N-[2-oxo-2-(1-pyrimidin-2-ylpiperidin-4-yl)ethyl]-3H-isoindole-1-carboxamide N-(3,4-dichlorophenyl)-2-[(6S)-2-methyl-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 6-(2-chloro-4-nitrophenyl)-3-[1-[(5Z,7E)-5,8-difluoroocta-5,7-dienyl]piperidin-4-yl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole 2-[3-azido-6-(4-butanoylpiperazin-1-yl)pyridin-2-yl]acetonitrile N-[(1S,3R)-3-[2-acetamidoethyl(methylsulfonyl)amino]cyclohexyl]thiophene-2-carboxamide 3-benzylsulfonyl-4,5-difluorobenzonitrile 6-(4,5-dimethylcyclohexa-1,3-dien-1-yl)-3-[2-hydroxy-2-(5-sulfanylidene-6H-isoquinolin-7-yl)propyl]pyrimidin-4-one N-[4-(4-aminophenoxy)pyridin-2-yl]acetamide ethane;4-[(E)-2-(4-hydroxyphenyl)ethenyl]phenol 3-(5-aminopyridin-2-yl)oxy-N-cyclohexyl-5-[1-methyl-3-[(Z)-prop-1-enyl]pyrazol-4-yl]benzamide 2-[2,6-dichloro-4-(3,5-dioxohexyl)phenyl]propanoic acid [6-(2,4-difluorophenyl)-3-methylpyridine-2-carbonyl]-(1H-indol-3-yl)carbamic acid 2-(1-benzylazetidin-3-yl)oxy-5-methylpyridine 1-(2,3-dihydropyrrol-1-yl)-6,7-dimethoxyisoquinoline 2-aminopyrazolo[1,5-a]pyridine-3-carboxamide;5-chloro-2-(1H-imidazol-5-ylmethoxy)-N-methylbenzamide N-(7-bromobenzo[g]isoquinolin-1-yl)-N',N'-dipropylethane-1,2-diamine 1-[(3aR,7aS)-2-ethylsulfonyl-5-methyl-1,3,3a,4,6,7,7a-octahydropyrrolo[3,4-c]pyridine;2,2,2-trifluoroacetic acid 5-chloro-6-(2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-7-yl)pyridazine-3-carbonitrile 2-(3,4-dimethoxyphenyl)-5-hydroxy-8,8,8-trimethylpyrano[2,3-h]chromene-9,10-dione (4-chloro-3-methoxyphenyl)phosphane 5-(3,4-dichlorophenyl)-1-(3-nitrophenyl)pyrazole 6-[[5-(3,4,5-trifluorophenyl)pyridin-2-yl]methoxy]-1H-indazole 1,4-dibromonaphthalene;N'-(diaminomethylidene)-2,5-dihydroxy-3,6-bis[1-(4-hydroxyphenyl)ethyl]benzenecarboximidamide 3-[4-(2,6-dichlorophenyl)-5-methyl-1,2,4-triazol-3-yl]propanoic acid 4-chloro-N-(2,6-dichlorophenyl)-3H-pyrrole-5-sulfonamide 3,4-bis(trifluoromethyl)benzene-1,2-dicarbonitrile (E)-3-[4-(2-methoxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)phenyl]but-2-enoic acid 1-(azidomethyl)-N-(2-hydroxyethyl)naphthalene-2-sulfonamide 2-[3,5-dichloro-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)anilino]ethanol 2-(5,6-dimethylpyridin-3-yl)quinazoline 1-(6-chloro-7,8-dihydronaphthalen-2-yl)ethanone N-[(6S)-5,6-dimethyl-4-[2-[3-(trifluoromethoxy)phenyl]acetyl]piperazin-2-yl]acetamide (2E,4Z)-5-[2,3-bis[(4-fluorophenyl)methoxy]phenyl]penta-2,4-dienal N-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-1,5-dimethylpyrrole-2-carboxamide 1-(1,3-benzodioxol-5-yl)-2,2-bis[4-methoxy-2-[(Z)-prop-1-enoxy]phenyl]ethanone 4-[3-(5-phenylpenta-1,3-dienyl)phenyl]butanoic acid 2-[2-hydroxyethyl(methyl)amino]-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-4-one 5-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-1,3-dihydrobenzimidazol-2-one;ethane 3-[(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-2,2-dimethylpropanamide 3-[(4,7-dimethyl-1H-imidazo[4,5-c]pyridin-2-yl)methylidene]-6-hydroxy-1H-indol-2-one 2-[7-amino-4-(furan-3-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]-N-[1-(2,3-dihydro-1H-inden-5-yl)ethyl]acetamide N-(1,3-benzothiazol-5-ylmethyl)-2-(2-fluorophenyl)imidazo[1,2-a]pyridine-7-carboxamide;ethane 4-(4-butoxyanilino)-1,5-dimethylanthracene-9,10-dione 4-chloro-3-[(2Z)-3,7-dimethylocta-2,6-dienoxy]phenol ethane;1,2,3-trimethoxy-4-propan-2-ylbenzene 2-amino-9-[(4R,5S)-4-hydroxy-3,7,11-trimethoxy-2-oxa-8-azatricyclo[8.6.0.03,8]hexadeca-1(10),11,13-trien-8-yl]-1H-purin-6-one 6-amino-5,6,7,8-tetrahydroacridine-1,3,4-tricarbonitrile 5-hydroxy-4,7-dimethylquinoline-2-carbonitrile 7-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-methoxy-5-methylpyrrolo[3,2-d]pyrimidine 2-[(E)-1,4,4-trihydroxybut-2-enyl]benzoic acid 2-[5-(azidomethyl)pyridin-3-yl]-4,6-bis[2-(dimethylamino)ethoxy]aniline 4-chloro-2,5,6,7,8,9-hexahydropyrazolo[3,4-c]isoquinoline 3-amino-6-azido-2-ethylquinazolin-4-one 3-[[(2S,4R)-4-(dimethylsulfamoylmethyl)oxolan-2-yl]methoxy]benzoic acid [5-fluoro-2,3-di(propan-2-yl)phenyl]methanethiol 4-(3,5-difluorophenyl)-6-(3,4-dimethoxyphenyl)-2H-pyrrolo[3,4-c]pyrazol-3-ol 1-[3,4-difluoro-2-(2-fluoro-4-methylanilino)phenyl]ethanol (3S)-N-[2,6-difluoro-4-methyl-3-[5-[3-[methyl-(2,2,6,6-tetramethylpiperidin-1-yl)amino]propoxy]quinazolin-8-yl]phenyl]-3-hydroxypyrrolidine-1-carboxamide 1-azido-2-[(1,3-dimethylindazol-5-yl)sulfonylamino]cyclopropane-1-carboxylic acid 4-bromo-N-[2,6-di(propan-2-yl)phenyl]-1H-pyrrole-3-carboxamide 5-tert-butyl-2-methyl-3,7-dihydropyrrolo[2,3-d]pyrimidin-4-one 1-[2-(3,4-dimethylanilino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-N,N-dimethyl-2-(5-methylthiophen-2-yl)ethanamine;formic acid (4R)-2,3-dimethyl-4-phenyl-5,10-bis[1-(2-sulfanylidene-3H-1,3,4-oxadiazol-5-yl)ethoxy]-6a,7,8,9,10,10a-hexahydrobenzo[g]quinoline-6,11,12-trione 2-[3,5-dibromo-4-(hydroxymethyl)phenyl]acetic acid 2-[3,5-bis(trifluoromethyl)phenyl]cyclohexane-1-carbonitrile N-(3,4-dichlorophenyl)-2,3-bis[(2R)-1-hydroxybutan-2-yl]benzimidazole-5-carboxamide 4-azidooxy-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide 2-[N-(2,4-dinitrophenyl)-4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]anilino]phenol 1-(difluoromethoxy)-6,8-dimethylnaphthalene 2-azido-4-(benzylamino)quinazoline-5,7-diol 4-methyl-3-nitro-N-[(Z)-pentylideneamino]benzamide 2-[(4-methoxyphenyl)methyl]-5,6-dihydroquinoline (2Z)-2-[4-(5-azidopentoxymethyl)phenyl]-N,5-diethylhepta-2,6-dienamide 2-(1,4,5,6-tetrahydropyrimidin-4-ylamino)benzamide N-(3,4-dihydronaphthalen-1-yl)-4-methoxypyridine-2-carboxamide 3-methoxy-N,2,5-trimethylaniline 3-[[(2S)-1-methylpyrrolidin-2-yl]methoxy]pyridine-2,6-dicarbonitrile 2-[2-(3,4-dimethoxyphenyl)ethyl]-N,N-bis(ethylsulfanyl)-6-sulfamoylpyridine-3-carboxamide (2R)-N-[(1S)-3-cyclohexyl-2-oxo-1-phenylpropyl]-4-(5,6,7,8-tetrahydroquinazolin-4-yl)butanamide N-(4-bromobutan-2-yl)-N-methoxycarbonyl-2,6-dinitrobenzamide 3-[(E)-1,2-difluoro-2-iodoethenyl]-6-(4-fluorophenyl)-5-methylpyrimidin-4-one 2-[4-(1H-indole-7-carbonyl)morpholin-3-yl]-3H-quinazolin-4-one 4-chloro-3,5,6-trifluoro-7-[1-[(1S)-2-(5-oxopyrrolidin-2-yl)ethoxy]ethenyl]quinoxaline-2-carboxylic acid 3-[2-(aminomethyl)-6-phenylphenyl]imino-4H-naphthalen-1-amine 1-N',2-N',3-tributylbenzene-1,2-dicarbohydrazide (3S)-4-tert-butylsulfanyl-N',2,6-trihydroxy-3-methoxybenzenecarboximidamide (2Z,5S)-5-[4-chloro-3-(trifluoromethyl)phenyl]-2-[[(E)-(4-hydroxyphenyl)methylideneamino]hydrazinylidene]-1,3-thiazolidin-4-one 5-amino-3-(4-chlorocyclohexyl)pyrazolo[1,5-a]pyrimidine-2-carbonitrile;propane 3-ethyl-N'-(1H-indazole-5-carbonyl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole-7-carboximidamide 4-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-5-methoxycarbonyl-2-[[2-(pyrazol-1-ylmethyl)phenyl]carbamoylamino]thiophene-3-carboxylic acid 3-[2-(dimethylamino)ethyl]-8-(5-fluoropyrimidine-4-carbonyl)-1,7-bis[2-(3-hydroxypropoxy)ethyl]purine-2,6-dione 1-[3-amino-2-(hydroxymethyl)prop-2-enoxy]-4-fluoroisoquinoline-3-carbonitrile 2-[(2R)-4-acetyl-2-methylpiperazin-1-yl]pyrimidine-5-carboxamide 7-cyclopentyloxy-6-ethoxy-4-oxo-N-(2,2,2-trifluoroethyl)-1H-quinoline-3-carboxamide 1-[2,6-di(propan-2-yl)phenyl]-3-[(E)-(3,5-dimethoxy-4-methylphenyl)methylideneamino]urea N-[2,6-difluoro-3-(propylsulfanylamino)phenyl]-5,7-diethyl-1H-indole-2-carboxamide 2-(5,6-dimethylnaphthalen-1-yl)pyridine 2-(3,4-dihydropyridin-6-yl)-N-[1-(5H-pyrrolo[3,2-d]pyrimidin-4-ylamino)butan-2-ylidene]prop-2-enamide 4-[(3,5-dimethylphenoxy)methyl]-1-(2-ethoxyphenyl)triazole 2-methyl-4,6-diphenyl-1H-triazine (E)-3-[6-[[(1S)-2,2,3,3,5,5,6,6-octadeuteriocyclohexyl]oxymethyl]pyridin-3-yl]prop-2-enoic acid 4-amino-3-[(E)-1-aminoprop-1-enyl]-7-fluoro-6-hydroxyquinoline-2-carboxamide;ethane [4-(ethylaminomethyl)piperidin-1-yl]-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methanone 3-(6,7-dihydroimidazo[2,1-b][1,3]thiazol-5-yl)-N-ethylaniline 6-[2-(dimethylamino)ethoxy]-3,4-dihydro-1H-quinazolin-2-one 4-(2-methylpropoxy)naphthalene-1,3-dione 3-[(4-carbamimidoylphenyl)methoxy]-2,6-dibromobenzoic acid 2-(3-aminophenyl)-6-(2-fluoroanilino)benzonitrile 2,2-dichloro-3-[4-(2-phenylethynyl)phenyl]cyclopropane-1,1-dicarbonitrile N-[(E)-benzylideneamino]-2-[(6R,7S)-5-oxo-3-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidin-7-yl]acetamide (7-tert-butyl-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepin-3-yl)methanol 4-[4-[4-(2,6-difluoro-4-pentoxyphenyl)cyclohexyl]cyclohexyl]-2,3-difluorophenol [[3-(6,8-dichloro-2H-chromene-4-carbonyl)phenyl]methylamino]urea N-cyclohexyl-2,6-dioxo-4-phenyl-1H-pyrimidine-5-carboxamide ethane;1-methoxypropan-2-one;6-[2-(1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]-1H-indole 4-(4-fluorophenyl)sulfanylbutanal;N-methylethanesulfinamide;[2-(piperidin-1-ylamino)phenyl]urea 2,3-dibromo-7-methyl-1H-indole 2-(9H-fluoren-1-yloxycarbonyl)benzoate 2-(5-fluoropyridin-3-yl)-4,6-diphenylpyrimidine N-[2,6-bis(3-phenylpentan-3-yl)phenyl]propanethioamide 2-methyl-N-[4-(pyrimidin-2-ylamino)phenyl]benzenesulfonamide 2-[(1S,3R)-3-aminocyclopentyl]oxy-4-methanimidoylbenzoic acid N-[2,6-bis(trifluoromethyl)phenyl]-3-hydroxy-1,5-dimethylpyridine-4-carboxamide ethane;4-(methylamino)naphthalene-1,2,3-trithiol 5-methyl-3-[4-(2,3,6-trichlorophenyl)sulfonylpiperazin-1-yl]-1H-indole 5-[(5,7-difluoro-1H-indol-2-yl)methyl]spiro[3a,4-dihydro-1H-indene-2,4'-piperidine] 5-[(4-azido-3,5-dimethylpyrazol-1-yl)methyl]-2-pyrimidin-2-yltetrazole 4-chloro-2-(4-methylphenyl)naphthalene-1,3-dione;ethane N-[5-cyano-2-[4-(1-ethylpyrazol-3-yl)piperidine-1-carbonyl]phenyl]ethenesulfonamide (1R)-6,7-dichloro-1-ethyl-5,10-dimethoxy-2-oxo-N-[4-(trifluoromethylsulfonylmethyl)phenyl]-3H-benzo[g]pteridine-8-carboxamide 1-(2-azidooxyethyl)-4-(4-chlorophenoxy)triazole (4aS,9aR)-3,4a,5,6,7,8,9,9a-octahydropyrido[2,3-b]azepine;4-(2H-azirin-3-ylmethoxy)-N-(1H-indazol-6-yl)benzamide 4-[3-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]benzonitrile 1-[4-[(1R,2S)-2-methylcyclopropanecarbonyl]phenyl]piperidine-3-carboxamide 3-chloro-4-[(2,5-dimethylphenyl)sulfonylamino]benzoic acid 1-[2,6-bis(trifluoromethyl)phenyl]-5-[4-(2,3-dihydropyridin-4-yl)phenyl]pyrazole N-azido-2-(3-hydroxyphenyl)propanamide (2-amino-6-phenoxypyrimidin-4-yl)oxyboronic acid;ethane 2-[[4,5-dichloro-3-(trifluoromethyl)pyrazole-1-carbonyl]amino]acetic acid 2-(4-chlorophenyl)-6-[(3-fluoropyridin-4-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-[2,4-dihydroxy-3,6-bis(3-methylbutanoylamino)phenyl]butyl-triethylazanium N-(2-methoxyphenyl)-4-oxo-3H-quinazoline-7-carboxamide 5-[5-(diethylamino)pyrazin-2-yl]-7,8-dihydronaphthalene-1,6-disulfonic acid N-azido-4-phenylbutanethioamide 3-[4-amino-7-[(2R,6S)-1,2,6-trimethylpiperidin-4-yl]pyrrolo[2,3-d]pyrimidin-5-yl]phenol 2-(3-cyclohexa-1,5-dien-1-ylpropanoyl)benzaldehyde 2-[(3R)-1-(4,6-dichloropyrimidin-5-yl)piperidin-3-yl]acetic acid 6-(2-cyclopentyloxyethoxy)imidazo[1,5-a]pyridine (NE)-N-[(5-methoxycarbonylfuran-2-yl)methylidene]-1,3-diphenylpyrazole-4-carboximidate 6-fluoro-5'-phenylspiro[cyclohexane-1,3'-isoindole]-2'-one (4S)-3-methylsulfonyl-2-(3-phenylpropanoylamino)-N-propan-2-yl-3,4,5,6-tetrahydropyridine-4-carboxamide 2-(4-benzo[g]quinoxalin-5-ylphenyl)propan-1-ol 2-(4-ethylpiperazin-1-yl)-6,7-difluoroquinoline (1R)-2-[4-[3,5-di(propan-2-yl)phenyl]pyridin-2-yl]oxy-N,N-dimethylcyclohexa-2,4-dien-1-amine 5-[(3S)-2,2-dimethylpentanoyl]oxy-1H-indole-2,7-dicarboxylic acid 2-azido-1,3-dichloro-5-(trifluoromethyl)benzene 2-[8-chloro-7-(4,5-dihydro-1H-imidazol-2-ylmethoxy)-9,10-dioxoanthracen-2-yl]acetic acid 3-[4-methyl-6-(propylamino)pyrimidin-2-yl]imidazo[1,2-b]pyridazine-7-carboxylic acid 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-9-phenyl-1,10-phenanthroline 1-(2,5-dimethylfuran-3-carbonyl)-N-[2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperidine-4-carboxamide (2-methylphenyl)-[1-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-yl]methanol 1-(2,6-difluorophenyl)sulfanyl-3-[4-[(3S)-3-methoxypyrrolidin-1-yl]phenyl]azetidine 2-[1,3-bis(4-fluorophenyl)propan-2-yl]-2-(3-pyridin-2-ylpyrazol-1-yl)acetamide N-butan-2-yl-5-[(E)-3-cyclopenta-1,4-dien-1-ylprop-1-enyl]pyridin-2-amine 2-methylpropane;7-[4-[(3R)-oxolan-3-yl]oxyphenyl]benzo[g]pteridine 4-[(3,5-difluorophenyl)methylamino]-N-methoxypyridine-2-carboxamide 4-(1H-imidazole-2-carbonyl)-1,4-diazepan-6-one;hydrochloride 2-(4-aminophenyl)-6-[(3-bromothiophen-2-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (Z)-1,3-diphenylprop-2-en-1-one;N-[[2-fluoro-6-methoxy-4-[5-(trifluoromethyl)pyridin-3-yl]phenyl]methyl]-N,2,2-trimethylpropanamide 5-azido-1,3-dibromo-2-(4-methylsulfanylphenyl)benzene 3-(3-chlorophenyl)-2-methyl-7-propylpyrazolo[1,5-a]pyrimidine 2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridine-4-carboxamide 3-(5,6-dimethoxypyridin-3-yl)cyclobutan-1-amine 3-(3,5-dimethyl-1H-pyrazol-4-yl)-6-methoxypyridin-2-amine;5-methanimidoylpyrimidine-4,6-diamine 1-[(4S)-3-[6-[[5-chloro-4-(methylamino)pyrimidin-2-yl]amino]pyridin-3-yl]-2-oxoimidazolidin-4-yl]piperidine-3-carboxamide (6R)-7-[[2-amino-5-chloro-4-fluoro-3-[(4-hydroxy-1-methylcyclohexanecarbonyl)amino]benzoyl]amino]-8-oxo-3-propanoylsulfanylundecanoic acid (5E)-2-phenylimino-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 3-bromo-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 2-ethoxycarbonyl-8-[(4-methyl-1,3-thiazol-2-yl)carbamoyl]-6-phenylimidazo[1,5-a]pyridine-7-carboxylic acid 2-(4-fluorophenyl)-6-(methylaminooxymethyl)oxan-3-ol 3-azido-5,6-dimethoxy-2-phenylquinoxaline 2-(3,5-difluorophenyl)sulfonyl-8-(4,6-dimethoxypyrimidin-2-yl)sulfanyl-9-methylidenedecanedioic acid 3-[2-(3,4-difluorophenyl)ethyl]-5-(1-methoxy-2-nitrosoethyl)-1H-indole N-[4-(diethylcarbamoyl)phenyl]-2,5-dihydroxybenzamide 2-(N-ethenylsulfonyl-4-hydroxyanilino)benzenesulfonic acid [2,4-dichloro-3-(2-ethylpyrazole-3-carbonyl)phenyl]-[4-hydroxy-4-[(2R)-2-methylpentoxy]piperidin-1-yl]methanone 2-(3,5-dichlorophenyl)imino-N'-ethyl-N-hydroxyethanimidamide 1-(3,4-dichlorophenyl)-5-[2-(2-fluorophenyl)sulfanylethylimino]pyrazolidin-3-one [2-[[4-[2-(aminomethyl)-3-fluoroprop-2-enoxy]phenyl]sulfonyl-[(3-chloro-5-methylcyclohexa-1,5-diene-1-carbonyl)amino]methylidene]cyclopentylidene]azanium 6,7-bis[(3-tert-butylphenyl)methyl]-1H-indene 3-N,5-N-dibutylbenzene-1,2,3,4,5-pentamine 5-[(1R)-2-chlorocyclohexa-2,4-dien-1-yl]-N-phenylthiophene-3-carboxamide N-[(2R,3S)-1-[2-(dimethylamino)acetyl]-2-(2-ethoxypyrazol-3-yl)piperidin-3-yl]-5-fluoropyridine-2-carboxamide 2-hydroxy-1,4-dimethoxyanthracene-9,10-dione [4-hydroxy-2-(trifluoromethyl)phenyl]iminocarbamic acid 2-[4-(1H-imidazole-5-carbonyl)piperazin-1-yl]-6-methylpyrimidin-4-amine 7-[4-chloro-3-(trifluoromethyl)phenyl]-2-ethoxy-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 7-(3,5-dimethoxyphenyl)-5-methylpyrido[4,3-b]indole 1-(4-azidooxybutyl)-3,5-difluorobenzene 3-[[2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)acetyl]amino]benzoic acid;hydrochloride N-azido-4,5-diethyltriazin-1-amine (5E)-2-imino-5-[(4-naphthalen-1-yloxyphenyl)methylidene]-1,3-thiazolidin-4-one 1-(2,6-dimethylphenyl)-5-[4-ethoxy-3-(trifluoromethyl)phenyl]pyrazole 7-(2,3-difluorophenyl)-1,4-oxazepane 6-[[5-chloro-2-(4-methylpiperidin-1-yl)pyridine-3-carbonyl]amino]-N-ethyl-8-(oxan-4-yl)imidazo[1,5-a]pyridine-7-carboxamide 2-(5-chloro-3-cyclopropyl-1,2-oxazol-4-yl)-N-[4-[methyl-[(Z)-(5-oxo-2H-furan-3-ylidene)amino]carbamoyl]phenyl]-2-(thiolan-1-ium-1-yl)acetamide (E)-N-(5-benzamidocyclohepta-1,3,6-trien-1-yl)but-2-enediamide 3-methoxy-6,7-dimethyldibenzothiophene 2-[(3Z)-4,5-bis(sulfanyloxy)hexa-1,3-dien-2-yl]benzenethiol 7-[3-(4-methylpiperazine-1-carbonyl)azetidin-1-yl]-5-oxo-8H-pyrido[2,3-d]pyrimidine-6-carboxylic acid 5-[(3S,4R)-1-acetyl-6-hydroxy-4-methoxycarbonyl-2-oxo-3-propan-2-ylpyrrolidin-3-yl]-N-diazo-1H-pyrrole-2-sulfonamide 4-[(1,3-dimethylindol-2-yl)sulfonylamino]-N-hydroxybenzamide 2-[4,6-dichloro-7-(2-cyclopropylbenzimidazol-1-yl)pyrido[2,3-b]pyrazin-3-yl]propan-2-ol (2R,4S)-N-[(Z)-1H-indol-3-ylmethylideneamino]-6-oxopiperidine-2-carboxamide 1-[(2-cyclopropylphenyl)methyl]-7H-purin-6-imine 2-[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]-4-thiophen-2-yl-1H-imidazole-5-carboxylic acid 4-[2-methoxy-5-(1H-pyrazolo[3,4-c]pyridine-6-carbonylamino)phenyl]piperazine-1-carboxylic acid 1-[(2Z,4E)-1-methoxyhexa-2,4-dien-3-yl]-6-phenoxyindazole 4-[1,3-bis(9H-fluoren-1-yl)-2-methoxypropan-2-yl]benzenesulfonic acid ethane;4-[4-[(3E)-hexa-1,3,5-trien-3-yl]oxybutoxy]benzoic acid N-[2-[(3S)-3,4-dimethylpiperazin-1-yl]phenyl]cyclopropanesulfonamide 4-amino-3-chloro-2-(4,5-dimethylimidazol-1-ium-2-ylidene)pyridine-1-carboximidamide (2S,4R)-4-(benzenesulfonamido)-1-[5-chloro-6-methyl-1-(3,4,5-trifluorophenyl)benzimidazol-2-yl]sulfonylpyrrolidine-2-carboxylic acid N-(3,4-difluorophenyl)-2-[1-methyl-5-(4-morpholin-4-ylphenyl)pyrazol-4-yl]acetamide 3-butan-2-yl-1,5-difluoro-2-methylbenzene;1-cyclopropyl-N'-(2-methoxyacetyl)-4-methylidenepiperidine-2-carbohydrazide 2-(4-cyano-3-fluorophenyl)-6-hydroxyhexanoic acid 2-methoxy-4-[(3S)-piperidin-3-yl]-1H-benzimidazole 6-methyl-4-(2H-triazol-4-yl)cyclohexa-1,3-dien-1-amine 2-[1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethylideneamino]guanidine;hydrochloride 1-[4-(cyclohexylmethyl)piperazine-1-carbonyl]quinolin-2-one;ethane 4-cyclopentyl-2-[(2-fluorophenyl)methylsulfanyl]-5-iodo-1H-pyrimidin-6-one 2-(4,5-dihydro-1H-imidazol-2-yl)-1-(3,4,6,7,8,9-hexahydrofuro[3,2-c]azocin-1-yl)ethanone 4-[(3Z)-penta-1,3-dien-2-yl]oxybenzenethiol 3,5-dimethoxybenzenecarboximidamide 4-(3,5-difluorophenyl)-7-methoxy-N'-methylspiro[1,2-dihydropyrrolo[3,2-b]quinoline-3,1'-cyclobutane]-5-carboximidamide;1-fluoropropane 1-(2,2-difluoroethoxy)-4-methyl-2-propan-2-ylbenzene (5S)-5-[2,6-difluoro-4-(1H-indol-3-yl)phenyl]-N-methoxy-4,5-dihydro-1,3-oxazol-2-amine 1-[5-[5-(3,5-dimethyl-1H-pyrazole-4-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-pyrazol-3-yl]ethanone 5-[[3-[3,4-dichloro-2-(cyclopropylcarbamoylamino)phenyl]-1,2-thiazol-5-yl]methylidene]-1,3-thiazolidine-3-carboxamide 3-[5-amino-6-(5,7-difluoroquinolin-4-yl)pyrazin-2-yl]cyclobutan-1-one 1-(2,5-dimethoxyphenyl)-3-[5-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)pyridin-2-yl]urea (E)-2,3-dimethyl-3-(2-methylidenehexanoylamino)-N-[[6-(trifluoromethyl)pyridin-2-yl]methoxy]but-2-enamide 4-(9H-fluoren-1-yl)-2-(1,3-thiazol-5-ylmethylideneamino)aniline 1-azido-2,3-bis(chloromethoxy)naphthalene 3-methyl-4-(5-nitrobenzotriazol-1-yl)piperidine-1-carboxylic acid 3-chloro-2-[(E)-2-methylhex-1-enoxy]pyridine N-[(4-nitrophenyl)methyl]-N-(2H-tetrazol-5-yl)hexadecanamide N-[4-amino-2,6-di(propan-2-yl)phenyl]-1-methoxyethenamine 3-(difluoromethyl)-5-[3-methyl-4-(4-methylimidazol-1-yl)phenyl]-N-propan-2-yl-1,2-oxazole-4-carboxamide 6-methyl-1'-[[3-(trifluoromethoxy)phenyl]methyl]spiro[2H-1,3-benzodioxine-4,3'-indole];hydrochloride ethane;1-methylsulfanyl-4-(4-propylphenyl)benzene 5-[2,4,6-trimethyl-N-(1,3-thiazol-5-yl)anilino]naphthalene-2-sulfonic acid (2S)-1-[3-[[6-amino-2-(4-fluorophenyl)pyrimidine-4-carboximidoyl]amino]piperidin-1-yl]butane-1,2-dione N-(4-bromo-2,5-dimethylphenyl)-N-naphthalen-1-ylbenzenesulfonamide 1-[2-[(Z)-2-amino-3,3,4,4,5,5,6,8,7,9,10,10,11,11-hexadecafluorodec-1-enyl]phenyl]ethanone 1-amino-3,3-bis(3-methylphenyl)propan-2-ol 2-(3-ethoxyphenyl)-6-methyl-7,7a-dihydroimidazo[1,5-b]pyridazine 4-[(2,4-dinitrophenyl)methoxy]butanoic acid 2-(4-azidooxypiperidin-1-yl)-5,6,7,8-tetrahydroquinoline 2-[3,5-dichloro-4-[(6-oxo-1H-pyridazine-3-carbonyl)amino]phenyl]propanoic acid 4-[(2-chlorophenoxy)methyl]-N'-hydroxypyridine-2-carboximidamide 3-[(2-bromo-5-chlorophenyl)methyl]-2,6-dihydropyran 3-methylsulfanyl-N'-phenylpyrazolo[1,5-a]pyrimidine-6-carbohydrazide N-(8-cyclohexyloxy-7,11-difluoro-1-methylidenebenzo[c]carbazol-5-yl)ethanimine 4-(2,6-dichlorophenyl)-5-fluoropyrimidine 2-azidosulfanyl-4-(2,5-dimethoxyphenyl)furan 2-(4-ethoxy-3,5-dimethoxyphenyl)quinoline 2-[3-[4-(difluoromethoxy)phenoxy]propylsulfanyl]-5-thiophen-2-ylthiophene N'-[(Z)-1,3-diaminoprop-2-enylidene]-2-(4-hydroxyphenyl)-5-methyl-6-pyridin-2-yloxybenzenecarboximidamide 3-[[2-chloro-6-(trifluoromethyl)phenyl]methylamino]benzoic acid 3-[4-(4-chlorophenoxy)-2-methylphenyl]-N,1-dimethyl-5-oxo-N-propanoylpyrazole-4-carboxamide 5-bromo-3-N-[(2R)-1,4-dioxan-2-yl]benzene-1,3-diamine (E)-N-ethoxy-3,3-dimethylpentan-1-imine;4-[2-fluoro-5-[3-[4-methyl-3-(1,2,4-triazol-1-yl)phenyl]-1,2,4-oxadiazol-5-yl]phenoxy]piperidine-1-carboxylic acid N-[2-(aminomethyl)phenyl]-4,6-dihydrazinylidenecyclohexa-2,5-dien-1-imine 3-(azidomethyl)-5-bromophenol (2E,4Z)-3-[5-(N,3,6-trimethylanilino)-1H-pyrazol-3-yl]hexa-2,4-dienal N-(2,5-dimethoxyphenyl)-4,7,7-trimethyl-3,5,6,8-tetrahydroisoquinoline-1-carboxamide 2-(5-methylcyclohexa-1,3-dien-1-yl)oxy-N-[[4-(trifluoromethoxy)phenyl]carbamothioyl]acetamide N'-[(1R)-2-hydroxy-5,7-dinitrochromen-4-ylidene]carbamimidate 3-(6-azidonaphthalen-2-yl)oxy-1H-indole 1-[1-(4-fluorophenyl)-5-hydroxy-6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl]ethanone [1-(2,6-dimethylphenyl)piperidin-4-ylidene]-methoxycarbonylazanium N-[2-(3,4-dichlorophenyl)propan-2-yl]-5-hydroxypyridine-3-carboxamide [2-bromo-4-fluoro-5-(3,4,6-trichloroimidazo[1,2-a]pyridin-8-yl)phenyl]methanol 5-[2-(4-bromophenoxy)phenyl]-1H-pyrazole 5-[[2,3,4-trimethoxy-6-(1,1,1-trifluoropentan-3-yl)phenyl]carbamoylamino]cyclohexa-1,5-diene-1-carboxylic acid 2-azido-5-cyclobutyloxypyrazine 4-[3,5-difluoro-2-(trifluoromethyl)phenyl]pyridine 2-[3,5-bis(trifluoromethyl)phenyl]-6-chloro-4-N-pyrimidin-4-ylpyrimidine-4,5-diamine 4-[4-(1,3-benzodioxol-5-yl)-2H-pyridin-1-yl]benzenesulfonamide N-methyl-1-(4-morpholin-4-ylphenyl)ethanamine;2,3,4,5-tetrahydro-1H-1,4-benzodiazepine 2-[8-(cyclopropylmethyl)-3,5,6,7,9,10-hexahydropyrimido[4,5-h][1]benzazepin-2-yl]phenol 4-chloro-3-[[2-methoxyethyl(propyl)amino]methyl]phenol (1R,3R)-3-[4-[(5-bromopyrimidin-2-yl)oxymethyl]piperidine-1-carbonyl]cyclopentane-1-carboxylic acid (2S)-1-[4-[4,6-bis(ethenyl)pyridin-3-yl]-N-methylanilino]propan-2-ol 1-[4-fluoro-3-methyl-5-(trifluoromethyl)phenyl]-2,2-dimethylpropan-1-one 3-[4-(azidomethyl)phenyl]-5,6-dihydro-1H-pyrrolo[2,3-b]pyridine (Z)-4-[(5E,7Z)-10-amino-8-methylundeca-5,7,11-trienyl]iminobut-2-en-1-amine;[3-methoxy-1-[4-(2-phenylethynyl)phenyl]piperidin-4-yl]-(4-propan-2-ylpiperazin-1-yl)methanone 2-chloro-N-(5-nitro-1,3-thiazol-2-yl)-4-(trifluoromethoxy)benzamide 4-benzyl-6,7-dimethoxy-2-(3-nitrophenyl)quinoline 2-(4-chlorophenyl)-1-[7-hydroxy-3,5-bis(trifluoromethyl)-6H-pyrazolo[4,3-b]pyridin-1-yl]ethanone (E,2Z)-3-[4-(dimethylamino)phenyl]iminopent-4-enoic acid N-[3-(2,4,6-trimethylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-ium-2-ylidene]hydroxylamine 1-(3,4-dimethoxyphenyl)-2-nitroethenol (4S)-3-[4-[1-[2-[4-(5,6-dichlorobenzimidazol-1-yl)phenyl]acetyl]piperidin-4-yl]butanoyl]azepane-4-carboxylic acid N-[2-bromo-4-chloro-3-(hydroxyiminomethyl)phenyl]-4-tert-butylbenzenesulfonamide 4-(2,3-dihydro-1H-indazole-6-carbonyl)morpholin-3-one [1-[(4R)-2,5-dimethyl-3-oxo-1,6-dihydrocyclohepta[c]pyrazole-4-carbonyl]azetidin-3-yl]methylcarbamic acid 6-(2,4-dimethylpyrimidine-5-carbonyl)-N-[1-(2-methoxyphenyl)cyclopropyl]spiro[3.3]heptane-2-carboxamide (2S)-4,6-difluoro-2-[3-[4-[5-methylsulfonyl-2-(trifluoromethyl)phenyl]piperidine-1-carbonyl]phenoxy]spiro[2H-1-benzofuran-3,4'-piperidine] N-[2-(1H-indol-3-yl)ethyl]-1,6-dimethyl-5-propan-2-yloxycyclohexa-2,4-diene-1-carboxamide 6,8-difluoro-N'-hydroxy-7-[methyl(2-methylsulfanylethyl)amino]quinazoline-4-carboximidamide 1-[(2R)-1-[4-(4-fluorophenoxy)benzoyl]piperidin-2-yl]ethanone N-(2-chlorophenyl)-2-[[1-ethyl-6-hydroxy-5-methanimidoyl-3-(4-methoxyphenyl)sulfonylindol-2-yl]amino]acetamide [4-[2-chloroethyl(methyl)amino]-3,5-difluorophenyl]urea 4-N,6-N-bis(4-aminophenyl)-1-N,1-N-diethyl-5H-pyrrolo[3,2-c]pyridine-1,4,6-triamine 1-cyclopropyl-6-fluoro-8-[(2S)-4-[3-(trifluoromethoxy)benzoyl]morpholin-2-yl]quinolin-4-one N-[1-(3,5-dimethyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]-2-fluoro-6-methoxybenzamide 3-[4-(1,1,1,2,3,3-hexadeuteriopropan-2-yl)phenyl]-2-phenyl-6H-cyclohepta[b]furan (3R)-3-[4-[(5-fluoropyridin-2-yl)oxymethyl]phenyl]hexanoic acid (2S,4R)-2,4-dibenzyl-6,7-bis[[(1S)-1-phenylethoxy]methyl]octanoic acid 1-[6-(cyclopropylmethoxy)-2-methoxypyridin-3-yl]-7-[(2-ethylphenyl)methylamino]pyrido[4,3-b]indole-5-carboxylic acid [2,5-dichloro-3-[4-(trifluoromethylsulfanyl)phenyl]phenyl]hydrazine 2-[4-[3,5-difluoro-6-(methoxymethyl)naphthalen-2-yl]phenyl]-5-hexylpyrimidine 1-[[4-(3,4-difluorophenyl)oxan-4-yl]methoxy]-5-ethylidenepyrrolidin-2-one 5-(2,4,6-trifluorophenyl)sulfanylpentanal 3-methyl-5-[4-(1-pyridin-2-yl-2,3-dihydrotriazolo[4,5-b]pyrazin-5-yl)phenyl]oxolan-2-one N-(4-butylcyclohexyl)-N,1-dimethylindazole-3-carboxamide N-[3,5-dichloro-4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1-(2-fluoroethyl)-5-oxopyrrolidine-3-carboxamide 5-(9H-fluoren-1-yl)furan-2-carboxylic acid N-methyl-N'-[5-(propanoylamino)pyridin-2-yl]oxamide 3-(2-benzylpiperidin-4-ylidene)prop-1-en-1-amine 2,3-diphenylbutane-2-sulfonic acid N-(2,6-dimethyl-4-propan-2-ylphenyl)but-3-enamide (3R,4R)-1-[2-(difluoromethoxy)ethyl]-N-[2-(furan-3-yl)ethyl]-4-phenylpyrrolidine-3-carboxamide;hydrochloride 1-(2-azidophenyl)-N,N-dimethylpiperidine-4-carboxamide 4-[(3S)-3-(cyclopropylmethoxy)pyrrolidine-1-carbonyl]-2,5-difluorobenzamide 3-(cyclopropanecarbonylamino)-N-(4,5,6,7-tetrahydro-1H-indazol-6-ylmethyl)benzamide N-[(3S,4R)-1-(cyclopropylmethylsulfonyl)-4-ethylpyrrolidin-3-yl]-3-phenylazetidine-1-carboxamide 2-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]-1H-pyrimidine-2,4-diamine 3-chloro-4-(2,5-difluorophenoxy)-N-[1-hydroxy-6-methoxy-1-[3-(trifluoromethylsulfanylamino)phenyl]hexan-2-yl]benzamide (1S,2R)-N-[(4-chlorophenyl)methyl]-1-[6-[[5-cyano-1-ethyl-6-oxopyridin-3-yl]amino]pyrimidin-4-yl]-N,2-dimethylcyclopropane-1-carboxamide 1-[(2S,3R)-4-methyl-3-phenylmorpholin-2-yl]ethanethiol 1,3-difluoro-2-[(E)-1-iodopent-1-enyl]benzene (4R)-1-[(2R,3S)-1,2,3,5,6,7-hexahydro-s-indacen-4-yl]-3-methylpiperidine N-[(1R)-3,4-dihydro-2H-chromen-8-yl]pyrazolo[5,1-b][1,3]thiazole-6-carboxamide 2-(4,5-diphenyl-1,3-oxazol-2-yl)benzamide [1-(4,5-dihydro-1H-imidazol-2-ylmethoxy)piperidin-4-yl]-(3-fluorophenyl)methanone 5-(4-methylphenyl)sulfonyloxypyridine-2-carboxylate N-ethenyl-4-methyl-N-[(3E)-1,6,6-trifluoro-5-(trifluoromethoxy)hexa-3,5-dien-2-yl]aniline 1-benzyl-5-(dimethylamino)-7H-pyrazolo[3,4-b]pyridin-6-one 1-methyl-2,3,4,5,6-pentapropylnaphthalene 1-azidooxy-6,7-diphenylheptane-2,3-dione 2-[(4E,5E)-5-ethylidene-4-(2-pyridin-3-ylprop-2-enylidene)-1H-pyrazol-3-yl]-7-pyrazin-2-yl-3H-imidazo[4,5-c]pyridine 2-[[4-[6-(3,5-dichlorophenyl)sulfanylpyridin-3-yl]oxy-1H-benzimidazol-2-yl]methoxy]ethylcarbamic acid [(3R)-4-phenyl-3-(pyridin-2-ylmethoxy)butanoyl]azanium 2-[(2S)-1,4-dioxan-2-yl]-N-(3-sulfamoylphenyl)propanamide 4-(4,5-dimethylpyridazin-3-yl)morpholine 4-(4-fluorophenyl)-N-[(Z)-(3-hydroxy-5-methoxy-2-nitrophenyl)methylideneamino]benzamide 5-phenyl-1,2-dihydropyrazolo[1,5-a]pyrimidine 3,4-di(nonyl)phthalate (E)-N',N'-dimethyl-3-[4-[1-(2-pentan-3-ylphenyl)propoxy]cyclohexyl]prop-2-ene-1,3-diamine 3-amino-N-cyclopropylbenzenesulfonamide N'-hydroxy-2-(oxolan-3-ylmethoxy)pyrimidine-4-carboximidamide 6-[5-[(5,5-dimethyloxolan-3-ylidene)methoxy]pentoxymethyl]pyridine-2-carbonitrile N-[4-(6,8-dihydrothieno[3,2-e]indole-2-carbonyl)phenyl]-2-ethyl-5H-pyrrolo[2,1-a]isoindole-7-carboxamide 4-[2-[4-(cyclohexylcarbamoyl)phenoxy]-6-morpholin-4-ylpyridin-3-yl]benzoic acid N-[[(2S,4R)-1-cyclohexyl-5-oxo-4-propan-2-ylpyrrolidin-2-yl]methyl]-3-[3-(trifluoromethoxy)phenyl]propanamide 3-chloro-N-cyclobutyl-2,4,5-trifluoroaniline 4-[3-(difluoromethoxy)phenyl]-1,2-thiazole [3-hydroxy-2,4,6-trimethyl-5-(2H-tetrazol-5-yl)phenyl]oxidanium (3Z,5E)-2-methylocta-1,3,5,7-tetraene;2-(1H-naphthalen-2-ylideneamino)propanoic acid 3-(2,4,6-trimethylbenzoyl)phthalic acid 6-[2,4-difluoro-3-(triazol-1-yl)phenyl]-5-ethynylpyrimidine-4-carboxamide [(2R)-1-(dimethylamino)-5-oxohexan-2-yl]oxymethylidene-phenylazanium 2-[(Z)-benzylsulfanylamino]propanamide;methanethiol 2-(3,4-dichlorophenyl)imino-5-[(1-methylindol-3-yl)methylidene]-1,3-thiazolidin-4-one 2-[(3R,4S)-1-[2-(benzenesulfinyloxy)acetyl]-3-methylpiperidin-4-yl]oxyacetic acid 4-[4-(6,7-dihydrobenzo[a]quinolizin-5-ium-11-yl)phenyl]benzoic acid N-[5-chloro-2,4-difluoro-3-(2-fluoropyridin-3-yl)phenyl]methanesulfonamide [2-(3-methylsulfanylphenyl)phenyl]-(6-methylcyclohexa-1,5-dien-1-yl)methanone 4-[2,3-dihydroxypropyl(1H-imidazol-5-yl)amino]benzoic acid 4-[3,5-bis(trifluoromethyl)phenyl]-2-sulfanylidene-1H-pyrimidine-6-carboxylic acid [3-(2,6-dihydroxyphenyl)propanoylamino]-hydroxyphosphinic acid N-(3,4-dichlorophenyl)sulfonyl-5-[(Z)-1-hydroxybut-2-enyl]pyridine-3-carboxamide 1-[4-fluoro-2-(trifluoromethyl)phenyl]-N,N'-dimethylethane-1,2-diamine N-(3,5-dimethoxyphenyl)-1H-pyrrole-2-carboxamide N-[2,6-dichloro-3-(1H-indole-2-carbonyl)phenyl]-4-methylbenzenesulfonamide (3S)-4-[2-(4-fluorophenyl)ethyl]-2,3,5-trimethoxyoxane 2-(5-azidopyridin-2-yl)oxy-6-methylsulfanylpyrazine N-(1-aminoisoquinolin-6-yl)formamide;hydrochloride 4-[3-[(6-chloro-2,3-dihydroindol-1-yl)methyl]furan-2-carbonyl]-3-methylpiperazin-2-one 3-(4-pyridin-2-yloxypiperidin-1-yl)benzonitrile 7-(3,4-dihydroxyphenyl)-2-[1-(2-piperidin-1-ylethoxy)propan-2-ylamino]thieno[3,2-b]pyridine-5-carboxamide 2-methyl-5-[4-(trifluoromethoxy)phenyl]-1,3,6,8a-tetrahydrocyclopenta[c]azete N-[2-(1H-indol-3-yl)ethyl]-4-nitro-N-phenylbenzamide 4-[2,3,5,6-tetradeuterio-4-hydroxy-6-(1H-imidazole-5-carbonyl)phenyl]benzonitrile N-cyclohexyl-2,5-dimethylpyrazolo[1,5-a]pyridine-3-carboxamide 5-(3,4-dimethoxyphenyl)-2-(3-methylbutanoylamino)thiophene-3-carboxylic acid;1-(methylamino)propane 1-azido-2,3-diphenylimidazolidine 3-bromo-N-cyclopropyl-4,6-dimethoxy-N'-(2,4,5-trifluorophenyl)benzenecarboximidamide 2-(4,6-diphenylpyridin-2-yl)-5-methylpyrimidine N-[(2,3-difluorophenyl)methyl]-N'-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]oxamide 2-[3-chloro-4-(5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonyl)phenoxy]acetamide 4-[3-(2,2-dimethylpropanoylamino)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-2-yl]benzamide 4-chlorobenzenethiol;1-[2,6-dimethyl-5-(2H-tetrazol-5-yl)pyrimidin-4-yl]-N,N-dimethylpiperidin-4-amine 5-[(E)-2-(3,4-difluorophenyl)ethenyl]-6-ethyl-4-hydroxypyran-2-one 4-(1,3-dimethylimidazol-1-ium-2-yl)benzonitrile 3-[4-(4-methylpiperazine-1-carbonyl)phenyl]thiophene-2-carboxamide 6-[3,5-bis(trifluoromethyl)phenyl]-2H-quinolizine N-[(2S)-5-[(4aS,6R)-8a-ethyl-1,3,4,4a,5,6,7,8-octahydroisoquinoline-2-carbonyl]-2-benzamido-4-oxopentanoyl]-N-(3-cyanophenyl)azetidine-3-carboxamide 2-ethylsulfanyl-5,6,7,8-tetrahydroquinazoline;hydrochloride N-[(2R)-1-[4-chloro-3-[2,6-dimethyl-4-(5-oxopyrrolidin-3-yl)phenyl]anilino]-3-hydroxypropan-2-yl]acetamide 3-azido-2-(4-chlorophenyl)sulfanyl-N-methylpropanamide N-(3-methylbutanoyl)-N-(2,4,6-trichlorophenyl)butanamide 4-(chloromethyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile N-[1-(8-fluoroquinolin-4-yl)cyclopentyl]-6-methoxypyridine-3-sulfonamide N-[5-(1,3,4,4a,5,6,7,8,8a-octahydroisoquinoline-2-carbonyl)-6-cyclopropyloxypyridin-3-yl]-4-methylbenzamide 2-azidooxy-3,5-dimethylsulfonylpyridine 5-chloro-2-N,4-N-bis[4-(dimethylamino)phenyl]pyrimidine-2,4-diamine 2-[(E)-[3,5-dimethyl-4-[3-oxo-4-phenyl-1-(pyridin-4-ylmethyl)piperazin-2-yl]iminohexylidene]amino]guanidine 2-(9,10-dioxoanthracen-1-yl)oxycarbonylbenzoic acid (E)-N-[2-[4-fluoro-5-(hydroxymethyl)-6-oxooxan-3-yl]ethynyl]-6,10,11-trioxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide 4-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-N-[(E)-1,3-dimethoxypropan-2-ylideneamino]pyridine-2-carboxamide 5-(2-hydroxyethyl)-2,4-dimethoxybenzamide 2-[4-[(1Z)-buta-1,3-dienyl]-5-methoxy-1H-pyrrol-3-yl]-N-[(1S)-1-(4-cyanophenyl)ethyl]acetamide N-[6-(3,4-difluorophenyl)imidazo[1,2-a]pyrazin-8-yl]piperazine-1-carboxamide;2-methoxyacetaldehyde N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-2-[2-oxo-2-(4-pyrrolidin-1-ylpiperidin-1-yl)ethyl]sulfanylacetamide N-(4,4-dimethylcyclohexyl)-3-oxo-1H-isoindole-2-carboxamide ethane;2-[4-[2-fluoro-6-methyl-3-(methyliminomethyl)phenoxy]butoxy]ethanol 3-[4-(aminomethyl)phenyl]thiophene-2-carboxylic acid;hydrochloride 3-methoxy-4-[2-(4-propylphenyl)ethynyl]aniline 2-[2,5-dichloro-N-(cyanomethyl)anilino]acetamide 1-[5-[(Z)-2-amino-3,4-dimethylpent-2-enoyl]thiophen-2-yl]ethanone 4-[[3-(4-fluorophenyl)imidazo[1,2-b]pyridazin-6-yl]methylamino]pyridine-2-carboxamide 2-[6-chloro-4-(1,5-dimethylpyrazol-3-yl)pyridin-2-yl]sulfanyl-N-(2-hydroxy-2-phenylethyl)acetamide 1-cyclohexyl-2-[4-(3,5-dimethylpyridin-4-yl)phenyl]ethanone;methane N-[(2,3,4,5,6-pentachlorophenyl)methyl]heptan-1-amine 2-bromo-4,5-difluoro-6-[[3-(trifluoromethyl)phenyl]methoxy]pyridine-3-carboxylic acid 2-[(2-butoxy-2-oxoethyl)-(4-chlorophenyl)sulfonylamino]benzoic acid 5-[4-fluoro-3-(2H-tetrazol-5-yl)phenyl]imidazolidine-2,4-dione 2-[2-(1,3,4-thiadiazol-2-ylamino)ethoxy]benzoic acid 2-methylbutane;6-(3,4,5-trichlorophenyl)naphthalene-1,4-dione (5Z)-2-(4-chlorophenyl)imino-5-[(1,3-diethoxy-5-nitropyrrol-2-yl)methylidene]-1,3-thiazolidin-4-one 2-(1,3-benzodioxol-5-yl)-6-methoxy-4,9-dihydro-3H-pyrazino[1,2-a]indole;N,N-dibutylcyclohexanamine 2-[N-(1,3-diethoxypropan-2-yl)-4-hydroxyanilino]acetic acid (3S)-3-methyl-1,2,5,6,7,8-hexahydropyrido[1,2-a]benzimidazole 1-bromo-3-chloroindole N-[2-(5-amino-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl)ethyl]-3,4-dimethoxybenzamide;hydrochloride (3R)-3-[(2S,4R)-5-hydroxy-4-methylpentanoyl]oxy-2-oxo-4-phenylbutanoic acid 5-(2-chloropyridin-4-yl)-3H-1,3-benzoxazol-2-one 5-chloro-N,4-dimethyl-2-(3-nitroanilino)benzamide 2-[[4-(2-hydroxyethyl)piperazin-1-yl]methyl]-3H-quinazolin-4-one 1-[2-(3,4-dihydroxyphenyl)quinazolin-4-yl]piperidine-3-carboxylic acid [1-ethylsulfonyl-3-(4-methoxyphenyl)indol-2-yl]urea 7-(1H-imidazol-5-yl)-2,3-dihydrothieno[3,4-b][1,4]dioxine (E)-3-[4-[2-amino-6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-ylamino)pyrimidin-4-yl]phenyl]prop-2-enamide (3R)-1-[5,6-difluoro-2-(propylaminomethyl)-2H-quinazolin-1-yl]azepan-3-ol 3-(2,6-dichloropyridin-4-yl)-5-oxo-7H-imidazo[1,2-c]imidazole-8-carbonitrile 6-[[(1R,2S)-2-hydroxycyclohexyl]amino]pyridazine-3-carboxamide 5-chloro-2-[(E)-1H-pyrrol-3-ylmethylideneamino]oxybenzoic acid 4-(2,6-difluorophenyl)-N-[5-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]pyridin-2-amine N-cyclohexyl-2,4-dinitro-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)aniline (2R)-1-[(3-benzylquinolin-4-yl)amino]-N-cyclohexylpropane-2-sulfonamide N-[6-(difluoromethyl)-3-nitropyridin-2-yl]-1H-pyrazole-5-carboxamide 4-chloro-5,6-difluoro-2,3-dihydroquinoline 4-[(4-methoxyphenyl)-(2,3,4,5,6-pentafluorophenyl)boranyl]benzoic acid 5-[2,4-difluoro-3-(trifluoromethoxy)phenyl]-1H-pyridin-2-one 6-amino-7-(3-hydroxynaphthalen-2-yl)iminoheptanoic acid 2-[4,5-bis(4-methylphenyl)-1H-imidazol-2-yl]-N-[3-bromo-5-(3-methoxy-3-oxopropanoyl)thiophen-2-yl]benzamide 2-cyclobutylsulfanyl-6-(2,4-dimethoxypyrimidin-5-yl)-8-[3-(trifluoromethyl)pyrazol-1-yl]pteridin-7-one 3-(5-carbamoyl-2-methoxyphenyl)propylcarbamic acid N-cyclohexyl-4,5-dimethyl-3-(6-propan-2-yloxypyridine-2-carbonyl)-1H-pyrrole-2-carboxamide 3-[(4-methoxy-6-methylpyridine-2-carbonyl)amino]propanoic acid N-methoxy-6-(2,3,5-trichlorophenoxy)hexanamide 2-N-[1-(3,4-difluorophenyl)butyl]pyrido[3,4-d]pyrimidine-2,4-diamine;ethane (3E)-4-amino-3-[[2-(2-chlorophenyl)sulfanylphenyl]methylidene]azete-2-thione 5-amino-7,8-difluoro-6H-imidazo[1,2-c]quinazoline-9-carboxylic acid 4-amino-6-chloro-3H-1,5-benzothiazepine-2-thione (E)-N,3-dimethyl-2-[4-methyl-1-oxo-3-phenyl-6-(3,3,3-trifluoroprop-1-ynyl)isoquinolin-2-yl]pent-3-enamide 3-[3-(3,5-difluorophenyl)propanoyl]chromen-2-one 5-(1H-imidazol-2-ylsulfonyl)benzenethiol 2-(N-ethenylsulfonylanilino)benzenesulfonic acid 4-[3,5-di(nonoxy)phenoxy]butan-1-ol (6R)-7-acetyl-10-ethoxycarbonyl-3-hexylsulfanyl-1-propanoyl-8,9-dihydropyrido[1,2-a]indole-6-carboxylic acid 2-azidooxycarbonylbenzoic acid N-(3,4-difluorophenyl)sulfonyl-N'-[5-methyl-1-[(4R)-oxepan-4-yl]pyrazolo[3,4-b]pyridin-4-yl]pentanediamide 2-N-[1-(3,5-dimethoxyphenyl)ethyl]pyrimidine-2,4-diamine N-[2-methoxy-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]methanesulfonamide N-[5-(2,6-dioxopiperidin-3-yl)-1,3,4-thiadiazol-2-yl]acetamide N-cyclopropyl-3,5-dimethoxy-2-(4-phenylanilino)benzamide 2-(7-bromoquinolin-4-yl)sulfanylacetohydrazide 3-[(2S,4R)-1-benzyl-4-[(4,6-dimethoxypyrimidin-5-yl)amino]pyrrolidin-2-yl]-1H-4,1,2-benzodioxazole-7-carboxylic acid N-[(4-fluorophenyl)methyl]-7-methoxy-1-[(3S,5R)-5-methyloxolan-3-yl]benzimidazole-2-carboxamide 3-(1H-benzimidazol-2-yl)-N-[6-[[4-[2-(1,5-dimethylpyrazol-3-yl)ethynyl]benzoyl]amino]hexan-3-yl]propanamide 2-[(3E)-3-chloropenta-1,3-dien-2-yl]oxycarbonylbenzoate 2-[4-(1H-indol-3-yl)pyrazol-1-yl]-2-methylpropanamide 2-[[4-(3,5-diphenyl-1H-1,2,4-triazol-4-ium-2-yl)-1,6-naphthyridin-7-yl]amino]pyridine-3-carbonitrile 7-(3,5-dimethylphenyl)-N-(4-fluorophenyl)-6-(methoxymethyl)-1H-pyrrolo[2,3-c]pyridin-4-amine 2-[(4S,5R)-3,3-difluoro-1-methylpiperidin-4-yl]-N-methyl-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 4-(2,6-difluorophenyl)-N-[3-fluoro-4-(2H-pyridin-1-ylmethoxy)phenyl]-5-(trifluoromethyl)pyrimidin-2-amine 4-[2-(5,6-dimethylpyrazin-2-yl)propanoyl]morpholine N-[4-[[[(2R)-1,4-dioxan-2-yl]methylamino]methyl]cyclohexyl]-5-ethoxy-6-fluoro-2-hydroxy-3-methoxybenzamide 1-[6-(dimethylsulfamoyl)pyrimidin-4-yl]pyrrolidine-3-carboxylic acid 2-azido-3,5-dibromopyridine 3,4-difluoro-2-(2-hydroxyethylamino)benzoic acid 2-(4-bromophenyl)-3,3a,5,6a-tetrahydro-1H-cyclopenta[c]pyrrole 2-[1-[(3R)-3-hydroxypyrrolidine-1-carbonyl]pyrazol-4-yl]-6H-pyrrolo[3,4-b]pyridin-5-one 2-(4-azido-3,5-dimethylphenyl)acetonitrile N-[4-chloro-3-(1,3-oxazole-5-carbonyl)phenyl]-2-fluorobenzamide 2,6-bis(4-fluorophenoxy)benzene-1,3,5-tricarbonitrile N-ethenyl-6,7-dimethoxyquinazolin-4-amine 2-[5-[(3,4-dihydroxyphenyl)methyl]pyridin-2-yl]-1H-pyrimidine-2,4-diol 2-[2,3-difluoro-4-(trifluoromethyl)phenoxy]naphthalene 5-methoxy-2,4-dinitrobenzoic acid;1-[1-(4-nitrophenyl)cyclopropyl]pyrrolidine (5Z)-2-[4-bromo-3,5-bis(trifluoromethyl)phenyl]imino-5-[(3-nitrophenyl)methylidene]-1,3-thiazolidin-4-one 2-[4-(1,3-benzothiazol-6-yl)piperazin-1-yl]-N-phenylacetamide;dihydrochloride (4Z)-N'-[5-[amino-[(Z)-2-aminoethenyl]amino]pyridin-3-yl]-N,1,7-trimethyl-6-propan-2-ylidenepurine-2-carboximidamide 4-amino-N-(3,4-dimethoxyphenyl)-5-ethylsulfanyl-1,2-thiazole-3-carboxamide 2-(2,3-dihydrofuro[3,4-b]pyridin-1-yl)-6-methoxypyrimidin-4-amine 4-bromo-2,5-dimethyl-3-(1H-pyrrol-3-yl)-2-[3-(trifluoromethoxy)phenyl]furan 2-(N-cyclohexyl-4-fluoroanilino)decanoic acid N-[3-(2-aminopyrimidin-4-yl)phenyl]-3,4-dichlorobenzenesulfonamide (2R)-2-ethenyl-5-fluoro-3,4-dihydrochromene-2,7-diol 2-[4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl]-4,5-dihydrothieno[3,2-d][1]benzazepine-6-carboxylic acid 1-(cyclohexylmethylamino)-3-(naphthalen-2-ylsulfanylmethyl)thiourea N-[1,4-bis(ethenyl)cyclohexa-2,4-dien-1-yl]-6,7-dimethoxy-5H-quinazolin-4-amine 1-(6-ethyl-2,3-dihydroindol-1-yl)-2-[5-methoxy-7-(4-methylimidazol-1-yl)thieno[3,2-b]pyridin-2-yl]ethanone 1-(2-benzoyl-4,5-dimethylphenoxy)-3-morpholin-4-ylpropan-2-one 2-cyclopentyl-3,5,7,8-tetramethoxychromene-4,6-dione 6-[5-cyclopropyl-4-(oxan-2-ylmethoxy)pyridine-3-carbonyl]-8a-ethyl-1,5,7,8-tetrahydro-[1,3]oxazolo[3,4-a]pyrazin-3-one 1-chloro-4-(disulfanyl)benzene;propane 5-[4-(difluoromethoxy)phenyl]thiophene-2-carboxylic acid ethane;N-[3-(1H-imidazol-5-yl)-2,6-dimethoxyphenyl]acetamide 4-[[6,8-dibromo-2-(4-phenylbutoxy)quinazolin-4-yl]amino]-3,5-dimethylbenzonitrile 4-[(3S,7R)-5-oxo-2-oxa-9-azatricyclo[12.4.0.03,8]octadeca-1(18),14,16-trien-9-yl]benzoic acid 1,5-dibromocyclohexa-1,3-diene;ethane 2-[1-[5-chloro-6-methyl-3-(triazol-2-yl)pyridin-2-yl]pyrazol-4-yl]acetaldehyde N-[3-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl]pyrazine-2-carboxamide (Z)-3-[6-bromo-5-methyl-1-[2-(oxan-4-yloxy)ethyl]indol-2-yl]prop-2-enal;fluoromethane (3R,4R)-4-[3,5-difluoro-2-[[2-methyl-6-[methyl(oxan-4-yl)amino]pyrimidine-4-carbonyl]amino]phenyl]piperidine-1-carboxylic acid 2-[5-(aminomethyl)pyridin-3-yl]-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-b]azepine-3-carbonitrile 1-(3,5-dimethylpiperazin-1-yl)-2-[4-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)piperidin-1-yl]ethane-1,2-dione 5-(2-iodophenyl)-7H-imidazo[1,2-b]pyridazine 2-[2-[5-fluoro-6-[3,4,5-trideuterio-7-(morpholin-4-ylmethyl)naphthalen-1-yl]oxypyridin-2-yl]oxan-4-yl]acetic acid [1-[2,6-dimethyl-4-(3-oxopropoxy)phenyl]pyrrol-3-yl]oxyboronic acid [(Z)-1H-indol-3-ylmethylideneamino]thiourea N-[2,6-dimethyl-4-(3-pyridin-3-ylphenyl)sulfanylphenyl]acetamide [1-(5-fluoro-2-propan-2-ylphenyl)sulfonylazetidin-3-ylidene]methanediol N-[(2-cyclohexylpyridin-3-yl)methyl]-1,5-naphthyridine-4-carboxamide 2-hydroxy-N,5-bis(4-methoxyphenyl)benzenesulfonamide 2-methyl-3,4-diphenylpentanoic acid [(Z)-3,5-diphenylhex-1-enyl]hydrazine 5-hydroxy-3-(2H-isoindol-1-yl)piperidine-2,6-dione (2-cyclopentyloxypyridine-3-carbonyl)iminoazanide N-[2,6-difluoro-3-(propylsulfanylamino)phenyl]thieno[3,2-d]pyrimidine-7-carboxamide 4-(dimethylcarbamoyloxy)benzenesulfonic acid 2-[1,6-diamino-4-(3-methoxyphenyl)cyclohexa-2,4-dien-1-yl]guanidine N-[3-[(3,4-dichlorophenyl)methylamino]-2-nitrophenyl]-1,5-naphthyridine-2-carboxamide 2-[(1R)-1-cyclohexa-2,4-dien-1-ylpropoxy]naphthalene N-[3-(2-amino-1,5-dicyano-6-oxopyridin-3-yl)phenyl]benzamide 2-[(5R)-3-cyclopropyl-7-fluoro-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]phenol 3-[4,5-dimethoxy-2-(2-methylphenyl)benzoyl]chromen-4-one N-(4,7-dimethyl-1,2,3,5-tetrahydro-s-indacen-6-yl)-3-[2-methylpropylsulfanyl(sulfinatoamino)methylidene]azetidine 3-ethyl-2-(3-methoxyphenyl)quinazolin-4-one 1-(4,5-dichlorocyclohexa-2,4-dien-1-yl)sulfonyl-N-methylpiperidine-3-carboxamide 2-[4-(trifluoromethoxy)phenyl]-1,3-dihydroimidazo[4,5-b]pyridine 5-azidooxycarbonyl-6-methylpyridine-2-carboxylic acid [4-(3,6-dimethyl-1-phenylpyrazolo[3,4-b]pyridine-4-carbonyl)piperazin-1-yl]-(4-ethoxy-2,5-dimethylphenyl)methanone 2-[6-[(2R)-2,4-dimethylpiperazine-1-carbonyl]-3H-imidazo[4,5-c]pyridin-2-yl]acetamide 2-chloro-4-[(Z)-[(4,6-diphenylpyrimidin-2-yl)hydrazinylidene]methyl]phenol N-[1-[(3R)-6-hydroxy-5,8-dimethoxy-1-oxo-2,9a-dihydroimidazo[1,2-c]quinazoline-3-carbonyl]piperidin-4-yl]-N-methylacetamide 4-chloro-N-(2,3-dihydrofuro[3,2-b]pyridin-7-yl)benzamide 4-chloro-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-6-phenylsulfanylpyrimidin-5-amine 4-(4,5,6-tribromopyridin-2-yl)morpholine 2-(4-fluorophenyl)-7-[(3S,5R)-3,4,5-trihydroxyhexyl]-3H-pyrrolo[3,4-b]quinolin-1-one 5-chloro-N-(2,3-dihydroxypropyl)-N-[2-methoxy-4-methyl-6-[(1R)-1-phenylethyl]pyridin-3-yl]thiophene-2-carboxamide 1-[5-[(4-fluorophenoxy)methyl]furan-2-carbonyl]pyrrolidine-3,4-dicarboxylic acid 4-(aminomethyl)-6,7-dihydrobenzo[a]quinolizin-5-ium 2-[3,5-dichloro-4-[(2-methylquinolin-8-yl)oxymethyl]phenyl]cyclohexane-1-carboxylic acid 2-[4-(3-bromopyridin-4-yl)phenyl]-3,8a-dihydroisoindole-1,3-dione 2-[4-[(1R)-2-oxocyclopentyl]phenyl]acetonitrile N-[4-methoxy-6-(pyrazole-1-carbonyl)-1,2-benzoxazol-3-yl]acetamide 1,4-dimethoxynaphthalene;ethane 2-[(3-chlorobenzoyl)amino]-5-methoxy-4-phenylthiophene-3-carboxylic acid 2-(3,4-dimethoxyanilino)quinoline-5,8-disulfonic acid 4-[(2E,4Z)-3-methylhepta-2,4,6-trien-2-yl]oxyaniline 3-(2,4-dichlorophenyl)sulfanyl-1-(1H-pyrrol-3-ylmethyl)pyrrolidine 4-(5,6-dihydro-1H-indol-3-yl)aniline 2-[4-methylsulfanyl-5-(2,2,3,3,4-pentafluorobutoxy)pyrimidin-2-yl]ethanol 2-[3,4-dichloro-5-(trifluoromethyl)phenyl]cyclopropane-1,1-dicarbonitrile (E)-1-[(5S,7R)-2-butylsulfanyl-5-phenyl-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazol-7-yl]-3-pyridin-3-ylprop-2-en-1-one 2-[2,4-difluoro-N-(1,3-thiazol-5-yl)anilino]acetic acid 1-(3,5-dibromophenyl)ethylurea;ethane 4-[6-(1H-pyrazol-5-yl)imidazo[2,1-b][1,3]thiazol-3-yl]phenol 3-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]benzonitrile 4-(1,3-benzothiazol-2-yl)cyclohexa-1,5-diene-1-sulfonic acid 1,6-dimethyl-2-oxo-5-[3-(trifluoromethoxy)phenyl]pyrimidine-4-carboxylic acid (2S)-3-[4-(4,6-dimethoxy-5-methylpyrimidin-2-yl)phenyl]-2-(1H-indol-3-ylmethylideneamino)propanoic acid 2-[4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)morpholin-3-yl]acetic acid 1-(2,5-difluorophenyl)-3-[4-fluoro-2-(trifluoromethyl)phenyl]propan-1-amine 6-methyl-3-(2,4,5-trifluorophenyl)-1H-pyrimidine-2,4-dione 3-hydroxy-4-methylpentane-1,2-dione;N-(2-propan-2-ylphenyl)acetamide 2-(3,4-dichlorophenyl)-N-[1-[4-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)cyclohexanecarbonyl]piperidin-4-yl]acetamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-hydroxy-N-methyl-2-phenylacetamide 2-[5,7-dichloro-2-(3-methylphenyl)quinolin-4-yl]propanoic acid 3-(2-methoxyethyl)-5,10,13-triazatricyclo[7.4.0.02,6]trideca-1(9),2(6),3,11-tetraen-12-one N-methyl-4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]benzamide 7-[(3R)-3,4-dimethylpiperazin-1-yl]-2-hydroxy-N-[4-hydroxy-3-(trifluoromethoxy)phenyl]-6-nitropyrido[1,2-a]pyrimidin-4-one 3-(2,5-dimethylpyrrolidin-1-yl)sulfonylpyridine 1-(2,5-dimethoxyphenyl)octane-1,1,4,4-tetraol 4-(2,1,3-benzothiadiazol-5-yl)-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 5-[(1R)-2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-oxoethyl]imidazolidine-2,4-dione [5-chloro-4-[2-(methylamino)pyridin-4-yl]pyridin-3-yl]-[4-(cyclopropanecarbonyl)piperazin-1-yl]methanone 2-chloro-5-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-ylamino)benzamide 2-[6-(6,7-dimethoxyquinolin-4-yl)oxypyridin-3-yl]acetic acid 2-(4-chlorophenyl)-3,5-diphenyl-3,6-dihydroimidazo[4,5-d]pyridazine 3-[4-(4,6-diphenylpyrimidin-2-yl)phenyl]phenol 1-(2,3-dihydro-1H-inden-5-yl)ethanone;ethane N-(2-bromophenyl)sulfanyl-2,4-dichloro-6-fluoroaniline (E)-N-tert-butylsulfanyl-1-[4-[[2,3-bis[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyridine-7-carbonyl]amino]piperidin-1-yl]methanesulfinamide;ethane 3-(2,6-difluorophenyl)-1-(3-hydroxypropyl)piperidine-4-carboxylic acid 2-(3,4-dimethoxyphenyl)-3-(3-methylphenyl)-6,7,8,9-tetrahydro-5H-[1,2]oxazolo[5,4-b]quinoline 2-methyl-4-[(3S)-1-[6-oxo-5-(trifluoromethyl)-1H-pyridazine-3-carbonyl]piperidin-3-yl]-1H-pyrimidin-6-one 1-[2,6-di(propan-2-yl)phenyl]-3-[4-(2,5-dimethylphenyl)-1H-pyrrol-3-yl]urea 2-(3-butylphenoxy)quinoline 6-(3,5-dimethoxy-2H-pyridin-1-yl)-1-ethyl-4-hydroxy-N-[5-(5-methylpyridin-2-yl)pentan-2-yl]pyrrolo[2,3-c]pyridine-3-carboxamide 3-(4,5-dimethyl-1H-pyrazole-3-carbonyl)-1,3,6,7,8,9,10,11,12a-octahydropyrido[2,1-a][2]benzazocine-2,4-dione (1S)-6,7,8-trimethoxy-5H-anthracene-1-carboxylic acid 2-[4,5-dimethoxy-3-[[4-(trifluoromethyl)anilino]methyl]indol-1-yl]acetic acid [2-azido-1-(4-tert-butylphenyl)ethoxy]methanethiol 3-[(4-chlorophenyl)methyl]-1-hexanoylpiperidine-2,6-dione 6-hydroxy-5-methyl-1,3-diphenyl-2H-pyrazolo[4,3-d]pyrimidin-7-one 6-bromo-4-[1-(3,5-dichloropyridin-2-yl)ethylamino]-8-methylpyrido[2,3-d]pyrimidin-7-one;ethane N-[2,5-difluoro-4-(3-oxo-1H-isoindol-2-yl)phenyl]-6-hydroxy-7-methoxyphthalazine-4-carboxamide 2-bromo-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-ylmethyl)benzamide [(2S,4R)-1-[[5-methyl-3-(6-methylpyridin-3-yl)triazolo[4,5-d]pyrimidin-7-yl]amino]-4-propoxypyrrolidine-2-carbonyl]oxidanium 2-[4-bromobutan-2-yl(propyl)amino]benzenesulfonic acid N-(1,1,2,2,3,3,4,4,5,6,7,8,8,9,9a-heptadecafluorononyl)-4-(trifluoromethyl)benzamide 4-amino-3,5,6-trichlorophthalic acid 2-(4,4,5,5,6,6,7,8,8,9,10,11,12,13,14,15,16,17-heptadecafluorooctyl)phenol (2-fluoropyridine-3-carbonyl)-methylidenephosphane [2-(1-azidopiperazin-2-yl)-5-fluoropyrimidin-4-yl]hydrazine 2-[(E)-hex-4-en-3-yl]-5,7-dimethoxy-6H-quinoline 1-(1,4-dihydropyridin-2-yl)-N-[1-[5-fluoro-6-(2-methoxyethoxy)-7-phenylmethoxyquinazolin-4-yl]pyrrolidin-3-yl]cyclopropane-1-carboxamide 3-[6-(azetidin-1-yl)purin-9-yl]propanal 5-azido-7-methoxy-6-(3,4,5-trifluorophenyl)quinazoline N-[5-(cyclopropylmethoxy)pyridin-2-yl]-6-methyl-8,9-dihydro-7H-pyrimido[4,5-b]azepin-4-amine;fluoroethane 2-[4,6-dichloro-5-(trifluoromethyl)pyrimidin-2-yl]sulfanyl-1-phenylethanone 4-[(5S,10bS)-2-chloro-7-methoxy-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-9-yl]-N-tert-butylbenzenesulfonamide N-(1H-indol-5-yl)-4-[[2-(pyridin-3-ylmethoxymethyl)piperidin-1-yl]methyl]benzamide 5-[(4-methoxybenzoyl)amino]-2-[3-(2H-tetrazol-5-yl)piperidin-1-yl]benzoic acid;2,2,2-trifluoroacetic acid 4-[6-(2,4,6-trimethylphenoxy)hexyl]benzene-1,3-diol N-azido-1,2,3,4-tetrahydroisoquinoline-6-carboxamide 2-[6,11-dimethyl-10-(1H-pyrazol-5-yl)-3,5,8,10-tetrazatricyclo[7.3.0.02,4]dodeca-1,3,6,8,11-pentaen-9-yl]propanoic acid (2R,3S)-3-[2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]-N'-pyridin-2-ylmorpholine-2-carbohydrazide (4-azido-1,3-diazetidin-1-yl)-[2-chloro-5-(3-chlorophenoxy)phenyl]methanone (1R,2S)-2-[4-[3-(1H-indol-6-ylmethoxy)phenyl]phenyl]cyclopropane-1-carboxylic acid 4-[3,5-dichloro-4-[(5-methyl-4-oxo-2,3-dihydrochromen-7-yl)oxy]phenyl]piperazine-1-carboxylic acid 1-(5-bromo-3,4-dihydroxy-2-methylphenyl)ethanone;N-but-3-yn-2-ylidenecyclohexa-2,4-diene-1-sulfonamide (1S,4R)-N-[2-(3-hydroxyazetidin-1-yl)pyrimidin-5-yl]-4-methoxy-1-methyl-2,3-dihydro-1H-indene-5-sulfonamide [(2S)-6-cyclopentyloxy-3,4-dihydro-2H-chromen-2-yl]methanamine 2-[4,5-bis(4-chlorophenyl)imidazol-1-id-2-yl]pyridine;iridium(3+) N-(3,5-difluorophenyl)-2-[(6R)-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 4-[1-(5,7,8,10,11-pentazatricyclo[7.4.0.02,6]trideca-1(13),2,4,6,9,11-hexaen-13-yl)piperidin-3-yl]phenol 4-[6-(4-methoxyphenyl)pyridazin-3-yl]piperazine-1-carboxylate 1-(2,4-difluorophenyl)-6-hydroxy-5-[(3R)-2-iminopiperidin-3-yl]pyrimidine-2,4-dione [(2S)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]carbamic acid 2-[5-[4,7-dichloro-6-(3-hydroxypropyl)quinazolin-2-yl]-1,3-thiazol-2-yl]phenol 1-[(3,5-dimethylphenyl)sulfanylamino]-N-methoxycyclopentane-1-carboxamide 2-methyl-1,3-bis(4-methylcyclohexa-1,5-dien-1-yl)benzene 5-(1,3-benzodioxol-4-yl)-N-[2-[2,6-di(propan-2-yl)phenyl]iminobut-3-en-2-yl]pyridine-3-carboxamide 2-[(6R)-2,6-dimethyloxan-4-yl]sulfanyl-7H-purine 2-[4-chloro-N-(3-methylbutyl)anilino]acetic acid 2-[(2E,5S)-2-[(Z)-1-(4-fluorophenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid [1-[6,7-dichloro-5-(2-fluorophenyl)-4-oxoquinazolin-3-yl]-3-methylidenepentan-2-yl]carbamic acid 4-[(3R)-1-(cyclopropanecarbonyl)piperidin-3-yl]-2-methyl-1H-pyrimidin-6-one 5-bromo-2-methylsulfonylpyridine 1-[(E)-3-cyclopentyloxy-2-methanimidoylprop-2-enyl]imidazole-4,5-diamine 4-[6-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]-9H-carbazol-3-yl]benzonitrile 1-[(3R)-3-[4-amino-5-[4-fluoro-2-(propan-2-yloxymethyl)phenyl]pyrrolo[2,1-f][1,2,4]triazin-7-yl]pyrrolidin-1-yl]prop-2-en-1-one 6-azido-4,5-dihydro-1H-1,3-benzodiazepine-2-carboxamide [4-azido-2,6-dichloro-3-(trifluoromethyl)phenyl]methanol 5-[(4-methylsulfanylphenyl)methylidene]-2-propylimino-1,3-thiazolidin-4-one (2S)-3,4-dihydroxy-1-(phenylmethoxycarbonylamino)butane-2-sulfonic acid 1-[2,5-di(propan-2-yl)phenoxy]pyrazole (2S)-N-[[3-fluoro-5-[2-[[(1R,2R)-1-hydroxy-4-methylsulfanylbutan-2-yl]amino]pyrimidin-4-yl]phenyl]methyl]oxolane-2-carboxamide (5S)-3-[4-[[1-(4-morpholin-4-ylsulfonylphenyl)cyclopropanecarbonyl]amino]-3-nitrophenyl]-5,6-dihydro-1H-pyrrolo[2,3-b]pyridine-7-carboxamide N-(1-bromobut-3-ynyl)-5-chloropyridine-2-sulfonamide N-methylsulfonyl-2,4,6-trinitro-N-(4-phenoxyphenyl)benzamide 4-(dibenzylamino)-5,6-bis(2-methylbutanoylamino)naphthalene-1,7-disulfonate 2-ethyl-4,7-dimethoxy-1H-benzimidazole ethane;methanamine;(1R)-N-methyl-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide N-(diaminomethylidene)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carboxamide;hydrochloride N-(3-hydroxypropyl)-2-[(4S)-1-[4-(2-methoxyphenyl)benzoyl]-3,4-dihydro-2H-quinolin-4-yl]acetamide 6-fluoro-7-(2,3,4,5,6-pentamethylphenyl)chromene-2,8-dione 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-7H-pyrrolo[2,3-d]pyrimidine 2-[1-azidoethyl(propan-2-ylamino)amino]aniline (4S)-1-tert-butyl-3,3-difluoro-4-(2-pyrimidin-5-ylpyridin-4-yl)piperidine-4-carboxylic acid 5-[4-(azidooxymethyl)phenoxy]benzimidazole [2-hydroxy-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methanol (2R)-N,N-diethyl-1-methylsulfonyl-4-[4-phenyl-5-(trifluoromethyl)pyrimidin-2-yl]piperazine-2-carboxamide 2-bromo-N-(1,5-dimethylpyrazol-3-yl)-N-[(4-oxo-3H-quinazolin-2-yl)methyl]benzamide 3-[(2-chloro-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carbonyl)amino]-1,1a,9b-tetrahydrocyclopropa[a]naphthalene-1-carboxylic acid 3-methyl-6,8a-dihydroisoindolo[2,1-a]indole N-[3-methylbutyl-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)amino]propanamide 2-[1-(4-cyclopropylphenyl)sulfonylpiperidin-3-yl]oxypyridine 2-(4-bromophenyl)-5-[(3S,7R)-7-hydroxy-8-(3-methylbut-2-enoyloxy)octyl]-1,3,4-oxadiazole-6-carboxylic acid 5-[4-chloro-2-(trifluoromethyl)phenyl]sulfanyl-6,8-dihydro-5H-imidazo[1,5-a]pyrazine (E)-N-benzylbut-2-enamide;3,3-dimethylpentanal 2-[(E)-2-cyano-3,3,3-trifluoroprop-1-enyl]benzoic acid 4-[2-(furan-2-yl)-1H-indole-3-carbonyl]morpholin-3-one 7-(4,6-dicyclohexyloxypyrimidin-5-yl)-N-[(2E,3Z)-2-ethylidenehexa-3,5-dienyl]pyrido[2,3-d]pyridazin-8-amine 4-chloro-N'-hydroxy-3-[(5S)-5H-imidazo[5,1-a]isoindol-5-yl]benzenecarboximidamide 2-[(6R,11bS)-4-acetyl-3-methoxy-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-7-yl]-1-(4-fluorophenyl)ethanone 5-[(E)-(2,4-dioxoquinazolin-1-yl)iminomethyl]benzene-1,3-diol 1-(4,5-dihydroimidazol-1-ylmethyl)isoquinoline 7-(1,3-benzodioxol-5-yl)-4-[[cyclobutylidenemethyl(ethyl)amino]methyl]chromene-2-thione [5-chloro-3-(trifluoromethyl)pyridin-2-yl]boronic acid 3-chloro-2,5-dimethyl-6H-pyrazolo[4,3-d]pyrimidine-7,8-dione 5-[(2E,4Z)-hexa-2,4-dienyl]-10-phenylacridin-9-one 3,4-dimethylnaphthalene;ethane N-[(1R)-2-cyclobutyloxyspiro[1,3-dihydroisoquinoline-4,1'-cyclopropane]-6-yl]-6-fluoropyridine-3-carboxamide 4-chloro-1-[(2R)-3-methoxybutan-2-yl]pyrazole 4-ethyl-1,3-diethyl-7-methoxyquinoxaline-2,5-dione (E)-4-chlorobut-2-ene;N-methyl-3,7-diphenylpyrazolo[1,5-a]pyrimidin-5-amine 5-[4-fluoro-3-(1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]-N-propan-2-ylpyridin-3-amine 6-(2,3-dimethylphenyl)iminocyclohexa-1,4-diene-1-carboxylic acid N-[1,3-dihydroxy-5-(4-methylphenoxy)cyclohexa-2,4-dien-1-ylidene]propane-2-sulfonamide 2-methyl-N-(3-phenylpropanoyl)but-3-enamide (7S)-N,4-dimethyl-N-phenyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-7-pyridin-3-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carboxamide (6R,9S)-2-amino-8-oxo-7-[(Z)-3-phenylprop-2-enoyl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-9-carboxylic acid N-[2,3-difluoro-4-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)phenyl]propane-1-sulfonamide 1-[2-(4-tert-butylphenyl)sulfonylethoxy]-3,5-dimethoxybenzene 2-(2,4-dimethoxypyrimidin-5-yl)-3-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine 1-(2,4-diaminophenyl)pyrrolidine-3-carboxamide 1-amino-4-[2,5-bis(4-hydroxybutoxy)phenyl]hexan-3-ol 3-[4-(5,6-difluoro-1H-benzimidazol-2-yl)-9H-fluoren-9-yl]pyridine-4-carboxylic acid ethane;2-hydroxy-2-(1,3,4-thiadiazol-2-yl)acetamide 4-[(3,5-dichloropyridin-2-yl)methylamino]-N'-hydroxybenzenecarboximidamide 7-fluoro-N',3-dimethyl-6-methylidenebenzo[c]chromene-8-carbohydrazide (1S)-2,2-difluoro-N-[(3R)-1-methylpyrrolidin-3-yl]-5-phenylcyclohexan-1-amine N-[2-(2,4-dimethoxyphenyl)ethyl]pent-1-en-3-amine;propane 2-fluoro-4-[6-[3-(3-fluoropropoxy)cyclobutyl]pyridin-3-yl]benzonitrile ethane;6-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-yl)thieno[2,3-d]pyrimidin-4-amine 1-[(2R,3S)-3-azido-2-methylpiperidin-1-yl]-4-(3-chlorophenyl)phthalazine N-azido-2-[4-(1,3-benzodioxol-5-yl)piperazin-1-yl]ethanamine N-[4-(2,3-dihydro-1H-pyrrolo[2,3-b]pyridine-2-carbonyl)phenyl]-2,6-dimethylbenzamide N-[2-[2-fluoro-4-[5-(trifluoromethyl)pyridin-2-yl]phenyl]ethyl]formamide N-[2-(diethylamino)ethyl]-4-phenyl-1H-pyrrole-3-carboxamide 4-[(1Z)-3,5-dimethylhexa-1,3,5-trienyl]benzoic acid 5-[(2R,3S)-4-ethyl-2-(hydroxymethyl)-3-methylpiperazine-1-carbonyl]-1H-pyridin-2-one 2-[(4S)-1-(3,5-dimethylphenyl)-1-methyl-6-(3-morpholin-4-ylpropoxy)-2-oxo-3,4-dihydroquinolin-4-yl]acetic acid 2-[N-(1,3-thiazol-5-yl)anilino]decanoic acid N-[3,4-difluoro-2-(4-methylpiperazine-1-carbonyl)phenyl]benzamide [(3aS,7aR)-5-methyl-2-[(1S)-1-phenylethyl]-3,3a,4,6,7,7a-hexahydro-1H-pyrrolo[3,4-c]pyridin-5-yl]-pyrrolidin-1-ylmethanone N-[5-methyl-2-(1H-pyrrole-3-carbonylamino)phenyl]-3-(trifluoromethyl)thiophene-2-carboxamide 3-[2-(2,4-dichlorophenyl)propyl]-5-pyrimidin-2-ylpyrazin-2-amine (1R,2S)-N,1-diphenyl-2-piperidin-3-yloxyethanamine;dihydrochloride 1-[2-(1H-imidazol-5-yl)ethenyl]-3,4-dihydroquinolin-2-one 6-chloro-3-(2-chloro-5-methylphenyl)sulfanylquinoline (2E)-5,6-dichloro-N'-[(E)-3-[(Z)-hydroxyiminomethyl]pent-3-enyl]-2-[4-iodo-2-(trifluoromethoxy)anilino]-7-(trifluoromethoxy)-1H-indole-3-carboximidamide 6-ethyl-2-(4-iodophenyl)-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one 2-(N-ethylsulfonyl-4-nitroanilino)benzenesulfonic acid N-[2-[4-(5-methylthiophen-3-yl)phenyl]propan-2-yl]acetamide [1-(3,4-dimethylbenzoyl)piperidin-2-yl]-(1H-imidazo[4,5-b]pyridin-7-yl)methanone 3-[(2-chlorophenyl)methyl]-4-ethoxybenzamide 3-amino-4-chloro-N-[(E)-1-ethylsulfanylbut-2-en-2-yl]benzamide 1-N',1-N'-dimethyl-6,7-dioxo-3,4-dihydro-2H-pyrrolo[3,4-b]indole-1,4-dicarboxamide;N'-ethylethane-1,2-diamine (2S,3R)-N-hydroxy-1-[(E)-7-phenylhept-5-enoyl]piperidine-2-carboxamide N-[4-(3,5-dimethylphenoxy)-2-hydroxybutyl]-4,6-bis[[4-fluoro-2-(trifluoromethyl)phenyl]methoxy]cyclohexa-1,3-diene-1-carboxamide 2-[(1S)-1-azidoethyl]-5-fluoro-1,3-dimethoxybenzene 2-(aminomethyl)-1-[[6-[[cyclohexylidene(propanoyloxy)methyl]amino]naphthalen-2-yl]methyl]benzimidazole-5-carboxylic acid (E)-1,3-diamino-2-[5-[4-[[3-(3,4-dimethoxyphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenoxy]pyridin-3-yl]prop-2-en-1-ol 1-[3-[2-(cyclopropylsulfonylamino)pyrimidin-4-yl]-5-(trifluoromethoxy)indazol-1-yl]-N'-hydroxymethanediamine N-(4-chlorophenyl)-1,2,3-trimethoxypropan-2-amine 6-[2-(dimethylamino)ethyl]-3,5-bis(4-methoxyphenyl)cyclohexa-1,5-diene-1,2,4-triamine 4-[(4-fluorophenyl)methyl]-1,3-thiazole;3-(2-oxopropoxy)cyclobutane-1-carboxylic acid 4-[3-amino-2,5-dioxo-6-(trifluoromethyl)imidazolidin-1-yl]benzonitrile 2-[3-(diethylamino)propylsulfanyl]-4-propyl-1H-pyrimidin-6-one 1-(3,4-dihydro-2H-pyrano[2,3-b]pyridin-4-yl)-7-methoxy-5-methylbenzimidazole 2-azido-1,4-difluorobenzene;ethane 2-[4-[4-[[4-(3,4-dichlorophenyl)piperazin-1-yl]methyl]-5H-cyclopenta[d]pyrimidine-7-carbonyl]piperazin-1-yl]acetamide N-[(3R,4S)-1-cyclopentyl-4-[2-(methoxymethyl)-1H-imidazol-5-yl]pyrrolidin-3-yl]oxane-4-carboxamide;dihydrochloride N-(3-cyclopropylphenyl)quinoline-6-carboxamide (5R)-N-(2,4-dimethylphenyl)-2-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-ylidene]-4-oxo-1,3-thiazinane-6-carboxamide 1-[2-[4,5-diamino-3,6-bis(ethoxymethyl)pyridin-2-yl]phenyl]-4-methyl-1-phenoxypentan-3-one 1-[2,5-dichloro-3-(methoxycarbonylamino)phenyl]-3-[1-oxo-4-phenyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethylidene]cyclohexanecarboximidoyl]urea N-[(1R,2S)-2-methylcyclohexyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 2-[4-[2-[[2-(4-methylphenyl)sulfanylacetyl]amino]ethoxy]phenyl]acetamide 2-(3,6-dimethoxycarbazol-9-yl)acetaldehyde;N-[6-[(4-ethoxypiperidin-1-yl)amino]hexyl]formamide N-[3-(trifluoromethyl)cyclohepta-1,4,6-trien-1-yl]quinazolin-4-amine (3S)-4,5-dihydroxy-1,2,6,8-tetramethoxy-3H-xanthene-9,10-dione 4-[(E)-3,7-diethyloct-5-enoxy]benzenesulfonate 4-[4-(difluoromethoxy)phenyl]-2,3,5-trimethylaniline 5-[2-(1H-benzimidazol-2-yl)acetyl]-N,N-dimethyl-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrole-2-carboxamide (1R,2S)-N-[8-amino-6-[4-(trifluoromethyl)pyridin-3-yl]isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 2-[3-fluoro-4-(5,7,8,12-tetrazatricyclo[7.4.0.02,6]trideca-1,3,5,7,9,11-hexaen-13-yloxy)phenoxy]propanoic acid (2R,6S)-2-(1H-indazol-5-yl)-4-[(2-methoxypyridin-3-yl)methyl]-6-phenylmorpholine 2-[(5S)-6,7-dimethoxy-4-oxooctanoyl]oxybenzoic acid 4-[2-(4-chlorophenyl)-3-hydroxypropyl]piperidine-1-carbonitrile 6-(7H-purin-2-yloxy)naphthalene-1,4-diamine 1-[4-(2-hydroxy-5-methylphenyl)piperazin-1-yl]ethanone 6-(2,4-dioxo-1H-pyrimidin-5-yl)isoquinoline-4-carboxylic acid 2-fluoro-4-[[6-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)hexanoylamino]methyl]benzoic acid 2-(4-butoxycarbonyl-N-ethenylsulfonylanilino)acetic acid 4-[(2,3-dihydro-1H-inden-5-ylamino)methyl]phenol 2-hydroxy-6-[4-(N-methylanilino)phenyl]cyclohepta-2,5-dien-1-one 4-(2,6-dimethoxyphenyl)-5-ethyl-2-[3-fluoro-4-(3-pyridin-4-ylpropylamino)phenyl]-1H-pyrazole-3-thione 5-chloro-2-[[4-(cyclopropanecarbonyl)piperazine-1-carbothioyl]amino]benzoic acid N-[4-[1,2,5,7-tetradeuterio-6-(difluoromethyl)-4H-indole-3-carbonyl]phenyl]ethenesulfonamide N-(4-methoxynaphthalen-1-yl)-2-methylidene-3,4-dihydronaphthalen-1-imine 4-methyl-5-(6-phenyl-3,4-dihydro-1H-pyrido[2,3-b]pyrazin-2-ylidene)pyrazol-1-amine 3-[3-(hydroxymethyl)phenyl]-1,4-dihydro-1,2,4-triazol-5-one 1-[(1,3-dioxoisoindol-2-yl)methoxy]-2H-anthracene-9,10-dione 4-[1-(2,3-dihydro-1H-inden-5-yl)imidazol-2-yl]phenol 4-(4,5-difluoro-2-methoxyphenyl)-1H-tetrazol-5-one (5S)-3,3,4,4,7,8-hexamethyl-2-phenyl-2,9-diazaspiro[4.5]decan-1-one 5-chloro-N'-[(E)-2,3-dimethylbutanoyl]pyridine-2-carbohydrazide 2-(4,5-dihydro-1H-imidazol-2-ylmethyl)-3-ethynyl-6-hydroxybenzoic acid (7S)-1',6-dimethylspiro[5H-pyrrolo[3,4-d]pyrimidine-7,3'-piperidine]-2-one 4-methoxy-2-[4-(methyliminomethyl)anilino]benzoate (5Z)-5-[[2,4-bis[[3-(difluoromethyl)phenoxy]methyl]phenyl]methylidene]imidazolidine-2,4-dione N-[4-(aminomethyl)phenyl]-N,7-dimethylthieno[3,2-d]pyrimidin-2-amine 4-[2,4,6-trimethyl-N-(3-nitrophenyl)anilino]benzenesulfonamide 1-cyclopropyl-2,3,4-trifluoro-5-(4-methoxyphenyl)benzene [1-[3-(4-methylpiperazin-1-yl)propoxy]naphthalen-2-yl]-phenyldiazene 4-N-[2-methyl-6-(1-oxophthalazin-2-yl)propyl]quinoline-3,4-dicarboxamide 6-methyl-5-[4-methyl-3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine (Z)-3-amino-2-[(2,4-dichlorophenoxy)methyl]but-2-enenitrile 4-(aziridine-2-carbonyl)-N-[3-(2,5-dimethylphenyl)propyl]piperazine-1-carboxamide 3-[4-(dimethylamino)phenyl]-4-methylcyclobut-3-ene-1,2-dione 5-[(5-bromopyrimidin-2-yl)amino]pyrazine-2-carboxamide 4-(2,2,6,6-tetramethylpiperidin-1-yl)sulfonylphenol N-(3,4-difluorophenyl)-6-methoxycarbonyl-3-methyl-2,4-dihydrothieno[3,4-b][1,5]benzodiazepine-5-carboxylate 4-[2-(furan-3-yl)ethynyl]-N',1-dimethylpyrazole-3-carbohydrazide 2-amino-4-[3,5-bis(trifluoromethyl)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile N-[4-(2,5-dioxopyrrolidin-1-yl)phenyl]acetamide 2-amino-7-(5-azidooxypentyl)-1H-purin-6-one 4-N-cyclohexyl-2-[methoxy(propanoyl)amino]-5,6,7,8-tetrahydrothieno[3,2-c]azepine-10-carboxamide (6S)-4,5,5a,6,7-hexahydro-3H-pyrrolo[1,2-c][1,3]oxazol-2-yl]-methanamine;dihydrochloride 2-fluoro-1,4-dimethoxybenzene;N-[(2S)-3-methylbutan-2-yl]-6-(oxan-4-yl)-1-benzofuran-3-carboxamide 3-[(6E)-6-ethylidene-1H-pyridine-2-carbonyl]benzonitrile [4-(2,6-difluoro-3,5-dimethoxyphenyl)phenyl]urea 3-(4-methylcyclohexyl)-6-[1-(4-methylsulfonylphenyl)ethyl]-1H-pyridin-2-one 1,3-bis(4-methylphenyl)sulfonylpropan-2-one N-[2,6-difluoro-4-(2-iodobutanoyl)phenyl]pyridine-3-carboxamide (3,5-difluorophenyl)-[4-[2-(6-methylpyrazin-2-yl)ethynyl]piperidin-1-yl]methanone N-(2,6-difluorophenyl)-4-[2-[(3,5-dimethoxyphenyl)carbamoylamino]cyclobuten-1-yl]benzamide 1-[(2R)-4,6-dimethyl-3,4a,5,7,8,9b-hexahydro-2H-pyrano[3,2-b]pyridin-2-yl]-3-(2-phenylethylamino)propan-1-one 2-methyl-6-[(4-morpholin-4-ylpiperidin-1-yl)methyl]-N-[3-(trifluoromethyl)phenyl]pyrimidin-4-amine 6-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]-1,3,9-triazaspiro[4.5]decane 4-(5,6-diaminohexylsulfanyl)aniline 2-[4-(benzenesulfonamido)piperidine-1-carbonyl]-6,7-dimethoxy-3H-1-benzofuran-2-carboxamide N-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-3-fluorophenyl]-1H-indole-2-carboxamide 1-[2,6-bis(3-methylimidazol-4-yl)phenyl]benzimidazole 5-[3-(4,6-diphenyl-1,4-dihydro-1,3,5-triazin-2-yl)naphthalen-1-yl]pyridine-3-carbonitrile 2-chloro-5-[2,4-difluoro-3-(2,2,2-trifluoroethylsulfanylmethoxy)phenyl]pyridine 5-(4,6-diphenyl-1,3,5-triazin-2-yl)-15-(8-ethenoxy-7H-naphthalen-1-ylidene)-9,14,18-triazaheptacyclo[12.10.1.02,11.03,8.019,27.017,22.026,28]heptacosa-1(29),2(11),3(8),4,6,9,12,17,19(28),21,23(29),24,26,28-dodecaene 3-[4-(5,6-dihydro-1,2,4-oxadiazol-3-yl)-3H-pyrrole-5-carbonyl]benzoic acid 1-(2-ethylphenyl)-5,7-dimethoxy-3,4-dihydronaphthalene-2,8-diol 1-[4-(difluoromethoxy)phenyl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine 5-[2,6-difluoro-3-(trifluoromethoxy)phenyl]imidazolidine-2,4-dione 2-(1-benzylpiperidin-4-ylidene)ethanimidamide 1-[3,5-dimethyl-4-(2,2,2-trifluoroethoxy)phenyl]-N,4-diethyl-6-hydroxy-2-oxopyridine-3-carboxamide (5E)-2-cyclopentylimino-5-[(1,3-diethoxynaphthalen-2-yl)methylidene]-1,3-thiazolidin-4-one 2-(4-fluorophenyl)-3-[1-methyl-5-(trifluoromethoxy)indol-2-yl]quinoxaline 2-tert-butyl-4-methoxy-6-[(3-phenylpyrazol-1-yl)iminomethyl]phenol [2-(4-hydroxyphenyl)cyclopentyl]carbamic acid 1-(2-nitroethenyl)-4-(5,6,7,8-tetrahydronaphthalen-1-yloxy)benzene 2-(5-bromo-3,4-diethoxyphenyl)prop-2-enamide 2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-N-[2-hydroxy-5-methyl-1-(3-phenylpropanoylamino)hexan-3-yl]acetamide 2-cyclopentyloxyimino-2-[2,6-difluoro-3-(4H-pyridin-1-ylmethyl)phenyl]acetic acid [4-(5-bromopyrrolo[2,1-f][1,2,4]triazin-4-yl)phenyl]carbamic acid 4-[2-amino-1-[6-(3-bromopyridin-2-yl)oxy-7-fluoro-4-methoxyisoquinolin-5-yl]ethyl]phenol 2-cyclohexyloxy-1,4-dimethylbenzene;propane (2R)-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxamide 1-methyl-6-(3,4,5-trifluorophenyl)-1,2,3,4-tetrahydroisoquinoline N-(6-anilinopyridin-2-yl)sulfanylcyclohexa-1,3-dien-5-yn-1-amine 1-[4,7-bis(1H-indol-3-yl)octa-2,6-dienoxy]propan-2-one 3-[2-(ethylamino)pyrimidin-4-yl]benzoic acid (5Z)-2-[3-chloro-4-[(3,5-difluorophenyl)methoxy]phenyl]imino-5-[[1,5-dimethyl-3-(trifluoromethyl)pyrazol-4-yl]methylidene]-1,3-thiazolidin-4-one 5-chloro-N,2,3,4-tetradeuterio-6-fluoro-N-methylbenzamide [1-[4-chloro-2-(4-methylphenyl)quinoline-3-carbonyl]piperidin-3-ylidene]-(5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)methanol (2-methoxyphenyl)-[3-methyl-5-[(6S,9R)-3-oxa-7,11-diazaspiro[5.6]dodecan-9-yl]pyridin-4-yl]methanone;2,2,2-trifluoroacetic acid 7-fluoro-8-phenylpyrido[3,4-b]pyrazine 3-(dimethylamino)-4,5,6,7-tetrafluoro-2-propylindole-1,6-disulfonic acid 2-(N-ethylsulfonyl-2-methoxyanilino)octanoic acid 4-methyl-2,7-bis(trifluoromethyl)quinazoline N-[3-[7-(4-methylpiperazine-1-carbonyl)-2,3-dihydropyrido[3,4-b][1,4]oxazin-4-yl]phenyl]acetamide 5-[[4-chloro-2-(1H-indol-3-yl)phenyl]methylamino]-6,7,8,9-tetrahydropyrimido[4,5-b]azepine-6,7-diol N-[2-oxo-2-(5-phenyl-1,3-dihydroisoindol-2-yl)ethyl]propanamide 6-[3,4-bis(phenylmethoxy)phenyl]pyridine-2,3-diamine 4-bromo-5,6-bis(ethenyl)-2-hydroxynaphthalene-1-carboxylic acid N-(1,3-benzothiazol-2-yl)prop-2-enamide 1-[4,5-bis(3-chlorophenyl)-2-(2,4-dimethoxyphenyl)-6-[2-(methylamino)pyrimidin-4-yl]pyridazin-3-yl]cyclopropan-1-amine;ethane 1-(3,4-dihydro-2H-chromen-6-yl)-4-[6-[4-(morpholine-4-carbonyl)phenoxy]pyridin-3-yl]butan-1-one 3-[[4-amino-2-(ethoxymethyl)phenoxy]methyl]benzonitrile N-[4-(3-methoxypropyl)phenyl]-5,6,7,8-tetrahydroquinazoline-2-carboxamide 2-[4-[6-(trifluoromethyl)pyridine-3-carbonyl]piperazin-1-yl]pyridine-3-carboxamide 4-methyl-2,6-bis(4-phenylphenyl)cyclohexa-1,5-dien-1-ol 4-[(2S,4R)-4-amino-1-[1-methyl-5-(pyrrolidine-1-carbonyl)pyrazole-3-carbonyl]pyrrolidin-2-yl]benzonitrile N-[(1R)-3-[3,5-bis(trifluoromethyl)phenoxy]cyclohexa-2,4-dien-1-yl]acetamide 2-(1,4-diazepane-1-carbonyl)-N-[5-methyl-6-(2-methylsulfonylphenyl)pyridin-3-yl]-1H-indole-6-carboxamide 5-N,8-N,1,3-tetramethylimidazo[4,5-h]quinazoline-2,8a-diamine (3R)-3-ethyl-5-(5-pyridin-2-ylthiophen-2-yl)sulfonyloxolan-2-one 4-[1-ethyl-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)pyrazol-4-yl]-N-phenylaniline 3-(dimethylamino)-4-methoxy-N-[[1-[(5-oxopyrrolidin-2-yl)methyl]pyrazol-4-yl]methyl]benzamide 3-(4,7-dimethylpyrazolo[1,5-a]pyridin-2-yl)oxy-N'-hydroxypropanimidamide (2R)-N-[(1S)-3,4-dihydro-1H-isochromen-1-yl]oxolane-2-carboxamide 3-[[1-(2,4-dihydroxyphenyl)pyrazole-3-carbonyl]amino]benzenesulfonic acid 2-methylpropane;3,4,5-trifluoro-6-(2-methoxyethoxy)benzenethiol 5-azidooxy-3-ethyl-2,6-dimethyl-4-phenylpyridine N-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)benzenesulfonamide 5-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxy-N-(4-propanoylphenyl)benzamide 1-[3-(1H-pyrazol-4-yl)piperidin-1-yl]ethanone 4-(2,6-difluorophenoxy)cyclohexa-1,5-dien-1-ol 1-(1,3-benzodioxol-5-yl)-2-[4-(2,6-dichlorobenzoyl)piperazine-1-carbonyl]ethanone 3-amino-N'-[2-(4,4-difluoropiperidin-1-yl)ethyl]-6-methoxypyridazine-4-carboximidamide 3-cyclohexyloxycarbonyl-4-[4-(4-methylphenyl)sulfonylbutanoylamino]benzoic acid (1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethanethiol 4-amino-1-butanoyl-N-(2,6-difluoro-3,5-dimethoxyphenyl)cyclohexa-2,4-diene-1-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-4-chloro-3-(2-cyclopropyl-2-oxoethyl)benzamide 5-fluoro-N-[3-(furan-2-yl)oxetan-3-yl]pyrimidin-4-amine 1,3-bis(4-tert-butylphenyl)-6-hydroxy-2-(3-methoxypropoxy)-5H-pyrazolo[3,4-d]pyrimidin-4-one 6-(4-chlorophenyl)hexanal;2,5-difluorobenzenethiol 3-(1H-benzimidazol-2-yl)-7-[4-chloro-N-(cyanomethylidene)carbamimidoyl]-5-[(2S)-1-hydroxypropan-2-yl]pyrazolo[1,5-a]pyrimidine-6-carboxylic acid 4-(2,3-dihydro-1H-pyrrolo[1,2-a]benzimidazole-9-carbonyl)benzoic acid 5-methyl-4-[4-(morpholin-2-ylamino)-1,3,6,10-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),4,8,11-tetraen-12-yl]furan-2-carboxylic acid ethane;2-[(3Z)-6-methylhepta-1,3,5-trien-4-yl]benzotriazole [3-hydroxy-3-(triazol-1-ylmethyl)pyrrolidin-1-yl]-phenylmethanone 1-[3-(difluoromethyl)phenyl]-3,4-dimethoxy-9H-pyrido[3,4-b]indole 6-[4-(azidomethyl)phenyl]-2-methoxyimidazo[1,2-b]pyridazine 1-[5-bromo-4-(2,4-dimethylpentoxy)pyridin-3-yl]propan-1-amine N-[(E)-(3,4-dihydroxyphenyl)methylideneamino]-2-[[5-(1H-indol-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide (2E,3R)-2-[[7-(4-chlorophenyl)-5-methyl-4,6-dioxopyrrolo[3,4-d]pyrimidin-1-yl]imino]-N,3-dihydroxybutanamide 5-[(4,6-dimethoxypyrimidin-2-yl)carbamothioylamino]pentanoic acid 2-[3-ethylsulfonyl-6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)pyridin-2-yl]-7-(trifluoromethyl)phthalazin-1-one 1-(2,4-diaminophenyl)propan-1-one 2-methoxy-6-(2-methylpropylimino)-5,7-dihydro-4H-thieno[3,2-c]pyridine-3-carbonitrile 4-[[6-(2,3-dihydro-1H-indol-5-yloxy)pyrimidin-4-yl]amino]benzenesulfonamide N-[(2S)-3,3-dimethylbutan-2-yl]-2-[4-(8-fluoroquinolin-4-yl)cyclohexyl]propanamide 1-azidooxy-3-chloro-2-ethylsulfanylbenzene (2S)-4-chloro-3-[[6-oxo-5-(trideuteriomethyl)benzo[c][1,8]naphthyridine-10-carbonyl]amino]butanoic acid N-[2-(2-hydroxypropan-2-yl)thieno[3,2-b]pyridin-7-yl]formamide 2-(6,7-dichloro-3-methylsulfanylnaphthalen-1-yl)acetamide 3-(1,6-dimethylpyridin-1-ium-2-yl)-8H-pyrido[4,3-b]indole 4-(3,4-dimethoxyphenyl)-2-hydroxybenzoic acid 1-(4-fluorophenyl)-2-[6-methyl-5-(1,3-oxazol-5-yl)isoquinolin-8-yl]ethanone 1-butyl-5,6-diethyl-N-[(2S)-4-methoxyimino-1-[3-(trifluoromethyl)phenyl]sulfonylpyrrolidin-2-yl]benzimidazole-2-carboxamide ethane;3-methylbutanoic acid;2-(7-methyloctyl)naphthalene 2-[5-chloro-6-(1,3-dioxolan-4-yl)pyridin-2-yl]-7-(2-fluorophenyl)imidazo[1,2-a]pyrimidine 1-[(Z)-3,4-diaminobut-2-enyl]-N-[1-(3,4-difluorophenyl)cyclopropyl]triazole-4-carboxamide 6-[5-[1-(dimethylamino)propan-2-yloxy]pyridine-3-carbonyl]-4,5-dihydrothieno[3,2-d][1]benzazepine-2-carboxylic acid 1-[(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)methyl]-4-phenylpiperidine-4-carboxamide 3-benzyl-4,5-dipropoxybenzenesulfonic acid 4-fluoro-N-[2-methyl-5-(6-morpholin-4-ylpyridazin-3-yl)pyridin-3-yl]benzamide N-[(2S)-1-amino-3,3-dimethyl-1-oxobutan-2-yl]-6-(2,5-difluorophenyl)-4-[(2-imino-1,3-oxazolidin-5-ylidene)methyl]pyridine-2-carboxamide N-[(2,3-dibromo-5-ethoxy-4-hydroxyphenyl)methylideneamino]benzamide 2-[4-(carbamoylsulfamoyl)-N-[(3-fluorophenyl)methyl]anilino]acetic acid 3-[4-[(E)-but-2-enoxy]-2,3-difluorophenyl]cyclopropane-1,1,2,2-tetracarbonitrile 4-azido-2-[(2-chlorophenyl)methoxy]-3-nitrophenol 3-[4-(furan-2-yl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]-1H-indole 7-amino-3-[5-(4,4-dimethylpiperidin-1-yl)sulfonylpyridin-2-yl]-6-fluoro-1H-quinolin-2-one 4-[(3R)-1-acetyl-5-oxopyrrolidin-3-yl]sulfanyl-N'-(2,6-dimethylphenyl)-2,2-dimethylbutanehydrazide (2-chlorophenyl)-[3-hydroxy-3-methyl-5-(trifluoromethoxy)piperidin-1-yl]methanone N-(3,4-dimethoxyphenyl)-2-[4-ethyl-6-oxo-1-(1H-pyrrol-2-yl)pyrimidin-5-yl]acetamide 1-[3-(2-methoxyethyl)pyrazin-2-yl]pyrazole-4-carboxamide 1-ethyl-2,3,5-triphenylpyrazole-4-carboxylic acid 4-chloro-5,6-dimethylnaphthalene-1,3,8-trithiol 2-(4-chlorophenyl)-1-(2,2-diethoxyethyl)piperazine;hydrochloride 3-[(2Z,4E)-3,7-dichlorohepta-2,4,6-trienyl]sulfonylbenzonitrile;ethane N-(4,5-dihydro-1,3-oxazol-2-yl)-4-[[4-fluoro-3-(4-methoxyphenyl)sulfonylphenoxy]methyl]benzamide 3-(methoxymethyl)-8-[5-(pyrrolidin-1-ylmethyl)pyridine-2-carbonyl]-6,7,9,10-tetrahydroazepino[2,1-c][1,4]benzodiazepin-11-one 2-[2,6-difluoro-N-(1-hydroxypropan-2-yl)anilino]sulfanyloxybenzoic acid 3-amino-4,5-dihydroxynaphthalene-2-sulfonic acid 3-cyclopropyl-5-[4-(4,6-dimethoxypyrimidin-2-yl)piperazin-1-yl]-[1,2,4]triazolo[4,3-a]pyridine (4E)-4-[5,6-difluoro-1-(4-fluorophenyl)sulfanylindol-2-yl]hepta-4,6-dienamide 5-[(2E,4Z)-hexa-2,4-dien-3-yl]oxy-1-(2-phenoxyphenyl)indazole 3-(1,2,4-triazol-1-yl)benzoic acid 1,2-dimethyl-6-[3-(4-phenylphenoxy)propoxy]isoquinolin-2-ium 4-[3-(N',N'-dimethylcarbamimidoyl)phenoxy]-6-methoxyquinoline-7-carboxamide [6-(1-cyclopropylethoxy)pyridin-3-yl]methanamine;ethane (5S)-1,6,6,9,11-pentamethyltricyclo[10.4.0.02,7]hexadeca-1(16),2,4,7,9,12,14-heptaene 1-[(2S)-4,4-difluoro-1-methoxybutan-2-yl]-3,5-bis(trifluoromethyl)benzene 1-azidooxysulfanyl-3,5-bis(3-methoxyphenoxy)benzene N-[2,4-dichloro-3-[(4-methylcyclohexyl)sulfamoyl]phenyl]acetamide 4-[[4-chloro-5-(2,3-dihydro-1H-inden-5-yloxy)pyridin-3-yl]carbamoylamino]-N-piperidin-3-ylbenzamide 1-[3-(cyclopropylmethoxy)-4-ethoxyphenyl]-2,5-dihydropyrido[4,3-b]indole 3-(5-azido-2,4-dimethylphenyl)piperidine 2-methyl-6-[4-(1,3-oxazol-5-ylmethyl)piperazin-1-yl]pyrimidine-4-carboxylic acid 5-amino-4-[3-methoxy-2-(naphthalen-1-yloxymethyl)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 2-[(3R,4S)-1-acetyl-5-oxo-4-propan-2-ylpyrrolidin-3-yl]benzonitrile 2-[(E)-3-oxo-3-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]prop-1-enyl]benzonitrile (2S)-3,4,6-trimethyl-1H-1,2,3,4-tetrahydroquinoline-2-carboxylic acid 6,9-dimethyl-7-[[4-(trifluoromethoxy)phenyl]carbamoylamino]benzo[g]quinoline-8-carboxamide 2-(dimethylamino)benzene-1,3-disulfonate 3-[6-[(2-methoxyphenyl)carbamoylamino]pyridin-4-yl]benzamide N-[4-(3,6-dihydro-2H-pyran-4-yl)phenyl]formamide;(2R,3S)-1-methoxy-5-[methyl-[2-[3-methylbutan-2-ylidene(prop-2-enoyl)amino]ethyl]amino]-3-phenylpentane-2-sulfonate 1-[(3,4-dimethoxyphenyl)methylamino]-3-propan-2-ylthiourea 1-ethyl-5-[2-ethoxy-4-(trifluoromethyl)phenyl]sulfanylpyridin-1-ium 6-[2-(3,4-difluorophenyl)ethyl]-1-fluoro-2-(trifluoromethoxy)naphthalene (4R)-1-(3,5-dimethylphenyl)-4-(2-ethoxybenzoyl)-3-methyl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 1-(5-cyclopropyl-1H-pyrazole-4-carbonyl)-N,N'-dimethylpyrrolidine-2-carbohydrazide 2-[(3S)-2,6-dioxopiperidin-3-yl]-5-methoxyisoindole-1,3-dione [(2S,4R)-1-benzyl-4-(3,5-dichlorophenyl)pyrrolidine-2-carbonyl]oxidanium 1-(2-azidophenoxy)-3-chloro-2,5-dimethylbenzene 1-[2-[5-bromo-4-(2,3-dichlorocyclopropyl)sulfonylthiophen-2-yl]ethynyl]pyrazole (1R)-2,2,2-trifluoro-N-[5-fluoro-4-methyl-3-(1H-pyrrolo[2,3-b]pyridine-6-carbonylamino)phenyl]-1-(3,4,5-trimethoxyphenyl)ethanesulfonamide 4-[2-[3,5-diethoxy-4-(methylamino)phenyl]ethenyl]-N,N-dipropylaniline 4-methoxy-2,5-diphenyl-1H-pyrazol-3-one N-[2-(ethylamino)pyridin-4-yl]-1,3-thiazole-5-carboxamide 2-(2-chloropyridin-4-yl)-N-[5-cyclopentyl-1-(2,6-dimethoxyphenyl)pyrazol-3-yl]acetamide 1-(3,5-diethylpyrazole-1-carbonyl)-2-methoxypyridin-4-one (E)-1,2-dichlorobut-2-en-1-one;8-ethylsulfonylquinoline (Z,2E)-N'-[4-amino-3-[2-methoxyethyl(oxan-4-yl)amino]phenyl]-2-hydrazinylidenepent-3-enimidamide 2-[3-(4-propan-2-ylphenyl)cyclohexyl]oxypyridine 1-N,4-dimethyl-3-(2-methylsulfonylphenyl)benzene-1,2-disulfonamide N-[3,5-difluoro-4-(2H-tetrazol-5-yl)phenyl]-2-methoxy-6-methylpyridine-3-carboxamide 1-(1H-indazol-4-yl)-6-(5-methyl-2-pyrrolidin-1-ylphenyl)-4,7-dihydropyrazolo[3,4-b]pyridine 2-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]cyclohexane-1,3-dione 7-benzylsulfanyl-N'-methyl-4,5,6,7,8,9-hexahydrothieno[2,3-b]azepine-2-carboximidamide 3-(5-acetylfuran-2-yl)-4-hydroxy-7,8-dihydrochromene-2-thione N-[5-(1H-imidazol-2-yl)-4,6-dimethylpyridin-3-yl]thiohydroxylamine 6-fluoro-4-morpholin-4-ylquinolin-3-amine [(2R,3S)-3-amino-1-oxobutan-2-yl]oxymethylideneazanium;dimethylphosphane 3-[1-(5,6-dimethylpyrazine-2-carbonyl)pyrrolidin-2-yl]-1H-benzimidazol-2-one 3-(2,3-dihydronaphthalene-2-carbonyl)-4H-pyrazolo[1,5-a]quinazolin-5-one 2-chloro-3-ethylaniline;5-methoxy-1,3-diphenylpyrazole 2-[1-(3-chloro-4-nitrophenyl)piperidin-4-yl]oxypyrimidine 3-(3,4-difluorophenyl)-2H-furo[2,3-d]pyrimidine 1-[2,4-dichloro-3-(6H-pyrimido[5,4-b]indol-9-yl)phenyl]ethanone 1-[3-(5-oxo-2-phenyl-4H-1,2,4-triazol-3-yl)propanoyl]pyrrolidine-2-carboxamide 2-ethyl-N,3-dimethylbenzimidazole-5-carboxamide N-ethylsulfonyl-2-(4-methoxyphenyl)acetamide (Z)-N-[3,5-dichloro-4-fluoro-2-(methylideneamino)phenyl]-1-phenylprop-1-en-1-amine;ethane 2-[1-(6-methoxyquinolin-4-yl)piperidin-3-yl]-N,N-dimethylacetamide 1-(4-azido-3,6-dimethoxy-2-phenylphenyl)ethanone 6-[4-amino-2-(4,5-dimethoxy-3-methylcyclohexa-1,5-dien-1-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]naphthalen-2-ol;ethane (2S)-3-hydroxy-N,2-dimethyl-4-oxo-5-phenylmethoxy-2-propanoylpentanamide 2-(3-azidophenyl)-3,4,5-trimethoxyphenol 2-[(5-ethoxypyrazin-2-yl)methylamino]pyridine-3-carbonitrile 4-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methylthieno[3,2-d]pyrimidine-2,4-diamine 1-(4-chlorophenyl)sulfonyl-3-[2-methyl-5-[2,3,7-trifluoro-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indol-1-yl]phenyl]urea 7-[(3R)-3,4-dimethylpiperazin-1-ium-1-ylidene]-1,2,8-trihydroxyxanthen-9-one 4-[6-(cyclobutylcarbamoyl)-1-phenylpyrazolo[3,4-b]pyridine-4-carbonyl]piperazine-1-carboxylic acid 5-(1,4-dioxaspiro[4.5]decan-8-yl)-3-methyl-1,2,4-thiadiazole 6-(2,5-difluorophenoxy)-N'-hydroxypyridine-4-carboximidamide 2-[(Z)-1H-indol-3-ylmethylideneamino]oxyacetic acid 6-[2,5-dimethyl-3-(2-propan-2-ylphenyl)hexa-1,4-dien-2-yl]naphthalene 4-(2-phenylethyl)piperidine-1,5-dicarboxylic acid 4-(6,8-difluoroquinoline-3-carbonyl)piperazine-1-carboxylate 1-[(2S,4R)-4-fluoro-6-(4-hydroxyphenyl)-5-methyl-2-propan-2-yl-3,4-dihydropyran-2-yl]pentan-1-one N-(5-fluoro-3-hydroxycyclohexa-2,4-dien-1-yl)-2-methoxybenzenesulfonamide 1-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethanone;ethane 2-amino-4-(3,4-difluorophenyl)-6-methylbenzene-1,3-disulfonic acid 4-[[3-(4-fluorophenoxy)-5-methoxy-N-propylanilino]methyl]phenol 1-[2,6-dimethyl-3-(1,2,4-triazol-1-yl)cyclohexa-1,5-dien-1-yl]butan-1-one 5-(4-methoxyphenyl)-6,7-dihydro-2H-imidazo[1,2-a]pyrimidine 2-[(4E)-3,5-dimethylhepta-1,4,6-trien-2-yl]-7-[2-(1H-imidazol-2-yl)ethyl]furo[3,2-g]chromene-5,8-dione 5-chloro-N-[1,3-dimethyl-2-oxo-5-(trifluoromethoxy)benzimidazol-6-yl]-3H-2-benzofuran-1-carboxamide 2-[4-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)piperazin-1-yl]-N,N-dimethylacetamide 2-[5,6-dimethoxy-1-(3-phenoxypropyl)benzimidazol-2-yl]ethanol N-(6-chloro-3,4-dihydronaphthalen-2-yl)benzenesulfonamide [1-(5-benzyl-4-phenyl-3,6-dihydro-2H-pyridine-1-carbonyl)piperidin-2-yl]carbamic acid 4-[1-(8-chloro-5-methylpyrazolo[1,5-a]quinazoline-2-carbonyl)piperidin-3-yl]benzonitrile 2-(diethylamino)-N-[4-[1-[1-[[4-[(4-fluorophenyl)methyl]piperazin-1-yl]amino]ethenylamino]ethenoxyiminomethyl]phenyl]acetamide 4-[4-aminobutyl(ethylamino)phosphoryl]-2-methoxyphenol N-azido-2,4-dichloro-6-methylsulfanylpyrimidine-5-carboxamide 4-[(3,4-dichlorophenyl)methyl]-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide N-[5,7-difluoro-1-[(4R)-2-methyloxepane-4-carbonyl]benzimidazol-2-yl]-2-methylpyridine-3-carboxamide 1-[5-(6,7,8,9-tetrahydro-5H-pyrazino[2,3-d]azepine-4-carbonyl)pyridin-2-yl]piperidin-4-one 7-chloro-2-[(3,5-dimethylphenyl)methylidene]-1,4-benzothiazepine;hydrochloride 1-azidosulfanyl-2,3,4,5,6-pentachlorobenzene (5Z)-5-[[1,2,4]triazolo[3,4-a]phthalazin-6-yl(1H-pyrazol-4-yl)methylidene]imidazolidine-2,4-dione 3-ethoxycarbonyl-6,7-dimethyl-2H-furo[2,3-g]indole-5-carboxylic acid 5-amino-3-[4-(N-phenylanilino)phenyl]dithiolene-2,4-dione [4-(azetidine-1-carbonyl)phenyl]-(3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazol-2-ylmethylidene)azanium (5Z)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-2-(2-oxochromen-6-yl)imino-1,3-thiazolidin-4-one 4-[(3R)-3-azidopyrrolidin-1-yl]sulfonyl-N,N-dimethylaniline 2-[(7R)-7-(4,5-dimethoxycyclohexa-1,3-dien-1-yl)-2-oxo-6-phenyl-1,3-oxazepan-3-ylidene]acetic acid 2,4-dichloropyrido[3,2-d]pyrimidine N-[(2S)-1-azido-3,3-dimethylbutan-2-yl]benzenesulfonamide 1-methyl-N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-yl)phenyl]-1,2,4-triazole-4-carboxamide ethane;N-[(1E,3Z)-2-fluorohexa-1,3,5-trienyl]-4-[(E)-prop-1-enyl]naphthalen-1-amine 1-[2,3-bis(ethenyl)-7-methoxynaphthalen-1-yl]octan-1-one 5-fluoro-N'-hydroxy-3-(3,4,5-trimethoxyanilino)pyrazine-2-carboximidamide 5-(2,3,4-trimethoxyphenyl)pyrimidine 4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)morpholine-4-carbonyl]-6-ethoxypyridine-2-carbonitrile (Z)-N-[5-tert-butyl-3-(2,4-difluorophenyl)sulfonylpyrazol-1-yl]-3-cyclopropyl-2-methanimidoyl-4-[4-methoxy-6-(triazol-2-yl)pyridin-2-yl]but-2-enamide 5-fluoro-3-[[4-(6-isocyanopyridine-2-carbonyl)piperazin-1-yl]methyl]-N,N-dipropylbenzamide 4-[2-(hydroxymethyl)pentoxy]benzenecarboximidamide 3-[6,7-dimethoxy-2-(2-methylpropyl)-9H-pyrimido[4,5-b]indol-4-yl]benzoic acid [4-(2,3-dimethylbenzimidazol-5-yl)sulfonylpiperazin-1-yl]-[2-hydroxy-4-(2H-tetrazol-5-yl)phenyl]methanone 3-[4-(cyclopentylsulfanylamino)phenyl]propanenitrile 2-[4-hydroxybutyl(methoxycarbonyl)amino]benzoic acid 4-[(4,5-dimethyl-1,3-oxazol-2-yl)methoxy]-N'-(pyridine-4-carboximidoyl)piperidine-1-carboximidamide 4-(8-bromo-7,9,9-trimethylfluoren-2-yl)cyclohexa-1,3-diene 6-[7-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]spiro[2.5]octane-2-carboxylic acid 2-[3,5-dichloro-4-[3-cyano-6-(1-cyclobutylpyrazol-4-yl)pyrazolo[1,5-a]pyridine-4-carbonyl]phenyl]sulfonylethanesulfonate 4-N-(2,3-difluorophenyl)sulfanyl-5-methoxypyrimidine-2,4-diamine 4-[(2,5-dimethylpyrazol-3-yl)amino]-6,7-dimethoxyquinoline-3-carbonitrile 1,2-dimethyl-3-[(E)-4-phenylbut-3-en-2-yl]benzene;ethane 4-(4-fluorophenyl)-3,7-dimethyl-5,8-dihydropyridazino[4,5-b]quinoxaline N-[2-(4-chlorophenyl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-N',N'-diethylpropane-1,3-diamine N-(3-acetamidophenyl)sulfonylbenzamide N-[2,4-dimethyl-5-(3,4,5-trimethoxyphenyl)pyrazol-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 1-(4-fluorophenyl)sulfonylpyrrolidine;2,3,6-trichloropyridine 2,6-difluoro-N-[1-(6-methoxypyridin-3-yl)ethyl]benzamide (3-propylthiophene-2-carbonyl)oxyboronic acid N-[4-(4,6-dimethylpyrimidin-2-yl)sulfanylphenyl]-3-ethoxy-2H-pyran-6-carboxamide 4-[1-(2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-2-methoxy-1H-pyrimidin-6-one N-[(2,4-dimethylphenyl)methyl]-6-methoxy-7-[3-[4-(oxan-2-ylmethylsulfonyl)piperazin-1-yl]propoxy]-1H-indole-4-carboxamide 4-[[3-(2,3-dichlorophenyl)sulfanylpyridin-2-yl]amino]piperidine-1-carboxylic acid [2-(triazolo[1,5-a]pyridin-3-yl)phenyl]methanamine N-[(2R)-3,3,3-trifluoro-1-[4-methyl-2-(2H-tetrazol-5-yl)phenyl]propan-2-yl]-7H-purin-6-amine 2-[3-(4,5-diphenyl-1,2,4-triazol-3-yl)propoxy]aniline 5-[[(2R)-2,6-dihydroxycyclohexyl]amino]-3H-2-benzofuran-1-one 1,4-difluorobenzene;N-[[2-(5-methylfuran-2-yl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-morpholin-4-ylpropanamide N-[3,5-dichloro-4-(trifluoromethyl)phenyl]-2-hydroxy-1,5-dimethyl-6-oxopyridine-3-carboxamide [7-(1H-indazole-3-carbonyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-3-yl]-pyrrolidin-1-ylmethanone 3-[4-(4,6-diphenyl-1,4-dihydropyrimidine-2-carbonyl)anilino]propylboronic acid N-(2,2,6-trimethyloxan-4-yl)-5-[1-(2,4,6-trifluorophenyl)ethyl]-1H-pyrazole-3-carboxamide 3-[6-(4,6-diaminopyridine-2-carbonyl)oxyhexyl]phthalic acid 1-[3-[(4,5-dimethylfuran-2-carbonyl)amino]propyl]triazole-4-carboxamide 4-[(3,5-dimethylphenyl)iminomethyl]-2-methoxyphenol 2-[4-(4-bromophenyl)phenyl]-N,N-di(ethyl)cyclopentan-1-amine 1-[4-(2,6-dimethylphenyl)piperazin-1-yl]-3-(5-ethoxypyridin-3-yl)propan-2-ol 2,4-di(nonyl)aniline 1-[6-(4-ethoxyphenoxy)pyrimidin-4-yl]-3-[2-methyl-1-(trifluoromethyl)cyclopropyl]urea 4-methylsulfanylthieno[3,2-d]pyrimidine 1-[4,5-dichloro-2-(3-chlorophenyl)imidazol-1-yl]propan-2-one N-(4-hydroxyphenyl)-2,3-dimethoxybenzenesulfonamide (E)-N-[4-(1,3-dihydroisoindol-2-yl)phenyl]-3-hydroxy-2-(3-methoxypyridin-1-ium-2-yl)-3-thiophen-2-ylprop-2-enethioamide 1-benzyl-3,5,6,7,8,8a-hexahydro-2H-quinoline 2-[(1Z)-buta-1,3-dienyl]-5-tert-butylpyridine;ethane N-[(3S,4R)-1-(2-amino-2-oxoethyl)-4-methoxypyrrolidin-3-yl]-5-cyanopyridine-2-carboxamide 3-[4-(2,3-dihydrofuro[2,3-c]pyridine-5-carbonyl)piperazin-1-yl]propanamide (5-chloro-1H-indol-2-yl)-(2,6-dimethoxypyridin-3-yl)methanone (Z)-N'-[[3-[4-fluoro-2-[(2S,6R)-1,2,3,5-tetramethyl-6-nitro-3a,4,6a-tetrahydrocyclopenta[b]pyrrol-6-yl]anilino]propylamino]methylidene]pent-2-enediamide 1-[4-(difluoromethoxy)phenyl]-N,2,3,6,7,8,9,10-octahydropyrimido[5,4-c]azocin-4-imine [5-amino-1,2-bis(4-methoxyphenyl)pyrrol-3-yl]methanol 1-[2-(6,7-dihydro-4H-pyrano[4,3-d][1,3]thiazol-2-yl)piperidine-1-carbonyl]pyrazole-3-carboxylic acid 4-[5-amino-2-(2,6-difluorophenyl)-1,3-thiazol-4-yl]benzoic acid 4-[5-amino-3,6-dimethyl-7-(2H-tetrazol-5-yl)pyrazolo[1,5-a]pyrimidin-2-yl]benzenesulfonamide 3-[4-(3,5-diphenyl-1,2,4-triazol-1-yl)butoxy]benzenecarboximidamide;hydrochloride 2-[[5-(2,3-dihydropyridin-4-yl)thiophen-2-yl]methyl]-1,3-thiazole N-[3-(diethylamino)propyl]-4-[6-[5-(1H-indol-3-yl)pentoxy]-1-benzofuran-2-yl]benzamide 5-methyl-4-[[2-(1H-pyrazole-4-carbonyl)phenyl]sulfamoyl]thiophene-3-carboxylic acid 3-[(2R)-2-(3,4-difluorophenyl)propyl]pyridine (3Z)-3-[(5E,7Z)-9-hydroxy-2,8-bis(hydroxymethyl)deca-3,5,7,9-tetraenylidene]-6-[4-(trifluoromethoxy)phenyl]-1H-indol-2-one 3-hydroxy-2-[4-(4-methylcyclohexanecarbonyl)piperazin-1-yl]-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one 4-hydroxy-6-[2,3,5-trimethyl-1-(1-phenylethoxy)indol-7-yl]-2H-isoquinolin-1-one 2-cyclobutyl-5-[(3R)-3-(3,4-dimethoxyphenyl)piperazine-1-carbonyl]benzaldehyde 2-amino-N-[(3R)-1-(diethylcarbamoyl)piperidin-3-yl]-5,6-dimethyl-4-(pyrrolidine-1-carbonyl)pyridine-3-carboxamide;hydrochloride (4-phenylpiperazin-1-yl)iodanuidylbenzene 4-[[(2,6-dichlorobenzoyl)amino]methyl]cyclohexane-1-carboxylic acid N-cyclohexyl-4-[[(2S)-oxolan-2-yl]methylamino]-6-pyridin-3-ylquinazoline-8-carboxamide 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidine-2-thione 2-(5-methylfuran-3-yl)-1,6-diphenylcyclohexa-2,4-dien-1-ol N-(2-aminoethyl)-4-[3-(2,6-dichlorophenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]cyclohexan-1-amine 1-(2,6-dichlorophenyl)-3-ethyl-3a,4,9b-tetrahydroindeno[5,c]pyrazole 2-[2-azidooxy-1-[2-(4-methylphenyl)ethoxy]ethoxy]acetaldehyde 2-bromo-4,5-diphenylimidazole;4,7-dimethylquinoline 5-[(2S)-1,3-dihydroxypropan-2-yl]-4-methylfuran-2-carboxylic acid 4-[2-(ethyliminomethyl)pyrrol-1-yl]benzenesulfonamide ethane;4-N-[3-(propan-2-ylamino)sulfanylphenyl]benzene-1,4-diamine 1-(4-cyclopropylpiperidine-1-carbonyl)indole-2,3-dione N-[3,5-dichloro-4-(2-methylpropoxy)phenyl]-2-(2-oxoazepan-1-yl)acetamide 4-[4-(2,6-dichloro-4-nitrophenyl)-1-(pyridine-3-carbonyl)pyrrolidin-3-yl]benzonitrile 2-azidosulfanyl-5-chloropyrimidine (5R)-3-[4-(difluoromethoxy)phenyl]-N,2-dimethyl-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carboxamide [4-(2,3-dichlorophenyl)piperazin-1-yl]-[3-ethoxy-5-methoxy-4-[2-(methylideneamino)ethenyl]thiophen-2-yl]methanone 1-[3-fluoro-2-(morpholin-4-ylmethyl)phenyl]pyrrolidine-2,5-dione 3-(5-bromocyclohepta-1,4,6-trien-1-yl)oxyaniline 2-[2,5-dimethyl-4-(3-nitrophenyl)piperazin-1-ium-1-ylidene]-1-naphthalen-1-ylethanone N-[4-[4-(aminomethyl)anilino]phenyl]acetamide N-(3,4-dihydro-2H-chromen-8-ylmethylideneamino)-6-phenylpyridazine-3-carboxamide 1-(2,4-dimethylphenyl)sulfonylsulfonylpiperidin-4-one 3-azido-5-(2,4-difluorophenyl)-1H-pyrazole 4-[3-(difluoromethyl)imidazo[1,2-b]pyridazin-6-yl]aniline 4-(3,5-dimethylpyrazol-1-yl)-2-[[4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl]methyl]-6-propan-2-ylidenecyclohexa-2,4-dien-1-one 1-(5-fluoropyridin-3-yl)-N-methylsulfonylcyclopropane-1-carboxamide 1-[(2S,5R)-4-[4-cyclobutyl-6-[[3,5-dimethyl-4-(5-methylthiophen-2-yl)phenyl]methoxy]pyrimidin-2-yl]-2,5-dimethylpiperazin-1-yl]ethanone 3-methyl-2,6-bis[(4-nitrophenyl)diazenyl]aniline (3R)-N-[2-azidooxy-4,6-bis(phenylmethoxy)phenyl]pyrrolidine-3-carboxamide N-[(2S)-1-methoxypropan-2-yl]-3,5-bis(sulfanylidene)cyclohexa-1,4-diene-1-carboxamide 3-[4-chloro-5-(2,3-dimethylanilino)pyrimidin-2-yl]sulfinamoyl-N,N-diethylpropanamide 2-[N-(4-chlorobutyl)-3-methylsulfanylanilino]acetamide N-[2-(4-ethylphenoxy)ethyl]-1-(2,3,5-trifluorophenyl)butan-1-amine 4-(2,3-dihydro-1H-inden-5-ylsulfonyl)morpholine 3-(2,5-dihydropyrrole-1-carbonyl)benzaldehyde;N-[4-[2-(dimethylamino)ethoxy]phenyl]-4,7-bis(hydroxymethyl)-N-methylcyclohepta-1,4,6-triene-1-carboxamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenoxy]-1,4-diethylcyclohexa-1,3-diene 7-(2,3-dihydrothiophen-5-yl)-3-phenylthieno[2,3-c]pyridine 5-(2,3-dihydro-1H-pyrazole-4-carbonylamino)pyridine-2-carboxamide 4-methyl-N-[3-methylidene-1-(3-nitrosocyclohexa-2,5-dien-1-yl)sulfonyl-2H-indol-6-yl]benzamide 4-[1-(6-ethoxynaphthalen-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carbonyl]piperazin-2-one (3S)-4-(cyclopropylmethoxy)-N-[[1,2-difluoro-7-(trifluoromethylsulfonylamino)naphthalen-2-yl]methyl]pyrrolidine-3-carboxamide 2-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-7-ethoxy-1,5-dihydropyrrolo[2,3-f]benzimidazole 2-[4-[(4E)-3,7-dihydro-2H-1-benzoxocin-5-yl]piperazin-1-yl]-N-methylethanamine 3,6-dimethyl-N-(2-methylpropanoyl)pyridine-2-carboxamide N-[3-[[2-(4-aminopiperidin-1-yl)anilino]methylidene]-2,5-dioxopyrrolidin-1-yl]acetamide (3S)-1'-benzylspiro[2H-indole-3,4'-piperidine] 3-chloro-2,4-dihydroxybenzoate N-[5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-7-yl(1H-pyrrol-3-ylmethyl)amino]acetamide 2-(azidomethyl)-5-(4,6-diphenylpyridin-3-yl)pyrimidine 6,7-difluoro-1-[4-(trifluoromethyl)phenyl]naphthalene 4-[6-fluoro-2-hydroxy-3-(piperidine-1,5-diylmethoxy)phenyl]benzonitrile 5-[(2E,4Z)-hepta-2,4-dien-3-yl]oxy-N'-hydroxypyrazine-2-carboximidamide (1E,3Z)-N'-[5-cyano-4-[2-methoxyethyl(propan-2-yl)amino]pyridin-2-yl]-1,3-bis(ethenyl)penta-1,3-diene-1,4-diamine [(2R,3S)-5,7-diethyl-1-methoxyimino-4-phenylnonan-2-yl]carbamic acid 1-[3-(4,6-dichlorocyclohexa-2,4-dien-1-yl)oxypropoxy]-3-ethylbenzene (7S)-N-[2-(1,3-benzodioxol-5-yloxy)ethyl]-5-methyl-7-pyridin-4-yl-6,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 2-(7,8-dihydroimidazo[1,2-a]pyridin-6-yl)phenol N-[4,5-dimethyl-2-(phenylsulfanylmethyl)furan-3-yl]benzenesulfonamide 3,5-dichloro-2-[3-methoxy-4-(2H-tetrazol-5-yl)phenyl]benzonitrile 2-(4-bromo-5-cyclopropyloxypentoxy)quinoline N-[5-[4-(2,3-dichlorophenyl)piperazine-1-carbonyl]-6-oxo-1H-pyridin-3-yl]acetamide 2-[(4S,7R)-3-methyl-5-oxo-7-thiophen-2-yl-6,7,8,9-tetrahydro-4H-pyrazolo[3,4-b]quinolin-1-yl]benzoic acid 5-[3-(1H-imidazo[4,5-b]pyridin-2-yl)phenyl]-N-pyrimidin-5-ylisoquinolin-3-amine 2-azidooxy-3-[2-(4-chlorophenyl)ethoxy]pyridine N-[5-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]pyridin-2-yl]-7-(dimethoxymethyl)-6-fluoro-1-(4-fluorophenyl)indazole-3-carboxamide 2-[3-methyl-1-(oxan-4-yl)pyrazol-4-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine 5-(8-fluoroimidazo[1,2-a]pyridine-6-carbonyl)-N-(4-hydroxyphenyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 3-[(4-fluorophenyl)methyl]-1-propan-2-ylpiperidine 2-(5-phenylmethoxypyrimidin-2-yl)oxypentanoate 2,6-dichloro-4-[(E)-2-cyclopentylethenyl]pyridine 1-benzyl-N',N'-dimethyl-5-phenylpyrazole-3-carbohydrazide N-[2-(ethylcarbamoyl)-4,6-difluorophenyl]pyridine-3-carboxamide 5-chloro-N'-[[(2,4-difluorophenyl)methyl-methylamino]methyl]-1H-indole-2-carboximidamide [3-[[5-amino-4-[(2E,4Z)-hexa-2,4-dienyl]-1H-pyrazol-3-yl]carbamoyl]phenyl]-dimethoxyphosphoryloxidanium 1-[2,4-bis(2-methylbutan-2-yl)phenyl]-N-[(Z)-3-hydroxyprop-1-enoxy]cyclopentane-1-carboxamide N-[(6-fluoro-2H-chromen-3-yl)methoxy]-1-benzofuran-6-amine 5-[(4E)-3,7-dimethylocta-2,4-dien-2-yl]-1-ethylindole 2-amino-7-[(1,5-dimethylpyrazol-4-yl)methyl]-5H-pyrrolo[3,2-d]pyrimidine-6-carbonitrile 2-N-butyl-4-(2,3-dihydroindol-1-ylsulfonyl)benzene-1,2-disulfonamide N-[(3,4-dichlorophenyl)methyl]-6-methoxyquinazolin-2-amine;propane ethane;2-methoxycarbonyl-3,5-dimethylphenolate (2E,6Z)-N,2-bis[[4-(diethylaminomethyl)phenyl]methylidene]-8-oxa-4,5-diaza-1-azanidacyclononan-3-imine;dichloroiron 2-[4-(2-phenylethylcarbamoylamino)pyrazole-1-carbonyl]pyrrolidine-1-carboxylic acid 2-(1H-imidazol-5-yl)-N-[3-methoxy-4-(trifluoromethoxy)phenyl]pyrimidine-4-carboxamide 7,8-dimethoxy-1-(2-phenylethyl)-4H-[1,2,4]triazolo[3,4-c][1,4]benzoxazin-3-one;ethane (6-chloropyridin-3-yl)-phenylcarbamic acid 2-N-[4-(4,5-dimethylimidazol-1-yl)phenyl]-7H-purine-2,6-diamine 1-amino-3,4-difluoro-5-methyl-2,6-bis[(4-methylphenyl)methoxy]benzene 1-phenylsulfanyl-3-(trichloromethylsulfonyl)benzene 1-(4,4-dimethylpent-2-en-3-yl)-N-methyl-3H-indene-2-carboxamide 5-azidooxy-4-hydroxy-2-phenylbenzoic acid 1-[4-(3-cyclopentyloxy-2,6-difluorophenyl)pyridin-2-yl]-2-methylpropan-2-ol 2-N,4-N,7-trimethylpyrazolo[1,5-a][1,3,5]triazine-2,4-diamine 4-cyclopropyl-2-(1,3,5-trimethylpyrazol-4-yl)aniline 4-[5-methyl-2,4-dioxo-6-(trifluoromethyl)thieno[3,2-d]pyrimidin-1-yl]benzoic acid (2R)-5-amino-2-[benzyl(benzyl)amino]pentanoic acid (5E)-2-cyclopentylimino-5-[[4-methoxy-3-nitro-5-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidin-4-one 5-[(4-fluorophenyl)methyl]-3,4-dihydro-2H-1,5-benzoxazepine-7-carboxylate ethane;(3Z)-pentacyclo[11.8.0.02,10.04,9.015,20]henicosa-1(21),2(10),4,6,8,11,13,15,17,19-decaene 3-[2-chloro-4-(methylamino)phenoxy]-N'-hydroxypyridine-2-carboximidamide 2-azido-3,4-dibromothiophene 4-(2,6-dichlorophenyl)-5-(4-methoxy-2-methylsulfonylphenyl)-N-[3-[1-propanoyl-6-(trifluoromethyl)piperidin-3-yl]phenyl]-1,2,4-triazole-3-carboxamide 2-cyclohexyl-6-[(4-methoxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3,7-dimethoxy-6-(3-methylbut-2-enyl)-2-phenyl-3a,4-dihydrobenzo[g]indole N-[(2S)-4,4-dimethylpentan-2-yl]sulfonylbenzamide 2-[4-chlorobutyl(3-methylbut-2-enyl)amino]phenol 2-(cyclopentylamino)oxybenzoic acid 3-(2,4-difluorophenyl)-N-ethyl-N-methylcyclobutan-1-amine (3-bromo-2,6-difluorophenyl)-triethylphosphanium 2-[4-(3,5-dimethylphenyl)sulfonylmorpholin-3-yl]ethanol N-[(5S)-3-amino-5-hydroxypentyl]-4,6-dimethoxypyrimidine-2-carboxamide 3-amino-5-(4-hexoxyphenyl)-1H-pyrazole-4-carboxamide 2-(4-hydroxy-3-propyl-5-sulfophenyl)propanoic acid 1-[3-azido-1-(4-fluorophenyl)propyl]-2,5-dimethoxybenzene 3-methylsulfanyl-6-(trifluoromethoxy)isoquinoline N-[2-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]cyclobutanamine N-benzyl-2-chloropyridine-3-carboxamide 2-[4,5-bis(4-fluorophenyl)imidazol-1-yl]ethanol 5-bromo-1,4-dihydroquinazoline 6-azido-N'-[4-(trifluoromethoxy)phenyl]hexanimidamide N-[1-(2,4-dichlorophenyl)ethyl]-5-(furan-2-yl)-3H-pyrrole-2-carboxamide;hydrochloride 4-[5-(1,3-thiazol-2-yl)pyrazin-2-yl]morpholine 2-[(3,4-difluorophenyl)methyl]isoquinolin-2-ium 1-[4-(6,7-dimethoxyquinolin-4-yl)oxy-2-fluorophenyl]-3-[5-(trifluoromethyl)pyridin-2-yl]urea 4-azidooxybenzoic acid 4-[6-(3,5-dimethyl-1H-pyrazol-4-yl)-7-oxo-8-propan-2-yloxy-1,8-naphthyridin-3-yl]cyclohexane-1-carboxylic acid 4-[(3R)-1-[(6-aminopyridin-2-yl)methyl]pyrrolidin-3-yl]oxy-N,N-dibutylbenzamide (7R)-5-methyl-6,11-dihydrobenzo[b][1]benzazepine;N'-(2-morpholin-4-ylethyl)propane-1,3-diamine 1-methyl-7-(3-propan-2-yloxyanilino)-6-prop-1-en-2-yl-3,4-dihydroquinolin-2-one 5-[4-(2,3-dihydropyridin-6-yl)phenyl]-2-ethoxypyridine 7-(3,5-dimethylphenyl)-N'-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]imidazo[1,2-a]pyridine-3-carbohydrazide N'-ethyl-4-[[(4-fluorophenyl)-(2,3,5,6-tetrafluorophenyl)methoxy]amino]piperidine-1-carboximidamide 2-chloro-3-cyclohexyloxycarbonylquinoline-4-carboxylic acid 2-[2-(1,3-benzodioxol-5-yloxy)-2-methoxyethyl]-4-bromo-1-methylimidazole 2-N,6-N,7-N-trimethyl-1H-pyrrolo[2,3-b]pyridine-2,4,6,7-tetramine 3-[1-(4-fluorophenyl)ethyl]-5-[5-fluoro-6-(2-hydroxypropan-2-yl)pyridin-3-yl]oxy-7H-pyrazolo[4,3-d]pyrimidine-6-thione 3-methylspiro[1,5,6,7-tetrahydropyrazolo[4,3-c]pyridine-4,1'-cycloheptane] 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-propylaniline 5-[4-methoxy-2-(trifluoromethyl)phenyl]-1,3-thiazole 2-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6H-cyclohepta[b]furan 2-[2-(aminomethyl)morpholin-4-yl]benzoic acid 2-[6-(9H-fluoren-1-yloxy)-5,7-dihydrofuro[3,4-d]pyrimidin-2-yl]-8-fluoroimidazo[1,2-a]pyridine 3-[2-(1,3-benzothiazol-6-yl)phenyl]-5-cyclopropyl-1,2,4-oxadiazole 4-N-[3-[[4-(furan-2-ylmethoxy)phenyl]methylideneamino]propyl]quinoline-3,4-dicarboxamide N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)spiro[3.3]heptane-2-carboxamide;hydrochloride [3-(cyclopentylmethoxy)-4-hydroxy-6-nitroindazol-1-yl]-morpholin-2-ylmethanone ethane;ethylbenzene;1-[1-(2-hydroxyethoxy)propan-2-yl]-3-phenylazetidin-3-ol N-(2,4-dichlorophenyl)sulfonyl-3-[1-hydroxy-2-oxo-2-(propan-2-ylamino)ethoxy]naphthalene-2-carboxamide N-benzyl-1',2-dimethylspiro[5,7-dihydropyrano[4,3-d]pyrimidine-8,3'-pyrrolidine]-2'-carboxamide;hydrochloride 3-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridine N-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-methoxypyrimidine-4-carboxamide 2,4-dibutyl-3-(4-phenylpiperazine-1-carbonyl)benzaldehyde 1-(2-methylpyridine-4-carbonyl)spiro[4H-quinoxaline-3,4'-piperidine]-2-one 3-cyclopropyl-2-fluoro-4-[7-methyl-6-[(1R)-2,2,2-trifluoro-1-hydroxyethoxy]pyrazolo[4,3-c]pyridin-1-yl]benzonitrile 3-methoxy-2,4,5,6,7-pentafluoro-1,9a-dihydrofluorene 2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methoxy]-N'-propan-2-ylpropanediamide [(4-methylpiperidin-1-ium-1-ylidene)amino]-[5-methylsulfonyl-6-[2,3,7-tris(sulfanylidene)-1,4-diazepin-5-ylidene]cyclohexa-1,3-dien-1-yl]azanide 4-(dihydroxymethyl)-1,7-bis[[3-(1H-pyrazol-5-yl)phenyl]sulfanylmethyl]chromen-2-one N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-2,4,6-trimethyl-N-(6-nitro-1,3-benzothiazol-2-yl)benzenesulfonamide 5-chloro-N-[(1S)-2,3-dihydro-1H-inden-1-yl]thiophene-2-carboxamide 6-[(2R,3S)-2-[(dimethylamino)methyl]-3-phenylmorpholine-4-carbonyl]pyridine-2-carboxamide 5-[(2R)-2,3-dihydroxybutyl]sulfanylpyridine-2,4-dicarboxylic acid N-[(2S)-1-amino-3,4-dioxobutan-2-yl]-5-methoxy-4-methylthiophene-2-carboxamide 2-methyl-1,4-diphenylcyclohexane-1-carbonitrile 4-ethoxy-N-(3-methylbut-2-enyl)-N-[(4-nitrophenyl)methyl]aniline 2,2-dimethyl-3-oxo-N-(4-pyrimidin-5-ylphenyl)propanamide N-[3-fluoro-5-(2-morpholin-4-ylpyrimidin-5-yl)phenyl]-1-propanoylpiperidine-3-carboxamide 1-[4-(6,7-dihydro-5H-pyrrolo[3,2-d]pyrimidin-4-yl)phenyl]-N'-methylpropane-1,3-diamine 2-(benzylideneamino)-4-phenylmethoxyphenol 6-ethenyl-N,2-dimethylnaphthalene-1-sulfinamide 1-[4-(2,6-dimethylmorpholine-4-carbonyl)-3-fluoroanilino]-N'-hydroxyimidazole-2-carboximidamide 1-(1,3-dioxol-4-yl)-6-methoxy-2H-isoquinoline N-[3-chloro-4-(2,5-dioxopyrrol-1-yl)phenyl]-2-(1-methylcyclopropyl)acetamide 4-(2,3-dihydroindol-1-yl)-N'-hydroxypyridine-2-carboximidamide (E,3R)-3-[6-[5-chloro-2-(oxan-4-ylmethoxy)pyridin-4-yl]-3-oxo-1H-isoindol-2-yl]-N'-formyl-3-phenylprop-2-enimidamide 1-[[3,5-bis(trifluoromethyl)phenyl]methylamino]-3-(cyclobutylsulfanylmethyl)thiourea 1-(4-bromophenyl)sulfonylpiperidine 2-[3-(4,5-dimethylpyridin-2-yl)oxypiperidin-1-yl]-6-fluoro-[1,3]thiazolo[4,5-b]pyridine 6-(cyclohexylamino)-1,3-dimethylpyrimidine-2,4-dione 1-(5,7,8,9-tetrahydrocarbazole-3-carbonyl)azetidine-3-carbonitrile (E)-3-(4,5-dihydro-1H-imidazol-2-ylamino)-1-phenylbut-2-en-1-one 5-chloro-N,4-dimethylfuran-2-sulfonamide 3-[[4-(1,2-dimethoxyethyl)phenyl]methoxy]-2-[(1E,5Z)-6-oxohexa-1,5-dienyl]benzoic acid 2-amino-3-[4-(trifluoromethyl)phenyl]-1H-indole-5-carbonitrile N-[2-(dimethylamino)ethyl]-4-(propanoylamino)benzamide 5-[2,5-bis(trifluoromethyl)phenyl]-4-[[4-chloro-6-[3-(diethylamino)propylcarbamoyl]quinolin-8-yl]oxymethyl]pyridine-2-carboxylic acid N-[3,5-bis(2-methoxyphenoxy)phenyl]-1,3-benzodioxole-4-sulfonamide 6-methyl-3-(1-methylpyridin-1-ium-2-yl)phenanthridine 5-[2-(4-aminooxypiperidin-1-yl)ethyl]-6,8-dibromo-3,3-dimethyl-11H-pyrano[2,3-b]acridine-2,7-dione 2-[4-(methoxymethyl)phenyl]-6,6a-dihydronaphtho[1,2-b]oxirene 2-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]phenol 1,3-diethyl-5-[(Z)-(3-methoxy-2H-isoquinolin-4-ylidene)methyl]-6-(trifluoromethyl)pyrimidine-2,4-dione 6-[2-aminoethyl(methyl)amino]-3,5,7-trihydroxychromen-4-one N-(3-ethylpyridin-4-yl)-5,6-difluoro-1H-indole-2-carboxamide N-[(2R,3S)-1-ethyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]-1H-pyrrole-3-carboxamide 3-[2-methoxyethyl(pyridin-4-yl)amino]piperidine-1-carboxylic acid 6-hydroxy-2,5,8-trimethylnaphthalene-1,4-dione N-[(4Z)-5-hydroxy-7,10-dioxo-2-(1-phenylpentylamino)undeca-4,8,10-trienyl]cycloheptanecarboxamide 2-[(2Z)-4-oxo-2-[(Z)-1-phenylpropylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 2-[3-azidooxy-1-(2,4-difluorophenyl)propyl]-N-hydroxyacetamide 2-[(3,5-difluorophenyl)carbamoylamino]-N-hydroxy-1,3-benzoxazole-6-carboxamide N-[(4-phenylcyclohexyl)methylidene]benzenesulfonamide 5-[2,6-dichloro-4-(2-methylpropanoyl)phenoxy]pentanedioic acid (5Z)-1',4'-difluorospiro[2H-indole-3,9'-xanthene]-4,8-dione 4-(N'-tert-butylcarbamimidoyl)benzoic acid 2-[(5Z)-5-[1-(benzenesulfonyl)-3-methylimidazolidin-2-ylidene]piperidin-3-yl]acetonitrile [3-(4,5-dimethylimidazol-1-yl)piperidin-1-yl]-(6-fluoroimidazo[1,2-a]pyridin-2-yl)methanone;formic acid N-(4-azidobutyl)-3-chlorobenzamide 3-chloro-5-[2-[[1-(4,4-dimethyl-2-oxopentyl)pyrazol-4-yl]amino]pyrimidin-4-yl]oxybenzenesulfinamide 3-methoxy-2-[4-(10,13,15-trichloro-3-tricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaenyl)piperazine-1-carbonyl]piperidine-1-carboxylic acid N-[1-(3-aminopropyl)-2,6-dioxopiperidin-4-ylidene]benzenesulfonamide 2-(3-chloro-4-propan-2-ylphenoxy)propanoic acid 1-[3,5-ditert-butyl-4-(methoxyamino)phenyl]propan-2-one 2-[(1,2-dimethylimidazole-4-carbonyl)amino]-5,6-dimethoxy-N-phenyl-1-benzofuran-3-carboxamide [(Z)-1-(1,5-dimethyl-6-oxopyridin-3-yl)prop-2-enylidene]azanium N-[(5S)-6-amino-5,7,8,9-tetrahydropyrimido[5,4-c]azepin-2-yl]-2-cyclobutylideneacetamide 3-[2,6-difluoro-4-(trifluoromethyl)phenyl]sulfonyloxy-1,2-thiazole-5-carboxylic acid 2-[1,3-bis(4-ethoxyphenyl)propyl]benzenesulfonate 3-[7-(6,8-dichloro-2-methyl-3,4-dihydro-1H-isoquinolin-4-yl)-3-oxoheptoxy]-5-fluoro-2-hydroxybenzoic acid 1-[4-(difluoromethyl)phenyl]pyrrolidine;N-[(6-pyrazol-1-ylpyridin-2-yl)methyl]acetamide 2-[5-carbamoyl-9-(quinolin-6-ylmethyl)carbazol-4-yl]oxyacetic acid N-(diaminomethylidene)-4,6-bis[4-ethyl-3-(2-hydroxyethoxy)phenyl]-1H-indole-2-carboxamide 5-[(4,5-dichloro-2-hydroxyphenyl)methylideneamino]pyridine-3-carboxylic acid 2-[(4-methylsulfinylphenyl)methyl]propanedinitrile 5-[(3R)-2,3-dihydroxyhexoxy]-1H-pyridin-2-one 4-azidooxy-N,6-dimethylbenzimidazole-1-carboxamide N-(4-bromophenyl)-2-[[5-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]pyridin-2-yl]methyl-methylamino]-N-ethylacetamide 3-(1H-indol-3-yl)propane-1,2-diol (4E)-2-cyclopropyl-N-[1-[3,5-dichloro-2-[(E)-3,3-dimethylbut-1-enyl]pyridin-4-yl]ethyl]-6,7-difluorohepta-2,4,6-trien-3-amine 3-(4-ethylpyridine-2-carbonyl)chromen-2-one 4-[2-(2,5-difluorophenyl)pyrrolidine-1-carbonyl]-N'-hydroxypyridine-2-carboximidamide 3-[2-(3-fluorophenyl)ethynyl]pyridine N-[5-(2-hydroxyethyl)-1,3-thiazol-2-yl]-2-(4-sulfamoylphenoxy)acetamide [(Z)-1,2-diamino-3-[5-methyl-4-(2,2,2-trifluoroethoxy)pyridin-3-yl]iminoprop-1-enyl]-[2-methoxy-6-(trifluoromethyl)pyridin-3-yl]azanium 2-[3,5-dichloro-4-(6-oxo-4-phenyl-1H-pyridazin-3-yl)phenoxy]acetic acid 1-(cyclohexen-1-yl)-5-(4-fluoro-2,3,6-trimethoxyphenyl)pentan-1-one 2-chloro-6-[2-(methylamino)pyridin-4-yl]oxybenzaldehyde 3-ethyl-6-[5-(4-morpholin-4-ylphenyl)-1,2,4-oxadiazol-3-yl]-3H-[1,2]oxazolo[4,5-c]pyridin-7-ium N-[5-(diethylaminomethyl)pyrazin-2-yl]-4-fluoro-3-hydroxysulfanylbenzamide N-[(3S,4R)-1-tert-butyl-3-[4-oxo-6-(trifluoromethyl)-5H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-4-yl]-2-(dimethylamino)acetamide (E)-4,8-dihydroxy-2,2,6,8-tetramethylnon-3-enoic acid;5-[2-[5-(3-ethoxyphenyl)thiophen-2-yl]ethynyl]pyridine-3-carboxylic acid 6-[1-(5,6,7,8-tetrahydroquinolin-2-yl)imidazol-4-yl]thieno[3,2-c]pyridine 3-benzyl-2,4-dimethyl-1,3-benzothiazole 4-(4-methoxyanilino)-1,3-dimethyl-6-oxopyridine-2-carboxamide (5R,7S)-2,3-dimethyl-4,5-diphenyl-1,4,6,7,8,9-hexahydropyrazolo[5,1-b]quinazoline 3-chloro-5-[7-(4,6-diphenylpyrimidin-2-yl)naphthalen-1-yl]benzonitrile 1-ethyl-4-[(2E,4Z)-3-methylhepta-2,4,6-trienoxy]benzene 5-[4-(3,5-dichloropyridin-4-yl)phenyl]sulfanyl-2H-triazole-4-carboxylic acid 1-(2,2,2-trifluoroethyl)-7H-pyrazolo[3,4-f]quinazoline (2R)-N-[4-fluoro-3-[7-methyl-5-oxo-8-(pyridin-2-ylmethoxy)imidazo[1,5-a]quinazolin-6-yl]phenyl]pyrrolidine-2-carboxamide ethane;1-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]ethanone (4E)-2,6-bis[2-ethylsulfanyl-5-methoxy-3-(trifluoromethoxy)phenyl]-N,4-dimethylhepta-1,4-dien-1-amine ethane;methanamine;(E)-4,5,6-trihydroxy-N-[[(Z)-2-pyridin-1-ium-3-ylethenyl]iminomethyl]hex-4-enamide N-[2,6-dichloro-4-(5,10,10-trifluorodecyl)phenyl]-4-fluoro-3-methoxybenzamide 2-chloro-1,4-difluorobenzene;5-[4-[3,4-dimethyl-6-(trifluoromethyl)-5H-1,2-oxazol-4-yl]phenyl]-N-methylthiophene-2-carboxamide 2-(3,5-dichlorophenyl)sulfonyl-1,4-dioxane;ethene 5-(cyclobutylmethoxy)-N-[1-(furan-2-carbonylamino)ethyl]pyridine-3-carboxamide 5-(4,7-dichloroindol-1-yl)sulfanylpyridin-2-amine 1-(4-azidophenoxy)-3-[4-fluoro-N-methyl-2,6-di(propan-2-yloxy)anilino]propan-2-ol 3-[2-(difluoromethoxy)phenyl]-1,5,6,7-tetrahydrocyclopenta[b]pyridine 2-fluoro-N-(3-methylphenyl)sulfonylbenzamide 4-amino-3-(9H-fluoren-1-yl)benzonitrile 1-[5,6-dichloro-3-fluoro-2-(triazin-4-yl)phenyl]ethanol 5-cyclopropyl-3-[2-hydroxy-4-(methoxyamino)phenyl]-N'-methanimidoylpyrazolo[1,5-a]pyrimidine-7-carboximidamide [2-[2-(2,3-dihydro-1H-indene-5-carbonylamino)ethyl]-4-(1-fluoropropan-2-yloxy)phenyl]azanium 2-methyl-N-(3-nitrophenyl)-4,5-bis[[2-(trifluoromethoxy)phenyl]methoxy]aniline 7-cyclopentyl-2,3-diethoxy-4,5-bis(phenylmethoxy)-6H-benzo[h]quinazoline 5-chloro-2-[1-[2,6-dichloro-4-(trifluoromethyl)phenyl]imidazol-4-yl]pyrimidine 2,4-dimethylbenzenesulfonic acid;N'-(3-fluorophenyl)-6-methoxy-N,1-bis[4-(trifluoromethyl)phenyl]cyclohexa-2,4-diene-1-carbohydrazide 2-[4-bromobutan-2-yl(pyridin-3-yl)amino]acetamide 2-[3-(cyclopropylmethoxy)phenyl]acetic acid N-[2-amino-1-(3,5-dichlorophenyl)ethenyl]-N-pent-4-enylformamide 2-(3-bromonaphthalen-1-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 1-[2,2-dimethylpropyl(methyl)amino]-3-(4-phenyltriazol-1-yl)propan-2-ol;hydrochloride 3-bromo-5-[1,6-bis(2-ethoxyethyl)-4-oxopyrazolo[3,4-d]pyridazin-5-yl]-N-[(4-chlorophenyl)methyl]benzenesulfonamide 5-[3,5-difluoro-4-(1-methylsulfanylpiperidin-4-yl)oxyphenyl]pyrimidine [(2S)-4,4-dimethyl-3-oxopentan-2-yl]sulfanium;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide [2-(2,4-difluoroanilino)-3H-benzimidazole-5-carbonyl]-methylazanium (3aR,7aS)-N-[1-(4-hydroxyphenyl)ethyl]-5-methyl-2-pyrimidin-2-yl-1,3,3a,6,7,7a-hexahydropyrrolo[3,4-c]pyridine-4-carboxamide 4-[(3,5-dimethoxyphenyl)sulfonyl-methylamino]benzenecarboximidamide;hydrochloride 7-(1,3-benzothiazol-6-ylamino)-2-cyclopropyl-[1,3]oxazolo[5,4-d]pyrimidine-6-carboxylic acid 2-[6-(2,5-dichlorophenyl)-1H-indol-3-yl]-N-[4-(1H-imidazol-5-ylmethyl)phenyl]acetamide 2-(4,5,6-trimethylpyrimidin-2-yl)sulfanylpropanedioic acid 5-[4-methyl-3,6-dioxo-2-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)cyclohexa-1,4-dien-1-yl]pyridine-3-carbonitrile N-[[3,5-bis(trifluoromethyl)phenyl]methoxy-dihydroxyphosphinothioyl]benzamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-6-propanoylpyridine-2-carboxamide 3-[(2R,4S)-4-azido-3,4-dimethylpentan-2-yl]phenol 2-methyl-4,6-dinitropyrimidine 2-(3,4-dimethylphenyl)spiro[4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-6,3'-pyrrolidine] 2-[2,6-dibromo-4-(5-oxo-2-sulfanylidene-3,6-dihydropyrimido[4,5-d]pyrimidin-4-yl)phenoxy]propanenitrile 6-(2,5-dimethylpyrrol-1-yl)quinazolin-4-amine 2-(4-methoxyanilino)-5,6,7,8-tetrahydro-3H-quinazolin-4-one ethane;4-ethenyl-3,5-bis(ethenyl)aniline N-(4-fluoro-3-nitrophenyl)sulfanylmethanamine 5-[1,3-dioxo-2-(trifluoromethyl)isoindol-5-yl]oxypyridine-3-carboxamide 1-benzyl-3,6,9,11-tetrahydropyrazolo[3,4-a]acridine (NE)-N-[2-imino-1-[4-methoxy-3-(trifluoromethyl)phenyl]ethylidene]hydroxylamine 4-[2,3,5,6-tetrafluoro-4-(trifluoromethyl)phenyl]cyclohexan-1-one 1-[[2-chloro-5-(dimethylamino)phenyl]methyl]indole-3-carboxylic acid N-[2,6-difluoro-4-(1H-pyrazol-5-yl)phenyl]-4-hydroxy-2-methoxybenzamide N-[4,6-dimethoxy-3-(propan-2-ylamino)quinoxaline-5-carboximidoyl]propanamide;dihydrochloride 6-(6-azidohexyl)benzene-1,2,3,4,5-pentol 3-[2-(benzylamino)ethyl]-2,5-dihydroxycyclohexa-2,4-dien-1-one 1-azido-2-(3-fluoro-5-methoxyphenyl)piperidine 2-chloro-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethyl)pyrimidine-4-carboxamide;dihydrochloride N-(2,4-difluorophenyl)-6-oxo-1H-pyrimidine-2-carboxamide;5-hydroxypentanoic acid 1-(3-benzylquinolin-5-yl)-N-methoxymethanamine 6-[3,5-dimethyl-1-(2-piperidin-4-ylethyl)pyrazol-4-yl]-3H-quinazolin-4-one;hydrochloride N-[3-(dimethylamino)propyl]-6,8-dihydroxy-1H-indole-2-carboxamide 2-amino-N-[1-(4,4-difluorocyclohexyl)imidazol-4-yl]thieno[3,2-d]pyrimidine-7-carboxamide 6-[[4-(cyclohexen-1-yl)-N-[2-hydroxy-3-[(E,3R)-7,7,7-trifluorohept-5-en-2-yl]phenyl]sulfonylanilino]methylideneamino]-4H-phthalazine-1,3-dione (1R,2S)-2-(5-fluoro-4-morpholin-4-ylpyridine-2-carbonyl)cyclohexane-1-carboxylic acid 5-(2,6-dichloro-4-fluorophenyl)-3H-1,3,4-thiadiazol-2-one 1-[6-(cyclohexylmethoxy)quinolin-8-yl]ethanone 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]acetic acid 1-azido-2,3-dibromo-4-(3-bromophenyl)benzene 6-(3,4-difluorophenyl)-2-methylimidazo[1,2-a]pyrazine 2-bromo-N-tert-butyl-3,4-dimethoxyaniline 2-(4-azidophenoxy)-1,3-benzothiazole 3-fluoro-2-(6-oxo-1,7-dihydropurin-8-yl)benzamide ethane;methanethiol;(E)-3,5,7,11-tetraoxo-N-[2-(pyridin-4-ylamino)-1H-inden-5-yl]hept-6-enamide N-azido-3,4-dihydroxybenzenesulfonamide 1-[5-(2,3,6,7,8,9,9a-octahydro-1H-quinolizine-4-carbonyl)-2-hydroxyphenyl]-4-methylpentan-1-one (2R,4S)-1-[(1S)-2-cyanocyclohexyl]-N-hydroxy-4-methoxypyrrolidine-2-carboxamide;N'-[1-(7H-purin-6-ylamino)propan-2-ylideneamino]ethanimidamide 3-(1H-benzimidazol-2-yl)-5-[1-(cyclohexylmethylamino)ethenyl]phenol;ethane N-(2,4-dichloropyrimidin-5-yl)-4-nitro-N-propylbenzamide (3aR,6R,7aS)-4-[(2S)-1-[2-methyl-5-(trifluoromethyl)pyrazole-3-carbonyl]piperidin-2-yl]-N-propan-2-yl-3,3a,5,6,7,7a-hexahydro-2H-furo[3,2-b]pyridine-6-carboxamide 2-[2-[4-(3,6-dihydroxyhexoxy)phenyl]-1,2,3,5-tetrahydropyrrolizin-7-yl]acetic acid 2,4-dihydroxy-5-[[3-(5-methylfuran-2-yl)-1-phenylpyrazol-4-ylidene]methyl]-N-phenylbenzamide 1-N',2-bis(4-fluorophenyl)ethanedihydrazide 5-[[7-(4,6-dimethylpyrimidin-2-yl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]piperidine-3-carboxylic acid 6-chloro-5-[(2,4,6-trifluorophenyl)methyl]-2H-triazolo[4,5-b]pyridine 1-[4-(6,7,8,9-tetrahydrodibenzofuran-2-yl)phenyl]ethanone 1-[4-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]phenyl]-3-methylidenepyrrolidine-3,4-diol 3-[(Z)-1-amino-3-iminoprop-1-enyl]-7-tert-butyl-1H-quinoxalin-2-one 2-[3,5-dimethyl-4-(oxiran-2-ylmethoxy)phenyl]acetaldehyde 2-[(Z)-[3-[2-(3,4-dimethoxyphenyl)ethylamino]-6H-benzo[c][1]benzoxepin-11-ylidene]methyl]phenol 2-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]-10H-cyclohepta[b]naphthalene 6-[(3S)-4-azido-3-methylpiperazine-1-carbonyl]pyridine-3-carbonitrile 7-[2-[(5-chloropyridin-2-yl)amino]acetyl]-N-[[1-(2,3-dihydroindol-1-ylsulfonylcarbamoyl)cyclopropyl]methyl]-8-oxo-1H-pyrrolo[1,2-a]quinoxaline-2-carboxamide 3-amino-4-(2,4-difluorophenyl)butanal;ethane 2-azido-7-methoxy-1-(3,4,5-trifluorophenyl)isoquinolin-2-ium 3-(4-aminophenyl)imino-6-methyl-1H-indol-2-one (E)-3-[2,5-dimethyl-4-(4-propanoylphenyl)thiophen-3-yl]prop-2-enenitrile (2S)-1,3,3-trimethyl-2-prop-2-enoxy-2H-indole 3-benzyl-5,6-diethoxy-1H-pyrimidine-2,4-dione (3-amino-6,7-dimethoxyquinoxalin-2-yl)-[4-chloro-2-hydroxy-5-(trifluoromethyl)phenyl]methanone 2-(3-fluoro-4-propan-2-yloxyphenyl)oxolane N-(2-aminoethyl)-3,4,6-trichloro-5-methoxybenzenesulfonamide;hydrochloride 7-[[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]methylamino]-1H-pyrido[4,3-b]indole-3-carboxylic acid 2-(2,4-dichlorophenoxy)-N-[1-oxo-5-propyl-8-(3,3,3-trifluoropropylsulfanylamino)phthalazin-6-yl]acetamide N-[(2S)-1,3-dihydroxypropan-2-yl]-6-methoxy-5H-cyclopenta[b]pyridine-7-carboxamide 1-[7,8-dimethyl-5-(2H-tetrazol-5-yl)-4,9-dihydropyren-1-yl]ethanone N-[3-(methylamino)phenyl]-2-nitrobenzamide 3-chloro-4-fluorobenzo[g][1,2]benzoxazole 4-methyl-6-[(1E)-2-pyridin-3-ylbuta-1,3-dienyl]pyridine-3-carboxylic acid N-ethyl-6-(furan-2-ylmethylamino)hexanamide 1-[2-(5-methoxy-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-3-yl)pyrimidin-4-yl]piperidine-3-carboxamide 2-(3,4-dimethoxyphenyl)-N-(5,6,7,8-tetrahydronaphthalen-1-ylsulfamoyl)acetamide 4-(2,6-dimethoxybenzoyl)-N'-hydroxypyridine-3-carboximidamide 3-[1,1-difluoro-5-(2-hydroxyethyl)cyclohexa-2,4-dien-1-yl]oxybenzonitrile 2-(3-fluoropyridin-4-yl)-N-[5-[[(E)-1,3-thiazolidin-5-ylidenemethylamino]methyl]pyridin-2-yl]oxyacetamide (1Z)-3,6-dimethylheptacyclo[d]triazole;ethane;2-(4-methylphenyl)sulfanylpentanoic acid 2-[6-(4,5-dimethylpyrazol-1-yl)pyridin-3-yl]-N-methoxysulfanyl-N-methylethanamine N'-(1-pyridin-3-ylpropan-2-ylideneamino)ethane-1,2-diamine 4-[(1R)-1-[4-amino-3,5-bis(methoxymethyl)phenyl]ethoxy]benzaldehyde;N-methylethanamine (7S)-8-cyclopropyl-2,7-dimethyl-5-oxo-6H-pyrido[3,4-b]pyrrolizine-1-carboxamide 1-benzyl-3-(2,4-dichloropyrimidin-5-yl)-1,3-dimethylurea 1-[(Z)-(2-hydroxy-3,5-dinitrophenyl)methylideneamino]-2-propan-2-ylguanidine 1-(2-fluorophenyl)sulfinylpyrrole N-[(1E)-3-[4-[2-(dimethylamino)ethoxy]phenyl]buta-1,3-dienyl]-N'-(1H-indol-5-yloxy)ethanimidamide 2-[3-[4-(2-aminoethyl)phenyl]pentan-3-yl]phenol;3,5-dimethoxycyclohexa-1,3-diene 4-[5-amino-1-[(3,4-dimethylphenyl)methyl]pyrazole-4-carbonyl]piperazin-2-one (E)-2-[(3Z,5Z)-6,8-dichloroocta-3,5-dienoxy]but-2-enenitrile;ethane 3-[(2,6-dimethylphenyl)carbamoylamino]benzoate 5-methyl-3,4-dihydro-2H-chromene;(2S)-2-methyl-1-phenyl-6-pyrrolidin-1-ylhexan-3-ol 4-N,8-dimethylanthracene-1,4-disulfonate N-[2-(5-phenyl-1,3,4-oxadiazol-2-yl)ethyl]-4H-pyrido[2,3-e][1,3]thiazin-8-imine 4-methyl-1-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxylic acid 2-[5-[3,5-dimethyl-4-(4-oxo-1,3-benzothiazin-2-yl)phenyl]pyridine-3-carbonyl]sulfanylacetic acid (6S)-N,1,2,3,6-pentamethyl-4,5,6,7-tetrahydroindazole-6-carboxamide 5-[4-amino-7-methyl-6-[4-(2,4,6-trifluorophenoxy)phenyl]pyrrolo[2,3-d]pyrimidin-5-yl]oxy-4-oxopentanoate (E)-2-[(3,4-dihydroxyphenyl)methyl]-4-(5-fluoropyridin-2-yl)but-3-enoic acid 1-N'-(5-bromopyridin-2-yl)butane-1,1,3-triamine N-(4,5-dimethyl-2-phenyldiazenylphenyl)-3-methoxybenzamide 5-[(2S,4R)-1-[2-cyclobutyl-6-oxo-4-(trifluoromethyl)pyrimidine-1-carbonyl]-4-fluoropyrrolidin-2-yl]-3H-1,3,4-oxadiazol-2-one 3-N-[5-(2,4-dimethylphenyl)sulfanyl-1,3,4-thiadiazol-2-yl]-5-(trifluoromethoxy)pyridine-2,3-diamine 2-[4-(3,5-dimethylphenyl)butan-2-yl]-N,N-diethylbenzamide 4-methyl-3-[(5S)-8-[2-(trifluoromethylsulfonyloxy)ethoxy]spiro[4,6-dihydro-3H-pyrimido[1,5-a]azepine-9,1'-cyclopropane]-5-yl]benzoic acid 5-fluoro-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3H-quinolin-4-one N-[1-(3,5-difluorophenyl)ethyl]-2-methoxybenzamide 3-[[4,6-bis(4-cyanophenyl)-1,3,5-triazin-2-yl]oxy]benzenesulfonic acid 2-(azidomethoxy)-6-[[4-(trifluoromethyl)cyclohexyl]methoxy]naphthalene N-methyl-1-(6-propan-2-ylpyrimidin-4-yl)piperidine-3-carboxamide N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]-3-propan-2-ylidenepiperazine-1-carboxamide 1-aminosulfanyl-2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]propan-2-ol N-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-sulfonamide 2-cyclopropylsulfonylnaphthalene 1-[2-(2,5-dioxoimidazolidin-4-yl)ethynyl]-3-(1-pyridin-4-ylpyrazol-4-yl)urea (4R,5S)-N-(cyclobutylmethyl)-6-(furan-2-yl)-8-(3-phenylpropanoyl)-2,8-diazaspiro[4.5]decane-4-carboxamide N-[2-(2,4-dichlorophenoxy)propanoyl]-3,6-diazabicyclo[3.1.0]hexane-6-carboxamide (2S)-4-[cyclohexyl-[(1R,3S)-3-naphthalen-1-yl-1-pyridin-3-ylsulfonylcyclopentyl]amino]-N-hydroxy-2-methoxybutanamide 1-[(2R)-5,6-dichloro-4-fluoro-2,3-dihydro-1H-inden-2-yl]pyrrolidine;3-methoxycyclobutane-1-carboxamide 3-N-[3,5-difluoro-2,4,6-tri(propan-2-yl)phenyl]-1-N,1-N-dimethylpentane-1,3-diamine;ethane 2-chloro-4-[3-[(4R)-5,5-dimethyl-1-(4-methylphenyl)sulfonyl-4H-pyrazol-3-yl]prop-2-enoylamino]benzoic acid [(2S)-1,3-dimethyl-2H-benzimidazol-5-yl]-(8-fluoro-1,3,4,6,7,9-hexahydropyrido[2,1-b]quinazolin-2-yl)methanone 3-[4-(1,2-dimethylcyclohexa-2,4-dien-1-yl)phenyl]benzonitrile N-[(2S)-1-(6-chloroimidazo[1,2-a]pyridin-3-yl)propan-2-yl]-6-cyclopentyloxypyrimidin-4-amine 4-[2-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]ethyl]benzonitrile 5-N,4-N-dimethyl-3-nitropyridine-2,4,5-triamine N-[(E)-1-[4-[2-(5-chloropyridin-3-yl)ethynyl]phenyl]prop-1-enyl]cycloheptanamine 5-[(4E)-4,7,8,9-tetramethylnona-1,4-dien-6-yn-3-yl]-2H-tetrazole 4-[4-(4-cyanophenyl)phenyl]benzenesulfonamide 3-[(2R)-1,1-difluoroethyl]-N'-[2-(4-methylphenyl)-6-pyrrolidin-1-ylpyrimidin-4-yl]oxybenzenecarboximidamide 6-amino-4-[2-(dimethylamino)phenyl]-4-methyl-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile 6-[3-(3,5-dichlorophenyl)pyrrolidine-1-carbonyl]pyridine-3-carbonitrile;4-(2-methyl-4-nitrophenoxy)benzoic acid (3S)-4,4,5,5-tetramethyl-2-phenoxyheptanamide 2-[3,5-bis(2,4-dimethylphenyl)phenyl]pyridine 4-fluoro-6-(3-pyridin-2-ylimidazo[1,5-a]pyrazin-8-yl)benzo[c][1]benzazepine 2-[(2,5-difluorophenyl)methyl]spiro[3,4-dihydroisoquinoline-1,4'-piperidine] 2-N,5,6-trimethyl-4-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]pyrimidine-2,4-diamine 5-bromo-3,7-dimethyl-2H-naphthalen-1-one 4-[azido(diphenyl)methyl]-2-chloropyridine 2-(aminomethyl)-5-[1,3-dioxo-4-(trifluoromethoxy)isoindol-2-yl]hexanoic acid [2-amino-5-(oxolan-3-yl)phenyl]methylideneazanium 2-(1H-indol-3-yl)-N'-phenylacetohydrazide 4-(6,8-dibromo-3H-1,5-benzodiazepine-7-carbonyl)morpholine-2-carboxylic acid 5-(cyclohexylmethoxy)-N'-[5-methyl-2-(4-oxo-1-phenyl-5H-pyrazolo[3,4-d]pyrimidin-6-yl)pyrazol-3-yl]furan-2-carbohydrazide 4-amino-6-[(3,5-dibromo-2-hydroxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-N,3-N-bis(2-propan-2-yloxyphenyl)pyrazine-2,3-dicarboxamide N-[4,5-dichloro-2-(8-fluoro-4-oxochromene-3-carbonyl)phenyl]methanesulfonamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-methoxypyrimidine-2-carboxamide 5-[1,2-dimethyl-4-(2-propan-2-ylphenyl)benzimidazol-5-yl]sulfanylpyridine-3-carbonitrile N-[(3-fluorophenyl)methyl]-6,7-dihydro-5H-pyrrolizine-1-carboxamide 1-amino-6-chloro-N,3-bis(4-fluorophenyl)indole-2-carboxamide N-ethylsulfonyl-4-[[(2S)-2,3,5,7,8-pentamethyl-1,2,3,4-tetrahydronaphthalen-6-yl]oxy]benzamide [(3S)-5,8-difluoro-3-propyl-2,3,4,9-tetrahydro-1H-carbazol-2-yl]methanol (2R,4S)-4-amino-2-phenylcyclohexane-1,3-dione 1-[2,4-bis(propan-2-ylperoxy)phenyl]naphthalene N-[5-(2,3-dimethylphenyl)-1H-pyrazol-4-yl]-6-fluoroquinoline-7-carboxamide 2,4-dimethyl-6-[1-(1H-pyrrol-3-yl)butan-2-yl]pyrimidine 4-[5-amino-6-(4-fluorophenyl)pyridin-2-yl]-N-methyl-1,3-thiazole-2-carboxamide;[(3S,4R)-2-(3-chloro-4-propoxybenzoyl)-4-hydroxypyrrolidin-3-yl]azanide;yttrium (E)-3-[2-[4-[(1R)-1-hydroxyethyl]anilino]pyrimidin-5-yl]-N-oxido-3-pyridin-3-ylprop-2-enamide 3-[2-cyclopropyl-1-[(Z,4E)-4-[5-ethylidene-7-fluoro-6-methoxy-2-oxo-1-(oxan-4-ylmethyl)quinolin-8-yl]hex-4-enoyl]azetidin-3-yl]benzonitrile (Z)-N'-[4-[2-[5-amino-8-fluoro-6-(methylamino)-3,4-dihydro-1H-isoquinolin-2-yl]ethoxy]phenyl]-3-(3-hydroxypropylimino)but-1-ene-1,5-diamine 2-[3,5-difluoro-4-(triazol-1-yl)anilino]quinoline-8-carboxylic acid 1-azido-3-[4-(9H-fluoren-1-yl)phenoxy]piperidine 6-ethyl-7-hydroxy-4H-1,3-benzodioxine-5,8-dione 2-[[3-(trifluoromethoxy)phenyl]carbamoylamino]spiro[1,4-dihydroquinoline-3,4'-piperidine]-6-carboxamide ethane;4-fluoro-N,1-dimethylpyrrolidine-2-carboxamide;6-[4-hydroxy-3,5-bis(methoxysulfanyl)phenyl]imino-2,4-dioxo-1H-pyrimidine-5-carbonitrile (2S,4S)-N-[(3,5-dimethylpyrazol-1-yl)methyl]-4-fluoropyrrolidine-2-carboxamide;hydrochloride N-[3-[(E)-2-methoxyethenyl]phenyl]-1H-pyrrole-2-carboxamide N-[4-chloro-3-(6-methoxypyrimidin-4-yl)phenyl]-2,5-difluoro-4-iodobenzenesulfonamide 4-ethylbenzoic acid;3-[1-(2-phenylpropyl)piperidin-4-yl]-3H-indene-1,2-dione 2-[3,5-diamino-6-(2,6-difluorophenyl)pyrazin-2-yl]phenol [7-cyclopropyloxy-2-(1,3-dimethylpyrazol-4-yl)-6-fluoroquinolin-5-yl]boronic acid (3aR,7aS)-2-[1-(4-fluorophenyl)ethyl]-5-methylsulfonyl-1,3,3a,6,7,7a-hexahydropyrrolo[3,4-c]pyridin-4-one 4-[[[5-(cyclopropylmethyl)-1,3-thiazol-2-yl]amino]methyl]benzenesulfonamide (2S)-N'-[6-methyl-5-[(1R,3R)-3-(quinolin-8-ylamino)cyclopentanecarbonyl]pyridin-2-yl]pyrrolidine-2-carbohydrazide N-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-2-methoxybenzenesulfonamide (2S,4R)-2-cyclohexyl-1-(2-methoxyethylamino)-4-phenylmethoxycyclopentane-1-carboxylic acid N-[(2R)-1-[(3S,4R)-3,4-dihydroxypyrrolidin-1-yl]-3-(4-fluorophenyl)butan-2-yl]-5-[4-(trifluoromethoxy)phenoxy]naphthalene-2-carboxamide 1-N,4-N,5-tripyridin-3-ylpyridine-2,4-dicarboxamide 4-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[[3-methoxy-5-(methylsulfanylamino)cyclohexa-2,4-dien-1-ylidene]amino]aniline 4-hydroxy-2-(N-octylanilino)benzoic acid 3-methyl-2-[(5-nitrofuran-2-yl)methylidene]butanedinitrile 2-(4-aminophenyl)-N-[(1R,3S)-3-cyclopropylcyclopentyl]acetamide;hydrochloride 3-(7-fluoro-1H-pyrrolo[2,3-c]pyridin-3-yl)azetidine-1-carboxylic acid 4-azido-N'-(3,4-dimethylphenyl)pyrimidine-2-carboximidamide 4-azidooxy-N,5-dimethylpyrimidine-2-carboxamide 1-[(3R,6S)-4-benzyl-2,8-diazaspiro[5.5]undecan-3-yl]ethanone;hydrochloride (3-chlorophenyl)methyl-diethyl-[[5-[4-ethoxycarbonylpiperazin-1-yl]pyrazin-2-yl]methyl]azanium (2S)-3-methyl-2-[N-(9H-thioxanthen-1-ylsulfonyl)anilino]butanoic acid 2-tert-butyl-N-(3,5-diethyl-1,3,4-thiadiazol-2-ylidene)pyridine-4-carboxamide 1-cyclohexa-1,3-dien-1-yl-2-[4-(2-methoxyethoxy)phenyl]-2-[6-(piperidin-3-ylamino)hexa-2,4-diynylamino]ethanol N-[4,5-bis(ethenyl)pyrimidin-2-yl]acetamide 5-[3-(2,4-dichlorophenyl)propyl]-2-ethylcycloheptane-1,4-dione 2-hydroxy-4,6-dimethyl-3-propanoyloxybenzenesulfonic acid 1-[3-[[2-(4-methylpiperazin-1-yl)thieno[3,2-d]pyrimidin-4-yl]amino]phenyl]prop-2-en-1-one 1-[4-(1,3-benzodioxol-5-ylmethoxy)phenyl]pyrazole N'-[(1Z)-buta-1,3-dienyl]-N-methylidene-4-phenylbenzenecarboximidamide 5-[(2,5-dimethylphenyl)sulfonylamino]-N'-hydroxypyridine-3-carboximidamide 2-[(4-bromophenyl)-diethoxyphosphorylmethyl]benzenesulfonic acid 1-azidosulfanyl-2,3,4-trimethoxybenzene 5-[4,6-bis(2-methylbutan-2-yl)-1,3,5-triazin-2-yl]-2-(oxolan-3-yloxymethyl)tetrazole 3-(azidomethyl)quinoline-4-carboxamide 1-cyclohexyl-5-(4-ethoxy-3,5-dimethoxyphenyl)pentan-2-one 1,7-dimethyl-5H-pyrazolo[4,3-c]quinolin-4-one [1-(4-azidooxy-3,5-difluorophenyl)-2-ethyl-7H-pyrrolo[3,2-d]pyrimidin-6-ylidene]methanamine 2-methyl-4-[(3E)-3-[(Z)-pent-3-enylidene]cyclopenta-1,4-dien-1-yl]butan-2-amine 5-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]pyridine-2-carbonitrile 3-(azidomethoxy)-2,6-difluorobenzenethiol 6-[2,5-dichloro-N-(4-hydroxybutyl)anilino]-4-hydroxynaphthalene-2-sulfonic acid 2-[5-methoxycarbonyl-3,6-dimethyl-1-(2-phenylethyl)-3a,4-dihydropyrrolo[3,4-c]pyrazol-4-yl]acetic acid 1-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[2-hydroxy-1-(1H-indol-6-yl)ethyl]urea 2-[(E)-4,4-dimethylpent-1-enoxy]benzaldehyde 6-(3-aminocyclobutyl)-N-[[2,4-difluoro-5-(1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl]methyl]pyrimidin-4-amine;dihydrochloride 2,3-dichloroquinoxaline 3-[(5S)-2,2-dimethylnonanoyl]-1H-quinolin-4-one 2-N-(3,4-dihydro-1H-isochromen-5-yl)-1,3,5-triazine-2,4,6-triamine 5-fluoro-2-[1'-(pyridine-4-carbonyl)spiro[3,4-dihydrochromene-2,4'-piperidine]-6-yl]oxybenzonitrile;2,2,2-trifluoroacetic acid 1-[(2,4-dichlorophenyl)methyl]-3-pyridin-4-ylpyrazolo[3,4-b]pyridine 2-(furan-2-ylmethylamino)-5-[(3-hydroxyphenyl)sulfonylamino]pyridine-3-carboxylic acid;2,2,2-trifluoroacetic acid N-[2-(4,5-dichloroimidazol-1-yl)ethyl]propanamide (5-amino-6-tert-butylsulfinylpyrazin-2-yl)-pyrrolidin-1-ylmethanone N-benzyl-5-chloro-2,4-dihydroxybenzenesulfonamide 2-[6-(dimethylamino)pyridin-3-yl]oxyethanesulfonic acid 5-[(2R)-2,3-dihydropyridine-2-carbonyl]-4-hydroxy-6-methoxypyran-2-one (2S,4S)-1-[3-(2,6-dichlorophenyl)propanoyl]-N-[(3-fluoro-5-methoxypyridin-2-yl)methyl]-4-hydroxypyrrolidine-2-carboxamide 2,3-bis(2,4-difluorophenyl)oxirane 3-[[4-(4-methylphenoxy)piperidin-1-yl]sulfonylamino]benzoic acid;hydrochloride N-[5-[6-fluoro-3-(7-pyridin-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclopropanecarboxamide N-[(4Z)-4-amino-4-cyclopropyliminobutoxy]-2-cyano-3-[3-ethyl-5-fluoro-4-(5,6,7,8-tetrahydronaphthalene-1-carbonyl)phenyl]benzamide 3-azido-2,4-difluoro-N-[(2S)-1-hydroxypropan-2-yl]benzamide 5-[4-[3-(3,5-difluoropyridin-2-yl)phenyl]sulfonylmorpholin-2-yl]-1H-pyrimidine-2,4-dione 3-methyl-2,4-dioxo-N'-[(3-phenylmethoxypyrazin-2-yl)methyl]pentanehydrazide 2-(dipropylamino)-N-[2-methyl-3-(trifluoromethoxy)phenyl]acetamide N-(2,4,5-trichlorophenyl)sulfanyl-1H-indole-3-carboxamide 1-[3,4-difluoro-2-(trifluoromethyl)phenyl]pyrrole N-[4-[(2E,4Z)-hepta-2,4,6-trien-3-yl]oxy-2,5-dimethylphenyl]furan-2-carboxamide N-(4-carbamoylphenyl)-3,5-dihydroimidazo[2,1-b]purine-7-carboxamide 3-[(Z)-1-iminobut-2-en-2-yl]-N-methyl-4-[1-methyl-5-(trifluoromethyl)pyrazol-4-yl]aniline 3,5-dichloro-N-[2-(4-methyl-6-oxo-1H-pyrimidin-2-yl)-5-phenylpyrazol-3-yl]benzamide 5-[4-(bromomethyl)phenyl]-1-tritylindazole 2-azidooxy-5,6-dimethylbenzo[de]isoquinoline-1,3-dione 2-[3,5-bis(trifluoromethyl)phenyl]cyclohepta-1,3,5-triene 2-[4-(3-ethoxyprop-1-enyl)phenyl]sulfonyl-5,6-dihydrothieno[3,2-b]pyrrole [3-(1,5-dimethylimidazol-2-yl)piperidin-1-yl]-(6-hydroxypyridin-3-yl)methanone 5-[2-ethoxy-5-(4,4,5,5-tetramethyloxaborolan-2-yl)phenyl]pyrimidine (E)-3-[3,5-bis(trifluoromethyl)phenyl]-1-[(4S)-2-pent-1-ynyloxepan-4-yl]prop-2-en-1-one 4-(1H-benzimidazole-2-carbonyl)-3,5-dihydro-2H-1,4-benzothiazepine (5S,7R)-N-[2-(4-chlorophenyl)ethyl]-1,5,7-trimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carboxamide 3-(1-chloroethenyl)-1H-quinoxalin-2-one 2-(3,4-difluorophenyl)-7-[4-(methylamino)-1H-pyrrole-2-carbonyl]cyclohepta-2,5-diene-1,4-dione;hydrochloride (4S)-3,6,9,10-tetrahydroxytricyclo[7.1.02,7]trideca-2(7),3,5-triene-8-carboxylic acid 6-(5-cyanopyridin-2-yl)oxy-N,1-dimethylindole-3-carboxamide;propane 4-[5-(aminomethyl)-1,2,4-oxadiazol-3-yl]benzene-1,3-diol 3-[5-chloro-2-(methylamino)phenyl]-N-(4-ethylpyridin-3-yl)imidazo[1,2-a]pyrazin-8-amine 5-(4-methylphenyl)sulfonyloxypentanoic acid [2-amino-5-(trifluoromethyl)phenyl]-[1-cyclopenta-2,4-dien-1-ylidene-3-[(4S)-4-[[1-cyclohexyl-2-(ethoxymethyl)benzimidazole-5-carbonyl]amino]piperidin-3-yl]prop-1-enyl]azanium N-(1,3-benzodioxol-5-ylmethylideneamino)-2-[1-[4-(trifluoromethoxy)phenyl]triazol-4-yl]quinoline-4-carboxamide [4-(4-methoxyphenyl)sulfanylphenyl]carbamic acid 5-fluoro-4-[1-[2-(methoxymethyl)pyrrolidine-1-carbonyl]cyclopropyl]-3H-2,1,3-benzoxadiazole-7-carboxylic acid 6-(cyclohexanecarbonylamino)imidazo[1,2-b]pyridazine-3-carboxylic acid 1-[4-fluoro-3,5-di(propan-2-yl)phenyl]piperidine 1-methylsulfonyl-4,5,6,7-tetrahydroindazole N-[5-(2,4-dihydroxy-5-propan-2-ylphenyl)-4-[1-(2,6-dimethylanilino)-3-methylbutyl]sulfanyl-1,3-thiazol-2-yl]acetamide 3-(4-fluorophenyl)-1-[2,2,2-trifluoro-1-(3-methoxyphenoxy)ethyl]azetidine;N-piperidin-4-ylcarbamate 2-[[1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]methoxy]pyridine-4-carbonitrile;hydrochloride (E)-3-(2,4-dihydroxyphenyl)-N-[1-[3-[4-(dimethylamino)quinazolin-2-yl]sulfanylpropoxy]-2-methylpropan-2-yl]prop-2-enamide N-(2,6-dioxopiperidin-3-yl)-1H-thieno[2,3-d]imidazole-5-carboxamide N-cyclohexyl-N-(2,3-dihydroxypropyl)benzamide 2-(4-tert-butylcyclohexa-1,3-dien-1-yl)sulfonyl-6-nitrobenzenesulfonamide 3-benzylsulfanyl-4,5-dichlorobenzenethiol 2-[(4,5-dimethylthiophene-3-carbonyl)amino]-1-ethyl-N-(1-hydroxypropan-2-yl)benzimidazole-5-carboxamide 2-amino-6-(3-hydroxyphenyl)pyridine-4-carbonitrile 4-fluoro-N-[(2S)-3-methylbutan-2-yl]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide 3-(2,4-dimethoxyphenyl)cyclopentan-1-one 2-[[4-(3,5-dichlorophenyl)sulfinylpiperazin-1-yl]methyl]-8a-methyl-6,7,8,9-tetrahydro-4H-imidazo[2,1-c][1,4]benzothiazine N-[2,3-difluoro-4-[4-(5-propan-2-yl-1H-pyrazol-4-yl)pyridin-2-yl]oxyphenyl]-4-ethylsulfanylbutane-1-sulfonamide N-[6-[(3R)-3-aminopiperidine-1-carbonyl]-4,5-dimethylpyridin-2-yl]acetamide 5-methoxy-N'-[2-(3-nitrophenoxy)ethyl]thiophene-2-carboximidamide 4-[2,6-difluoro-3-[(5-oxo-1H-tetrazol-4-yl)methoxy]phenyl]-6-ethynyl-7-fluoro-1-(oxan-2-yl)quinolin-2-one 3-benzylsulfanyl-1,2,4,5-tetrafluorobenzene 2-[(2Z)-2-[(3,5-dichlorophenyl)methylidene]hydrazinyl]-4-(2,6-dimethoxyphenyl)-1H-pyrimidin-6-one 3-benzylsulfanyl-5-[(2R)-pentan-2-yl]-8H-[1,2,4]triazolo[4,3-a]pyrimidin-7-one 2-chloro-3-fluoro-4-(methylamino)benzenesulfonamide;4-[(6S,9S,13R,14S)-17-ethyl-13-methyl-7,8,11,12,15,16-hexahydrocyclopenta[a]phenanthrene-2,3-dimethoxy-1-carbonyl]benzaldehyde (2S,4R)-N-[1-[[6-amino-5-(trifluoromethyl)pyridin-3-yl]methoxy]naphthalen-2-yl]-4-benzamidopyrrolidine-2-carboxamide N-(4-chlorophenyl)-N'-[1-(4-methoxy-3-methylbenzoyl)piperidin-4-yl]oxamide [(2S)-1-[[2-methyl-7-[3-(trifluoromethoxy)phenyl]pyrazolo[4,3-c]pyridin-4-yl]amino]butan-2-yl]carbamic acid 2-[(3Z)-3-ethoxyiminoindol-2-yl]-5,7-dimethoxy-3H-quinazolin-4-one N-methyl-2-(4-propoxyphenoxy)acetamide N-[3,5-bis(trifluoromethyl)phenyl]-6-azidooxy-1-(4-ethylsulfonylpiperazin-1-yl)cyclohexa-2,4-diene-1-carboxamide 5-benzyl-3,4-dichloro-1-propan-2-ylindazole N-[3,4-difluoro-5-[2-(methylamino)pyrimidin-4-yl]oxyphenyl]benzenesulfonamide 1-methylsulfinylindole-3-carboxylic acid 3-(4-chlorophenyl)-N'-hydroxy-5-[2-[methyl(propan-2-yl)amino]ethoxy]pyridazine-4-carboximidamide 1,4-dimethyl-2-oxo-N-(5-thiophen-3-yl-1H-pyrazol-3-yl)quinoline-6-carboxamide (Z)-1-[1-[5-chloro-6-methyl-4-(oxan-2-yloxy)pyridin-3-yl]ethylideneamino]ethenethiol 1-(4,6-dimethylpyrimidin-2-yl)-1,3,5-triazepane ethane;N-[3-(4-methylpiperazine-1-carbonyl)-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl]formamide 2-[1,3-benzodioxol-5-ylmethoxy(ethyl)amino]acetamide N'-hydroxy-5,6-dimethyl-3-[2-(oxolan-2-ylmethylamino)ethoxy]pyridazine-4-carboximidamide 6-benzyl-3-(piperidin-4-ylmethoxy)-1,2-dihydro-[1,2,4]triazolo[4,3-b]pyridazine 5-methoxy-4-[1-(2,3,6-trifluoro-4-methylphenyl)cyclopropyl]benzaldehyde N-[2-(2,6-dimethylphenyl)pyrazol-3-yl]-2-(3-ethoxycyclobutyl)acetamide 4-[(2,3-dichlorophenyl)methyl]-1H-pyrimidine-2,4-diamine N-[3-[5-chloro-2-[(6-fluorocyclohexa-1,3-dien-1-yl)amino]pyridin-4-yl]phenyl]prop-2-enamide 2-[4-fluoro-3,5-di(propanoyl)phenyl]acetate 1-bromo-3,7-dimethyl-2H-purine 3-[4-(6-fluoro-1H-indole-2-carbonyl)piperazin-1-yl]propanoic acid 4-[2-(azidomethyl)pyrrolidine-1-carbonyl]benzenesulfonamide N-[(Z)-1-amino-3,4,5-trimethylhept-2-en-2-yl]-2-cyanobenzamide 3-(5-chloro-2-morpholin-4-ylpyridin-4-yl)-1,6,7-triazabicyclo[4.2.0]octa-2,4-dien-8-ol 2-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine;6-propan-2-ylisoquinoline 4-[[2-ethyl-3,5-dimethyl-6-(1-methylcyclopropyl)benzimidazol-4-yl]oxymethyl]benzonitrile N-[2-(1H-indole-3-carbonyl)phenyl]thiophene-2-sulfonamide N-[2-(diethylamino)ethyl]-6,8-dimethoxy-1H-indazole-5-carboxamide ethane;(2E,5Z)-6-imino-4-[(methylideneamino)-phenylmethyl]hexa-2,5-dien-3-ol 2-(N-(4-aminophenyl)anilino)acetonitrile 2-(2-chlorophenyl)-1,3-benzothiazole 4-chloro-5-(3,7-dimethylocta-2,6-dienoxy)pyridine-2,3-diamine (1R)-N-[5-tert-butyl-2-hydroxy-3-[(4-methoxyphenyl)methylideneamino]phenyl]-1,2,3,4-tetrahydroisoquinoline-1-carboxamide 4-[2,5-bis(trifluoromethyl)anilino]-6-oxo-1H-pyrimidine-5-carbonitrile 4-[2-(furan-3-yl)phenyl]-3,8a-dihydroquinoxaline 2-(1H-indol-4-ylsulfonyl)cyclohexan-1-one 1-[6-(3,4-dimethoxyphenyl)pyrimidine-4-carbonyl]piperidine-2-carboxylic acid (2S)-3-[4-(3,6-dioxocyclohexa-1,4-dien-1-yl)phenyl]-2-[[2,5-bis(trifluoromethyl)benzoyl]amino]propanoic acid 4-[3-(1H-indazol-4-yl)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile 6-[(3S,5R)-2,7-diazaspiro[4.4]nonan-7-yl]-N-pyridin-3-ylpyrazine-2-carboxamide;dihydrochloride 2-chloro-N,4-dimethyl-6-oxo-1H-pyrimidine-5-carboxamide 1-[(4-chloro-2,5-dimethylpyrazol-3-yl)methyl]-3-cyclopropylpyrrolidine;formic acid 2-(N-acetylanilino)-2,4-dimethylpentanoic acid (3R,4S)-1-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzoyl]-N'-(3-hydroxypropylsulfonyl)-4-methoxypyrrolidine-3-carbohydrazide 2-(1H-indol-3-yl)-N-methylsulfonyl-3-oxopentanamide 4-[1-azido-2,3-bis(4-methylphenyl)propan-2-yl]pyridine 2-[4-(2,3-dihydroxypropylsulfanyl)phenyl]acetaldehyde 1-(2,4-difluorophenyl)sulfonyl-3-[5-fluoro-1,8-dimethyl-2-(trifluoromethyl)-3H-imidazo[1,2-a]pyridin-6-ylidene]urea 6-[6-chloro-1-(oxan-2-yl)indazol-3-yl]imidazo[1,5-a]pyridine 2-(1,4-diazepin-1-yl)benzenesulfonamide (3S)-3-[5-chloro-2-ethyl-4-[(Z)-2-pyridin-3-ylethenyl]phenyl]-1-methylpyrrolidine 3-ethyl-2,4-dimethoxyquinoline 1-[2-methoxy-3,4-di(propan-2-yl)phenyl]ethylidenehydrazine (2Z)-3,4-dimethyl-1-phenyl-4H-[1]benzoxepino[5,4-c]pyrrole 4-[2-amino-6-[3-(diethylamino)propoxy]pyridin-4-yl]oxy-N,3,5-trimethoxybenzamide 3-(4,5-dihydro-1H-imidazol-2-yl)-N-[[6-methoxy-1-[(Z)-prop-1-enyl]benzimidazol-2-yl]methyl]but-3-enamide 1-[4,5-bis(4-bromophenyl)-1H-imidazol-2-yl]propan-2-amine 2-N,6-N-bis[4-(diethylamino)phenyl]pyridine-2,6-dicarboxamide 4-(N'-ethylcarbamimidoyl)-2-fluorobenzoic acid 1-benzyl-4-[(4Z,6E)-5-methylidenedeca-2,6,8-trien-3-yl]piperazine 6-chloro-5-(2,4-difluorophenyl)sulfanyl-3-(1H-indol-7-ylmethyl)pyrimidin-4-one [2-(4,6-diphenyl-1,3,5-triazin-2-yl)-9H-fluoren-1-yl]boronic acid [[2-(4,4-diphenylbutoxymethyl)benzoyl]-methylamino]carbamodithioic acid 2-chloro-4,6-bis(3,5-dimethylpyrazol-1-yl)-5-[2-(1,3,5-triazin-2-yl)propan-2-yl]pyrimidine 7-(2,5-dimethylphenyl)-1H-pyrazolo[3,4-c]quinoline 2-[3,5-dimethyl-4-(1H-pyrrole-3-carbonylamino)pyrazol-1-yl]acetic acid (5Z)-2-(4-ethylphenyl)imino-5-[(3-iodonaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one (2S)-4-[3,5-bis(trifluoromethyl)benzoyl]-1,4-diazepane-2-carboxylic acid 2-(cyclopentylsulfanylamino)-N'-hydroxypyridine-4-carboximidamide 7-[(1S)-1-azidoethyl]-2-chlorothieno[3,2-b]pyridine N-[2-[4-hydroxy-3,5-di(propan-2-yl)phenyl]-1H-imidazol-5-yl]acetamide 1-azido-4-phenylpiperidine 6-[(E)-3-[4,5-bis(ethylsulfonyl)thiophen-2-yl]prop-1-enyl]pyridine-3-carbonitrile 4-[2,6-diethyl-5-(2-methylpropyl)pyrimidin-4-yl]butanoic acid N-[1-(2-hydroxy-1H-indol-3-yl)ethylideneamino]-4,5,6,7,8,9-hexahydro-1H-cycloocta[b]pyrrole-2-carboxamide 1-(4-chloro-3-methoxyphenyl)pentan-2-one 4-[3,5-dichloro-2-(hydroxymethyl)phenyl]butanenitrile N-(1,3-thiazol-2-yl)-4-[6-(trifluoromethoxy)-1H-benzimidazol-2-yl]benzenesulfonamide 1-[[2,6-di(propan-2-yl)phenyl]methylideneamino]naphthalen-2-ol 2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)-N-(1H-pyrrol-2-ylmethylideneamino)benzamide 2-(3,5-dichlorophenyl)-1-[4-(methylamino)piperidin-1-yl]ethanone 2-(N-ethylsulfonyl-2,4,6-trimethylanilino)octanoic acid 1-[3-azido-2,6-di(propan-2-yl)phenyl]imidazole 7-[(2-bromophenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 2-methylsulfinyl-N-(6H-pyrrolo[3,4-c]pyrazol-1-yl)acetamide 2-bromo-N-(4,5-dimethyl-1,3-thiazol-2-yl)-6-fluorobenzamide 1-[1-[2,6-dichloro-4-(3,5-dimethylpyrazol-1-yl)benzoyl]piperidin-4-yl]-N-pyridin-3-ylpiperidine-4-carboxamide 1-[(5E,7Z)-4-methylcyclodeca-2,5,7-trien-1-yl]naphthalene 1-[2-(cyclopropylmethylamino)ethyl]-6,7-difluoro-3-[[1-(hydroxymethyl)cyclobutyl]methoxyimino]quinazolin-4-one 3-[1-(4,5-dimethoxy-2-propylphenyl)-3,6-dihydro-2H-pyridin-4-yl]-8-fluoro-7-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-c]pyrimidine 1,3-dimethyl-N-[4-(2-methylphenyl)cyclohexa-1,5-dien-1-yl]-6H-cyclohepta[c]pyrazole-5-carboxamide 7-methyl-2-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine 2-(3,4-dimethylphenyl)-N-[1-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylsulfanyl)ethyl]piperidin-4-yl]acetamide ethane;7-[5-(6-methylpyridin-2-yl)oxypyrimidin-4-yl]-3,9a-dihydrofuro[3,2-c]pyridine 4-cyclohexa-2,4-dien-1-yl-N-[4-(trifluoromethoxy)phenyl]piperazine-1-carboxamide [3-[2-fluoro-4-(hydroxymethyl)phenyl]piperidin-1-yl]-phenylmethanone 4-[3,5-bis(trifluoromethyl)phenyl]sulfanylmorpholine 4-[7-ethyl-1,6-dimethoxy-3-(2-piperidin-2-ylethenyl)naphthalen-2-yl]-N-[2-(1,3-oxazol-5-yl)phenyl]pyrimidin-2-amine N-benzylsulfonyl-1,3-benzodioxol-5-carboxamide (1R)-3-[(2S,5R)-2-methyl-6-[4-(1H-pyrazol-4-ylamino)pyrimidin-2-yl]-3,4,5-triphenylcyclohexa-1,5-dien-1-yl]oxycyclohexane-1-carboxylic acid N-[1-[1-(2,3-dihydroindole-1-carbonyl)cyclopropyl]ethyl]benzenesulfonamide N-[(3R,4S)-1-azido-4-[4-(6-methylquinolin-5-yl)phenyl]pyrrolidin-3-yl]propane-2-sulfonamide 4-[(6R)-7-amino-2-chloro-3,6,8,9-tetrahydrofuro[2,3-e]indole-5-carbonyl]-N'-ethylpiperazine-1-carboximidamide;dihydrochloride [3-fluoro-2-(1H-indol-4-yl)phenyl]methanamine 4-[(3R,5S)-3-amino-5-methylpiperidin-1-yl]-N-methoxy-N-propan-2-ylpyridine-3-carboxamide (5R)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-N-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 1-[5-chloro-2-(3-methoxypropylsulfonyl)phenyl]-4-hydroxy-6,7-dihydro-5H-pyrazolo[4,3-c]pyridine (4-chlorophenyl)methylsulfanium;ethane N-methyl-N'-(2,3,4,5-tetrafluorophenyl)pyrrolidine-1-carboximidamide 1-(2-azidosulfanylpyridin-4-yl)benzimidazole 5-[1-(dimethylamino)propan-2-yl]-3H-1,3,4-thiadiazol-2-one [5-amino-1-(4-bromophenyl)pyrazol-3-yl]-(2,6-difluorophenyl)methanone 3-[4-fluoro-2-(hydroxymethyl)anilino]sulfanylbenzaldehyde (2R)-1-[3-ethylsulfonyl-5-[4-(trifluoromethoxy)phenyl]pyridine-2-carbonyl]-N-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidine-2-carboxamide [4-[5-(2-bromophenyl)-1H-pyrazole-3-carbonyl]piperazin-1-yl]-phenylmethanone 1-[2,6-di(propan-2-yl)phenyl]-3-[[4-[5-isocyano-2-[(2S)-1,1,1-trifluoropropan-2-yl]oxypyridin-4-yl]phenyl]methyl]urea 2-methyl-3-[4-(pyridine-4-carbonylamino)phenyl]sulfonylpropanoic acid 2-benzylsulfanyl-N'-(4,6-dimethylpyrimidin-5-yl)ethanimidamide 3-[4-[(4-chloro-5,6-dihydro-1H-pyrrolo[2,3-b]pyridine-7-carbonyl)amino]pyrazol-1-yl]propanoic acid N-[(4-bromophenyl)methyl]spiro[1,4-dihydroquinoline-3,4'-piperidine]-2-imine 2-[(E)-3-(1H-benzimidazol-4-yloxy)prop-1-enyl]phenol [3-(4-azidophenyl)pyrrolidin-1-yl]-methylborinic acid 1,2-diamino-4-[3-(aminomethyl)phenyl]-6-oxopyridine-3,5-dicarbonitrile 1-[(E)-5-methylhex-2-en-3-yl]pyrene 6-[(5Z)-5-[(3,4-difluorophenyl)methylidene]furan-2-yl]-N-(pyridin-3-ylmethyl)pyridazine-3-carboxamide [4-[2,3-dihydroxypropyl(ethenylsulfonyl)amino]phenyl]sulfonylurea N-(cyclohexylmethyl)-6-oxo-4,5,7,8-tetrahydropyrazolo[1,5-a][1,3]diazepine-2-carboxamide 2-[4,6-bis(dimethylamino)pyrimidin-1-ium-2-yl]oxyethanol;bromide N-[2,5-difluoro-4-(2-fluoro-5-phenylanilino)phenyl]sulfanylcyclopropanesulfinamide 2-azidosulfanyl-4-(2,5-difluorophenyl)-1,3-thiazole 4-(3,5-dichlorophenyl)-1H-pyrimidine-2,4-diamine 1-(3,4-difluorophenyl)-5-hydroxy-2,6-bis[2-(4-nitrophenoxy)ethyl]-N',1-dioxo-1,2,6-thiadiazinane-3-carbohydrazide 4-[4-(dimethylamino)-N-hexadecylanilino]benzenesulfonic acid 2-amino-1-[(4S)-3-cyclopropyl-4-methoxypyrrolidin-1-yl]-4-methyl-1,4-dihydrothieno[3,2-d]pyrimidine-6-carboxylic acid 1-[3-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]ethanone 2-[[6-(chloromethyl)-1,3-benzothiazol-2-yl]amino]acetic acid 1-[4-(1,3,5-triazin-2-yl)phenyl]propane-2,3-dione N-[(E)-butylideneamino]-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxamide 3-[[5-chloro-6-(2,2,2-trifluoroethoxy)pyridine-3-carbonyl]amino]cyclobutane-1-carboxylate 5-[2,6-dichloro-4-(2-phenoxyethoxy)phenyl]imidazolidine-2,4-dione 3-[2-(6-carboxy-4,5-dimethyl-1H-benzimidazol-2-yl)butyl]benzoic acid 6-methoxy-2,5-diphenyl-1H-pyrimidine-4-thione 5-(1H-pyrazol-5-yl)-2-[4-(3-pyrrolidin-1-ylpropoxy)anilino]thiophene-3-carboxamide 1-[(2S)-3-(4-chlorophenoxy)-2-methylpropanoyl]piperidine-4-carboxamide 5-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-[2-(2-fluorophenyl)ethyl]-1H-indole-3-carboxamide ethane;2-methylpropanoic acid;5-phenyl-3H-1,4-benzodiazepine 2-[(3Z,5E)-3,6-bis(methylsulfanyl)hexa-1,3,5-trien-4-yl]oxy-3H-pyrido[3,4-d]pyrimidin-4-one [3-(difluoromethoxy)phenyl]-[7-hydroxy-3,5-bis(trifluoromethyl)-1H-indol-2-yl]methanone 1-azidosulfanyl-4-chloro-2-fluorobenzene (Z)-2-[amino-[4-(dimethylamino)phenyl]methyl]-3-[2,5-difluoro-N-formyl-6-(trifluoromethoxy)anilino]-N'-[1-(3-methanimidoylphenyl)ethyl]prop-2-enimidamide 2-bromo-4-phenylbenzoic acid;hydrate 2-[(4-methoxyphenyl)methyl]-6-methyl-4-[5-(trifluoromethyl)pyridin-2-yl]morpholine 3-[2,4-dimethyl-5-(trifluoromethyl)phenyl]imino-5-morpholin-4-ylpentan-1-ol 5-(1,3-benzodioxol-5-yl)penta-2,4-diynal 2-[1-carboxyethyl-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)amino]octanoic acid 4-[2,2-dimethoxyethyl(1,3-thiazol-5-yl)amino]benzenesulfonamide 5-methyl-4,6-diphenyl-1,2-dihydropyridazine 3-chloro-4-[4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]aniline 1-(5-fluoro-2,3-dihydroindol-1-yl)-4-[3-fluoro-5-(trifluoromethyl)phenyl]butan-1-one 4-methyl-2-(3-phenylphenyl)-6H-pyrazolo[1,5-a][1,3,5]triazin-7-one N-[3,5-bis(trifluoromethyl)phenyl]-2-methoxy-4-oxobutanamide 1-[2-(1,3-benzodioxol-5-yloxy)ethyl]-N'-hydroxyimidazole-2-carboximidamide 7-chloro-2,3,4,5-tetrahydro-1H-pyrido[3,2-b]indole 3-[4-[(3R,5S)-3,5-dimethylmorpholine-4-carbonyl]phenyl]propanenitrile 4-[2,3-dichloro-4-(4-chlorophenyl)phenoxy]butanoic acid (NE)-N-[amino(thiophen-3-yl)methylidene]-4-oxopyrrolidine-2-carboxamide 4-[(2S)-1-azidopropan-2-yl]-5-bromo-N'-hydroxypyridine-2-carboximidamide 3-amino-2,4-dichloro-6-(trifluoromethoxy)benzenethiol 3-chloro-N-[4-(dimethylamino)phenyl]-5-fluoro-2,6-dioxopiperidine-1-carboxamide N-azido-2,5-bis(trifluoromethyl)benzenesulfonamide 1-N-(3,4-dimethoxyphenyl)sulfanyl-2-N-piperidin-1-ium-1-ylpropane-1,2-diimine N-[(6R)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl]cyclopropanecarboxamide N-[5-[2-(4-azidophenoxy)ethyl]-1,3-thiazol-2-yl]-6-bromo-1H-indole-2-carboxamide [2-(dimethylamino)-4-[1-[4-(3,5-diphenylpyrazol-1-yl)benzoyl]azetidin-3-yl]oxybutylidene]oxidanium 2-[4-(4-methylpiperazin-1-yl)phenyl]ethanimidamide 2-[(3,5-dimethylphenoxy)methyl]-7-fluoro-1H-imidazo[4,5-b]pyridine 2-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylcarbamoylsulfamoyl)butanamide 3-(2,5-dichlorophenyl)-4-propyl-2H-pyrazolo[3,4-b]pyridine N-[1-amino-3,3-dimethyl-4-(2-oxa-8-azatricyclo[7.5.0.03,7]tetradeca-1(9),10,12-trien-13-yl)butylidene]-4-pyridin-3-ylsulfonylpiperazine-1-carboxamide (2E,4Z)-2-[2-[4-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]oxypiperidine-1-carbonyl]phenoxy]hepta-2,4,6-trienamide (6S,9R)-2-butylsulfanyl-6-methyl-9-pyridin-3-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one N-[(4E,5Z)-2-[1-(1H-imidazol-5-ylmethylidene)indol-1-ium-3-yl]-6-methoxy-1-oxohexa-4,5-dien-3-yl]-1-oxidoazepane-4-carboxamide 4-[6-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]pyrimidin-4-yl]oxynaphthalene-1-carboxamide [(1S)-5-benzylsulfanyl-4,6-difluoro-2,3-dihydro-1H-inden-1-yl]carbamic acid 5-[(4,6-dichloropyrimidin-2-yl)amino]thiophene-3-carboxylate N-(1-cyclohexylethenyl)-5-[3-(4-pyridin-2-yl-1H-indol-2-yl)-1H-indazol-5-yl]pyridin-3-amine 3-[[3-(4-butoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]chromene-2,4-dione 4-[(3,5-difluorophenyl)methylamino]-2-propan-2-yl-1H-pyrimidin-6-one (2R)-N'-[1-[5-fluoro-2-hydroxy-4-(triazol-1-ylmethyl)phenyl]ethylideneamino]butanediamide 2-(1,3-benzothiazol-5-ylmethyl)-5-chloro-3H-isoindol-1-one 5-amino-2,7,9,11,13-pentazatricyclo[8.4.0.03,7]tetradeca-1(10),3,5,11,14-pentaen-6-one;hydrochloride 1-[(2R,3S)-6,8-difluoro-11-hydroxy-2-methyl-9-oxa-1,12-diazatricyclo[8.4.0.03,7]tetradeca-10,13-diene-13-carbonyl]piperidine-4-carbonitrile 6-(2,4-dimethylpiperazin-1-yl)-N'-hydroxypyridine-2-carboximidamide ethane;4-(2-methylphenyl)-1,3-bis[(2E)-penta-2,4-dien-2-yl]-5-propan-2-ylidenepyrazole N-[(1S)-2-ethoxy-1-[4-fluoro-3-(4-methylphenyl)phenyl]ethyl]-3,5-diethyl-4-methoxybenzamide 2-methyliodanuidylbenzo[de]isoquinoline N-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]-3,4-bis(trifluoromethoxy)benzamide [2-(3,4-dimethoxyphenyl)cyclopropyl]-spiro[2H-furo[3,2-b]pyridine-5,3'-pyrrolidine]-1'-ylmethanone 1-methyl-5-(pyrrolidine-1-carbonyl)pyrido[2,3-d]pyrimidine-4,7-dione N-[3,5-dichloro-4-(2-methylsulfanylphenoxy)phenyl]hydroxylamine [2-(4-amino-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carbonyl)pyridin-4-yl]methylcarbamic acid 2-(2,4-dichlorophenyl)-3-methylquinoline (2S)-2-[1-hydroxy-4,5-dimethoxy-3-phenyl-2-(trifluoromethyl)pyridin-1-ium-4-carbonyl]pyrrolidine-1-carboxylate 5-fluoro-3,4,6-triphenylpyridazine (5E)-1-(4-chlorophenyl)-2,6-dimethylhepta-2,5-diene-3,7-dione 2-[4,5-bis(trifluoromethyl)pyrazol-1-yl]pyridine 5-benzyl-2,4-dimethoxy-6-[(2R)-1-phenylpropan-2-yl]pyrimidine [1-(1,4-dimethylpiperidine-4-carbonyl)pyrrolidin-3-yl]-[2-(triazol-1-yl)phenyl]methanone N-(4,4-dimethylcyclohexyl)-5-methanimidoyl-2-N-[(1-prop-2-enoylpiperidin-3-yl)methoxy]pyrimidine-2,4-diamine N-(2,4-dimethylphenyl)-3,5-difluoro-6-iodo-2H-pyrimidin-1-amine 2-(3,5-dimethylphenyl)-2-(6-fluoroimidazo[1,2-a]pyridine-2-carbonyl)pentanedioic acid 2-[(1-cyclopropylsulfonylpiperidin-4-yl)amino]-4,5-dimethylthiophene-3-carbonitrile 2-(aminomethyl)-5,6-dichloro-1,3,4-triphenylcyclohexa-2,4-dien-1-ol 2-[1-(2,6-dimethylphenyl)ethenylimino]propanedioic acid 3-[(4R)-7,8-dimethoxy-2,10b-dimethyl-6,11-dihydro-5H-imidazo[2,1-a]isoquinolin-4-yl]phenol N-(2,6-dimethylphenyl)-1-[5-[[2-fluoro-4-(2H-tetrazol-5-yl)benzoyl]amino]pyridine-3-carbonyl]piperidine-2-carboxamide 4-chloro-6-(3-methoxyphenyl)-2H-isoindole 6-chloro-1-methyl-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-7-one 1-(3,4-dimethoxyphenyl)hexane-2-sulfonamide (4R)-1-tert-butyl-4-methyliodanuidyl-3,4,5,6-tetrahydro-2H-quinoline 4-[(E)-2-(5,6-dimethoxypyridin-3-yl)ethenyl]-N'-ethyl-N-methylidenebenzenecarboximidamide;methane 2-[4-(dimethylamino)phenoxy]-5-[2-(3-fluorophenyl)ethyl]pyridine-3-carboxamide;hydrochloride 2-N-(3-azidopropyl)-2-N,6-N-dibenzyl-1H-indole-2,6-diamine N-[[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]methoxy]-3-(6-phenylquinolin-8-yl)benzamide 3-methoxy-5,5-diphenylpyrrolidine-2,4-dione 4-(7-azatricyclo[10.4.0.02,9]hexadeca-1(16),2,4,6,8,12,14-heptaen-11-ylamino)-N-[3-(dimethylcarbamoyl)phenyl]benzamide 1-azidooxy-2,4-dinitrobenzene N-[4-chloro-3-(trifluoromethyl)phenyl]sulfanyl-5-ethoxypentanamide 2-(4-methylphenyl)sulfanyloxyacetamide 6-[2,4-bis(trifluoromethyl)phenyl]-N-(2H-tetrazol-5-ylmethyl)pyridine-3-carboxamide 6-azido-5-fluoro-2,3-dimethoxyphenol N-[5-(1,4-dimethyl-6-oxopyridazin-3-yl)-2H-triazol-4-yl]benzenesulfonamide N-butylsulfanyl-5,6-difluoro-1H-indole-2-carboxamide 2-[4-ethoxycarbonyl-N-(3-methylbut-2-enyl)anilino]propanoic acid 2-(3,5-difluorophenyl)-1,3-benzothiazole N-(2,5-dioxopyrrolidin-1-yl)-1'-(pyridine-4-carbonyl)spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide (1S,3R)-3-[2-methyl-6-[1-methyl-5-[[[(1R)-1-thiophen-2-ylethyl]amino]methyl]triazol-4-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid N-(3,4-dihydro-2H-chromen-3-yl)-1-methoxy-2,2,6,6-tetramethylpiperidine-4-carboxamide 6-[3-(2,4-difluorophenyl)butanoyl]-N-(2-methoxyethyl)-N,1-dimethyl-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine-4-carboxamide (E)-3-[4-[(Z)-1-aminopent-2-enyl]phenyl]prop-2-enoic acid N-cyclohexyl-N-[2-(cyclopropylamino)-5-pyridin-3-ylphenyl]formamide 2,6-dichloro-N-[(2R)-1-hydroxypropan-2-yl]benzamide 1-azido-4,5-bis(chloromethyl)-2-nitrobenzene ethane;2-fluoro-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]diazenyl]phenol 2-(2,4-dimethylphenyl)-N-[5-(trifluoromethoxy)pyridin-3-yl]acetamide 3-chloro-6-methoxynaphtho[2,1-b][1]benzofuran (3-aminopyrrolidin-1-yl)-[5,6-bis(4-chlorophenyl)furo[2,3-d]pyrimidin-4-yl]methanone [4-chloro-3-(difluoromethyl)phenyl]-ethoxyphosphinate (3R)-N'-[amino-[2,2-dimethylpropanoyl(3-pyridin-4-ylpropyl)amino]methylidene]-1-[5-chloro-6-[3-(trifluoromethoxy)phenoxy]pyridin-3-yl]pyrrolidine-3-carboximidamide 4-chloro-5-(1,3-thiazol-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-6-amine;formamide 4-N,4-N-diethyl-2,6-bis(5-nitropyridin-2-yl)pyrimidine-4,5-diamine 2-[(3E)-3,5-diethylhexa-1,3,5-trien-2-yl]oxynaphthalene 2-(4-chlorophenyl)-N-[3,5-difluoro-4-(8-methoxyquinolin-7-yl)oxyphenyl]acetamide 2-[(E)-but-1-enyl]-5-ethylidene-7-methyl-3-propan-2-ylisoquinoline 1-[4-[2-[5-(1H-pyrrole-2-carbonyl)pyridin-3-yl]ethynyl]phenyl]cyclopropane-1-carboxylic acid (2S)-2-[9H-fluorene-1-carbonyl(methyl)amino]-3-phenylpropanoic acid 4-azidooxy-1,2-dimethylindole 3-[(1S)-2,2-dimethylcyclopentyl]benzaldehyde 2-[4-(1H-indazole-3-carbonyl)piperazin-1-yl]-N-propan-2-ylpyrimidine-5-carboxamide N-[1,2-diamino-4-(3,5-dihydroxyphenyl)-2,4-dioxobutyl]-2-methoxybenzamide (3R,4S)-1-[5-[6-amino-8-(ethylsulfanylmethoxy)purin-9-yl]oxolane-2-carbonyl]-4-fluoropyrrolidine-3-carboxamide (5-oxo-4H-tetrazolo[1,5-a]quinazolin-7-yl)methanesulfonamide 2-(N-(4-nitrobenzoyl)anilino)benzenesulfonic acid [3-(azidomethyl)-4,5-difluorophenyl]carbamic acid N-[[1-(3,4-difluorophenyl)pyrrolidin-3-yl]methyl]imidazo[1,2-b]pyridazine-6-carboxamide 4-[[2,6-difluoro-N-(3-methylbut-1-en-2-yl)anilino]methyl]-N'-hydroxybenzenecarboximidamide 5-[(3,4-dichlorophenoxy)methyl]-1H-tetrazolo[1,5-a]pyridine 5-[3,5-difluoro-4-(2H-triazolo[1,5-a]pyrimidin-6-yl)phenyl]-7-fluoropyrido[2,3-b]pyrazine N-[1-(4-methoxyphenyl)ethyl]-3-[[6-oxo-4-(trifluoromethyl)-1H-pyrimidin-2-yl]sulfanyl]propanamide 2-[4,7-bis(dimethylamino)chromen-4-yl]-1H-benzimidazole-5-carboxamide 2-(6,7,8-trimethoxyquinolin-4-yl)piperazine-1-carboxylate 2-[4-bromo-N-(1,3-thiazol-5-yl)anilino]acetic acid 2-[(E)-3-(5,6-dimethoxycyclohexa-1,3-dien-1-yl)prop-2-enoyl]benzenesulfinic acid 2-[3-(4-aminophenyl)propyl]decanedioic acid 1-[(Z)-2,3-difluorobut-2-enyl]-4-[(3R)-3-methylpent-1-ynyl]benzene 7-[(3,5-dimethylphenyl)methoxy]-8-methoxy-2-pyridin-3-ylchromen-4-one 1,3-diazidonaphthalene;hydrochloride (E)-2-cyano-3-[5,8-diethoxy-4-oxo-1,7-bis(phenylmethoxy)quinolin-6-yl]prop-2-enoic acid 5-[2-(3,4-difluorophenyl)pyridin-4-yl]oxy-3H-1,3-benzothiazol-2-one 7-[(1R,2S)-2-[[4-chloro-3-[4-(trifluoromethylsulfonyl)phenyl]phenyl]methoxy]cyclopentyl]heptanoic acid 2-[4-fluoro-6-[2-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-3-yl)ethynyl]pyridin-2-yl]ethanamine 2-cyclopropylimino-5-[(4,6-dimethoxypyrimidin-2-yl)methylidene]-1,3-thiazolidin-4-one 1-(2,4-dichlorophenyl)-5-methylsulfonylbenzo[g]indazole N-[1-(2,3-dihydro-1H-pyrrol-5-yl)ethylidene]-4-propan-2-ylaniline 1-bromo-2,3-diethynylbenzene;ethane N-(4,6-dimethoxypyrimidin-2-yl)-4-[2,4,7-tris(sulfanylidene)-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidin-5-yl]benzamide 3-fluoro-6-(4-propylcyclohexyl)-2-(trifluoromethoxy)phenol 2-(4-chlorophenyl)-3-methyl-1-[4-methyl-5-(trifluoromethylsulfanyl)thiophen-2-yl]sulfonylazetidine N-(4,5-dihydropyrimidin-2-yl)-1H-indole-6-sulfonamide 3-[5-azido-2,4-bis(phenylmethoxy)phenyl]sulfonylphenol N-[4-methyl-3-[(2E,4Z)-2-methylhexa-2,4-dienoyl]phenyl]pyridine-3-carboxamide (1S,2R)-N-[6-fluoro-5-(4-hydroxyphenyl)-3-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-fluorocyclopropane-1-carboxamide 5-(azidomethyl)-2,3,4,6-tetrabromopyridine [1-[2,4-bis(trifluoromethyl)phenyl]pyrrolidin-3-ylidene]carbamic acid 4-[5-(3-aminoanilino)-2H-triazol-4-yl]-1,3-thiazole-2-carboxylic acid 4-[1-(2,6-difluorophenyl)ethyl]-N'-methanimidoylthieno[3,2-c]pyridine-7-carboximidamide [3-(1-aminoethyl)phenyl]-[4-(2,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methanone;dihydrochloride 4-[2-(1H-inden-5-yl)propan-2-yl]naphthalene 2-[3,4-bis(ethenyl)cyclohexa-1,5-dien-1-yl]-N-cyclohexa-1,3-dien-1-ylaniline;toluene 6-[2,5-difluoro-3-(pyrrolidine-1-carbonyl)phenyl]-4-hydroxy-1H-pyridin-2-one 2-[4-[2-(aminomethyl)-3-fluoroprop-2-enoxy]phenyl]-N'-ethylprop-2-enehydrazide 2-[[2,6-dichloro-4-(trifluoromethyl)phenyl]methylsulfanylamino]-3,3-diethylbutanal 1-[2-fluoro-5-(trifluoromethyl)phenyl]-N-methoxymethanamine 4-[2,3-dihydroxypropyl(1H-indole-5-carbonyl)amino]-2-hydroxybenzoic acid 1-[2,5-dimethyl-3-(methylideneamino)pyrrol-1-yl]-2-phenylethanone N-[3-methoxy-2,6-di(propan-2-yl)phenyl]-1H-benzimidazole-2-carboxamide 2-[(6S,9aS)-1-hydroxy-3,4,8,9a-tetrahydro-2H-indeno[1,2-b]pyridin-6-yl]ethanol 6-bromo-N-[(1S,3R)-3-methylcyclohexyl]pyridine-2-carboxamide (5S)-2-phenylimino-5-propan-2-yl-1,3-thiazolidin-4-one [5-(hydroxyamino)pyridine-3-carbonyl]azanium 1-cyclopropyl-3-[2-(5-methoxy-2,4-dioxopyrimidin-1-yl)ethyl]urea 6-[(2R)-2-ethylpiperazine-1-carbonyl]-3,4-dihydroisochromen-1-one [(4-fluorophenyl)methyl]-(4-methoxy-6,7-dihydropyrrolo[3,2-d]pyrimidin-5-ylidene)azanium 6-(4-hydroxyphenyl)-2,3,5-trimethoxyphenol 2-[4-(methylamino)cyclohexyl]oxy-4,6-diphenylbenzaldehyde 2-[(1S)-2-cyclohexyloxy-1,3-dihydroinden-1-yl]acetonitrile 5-amino-4-(3-chloro-2,6-difluorophenyl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione [1-[4-[(2E,5Z)-6-methylideneocta-2,5-dien-3-yl]oxyphenyl]pyrazol-4-yl]methanol 2-fluoro-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)acetamide (3E)-4-amino-3-[(2,5-difluoro-4-hydroxyphenyl)methylidene]azete-2-thione 1-[(2,3-dimethylphenyl)-(4-fluorophenyl)methyl]-3-(2-hydroxyethylamino)thiourea 2-amino-6,8-dibromoimidazo[1,2-a]pyridine-7-carboxylic acid 2-[(3S)-1-cyclohexylpyrrolidine-3-carbonyl]-6-methoxy-5-methyl-3,4-dihydro-1H-isoquinoline-8-carboxylic acid N-(4-chlorobutyl)-N-(4,5-dimethyl-2-phenyldiazenylphenyl)benzenesulfonamide N-(3-iodopropyl)-2,6-dimethoxybenzamide 2,7-dichloro-6-(6-fluoroimidazo[1,2-a]pyridin-2-yl)purine 4-[3-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-N-ethyl-5-methylpyrimidin-2-amine N-(4-methoxyphenyl)-2-methyl-N'-[5-[1-[4-(trifluoromethylsulfanyl)anilino]ethenyl]pyrazin-2-yl]propanediamide 2-amino-N-[5-(3,4-dimethoxyphenyl)sulfanylpyrimidin-1-ium-2-yl]acetamide 2-(6,7-dimethoxyquinolin-4-yl)oxyaniline N-benzyl-6-[3-(dimethylamino)propylamino]pyridine-2-carboxamide 3,5-dimethyl-1-[(2S)-3,4,7-trihydroxy-6-phenylmethoxyoctan-2-yl]pyrazole-4-carbonitrile 3-[4-[1-(cyclohexylamino)ethyl]piperidin-1-yl]aniline 4-[(2,3-dichlorophenyl)methylamino]-6-[1-[(Z)-ethylideneamino]ethenylsulfanyl]pyrimidin-5-ol N-[(1R,2S)-1-cyclobutyloxy-1-(3-methoxyphenyl)propan-2-yl]-6-oxo-1H-pyrimidine-4-carboxamide 2-[(5R)-3-chloro-5-cyano-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonyl]-4-[2-(2-pyrrolidin-1-ylethoxy)phenyl]benzamide 6-azidosulfanylhex-5-enylbenzene (2S)-1-[[6-azido-3,5-bis(trifluoromethyl)pyridin-2-yl]amino]propan-2-ol 7-[[4-chloro-2-(methoxymethyl)phenyl]methylamino]-1,3,6-trimethylpurine-2,8-dione (5Z)-2-(4,6-dimethylpyrimidin-2-yl)imino-5-[[3-fluoro-2-hydroxy-5-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidin-4-one 4-[[5-chloro-4-(methylamino)pyrimidin-2-yl]amino]benzamide 2-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl)-5-propan-2-yloxyaniline;methanamine 2-[4-(2,5-dimethylpyrrolidine-1-carbonyl)piperidin-1-yl]sulfonylbenzoic acid 7-[(E)-1,2-bis(benzenesulfonyl)but-1-enyl]-5,6-dihydro-3H-imidazo[4,5-b]pyridine 1-[6-[2-(3,4-dihydro-2H-pyrido[2,3-b]pyrazin-1-yl)ethyl]pyridazin-3-yl]pyrrolidin-2-one 2-[3,5-bis(trifluoromethyl)phenyl]sulfonylbenzenethiol 4-(2,6-dibromophenyl)-5-propan-2-yl-1H-pyrimidine-2,4-diamine 3-azido-N,5-ditert-butyl-4-(2-methylpropoxy)benzenesulfonamide N-[(2S)-4-amino-3,4-dioxo-1-phenylbutan-2-yl]-5-pyridin-2-ylpyrazole-1-carboxamide N-[2-(3-cyanoazetidin-1-yl)ethyl]-4-oxochromene-6-carboxamide 2-(difluoromethyl)-3,5-bis[4-(trideuteriomethoxy)phenyl]pyrazine 4-[(2R,5R)-5-azidopyrrolidin-2-yl]oxyaniline (3S)-4-methyl-3,5-diphenylfuran N'-hydroxy-4-[2-methoxyethyl(1-sulfanylpropan-2-yl)amino]pyridine-2-carboximidamide 3-[2-(ethylamino)-5-methylphenyl]thiophene-2-carboxylic acid 6-[(2S)-4-aminobutan-2-yl]oxypyridine-3-carboxylic acid 5-chloro-2,6-dimethyl-N-(3,4,5-trifluorophenyl)pyridine-3-carboxamide 4-methyl-6-(3-methylphenyl)benzene-1,2,3,5-tetrol (3S,4R)-4-phenyl-1-[2-[4-(trifluoromethyl)anilino]pyrimidin-5-yl]pyrrolidine-3-carboxylic acid 3-azidosulfanyl-5,6-dichloroimidazo[4,5-b]pyridine 2-[(6-nitro-1,3-benzothiazol-2-yl)-propylamino]acetic acid 5-[2-(4,6-dimethoxycyclohexa-1,3-dien-1-yl)ethynyl]-4-N-(4-morpholin-4-ylphenyl)pyrimidine-2,4-diamine 4-[1-(oxan-2-yl)indazol-5-yl]sulfonylmorpholine 7-(3,4-dimethoxyphenyl)-N-hydroxyheptanamide 1-[4-(3,5-ditert-butyl-4-methoxyphenyl)piperazin-1-yl]prop-2-en-1-one N'-hydroxy-4,5-dimethylnaphthalene-2-carboximidamide 1-(benzenesulfonyl)-7,8-diethoxy-3H-imidazo[4,5-c]quinolin-2-one 1-(4,5-dimethylcyclohexa-2,4-dien-1-ylidene)-3-(4-ethoxyphenyl)urea 2-methyl-5,6,8,9-tetrahydrocyclohepta[b]indole [(Z)-3-amino-1-[2-(5,6-dimethyl-1H-benzimidazol-2-yl)quinolin-7-yl]prop-2-enylidene]azanium 3,4-dimethyl-2-phenyl-5H-1,4-benzothiazepine ethane;4-[2-fluoro-5-(trifluoromethyl)phenyl]-2,6-dipyridin-3-ylpyridine N-[(1R)-2,3-dihydro-1H-inden-1-yl]propanamide 1-azido-3-benzyl-4,5-dimethylimidazole-2-thione 3,5-dichloro-N-methyl-4-(2-phenylethenyl)aniline (3Z)-5,7-dichloro-6-methyl-2-phenylmethoxyhepta-1,3,5-triene;ethane (Z)-3-(2,5-dimethoxyphenyl)-N'-[1-(methylamino)ethenyl]but-2-enimidamide N-[2-(6,7-dimethoxyquinolin-4-yl)-3H-benzimidazol-5-yl]-2,2,4-trimethylpentanamide [2-fluoro-4-[5-(trifluoromethyl)pyrimidin-2-yl]oxyphenyl]-[3-methyl-4-[(pyridin-2-ylamino)methyl]piperazin-1-yl]methanone N-[(1E,3Z)-2-butan-2-ylidenecyclopentyl]-7-methoxyquinoxaline-6-carboxamide 4-[2,3-dihydroxypropyl(1,3-thiazol-5-yl)amino]benzenesulfonic acid 2,5-bis(6-methylpyridin-3-yl)quinoline 2-[(3E)-hexa-1,3,5-trien-3-yl]-5-phenylcyclohepta-1,4,6-triene (3aR,7aR)-1-[2-methyl-5-(1-methyltriazol-4-yl)benzoyl]-3,3a,4,6,7,7a-hexahydro-2H-pyrrolo[3,2-b]pyridin-5-one 3-[1-[(E)-but-2-en-2-yl]sulfanylethenyl]-N,N'-dipropylbenzenecarboximidamide 2-amino-6-[3-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]oxyphenyl]pyridine-3-carbonitrile 3-methyl-4-[6-(6,8,10-triazatetracyclo[7.6.0.02,7.011,15]pentadeca-1(9),2,4,5,7,11(15)-hexaen-13-yl)imidazo[1,2-a]pyridin-2-yl]morpholine 2-(4,4,5,5,6,7,7,8,8,9,10,11,12,12,14,15,16,17-hexadecafluorooctoxy)benzenesulfonic acid N-(2,4-dinitrophenyl)-3-pyridin-1-ium-4-yl-5H-pyrrolo[3,2-c]pyridine-7-carboxamide 2-[2-fluoro-5-(trifluoromethyl)phenyl]sulfanyl-N'-hydroxypyrimidine-4-carboximidamide (E)-3-[4-fluoro-2-methyl-6-(1,5-naphthyridin-8-ylamino)phenyl]-N-hydroxyprop-2-enamide N-(furan-2-ylmethyl)-7-[4-(1,3-thiazole-5-carbonylamino)benzoyl]-3,8a-dihydroindolizine-1-carboxamide 1-[(3-chloro-2,5-dimethoxyphenyl)sulfanylamino]-3-cyclopropylazetidin-2-one 4-methyl-2,3-di(propan-2-yl)quinoline 3-[2,4-dimethyl-5-(3,3,6-trimethyl-1H-indene-2-carbonyl)phenyl]propanoic acid 6-bromo-8-ethyl-2-(furan-3-yl)chromen-4-one 4-bromo-1-[(4-methoxyphenyl)sulfonylamino]indole-7-carboxamide (4Z)-3,5,7-trimethyl-2-[1-[2-[methyl-(1-phenylpiperidin-3-ylidene)amino]oxyethylamino]ethenyl]hepta-4,6-dienal 3-[2,4-dichloro-N-(2-methylpropanoyl)anilino]butanoic acid 5-[4-amino-2,6-dichloro-3-(4-fluorophenyl)quinoline-7-carbonyl]-3-fluorocyclohexa-1,3-diene-1-sulfonamide 3-[5-(1,4-diazepane-1-carboximidoyl)thiophen-2-yl]benzoic acid 3-(4-nitrophenyl)sulfonyl-3-azaspiro[5.5]undecane 6-[(1R)-4-[(3S,5S)-3,5-dimethylpiperazin-1-yl]cyclohexa-2,4-dien-1-yl]oxy-N'-hydrazinylidenepyridine-2-carboximidamide 4-[(E)-1-(1,3-benzodioxol-5-yloxy)but-2-en-2-yl]pyridine [2-(3,4-dichlorophenyl)quinolin-4-yl]-(1-methylpyrrol-3-yl)methanone N'-(2,4-dioxo-1H-pyrimidin-5-yl)-N,N-bis(pyridin-3-ylmethylideneamino)ethanimidamide 2-[[(3,5-dibromophenyl)methyl-methylcarbamothioyl]amino]-N-phenylacetamide 1-[(3S)-1-[4-[2-amino-5-(trifluoromethyl)benzimidazol-1-yl]phenyl]pyrrolidin-3-yl]ethanone N-[(2E,4Z)-6-(2-chloro-5-fluorophenyl)-1-hydroxyhepta-2,4,6-trienylidene]-3-methylbutanamide N-[1,4]benzodioxino[2,3-f]quinazoline-9-carboxamide N-(2,6-dichlorophenyl)-5-[3-[(3Z)-hexa-1,3,5-trienyl]sulfanylcyclobutyl]pentanethioamide 2,6-dibromo-4-[(Z)-hydroxyiminomethyl]phenol N-(5-methoxycyclohepta-1,3,6-trien-1-yl)propanamide;2-[2-(3,4,5-trihydroxyphenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]acetaldehyde 2-[4-[(5-cyclopropyl-1,2-oxazol-3-yl)methoxy]phenyl]ethanamine 1-(4,6-dimethylpyrimidin-2-yl)oxy-3-[3-[2-(trifluoromethoxy)phenyl]imidazolidin-1-ium-1-yl]propan-2-ol 2-[(2,6-dichlorobenzoyl)amino]oxypentanoic acid 2-(ethylamino)-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one;hydrochloride 5-[(1S)-1-azidoethyl]-3,4-difluorobenzene-1,2-diol 4-methylbenzenesulfonate;1,2,3,4,5-pentafluorobenzene-6-ide;tungsten(4+) 1-(2,5-dimethylphenyl)piperazine;ethene 2-[(Z)-1,3-diphenylprop-2-enylideneamino]guanidine 2-[(5R)-2-(methoxymethyl)-7-oxo-1,4-diazepan-1-ium-1-ylidene]acetaldehyde;trifluoromethanesulfonate 1-[4-(dimethylamino)phenyl]sulfonylpyrrolidine-2,5-dione N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-5-nitrofuran-2-carboxamide 4-methyl-2-[4-(5,6,7,8-tetrahydroquinazolin-2-ylsulfanyl)butoxy]-1H-pyrimidin-6-one N-cyclopropylsulfonyl-1'-(3,5-dimethoxybenzoyl)spiro[4,7-dihydropyrano[4,3-c]pyrazole-6,4'-piperidine]-2-carboxamide (4S)-1-(5-chloro-1,3-benzothiazol-2-yl)-3-methyl-4-thiophen-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 5-chloro-2,3,4,6-tetradeuterio-N-(1H-pyrrolo[2,3-b]pyridin-3-ylmethylideneamino)benzamide 1-[2,4-bis(2-hydroxyethoxy)phenyl]-2-bromo-3-phenylpropan-1-one N-[4-(cyclohexa-1,3-dien-5-yn-1-ylmethoxy)phenyl]-1,2-oxazole-5-carboxamide N-[(E)-1H-indol-3-ylmethylideneamino]-2,4-dinitroaniline 5-ethyl-N'-(3-methylphenyl)pyrrolidine-2-carboximidamide;dihydrochloride N-(2,4-dinitrophenyl)-N-propylbenzenesulfonamide N-[(4S)-1,2,3,4,5,6-hexahydroacridin-9-yl]thiophene-2-carboxamide 6-[(4R)-3,3-difluoropiperidin-4-yl]oxyisoquinoline 6-[1-(cyclopropylmethyl)pyrazol-4-yl]-N-(piperidin-3-ylmethyl)quinoxaline-2-carboxamide 2-[1-(4-hydroxybenzoyl)-5-oxopyrrolidin-3-yl]isoindole-1,3-dione 4-[[(2S,3R)-3-hydroxypiperidine-2-carbonyl]amino]benzoic acid N-[3-(benzenesulfonyl)phenyl]sulfonyl-6-methylpyridine-2-carboxamide 4-[[1-(2,6-dichlorophenyl)pyrrolidin-3-yl]methylamino]-N-methylpyridine-3-carboxamide 1-azidooxy-2-phenylnaphthalene (2R)-1-[4-amino-3-chloro-5-fluoro-6-[4-(trifluoromethylsulfonyl)piperazine-1-carbonyl]pyridin-2-yl]-N-[4-cyano-3-(trifluoromethyl)phenyl]-N,1-dimethylpyrrolidine-2-carboxamide 2-[4,5-bis(4-methoxyphenyl)-1H-imidazol-3-ium-3-yl]phenol 4-[3-chloropropyl(propyl)amino]benzenesulfonic acid 3-[5-(2,6-difluorophenyl)sulfonyl-1H-pyrazol-4-yl]-1-methoxyazetidine 7-cyclopentyl-2-(4-fluorophenyl)-6-oxo-N-pyridin-3-yl-5H-furo[3,4-b]pyridine-3-carboxamide 5-(2,3-dihydro-1H-isoindole-4-carbonyl)-N-methylthiophene-3-sulfonamide 4-[(2S)-1-[(3R,5R)-3,4-dihydroxy-5-(6-methylpyrazin-2-yl)oxolan-2-yl]-3-oxobutan-2-yl]benzonitrile ethane;2-(3-fluorophenyl)-5-[4-[(1-hydroxycyclobutyl)methoxy]-3,5-dimethylphenyl]pyridine-4-carboxylic acid 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[N'-hydroxy-N-[(4-methoxyphenyl)methyl]carbamimidoyl]urea N-methyl-2-oxo-3,4-dihydrochromene-5-carboxamide 3-[3-fluoro-5-(2-piperidin-1-ylethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 6-(4-but-3-enylphenyl)-1,2,3-trifluoronaphthalene 4-azido-5-methyl-N-[2,2,2-trifluoro-1-(3-methoxyphenyl)ethyl]pyrimidin-2-amine 1-(2,3-dimethoxyphenyl)sulfonyl-N-[4-(1H-pyrazol-5-yl)phenyl]azetidine-2-carboxamide 2-chloro-4,5-difluoro-3-pyridin-2-ylbenzamide [3-(2,6-difluorophenoxy)phenyl]methylcarbamic acid N-(2,6-dichloro-4-nitrophenyl)-N-(1,3-thiazol-5-yl)acetamide 2,5-ditert-butyl-4-(5-ethoxypyridin-3-yl)-6-methylpyrimidine 3-(4,6-dimethoxypyrimidin-2-yl)azetidine-1-carboxylic acid 3,4-dichloro-N-[(2R)-1-cyclopentyloxy-3-phenylpropan-2-yl]benzamide 4-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[[2-methyl-4-[6-(trifluoromethoxy)pyridin-2-yl]phenyl]methyl]aniline 6-(7,8-dihydronaphthalen-1-yl)-3-[4-(4-fluorophenoxy)phenyl]thieno[2,3-c]pyrrole 1-[4-chloro-3-(trifluoromethyl)phenyl]piperidine;N-[2,2-dimethoxyethyl(pyridin-4-ylmethyl)amino]formamide 2-methyl-N-[(4-methylphenyl)methoxy]-2,3-dihydro-1H-benzimidazole-5-carboxamide 5-chloro-4,8-dimethyl-3-pentylisoquinoline 1-[5-fluoro-2-(2H-thiopyran-6-yl)phenyl]pentan-3-one N-(1H-indol-3-ylmethylideneamino)-5-methoxyquinoline-8-carboxamide N-[(3R,4S)-1-benzyl-3-methoxypiperidin-4-yl]-5-chloropyridine-2-carboxamide 4-(2,5-dimethylpyrrol-1-yl)-N-[3-[6-[2-(trifluoromethoxy)anilino]pyridin-2-yl]oxolan-3-yl]benzamide 3,4-dichloro-2-methoxy-N-prop-1-en-2-ylaniline 5-(5,6-dimethoxypyridin-3-yl)-N-[4-fluoro-2-methoxy-7-(1H-pyrazol-4-yl)-1,3-benzothiazol-5-yl]-1,3-oxazole-2-carboxamide (3E,5Z)-hepta-1,3,5-triene;(6S,8R)-7-hydroxy-9,10-dioxo-N-[[4-(2,2,2-trifluoroethoxy)phenyl]methyl]-4-oxa-1,7-diazatricyclo[8.4.0.03,8]tetradeca-9,11,13-triene-12-carboxamide 2-(2,5-dimethylphenyl)-N-[[4-[1-(2-fluoroethylamino)ethenyl]phenyl]methyl]acetamide;methoxymethane N-[2-(1H-indol-3-yl)ethyl]-N-methyl-3,5-bis(trifluoromethyl)aniline 1-[2-azidooxy-5-(trifluoromethyl)phenyl]ethanone 3-(azidomethyl)-6,8,10-triazatetracyclo[7.5.0.02,7.011,13]tetradeca-1,4,6,9,11-pentaene N-[(2S)-1,4-dioxan-2-yl]-6-[(4-fluorophenyl)methoxy]pyridine-3-carboxamide N-[(3S)-4,4-dimethylpentan-3-yl]-1H-pyrrole-2-carboxamide;6-fluoro-2-morpholin-4-ylsulfonyl-3H-quinazolin-4-one (1E)-2,3-dimethylpentacyclo[b]naphthalene;ethane 2-methylsulfanyl-N-(1H-pyrazol-5-yl)acetamide N-[1-(5-ethylpyrimidin-2-yl)piperidin-4-ylidene]nitramide N-(6-cyanopyridazin-3-yl)-2-[4,5,7-trichloro-1-methyl-3-oxoinden-2-ylidene]acetamide 4-[3-bromo-7-[(5-methylpyrrolidin-2-ylidene)amino]pyrazolo[1,5-a]pyrimidin-5-yl]-N-benzylpiperidine-1-carboxamide 4-[5-(1H-pyrazole-5-carbonylamino)pyridin-2-yl]oxybenzoic acid 2,4-bis(1,3-benzodioxol-5-yl)-6H-pyrido[2,1-a]isoindole 2,3-dichlorobenzamide;2-[3-(4-fluorophenoxy)azetidin-1-yl]sulfonylpyridine 3-[4-(difluoromethyl)phenyl]-1H-pyridazine-2,5-diamine 2-[(4-butylsulfanylphenyl)sulfonylamino]acetic acid 4-[(1-methylbenzimidazole-2-carbonyl)amino]cyclohexane-1-carboxylic acid 5-bromo-4,8-dichlorobenzo[b]carbazole N-[(1R,3S)-3-hydroxycyclopentyl]quinoline-7-carboxamide N-[1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)piperidin-4-yl]acetamide 4-N-[3-(2,3-difluorophenyl)propyl]pyridine-2,4-dicarboxamide (3-chlorophenyl)sulfanylmethanesulfinic acid 2-[(4S,5R)-3-acetyl-6,10-dihydroxy-8-oxodecanoyl]benzamide (E)-1-cyclohexa-2,4-dien-1-ylbut-1-ene-1,3-diol;ethane 2-[4-(2-methylbutan-2-ylamino)cyclohexa-1,3-dien-1-yl]-2-oxo-N-propan-2-ylacetamide;5-methylidene-7-[2-(1-sulfanylethoxy)phenyl]hepta-1,6-dienethiol (3R)-N-[(3S,7R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-3-methoxy-1-[4-(trifluoromethyl)phenyl]sulfonylpyrrolidine-3-carboxamide [(E)-2,3-dihydro-1H-imidazo[1,2-c]quinazolin-5-ylidenemethyl]phosphonic acid 5-(2,3-dimethylindole-1-carbonyl)pyridine-3-sulfinate (2R)-N-[3,5-bis[(4-aminophenyl)methoxy]phenyl]pyrrolidine-2-carboxamide [(3S)-1-[4-cyclopentyloxy-5,7-difluoro-8-(propan-2-ylamino)quinoline-3-carbonyl]pyrrolidin-3-yl]carbamic acid 1-[(5R,6S)-6-ethylcyclohexa-2,4-dien-1-yl]imidazole 4-(methylaminomethyl)-2-[3-(pyridin-4-ylamino)prop-1-ynyl]phenol 2-[3-(4,5-dihydroimidazol-1-yl)-N-methoxyanilino]pyrimidine-4-carbonitrile 2-methyl-N'-[3-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl]-2-pyridin-2-ylbutanediamide 5-(3,5-difluorophenyl)-N'-hydrazinylthiophene-2-carboximidamide N-[(3R)-1,1-dioxothiolan-3-yl]-2,2-dimethyl-4H-benzo[g]chromene-6-carboxamide 4-(4-benzyl-1,3-thiazol-2-yl)-2,6-ditert-butylphenol [4-amino-2-chloro-6-(3,5-dimethylpiperazin-1-yl)pyrimidin-5-yl]-cyclohexa-1,3-dien-1-ylmethanone 2-[4-(difluoromethyl)benzoyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-5-carboxylic acid 2-[6-(trifluoromethoxy)naphthalen-1-yl]benzotriazole (5E)-5-[[1-(2,4-dinitrophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-imino-1,3-thiazolidin-4-one N-butyl-2-[2-(cycloheptylamino)ethoxy]benzamide 2-hydroxyimino-3-(1,3-thiazol-2-yl)-5H-chromeno[4,3-b]pyridine-8-carboxamide 4-[3,5-bis(4-methoxyphenyl)pyrazol-1-yl]benzenesulfinate 6-methyl-3,4-dihydronaphthalene;1,2,8-trihydroxy-9H-xanthene-9-carboxylic acid 4-chloro-N,3-dihydroxybenzenecarboximidate 5-[4-[2,3-difluoro-5-(2-methylsulfonylethoxy)phenyl]piperidine-1-carbonyl]-7-piperidin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide 6-amino-9-[2-[2-(4-hydroxyphenyl)hydrazinyl]ethyl]purine-8-thiol 1-[3-fluoro-4-[[1-(1H-indazol-5-yl)triazolo[4,5-b]pyridin-7-yl]oxymethyl]phenyl]-N,N-dimethylmethanamine N-methyl-1-[[4-(trifluoromethoxy)phenyl]methylideneamino]ethanamine (2R)-1-[4-(3,5-dichlorophenyl)piperazin-1-yl]-3-[(E)-2-naphthalen-1-ylethenyl]sulfanylpropane-1,2-dione 4-[2,5-dichloro-N-(3-methylbutyl)anilino]benzenesulfonic acid 2-[(6-methylpyridin-2-yl)oxymethyl]-8-(thiophen-3-ylmethyl)-5-oxa-2-azaspiro[3.4]octane;2,2,2-trifluoroacetic acid 2-(6,8-dihydroxy-4-oxoquinazolin-3-yl)-N-[1-methyl-3-phenyl-5-(prop-2-enoylamino)pyrazol-4-yl]acetamide N-[(3-benzylimidazol-4-yl)methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide 3-(4,5-dihydroimidazol-1-yl)-6-N-naphthalen-2-yl-4-N-phenylbenzene-1,4,6-triamine 4-[5-(furan-2-ylmethylamino)-1,3,4-thiadiazol-2-yl]phenol (2S)-3-(4-methylphenyl)-1,2-diphenylpropan-1-one 2-[3-(2,5-difluorophenyl)-4-oxoquinazolin-7-yl]-N-(oxolan-2-ylmethyl)acetamide 2-(3-chlorophenyl)-5,6-dimethoxy-1H-benzimidazole 1-(2,5-dimethylphenyl)-3-[4-[7-(4-hydroxyphenoxy)-1,6-naphthyridin-2-yl]phenyl]urea 2-[8,14-difluoro-3-thiapentacyclo[11.7.0.02,10.04,9.015,20]icosa-1(13),2(10),4(9),5,7,11,15,17,19-nonaen-6-yl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 6-[(3-chlorophenyl)methyl]-2,4,5-trifluorocyclohexa-1,3-diene-1,3-disulfonamide N-[(6R)-7-amino-5,6-dimethyl-4-(2,3,4-trifluorophenyl)octan-4-yl]pyridine-3-carboxamide 2-(3,4-dihydropyridin-2-yl)thieno[3,2-c]quinoline 2-(2,4-dihydroxyphenyl)-3,5-bis[4-(oxiran-2-ylmethoxy)phenyl]phenol 2-[4-methylsulfanyl-N-(2-methylpropyl)anilino]ethanol 3-[1-(2,3-dihydroindol-1-yl)ethoxymethyl]aniline N-(2,4-dimethylphenyl)sulfonyl-1-propanoylpyrrolidine-3-carboxamide 1-N'-cyclopropyl-5-(3,4-dichlorophenyl)-3-N'-[2-methoxy-6-methyl-4-[4-(trifluoromethyl)imidazol-1-yl]benzoyl]-5,6-dihydro-4H-pyrazolo[3,4-e]indazole-1,3-dicarboxamide 5-(methylaminosulfanyl)benzo[c]acridine 6-[(2R)-butan-2-yl]oxy-2,3-dihydronaphthalene [2-(4-phenylbenzenecarboximidoyl)pyridin-3-yl]boronic acid 3-[(4R,9aR)-8-(2-methoxyethyl)-1-oxospiro[6,7,9,9a-tetrahydro-5H-[1,3]oxazolo[3,4-a]pyridine-1,3'-piperidine]-4-yl]benzonitrile;2,2,2-trifluoroacetic acid 1-[(2S)-1,1-difluoro-3-hydroxypropan-2-yl]-4-methoxy-6-(3-nitrophenyl)pyrimidin-2-one 1-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethanone 1-[7-[(1Z)-buta-1,3-dienyl]sulfanyl-2,5-dimethylpyrazolo[1,5-a]pyrimidin-6-yl]ethanone 3-azido-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine (2E)-6-[3-(2,4-difluorophenyl)oxetan-3-yl]-2-ethylidene-1H-pyrimidine [3-(ethylamino)azetidin-1-yl]-[6-methoxy-2-[4-(propan-2-ylamino)phenyl]-7,8-dihydroquinolin-5-yl]methanone 5-[(E)-2-methylbut-1-enyl]-3-(4-morpholin-4-ylcyclohexyl)-7,8,9,10-tetrahydrobenzo[b]carbazole-6-carboxylic acid 5-(3,4-difluorophenyl)-2-methyl-N-[1-[4-(trifluoromethoxy)phenyl]ethyl]pyrazole-3-carboxamide 4-N,6-dimethyl-2-N-[5-methyl-3-(oxan-4-yl)-1,2-oxazol-4-yl]pyrimidine-2,4-diamine (E)-N',2,3,3-tetramethylhex-4-enimidamide;3-(4-propanoylphenyl)imidazolidine-2,4-dione [4-(difluoromethoxy)phenyl]-[3-methylsulfanyl-4-[(4-pyridazin-4-ylpiperazin-1-yl)methyl]pyrrolidin-1-yl]methanone 2,4-dimethyl-N-(6-propanoylpyridin-3-yl)-1,3-thiazole-5-carboxamide (7R)-N-(4-ethoxyphenyl)-5-oxo-2-propan-2-ylidene-1,3-diazinane-6-carboxamide (E)-1-[10-chloro-2-(4-methylpiperazin-1-yl)sulfonyl-12,14-diazatricyclo[9.5.0.03,8]hexadeca-1(11),3,5,7,12,15-hexaen-13-yl]-N',N-dimethylethene-1,2-diamine (2R)-1,4,5-trihydroxy-6-methyl-7-[(Z)-3-phenylprop-2-enoyl]oxy-3,3a,4,9b-tetrahydro-2H-benzo[g]indole-2-carboxylic acid N-[6-(difluoromethoxy)pyridin-3-yl]benzenesulfonamide 6-(hydroxymethyl)-1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazole-7-carboxylic acid N-[4-methoxy-3-(2-pyrrolidin-1-ylethoxy)phenyl]-6-pyridin-2-ylpyridine-3-carboxamide 2-[[4-(5,8-dimethylpyrazolo[1,5-a][1,3,5]triazin-2-yl)piperazin-1-yl]methyl]-6,7,8,9-tetrahydropyrido[3,2-b]indolizine (1E,3Z)-2-[(Z)-2-phenylethenyl]penta-1,3-dien-1-amine 2-[3,5-dichloro-4-(5-methylthieno[3,2-d]pyrimidin-4-yl)oxyphenyl]-1,1-difluoro-3-oxopropane-2-sulfonic acid 3-[5-chloro-2-(4,6-dimethylpyrimidine-5-carbonyl)phenoxy]propanoic acid 2-[(E)-[4-[(1S)-1-[3-bromo-5-fluoro-2-methoxy-6-methyl-7H-cyclopenta[b]pyridin-1-yl]ethyl]piperazin-1-yl]iminomethyl]phenol 3-[1-(4,5-dihydro-1,2-oxazole-3-carbonyl)-6-fluoropiperidin-3-yl]benzamide 1-cyclohexa-2,4-dien-1-ylsulfanyl-5H-pyrazolo[3,4-d]pyrimidin-4-one (5R,7S)-N-[2-(4-fluorophenyl)-1-[3-methoxy-4-[4-(trifluoromethyl)phenoxy]piperidin-1-yl]ethylidene]-7-methyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 2-[(4S)-4-benzyl-6,8-dimethoxy-1,3-dihydroisoquinolin-2-yl]acetic acid 4-[(1S)-5-acetylcyclohex-3-en-1-yl]oxycarbonylbenzoic acid ethane;4-[3-[4-(2-fluoro-5,6,7,8-tetrahydroquinolin-5-yl)piperazin-1-yl]propoxy]benzoic acid 3-[2-(1H-indol-3-yl)ethynyl]benzenesulfonamide (3R)-2,3-difluorobutanal;3-N-methyl-1H-indazole-5-carbohydrazide (Z)-4,7-dihydroxy-1-[3-[2-(methylamino)ethoxy]phenyl]hept-5-en-3-one 2-methyl-5,12-dihydrobenzo[b]acridine;1,4-xylene 2-[(3,5-dichlorophenyl)methyl]-4-oxopentanoic acid 5-[4-(azidomethyl)phenyl]-2-thiophen-3-ylpyridine 3-(5-chloropyridin-2-yl)sulfanyloxyaniline 3-[5-(1,2,4-triazol-1-yl)pentanoylamino]butanoic acid 1-cyclopentyl-7-(diethylamino)-6-fluoro-N,4-dioxoquinoline-3-carboxamide 1-(2,6-difluorobenzoyl)-N-[4-[[3-ethoxy-4-(7-oxooxocan-4-yl)phenyl]sulfamoyl]phenyl]piperidine-3-carboxamide N-methoxy-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxamide 1-[(6-chloro-1,3-benzodioxol-5-yl)sulfanyl]-2,3-dihydroindole 1-methoxy-4-[2,3,7-tris(ethenyl)anthracen-9-yl]oxybenzene N-[(2R)-1-amino-3,3-dimethyl-1-oxobutan-2-yl]-4-(3-chlorophenyl)cyclohexane-1-carboxamide;(E)-but-2-ene 2-[(3S,4R)-1-[4-cyano-3-(trifluoromethyl)phenyl]-4-hydroxypiperidin-3-yl]acetamide (2E)-1,3-bis[(4-chlorophenyl)sulfonyl]penta-2,4-dien-2-ol 1-[6-cyclohexyloxy-2,4-bis(2-methoxyphenyl)pyridine-3-carbonyl]piperidin-4-one N-[6,7-diamino-5-(2-methylpropanimidoyl)isoquinolin-3-yl]cyclobutanecarboxamide N-(2,3-dimethylphenyl)-1-ethylpiperidine-4-carboxamide 6-cyclohexyloxycarbonyl-1,4-dimethylindole-2-carboxylate (2S,4R)-1-[1-[(3R)-1-propanoylazepane-3-carbonyl]piperidin-4-yl]-N-quinolin-5-ylsulfonyl-4-[4-(trifluoromethyl)phenyl]pyrrolidine-2-carboxamide 4-[(4-aminophenyl)sulfonylmethyl]benzaldehyde 5-[(1S)-1-azidopropoxy]-3,4-dihydro-2H-naphthalen-1-one 2-[5,6-dichloro-1-(4-cyclobutylphenyl)sulfonylindol-3-yl]propanoic acid N-[1-(diethylamino)propan-2-yl]-3-methoxy-4,6,7,8-tetrahydrofuro[3,2-c]azepine-5-carboxamide 6-(2,4-difluorophenyl)-5H-thieno[3,2-b]pyridine (3R)-5-[3-[5,6-dimethyl-2-(pyridine-4-carbonylamino)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-2,5-dioxopyrrolidine-3-carboxamide 2-azidosulfanyl-1,3-bis[(4-chlorophenyl)methyl]benzene 2-[4-(dipropylamino)anilino]acetic acid (2S)-1-[(3R)-1,2-dihydroxyheptan-3-yl]-N-[4-[5-fluoro-6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]-2-oxo-4H-pyrido[3,2-d]pyrimidine-3-carboxamide 4-[5-[(4R)-3,8-dimethyl-2-oxooxepin-4-yl]sulfanylthiophen-2-yl]benzoic acid 2-bromo-1,3,5-triphenylbenzene 1-azido-2,3,4-trifluoro-9H-fluorene N-[5-(2-aminopyrimidin-4-yl)oxy-6-methylpyridin-3-yl]-1H-indole-3-carboxamide;ethane (2E)-4,5-dimethylhepta-2,6-diene;ethane;9-ethoxy-2H-naphtho[2,1-f]isoquinolin-10-one 3-[(2E)-penta-2,4-dienoyl]chromen-4-one 4-[5-amino-6-chloro-2-(difluoromethyl)-1-hydroxyindol-3-yl]benzoic acid (2R,3S)-2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-N-(5-propan-2-yl-1H-pyrazol-3-yl)butane-3-sulfonamide N-azido-4-phenylcyclohexa-1,5-dien-1-amine 4-N,6-dimethylquinoline-2,4-diamine 3-azidooxy-N,N-dibenzylpropanamide 3-(2-diazohydrazinyl)-N,N-dimethylbenzamide (6S)-1,3-bis(methylamino)-6-naphthalen-2-ylpyrrolidine-2,5-dione (6-aminopyridin-3-yl)-[4-(1H-indole-2-carbonyl)piperazin-1-yl]methanone 7-chloro-1-ethoxyphenazine 2-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]isoindole-1,3-dione 4-(2,5-dioxopyrrol-1-yl)oxy-N-[2-(4-hydroxy-3-methoxyphenyl)ethyl]butanamide 2-[4-(cyclopropanecarbonyl)piperazin-1-yl]quinoline-6,8-dicarboxylic acid [4-(methoxyamino)piperidin-1-yl]-[4-methyl-5-(2-methylpyridin-3-yl)thiophen-2-yl]methanone 3-hydroxy-2-[(4-methylbenzoyl)amino]propanethioyloxidanium 2-[(6-hydroxy-1H-indol-3-yl)diazenyl]benzoic acid N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-5-methoxybenzamide;formic acid 6-(cyclopentylmethylamino)-N'-hydroxy-3-nitropyridine-2-carboximidamide N-(5,6-dimethoxypyridin-3-yl)-2-[2-(2-methylsulfonylpyrimidin-4-yl)phenyl]-1H-indole-6-carboxamide 1-[4-methylsulfanyl-3-[(Z)-prop-1-enoxy]pyridin-2-yl]oxycyclobutane-1-carboxylic acid 4-[2-(cyclohexylamino)pyrimidin-5-yl]cyclohexan-1-one 2-[1,3-bis(9H-fluoren-1-yl)propan-2-yl]oxypyrimidine 6-benzyl-1,3,9,11,12-pentazatetracyclo[8.7.0.02,7.013,17]heptadeca-2(7),10,13,15-tetraene 3-chloro-4-[4-(cyclopropylmethoxy)piperidin-1-yl]aniline 3-(4-methoxypyridin-2-yl)-4,5-diphenyl-1,3,5-triazine 5-hydroxy-2,3,4-trimethylbenzenesulfonic acid (4Z)-2-[5-fluoro-3-methyl-1-(2,2,2-trifluoroethyl)indol-2-ylidene]-3-hydroxypropanoic acid 4-[2-methylbutanoyl(pyridin-3-yl)amino]benzenesulfonic acid 4-[5-[3-(cyclopropylcarbamoylamino)phenyl]pyrimidin-2-yl]benzamide 4-bromo-2,6-bis[(E)-3-oxobut-1-enyl]benzaldehyde 4-(5-oxo-2,3-dihydrothieno[3,4-b][1,4]dioxin-7-yl)butanamide 2-(5-chloropyridin-3-yl)-N-[2,4-dimethoxy-7-(1-methylpyrrolidin-3-yl)oxyquinazolin-6-yl]acetamide 2,6-dimethyl-4-[(1R)-1-propanoylpiperidin-3-yl]pyridine-3-carbonitrile 6,7-dimethoxy-1-(3-morpholin-4-ylpropyl)quinazoline-2,4-dione 2-bromo-5-(10,10,10-trifluorodecyl)benzoic acid N-[2-(4-amino-5-hydroxy-6,7-dihydropyrrolo[3,4-d]pyrimidin-2-yl)phenyl]-4-chlorobenzenesulfonamide (E)-1-cyclopentyl-3-[5-[2-fluoro-4-[2-[methyl(oxolan-3-yl)amino]ethoxy]phenyl]thiophen-2-yl]prop-2-en-1-one 4-[2,5-dimethyl-1-(4-nitrophenyl)hexan-3-yl]cyclohepta-1,4,6-triene 2-(4-cyanoanilino)-N'-[2-methoxy-5-[1-(oxidoamino)ethenyl]phenyl]-5H-pyrrolo[3,2-d]pyrimidine-6-carbohydrazide 5-bromo-2-[(4E,6Z)-3-methylideneocta-1,4,6-trienyl]furan [4-chloro-2-(hydroxymethyl)indol-1-yl]-naphthalen-1-ylmethanone 6-fluoro-3,4-dihydro-1H-isoquinoline;hydrochloride 1-(3,5-dichlorophenyl)-5-hydroxy-2H-pyrimidine 4-[(3E,5Z)-hepta-1,3,5-trien-2-yl]oxybenzenecarboximidamide 1-[3,3-difluoro-5-(4-methylphenyl)cyclohexa-1,5-dien-1-yl]pentan-2-one 2-[(4E)-3-ethoxycarbonyl-4-hydroxyiminopentyl]pyridine-4-carboxylic acid (2-fluorophenyl)-[7-[3-methoxypropyl(methyl)amino]furo[3,2-b]pyridin-5-yl]methanone 1-[2-(4-chlorophenyl)ethyl]-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carbonylamino)thiourea 5-cyclopropyl-4-(7-ethoxynaphthalene-2-carbonyl)morpholin-3-one N-[5-cyano-4-(furan-2-yl)pyrimidin-2-yl]-2-(2,6-difluorophenyl)acetamide 3-[6-(2-methylhexan-2-ylamino)pyrimidin-4-yl]benzimidazole-5-carbonitrile 1,3-bis(2-chlorophenyl)thiourea 1-[2,6-di(propan-2-yl)phenyl]-3-[2-[5-fluoro-4-(7-fluoro-2-methylindazol-5-yl)cyclohexa-1,3-dien-1-yl]ethyl]urea (2S)-3-[1H-indol-7-ylmethylideneamino]-1,4-dihydro-2,4-benzodiazepine-5,6-dione 2-bromo-1,3-dichloronaphthalene 4-(3,5-dimethylphenyl)-1-[5-(trifluoromethoxy)pyridin-2-yl]butan-2-one (Z)-1-N,1-N'-bis[[4-(trifluoromethyl)phenyl]diazenyl]ethene-1,1-disulfonamide (4S)-4-[(1S)-1-[3-[3,5-bis(trifluoromethyl)phenyl]-2H-pyridin-6-yl]-1-chloroethyl]pyrrolidine-2,5-dione 3-(2,6-dichlorophenyl)oxirane-2,2-dicarbonitrile 1-azidooxy-2,3-difluoro-4-phenylbenzene 6-[(3,5-difluorophenyl)methyl]quinoline 2-(6,7-dimethoxynaphthalen-1-yl)acetic acid [(2R,3S)-2-(hydroxymethyl)-4,5,7,8-tetrahydrooxepino[4,5-c]pyrazol-3-yl]-(4-pyrazin-2-ylpiperidin-1-yl)methanone 3-[4-(2,6-difluorophenyl)-1H-indole-2-carbonyl]-5-phenylcyclohexa-2,4-diene-1-sulfonamide 4-[(2R)-2,3-dihydroxypropoxy]-5-[[4-hydroxy-6-(hydroxymethyl)oxan-2-yl]amino]benzene-1,3-disulfonic acid 3,5-bis[1,2-dihydropyridin-6-yl(phenyl)methylidene]-1H-pyrrol-4-one N-[(1S)-1-phenylethyl]pyrrolidine-2-carboxamide (2Z)-2-[amino(phenyl)methylidene]-4-[[5-[2-(diethylcarbamoyl)benzimidazol-1-yl]thiophen-3-yl]methylimino]cyclohexan-1-one 1-azido-4-[(4-ethoxyphenyl)methyl]piperazine (4R)-2-[6-[[1-(3,5-difluoropyridin-4-yl)azetidin-3-ylidene]methylamino]pyrimidin-4-yl]-4-hydroxy-N',2-dimethyl-N,3-dipropoxybutanimidamide (3Z)-6-methyl-5-[1-(2-methyl-4,6-diphenyl-1H-pyrimidin-2-yl)piperidin-4-yl]hexa-3,5-dienoic acid 5-(4,6-dimethylpyrimidin-2-yl)oxyquinoline 4-bromo-1,2,3,5,6-pentafluorobenzene 2-fluoro-1,4-dimethylbenzene;2-[3-(4-methoxyphenyl)-4-oxochromen-8-yl]acetaldehyde (2Z)-N'-hydroxy-1-phenyl-2-[3-[(4-propan-2-ylsulfonylpiperazine-1-carbonyl)amino]pyridin-2-ylidene]ethanediamide 2-cyclohepta-1,3,5-trien-1-yl-4-phenyl-6,7-dihydro-5H-[1]benzofuro[2,3-d]pyrimidine;ethane [2-[4,6-diamino-5-(methyliminomethyl)pyrimidin-1-ium-3-yl]phenyl]methanol 2-[4-amino-7-methyl-5-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidin-6-yl]phenol N-[4-(2,3-dihydro-1H-inden-5-yloxy)-3-methylphenyl]-4-hydroxy-6-oxo-1H-pyridine-3-carboxamide 4-bromo-N-(5-chloropyridin-2-yl)-3-fluorobenzenesulfonamide 1-[(5S)-3,5,6-trimethylcyclohexa-2,4-dien-1-yl]naphthalene 2-[1-(4-aminophenoxy)hexoxy]-6-methylaniline (2S,3R)-3-[[4-(2-methylpyridin-4-yl)oxypiperidine-1-carbonyl]amino]oxolane-2-carboxylic acid 5-[(2Z,3E)-1-(4-acetyloxyphenyl)-4-methylidenehexa-2,3-dien-2-yl]thiophene-2-carboxylic acid 4-(4-chlorophenoxy)benzene-1,2-dicarboxamide;hydrochloride 1-[3,5-bis(difluoromethyl)-4H-pyrimidin-2-yl]ethanol 3-[2-methylpropyl(pyridin-2-yl)amino]propane-1,2-diol 1-(3-chlorophenyl)pyrrole;ethane 1-[3-(dimethylamino)butyl]-N,5-dihydrocyclohepta[b]pyrrole-2-carboxamide 3-[2,4-dimethylpentyl(formyl)amino]-4-ethoxy-5-(hydroxymethyl)benzoic acid 3-chloro-N'-hydroxy-2-(3-methylpyrazol-1-yl)pyridine-4-carboximidamide 2-chloro-N-(4,6-dimethylpyrimidin-5-yl)quinoline-3-carboxamide 3-methylsulfanyl-6,7-dihydro-5H-[1,2]oxazolo[4,3-c]pyridine-4-carboxylic acid 2-[6-(4-methoxy-N,3-dimethylanilino)pyrazin-2-yl]cyclohexa-1,5-dien-1-ol 2-[1,3-dioxo-5-(1H-pyrazolo[4,3-b]pyridine-6-carbonylamino)isoindol-2-yl]acetic acid 2-[4-(3,5-diethylpyridin-2-yl)piperazine-1-carbonyl]-7H-thieno[3,4-b]pyrazin-5-one;ethane 1-(5,8-difluoro-2-hexan-3-ylimidazo[1,2-a]pyridine-6-carbonyl)pyrrolidine-2-carboxamide 5-[2,3-difluoro-4-(trifluoromethyl)phenyl]-1H-pyrazol-3-amine [(2-cyclohexa-1,5-dien-1-ylphenyl)methylideneamino]thiourea N-[(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-2,1,3-benzothiadiazol-6-amine 4-[(6R,8aR)-1-benzyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-6-carbonyl]benzoic acid N-(5,6-diethyl-4-fluoropyridin-2-yl)ethanimine 5-chloro-3,4-dihydro-1H-pyrido[4,3-b]indole-2-carboxylate 3-[(2S)-1,4-bis(diphenylphosphanylmethoxy)butan-2-yl]phenol (4S,5R)-6-[2-methylpropanoyl-(2-methylpyridin-3-yl)amino]oxy-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid 4-azido-3,3-dimethylnaphthalene-1,2-disulfonic acid 3-amino-6-(4,5-dimethyl-1H-pyrazol-3-yl)-2-fluorobenzonitrile 2-[(3S)-4-benzylmorpholin-3-yl]-6-pyridin-4-ylimidazo[1,2-a]pyrazin-8-amine N-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-2-phenylethanesulfonamide N-[4-(2,3-dihydro-1H-indene-5-carbonyl)phenyl]-5-fluoropyridine-3-carboxamide 4-amino-5-(2-pyridin-3-ylethoxy)cyclohepta-2,4,6-triene-1-carboxylic acid 4-[2-(6,7-dimethoxyquinazolin-4-yl)oxyethyl]aniline [2-(4,5,6-trifluoronaphthalene-1-carbonyl)naphthalen-1-yl]oxy-(trihydroxymethyl)phosphinic acid (3S,4R)-1-[2-(2-chlorophenyl)ethyl]-4-(3,5-difluorophenyl)-N-methylpyrrolidine-3-carboxamide (E)-1,4-difluoro-3-phenylbut-2-en-1-ol 2-[4-chlorobutyl(cyclohexyl)amino]phenol 1-[5-amino-2-(4-ethoxyphenyl)phenyl]-3,4-diphenylbutan-2-one (3R,5S)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]naphthalen-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol 3-[3-oxo-6-[4-[(4-phenylthiophen-2-yl)methoxy]piperidine-1-carbonyl]-1H-isoindol-2-yl]piperidine-2,6-dione [6-(2,5-dichlorophenyl)-3-methyl-7H-[1,2]oxazolo[5,4-d]pyrimidine-4-carbonyl]oxidanium 2-[4,5,7-trideuterio-6-(2,3,4,5-tetradeuteriopyrrol-1-yl)dibenzothiophen-4-yl]pyridine 1-[4-chloro-3-(trifluoromethyl)phenyl]pyrrolidine;2-[2,6-dimethoxy-4-(piperidin-4-ylamino)sulfanylphenoxy]acetic acid 5-chloro-4-[(2S,3R)-6-(3,5-dimethylpyrazol-1-yl)-3-hydroxy-2-methyl-3-phenylmorpholin-4-yl]pyridine-3-carbonitrile N-[5-(2,4-dichlorophenyl)-3H-1,3,4-oxadiazol-2-ylidene]formamide 2-[4-amino-3-(2,5-dimethylphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-N,N-dimethylacetamide 2-[4-(aminomethyl)-1,3-thiazol-2-yl]-N-(6-pyrrolidin-1-ylpyridin-3-yl)acetamide 2-[4-(2,3-dihydropyrazin-5-yl)phenyl]-6,7-dihydro-1H-pyrrolo[2,3-c]pyridine 2-[2-(2,5-difluorophenyl)morpholin-4-yl]ethanamine 2-[3-fluoro-4-(pyrrolidine-1-carbonyl)phenyl]acetic acid N-[2-(diethylamino)pyrimidin-5-yl]-4-methoxy-6-methylcyclohepta-1,3,5-triene-1-carboxamide 1-[2-(5,6-dimethylpyridin-3-yl)acetyl]-N-phenylpyrrolidine-2-carboxamide 3-[N-(2,4-dichloropyrimidin-5-yl)-4-(pyridin-2-ylsulfamoyl)anilino]propanoic acid 4-[5-bromo-1,2-di(propan-2-yl)pyrrole-3-carbonyl]piperazine-1-carboxylic acid N-[2-amino-1-(furan-3-yl)ethyl]-4-methoxybenzamide 6-(4,5-dimethylimidazol-1-yl)pyridine-3-carboxamide 5-[2,2-dimethylpropoxy(hydroxy)methyl]naphthalene-1-carboxylic acid 5-cyclopropyl-4,6-diethyl-2H-1,3,4-oxadiazine 4-[[2-(3,5-dibromopyridin-4-yl)ethyl-methylamino]methyl]-N'-hydroxybenzenecarboximidamide 2-(3,6-dihydro-2H-pyran-4-yl)-N-[1-(furan-2-ylmethyl)piperidin-4-yl]propanamide 5-(3,5-dichlorophenyl)-1-methyl-N-[1-[6-[(4-methylpiperazine-1-carbonyl)amino]pyrimidin-4-yl]cyclopropyl]pyrazole-4-carboxamide 2-(4,5-dihydroimidazol-1-yl)-N,N-diphenylaniline N-[5-(2-aminoquinazolin-6-yl)pyridin-3-yl]formamide;methoxyethane [(1R)-2,3,4,9-tetrahydropyrano[3,4-b]indole-1-carbonyl]carbamic acid N-[(E)-1-naphthalen-2-ylpentylideneamino]aniline 4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-2-methoxyaniline 2-(4,4-dimethylcyclohexen-1-yl)-N-[3-[[5-(1H-indazol-6-ylamino)pyrimidin-4-yl]amino]phenyl]acetamide 2-amino-5-(3-chlorophenyl)-5,8-dihydro-1H-imidazo[4,5-g]quinazoline-7-carboxylic acid 2-bromo-1-[4-(chloromethyl)phenoxy]cyclohexa-3,5-diene-1,3-dicarboxylic acid 3-(5-aminopyridine-2-carbonyl)benzoic acid (1-methoxycyclopropyl)-[3-methoxy-2,5-dimethyl-4-[[4-(oxan-4-ylamino)-6-phenylpyridine-2-carbonyl]amino]phenyl]azanium N-methyl-3,4-bis[(2-methylpropan-2-yl)oxy]benzenesulfonamide (4R)-1-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-3-(1,3-thiazol-4-ylmethyl)imidazolidine-2,4-dione 2-(1-ethylpyrazol-4-yl)-N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)propyl]acetamide;dihydrochloride 3,4-dimethyl-2-methylimino-6-[(Z)-prop-1-enyl]-1H-quinazolin-7-one N-[1-(furan-2-carbonyl)azetidin-3-yl]-N-[2-[5-methoxy-6-(trifluoromethyl)pyridin-3-yl]ethyl]methanesulfonamide 3-[5-methoxycarbonyl-4-methyl-2-(2,4,6-trichlorophenyl)-1,4-dihydropyrimidine-6-carbonyl]piperidine-1-carboxylic acid (2R)-1-[4-[7-chloro-3-[3-methyl-4-(1,1,4-trioxo-1,2,5-thiadiazolidin-2-yl)phenyl]imidazo[4,5-b]pyridin-2-yl]phenyl]sulfonylpyrrolidine-2-carboxylic acid [7-azido-1,2,3-trimethyl-5-phenyl-6-(trifluoromethoxy)indol-4-yl]-(3-hydroxyazetidin-1-yl)methanone 3-N,4-N-dimethyl-2-(5H-pyrrolo[2,3-b]pyrazin-6-yl)butane-1,3-diamine 2-hydroxy-6-(hydroxymethyl)-1,2-dihydronaphthalene-1,4,5,6,7-pentol 1,3-bis(4-methylphenyl)propan-2-one 1-[5-[(2-propan-2-ylphenoxy)methyl]furan-3-carbonyl]-N-[3-(4H-triazol-2-ium-2-yl)cyclobutyl]pyrrolidine-2-carboxamide 1-[(2-fluorophenyl)methylamino]-3,4-dihydro-2H-naphthalen-1-ol 5-azidooxy-N,N,2-trimethylaniline 3-[4,6-di(propanoyloxy)pyrimidine-5-carbonyl]piperazine-1-carboxylic acid 3-[1-(4-hydroxybutoxy)-3-oxohexan-2-yl]sulfanylbenzoic acid 3-(2,4-dioxopyrimidin-1-yl)butanedioic acid 1-[(1R)-6-fluoro-3,4-dihydro-1H-isochromen-1-yl]pyrrole (2-azido-2,3,4,6-tetramethylphenyl)carbamic acid 3-[4-[3-(aminomethyl)phenyl]-2-hydroxyphenyl]-4H-1,2,4-oxadiazol-5-one;hydrochloride N-[4-(diethylamino)phenyl]-2,4-dimethylpentanamide;ethane 2-cyclopropyl-6,6-dimethyl-1-pyridin-3-ylheptan-4-ol 1-azidooxy-3,4-dimethylnaphthalene 2-[N'-(3,4-dimethoxyphenyl)carbamimidoyl]benzamide 3-[1-methyl-2-(methylamino)benzimidazole-5-carbonyl]oxybutanoic acid 2-N-(4-aminophenyl)-3H-benzimidazole-1,2-diamine 2-[[3-(aminomethyl)piperidin-1-yl]methyl]quinoline-4-carboxamide 1-[3-(4-chlorophenyl)sulfanylphenyl]propan-2-one 2-[(E)-1-(4-aminophenyl)ethylideneamino]oxyacetic acid (2S)-6,8-dimethyl-N-propan-2-ylspiro[1,4-dihydroquinoxaline-3,4'-thiane]-2-imine [3-[(7,8-dimethoxy-2-methylquinoline-5-carbonyl)amino]-6-iminocycloocta-1,4,7-trien-1-yl]methylideneazanium N-[1-(6-aminopyridazin-3-yl)pyrrolidin-3-yl]-5-chloro-7,8-dihydronaphthalene-2-carboxamide 4-(4-ethyl-2,6-dimethylphenyl)sulfonylmorpholine N-(1,3-benzodioxol-5-ylmethylideneamino)-6-fluoro-4-oxospiro[1H-quinoline-3,4'-piperidine]-2-carboxamide 2,6-dichloro-4-[(Z)-[5-fluoro-1,4-bis[3-(trifluoromethyl)phenyl]butylidene]amino]phenol 2-[3-(1,2-benzoxazol-6-yl)phenyl]propanoic acid 1-[7-(4-fluorophenyl)-8,9-dihydropurin-6-yl]butan-2-amine N-[2,6-di(propan-2-yl)phenyl]-1-[4-[[6-(trifluoromethoxy)cyclohexa-2,4-dien-1-ylidene]amino]phenyl]propan-2-imine N-[(1S,2R)-3-ethylcyclohex-3-en-1-yl]-3-methoxy-4-phenoxybenzamide N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-N'-methanimidoylethane-1,2-diamine 2-[2,6-bis(2,4-dimethylphenyl)pyridin-4-yl]ethanol 1,5-dibromo-3-(2-methyl-4-nitrophenyl)-6,7-dihydroindole 1-[5-tert-butyl-2-(oxan-4-yl)pyrazol-3-yl]-3-[7-[2-(diethylamino)pyrimidin-5-yl]pyrazolo[1,5-a]pyridin-6-yl]urea 2-(3,5-difluorophenyl)-6-(4-propylcyclohexyl)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene N-[6-(2,4-difluorophenoxy)pyridin-3-yl]-1-(3-methoxypropoxy)methanimidate 2-[(6R)-6-methyl-5,6-dihydrobenzo[f][1]benzothiol-7-yl]pyridine 4-(2,5-difluorophenyl)butyl-[2-(3,4-dihydroxy-6-oxoxanthen-9-yl)oxyethyl]azanium 3-[(1S)-1-aminoethyl]-6-[2,3-dichloro-4-[(E)-3-hydroxyprop-1-enyl]phenyl]-8-fluoroquinazolin-4-one;oxolane (3S)-1-[2,2-dichloro-5-fluoro-4-(1-methylcyclopropanecarbonyl)oxy-3H-1-benzofuran-7-yl]pyrrolidine-3-carboxylate 4-(methoxymethyl)-N-(2-methoxyethylsulfanyl)aniline 1-N,2-N-dimethyl-4-N-(4-propoxyphenyl)benzene-1,2,4-triamine 2-(4,6-diphenylpyrimidin-5-yl)-1H-benzimidazole 1-(1,3-benzodioxol-5-ylmethyl)-N-[[3-methoxy-4-(1-methoxypropan-2-yloxy)phenyl]methylideneamino]piperidine-4-carboxamide 2,3-bis(ethenyl)-N-methyl-5,6-dihydroimidazo[1,2-a]pyridine-6-carboxamide 3-(cyclopropylmethoxy)-4-[3-[2-(5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-3-yl)ethynyl]phenyl]benzoic acid 5-fluoro-2-methoxypyridine;N-[(1R)-1-phenylethyl]naphthalene-2-carboxamide N-(4,6-dimethylpyrimidin-2-yl)-4-[prop-2-enoyl(1,3-thiazol-5-yl)amino]benzenesulfonamide 1-(2-acetylsulfanylethoxy)-7,10,11,12-tetrahydro-6H-benzo[c][1]benzazocine-5-carboxylic acid 1-cyclobutyl-6-hydroxy-5-[(Z)-pyrrolo[2,3-b]pyridin-4-ylidenemethyl]pyrimidine-2,4-dione 2,4-dibromo-6-ethenyl-N-ethenylaniline 2-(1,3-benzodioxol-5-yl)-N-[4-[2-hydroxy-3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl]acetamide 1-(4-chlorophenyl)-N,3-dimethylcyclobutan-1-amine;ethane 2-methyl-1,4-bis[(4-propan-2-ylcyclohexa-1,5-dien-1-yl)oxy]benzene 2,6-dimethylnaphthalene;ethane;5-(4-ethenylphenyl)-7H-purin-8-imine N-[2,4,6-trichloro-3-[[3-(trifluoromethyl)phenyl]methoxy]phenyl]acetamide N-[(1S)-6,7-difluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]-6-methoxy-7-(oxan-4-ylmethoxy)quinoline-5-carboxamide 2-(1H-indol-3-ylmethylideneamino)phenol 3-(4-acetylphenyl)-7-fluoro-N,N-dimethylindolizine-2-carboxamide;ethane 2-cycloheptyl-5-methylbenzoic acid N-[4-[2-[(3-chlorophenoxy)methyl]piperidin-1-yl]but-1-en-2-yl]hydroxylamine (2R)-N,4,5-trimethyl-1-[3-methyl-5-[6-methylidene-11-(4-methylphenyl)indolo[1,2-a]quinolin-10-ium-12-yl]thiophen-2-yl]hexan-2-amine (2E)-2-[5-ethylsulfonyl-6-[3-methanimidoyl-4-(trifluoromethoxy)phenoxy]pyridin-3-yl]-1-[6-(3-fluorooxetan-3-yl)pyridin-2-yl]penta-2,4-dien-1-one 4-N,6-dimethyl-2-N-[(2E)-2-[(methylideneamino)-(1-piperidin-3-ylpyrazol-4-yl)methoxy]penta-2,4-dienyl]pyrimidine-2,4-diamine 3-(2,4-dimethoxyphenyl)-7-[4-fluoro-3-(hydroxymethyl)anilino]quinoxaline-6-carbonitrile 2-[5-[5-(4,5-dihydro-1H-imidazol-2-yl)pyrazin-2-yl]benzimidazol-1-yl]acetic acid (2S)-N-[4-[4-cyanobutyl(methyl)amino]phenyl]sulfanyloxy-N,3-dihydroxy-2-(1H-indol-6-ylmethylideneamino)propanamide 2-(1,4-dimethyl-5,6-dihydronaphthalen-2-yl)dibenzothiophene 2-bromo-3,5-dichloropyridine 5-[(2R,3S)-3-butylpiperidin-1-yl]sulfonylisoquinoline;hydrochloride 2-tert-butyl-4-ethoxyisoquinolin-2-ium;chloroethane 5-benzylsulfanyl-2-bromofuran 4-[2-(5-cyanopyridin-3-yl)-6-fluorophenoxy]-N,N-dimethylpiperidine-1-sulfonamide 1-cyclopentyloxy-4-(2,5-difluorophenyl)-N-methylbutan-2-amine 1-[4-(6-tert-butylpyridazin-3-yl)piperidine-1-carbonyl]cyclopropane-1-carbonitrile 5-[4-azidooxy-3-(1H-pyrrol-2-yl)phenyl]-2-methoxypyridine [2-(azidomethyl)-4,6-bis(hydroxymethyl)pyridin-3-yl]-pyrrolidin-1-ylmethanone 1-[7-(difluoromethyl)-5-fluoro-1H-indol-2-yl]ethanone 1-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)piperazin-1-yl]prop-2-en-1-one 3-bromo-5-methylthieno[2,3-d]pyrimidin-4-one N-cyclohexyl-3-(4,6-dimethoxypyrimidin-2-yl)sulfanylpropanamide N-[2-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-6-methoxypyridine-3-carboxamide 1-[(3S)-3-[2,6-difluoro-4-(methanesulfonamido)phenoxy]pyrrolidin-1-yl]-3-morpholin-4-ylpropan-2-ol 2-(2,6-difluoro-4-methylphenyl)-5-pentoxybenzonitrile (E)-3-[1-[4-cyano-2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-enoic acid N-[1-(5-chloropyridine-2-carbonyl)piperidin-3-yl]tricyclo[4.3.0.02,4]nona-1(6),7-diene-8-carboxamide N-benzyl-2,4-dimethoxy-N-methylpyrimidine-5-carboxamide N-(1-aminoethylidene)-2,3-dihydroanthracene-9-carboxamide 3-amino-5-[(1R,2S)-2-piperidin-4-ylcyclopropanecarbonyl]benzaldehyde 2-[(3R)-1-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yloxy)phenyl]pyrrolidin-3-yl]acetic acid 3-(3-azidooxypropyl)benzonitrile 3-[4-(2,5-dimethoxyphenyl)benzotriazol-1-yl]phenol 6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]cyclohexa-1,3-diene-1-carboxylic acid 3-[(4-bromo-2,5-dimethylphenyl)sulfonylamino]benzoic acid 2-[4-(3,4-dihydropyridin-6-yl)phenyl]-1-(4-methoxycyclohexa-1,5-dien-1-yl)benzimidazole 2-[[3-(aminomethyl)phenyl]-naphthalen-1-ylsulfonylamino]acetic acid 3-[2,4-bis(trifluoromethyl)phenyl]-N-cyclohexylcyclobutan-1-amine 4-[(Z)-2-amino-1-[(2R,5S)-2,7-dimethyl-5-naphthalen-1-ylheptoxy]ethenyl]-3-chlorobenzaldehyde 2-[[4-amino-3-(2-methoxypyridin-4-yl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]-8-fluoro-7-[(E)-prop-1-enyl]-3H-pyrrolo[3,2-e]indole-1-carboxamide 2-(azidooxymethyl)-1,3-difluoro-5-[4-(trifluoromethoxy)phenyl]benzene 5-(4-chlorophenyl)-N-cyanopentanamide;ethane;3-methyl-1,2-dihydroindene 5-chloro-N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]thiophene-2-sulfonamide 3-[[5-(2,4-difluorophenyl)-2-methylphenyl]methyl]-4H-pyrimidine 1,6-dimethyl-5H-pyrazolo[3,4-d]pyrimidine-3,4,7-trithione 1-cyclopropyl-3-[4-(2,6-dimethoxyphenyl)-5-(5-hydroxypyridin-3-yl)-1,2,4-triazol-3-yl]piperidin-4-ol 3-ethylsulfanyl-7-(trifluoromethoxy)imidazo[1,2-a]pyridine 3,8-dibutylphenoxazine-10-carboxylic acid 5-azido-7,8-dihydronaphthalene-2-thiol 4-(5,6-dimethylpyridin-3-yl)-7H-furo[2,3-c]pyridine-2,3-diamine 5-[1,2,4-triazol-1-ylmethyl(thian-4-yl)amino]furan-2-carboxylic acid [1-[2-[1-(3,4-dimethylphenyl)ethylideneamino]oxy-5-fluoropyridin-4-yl]piperidin-4-yl]methanamine (2Z)-N-[(1S,3R)-3-methylcyclopentyl]-2-[(6-nitro-1H-benzimidazol-2-yl)imino]-1-oxo-4a,5,8,9,10,11-hexahydroindolo[2,3-b]quinoline-3-carboxamide 2-[(2Z)-2-[(5-chloro-3,4-dimethoxyphenyl)methylidene]hydrazinyl]-N-pyridin-3-yl-1,3-thiazole-5-carboxamide N-[2-(3-tert-butylphenyl)sulfanylethyl]-1-pyrrolidin-1-ylmethanesulfonamide 2-ethenyl-4-(5,6,7,8-tetrahydronaphthalen-1-yl)benzonitrile 2-(9,10-dioxoanthracen-1-yl)oxyacetamide N-[2,4-dinitro-6-(trifluoromethyl)phenyl]acetamide N-[2,4-dimethyl-5-[(5R)-3-(trifluoromethoxy)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-5-carbonyl]phenyl]formamide 4-(2,6-difluorophenyl)-2-[5-[(1R,5S)-3-(9H-fluoren-9-ylmethoxycarbonylamino)-6-bicyclo[3.1.0]hexanyl]-1,3,4-oxadiazol-2-yl]butanenitrile 4-[[5-amino-2-[2,6-dichloro-3-fluoro-4-(5,5,5-trifluoropentoxy)phenyl]imidazol-1-yl]methyl]benzenesulfonamide 6-chloro-3,4-dihydrocarbazole (2R)-1-[6-amino-5-[4-amino-3-(difluoromethyl)phenyl]pyrazine-2-carbonyl]pyrrolidine-2-carboxylic acid 1-[4-(5-fluoropentoxy)phenyl]ethanone N-[2,4-difluoro-3-(pyrimidine-5-carbonylamino)phenyl]carbamate (2R,3S)-3-benzyl-N-(1H-indazole-5-carbonyl)piperidine-2-carboxamide 5-[5,8-bis(4-chlorophenyl)imidazo[1,2-b]pyridazine-7-carbonyl]pyridine-3-carbonitrile (6S)-7-acetyl-3-butylsulfanyl-6-(2,5-dimethoxyphenyl)-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one [4-(6-aminopyridin-3-yl)piperidin-1-yl]-[2-(2-hydroxy-2-methylpropanoyl)-5,7-dihydro-4H-pyrano[3,4-c]pyrazol-7-yl]methanone (2S)-1-[4-[4-amino-7-methyl-5-[4-(pyrrolidine-1-carbonyl)phenyl]pyrrolo[3,2-d]pyrimidin-6-yl]piperidin-1-yl]-2-hydroxy-2-phenylethanone 2-(1,4-dioxan-2-yl)-N-[2-[4-[(Z)-hydroxyiminomethyl]phenyl]ethynyl]benzamide 5-(2,4-dichlorophenoxy)carbonyl-1H-pyrrole-3-carboxylic acid 2-[8-(4-chlorophenyl)-9H-pyrido[3,4-b]indol-1-yl]acetic acid;formic acid 4-(2-diazohydrazinyl)-N',5-dimethylpyridine-3-carboximidamide 2-[[(4,5-dichloro-1H-imidazole-2-carbonyl)amino]methyl]-N,3-diethoxy-N-methylbenzamide 3-[2-(benzylamino)ethyl]phenol;ethane (2R,5S)-N-methyl-4-oxo-1,3,9-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-10,13,15-triene-5-carboxamide;hydrochloride 3-[2-(benzenesulfonamido)phenyl]benzoate 6-chloro-N,3-dimethyl-5-oxo-7H-thieno[2,3-b]pyridine-2-carboxamide N-[5-(2,3-dihydroxypropoxy)-2-[6-[[1-[4-[dimethylsulfanyl(methylsulfonyl)amino]butyl]piperidin-4-yl]-methylamino]pyridine-3-carboximidoyl]phenyl]cyclopropanecarboxamide N-[1-(2,4-dichlorophenyl)ethenyl]piperidine-3-carboxamide [3-(4,5-dihydro-1H-imidazol-2-yl)cyclohexa-2,4-dien-1-ylidene]-phenyloxidanium (4R)-4-(2,3-dihydroindole-1-carbonyl)-5-[2-[1-(4-fluorophenyl)pyrazol-3-yl]-2-oxoethyl]-1-(2-methoxyphenyl)pyrrolidine-2,3-dione 2-(4,5-dimethylfuran-2-carbonyl)-N-[1-(pyridine-3-carbonyl)piperidin-3-yl]acetamide 4-[7-(4-chlorophenyl)-5-methylspiro[6H-pyrrolo[2,1-c][1,2,4]triazine-8,3'-pyrrolidine]-1'-yl]-N-hydroxybenzamide;ethane 2-[1,4-dimethyl-5-(naphthalene-2-carbonyl)-2-oxoquinolin-3-yl]acetic acid 2-N-methyl-5,6,8-triazatricyclo[7.4.0.03,7]trideca-1(9),2,4,6,10,12-hexaene-2,4-diamine 1-[(3-chlorophenyl)methylamino]-3-decylthiourea N-(5-chloro-2-methoxyphenyl)-1H-indole-7-carboxamide 2-[4-(N,3-dimethylanilino)-3,5-difluorophenyl]benzene-1,4-diamine 4-(1-azidoethyl)-6-[2,4-bis(trifluoromethyl)phenyl]pyrimidine 2-[(3,5-difluorophenyl)methyl]-N-(2-hydroxypropyl)thieno[3,2-b]pyridine-7-carboxamide 3-N-azido-6-N,2-diphenylbenzene-1,3,5,6-tetramine 1-[4-[2-(dimethylamino)ethyl]phenyl]-3-[2-fluoro-5-nitro-6-(2,2,2-trifluoroacetyl)pyridin-3-yl]urea 2-methoxy-1,4-dimethylbenzene;4-(methoxymethyl)heptane 2-[[(1R,3S)-3-(cyanomethylcarbamoyl)cyclohexanecarbonyl]amino]acetic acid;6-fluoro-2-(4-formamidophenyl)imidazo[1,2-a]pyridine-3-carboxamide 1-azido-2,3,4-trifluoro-5-methylsulfanylbenzene [4-(5-ethylpyrimidin-2-yl)oxypiperidin-1-yl]-(4-propan-2-ylfuran-3-yl)methanone 4-[(3R)-3-methylmorpholine-4-carbonyl]-1H-quinolin-2-one 2-[4-(dimethylamino)piperidine-1-carboximidoyl]benzene-1,3-diamine;ethane 3-[5-(trifluoromethyl)tetrazolo[1,5-a]quinolin-2-yl]phenol (1Z)-2,3,6,8-tetrafluoro-7-[4-(methoxymethyl)cyclohexylidene]-1-prop-2-enylideneanthracene 1-methyl-N-[[4-(piperidine-1-carbonyl)cyclohexa-2,4-dien-1-yl]methyl]indole-7-carboxamide 6-[(1R)-2,2,2-trifluoroethoxy]-N-[4-(triazol-2-yl)phenyl]pyridine-3-carboxamide 1-(5-tert-butylpyrazol-2-id-3-yl)isoquinoline;(Z)-6,6-difluoro-7-hydroxy-N-methanimidoyl-4-oxohept-5-enamide;iridium (2R)-3-azido-1-[(5S,7S)-4,5-dimethyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidine-2-carbonyl]pyrrolidine-2-carboxylic acid 4-[(Z)-3,4-dimethylpenta-1,4-dienyl]-N-(4-ethoxyphenyl)piperazine-1-carboxamide;3-[3-[3,5-dimethyl-2-[3-[(5-phenylpentanoylamino)methyl]phenyl]phenoxy]propyl]benzaldehyde ethane;N-[1-(2-hydroxypropanoyl)pyrrolidin-3-yl]benzamide 1-(2,3-difluorophenyl)-4H-indeno[1,2-c]pyrazole 5-(2-iodoethynyl)-1H-pyrrolo[3,2-b]pyridine 4-chloro-6-(1H-indol-3-yl)-N,N-dimethyl-1H-benzimidazole-2-carboxamide N-(cyclopropylmethoxy)-3-(5-propan-2-yl-1,3-thiazol-4-yl)aniline;formaldehyde N-(2,4-dimethylphenyl)-3-[(4-ethoxyphenyl)sulfonylamino]-5-hydroxy-7-oxo-8H-naphthalene-1-carboxamide 5-[2-[(3R)-3-fluoropiperidine-1-carbonyl]thieno[3,2-b]pyridin-7-yl]oxyisoquinoline-8-carboxamide 1-[3-(2,6-dichlorophenyl)propanoyl]-5-hydroxyimidazolidine-2,4-dione 1-(2,4,5-trimethylphenyl)sulfonylnaphthalene 2-[1-[3,5-diethyl-4-(4-methoxyphenyl)phenyl]ethylideneamino]oxycarbonyl-2-methylpropanoic acid [4-fluoro-2-(trifluoromethyl)phenyl]azanium 6-[4-amino-3-(1,2,5-oxadiazole-3-carboximidoyl)phenoxy]hexanoic acid (3E)-5,6-dimethylhepta-1,3,5-triene;2,5-dimethyl-1-[(Z)-prop-1-enoxy]-4-[(E)-prop-1-enyl]benzene;ethane 6-cyclohexyloxycarbonyl-3,4-dihydro-2H-chromene-5-carboxylate N-(2,2-diethoxyethyl)-1,3-thiazol-5-amine N-[3,4-dihydroxy-2-(3-methoxyphenyl)butan-2-yl]formamide 3-azido-1-[2,6-difluoro-4-(trifluoromethyl)phenyl]sulfonyl-5-ethylpiperidine N-methyl-6-(4-propanoylpiperazin-1-yl)pyridine-3-carboxamide 3-(1H-indol-2-yl)indole-6-carboxylic acid (3R,4S)-4-benzyl-2-tert-butyl-5-hydroxypiperidine-1-carboxylic acid 1-[4-(N,4-dimethylanilino)butanoyl]piperidine-2-carboxylate 1-[[4-chloro-2,5-difluoro-3-(phenylmethoxycarbonylamino)phenyl]methylsulfanyl]cyclopentane-1-carboxylic acid 1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)piperidine-3-carboxamide;dihydrochloride 2-[N-(4-chlorobutyl)-4,5-dimethyl-2-phenyldiazenylanilino]acetic acid N-[2,4-dihydroxy-3-[(1Z)-1-(methylamino)buta-1,3-dien-2-yl]phenyl]acetamide (1Z,3E)-4-[1-[(4-chlorophenyl)methyl]-5,6-dihydro-2H-naphthalen-1-id-4-yl]-N'-ethenyl-N-ethylidene-3-methylbuta-1,3-diene-1-carboximidamide;ethane 5-(2,4-dimethoxyphenyl)-N'-[(E)-1H-indol-3-ylmethylideneamino]-7-methoxy-1-benzofuran-3-carboximidamide 4-bromo-2-[[1,5-dimethyl-6-(piperidine-3-carbonyl)benzimidazol-2-yl]methoxy]benzoic acid (5Z)-2-(4-bromophenyl)imino-5-[[1,3-diethoxy-6-(trifluoromethyl)naphthalen-2-yl]methylidene]-1,3-thiazolidin-4-one [5-(aminomethyl)oxolan-2-yl]-[4-[6-chloro-7-fluoro-8-(fluoromethoxy)-1,5-naphthyridin-3-yl]piperazin-1-yl]methanone (3R,4S)-1-(5-bromo-2-methylpyridin-3-yl)-N,N-diethyl-4-hydroxypiperidine-3-carboxamide 2-[4-(difluoromethyl)phenyl]-6-fluoro-1H-benzimidazole 1-[1-(3-chlorophenyl)ethyl]pyridin-4-one 2-tert-butyl-4,6-bis(trifluoromethoxy)aniline 2-[4-(1H-imidazol-5-ylsulfonyl)phenoxy]-N,N-dimethylethanamine [(5aS,8aR)-1-[2-(4-fluorophenyl)ethyl]-2,2-dioxo-3,4,5a,6,8,8a-hexahydropyrrolo[3,4-f][1,4,5]oxathiazepin-7-yl]-piperidin-1-ylmethanone 3,5-dimethyl-4-oxo-2H-1,6-naphthyridine-7-carboxamide 2-[(5,6-dimethylpyridine-3-carbonyl)amino]-9-(4-hydroxycyclohexa-1,3-dien-1-yl)nonanoic acid 2-(4-ethylpiperidin-1-yl)-N'-hydroxypyrimidine-4-carboximidamide 2-[4-methoxy-5-(trifluoromethyl)pyrimidin-2-yl]benzenesulfonamide 3-[6-[4-(2,5-dichloropyridin-3-yl)piperazin-1-yl]hexanoyl]-7-hydroxy-1H-quinolin-2-one 4-chlorobenzenethiol;6,7-difluoro-2,4-bis(methoxycarbonyl)-1H-indole-3-carboxylic acid 4-[5-(2,3-difluorophenyl)-6-ethoxypyridin-3-yl]sulfonyl-2-methyl-2,7-naphthyridin-1-one N-cyclopentyl-2,6-difluorobenzenesulfonamide (2R)-N'-[4-chloro-3-(trifluoromethyl)phenyl]-2-[4-cyano-3-(trifluoromethyl)phenyl]-1-(2,2-dioxopropanoyl)piperidine-4-carbohydrazide 2-[1-(2,4-dichlorophenyl)ethenyl]aniline 6-[(3,4-dichlorophenyl)methylamino]-1-propylcyclohexa-2,4-diene-1-carbonitrile 4-(8,8-dimethyl-3,4a,5,7,9b-hexahydro-2H-pyrano[3,2-c]pyridine-6-carbonyl)benzoic acid 2-[[4,4-dimethyl-6-(4-nitrophenyl)-1,3,5-triazin-2-yl]sulfanyl]-N-(4-methoxyphenyl)acetamide 2,2-difluoro-N-[3-(4-methoxyphenyl)sulfanylpropyl]-3-(4-piperidin-1-ylpiperidin-1-yl)propanamide 7-[4-(2,5-dioxopyrrolidin-1-yl)cyclohexyl]oxyquinoline-8-carboxamide (2S)-4-methylsulfanyl-1-[3-phenyl-4-(pyridine-2-carbonyloxyamino)butyl]pyrrolidine-2-carboxylic acid N-[4-amino-3,4-dioxo-1-(1H-pyrrol-2-yl)butan-2-yl]-2-pyrazin-2-ylpyrazole-3-carboxamide 7-(4-chlorophenyl)-N,2-dimethyl-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide 2-(3,5-dimethylphenyl)-4-[1,3,4-thiadiazol-3-ium-3-yliminomethyl]-5-thiophen-2-yl-1H-pyrazole-3-thione 1,3-difluorobenzene;N-ethylethanamine;4-[5-methoxy-2-(trifluoromethyl)indol-1-yl]butanenitrile 6-[3-(4-methylphenoxy)azetidin-1-yl]pyridine-2-carboxylic acid [2-azido-5-(1H-indol-2-yl)phenyl]methanol N-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-1-cyanocyclopropane-1-carboxamide 2-[[4-[[5-bromo-2-(tetrazol-1-yl)phenyl]methoxy]piperidin-1-yl]methyl]-3H-thieno[3,2-d]pyrimidin-4-one (3Z)-6-fluoro-N,5-dimethylhexa-1,3,5-trien-2-amine;[3-[[4-(2H-tetrazol-5-yl)phenyl]methoxy]naphthalen-2-yl]methanimine N-[4-[2-chloroethylsulfonyl(methylamino)amino]naphthalen-1-yl]acetamide 2-(2,6-dioxopiperidin-3-yl)-4-[2-methoxyethyl(1,1,2,2,2-pentafluoroethyl)amino]isoindole-1,3-dione;propane 4-chloro-N,5-bis(4-chlorophenyl)-1,3-thiazole-2-carboxamide 2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-N-methoxyacetamide (2S)-N-[2,4-difluoro-3-(8-methoxy-1,7-naphthyridin-6-yl)phenyl]piperidine-2-carboxamide 3-bromo-N-[[(2R,6S)-2,4-dimethylmorpholin-6-yl]methyl]quinoline-7-carboxamide N-[5-cyano-2-methyl-4-(trifluoromethoxy)phenyl]-1,3,4,7-tetrahydropyrazolo[3,4-d]pyrimidine-6-carboxamide 5-(2,3-dichlorophenyl)-N-[[4-(trifluoromethylsulfonyl)phenyl]methyl]-7H-pyrrolo[3,2-d]pyrimidin-2-amine 2-[4-methyl-N-(1,3-thiazol-5-yl)anilino]decanoic acid 4-[2,3-difluoro-4-(trifluoromethoxy)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-tert-butyl-5-methyl-6H-[1,3]thiazolo[4,5-d]pyrimidin-7-one N-azido-3,5-bis(trifluoromethyl)benzamide 4-[3-(6,7-dimethoxyquinazolin-2-yl)oxyphenyl]-1H-imidazole-5-carboxamide (3R)-N-[2-[4-(furan-2-yl)piperidin-1-yl]ethyl]-5-phenyl-3,6-dihydro-2H-pyridine-1-carboxamide 3-bromo-7-methoxypyrazolo[1,5-a]pyrimidine 4-[(3S)-3-methylpyrrolidine-1-carbonyl]benzoic acid 2-[(5-bromothiophene-2-carbonyl)amino]-3,4-dihydro-1H-isoquinoline-4-carboxylic acid 5-(4-chlorophenyl)-2,3-dihydro-1H-tetrazolo[1,5-a]pyrimidine N-[(2S,3R)-4-(1H-indole-6-carbonylamino)-2,3-dihydro-1H-inden-2-yl]carbamate 4-[azido(ethoxy)methyl]-1-nitro-2-phenylbenzene 2-(aminomethyl)-5,6-ditert-butyl-4-[(E)-2-phenylethenoxy]phenol 4-(3,5-dimethoxyphenyl)piperazine 2-azido-1,3-bis[2-(trifluoromethyl)phenyl]propan-1-one 2-(1,3-benzothiazol-6-yl)-N'-hydroxy-1,5-dihydropyrazole-4-carboximidamide 5-[2,2-dimethoxyethyl(1-phenylpropan-2-yl)amino]naphthalene-2-sulfonic acid 5-bromo-4-[(4,6-dimethylcyclohexa-1,3-dien-1-yl)amino]-1H-pyrimidin-6-one 4-[5-fluoro-3-(piperidine-1-carbonyl)quinolin-2-yl]piperazine-1-sulfonamide 1,3-dibromo-5-chloro-4-[1-(trifluoromethoxy)ethyl]-2H-benzimidazole 2-[(3,4-dichlorophenyl)methylamino]-5,6,7,8-tetrahydroquinazoline-6-carboxylate N-(1,3-benzothiazol-2-yl)-2-(3-hydroxypyrrolidin-1-yl)acetamide 7-(4,8-dichloro-5,6,7,9-tetrahydroimidazo[1,2-a][1,4]diazepine-2-carbonyl)-5H-pyrrolo[3,2-d]pyrimidine-2-carbonitrile [4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carbonyl)morpholin-3-yl]methanol 6-(2,3-dihydro-1H-indene-2-carbonyl)spiro[1,4-dihydroquinoxaline-3,3'-piperidine]-2-one 3-[(1S,5R)-6,7-dimethoxy-2-azabicyclo[4.2.0]octan-2-yl]phenol 2-amino-5,6-dihydropyrrolo[1,2-a]quinoxaline-9-carboxylic acid N-[2,4-difluoro-3-[5-(furan-2-yl)pyrazolo[3,4-b]pyridine-2-carbonyl]phenyl]-1-benzothiophene-6-sulfonamide 2-[(5R)-4,7-dioxo-3-(2-phenylethylsulfanyl)-6H-pyrazolo[4,3-d]pyrimidin-5-yl]-N-prop-1-en-2-ylacetamide 2-(4-methoxybutyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine (2S,3R)-1-[4-[2-chloro-4-[(1S)-1-hydroxyethyl]phenyl]piperidin-1-yl]-3-methylpyrrolidine-2-carboxamide N-[1-[3,5-dimethyl-4-(4-phenylphenyl)cyclohexa-2,4-dien-1-yl]ethyl]benzenesulfonamide [(5Z)-5-[(3-bromophenyl)methylidene]oxolan-2-yl]phosphane 4-bromo-5-chloro-2-(4,6-dimethoxypyrimidin-2-yl)phenol N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methylideneamino]benzamide 2-[2-[[5,6-bis(4-methoxyphenyl)pyridazine-3-carbonyl]amino]ethyl]-1,3-thiazole-4-carboxylate 1,2-dichlorobenzene;N'-(cyclohexa-2,4-dien-1-ylmethyl)-N-[5-(2-oxo-3H-1,3,4-oxadiazol-5-yl)pentanoyl]ethanimidamide N-(4-azidonaphthalen-1-yl)-4-[(2,4-dichlorophenyl)methoxy]benzamide 3-amino-N'-[(1S)-1-cyanoethyl]pyrazine-2-carboximidamide 2-(hydroxymethyl)-6-[1,3-dioxo-4-(trifluoromethoxy)isoindol-2-yl]oxane-4,5-dione 2-[(2,5-dimethylphenyl)sulfonyl-(3-ethoxypropyl)amino]acetic acid 4-(5-aminopyridin-2-yl)piperazine-1-carboxylic acid 3-azidooxy-4,5,6-trifluorobenzene-1,2-dicarbonitrile 4-[1-(2-amino-6-oxo-5H-pyrimido[4,5-d]pyrimidin-4-yl)piperidin-3-yl]benzonitrile;ethane N'-(2,4-dimethylphenyl)sulfanyl-1-propylindole-3-carbohydrazide 2-(3,6-dihydro-2H-pyran-4-yl)-N-[1-hydroxy-5-(2H-triazol-4-yl)pentan-2-yl]pyridine-4-carboxamide 2-(cyclopropylmethylamino)-5,6,7,8-tetrahydroquinazoline-4-carbonitrile;hydrochloride N-[5,6-difluoro-1-(4-fluorophenyl)sulfonylbenzimidazol-2-yl]quinoline-8-carboxamide (2S)-6-[(1R,3aR,7aS)-5-hydroxy-2,3,3a,4,9,10,10a-octahydro-1H-cyclopenta[b]chromene-1-carbonyl]-N-methyl-1,2,3,4-tetrahydronaphthalene-2-carboxamide 2-cyclopropyl-N-(1H-imidazol-5-ylmethylideneamino)pyrazolo[1,5-a]pyrimidine-6-carboxamide 3-[(Z)-(5-aminosulfanyl-2-oxo-1H-indol-3-ylidene)methyl]-N,N-dimethylbenzamide 2-bromo-5-(1,3,4,7-tetrahydropyrido[4,3-b]indole-2-carbonyl)benzaldehyde 4-[3-(cyclopentanecarbonyl)-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-1-carbonyl]-N-methylbenzamide 1,2-diamino-4-[2-fluoro-3-methoxy-6-(trifluoromethyl)phenyl]-6-oxopyridine-3,5-dicarbonitrile 4-[5-(aminomethyl)-1,2,4-oxadiazol-3-yl]-6-ethoxy-2-fluoro-3-(1H-indazole-7-carbonylamino)benzoic acid (5E)-4,7-dimethyl-N-phenyldeca-5,8-dienamide 6-[1-[6,7-dimethoxy-2-(4-methylphenyl)quinazolin-4-yl]piperidin-3-yl]naphthalene-2-carboxylic acid (3-bromo-5,7,7-trimethylcyclohepta-1,4,6-trien-1-yl)-phenylmethanone 3-[(2Z,4E)-hepta-2,4-dienyl]-2-N-phenylimidazo[1,2-a]pyridine-2,8-diamine (1R,3S)-2-[4-chloro-N-[2-[3-[[6-(2-hydroxyethylcarbamoylamino)pyrimidine-4-carbonyl]amino]phenyl]ethyl]anilino]cyclohexane-1-carboxamide (2E)-3,7-dimethyl-6-oxo-N-[4-(trifluoromethoxy)phenyl]nona-2,8-dienamide 1-(3,4-dimethoxyphenyl)-6-methylheptan-2-ol 4-hydroxy-2,5-dimethyl-3-pent-1-ynylbenzoic acid (2R)-N,3-dibenzylhexan-2-amine 4-(3,5-dimethylphenyl)-2-phenylpyridine;1-ethynyl-2-fluoro-4-methylbenzene;N-[2-(3H-indol-6-id-5-yloxy)ethyl]formamide 3-(4-amino-2-oxopyrimidin-1-yl)piperidine-2,6-dione N-[3-fluoro-5-(2-pyridin-4-ylthieno[3,2-d]pyrimidin-4-yl)phenyl]propane-1-sulfonamide 6-bromo-2-methyl-4,5,7,8-tetrahydropyrazolo[1,5-d][1,4]diazepine;hydrochloride 3-[(2-acetamidophenyl)sulfonyl-aminoaminoaminomethyl]pyridine-4-carboxylic acid 2-[4,5-bis(2-methylpropyl)-1H-imidazol-3-ium-2-yl]pyridine;tetrafluoroborate 2-(3-fluorophenyl)-N-[4-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide N-[3-(5,6-diethylthieno[2,3-d]pyrimidin-4-yl)phenyl]-2-oxoacetamide 6-[(5-chlorothiophene-2-carbonyl)amino]-N-methyl-1H-indole-3-carboxamide 2-[4,5-dihydroxy-3-(2-methylpropyl)-6-oxopyran-2-yl]sulfanylacetaldehyde 3-[(2S,4S)-2-methyloxan-4-yl]oxybenzoic acid [(3Z)-4-acetylhexa-1,3,5-trien-2-yl]-bis(4-fluorophenyl)borane 6-amino-7-[(1,3-diethyl-5,5-dioxopyrrolidin-2-ylidene)methyl]-1H-quinolin-2-one 4-methoxycarbonyloxybenzoic acid;3-(5-oxo-2,7-dihydrothieno[3,4-d]pyrimidin-6-yl)propanoate N-[(4S)-3,4-dihydro-2H-chromen-4-yl]-2-(3-propanoylphenyl)acetamide N-(2,6-dichlorophenyl)acetamide;ethane 2-(4-hydroxyphenyl)imino-5H-quinazolin-7-one 2-[5-[(1R)-1-aminoethyl]-3-phenyl-1,2,4-triazol-1-yl]benzonitrile;hydrochloride 5-(5-chlorohexoxy)-7-ethylquinoline (5S)-3-[2,6-difluoro-4-(iodoamino)phenyl]-N-[1-(4-methoxybutanoyl)piperidin-4-yl]-1,3-oxazolidine-5-carboxamide N-[5-tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-5-oxo-1,4-dihydro-1,2,4-triazole-3-carboxamide 2-[1-[(6-bromoimidazo[4,5-b]pyridin-3-yl)methoxy]ethenyl]aniline N-[2-amino-5-(dimethylamino)phenyl]formamide 6-[4-[2-(4-methylphenyl)ethyl]-1,3-thiazol-5-yl]pyridine-2-carboxylic acid 2-chloro-6-[3-(4-chlorophenyl)propyl]-5,7-dihydropyrrolo[3,4-d]pyrimidine 2-[N-(2-bromophenyl)-3-methylsulfanylanilino]ethanol 5-(1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-inden-1-ol 1-(6,7-dihydro-4H-furo[3,2-c]pyridin-5-yl)-2-[[5-ethoxy-8-methyl-2-(oxan-4-yl)imidazo[1,2-a]pyrazin-3-yl]amino]-2-oxoethanesulfonamide 2-amino-6-[5-[1-(3,5-dimethylphenyl)propan-2-yl]-1,3-thiazol-2-yl]phenol 2-ethoxy-4,6-diiodobenzaldehyde (1S,2R)-N-[4-[6-amino-5-(difluoromethyl)pyridin-3-yl]phenyl]-2-(fluoromethoxycarbonyl)cyclopropane-1-carboxylic acid 6-methyl-2-[1-(4-methylsulfonylphenyl)propan-2-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine 2-[(1E,3Z)-1-(cyclohexa-1,5-dien-1-ylmethylideneamino)penta-1,3-dienoxy]benzonitrile N-[(E)-1-(1H-benzimidazol-2-yl)ethylideneamino]-4-hydroxypyrrolidine-3-carboxamide 2-(4,5-dimethylpyridin-2-yl)-5-(1H-imidazol-5-ylmethyl)pyrazine (2E)-N,2-dimethyl-3-[[4-(4-methylphenyl)piperidin-1-yl]sulfonylamino]penta-2,4-dienamide;ethane N-[3-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)phenyl]-N'-ethyl-2-(3-fluorophenyl)propanediamide 7-(3,4-dihydroquinoline-8-carbonyl)-2-ethyl-6,8-dimethoxy-3,4-dihydroisoquinolin-1-one 5-methyl-3-(4-methylcyclohexyl)oxy-7H-pyrrolo[2,1-c][1,2,4]triazine 3-amino-N'-[[3-chloro-5-(trifluoromethyl)phenyl]carbamoyl]benzenecarboximidamide N-methyl-4-oxo-6,7,8,9-tetrahydroquinolizine-1-carboxamide N-[2,4-difluoro-3-[5-(1-pyridin-2-ylindazol-6-yl)-1,2,4-oxadiazol-3-yl]phenyl]propane-1-sulfonamide 5-[3-(cyclopropylmethoxy)-4-fluorophenyl]-6-ethenylpyrimidine-2,4-diamine 4-[N'-(6,7-dimethoxyquinazolin-4-yl)carbamimidoyl]benzamide 6-[1,2-dimethyl-4-(5-pyrrolidin-3-yloxypyridin-2-yl)piperazin-1-ium-1-yl]-7H-purine 2-[5-carbamoyl-9-(3-chlorophenyl)carbazol-4-yl]oxyacetic acid (5Z)-5-[(4-ethylphenyl)methylidene]-2-imino-1,3-thiazolidin-4-one N-[4-fluoro-3-(trifluoromethyl)phenyl]-2-[[6-oxo-4-(propan-2-ylsulfanylmethyl)-1H-pyrimidin-2-yl]sulfanyl]butanamide 7-[3-fluoro-4-[(2S)-2-methylpyrrolidin-1-yl]phenyl]-6,8,9,10-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine 5-(4-methoxyphenyl)-3,6-dihydro-1H-pyrrolo[2,3-b]pyrrole 2-[(3-ethylphenyl)methoxy]-1-(4-heptan-4-ylpiperazin-1-yl)ethanone 1-[(6-chloropyridin-3-yl)methylamino]-2,5-dihydropyrido[3,4-e][1,2,4]triazine-7-carboxamide (2E,5Z)-5-[(2-bromophenyl)methylidene]-3-[(2,4-dichlorophenyl)methyl]-2-hydroxyiminocyclopentan-1-one (3R)-5-amino-1-[6-azido-2,4-bis(trifluoromethyl)pyridin-3-yl]-3-tert-butylpyrazole-4-carbonitrile 4-[2,3-difluoro-6-(methoxymethyl)-4-nitrophenoxy]butanal (2S)-N,3-dimethylbutanamide;7-(2,6-dimethylpyridin-4-yl)-5-[1-[(6-fluoropyridin-3-yl)methyl]pyrazol-4-yl]pyrrolo[1,2-b]pyridazine (4Z)-N-tert-butyl-2,3,7-trimethyl-5H-1-benzazonin-6-imine 2-[4-[(3R)-1-ethylpiperidin-3-yl]oxyphenyl]indazole 3-(3,4,5-trimethoxyphenyl)piperidine-2-carboxamide 2-(3,5-dimethylphenyl)sulfanyl-5-[(4-nitrobenzoyl)amino]benzoic acid N-benzyl-N-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-ylmethyl)-2-pyrrolidin-1-ylpropanamide (E)-3,5-dihydroxy-2-methyl-6-naphthalen-2-ylhex-5-enal N-[[2-(3,5-dimethylpyridine-4-carbonyl)-2-azaspiro[4.5]decan-8-yl]methyl]pyridine-2-carboxamide;hydrochloride 1-[4-(dimethylamino)phenyl]-6-methyl-4H-pyridazin-3-one 4-[[1-(6,7-dimethoxyquinazolin-4-yl)piperidin-3-ylidene]-ethylamino]benzonitrile 2-(4-bromophenyl)-N-tert-butyl-5-(3-methoxyphenyl)-1H-pyrrole-3-carboxamide 6-(3,3-dichloroprop-2-enoxy)-7-methyl-1,4-benzothiazin-3-one (2S)-3,4-dimethyl-1-phenyl-N-(pyridin-3-ylmethylideneamino)-5-sulfanylidenepyrrolidine-2-carboxamide 3-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]-N',N'-bis[1-(N,3-dimethylanilino)ethenyl]benzenecarboximidamide 4-[3,5-bis(trifluoromethyl)phenyl]sulfonylpiperazine-1-carboximidamide 1-cyclopropyl-5-[(3S,4R)-3-hydroxypiperidine-4-carbonyl]pyridin-2-one;hydrochloride 4-(6-ethynyl-1,3-benzothiazol-2-yl)phenol (7-fluoro-2,3-dihydroindol-1-yl)-[6-methoxy-4-[[2-methyl-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]pentanoylamino]pyridine-4-carbonyl]amino]-2H-pyrazolo[1,5-a]pyridin-3-yl]carbamic acid 2-[5-[2-amino-5-(1,3-dioxolan-2-yl)pyrimidin-4-yl]-6-methoxypyridin-2-yl]-N-propylacetamide 6-methyl-4-(trifluoromethoxy)quinoline 3-[(7-bromopyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]propane-1-sulfonic acid (3R,5S)-4-azido-3,5-dibenzylmorpholine 1-[5-(2-methoxypyridine-3-carboximidoyl)thiophen-3-yl]ethanone N-(6-oxobenzo[c]chromen-3-yl)propanamide 1-[5-(2-phenylethynyl)pyridin-3-yl]piperidine-3-carboxamide 4-(1,3-benzothiazol-6-yl)benzene-1,2-diamine 4-tert-butyl-1,3-bis(phenylsulfanyl)imidazolidine-2-thione 1-[4-[2-(dimethylamino)ethyl]phenyl]-6,7-dihydropyrrolo[2,3-c]pyridine-5-carboxylate N-[(3R)-4,5,6,7-tetrahydro-1-benzothiophen-3-yl]cyclopropanesulfonamide 1-(2,3-dihydro-1H-inden-2-yl)-6-propan-2-yl-4-thiophen-2-yl-[1,2]oxazolo[5,4-d]pyrimidine (6R)-6-tert-butyl-2-[(3-ethoxyphenyl)methylideneamino]-N,4-dihydroxy-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-9-carboxamide N-(3,4-dimethoxyphenyl)-2-[6-ethyl-7-(3-fluorophenyl)-2-oxo-1,3-dihydroimidazo[1,2-b]pyrazol-3-yl]acetamide 3-chloro-5-(1H-indol-4-yl)phenol 2-[N-(carboxymethyl)-3,5-dichloroanilino]propanoic acid [4-[3,5-difluoro-2-(trifluoromethyl)phenyl]phenyl]-hydroxyazanium N'-(1-benzothiophen-5-yl)benzenecarboximidamide N-(2,6-dimethylphenyl)-4-[[5-(1H-indol-3-yl)-4-(oxolan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide 5-amino-2-butoxy-8H-[1,2,4]triazolo[4,3-c]pyrimidin-7-one 4-[3-(trifluoromethyl)phenyl]-2,5-bis(sulfanylidene)imidazolidin-4-one 3-[(2R)-1-[(2S)-2-methylpyrrolidine-1-carbonyl]-4,5-dihydro-2H-indol-6-yl]-N-propan-2-ylbenzamide (2R)-3-[1-(1-azidonaphthalen-2-yl)sulfonylindol-6-yl]-2-methoxypropanoic acid 5-(1,3-benzodioxol-4-yl)-6-[3-fluoro-4-[3-(trifluoromethoxy)phenyl]phenyl]sulfonylhexan-2-one 2-[(4R)-1-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]benzoic acid 2-[5-chloro-1-(6,7,8,9-tetrahydro-5H-carbazole-4-carbonyl)indol-3-yl]propanamide (2S)-1,1,1-trifluoro-3,4-dihydro-2H-phenanthrene-2-carboxylic acid N-[4-cyano-2-(trifluoromethyl)phenyl]-1-methyl-5-oxopyrrolidine-3-carboxamide N-(1,3-benzodioxol-5-ylmethyl)-6-[2-hydroxyethyl(methyl)amino]-1H-indole-3-carboxamide 7-N,2-bis(3-chlorophenyl)-5-N,4-dimethyl-3H-1,4-benzoxazine-2,5-dicarboximidamide 3-azido-2,6-dihydropyrrolo[2,3-c]carbazole N-cyclohexyl-4-[(2E)-2-ethenylpenta-2,4-dienoxy]pyridin-3-amine;ethane (4S)-4-methyl-1,3-diphenylimidazolidin-2-one 4-[1-amino-2-[6-(3,5-difluorophenyl)pyridin-2-yl]-2-cyclopropylethenyl]-N-methoxyaniline 6-(2,3-dihydroindol-1-yl)pyridazine-4-carbonitrile 3-[2,5-dimethyl-1-(3-methylbut-2-enyl)pyrrole-3-carbonyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carboxamide 1-cyclopropylsulfonyl-3,5-dimethylpyrrolo[2,3-b]pyridine (2S,5R)-5-[[[1-(cyclohexa-1,3-dien-1-ylmethoxycarbonylamino)-4-fluorobutan-2-yl]amino]methyl]pyrrolidine-2-carboxylic acid 1-[(4aS,8R)-6-(3-methoxyphenyl)sulfonyl-4a-methyl-8,9,10,11-tetrahydropyrano[2,3-h]isoquinoline 3-[(2Z,4E)-hepta-2,4,6-trien-4-yl]oxy-1,5-dimethylpyrazole 4-chloro-1-(2,6-difluorophenyl)-N-[3-methyl-5-(trifluoromethyl)phenyl]pyrazole-3-carboxamide (4Z)-2-[6-[ethyl(2-hydroxyethyl)amino]pyridin-3-yl]-4-hydrazinylidene-8-methoxythieno[2,3-c]quinoline-5,7-dione N-[2-(azetidine-1-carbonyl)-5,6-dihydrofuro[3,2-b]pyridin-4-yl]cyclopropanecarboxamide N-[(3S,7R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-1-butan-2-yltriazole-4-carboxamide 2-(4-bromo-6,7-dichloro-1H-benzimidazole-5-carbonyl)cyclohexan-1-one [(2S)-2-[methyl-(5,6,7,8-tetrahydroquinolin-8-ylamino)carbamoyl]pyrrolidine-1-carbonyl]-methylidyneazanium 2-[(3,4-dichlorophenyl)methyl]-6-(4-piperazin-1-ylsulfonylphenyl)imidazo[1,2-a]pyrazine 2-tert-butyl-7-[(4-cyclohexyloxy-3-methoxyphenyl)methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one (2S)-1-N,2-N-bis[4-(1H-imidazol-5-ylmethylamino)phenyl]benzene-1,2-dicarboxamide 1-(cyclohexylmethyl)-3,7-difluoroquinolin-4-one 1-[3-(2,3-dihydropyridin-5-yl)phenyl]-N-methylethenamine 2-amino-6-chloro-3-fluoro-N,N'-diphenylbenzenecarboximidamide 7-methyl-2,3-diphenyl-2H-benzo[g]quinoxaline 2-(4-methylphenyl)-5H-pyrido[3,2-b]indole 1-[(3R)-1,4-dihydroxy-5-phenylpentan-3-yl]pyrrolidine-2-carboxylic acid 4-(2-chloro-6-methoxyphenyl)-7-fluoroquinoline 1-[2-(3-ethylhexan-2-ylamino)pyrimidin-5-yl]ethenol ethane;4-[5-methyl-7-(2,4,6-trifluorophenyl)heptanoyl]benzaldehyde 2-(N-butanoyl-4,5-dimethyl-2-phenyldiazenylanilino)acetamide 3-amino-N'-[2,4-dimethyl-6-(2,4,5-trifluorophenyl)phenyl]pyrrolidine-1-carboximidamide 5-[7-[(Z)-1,3-diaminopent-2-en-4-ynylideneamino]imidazo[1,2-a]pyridin-3-yl]pyridine-3-carbonitrile ethane;3-ethyl-2,4-dimethoxyphenol 1-azido-5,7-dimethoxy-3-[2-(trifluoromethyl)phenyl]sulfonylnaphthalene 2-(4-bromophenyl)benzenesulfinate [5-chloro-2-(hydroxymethyl)phenyl]methylidene-[3-[[1-[1,3-dioxobenzo[de]isoquinolin-2-yl]-3-methoxypropan-2-yl]amino]-4-methylsulfanylbutyl]azanium 1,2-diethyl-N'-methanimidoyl-5,6-dimethoxyindole-3-carboximidamide N-butyl-5,6-diphenylpyrimidin-2-amine;[3-methoxy-4-(2H-tetrazol-5-yl)phenyl]-piperazin-1-ylmethanone (5S)-2-[2-chloro-5-(trifluoromethyl)phenyl]imino-5-ethoxy-1,3-thiazolidin-4-one 2-(2-azido-5,6,7,8-tetrahydronaphthalen-1-yl)thiophene 4-[[4-(2,6-dimethylpyridin-4-yl)piperidin-1-yl]methyl]-3-ethoxyphenol 2-(4,5-dichloro-2,3,6-trimethylphenyl)propanedioic acid 2-[4-methyl-3-(1,6,8-triazatricyclo[7.3.0.03,7]dodeca-9,11-dien-8-yl)phenyl]pyridine-4-carboxylic acid 4-[1,2,3-trimethyl-7-(piperidin-4-ylmethoxy)indolizine 4-chloro-3,5-bis(4-hydroxyphenyl)-2H-1,3-oxazole-2-carboxylic acid 5-bromo-4-methyl-2-[(2Z)-penta-2,4-dien-2-yl]sulfonylpyrimidine 2-(4-chlorophenyl)-N-[4-[5-fluoro-6-methoxy-1-(3,3,3-trifluoropropyl)benzimidazol-2-yl]cyclohexa-2,4-dien-1-ylidene]acetamide 1,4-diphenylpiperazine;hydrate 3-(1,3-benzothiazol-2-yl)-4H-chromene-6-carboxylate N-[[4-(3,5-dimethylpyridin-2-yl)morpholin-2-yl]methyl]pyrimidin-2-amine;formic acid 3-[5-[[4-[(Z)-1-amino-2-hydrazinylethenyl]piperidin-1-yl]methyl]-6-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione 3-[2,5-dihydroxy-6-methyl-4-(methylideneamino)cyclohexa-1,3-dien-1-yl]oxycarbonylphthalic acid 5-chloro-N'-[(3S)-1-oxo-3,4-dihydroisochromene-3-carbonyl]pyrazine-2-carbohydrazide 3-chloro-5,7-dimethyl-N-[(6R)-2-oxoazepan-1-yl]quinoline-6-carboxamide (4S,5R)-2-benzoyl-4-methyl-1,3-dioxolan-2-one;methanol N-[5-(azidomethyl)pyridin-2-yl]-5,7-dichloroquinazolin-4-amine 1-[5-(2,6-difluorophenyl)pyridin-2-yl]-7H-pyrazolo[3,4-d]pyrimidine-6-thione N-[3-ethyl-4-methoxy-5-(2-nitropyridin-3-yl)phenyl]-3-(trifluoromethoxy)aniline [3-[4-(4-oxocyclohexyl)piperidine-1-carbonyl]phenyl]azanium 4-(3-ethenyl-2,6-dimethoxyphenyl)-N,N-bis[2-(2-hydroxybutoxy)propan-2-yl]aniline 5-chloro-2,4-dimethoxy-N-[6-(propanoylamino)pyridin-3-yl]benzamide (4-methyl-2,5-diphenylpyrazol-3-yl)phosphonic acid 2-[N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-methoxyanilino]octanoic acid 2-[4-(diethylamino)phenyl]-5-(2H-indol-3-yl)-4H-1,2,4-triazol-3-one 5-methoxy-N-[(1E)-2,4,6,7-tetrachlorocycloocta-1,3,7-trien-1-yl]-1H-indazole-3-carboxamide 1,3-dimethylcyclohexane;ethane;(7E)-2-methyl-9-[(4Z,6Z)-5-propan-2-ylidenenona-4,6-dien-2-ylidene]-10H-phenanthridine 2-[5-(8,9,10,11,15,16,18-hexazatetracyclo[8.7.0.02,6.012,17]heptadeca-1(17),2,4,6,8,13,15-heptaen-11-yl)pyridin-3-yl]acetonitrile 4-benzylsulfanylcycloheptane-1,3-dione N-(5-bromothiophen-2-yl)sulfonylacetamide 2-(2,5-dimethoxyphenyl)-1-[3-methylsulfanyl-4-(pyrrolidine-1-carbonyl)-5,6,7,8-tetrahydroquinolin-8-yl]ethanone ethane;2-(4-ethyl-3,5-dimethyl-1H-pyrazol-2-ium-2-yl)-N'-propan-2-ylidenebenzenecarboximidamide 1-[3-(difluoromethoxy)phenyl]-6,7-dihydro-5H-cyclopenta[d]pyridazine 2-(2,4-dichlorophenyl)-5-methylpyrazine;ethane N-[(E)-1-aminoethylidenecarbamothioyl]benzamide 2-(1,3,5-trimethylpyrazole-4-carbonyl)pentanedioic acid 5-[(4R)-7,11-dihydropyrrolo[2,1-c][1,4]benzodiazepine-6-carbonyl]-2-methoxybenzaldehyde (2S)-1-[3,5-difluoro-4-(2-hydroxypropan-2-yl)phenyl]-2-(4-methoxyphenyl)pyrrolidine-3-carbonitrile 1-bromo-2-(3-chloropropoxy)-4-methylbenzene 2-[5-azidooxy-6-(trifluoromethyl)pyridin-3-yl]ethanol [2-(4-ethoxyphenyl)sulfanylpyrrolidin-1-yl]-(4-methylpiperazin-1-yl)methanone 1-[2,6-di(propan-2-yl)phenyl]-5H-pyrazolo[4,3-c]pyridine 1-[4-(5-azido-2,3-dimethylbenzimidazol-4-yl)phenyl]ethanone 1-[4-(azidomethyl)phenyl]indole [2-chloro-6-(trifluoromethyl)pyridin-4-yl]-pyrrolidin-1-ylmethanone 3-azido-7-chloro-2,6-naphthyridin-1-amine 3-azidooxysulfonyl-6,7-difluoronaphthalene-2-sulfonic acid 2-(4-acetamidobutanoylamino)benzenesulfonic acid 6-(4-aminopyridin-3-yl)-2H-1,4-benzoxazine-3-carboxylic acid;cyclohexane 2-(2-bromo-4,5-dimethoxyphenyl)-N,1,3-triphenylimidazolidine-2-carboxamide 2-(cyclopenten-1-yl)-N'-hydroxypyrimidine-4-carboximidamide 2-chloro-N-methyl-5,6-diphenylpyrimidine-4-carboxamide 2-[4-(carbamoylsulfamoyl)-N-methoxycarbonylanilino]acetic acid 3-[2-(2,5-dimethylpyrazol-3-yl)ethoxy]-N'-hydroxypyrazine-2-carboximidamide 3-(6,7,8a,9,10,11-hexahydrobenzo[d][1]benzazepin-5-yl)-N-methylpropan-1-amine 1-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl)-7-methoxy-3-phenylquinoxalin-2-one (3S)-1,2-dibenzyl-6-[4-[2-methoxyethyl(pyridin-2-ylmethyl)amino]butyl]piperidine-3-carboxylic acid 3-[(5-methoxyfuran-2-yl)methyl]quinazolin-4-one 3-[(3,4-dimethoxyphenyl)methyl]-6-(furan-2-yl)-1H-pyrimidine-2,4-dione (4-bromo-2-iodophenyl)methanol 3-ethylsulfanyl-6-(1-methoxyethenyl)pyridazine;N-(2,4,5-trichlorophenyl)acetamide 6-[2,3,5-trihydroxy-4-(hydroxymethyl)phenyl]hexanoic acid 2-(4,4-difluoro-1-methylpiperidine-3-carbonyl)benzoic acid N-[4-(2,3-dichloro-7-methoxyquinoline-6-carbonyl)-1,3-thiazol-2-yl]butane-1-sulfonamide 1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]piperazine-2-carboxylic acid 1-(2,4-difluorophenyl)sulfonyl-3-methoxypyrazolo[3,4-c]pyridine 5-[(3S)-1,3-dimethyl-6-propan-2-ylpiperidin-3-yl]-7-methoxy-3H-imidazo[4,5-b]pyridine;ethane N-(3,5-dichlorophenyl)-1-ethylsulfonylpyrrolidine-2-carboxamide 2-[5-methyl-4-(oxolan-3-yl)-1,2,4-triazol-3-yl]pyridine 6-chloro-2-(3-methylsulfonylphenyl)quinoline 2-[7-(1,3-benzoxazol-5-yl)pyrido[4,3-d]pyrimidin-2-yl]oxy-N-methylethanamine;ethane 6-[[(1R)-5-phenylpentyl]amino]hexane-2,3-dione (3-phenylmethoxyphenyl)phosphane 3-aminosulfanyl-N'-[2,6-difluoro-4-(trifluoromethoxy)phenyl]benzohydrazide;hydrochloride ethane;[5-methyl-2-(4-pent-1-ynylphenyl)phenyl]phosphane 6-hydroxy-N-[4-(pyridin-3-ylsulfanylamino)phenyl]-2,3-dihydroindole-1-carboxamide [1-(2,6-dichlorophenyl)sulfonylpiperidin-3-yl]methanamine 4-[1,3-benzodioxol-5-yloxy(2H-pyran-2-yl)amino]-N-(2,6-difluorophenyl)benzamide 4-(2,6-dimethylpyridin-3-yl)-5-methoxycarbonyl-6-[1-(pyridine-2-carbonyl)piperidin-3-yl]-2,3-dihydropyridine-1-carboxylic acid 1-(3-bromopyridin-4-yl)-N,6,7-trimethoxyisoquinoline-4-carboxamide 2-(1,3,4,6,7,8,9,10,11,12,14,15-decahydrocyclopenta[a]phenanthren-16-yl)ethanol 1-[(4-cyclopropylphenyl)methyl]pyrrolidine;N-(2,3-dihydro-1H-inden-5-ylsulfonyl)formamide 3-amino-N-(4,5-dihydroimidazol-1-yl)-6-(2-hydroxyphenyl)pyrazine-2-carboxamide N-(1-methylpiperidin-4-yl)-N'-[4-[2-(3-methylpyridin-2-yl)ethenyl]phenyl]butanediamide 1-[2-(1,3-dihydroisoindol-2-yl)ethoxy]cyclobutan-1-amine 5-[4-(methylamino)piperidine-1-carbonyl]-3H-1,3,4-thiadiazol-2-one 3-(1-azido-1H-inden-2-yl)-6-phenylhexanenitrile (2S)-3-(4-methylphenyl)sulfonyl-2-[4-(pyridine-2-carbonyloxy)phenoxy]butanoic acid N-[3,4-dichloro-2-(propan-2-ylsulfamoyl)phenyl]piperidine-3-carboxamide 2-[4-[2,6-dichloro-3-(4,5-dihydrobenzotriazol-1-yl)phenoxy]phenyl]acetonitrile (3E,5Z)-1-amino-5-bromo-7-ethylsulfonyl-N'-methylidene-2-oxo-4-phenylpyrrolo[3,2-c]quinoline-3-carboximidamide 2-ethyl-4,6-dimethoxyquinoline 5-[2-(diethylamino)pyridin-3-yl]-1,3-benzoxazol-4-amine 4-(2-methylbutoxy)carbonylbenzoic acid 1-(4-chlorophenyl)-5-[[2-fluoro-6-methoxy-4-[2-(3,3,3-trifluoropropylamino)pyrimidin-4-yl]phenoxy]methyl]-3-methylpyrazole-4-carbonitrile 1-(3,4-difluorophenyl)sulfonyl-N-[(2R)-5-methyl-4-oxo-7-piperazin-1-yl-2,3-dihydro-1H-1,5-benzodiazepin-8-yl]piperidine-2-carboxamide 2-[4-[1,3-bis(sulfanyl)propoxycarbonyl]phenyl]acetic acid 1-N,1-N'-dicyclohexyl-2-N-phenylbutane-1,1-diamine 3-[[[4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]benzoyl]amino]carbamoyl]benzoic acid 4-bromo-3-(bromomethyl)pyridine N-cyclobutyl-2,4,6-trimethylbenzamide 2-ethyl-6-[4-(4-propoxyphenoxy)phenyl]pyridine 2-[2-(furan-3-yl)pyridine-4-carbonyl]spiro[6,7-dihydropyrrolo[1,2-a]pyrimidine-8,3'-pyrrolidine]-5-one;2,2,2-trifluoroacetic acid 1-[4-methyl-3,5-bis(methylamino)phenyl]ethanone [5-(4-fluorophenoxy)-1,2-oxazol-3-yl]-(4-methoxyphenyl)methanone 2,3-dimethyl-5-[4-(trifluoromethoxy)phenyl]-1H-indole 5-[4-(2,3-dichlorophenyl)piperazine-1-carbonyl]-1H-pyrrole-2-carbonitrile 1-[2-(4-methylcyclohexyl)oxyethyl]pyrazolo[3,4-c]pyridine 1-[3-(7-chlorospiro[2H-indole-3,4'-oxane]-5-yl)oxypropyl]imidazolidine-2,4-dione 3-[(4-fluorophenyl)methyl]-5-(hydroxymethoxymethylidene)-2,6-dioxopyrimidine-4-carboxylic acid N-azido-2-[[4-fluoro-3-(trifluoromethyl)phenyl]methoxy]pyridine-3-carboxamide N-[5-(difluoromethyl)-1H-pyrazol-3-yl]-2,6-difluoro-4-[7-hydroxy-8-(trifluoromethoxy)quinazolin-4-yl]benzamide 2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-3H-quinazolin-4-one 1-[2-(4-hydroxy-3,5-dimethylphenyl)pyridin-4-yl]ethanone 5-(3,5-difluorophenyl)-1-[(2R)-oxan-2-yl]indazole 5-azido-4-(2,4-dichlorophenyl)-1H-pyrazole (Z)-4,4-dimethylpent-2-ene;3-[2-(3-ethylheptan-3-yl)phenyl]pyridine 1-azidosulfanyl-3,5-dichlorobenzene 6-bromo-N,2-dimethylquinazolin-4-amine 2-[4-(3-bromocyclobutyl)-1H-benzimidazol-2-yl]-N,N-dimethylethanamine 6-chloro-7,8-dimethoxy-4H-1,3-benzodioxine 2-[5-(1H-pyrazol-4-yl)pyridin-3-yl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione 5-[3,5-difluoro-4-(trifluoromethyl)phenyl]sulfonyl-2-methoxypyridine-4-carbonitrile 4-[(6-fluoro-1H-indazol-5-yl)amino]cyclohexan-1-ol 2-azido-4,5-diphenylpyrazole 5-chloro-N'-hydroxy-1H-indole-2-carboximidamide 4-[(2Z,5S)-2-[(E)-3-methylbutan-2-ylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]benzenesulfonamide 3-methyl-4,5,6,7-tetrahydrobenzo[d][1]benzazepine 5-[3-(1,2,3,6-tetrahydropyridin-4-yl)phenyl]pyrimidine 4-[(1R,2S)-2-cyclohexylcyclopropanecarbonyl]benzaldehyde 1-[(2-methylpropan-2-yl)oxy]pyrene N'-(3,5-difluorophenyl)-2,2-dimethylpropanehydrazide N-[(E)-1-cyclohexa-2,4-dien-1-ylidene-3-hydroxyprop-1-enyl]benzamide 4-[1,1,2,3,3,3-hexafluoropropyl(1,3-thiazol-5-yl)amino]butan-1-ol N-[6-(2,4-difluorophenoxy)pyridine-3-carbonyl]morpholine-4-carboxamide 1-[(2E)-4,5-dimethylhexa-2,4-dien-3-yl]sulfanyl-2-phenylbenzene 2-[4-chlorobutyl(phenacyl)amino]benzenesulfonic acid 3-[(Z)-1,2-bis(benzenesulfonyl)but-2-enyl]pyridine 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazol-1-ium;iron(2+);dichloride (E)-3-[2-methoxy-5-(trifluoromethyl)phenyl]-2-sulfanylprop-2-enoic acid (2S)-N,3-dimethyl-1-(6-oxo-2-pyridin-4-yl-1H-pyrimidine-5-carbonyl)pyrrolidine-2-carboxamide 6-chloro-N,5-dimethyl-2,3,4,9-tetrahydro-1H-carbazole-1-sulfonamide 1-[5-chloro-2-(3-methoxyanilino)phenyl]butan-1-ol;ethane 6-chloro-N-[2,4-difluoro-5-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]phenyl]pyridine-3-carboxamide 2-azido-3,4,6,7-tetramethylthiochromene 4-(3-azidopyridin-2-yl)oxybenzonitrile 2-methyl-5-(1,3-thiazol-2-yl)benzenesulfonamide 2-(4-chloroanilino)-1,3-diethylbenzimidazol-1-ium-5-carboxylate 4-[5-(2-aminopyrimidin-4-yl)imidazo[1,2-c]pyrimidin-8-yl]benzaldehyde;methanamine 2-(4-chlorobutyl)isoindole-1,3-dione 1-(4,6-dimethylpyrimidin-2-yl)-3-[(Z)-[3-fluoro-4-[1-[4-(trifluoromethoxy)phenyl]-1,2,4-triazol-3-yl]phenyl]methylideneamino]thiourea 4-amino-2-[2,3-bis(4-methylphenyl)propanoyl]-6-methoxycarbonylbenzoate 5-(3,4-difluorophenyl)sulfonyl-N-[(1R,2S)-2-hydroxycyclooctyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide N-(4,5-difluorocyclohexa-1,3-dien-1-yl)-6-methoxy-7-[[2-(1,3,4-oxadiazol-2-yl)phenyl]methoxy]quinoline-3-carboxamide N'-hydroxy-5,6-dihydroimidazo[2,1-b][3]benzazepine-11-carboximidamide [(2S,4R)-1-[(5-bromo-3H-thiadiazol-2-yl)methyl]-4-fluoropyrrolidin-2-yl]methanol 2-ethyl-1,3-bis[2-(4-methoxyphenyl)ethynyl]benzene 1,5-bis(ethylsulfanyl)anthracene [4-(1H-imidazol-2-ylmethylamino)piperidin-1-yl]-[5-methoxy-6-(quinolin-8-ylmethoxy)pyridin-3-yl]methanone 2-(cyclohexa-1,5-dien-1-ylamino)-7H-purine-6-carbonitrile 3-(1H-benzimidazol-2-yl)-N-ethyl-6,7-dihydro-5H-cyclopenta[c]pyridine-7-carboxamide 5-[3,4,6-tris(hydroxymethyl)pyridin-2-yl]sulfanylpentanenitrile 5-[4-(6-aminopurin-9-yl)butoxy]-2,3-dihydro-1H-indene-1,2-disulfonate 4-[4,5-bis(2-methoxyethyl)-1H-imidazol-2-yl]phenol N-[[1-(4-ethylphenyl)-2,6-difluoro-3H-azepin-4-yl]methylidene]hydroxylamine 6-[(4,5-dimethylpyridin-2-yl)amino]-7-nitro-3H-quinazolin-4-one N-[[(4aS,5S)-8-(3-chloro-5-fluorophenyl)sulfonyl-9-cyclopentyl-2,4,4a,5-tetrahydropyrano[3,2-c]quinolin-5-yl]methyl]propanamide 3-[(3,4-dimethoxyphenyl)methylidene]-2-methyl-5-methylsulfanyl-1H-indole 2-methyl-5-[(2Z)-4-methylidene-1,3,6,8-tetrahydrocyclohepta[b]pyrrol-7-yl]benzaldehyde 2-[6-chloro-1-(cyclopropylmethoxy)naphthalen-2-yl]benzo[g][1,3]benzothiazole 4-[1-(3-fluorophenyl)imidazol-2-yl]-5,6,7,8-tetrahydroisoquinoline;dihydrochloride 1-(2-aminophenyl)-3-hydroxydodecane-5,6-dione 5-chloro-6-(2,4,5-trimethylphenyl)-1H-imidazo[4,5-b]pyridine 2-[3,5-bis(trifluoromethyl)phenyl]-1-ethoxyethanol (E)-N'-(4-aminonaphthalen-1-yl)-3-pyridin-2-ylprop-2-enimidamide N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]-1,7-naphthyridine-6-carboxamide 2-[3-(1-pyridin-3-ylsulfinylcyclopropyl)-5-(trifluoromethyl)phenyl]acetic acid 4-methoxy-N'-[2-(3,5,6-trimethylpyridin-2-yl)ethyl]benzenecarboximidamide (E)-3-[3,5-difluoro-4-[7-[(2-methylcyclopentyl)amino]heptyl]phenyl]-N-hydroxyprop-2-enamide N-[4-(1-benzyltriazol-4-yl)phenyl]sulfanyl-2,3-dihydro-1H-indole-7-carboxamide 2-ethyl-N,4,5-trimethoxybenzamide N-[5-chloro-4-(2,6-dimethoxyphenyl)pyridin-3-yl]-1-ethoxy-N',4-dimethylbenzenecarboximidamide 5-benzyl-N-[4-fluoro-3-(1,2-oxazol-3-yl)phenyl]pyrazine-2-carboxamide 3-[(2R,4R)-2-phenyloxan-4-yl]oxypyridine 1-[4-(benzenesulfinyl)phenyl]-2,6-difluoro-3-(trideuteriomethyl)benzene N-[(3S,5R)-5-hydroxy-6-(quinoline-4-carbonylamino)hexan-3-yl]-1H-indole-2-carboxamide 2-amino-3,5-dimethyl-6-(trifluoromethoxy)benzonitrile 4-[(3S)-4-[2-(oxolan-3-ylmethoxy)ethyl]morpholin-3-yl]benzamide 2-azido-N-[(3,4-dichlorophenyl)methyl]-5-hydroxy-6-oxo-1H-pyrimidine-4-carboxamide 6-methoxy-N-[2,4,7-trioxo-8-[(3R)-piperidin-3-yl]oxy-3H-pteridin-1-yl]pyridine-3-carboxamide;hydrochloride 2-[2-amino-5-(4-methoxyphenyl)-1,3-thiazol-4-yl]acetamide N-[5,6-dihydroxy-2-[4-(trifluoromethyl)phenyl]benzimidazol-1-yl]benzamide N-[3-[2-(3,4-dichlorophenoxy)ethyl-propylamino]propyl]-5-methyl-1-phenyltriazole-4-carboxamide;hydrochloride N-[5,8-bis(2-methylphenyl)quinolin-7-yl]acetamide (2E,4Z)-N-[5-chloro-6-(1H-imidazol-2-yl)pyridin-3-yl]-2-methanimidoylhexa-2,4-dienamide 1-azido-6,7-dimethyl-3-phenyldibenzothiophene 3-azido-4,5,6,7-tetrahydrobenzimidazole N-(4,6-dimethylpyridin-2-yl)-3-[1,1-dioxo-4-[4-(trifluoromethoxy)phenyl]-1,2,5-thiadiazol-3-yl]propanamide N-[1-[1-(3-hydroxyazetidine-1-carbonyl)piperidin-4-yl]ethyl]naphthalene-2-sulfonamide 4-[(E)-3-amino-2-cyano-3-oxoprop-1-enyl]-N-tert-butylbenzamide 4-bromo-3-[(E)-4-phenylbut-2-enoxy]benzaldehyde 2-[(1S)-5-methoxy-3,4-dihydronaphthalen-2-yl]benzotriazole 1-[5-(cyclopropylamino)-4,6-diethoxypyridin-2-yl]ethanol N-ethenyl-4,5-dinitrofuran-2-amine 5-bromo-2-[1-(3,4-dimethylphenyl)ethylidene]cyclohexan-1-one 2-[(4S)-6,8-dichloro-1,2,3,4-tetrahydroquinolin-4-yl]butanoic acid N-[[4-(hydroxymethyl)oxan-4-yl]methyl]-2-oxopyridine-1-carboxamide 3-[4-(9H-fluorene-1-carbonyl)-2-methylpiperazin-1-yl]-5,6-diphenylpyrazine-2-carboxamide 2-[(2S)-1-methylpyrrolidin-2-yl]-N-propan-2-yloxy-5-pyrrolidin-3-ylbenzamide 1-[5-(trifluoromethyl)pyridin-2-yl]propane-2-thiol N-methoxy-N-(3-phenylpropyl)benzenesulfonamide 2-N,4-N-bis(1-benzofuran-3-ylmethylideneamino)benzene-1,2,4-triamine (2R)-2-[(1S)-1-(2,4-dichlorophenyl)ethyl]cyclohexan-1-one 6-[(4S)-4-methyloctoxy]-1,3,5-triazine-2,4-diamine 2,3-diphenylinden-1-imine 5-[[4-chloro-2,6-di(propan-2-yl)phenyl]carbamoylamino]pyridine-3-carboxylic acid 4-N-[(2E,4Z)-hepta-2,4-dienyl]-6-propan-2-ylpyrimidine-2,4-diamine 4-[2-[(1R,3S)-6-fluoro-1-methyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-4-pyridin-2-ylpyrazolidin-1-yl]benzonitrile 1-methyliodanuidylbutoxybenzene (3E)-4-amino-3-[(2,5-dimethoxyphenyl)methylidene]azete-2-thione 1-(4-methylpiperazin-1-yl)sulfonylnaphthalene-2,3-diol 4-(2,3,3a,4,6,7,7a-octahydro-1H-pyrrolo[3,4-c]pyridine-5-carbonyl)-N'-cyclopropylsulfanyl-3-fluorobenzohydrazide N-[5-chloro-4-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-(4-fluorophenyl)-3-oxo-2H-pyrazole-4-carboxamide 2-(4,5-dichlorothiophen-3-yl)imino-1H-pyrimidine-4,6-dione [2-[3-(trifluoromethyl)phenoxy]phenyl]boronic acid (6E)-N,2-dimethylocta-1,3,6-trien-4-amine;1-[4-(4,5-dihydrofuro[3,4-c]pyrazol-2-yloxy)phenyl]ethanone 7-benzyl-5,7-diazaspiro[2.4]heptan-6-one [1-(4,4-diethylcyclohexen-1-yl)-2,2-dimethoxyethylidene]hydrazine ethane;4-(methylsulfonimidoyl)benzenethiol 2-[(4-oxo-1,5,6,7-tetrahydroindole-3-carbonyl)amino]propanoic acid N-[(1R,2S)-2-hydroxycyclohexyl]-6-methoxypyridine-3-carboxamide 3-(2,4-dimethylphenyl)-1-(4-fluorophenyl)prop-2-en-1-one 3-[1-(azidomethyl)cyclohexa-2,4-dien-1-yl]-5-(3-chloro-2-fluorophenyl)pyridine 3-amino-4,5-dimethoxybenzoic acid;2-[(6-bromopyridin-3-yl)methoxy]-6-(ethylideneamino)pyridine 2-[3-(6,8-dihydrobenzo[c]chromen-2-yloxy)propyl]piperidine 2-(methylamino)-5,6,7,8-tetrahydrothieno[3,2-b]azepine-4-carbonitrile N-butyl-2,6-dibromopyrimidin-4-amine 2-[3,5-bis(trifluoromethyl)phenyl]-1-[4-ethoxy-3-(1H-indol-2-yl)phenyl]guanidine 6-(3,4-dihydroxyphenyl)-2-[1-(piperidine-1-carbonyl)indol-5-yl]pyran-4-one N-(2,4-dichloropyrimidin-5-yl)-N-[1-phenylpropan-2-ylideneamino]-2H-tetrazol-5-amine 2-amino-8a-[4-fluoro-3-(trifluoromethoxy)phenyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carbonitrile N-(furan-2-ylmethyl)-4,9-dioxobenzo[f][1]benzofuran-5-carboxamide 4-chloro-N-[3-(2H-tetrazol-5-yl)phenyl]benzamide N-[2-(3-chlorophenoxy)propyl]ethanamine;(4S,5R)-4,5-dihydroxy-3,7,7-trimethyloctanamide 4-[6-ethylsulfonyl-2,3-difluoro-5-(pyridine-2-carbonyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-6-carbonitrile 1,2-diamino-6-oxo-4-(5-pyridin-3-ylfuran-2-yl)pyridine-3,5-dicarbonitrile 1-butyl-3-[(4Z)-2-methylhepta-2,4,6-trien-3-yl]benzene;ethane N-methyl-4-[3-(methylamino)-2,5-dioxopyrrol-1-yl]-N-(pyridin-2-ylcarbamoyl)benzamide N-[(3S)-1-azabicyclo[2.2.0]hexan-3-yl]-6-fluoro-4-oxochromene-2-carboxamide 5-amino-2,4-dimethylthiophene-3-carboxylic acid N-(2,3-dihydroindol-1-yl)-4-[5-(piperidin-3-ylmethoxy)pyridin-3-yl]benzamide N-[(3R,4S)-1-cyclopentyl-4-methoxypyrrolidin-3-yl]-2-(oxan-4-ylsulfamoyl)benzamide;hydrochloride (1S)-3-[2-(cyclopropylmethoxy)pyridin-4-yl]-N,N-dimethyl-1-spiro[3.5]nonan-9-ylpropan-1-amine N-ethylsulfonyl-2,4,6-trimethyl-N-[(4-nitrophenyl)methoxy]benzenesulfonamide (2Z,4E)-5-(1-ethylpiperidin-3-yl)-7-(2-methoxyphenyl)hepta-2,4-dienal 1-(4-azidophenyl)-N,2-dimethylpropan-1-imine (2S,5R)-4-acetyloxy-5-(3,4-dihydro-1H-isoquinoline-2-carbonylamino)-2-methoxy-6-(phenylcarbamoyl)hexanoic acid N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-ethoxypyrimidine-5-carboxamide N'-[(1R)-2,3-dihydro-1H-inden-1-yl]-6-hydroxy-1,4-dioxonaphthalene-2-carboximidamide (2S)-4-[3,5-bis[[6-(2-propoxyethylamino)pyridine-2-carbonyl]amino]phenyl]-1-butanoylpyrrolidine-2-carboxylic acid 2-(methoxycarbonylamino)benzenesulfonate 2-(4-azidophenoxy)-N-[(1R,5S)-3-(5-methylpyrazole-1-carbonyl)-6-bicyclo[3.2.0]heptanyl]acetamide N-(4,6-dimethylpyrimidin-2-yl)sulfanyl-N-(2H-tetrazol-5-yl)butanamide 1-[3,5-bis(trifluoromethyl)phenyl]-N-(4-cyclopentylphenyl)cyclopropane-1-carboxamide 1-[2-azido-4,5-dimethoxy-3-(trifluoromethyl)phenyl]imidazole 5-[[4-(4-tert-butylpiperidine-1-carbonyl)phenyl]methoxy]-6-methanimidoylpyrimidine-4,7-diamine 5-(2,6-difluorophenyl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-one (Z)-3-[3,5-bis(trifluoromethyl)phenyl]prop-2-enoic acid (2R)-6,15,16,17,21-hexamethylpentacyclo[11.7.0.02,10.05,9.014,18]icosa-1(13),2(10),3,5(9),6,11,14(18),18-heptaene N-[3,5-bis(trifluoromethyl)phenyl]-4-tert-butylbenzamide [2-fluoro-6-(trifluoromethyl)phenyl]-[[6-[4-[3-[2-(prop-1-en-2-ylamino)ethoxy]benzoyl]piperazine-1-carbonyl]pyridine-3-carboximidoyl]iodanuidylmethylidene]azanium 4-(2-oxo-1H-quinolin-3-yl)piperazine-1-carboxylic acid 1-[2,6-bis(trifluoromethyl)phenyl]hexane-3,4-dione 2-amino-N'-[3-(4-cyclopropylsulfanylphenyl)sulfanylphenyl]pyridine-3-carboximidamide (3S)-4-amino-2,2,5,6,7-pentamethyl-1-(4-propan-2-yloxyphenyl)heptan-3-ol ethane;1-ethylpiperidine;methanamine;4-[[5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl(propan-2-yl)amino]methyl]benzoic acid 4-[(2,6-difluorophenyl)methyl]-3,5,7,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,6,11-pentaen-13-one (3-fluorophenyl)-(5H-pyrrolo[2,3-b]pyrazin-7-ylmethylamino)methanol 1,5-dimethyl-3-(pyridin-2-ylamino)pyrazole-4-carboxamide N-[(Z)-2,4-difluorohex-3-enyl]-N-methylbenzenesulfonamide [1-(3,3-dimethylmorpholin-4-yl)cyclopentyl]-(6-pyridin-2-ylindolizin-5-yl)methanone;2,2,2-trifluoroacetic acid 1-[2-(4-tert-butylphenyl)cyclopropyl]naphthalene (E)-2-[[5-chloro-6-(methylamino)pyrimidin-4-yl]amino]but-1-ene-1,3-diol 4-[[2,6-di(propan-2-yl)phenyl]iminomethyl]benzene-1,3-diol 2-[4-chloro-5-[(4R)-2,2-dimethyl-1,3-oxazolidin-4-yl]thiophen-2-yl]sulfanylpyridine 2-[2-ethyl-6-methyl-4-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-3-yl)phenoxy]acetic acid;6-methoxy-N-pentan-3-ylpyridazine-3-carboxamide 6-N-[3-(2-aminoethyl)phenyl]-4-chloroquinazoline-2,7-diamine;hydrochloride (2S)-N-[3,5-bis(trifluoromethyl)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]sulfanylpyrrolidine-2-carboxamide [4-(6-bromo-13-chloro-8-hydroxy-4-azatricyclo[9.4.0.03,7]pentadeca-1(11),3(7),5,12,14-pentaen-2-yl)piperidin-1-yl]-[2-(methoxymethylamino)cyclopropyl]methanone 4-[2,2-dimethoxyethyl(3-methylbut-2-enyl)amino]benzoic acid N'-[3-chloro-4-(trifluoromethyl)phenyl]-N,N'-diethylpropane-1,3-diamine (2R)-1,5,6-trimethyl-N-[4-(trifluoromethoxy)phenyl]piperidine-2-carboxamide (Z)-2-(3-phenylpropylsulfonyloxymethylamino)but-2-enoate N-butan-2-yl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide;ethane 2-tert-butyl-5,7-dichloroquinoline 1-[6-(trifluoromethyl)pyridin-3-yl]piperidine-4-carboxamide 1-[3-[4-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazine-1-carbonyl]phenyl]ethanone 5-(aziridine-1-carbonyl)-N,2,4-trimethylpyrazole-3-sulfonamide 1-[6-(2-fluorophenyl)imidazo[1,2-a]pyridin-8-yl]-2H-pyrazine N-(5,6-dihydronaphthalen-2-yl)-4-[(4S)-2-methylcyclopropen-1-yl]butanamide 2-[[(3,5-dimethylbenzoyl)-[6-oxo-4-(trifluoromethoxy)piperidin-3-yl]amino]methyl]benzamide 2-[6,7-difluoro-5-(4-pentoxyphenyl)naphthalen-2-yl]oxane 3-(4,6-diphenylpyrimidin-2-yl)-5-nitrobenzonitrile 1-[2-[2,4,6-trichloro-N-(2,3-dihydroxypropyl)anilino]ethyl]pyrrolidine-2,5-dione N-(2,6-difluorophenyl)-2,4,6-trimethyl-N-(3-methylbut-2-enyl)benzamide ethane;[2-methyl-4-(1-pyrimidin-2-ylethenyl)phenyl]-[4-(pyrrolidin-1-ylamino)piperidin-1-yl]methanone N-(3,5-dichlorophenyl)-2-[4-methyl-6-oxo-1-[[4-(trifluoromethoxy)phenyl]methyl]pyrimidin-5-yl]acetamide 3-[4-hydroxybutyl(3-methylbut-2-enyl)amino]phenol 1-(2,5-dimethoxyphenyl)-N-[2-[(4-oxo-3H-quinazolin-2-yl)methyl-propan-2-ylamino]ethyl]cyclopentane-1-carboxamide ethane;6-methyl-4-(3,3,4,5,7,8-hexamethylnaphthalen-1-yl)isoquinoline N-[(3,5-dimethoxyphenyl)methyl]-2-pyrrolidin-1-ylsulfonylcyclohexane-1-carboxamide N-[5-(benzimidazol-1-yl)isoquinolin-3-yl]propanamide N'-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-phenylpropanimidamide N-[[2,6-dimethyl-4-[(Z)-1H-pyrazol-5-yliminomethyl]phenyl]methyl]benzenesulfonamide (E)-3-[4-hydroxy-2,6-dimethyl-3-(1-phenylethoxycarbonylamino)pyridin-1-ium-1-yl]prop-2-enoic acid 3-(4-methylphenoxy)-6-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-2-yl]pyridazine-4-carbonitrile N-methyl-6-(4,4,5,5-tetramethyloxaborolan-2-yl)pyridin-3-amine N-(3,4-dihydropyridin-2-yl)-2-iodobenzamide (2S)-1-(2,2-difluoroethyl)-4-[7-(8-methylnaphthalen-1-yl)-2-(2-oxoimidazolidin-1-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]piperazine-2-carbonitrile N-[(1S)-2-oxocyclohexyl]naphthalene-1-carboxamide N-[(2R,3S)-5-methyl-1-sulfanylidenepent-4-en-2-yl]benzenesulfinamide N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-4-(4-fluorophenyl)piperazine-1-carboxamide;formic acid 4-(cyclopropanecarbonylamino)-2,3-dihydro-1H-indole-5-carboxylic acid 1-[4-(azidomethyl)phenyl]sulfonyl-3-(trifluoromethoxy)benzene [3-(1,4-dihydropyrimidin-2-ylamino)cyclobutyl]-[2-methyl-6-(1,2,4-triazol-1-yl)pyridin-3-yl]methanone [3-(2,4-dichlorophenyl)cyclopentyl]methanamine (3R)-3-amino-4-[5-fluoro-6-(2,2,2-trifluoroethylsulfanyl)pyridin-3-yl]butanoic acid 5-(2,6-dichlorophenyl)-4-[4-ethyl-3-[hydroxy(methylamino)methoxy]phenyl]-N-[(1R)-1-naphthalen-1-ylethyl]-1,2,4-triazole-3-carboxamide N-[4-(7-hydroxyquinolin-4-yl)oxycyclohexa-1,3-dien-1-yl]pyridine-2-carboxamide 2-[3-bromo-4-(2H-pyridin-1-yl)phenyl]sulfanylpyrazine N-benzyl-2,4,6-trimethyl-N-(1-phenylethyl)aniline 4-[1-[(3S)-piperidine-3-carbonyl]azetidin-3-yl]oxypyridine-2-carboxamide 4-[1,3-dioxo-7-[[2-(trifluoromethyl)phenyl]carbamoyloxy]isoindol-2-yl]benzoic acid 6-(3,4-dihydropyridin-5-yl)-8-methylquinazoline;ethane 3-[(2E)-3,7-dimethylocta-2,6-dienoxy]benzaldehyde 3-[[2-[5-(aminomethyl)pyridin-2-yl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]sulfonyl]benzamide 6-[2,3-bis(sulfanyl)anilino]hexanenitrile 1-ethyl-3-[(E)-N'-(2,4,6-trichlorophenyl)carbamimidoyl]urea [2,2-difluoroethyl(3-methoxypropyl)amino]-[1-(1H-indazole-5-carbonyl)piperidin-4-yl]-oxoazanium 2-[1-(2,6-dichlorophenyl)propan-2-yl]-4-methoxypyrimidine 1-[[5-(4-fluorophenyl)triazolo[4,5-b]pyrazin-3-yl]methyl]cyclohexan-1-amine;hydrochloride 2-[(4-methoxyphenyl)sulfanylmethylidene]propanedinitrile 2-N-cyclohexyl-4-N-[3-fluoro-5-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine 4-chloro-N-[1-(3,5-difluorophenyl)propyl]-2-iodoaniline 2-[[3,4-bis(trifluoromethyl)phenoxy]methyl]pyridine N-[4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]-2-methoxy-N-(4-nitrobenzoyl)acetamide 2-[(4-chlorophenyl)sulfanylmethyl]-7,8-dihydro-3H-pyrimido[5,4-b]pyrrolizin-4-one N-[4-(5,6,7,8-tetrahydronaphthalene-1-carbonyl)thiophen-2-yl]benzenesulfonamide [3-(2,6-dioxopiperidin-1-yl)phenyl]phosphonic acid 2-cyclopropyloxy-6-fluoro-N-[4-(3-phenylmethoxyazetidine-1-carbonyl)phenyl]benzamide N-[(1S,2R)-1-hydroxy-3-oxo-2-phenylcyclohexyl]imidazo[1,5-a]pyridine-2-carboxamide 2-chloro-N-[(Z)-3,5-dimethylheptan-4-ylideneamino]-7-fluoro-3H-benzimidazole-5-carboxamide N'-[[(4-aminocyclohexyl)amino]-(2,3,5,6-tetrafluorophenyl)methyl]propanediamide (2Z)-3,5-bis[4-(diethylamino)phenyl]-N-ethyl-2-hydroxyiminopentanamide;N-[(1S)-1-(4-fluoro-3-methoxyphenyl)ethyl]acetamide 7-methoxy-5-(5-morpholin-4-ylpyridin-2-yl)cinnoline-3,8-dione 1-[4-(5-bromopyridin-3-yl)oxyphenyl]ethanimine [4-(3,4-dihydro-2H-chromen-8-ylmethyl)piperazin-1-yl]-(5-methylpyrazin-2-yl)methanone (2S)-5-[(E)-4-benzoyloxybut-3-enoyl]oxy-2-(4-chlorophenyl)hexanoic acid 2-[N-(3-methylbut-2-enyl)-4-[(2-phenylpyrazol-3-yl)sulfamoyl]anilino]octanoic acid 5-methylsulfinyl-N-[2-(pyridine-3-carbonylamino)ethyl]pyridine-3-carboxamide 4-azidooxy-2-benzylperoxy-1-chlorobenzene 3,3-dimethylpentane;6-[(4R)-2,7-dimethyloct-5-en-4-yl]quinoline [2-[4-(6,8-dichloro-7-fluoroquinazolin-4-yl)piperazin-1-yl]phenyl]methanediamine N-(4,5-dimethoxypyridin-2-yl)-3-[(1S,4R)-4-hydroxy-2-azabicyclo[2.2.0]hexan-2-yl]propanamide 2-[(1,5-dimethylpyrazole-4-carbonyl)amino]-9-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)-3H-purine-6-carboxamide 2-[1-(4,4-difluorocyclohexyl)ethyl]-6-[3-hydroxy-4-[4-hydroxy-2-(trifluoromethoxy)phenoxy]phenyl]-8-propan-2-ylimidazo[1,5-a]pyrimidin-7-one 4-ethyl-2,3-bis(1H-imidazol-2-yl)phenol 2-ethoxy-6-fluoro-N'-hydroxy-3-methylbenzenecarboximidamide 1-[7-azido-5-(2,4,6-trimethylphenyl)-9H-fluoren-2-yl]-2,3-diethoxyindole (7R)-2,3-bis(ethenyl)-8-methylidene-9-propan-2-yl-11H-benzo[a]fluorene N-[6-(2,4-difluorophenyl)imidazo[1,2-a]pyridin-8-yl]-3-ethoxysulfanylcyclobutane-1-carboxamide N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]-3-morpholin-4-ylazetidine-1-sulfinamide 3-(1H-benzimidazole-2-carbonylamino)propanoic acid 1-[(3,5-dichloropyridin-4-yl)methyl]pyrrolidine-2-carboxylate 1-[(1R,2S)-2-hydroxycyclohexyl]-3-[4-methoxy-6-methyl-5-(pyrrolidine-1-carbonyl)pyridin-2-yl]urea N-[1-(4-bromophenyl)ethyl]-2-cyanopyridine-3-carboxamide N-[[4-(furan-3-yl)thiophen-2-yl]methyl]formamide (3S)-2,2-dichloro-6-fluoro-7-formyl-1,3-dihydroindene-4-carboxylic acid;N-[(3R)-1,1-dioxothiolan-3-yl]-5-methoxypyridine-2-carboxamide 2-[5-(4-tert-butylphenyl)-4,4-dimethyl-3H-pyrazol-2-yl]pyridine N-[2,6-di(propan-2-yl)phenyl]-4-ethynylcyclohexane-1-carboxamide [(4aS)-6,7,8,9,10,11b-hexahydro-5aH-pyrido[1,2-h]pteridine-4-carbonyl]-methylazanium 1-[(2S,4R)-4-azido-5-chloro-2,3-dihydroindol-1-yl]ethanone N-[2-(5,7-dimethylimidazo[1,2-a]pyridin-3-yl)ethyl]cyclohexanecarboxamide N-(diaminomethylidene)-3,5-dihydroxy-2-oxo-6-phenylchromene-8-carboxamide;N,2-dimethylpropane-2-sulfonamide 2-(4-fluorophenyl)-6,7-dimethoxy-3H-quinazolin-4-one 2-[2-chloro-4-(trifluoromethyl)phenyl]-1,3-benzothiazole 2-[[4,6-dichloro-1-(4-fluorophenyl)benzimidazol-2-yl]methoxycarbonylamino]acetic acid N-(2,6-dichloro-3-nitrophenyl)-5-methyl-1H-indazole-3-carboxamide ethane;2-[4-(trifluoromethyl)phenyl]sulfonylcyclohexan-1-one N-(2,4-dichloropyrimidin-5-yl)-3-oxobutanamide 3-(1,3-benzodioxol-5-ylmethylideneamino)pyridine-2-carboxylic acid N-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]propanamide 7,10-dimethoxy-2-[2-(5-nitrofuran-3-yl)ethyl]-6H-1,4-benzoxazepine 4-(1,3-benzothiazol-2-yl)-5-imino-1-[4-(trifluoromethoxy)phenyl]-2H-pyrrol-3-ol 4-[(E)-2-chloroprop-1-enyl]sulfanylphenol N-ethenyl-1,2-difluoro-6-[4-(4-methylcyclohexyl)phenyl]naphthalene-5-carboxamide 4-hydroxy-6-methoxy-5-(2-methyliminoethanehydrazonoyl)pyridine-3-carboxamide 1-cyclopropyl-7-[4-(6,6-dimethylazepane-2-carbonyl)piperazin-1-yl]-6-fluoro-8-methoxy-5H-pyrazolo[4,3-c]quinolin-4-one 1-[5-methyl-3-[(2-methyl-6-morpholin-4-ylpyrimidine-4-carbonyl)amino]pyridin-2-yl]piperidine-4-carboxylic acid N-[(Z)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-3-methoxybenzamide 4-(6,7-dimethoxyquinazolin-4-yl)morpholine 1-(7,8-dihydrothieno[2,3-b][1,5]benzothiazepin-4-yl)propan-2-one 4-[2-[2-(ethylamino)pyridin-3-yl]ethynyl]benzamide N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-3-morpholin-4-ylsulfonylbenzamide 2-amino-5,6-dichloro-3H-quinazolin-4-one 2-[4-[1-(1,3-benzodioxol-5-yl)cyclopropyl]piperazin-1-yl]-6-methanimidoyl-N,N-dimethylpyridine-4-carboxamide N-[(2S)-3,3-dimethylbutan-2-yl]-4-fluorobenzamide 4-[5-(3,5-dimethoxyphenyl)pentanoyl]-3-nitrobenzonitrile 5-amino-1-(oxan-4-yl)-6H-pyrazolo[4,3-d]pyrimidine-7-thione 5-(1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl)benzene-1,3-dicarboxylic acid 2-[(3-methylphenyl)methyl]-N-propan-2-yl-3H-pyrazole-4-carboxamide 2-[1'-(cyclopropanecarbonyl)spiro[1,3-dihydroisoquinoline-4,4'-piperidine]-2-yl]acetic acid;2,2,2-trifluoroacetic acid 6-azido-2-chlorobenzenesulfonamide 4-[2,3-dichloro-5-[(1S)-1-hydroxyethyl]phenyl]pyridine-3-carbonitrile 4-(1,3-benzodioxol-5-yl)-2-iminopyrrolidine-1-carboxylic acid N-[2-methyl-3-(1H-pyrrol-2-yl)butan-2-yl]benzamide (2R,3S)-5-chloro-N,N'-dimethyl-1-pyridin-4-yloxycarbonylpiperidine-2-carbohydrazide N-[(3,4-difluorophenyl)methyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide 4-tert-butyl-2-[(E)-[[6-(2,6-dimethoxyphenyl)pyridin-3-yl]hydrazinylidene]methyl]phenol (4R)-4-[3,5-bis(trifluoromethyl)phenyl]pyrrolidine-2-carboxylic acid 2-amino-4,5-difluoro-N'-phenylbenzenecarboximidamide (4-chlorophenyl)sulfonyl-(2,3-dihydro-1H-inden-5-ylsulfanylmethoxycarbonyl)azanium 4-[2-(4,5-dimethylfuran-3-carbonyl)oxyethoxy]benzoic acid 5-[3,4-dichloro-2-(methylamino)phenyl]pyrimidine-2,4-diamine 6-(4-cyclopropyl-5H-1,3-thiazol-2-yl)pyridine-2-sulfonamide 1-azido-5,6,7,8-tetrahydroisoquinoline-4-carboxamide 1-(4-methylphenyl)-N,N'-bis[3-(trifluoromethylsulfanyl)but-3-enyl]ethane-1,2-diamine 2-tert-butyl-6-(phenyliminomethyl)phenol;dichlorotitanium 2-[6-(benzylamino)pyridine-3-carbonyl]-1,4-dihydroisoquinolin-5-one 3-[5-[4-(azidomethyl)phenyl]thiophen-2-yl]-1,1-dimethylurea (2R,3S)-2-ethyl-N'-[(5-methoxypyrimidin-4-yl)methyl]-3-(1-methylpyrazol-4-yl)butanediamide 4-(3,5-dimethylphenyl)-2,6-bis(trifluoromethyl)pyridine 1-azidooxy-3,5,6-trimethyl-4-(2,4,6-trichlorophenoxy)benzene 4-chloro-2-[[(3R)-3-fluoropyrrolidin-1-yl]methoxy]benzoic acid 4-[2-(benzylideneamino)propanoylamino]benzenesulfonic acid 3-[1-[6-chloro-5-(methylamino)pyridine-2-carbonyl]piperidin-4-yl]-1,4-dihydro-1,2,4-triazol-5-one 4-fluoro-5-methylsulfanyl-2-(1,3-thiazol-4-yl)benzoic acid 3-[2-cyclohexyl-1-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-yl]-N,N-diethylpropan-1-amine;hydrobromide N-[5-[4-fluoro-3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]cyclopropanecarboxamide 1-[2-(3,5-difluorophenyl)acetyl]-N-hydroxy-N'-methylpiperidine-4-carboximidamide N-[1-(2,6-dioxopiperidin-3-yl)-2-hydroxyindol-3-yl]imino-2,5-dimethoxybenzamide 3-(3,4-dimethoxyphenyl)-N-[2-(1H-indol-3-yl)ethyl]prop-2-enamide;uranium(2+) (Z)-N,4-dimethylpent-2-enamide;3-ethyl-5-fluoro-7-methyl-1H-indole;(E)-8-methoxy-6-methylidenenon-4-ene 7-[2-(3,5-dimethoxyphenyl)ethynyl]-1,4,4,5-tetrahydroxyimidazolidin-2-one 4-[(2,5-dimethoxyphenyl)methyl]-6-fluoro-7-pyrazol-1-ylchromen-2-one N-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]formamide;ethane 4-(cyclopentylmethylamino)benzenesulfonamide 3-[1-(2,6-dichlorophenyl)ethenyl]-4H-1,2,4-oxadiazol-5-one 1-(4-chlorophenyl)-3-[(Z)-prop-1-enyl]piperazine;ethane 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[(5-methoxypyrazin-2-yl)methylidene]urea 1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxycarbonylnaphthalene-2-carboxylic acid N-[(2S)-1-[3-cyclohexylpropanoyl(2,4-dihydroxybutyl)amino]-2-methoxypropan-2-yl]-5-[(E)-ethylideneamino]-1H-pyrazole-3-carboxamide 4-[2,3-difluoro-5-(1,3-thiazol-2-ylmethoxy)phenyl]pyrimidin-2-amine N-(2,4-difluorophenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidine-7-carboxamide 2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-(1-phenylcyclopentyl)acetamide 2-(4-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole 5-amino-4-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one 4-[5-[(2R)-2-(methylaminomethyl)morpholine-4-carbonyl]pyridin-3-yl]oxypiperidine-1-carboxylate 1-[(3-methoxyphenyl)methyl]-2-oxo-N-propan-2-ylpyridine-4-carboxamide 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[chromene-2,4'-piperidine] N-[3-methyl-2-(4-phenylcyclohexa-1,5-dien-1-yl)phenyl]pentanamide 7-ethyl-N-methylidene-6-[3-(2,2,2-trifluoroethoxy)azetidine-1-carbonyl]indolizine-5-carboxamide 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-1-yl]-5-propoxypyridine 2-azido-5-[(4-methylphenyl)sulfonylamino]pyridine-3-carboxylic acid 3-[3-azidooxypropyl(3-phenylpropanoyl)amino]benzoic acid 4-amino-3,5-diiodobenzoate 2-(3,5-dibromo-2-hydroxyphenyl)benzo[e]benzotriazole-4,6-disulfonic acid 2-[3-(4,7,10-triazatricyclo[7.5.0.02,6]tetradeca-1(9),2(6),3,11-tetraen-12-yl)phenyl]propanoic acid 1-[2-(4-fluorophenyl)ethyl]-3,3a,5,6a-tetrahydropyrrolo[3,2-b]pyrrole 1-azido-5,6-dimethoxy-2H-acenaphthylene 5-[3-(1H-benzimidazol-2-yl)propanoyl]pyridine-3-carboxamide;acetic acid N-[(3R)-1-acetylpiperidin-3-yl]-2-[7-amino-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]acetamide 4-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]-1H-pyrrole-3-carbonitrile 4-bromo-2-[(E)-1,3-diaminoprop-2-enylidene]-N-(5-chloropyridin-2-yl)pyrrolidine-1-carboxamide 2-(3,4-difluorophenyl)-1-(methylamino)propan-2-ol 4-(azidomethyl)-2-chloro-3-fluorophenol N-[2-(2-methylpropanoylamino)ethyl]quinoline-3-carboxamide N-[(5Z)-3-[4-[[3,5-bis(trifluoromethyl)phenyl]methoxy]phenyl]-5-(2H-tetrazol-5-ylmethylidene)pyrrol-2-yl]hydroxylamine 1-[3-amino-5-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl]ethanone N-[4-methylsulfanyl-2-(trifluoromethyl)phenyl]carbamate 2-[4-(6-fluoropyridin-3-yl)phenyl]acetic acid 3-methoxy-4,6-diphenylbenzene-1,2-dicarbonitrile [5-(3,4-dimethoxyphenyl)tetrazol-1-yl]-[2-fluoro-6-[3-[6-(trifluoromethyl)pyridin-2-yl]phenoxy]pyridin-3-yl]methanone 1-(4,5,6-trimethyl-3H-isoindol-1-yl)ethanone N-[(3S,4R)-1-[5-[1-(cyclopropylmethoxy)ethyl]-2-fluorophenyl]-4-(hydroxymethyl)piperidin-3-yl]methanesulfonamide N-(4,5-dimethylpyrimidin-2-yl)-4-[2-ethoxypropyl(methylsulfonyl)amino]benzenesulfonamide 7-(3,4-dihydro-2H-chromene-6-carbonylamino)heptanoic acid 3-methylsulfanyl-4-[(2E,7Z)-nona-2,7-dien-5-ynoxy]-1-propanoyl-N-thiophen-2-ylpyrrolo[2,3-b]pyridine-2-carboxamide N'-amino-4-(2,5-dimethoxyphenyl)-1,3-thiazole-5-carboximidamide 2-[3-(4-fluorophenyl)-4-oxothiochromene-7-carbonyl]oxyacetic acid 3-chloro-N'-(1H-pyrazole-5-carbonyl)benzohydrazide 2-(5,6-dichloroindole-1-carbonyl)cyclopentane-1-carboxylic acid 5-[4-methoxy-3,5-bis(trifluoromethyl)phenyl]imidazolidine-2,4-dione N-[3,5-di(propanoyl)phenyl]-3-(3-methoxyphenyl)butanamide [(3S)-6-bromo-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methanol [6-(2,4-dimethylphenoxy)-1H-benzimidazol-2-yl]carbamic acid N-(4-chlorophenyl)-5-[4-hydroxy-2-(trifluoromethyl)anilino]naphthalene-1-sulfonamide 3-(6,7-dimethoxy-2H-quinoline-1-carbonyl)benzoic acid 2-amino-7-[3-fluoro-4-(methylamino)phenyl]-9-(oxan-4-yl)-1H-purine-6,8-dione 2-[4-(2,6-dioxopiperidin-3-yl)-2-formylphenyl]iminoacetamide N-[(3S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethoxy)piperidin-3-yl]acetamide 3-[2,4-dihydroxy-5-(5-methylsulfanylthiophen-2-yl)phenyl]propanamide 4-fluoro-N-[1-(5-ethylfuran-2-carbonyl)piperidin-3-yl]-3,5-dimethoxybenzamide 2-[5-amino-4-[(Z)-1,3-dichloroprop-1-enyl]-6-methylpyrimidin-2-yl]phenol [(4aR,7aS)-2-methyl-3,4a,5,6,7,7a-hexahydrocyclopenta[b][1,4]oxazin-4-yl]-(5-chloropyrimidin-2-yl)methanone (3S)-2-[6,7-difluoro-5-[4-[1-methyl-5-(morpholine-4-carbonyl)pyrazol-4-yl]phenyl]-1H-indole-3-carbonyl]-N'-hydroxy-3-propan-2-ylbutanediamide 2-[[5-chloro-2-(6-fluoro-7-methyl-1H-indole-3-carbonyl)phenyl]sulfonylamino]acetic acid 3-[4-(3,5-dimethylpiperidin-1-yl)-2,6-dioxopiperidin-3-yl]phthalic acid 3-[2-(4-fluorophenyl)ethyl]-1,5-dimethylimidazolidine-2,4-dione 3-[4-(N'-hydroxycarbamimidoyl)phenyl]-2,5-dimethylfuran-4-carboxylic acid 1-[4-(2,5-difluorophenyl)-2-methylbutan-2-yl]piperidine 5-[(4Z)-1,2-dimethyl-6-oxoocta-2,4-dien-3-yl]oxycarbonylpyridine-2-carboxylic acid 4-amino-6-[(2,3,5,7,8-pentamethyl-1-benzofuran-5-yl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 1-(3,4-dimethoxyphenyl)-2-methyl-3H-pyridazin-6-one [1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]-pyrrolidin-1-ylmethanone 2-(3,5-dichlorophenyl)-4H-[1,3]thiazolo[5,4-c]pyridine-6-carboxamide 1-bromo-3-(10,10-dimethylundecoxy)benzene 4-(azidomethyl)-N-[2,6-dibromo-3-[difluoro(phenyl)methoxy]phenyl]benzenesulfonamide N-[(3S,4R)-1-(2,5-dimethylpyrimidin-4-yl)-4-phenylpyrrolidin-3-yl]-1,7-naphthyridine-3-carboxamide 2-(N-naphthalen-1-yl-4-propylanilino)acetonitrile 1,3-dimethyl-5-[4-[2-(oxan-4-yloxy)ethyl]piperazine-1-carbonyl]benzimidazol-2-one;formic acid 1-(3,5-dimethoxyphenyl)-6,8,9,10-tetrahydrocycloocta[b]indole 6-[(Z,2E)-2-ethylidenepent-3-enyl]-4H-1,4-benzoxazin-3-one 1,3-dimethyl-4-[(4R)-6-oxo-7-phenyl-2,5,8,11,14-pentazatricyclo[8.4.0.02,6]tetradeca-1(10),3,13-trien-12-yl]piperazine-2,5-dione 3-[8-amino-2,3-bis(quinolin-7-ylmethyl)imidazo[1,2-a]pyrazin-6-yl]phenol [7-(hydroxymethyl)-3,4a,5,6,7,8,9,10,11a-decahydro-2H-cyclopenta[b][1]benzazepin-1-yl]methanol 7-fluoro-4-(4,5,6-trichloropyrimidin-2-yl)quinoline 4-[7,8-bis(ethenyl)-6-iminodibenzothiophen-2-yl]benzaldehyde 4-(3,5-diphenyl-1H-pyrazol-4-yl)morpholine 4-hydroxy-1,7-diphenylheptan-3-one 3-[4-(4-methylimidazol-1-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-5-pyrimidin-5-yl-2H-pyrazolo[3,4-b]pyridine N-butyl-3-[5-fluoro-1-methyl-6-(pyrrolidin-1-ylmethyl)indol-2-yl]benzamide 4-(4-ethylphenyl)sulfanylpiperidine 4-hydroxy-3-methoxy-N-(1H-pyrrolo[2,3-b]pyridin-5-yl)benzamide 1-[4-(methoxymethyl)phenyl]sulfonyl-5,8-diazaspiro[3.5]nonane N-[5,6-dimethoxy-2-(1H-pyrazolo[3,4-b]pyridin-5-yl)pyrimidin-4-yl]ethanesulfonamide 1-(2,4-dichloro-3-methylphenyl)-N-[6-(3,4-dimethoxycyclohexa-1,5-dien-1-yl)pyridin-3-yl]ethanimine 5-[[2-(4,6-dimethoxypyrimidin-2-yl)sulfanylacetyl]amino]-1,3-thiazole-4-carboxylic acid 1-[(4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]-2,7-dicyclohexyloxynaphthalene-2,3-diol 4-[1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one 1-[2,6-di(propan-2-yl)phenyl]pyrrole-2,5-dione;rhodium(3+) 4-[5-[2-(2,6-dichlorophenyl)ethyl]pyridin-3-yl]benzaldehyde 4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]benzoic acid N-(cyclopropylmethyl)-2,6-difluoro-4-[3-methanimidoyl-5-[1-(methylideneamino)ethoxy]phenyl]benzamide 2-[[3,5-difluoro-4-(1H-indol-3-yl)phenyl]methoxy]ethanamine 1-methyl-2,3-bis[(4-phenylphenoxy)methoxy]benzene N-[(Z)-(4-hydroxyphenyl)methylideneamino]-3,4-dihydro-2H-1,5-benzodioxepine-7-carboxamide 3-azido-1-[(2,6-dichlorophenyl)methyl]pyrazole N-[(3R)-1-(6-chloroimidazo[1,2-a]pyridine-2-carbonyl)piperidin-3-yl]benzamide N-azido-1,3-benzoxazol-5-amine (2E)-1-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-N'-[1-[3-[(3E,6Z)-octa-1,3,6-trien-3-yl]oxycyclobutyl]ethylideneamino]penta-2,4-diene-1,5-diamine (Z)-N,3-dimethylbutan-1-imine;ethane;2-methylpropane;(E)-3-pyridin-4-ylhex-2-enal [4-(3,5-dichlorophenyl)piperazin-1-yl]-spiro[2H-indole-3,7'-6H-furo[2,3-f][1,3]benzodioxole] 2-[[7-hydroxy-4-(trifluoromethyl)-1H-indole-2-carbonyl]amino]acetic acid N-[4-(5-chlorothiophene-2-carbonyl)piperazin-1-yl]sulfonyl-3,4,5-trimethoxybenzamide (4R)-4-ethyl-2,6,7-trimethyl-N'-[3-[3-(trifluoromethoxy)anilino]pyrazin-2-yl]heptanediamide 2-[4-chloro-3-methylsulfonyl-5-(trifluoromethyl)phenyl]ethanol 3-[5-(4,4-difluoropiperidine-1-carbonyl)thiophen-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile 3-(3,4-dimethoxyphenyl)-1-phenylpropan-1-one;ethane 1,2-diamino-4-[3-methoxy-5-nitro-4-(trifluoromethoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile 2-[(3R)-piperidin-3-yl]-5-phenyl-3H-thieno[2,3-d]pyrimidin-4-one 5-[6-(2,4-difluorophenyl)pyrazin-2-yl]-3H-1,3,4-oxadiazol-2-one 3-[(2R,6S)-9-fluoro-2-methylnonan-4-yl]pyridine (1R,2R)-2-[(2S)-3-methylbutan-2-yl]-N-[1-[6-(1-methylpyrazol-4-yl)isoquinolin-3-yl]ethyl]cyclopropane-1-carboxamide N-[1-(4-chlorophenyl)cyclobutyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide N-(3,5-dimethylphenyl)sulfonyl-1'-[2-(4-fluorophenoxy)ethyl]spiro[4,7-dihydropyrano[4,3-c]pyrazole-6,4'-piperidine]-3-carboxamide 3-(2-azidophenyl)-1,1,1-trifluoro-2-[4-(trifluoromethylsulfanyloxy)phenoxy]propan-2-ol (1R,6S)-3-(4-methylcyclohexen-1-yl)oxycarbonyl-7-oxo-2-phenylsulfanyl-8H-1,8-naphthyridine-6-carboxylic acid 6-(1H-benzimidazol-4-ylmethyl)-2-thiophen-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-[(2R,4S)-1-benzyl-2-(4-chlorophenyl)piperidin-4-yl]acetonitrile 5-bromo-3-(methoxymethyl)-1,4-dihydrothieno[2,3-d]pyrimidin-2-one (Z)-N'-[4-chloro-3-(trifluoromethyl)phenyl]-2-hydrazinylidenebut-3-enimidamide 1-[5-(4-bromophenyl)-3-propyl-2,3-dihydrothiophen-2-yl]cyclohexa-2,4-diene-1-carboxylic acid 1-[3,5-bis(trifluoromethyl)phenyl]-2-methylpropan-2-amine N-[1-(6-aminopyrimidin-4-yl)cyclopentyl]acetamide 3-fluoro-4-[(6S)-2,3,3a,5,6,7,7a-octahydropyrrolo[1,2-c]imidazol-1-yl]aniline 2-[3-(4-cyclopentylpiperidine-1-carbonyl)phenoxy]acetic acid [(3-chloro-1H-indole-2-carbonyl)amino]carbamodithioic acid (2R)-3-[3-oxo-7-[4-(trifluoromethyl)phenyl]-1H-isoindol-2-yl]-2-(2,3,5,6-tetradeuteriophenoxy)cyclobutan-1-one N-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-ethyl-5-oxo-4H-pyrazolo[1,5-a]quinazoline-6-carboxamide N-[4-chloro-3-(5-ethoxy-1,2,4-triazol-3-yl)phenyl]-6-(1H-indol-4-ylmethylamino)pyridine-2-carboxamide N-(4-fluorophenyl)-3-(4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-b]pyridin-5-yl)pyrrolidine-1-carboxamide 2-[2-methyl-4-(trifluoromethoxy)phenyl]benzo[g][1,3]benzoxazole 7-(2,3-dihydropyridin-6-yl)-9,9-dimethylfluorene;ethane;9-(4-methylphenyl)phenanthrene 7-(6-methylheptan-3-yl)naphthalene-2-carboxamide 3,7-dimethylbenzo[f][1]benzoxepine;ethane 1-(2,6-dichlorophenyl)cyclopentane-1-carboxylic acid ethane;1-(2-hydroxyphenyl)-4-methylpentan-3-one 2,6-bis[(4-methylphenyl)sulfonylamino]benzenesulfonic acid N-[(1R)-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-1-yl]-2-[4-(4-chloro-2-fluorophenyl)cyclohexylidene]acetamide 2-methyl-3-[4-(6,7,8,9-tetrahydro-5H-carbazole-2-carbonyl)piperidine-1-carbonyl]pyridine-4-carboxamide 4-chloro-2,6-dimethoxy-N-[(E)-pyridin-2-yliminomethyl]benzamide;hydrochloride [(2R,6S)-1-benzyl-3,4,5-trihydroxy-6-methoxyoxan-2-yl]oxy-bis(prop-2-ynoxy)phosphane [3-[4-(2,3-dihydro-1H-inden-5-yloxy)pyridin-3-yl]oxiran-2-ylidene]azanium 2-[3-[4-(difluoromethoxy)phenyl]propyl]pyrrolidine N-[4-amino-3,5-bis(trifluoromethyl)phenyl]formamide;1-(2-azidoethyl)-2-(trifluoromethoxy)benzene (7R)-N,N-dimethyl-4-oxo-5-[4-[(2-phenoxyphenyl)carbamoyl]phenyl]-6,7-dihydropyrazolo[1,5-a]pyrazine-3-carboxamide 4-(2,3-dimethylimidazol-4-yl)-6-[5-(2,2,2-trifluoroethoxymethyl)thiophen-2-yl]pyrimidine N-(3,4-diethylphenyl)acetamide;ethane;3-[2-methoxy-5-(trifluoromethoxy)phenyl]butanal [2-(6,8-dimethoxyquinolin-4-yl)-3,7-dihydro-1H-pyrrolo[2,3-b]pyridin-5-ylidene]methanediol 1-[1-(2-chlorophenyl)sulfonylpiperidin-4-yl]-5H-pyrazolo[3,4-d]pyrimidin-4-one 4-chloro-5-[5-[(2R)-butan-2-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]-N-ethyl-N-[(4-methoxyphenyl)methyl]-3-methylthiophene-2-sulfonamide (4Z)-2-methylsulfanyl-4-[[2-(pyridin-3-ylmethoxymethyl)phenyl]methylidene]-1,3-oxazol-5-one 3-[2,4,6-tribromo-N-(3-methylbutyl)anilino]propanoic acid N-(6,7-dimethoxyquinazolin-4-yl)-5-(furan-2-yl)-1H-pyrazole-3-carboxamide 2-(4,5-dimethoxy-3,6-dimethylcyclohexa-1,3-dien-1-yl)oxybenzoic acid 3-bromo-N-methylbenzenesulfinamide 1-cyclopentyl-3-[4-methanimidoyl-5-[(5-pyridin-2-yloxyfuran-2-carbonyl)amino]thiophene-2-carbonyl]imidazolidin-2-one N-[4-chloro-3-(trifluoromethyl)phenyl]-2,6-difluorobenzamide 4-amino-5-(1-chloroethenyl)-6-(pyridine-3-carboximidoyl)pyridazine-3,7-dione 2-[3-(4-ethylpiperidin-1-ium-1-ylidene)-5-fluoro-2,6-dimethoxyxanthen-9-yl]-N-(pyridin-3-ylmethyl)benzamide 3-amino-1-[4-(azidomethyl)cyclohexylidene]-N,2-dibenzylbenzimidazol-5-amine 5-[[6-methoxy-4-(2,2,2-trifluoroethylamino)quinazolin-7-yl]oxymethyl]-3-(methylideneamino)pentanal N-(3,4,5-trimethyl-1H-indol-2-yl)benzamide [2-hydroxy-5,7-dimethyl-4-oxo-3-[(E)-2-(4-pyridin-2-ylpiperazin-1-ium-1-ylidene)ethylideneamino]quinazolin-6-yl]azanide 3-[2,6-difluoro-4-(methylsulfanylamino)phenyl]-N-(5-morpholin-4-ylpyridin-3-yl)imidazo[1,5-a]pyrazine-8-carboxamide;methanol 1-[(2S,4R)-1,2,3,4-tetrahydronaphthalen-2-yl]imidazole 7-[2-(4-chlorophenyl)ethyl]-1,3-dimethylpurine-2,6-dione 2-(2,4,6-trimethylphenyl)iminopyrazolidine-3,5-dione N-[2-methoxy-5-(4-methylimidazol-1-yl)-3,6-didehydrocyclohexa-1,5-dien-1-yl]benzamide 2-[8-amino-6-(4,5,7-trifluoro-1H-indol-3-yl)imidazo[1,2-b]pyridazin-3-yl]phenol 2-(N-benzoyl-4-chloroanilino)propanoic acid 1-(4-azidobutyl)anthracene 2-[3-(1,4-diazepan-1-ylsulfonyl)phenyl]ethylcarbamic acid (5-chloropyridin-2-yl)-[3-fluoro-4-[2-(trifluoromethoxy)phenoxy]pyrrolidin-1-yl]methanone (7S)-N-[(Z)-1H-indol-3-ylmethylideneamino]-5-methyl-7-phenyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide N-(2-chloroacetyl)-N-[4-(dimethylsulfamoyl)phenyl]hexadecanamide 5-amino-3-methoxycarbonylpyridine-2-carboxylic acid N-(4,4-difluorocyclohexyl)-4-methyl-2-propanoylbenzenesulfonamide (3S)-1-[2-[4-(3,5-dichloropyridin-4-yl)piperazine-1-carbonyl]-3-fluorobenzoyl]pyrrolidine-3-carboxamide 1-(5,6,7,8-tetrahydroquinolin-4-yl)azepane;dihydrochloride 5-bromo-3-ethoxy-2,6-difluoropyridine (3R)-4-(4,6-dimethylpyrimidin-2-yl)-3-(phenoxymethyl)piperidine-1-carboxylic acid N-ethyl-2-[[5-oxo-4-(3,4,5-trimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide 2-(4-butan-2-ylcyclohexyl)-5,6,7,8-tetrahydroquinoline 3-methyl-5,6-bis(4-methylphenyl)-9H-[1]benzofuro[3,2-b]pyridine ethane;4-N-(3-fluorophenyl)-2,3,5,6-tetramethylbenzene-1,4-diamine 5-(1-ethyl-4-fluoropiperidin-2-yl)oxypyridine-3-carbonitrile 2-azido-N,N'-dimethylthieno[2,3-d]pyrimidine-5-carbohydrazide 2-ethoxy-1H-indole-7-carboximidamide 1-[(E)-2-[4-amino-5-[3-fluoro-5-methyl-2-(oxan-4-yloxy)phenyl]pyrrolo[2,1-f][1,2,4]triazin-7-yl]ethenyl]cyclopropane-1-carbonitrile N-[(1Z)-2-hydroxy-4-(4,6,7,8-tetrahydroimidazo[2,1-c][1,4]oxazin-3-yl)buta-1,3-dienyl]benzamide 1-(3-methoxyphenyl)sulfonylcycloheptane ethane;ethene;1-[(3E)-hexa-1,3,5-trien-3-yl]oxypropan-2-one;1-methyl-4-phenylbenzene 2-[(4-fluorophenyl)methyl]-5,6-bis(1H-inden-1-yl)isoindole 5-[4-methyl-2-(4-phenylmethoxyanilino)pyrimidin-5-yl]pentanal N-[1-(2,3-dihydro-1H-inden-2-yl)ethoxy]-6-methyl-3-[4-(trifluoromethylsulfanyl)anilino]pyridazine-4-carboxamide 3-[[4,5-bis(ethenyl)-2-methoxyphenoxy]methyl]-N,N-dimethylaniline 1-[3-(4-propanoylphenyl)sulfanylcyclobutyl]azetidine-3-carboxylic acid 2-[4-(dimethylamino)phenyl]-1-(6,7-dimethyl-1H-indol-3-yl)butan-1-one 5-[4-amino-3,6-bis(ethenyl)pyridin-2-yl]-N'-methanimidoylfuran-2-carboximidamide 4-[5-(3,5-dimethoxyphenyl)hex-1-enyl]oxane-2,6-dione (2S)-2-[1-(dimethylamino)isoquinoline-3-carbonyl]piperidine-4-carbonitrile 1-[4-[2-[2-(4-tert-butylphenyl)ethynyl]-6,7-dihydrothieno[3,2-b]pyridin-5-yl]piperidin-1-yl]ethanone 2-[3,5-dichloro-4-(6-fluoroindol-1-yl)phenyl]acetic acid 5-[2,3-bis(ethenyl)phenoxy]-N,4-dimethoxypentanamide 2-[4-(2,3-dimethylpentan-2-yl)benzoyl]benzoic acid N-benzyl-3-[5-(difluoromethoxy)tetrazol-1-yl]propanamide N-[(2,6-dichlorophenyl)methyl]-3-ethenyl-1,2-oxazole-5-carboxamide 2-(4-fluorophenyl)sulfonyloxypropanedioic acid N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]-6-methylquinoline-7-carboxamide (E)-4-[[2-(ethenylamino)acetyl]amino]-1-[3-(trifluoromethoxy)phenyl]but-3-ene-2-sulfonic acid 2-(3,4-dihydro-1H-isoquinolin-2-yl)-7-(oxan-4-ylamino)quinoline-3-carbonitrile N-[4-amino-3-(cyclohexa-1,5-dien-1-ylmethoxy)phenyl]-2-(3,4-dichlorophenoxy)acetamide 3-[4-(2,6-dimethoxyphenyl)phenyl]propylphosphonic acid (E)-3-[4-[1,2,5]oxadiazol-3-ylmethoxycarbonyl-[4-(trifluoromethyl)benzoyl]amino]prop-2-enoic acid 4-(furan-2-yl)-3H-pyrazolo[1,5-a][1,3,5]triazin-2-one (2R)-3-methyl-1,4-dioxospiro[2,5-dihydropyrido[2,1-f][1,2,4]triazine-6,1'-cyclohexane]-7-carboxamide 2-[7-[3-(4,5-dimethyl-1H-imidazol-2-yl)phenyl]-6-fluoroisoquinolin-3-yl]-2-oxoacetaldehyde [4-[(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)methoxy]piperidin-1-yl]-(oxolan-2-yl)methanone 7-(3,5-dimethylcyclohexen-1-yl)pyrido[2,3-b]pyrazine (2S)-2,4-bis[4-chloro-2-[2-[2-(cyclopropylamino)ethoxy]ethyl-methylamino]phenyl]butan-1-ol 3-(5-propan-2-ylthiophen-3-yl)-1H-indole 5-[(5-fluoropyridine-2-carbonyl)amino]-3H-1,4-benzodiazepine-7-carboxylic acid 1-(6-methyl-2,3,4,5-tetrahydroindol-1-yl)-2-[3-(tetrazol-1-yl)azetidin-1-yl]ethanone 7-(2,5-dimethyl-3H-furan-2-yl)-N-[2-(dimethylamino)phenyl]heptanamide 1-[3-(benzylamino)-2,2-difluorocyclobutyl]ethanone 3-[(2E)-2-(6,7,8,9-tetrahydrocarbazol-3-ylmethylidene)hydrazinyl]benzoic acid 7-(6,8-difluoro-1-iodoquinazolin-4-ylidene)-3,5-bis[2-(2-methylpyridin-3-yl)ethenyl]fluoren-9-ol N-[2-(3,5-dimethylanilino)pyrimidin-4-yl]acetamide 4-(benzenesulfonyl)-1-N,3-N-bis[2-[butyl-[3-(methylideneamino)propyl]amino]ethyl]benzene-1,3-diamine 2-cyclohexyl-4-methoxycarbonylbenzenesulfonic acid 4-[(3,5-difluorophenyl)methyl]-N-[2-ethoxy-5-[(E)-prop-1-enyl]pyridin-3-yl]piperazine-1-carboxamide 6-chloro-N-[[2-(furan-3-yl)pyridin-4-yl]methyl]pyrimidin-4-amine 6-methoxy-4-oxo-5,7-dihydro-3H-1,3-benzoxazine-2-thione N-[2-[N-ethylsulfonyl-4-(pyridin-2-ylsulfamoyl)anilino]ethyl]acetamide 2-[(4E,5Z)-3-ethylidenehepta-1,5-dien-4-yl]-6-methoxy-N-(3-propanoylphenyl)pyridine-4-carboxamide 6-[2-(2,3,4,5-tetrafluorophenyl)ethyl]-2,3,4,5-tetrahydropyridine 2-(3-chlorophenyl)sulfonyl-8-(dimethylsulfamoyl)-7-hydroxy-5,6-dihydro-4H-1,3-benzothiazole (E)-3-[4-(2,6-dimethoxyphenyl)-1,3-thiazol-5-yl]prop-2-enoic acid N-(2,3-dioxopropyl)-N-[4-[(2-phenylpyrazol-3-yl)sulfamoyl]phenyl]butanamide (2S)-1-azido-3-[1-(6-fluoronaphthalen-2-yl)sulfonylpiperidin-4-yl]propan-2-ol [3-(2-hydroxyethylamino)cyclopentyl]-spiro[3,4-dihydrochromene-2,3'-pyrrolidine]-1'-ylmethanone 4-[3-(5,7-dimethyl-1H-indole-2-carbonyl)phenyl]-1-methylimidazolidin-2-one 1-(2,3,4a,5,7,8,8a-octahydropyrano[3,4-b]pyrazin-1-yl)-3-[6-(1H-pyrazol-5-yl)isoquinolin-3-yl]propan-2-one (5R,10S)-9-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-7-oxa-2,13-diazaspiro[4.6]undecan-10-one 4-[(2R)-4-tert-butylsulfanylpiperazine-2-carbonyl]-2-N,5-N-diethylpyridine-2,5-dicarboximidamide [6-amino-2,3-bis(methylideneamino)phenyl]-ethylazanium N-[2,4-difluoro-3-[5-(furan-3-yl)pyridin-2-yl]oxyphenyl]-6-oxo-1H-pyridazine-5-carboxamide 4-[[4-(4,5-dimethylpyridin-2-yl)piperazin-1-yl]methyl]benzamide (6R)-7-amino-3-(5-tert-butylthiophene-2-carbonyl)-2-[4-(dimethylcarbamoyloxymethyl)phenyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-9-olate N-(2-methyl-1,3-dihydroisoindole-5-carbothioyl)benzamide 2-bromo-N-(3-methylsulfanylphenyl)-N-prop-2-enylbenzamide 1-[(3R)-1-acetylpiperidin-3-yl]-N-methoxy-5H-pyrrolo[2,3-b]pyrazine-2-carboxamide (4-methoxyphenyl)iodanium;tetrafluoroborate 2-[1-(3,4-dichlorophenyl)-5-(trifluoromethylsulfanyloxy)pyrazole-4-carbonyl]propanedinitrile (2S,5S)-5-azido-1-[5-(trifluoromethyl)pyridin-2-yl]piperidine-2-carboxylic acid 2-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,11-tetraen-3-ylamino)pyrazol-1-yl]acetaldehyde 2-[(3R)-7-fluoro-5-methyl-4-oxo-2,3-dihydropyrido[3,2-b][1,4]oxazepin-3-yl]-N-propan-2-ylacetamide (E)-3-[4-[2-[6-(diethylaminomethoxy)pyridin-2-yl]thieno[2,3-b]pyridin-5-yl]phenyl]prop-2-enoic acid N-[4-(chloromethyl)phenyl]-2-hydroxy-3,3a,4,5-tetrahydro-1H-indole-2-carboxamide N-[5-chloro-2-[4-(3,5-dimethylphenyl)piperazin-1-yl]phenyl]sulfanyl-4-fluoroaniline 2-azido-6,7-dimethoxyquinazoline 2-[4-(cyclohexanecarbonyl)piperidin-1-yl]-1,3-thiazole-5-carboxamide 3-[(4R,7S)-4-benzyl-1-methoxycarbonyl-5-oxopyrrolidine-2-carbonyl]-1H-indole-6-carboxylic acid 1-[2-(dimethylamino)ethyl]-5-(4-oxo-3H-quinazolin-2-yl)indole-7-carboxamide 5-(2,6-dimethoxyphenyl)sulfanyl-2-hydroxyisoindole 3-(azidomethyl)-2,4-dichloroaniline 3-(2,6-diphenylanilino)butanoic acid 2-(cyclohexylmethoxy)-N-[1,2,4]triazolo[5,1-b][1,3]thiazole-5-carboxamide 4-[5,6-dichloro-2-(hydroxymethyl)pyridin-3-yl]benzonitrile 1-cyclopropyl-6,7-difluoro-N-[5-(3-methoxyazetidin-1-yl)pyridin-2-yl]sulfonylquinolin-4-imine ethane;3-methyl-7-phenyl-2,4-dihydro-1H-benzo[f]quinoxaline 1-(2-methylsulfonylethynoxy)-3-phenylbenzene 2-(5-methoxypyridin-3-yl)-4-propan-2-ylpyridine ethene;2-methyl-7-(2-phenylpropyl)naphthalene 2-[6,7-dimethyl-8-(N'-propanoylcarbamimidoyl)naphthalen-1-yl]acetic acid 2-[(5S,10bR)-7-methoxy-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-methoxyphenol (3R)-6,8-dichloro-2-[[5-(cyclopropylmethoxy)pyridin-2-yl]methylsulfinyl]-4,5-dihydro-3H-1-benzazepine 1,2-bis(3,4-diethylphenyl)guanidine;hydrochloride 3-(6-bromonaphthalen-2-yl)sulfanylpropanenitrile 2-[(2Z,5R)-2-[(Z)-[4-(2-fluorophenoxy)phenyl]methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid [3-(5-amino-1,2,4-oxadiazol-3-yl)azetidin-1-yl]-[4-(4-methoxyphenyl)cyclohexa-1,3-dien-1-yl]methanone 4-[3-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)anilino]benzenesulfonic acid (Z)-N-[[4-chloro-3-(5-oxo-1,2,4-oxadiazolidine-4-carbonyl)phenyl]methyl]-4-(2-hydroxyethylamino)but-2-enamide 4-(3,5-dimethoxyphenyl)sulfanyl-2-ethoxypyridine 2-[(6S,7R)-7-(4-chloro-3-methoxyphenyl)-1,4-oxazepane-6-carbonyl]-5H-pyrrolo[2,3-b]pyrazine-7-carbonitrile 2-[5-bromo-4-(1,3-dioxan-2-yl)-6-methoxypyridin-2-yl]benzoate (2S)-4-[2,6-dimethoxy-4-(3-oxomorpholin-4-yl)benzoyl]-2,5-dimethylpiperazine-1-carboxylic acid (2S,5R)-1-[3,5-bis(trifluoromethyl)phenyl]sulfonyl-5-N-phenyl-4-N-propan-2-ylpiperazine-2,5-dicarboxamide 2-(4-but-3-enylphenyl)-6,7-difluoronaphthalene N-[(2S)-1-cyclohexa-1,3-dien-5-yn-1-yl-3-(3,5-difluorophenyl)-4-[(3-ethylphenyl)methylamino]butan-2-yl]pyridine-4-carboxamide (3aR,6aS)-2-[2-[4-(trifluoromethyl)phenyl]acetyl]-5-[(E)-2,3,3a,4,5,6,6a-octahydrocyclopenta[b]furan-3-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-5-carboxylic acid 4-bromo-2,6-dichloro-N'-hydroxybenzenecarboximidamide N-(diaminomethylideneamino)-2,4,6-triiodobenzamide 6-[4-(3,4-dichlorophenyl)sulfonylpiperazine-1-carbonyl]-2H-isoquinolin-1-one 5-fluoro-N'-[(4-fluorophenyl)methyl]-2,3-dihydropyridine-6-carboximidamide 3-[2-(1H-indol-5-yl)ethoxy]propanal 3-(1,2,5-oxadiazol-3-yl)-6-[(4-phenylpyridin-2-yl)amino]-2H-naphthalen-1-one 3-(2,4,5-trimethylphenyl)-1,3,5-oxadiazinan-2-one 5-bromo-2,4-dimethylphenol;ethane 2-[6-(3,5-dichlorophenyl)-1H-benzimidazol-2-yl]ethanamine 3-(1,2,4-triazol-1-yl)-5-(trifluoromethyl)benzoic acid 2-[1-(3,5-difluorophenyl)-4,6-difluorobenzimidazole-2-carbonyl]oxyethylazanium (2R,4S)-N-[1-[(4-cyanophenyl)methyl]pyrazol-4-yl]-4-hydroxypiperidine-2-carboxamide 2-(3,4-dichlorophenyl)-6-methyl-8-pyrimidin-5-yloxypyrido[2,3-d]pyrimidin-7-one 2-tert-butyl-6-[(2,4-dihydroxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-[2,6-difluoro-4-(methoxyamino)phenyl]propanamide;4-(4-ethylphenyl)piperazine 5-[[(Z)-3,4,5-trihydroxyoct-3-enyl]amino]benzene-1,2,3-triol 5-(methylamino)pyrazolo[1,5-a]pyridine-3-carbonitrile;6-piperidin-4-yloxyimidazo[2,1-b][1,3]thiazole 2-benzylsulfanyl-N,N-dibutylacetamide 4-hydroxy-N,5-dimethyl-2-[[2-[(E)-3-oxoprop-1-enyl]cyclohepta-2,4,6-triene-1-carbonyl]amino]benzamide 5-[(Z)-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)iminomethyl]benzene-1,3-diol 1-[(6,7-dimethylnaphthalen-2-yl)methyl]pyrrole (3E)-5-bromo-3-[(4Z,6Z)-4-ethylundeca-4,6,8-trienylidene]-1H-indol-2-one 5-fluoro-N-[[1-(3-methylbutanoyl)piperidin-4-yl]methyl]pyridine-2-carboxamide (6S,9aS)-N-benzyl-2-[(2R)-butan-2-yl]-8-[(4-hydroxyphenyl)methyl]-6-[(3-methoxyphenyl)methyl]-4a,7,8,9a-tetrahydropurine-6-carboxamide 1-methyl-4-[6-[(5R)-5-(1H-pyrazol-5-ylamino)cyclohexen-1-yl]pyridin-3-yl]piperazin-2-one 3-methoxy-1-[(E)-2-nitroethenyl]-9H-fluorene N-[1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl]pyrrolidine-3-carboxamide 3-[4,5-dihydroxy-6-(4-nitroanilino)-1H-pyrrolo[2,3-c]pyridine-2-carbonyl]oxyazetidine-1-carboxylic acid 2-[5-(cyclopentyloxymethyl)-3-(3,5-difluorophenyl)pyrazol-1-yl]ethanol;5-oxo-4H-pyrazolo[1,5-a]quinazoline-3-carbonitrile 2-[6-bromo-1-(4-ethylcyclohexen-1-yl)-5-fluoronaphthalen-2-yl]oxyacetic acid N-(6-fluoro-2,2-dimethyl-1,3-benzodioxol-5-yl)-4-phenylpyrimidine-5-carboxamide N-[5-cyano-2-(4,6-dimethylpyrimidin-2-yl)pyrazol-3-yl]-1H-indazole-5-sulfonamide 4-[(3S)-4-cyclopropylmorpholin-3-yl]-2-methylpyrazole-3-carboxamide 2-[3-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]indol-1-ium-3-ylidene]propanedinitrile;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide 4-N,4-N,6-trimethylthieno[2,3-d]pyrimidine-2,4-diamine N-[1-(4-methylsulfonylphenyl)ethenyl]butanamide [4-methoxy-2-(3,6,7,8-tetrahydrocyclohepta[d]imidazol-2-yl)phenyl]boronic acid 6-[1-(dimethylamino)ethyl]-5-fluoro-2,3-dihydroinden-1-one;N'-methyl-N-[(4-oxo-3H-quinazolin-7-yl)methyl]acetohydrazide N-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-3-yl]-5-propan-2-yl-7,8-dihydroquinoline-6-carboxamide [2-hydroxy-3-[[4-methoxycarbonyl-2-(oxan-4-ylamino)phenyl]diazenyl]phenyl]chloranium 5-amino-3-[2-(3,4-difluorophenyl)ethyl]-1H-indole-6-carbonitrile;ethane (6R)-N-benzyl-10-ethoxy-8,11,14-triazatetracyclo[7.6.0.02,7.010,15]pentadeca-1,9,12,14-tetraen-13-amine 3-[4-(1,2-dihydroimidazo[4,5-b]pyrazin-5-yl)pyrazol-1-yl]propanenitrile;hydrochloride 3-[5-(1,4-diazepan-1-yl)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenol N-(furan-2-ylmethylideneamino)-3,4-dihydronaphthalene-1-sulfonamide 1-[3,5-dichloro-2-hydroxy-4-(trifluoromethyl)phenyl]ethanone 7-(2,6-dichloro-3,5-dimethoxyphenyl)-5H-pyrimido[4,5-d][2]benzazepine (3-chloro-4-iodophenyl)boronic acid 1-(3,4-dihydro-2H-1,5-benzodioxepine-7-carbonyl)piperidine-2-carboxamide 3-(4,5-dimethylfuran-2-yl)-3-iminopropanenitrile (2S)-2,5-diamino-6-[[benzyl-[[1-[3-(carboxymethoxy)propanoyl]pyrrolidine-2-carbonyl]amino]carbamothioyl]amino]hexanoic acid 2-methyl-5-[[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yloxy)piperidine-1-carbonyl]amino]benzoic acid 2-[4-(benzimidazol-1-yl)phenyl]propanamide (1R)-2,2-difluoro-N-[4-[5-[3-(propanoylamino)phenyl]pyrazolo[3,4-b]pyridin-2-yl]cyclohexa-1,3-dien-1-yl]cyclopropane-1-carboxamide ethane;N-[(E)-1-(4-methylphenyl)prop-1-enyl]-3-nitrobenzamide 2-[4-(4,6-dimorpholin-4-yl-1H-pyrrolo[3,2-c]pyridin-2-yl)-1H-benzimidazol-2-yl]-5-thiophen-2-ylphenol [(2S,4R)-1-[5-fluoro-6-(3H-inden-1-yloxymethyl)pyrimidin-4-yl]-4-hydroxypyrrolidin-2-yl]methanol 3-(3,4-dichlorophenyl)-1-(2-piperidin-1-ylethyl)indole 7-[1-(cyclopropylmethylamino)-2,3-dihydro-1H-inden-4-yl]-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-5-carboxamide N-(2-methoxy-4-nitrophenyl)-1-pyridin-3-ylethanimine 6-[(2S)-1,1-difluoropropan-2-yl]oxy-5-methylpyridine-3-carboxylic acid (Z)-2-cyano-3-[5-methoxy-2-(trifluoromethyl)phenyl]prop-2-enamide 5-(2-bromophenyl)imino-4,6-dihydroxyiminocyclohex-2-en-1-one 4-N-azidooxy-1,2-dimethylbenzene-1,4-disulfonamide N-[5-(3,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-4-(morpholin-4-ylmethyl)benzamide 5-fluoro-2-[[3-(trifluoromethyl)pyridin-2-yl]amino]benzonitrile 2-tert-butyl-7-[(1-methoxypyridin-1-ium-3-yl)methyl]-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 4-[(1,3-benzodioxol-5-ylmethylamino)methyl]-N'-hydroxypyridine-2-carboximidamide N-methyl-6-[2-(methylamino)ethoxy]pyridine-3-carboxamide 3-azido-2-(9H-fluoren-1-ylmethoxy)thiophene 4-azido-1,2,3-trifluoronaphthalene 1-N-(3,5-dichlorophenyl)sulfanyl-2-N,2-N-diethylpropane-1,2-diamine 7-[(E)-(2,3-dimethoxyphenyl)methylideneamino]sulfanyl-3-(naphthalene-2-carbonyl)-1H-quinazoline-2,4-dione 4-[4-(diethoxyphosphorylmethyl)piperidine-1-carbonyl]phenol 3-(2,4-difluorophenyl)-5-hydroxy-8-oxa-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-12-one (7Z)-3,4-bis[2-chloroethyl(methylsulfonylamino)oxy]-9H-fluoren-1-amine N-[4,5-bis(ethenyl)cyclohepta-1,3,6-trien-1-yl]benzamide 4-[(2,3-dimethylcyclopentyl)amino]pyridine-2-carbonitrile 4-ethyliodanuidyl-N',N'-dimethylbenzenecarboximidamide N-(4-chlorophenyl)-2,5-dimethylhexanamide 1-[4-chloro-3-(5-ethoxycarbonylcyclohexa-2,4-dien-1-yl)oxyphenyl]pyrrolidine-3-carboxylic acid ethane;3-(1,4-oxazepan-4-ylmethyl)benzoic acid [7-(2,3-dimethylphenyl)sulfonyl-4a-(hydroxymethyl)-1,3,4,5,6,8,8a-octahydro-2,7-naphthyridin-2-yl]-cyclohexylmethanone (2S)-3-[4-(trifluoromethyl)phenyl]sulfonyloxybutanedioic acid N-(6-fluoropyridin-3-yl)-1,2,4-oxadiazole-5-carboxamide N-(4-chlorophenyl)-2,5-dimethoxybenzenecarboximidate 2-[(Z)-1-cyano-3-cyclopropylbut-2-enyl]sulfanyl-4-methyl-N-phenylbenzamide 1-(2-hydroxy-3H-pyrrol-4-yl)-5-methyl-N-[(Z)-5-oxopent-3-en-2-ylideneamino]pyrazole-3-carboxamide 6-[2,3-dichloro-4-(3-morpholin-4-ylsulfonylpropoxy)phenyl]pyridine-2-carboxamide 2-[4-(1H-indole-3-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 2-[4-methoxycarbonyl-N-(1,3-thiazol-5-yl)anilino]octanoic acid 1-(6-methylpyridine-3-carbonyl)piperidine-4-carboxylic acid;2,2,2-trifluoroacetic acid (3S)-1'-(4-methylsulfonylphenyl)spiro[1H-indole-3,3'-piperidine]-2-one 5-[4-(3,5-dichlorophenyl)piperazin-1-yl]pyridazine N-(4-chlorophenyl)formamide;ethane;3-[7-methoxy-1,1-dimethyl-2-(naphthalene-2-carbonylamino)inden-5-yl]propanoic acid N-[(3S,4R)-1-(2-cyclohexylacetyl)-4-(5-methyl-1H-1,2,4-triazol-3-yl)pyrrolidin-3-yl]oxane-4-carboxamide 5-[(2-ethoxyphenyl)methylidene]imidazolidine-2,4-dione 5-(7,8-dimethoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-N'-piperidin-4-yl-3-propan-2-ylpyrazolo[1,5-a]pyrimidine-7-carboximidamide;hydrochloride N-[3-[7-[(2,6-difluorophenyl)methoxy]-1H-indazol-3-yl]phenyl]propanamide 4-[(E)-2-[5-methylsulfonyl-2-(trifluoromethoxy)phenyl]ethenyl]benzoic acid 1-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylacetyl]-N-(2-fluoropyridin-3-yl)-4-phenylpiperidine-4-carboxamide 3-(2-azidooxy-5-methylphenyl)-N,N-diethylpropanamide 2-(4-methoxy-N-propylanilino)octanoic acid 6-chloro-1,3-dimethylimidazo[4,5-b]pyridin-2-one 3-methyl-4-[[2-(trifluoromethyl)phenyl]diazenyl]aniline 4-[7-amino-8-butan-2-yloxy-6-(3,3-difluorocyclobutyl)imidazo[1,5-a]pyrazin-3-yl]benzaldehyde;5-methoxy-2-pyridin-2-ylpyrimidine (1S)-2,2-difluoro-6-(4-nitrophenyl)sulfonylcyclohexan-1-ol N-(4,5-dihydrothieno[3,2-d][1]benzoxepin-9b-ylmethylideneamino)propanamide 1-azido-2,3-bis(chloromethyl)-4-methoxybenzene N-methoxy-6,7-dihydrobenzo[a]quinolizin-11-ium-9-imine 2-(azetidin-1-yl)-6-bromopyrido[3,4-d]pyrimidine 1-azido-6-(trifluoromethoxy)naphthalene 1-(5,8-dichloro-4,6,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-11-yl)pyrrolidine-2,5-dione 3-(2-methoxy-5,7-dimethylquinolin-6-yl)-N-[4-methyl-5-(trifluoromethyl)pyridin-2-yl]benzamide N-(4,5-dimethyl-1H-pyrazol-3-yl)-2-[(4-phenyl-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide 2-[(3S)-4-[5-[2-(methylaminomethyl)phenyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl]morpholin-3-yl]acetamide N-methyl-4-[(2S,3R)-2-[[4-(1,3-thiazol-5-yl)phenoxy]methyl]-4-(trifluoromethoxy)pentanoyl]piperazine-1-carboxamide 2-[(E)-4,5-difluoronon-5-enyl]naphthalene N-[4-[2-[(3Z,5E)-3,6-dimethylhepta-1,3,5-trien-4-yl]-5H-pyrrolo[2,3-b]pyrazine-7-carbonyl]pyridin-2-yl]methanesulfonamide 2-azidosulfanyl-1,3-dinitrobenzene N-[(3,4-dimethylphenyl)methoxy]-2-(5-methylpyridazin-3-yl)propanamide (2E)-N,5,8-trimethyl-3-[[4-[(Z)-1-(3-morpholin-4-ylpropylamino)pent-1-enyl]phenyl]methyl]-N-[(4-methylsulfonylphenyl)methoxymethyl]deca-2,4,6-trienethioamide 5-(2-cyanophenyl)-2H-triazole-4-carboxylic acid 2-azido-5,8-difluoroquinoline 2-[2,6-dimethyl-4-(1H-pyrazol-5-yl)phenoxy]acetic acid;ethane 2-[3,5-bis(trifluoromethyl)phenyl]-2-methoxyacetaldehyde;1-butan-2-ylidene-4-fluorocyclohexane 2-(1,3-benzothiazol-4-ylsulfonylamino)thiophene-3-carboxylic acid N-methyl-1,3,5-tri(propan-2-yloxy)benzenesulfonamide N-[3-(dimethylamino)propyl]-1,2-dimethylindole-5-carboxamide 3-methyl-1,2-diphenyl-4H-pyrimidine N-[(3R,4S)-1-[6-amino-5-(trifluoromethyl)pyrimidin-4-yl]-4-hydroxypyrrolidin-3-yl]acetamide N-[6,7-dichloro-5-(hydroxymethyl)pyridin-2-yl]quinoline-4-carboxamide 2-[(1R)-1-azidoethyl]-5-fluoro-3,4,6-trimethoxypyridine [5-cyclopropyl-4-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonylamino)pyridine-3-carbonyl]carbamic acid 2-[4-(3,5-difluorophenyl)piperazine-1-carbonyl]-7-thia-4,10,12-triazatricyclo[6.4.0.02,6]dodeca-1(8),9,11-trien-3-one;hydrochloride 6-methoxy-3,9-dimethyl-2H-benzo[f]isoindole-1,3'-dione 1-N,3-N-bis[(E)-(4-hydroxyphenyl)methylideneamino]benzene-1,3-dicarboxamide;cyclopenta-2,4-dien-1-one N-[(3-cyanophenyl)methyl]spiro[2.5]octane-6-carboxamide;propane 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;ethane 2,3-diamino-N-ethylbenzamide 4-(1,3,3a,5,6,6a-hexahydrocyclopenta[c]pyrrol-2-yl)-N'-hydroxypyridine-2-carboximidamide 3-[(4-methylphenoxy)methyl]-2,3-dihydrothieno[3,4-b][1,4]oxazine N-[(2S)-2-[4-(cyclobutylmethoxy)phenyl]-2-hydroxyethyl]-6,7-dihydro-1H-benzimidazole-4-carboxamide 2-(7,8-dihydronaphthalen-1-yl)benzenesulfonic acid N-methyl-N-[1-(6-methylpyridin-2-yl)ethyl]-3,5-bis(trifluoromethyl)aniline 3-N,7-N-bis(2-aminophenyl)naphthalene-2,7-disulfonamide 4-(2,6-dichlorophenyl)-5H-1,3-thiazole-4-carboxylic acid 4-(5,7-difluoro-2H-1,3-benzoxazol-6-yl)-N'-methanimidoylpyridine-3-carboximidamide (6S)-7-[[2-(4-aminophenyl)-1,3-benzoxazol-5-yl]methoxy]-3-ethoxy-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-[4-(2,6-difluorophenoxy)piperidine-1-carbonyl]benzoic acid 3-[4-[2-(8-fluoro-5-methyl-1,4-dihydroquinoxaline-6-carbonyl)-3-oxo-1H-isoindol-5-yl]piperazin-1-yl]azetidine-1-carboxylic acid 4-[3-[2-(dimethylamino)ethyl]phenyl]-1,2,5-oxadiazol-3-amine;hydrochloride N-(1,3-benzodioxol-5-yl)-2-(3-cyclopropylindol-1-yl)-N-methylacetamide 2-[(3,4-dimethylphenyl)sulfonylamino]-6-thiophen-2-yloxycyclohexene-1-carboxamide 1-(2,4-dinitrophenyl)piperidine 4-[2,3-bis(ethenyl)phenyl]-7-methoxyquinoline (5Z)-3-(5,6,7-trimethoxyquinolin-4-yl)oxy-2,7-dihydrochromene-2-carboxylic acid [2-[(2S)-1-(4-ethylphenyl)sulfonylpiperidin-2-yl]acetyl]carbamic acid 4-(2,5-dioxo-1,3-thiazolidin-3-yl)-N-[2-fluoro-5-methoxy-4-(1,1,1-trifluoropropan-2-ylideneamino)phenyl]butanamide 1-(2,6-difluorophenyl)-3-[4-methyl-5-oxo-1-propan-2-yl-7-[[[1-[[4-(trifluoromethoxy)phenyl]methyl]piperidin-4-yl]amino]methyl]-4H-pyrazolo[3,4-b]pyridin-6-yl]urea (2S)-3-cyclohexa-1,5-dien-1-yl-2-[[6-methoxycarbonyl-7-propanoyl-4-[3-[(E)-2-pyridin-2-ylethenyl]phenyl]-2,3-dihydroquinoxalin-1-yl]sulfonylamino]propanoic acid N-[5-(2,3-dihydro-1H-inden-4-yl)-2-formamidophenyl]acetamide N'-hydroxy-3-[methyl(2,2,2-trifluoroethyl)amino]pyrazine-2-carboximidamide 2-[4-hydroxy-5,8-dimethyl-3-(phenylsulfanylmethyl)naphthalen-1-yl]oxyacetic acid 2-(6,8-difluoro-3,4-dihydro-2H-quinoline-1-carbonyl)-N,5-dimethylpyrazole-3-carboxamide (3-bromophenyl)methanetriamine;4,4,5,5,6,7,8,9,10,11,12,13,14,15,16,17-hexadecafluoro-2-[4-(2-methylpropoxy)benzoyl]-1-oxa-3-azoniacyclohexadec-2-ene 4-(2-methoxyphenyl)-N,2-dimethylbutanamide (2-butan-2-yl-1-methylcyclopenta-2,4-dien-1-yl)benzene 2-[4-(cyclobutylsulfanylamino)phenyl]-N-[(3S,5Z)-5-methylidenehepta-1,6-dien-2-yl]quinazoline-7-carboxamide (5E)-1-(4,6-dimethylpyrimidin-2-yl)-4,7-dihydropyrazolo[3,4-d]pyrimidin-6-one 3-[6,7-dimethoxy-2-[4-(trifluoromethyl)phenyl]quinolin-4-yl]-3-oxopropanoate N-(cyclopropylmethyl)-1'-(pyridine-3-carbonyl)spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 5-fluoro-2-[[(3Z,4E)-6-methoxy-1-pyridin-3-ylhepta-3,4,6-trien-2-ylidene]amino]phenol N-[4-(1,3-oxazol-5-yl)phenyl]-N-[(4-nitrophenyl)methyl]benzamide 2-[[7-(benzylamino)-1-oxo-3,4-dihydroisoquinolin-2-yl]methyl]-N-tert-butyl-3H-benzimidazole-5-carboxamide 6-[3-(oxan-4-ylmethoxy)phenyl]-4,5-dihydro-1H-pyrimidine (2S)-3-[[4,5-dimethyl-1-[4-(trifluoromethoxy)phenyl]pyrazole-3-carbonyl]amino]-2-hydroxypropanoic acid 2-methyl-4-(1,3-thiazol-5-yl)pyrimidine-5-carboxylic acid 1-[[2,5-difluoro-4-(2-hydroxypropan-2-yl)phenyl]sulfamoyl]piperidine-3-carboxylic acid (6R)-5-amino-3-methyl-7,9-dihydro-6H-[1]benzothiolo[2,3-d]pyrimidine-4-thione (6S)-7-acetyl-6-[5-chloro-2,3-bis(phenylmethoxy)phenyl]-1,4-oxazepane-4-carboxylic acid 2-benzylsulfanyl-N,N',N'-trimethylbenzohydrazide 2-(4-fluorophenyl)-N-[2-[5-methyl-6-(trifluoromethyl)pyridin-3-yl]propan-2-yl]acetamide ethane;1-[4-(5-phenylsulfanylquinolin-8-yl)sulfanylpiperidin-1-yl]butan-2-one N-[(1S,3R)-3-[[4-(1H-pyrazol-5-ylmethylcarbamoylamino)benzoyl]amino]cyclohexyl]pyrazine-2-carboxamide N-[1-[2-(2-hydroxyphenyl)-7-methylquinazolin-4-yl]piperidin-3-yl]cyclopropanecarboxamide 2-fluoro-5-methylbenzenesulfonamide 7-(2,3-dimethylphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 4-(3,5-difluoroanilino)-7H-purine-6-carboxamide 1-[2,3-difluoro-4-(2-hydroxy-4-methylphenyl)sulfanyloxyphenyl]ethanone;ethane 4-(2,3-dihydro-1H-inden-5-yloxy)-1H-triazole-5-carboxylic acid 3-[[(2S)-3,5-dimethyloxan-2-yl]methoxymethyl]benzamide 2-[(3,4-dimethoxyphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrile 2-[7-[(3,5-dimethoxyphenyl)sulfonylamino]-6H-pyrido[2,1-c][1,2,4]triazin-9-ium-10-yl]-N,N-dimethylacetamide 2-azido-N,3,4,5,6-pentamethylaniline 5-[(2,4-dichloropyrimidin-5-yl)-(4-nitrobenzoyl)amino]naphthalene-2-sulfonic acid (3Z)-N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]imino-4-methoxybutanamide N'-[1-[5-(diethylamino)pentanoyl]azepan-4-yl]benzohydrazide 1-[6-(3-cyclopentylpropanoyl)pyridin-2-yl]but-3-en-2-one 5-(2,3-dichlorophenoxy)-N'-hydroxypyrazine-2-carboximidamide [(1S,3R)-2,2-dimethyl-3-phenylcyclopropyl]-spiro[4H-isoquinoline-3,4'-piperidine]-1'-ylmethanone 2-[1,3-benzoxazol-2-ylmethyl-[(2S)-2-hydroxy-2-phenylethyl]amino]acetic acid 2,4-dioxo-1H-pyrimidine-5-sulfonamide 1-[4-(2-bromophenyl)piperazine-1-carbonyl]cyclohexan-1-ol 2-[3-[(5R)-3-amino-5-methylpiperidin-1-yl]-6-[hydroxy-(4-morpholin-4-ylphenyl)methyl]-5,8-dihydroimidazo[1,2-a]pyrazin-7-yl]acetamide N-[2,6-difluoro-4-(triazolo[1,5-a]pyridin-8-yl)phenyl]-2-methoxybenzamide 3-(2,6-dimethylphenyl)-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-4-one 2-(2-chlorophenyl)-5-methylfuran 5-[2-(2,3-dimethylimidazol-4-yl)ethynyl]pyridine-3-carbonitrile N-(4-anilinophenyl)-2,6-dichloro-N-propylpyrimidin-4-amine 2-[5-(4-hydroxyphenyl)-2-oxo-1H-pyrrol-3-yl]propanoic acid N-(5-acetamido-3,4-dimethoxycyclohexa-1,5-dien-1-yl)benzamide 3,5-dimethyl-4-(2,4,6-triphenylcyclohexa-1,3-dien-1-yl)phenol 3-(2,6-dioxopiperidin-3-yl)-4-hydroxy-1-oxo-N-phenyl-2H-isoquinoline-7-carboxamide 2-(2,6-dioxopiperidin-3-yl)-5-[4-(1-methylidene-3-phenyl-2H-isoquinolin-7-yl)piperazin-1-yl]isoindole-1,3-dione (2S)-N-[5-[4,5-bis(ethenyl)-1H-pyrrol-3-yl]pent-4-ynyl]-N'-ethyl-4,4-difluoro-N-propan-2-ylpyrrolidine-2-carboximidamide 5-amino-3-(4-bromophenyl)-2,6-dihydropyrazolo[4,3-d]pyrimidin-7-one 3-(4-chlorophenyl)sulfanyl-2,5-dihydroxybenzoic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-[4-(diethylaminomethylideneamino)phenoxy]acetamide N-(4-acetylphenyl)sulfonyl-6-fluoronaphthalene-2-carboxamide N-[1-(cyclohexa-2,4-dien-1-ylmethyl)piperidin-3-yl]-6-[4-(4-fluorophenyl)piperazine-1-carbonyl]-4,5-dihydrothieno[3,2-d][1]benzazepine-2-carboxamide 3-(2,4-difluorophenyl)-5-[[6-ethyl-7-(hydroxymethyl)-8-methoxy-4H-imidazo[1,5-a][1,4]benzodiazepin-3-yl]methylamino]thiophene-2-carboxylic acid 4-[5-(azetidine-1-carbonyl)pyrazin-2-yl]oxypiperidine-1-carboxylate 2-[(2-chloroacetyl)amino]-3-hydroxybenzoic acid 2-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]acetic acid 4-[3,5-difluoro-4-(4-methylpiperazine-1-carbonyl)phenyl]-5,8-dimethoxychromen-2-one N-[1-[2-[(3,5-dimethoxyphenyl)methyl]-6-hydroxy-3,4-dihydro-1H-isoquinolin-7-yl]cyclopropyl]acetamide 3-[(3E)-hexa-1,3,5-trien-3-yl]sulfonyl-N-prop-2-ynoxybenzamide N-[3-[(7-bromo-4,6-dihydroimidazo[2,1-c][1,4]oxazin-5-yl)methylamino]phenyl]butanamide 5-phenyl-2-(4-piperazin-1-ylcyclohexen-1-yl)pyrimidine [2-(3,5-dimethylphenyl)cyclopropyl]-(4-methylpiperidin-1-yl)methanone 3-(3-cyclopropylpropoxy)-5-[2-[1-methylidene-3-[6-methyl-7-oxo-4-(trifluoromethyl)pyrazolo[3,4-d]pyridazin-2-yl]pyrazol-1-ium-2-yl]ethoxy]benzonitrile (3S)-N'-ethyl-2,3-dihydroxy-4,5-bis[(3R)-3-phenylbutanoyl]benzohydrazide 2-[[1-(5-chloropyrimidin-4-yl)piperidin-3-ylidene]methylsulfonyl]-5-fluoropyridine 2-amino-1-[4-(3,5-dimethoxyphenyl)piperidin-1-yl]propan-1-one;hydrochloride 1-(3,4-dihydro-2H-naphthalen-1-ylidene)pyrrol-1-ium 2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-1-[4-[2-[2-fluoroethoxymethyl-[(3R)-oxolan-3-yl]amino]ethyl]phenyl]guanidine 2-[(7R)-6-methoxycarbonyl-5-oxo-4,7-dihydro-1H-pyrazolo[3,4-b]pyridin-7-yl]acetic acid 2-[(1S)-1,2-diphenylethyl]iminopropanedinitrile 2-[2-(4-methoxyphenyl)sulfonylethyl]benzoic acid 3-[(7-chloro-1,8-naphthyridin-4-yl)oxy]benzamide;ethane 5-[(4R)-2-amino-1,4-dihydro-[1,3,5]triazino[1,2-a]benzimidazol-4-yl]-2,6-dichloropyridin-3-ol 3-azido-1-chloroisoquinoline (2R)-1-N,3-N-bis[2-(dimethylamino)ethyl]-4-phenylmethoxybutane-1,3-diamine 3-[4-(1,5-dihydroimidazo[1,2-b]pyrazole-7-carbonyl)piperazin-1-yl]-3-phenylpropanenitrile 2-amino-5,7-dimethyl-8,9-dihydropyrido[3,4-b]indole-3-carboxylic acid 2-hydroxy-5-[methylsulfonyl(octyl)amino]benzoic acid 3-[4,6-diamino-5-(7-cyanoimidazo[1,2-a]pyrimidine-2-carbonyl)pyridin-2-yl]benzenesulfonamide 2,4-diaminopyrimidine-5-carbonitrile;2-ethyl-N-[[3-(4-fluorophenyl)phenyl]methyl]-1H-benzimidazole-4-carboxamide 4-(5,6-dihydro-1H-pyrrolo[2,3-b]pyridin-2-yl)-1,3,7-trimethylpyrrolo[3,4-c]pyridazine (7-methyl-1,3-benzodioxol-5-yl)phosphane 5-(azidomethyl)-1,3-diethoxybenzene 2-(2-hydroxyethyl)-6,8-dimethoxy-3H-quinoline-4-thione 4-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylamino)piperidine-1-carboxylate 2-methyl-4-[2-(3,4,5-trifluorophenyl)ethynyl]benzoic acid 6-methyl-4,11,18-triazapentacyclo[8.7.0.02,8.03,8.012,16]heptadeca-1(10),2(8),3(8),6,9,11,13,15-octaene 3-[2-(3,4-dimethoxyphenyl)ethynyl]-1-hydroxy-N-methylpyrrolo[1,2-a]pyrazine-6-carboxamide [(3S)-1-methylpyrrolidin-3-yl]-[4-(6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-2-ylamino)phenyl]methanol 2-[5-tert-butyl-4-(methoxymethylamino)pyridin-3-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one (3R)-2-hydroxy-4,6-dimethyl-7-(naphthalen-1-ylmethoxy)-3H-benzo[g]chromen-1-ium 5-[5-azidooxy-1,3-diethyl-2,6-dimethyl-4-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine 3-[2,4-dihydroxy-5-(3-methylbutanoylamino)phenyl]-5-(4-piperidin-1-ylsulfonylbenzoyl)-1H-indole-7-carboxamide (1R)-1-(2,4-difluorophenyl)-N,N,2-trimethylpropan-1-amine;hydrochloride N-ethenyl-2,5-bis[(2Z)-2-ethylidenebutoxy]aniline N-[6-cyano-2,5-di(piperidine-1-carbonyl)pyridin-3-yl]nitramide 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)quinoline 1-[(3R)-3-azidopiperidin-1-yl]-2-methoxyisoquinolin-2-ium [(1-benzylpyrazol-4-yl)amino]-phenylmethanol N-ethyl-4-(methylamino)-6,7-dihydronaphthalene-1-sulfinamide 3-[3-(2-azidoethynyl)-5-chlorophenyl]-4,5-dihydro-1H-pyridazin-6-one 4-(3-aminopiperidin-1-yl)-5-propan-2-yl-N-pyridin-2-ylpyrimidine-2-carboxamide 4-(benzylsulfinylamino)benzoic acid N-[3-[[2-(3,5-dimethylanilino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]phenyl]-2-(trifluoromethoxy)benzamide 4-chloro-1,5-dimethyl-N-(oxolan-2-ylmethoxy)pyrazole-3-carboxamide 3-methyl-4-(1,2,6-trifluoronaphthalen-2-yl)benzamide 5-chloro-2,3-difluoroaniline;N-methylformamide;1-[4-(6-oxooxepan-2-yl)phenyl]ethanone N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[2,6-di(propan-2-yl)benzoyl]benzohydrazide ethene;(4S)-2,3,5-trimethylhexanal;(4-pentoxyphenyl)methanimine 2-benzyl-4,6-dichloroquinoline;methoxyethane 6-(furan-2-yl)-8-[1-methoxy-4,5-bis(phenylmethoxy)pyridin-1-ium-2-yl]-7H-purine 5-amino-4-[7-(2,3-dimethylmorpholine-4-carbonyl)furo[3,2-b]pyridin-2-yl]-2-fluorobenzoate N-(2,3-dihydroxypropyl)-1H-indole-4-carboxamide (2S)-2,5-diamino-N-[3-(4-methoxyphenyl)propanoyl]pentanamide;hydrochloride N-[5-cyclopropyl-1-(4,6-dimethylpyridin-2-yl)pyrazol-3-yl]-4-methylbenzenesulfonamide N-(5-bromopyridin-2-yl)-4-nitro-N-(3-oxopropanoyl)benzamide N-[4,6-bis(3-cyanophenyl)pyrimidin-2-yl]-1H-indazole-3-carboxamide 3-azidooxy-6-[2,5-dimethyl-4-(trifluoromethyl)phenoxy]pyridazine 4-[(E)-2,3-dimethylbut-1-enyl]benzamide 2-[1,3-benzodioxol-5-yl(hydroxy)methylidene]butanedioate 2-[3-(methoxymethyl)-4-[(E,1S)-1-phenylethoxyiminomethyl]pyridin-2-yl]sulfanyl-6-oxo-1H-pyrimidine-5-carbonitrile 1-[4-(3,5-dichloroanilino)piperidin-1-yl]ethanone;formic acid 5-(3,4-dichlorophenyl)-N-[3-methyl-1-(2H-tetrazol-5-ylmethoxy)butan-2-yl]-1,3-thiazole-2-carboxamide 2-azidooxy-N-methyl-6-(trifluoromethyl)aniline (3S,4R)-1-[2-[(4-fluorophenoxy)methyl]phenyl]sulfonyl-4-hydroxy-4-propylpiperidine-3-carboxylic acid (1R)-2,3-bis(4-bromophenyl)cyclopropane-1,1-dicarbonitrile 4-[6-methoxy-5-[[2-methyl-3,5-di(propan-2-yl)pyrazole-3-carbonyl]amino]pyridazin-3-yl]piperazine-1-carboxylic acid 2-[4-bromobutan-2-yl(nonanoyl)amino]benzoic acid 4-(3,5-dibromoanilino)-N'-hydroxypyridine-2-carboximidamide N-[3,5-difluoro-4-(7H-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3,4-bis(ethenyl)benzenesulfonamide 6-[5-(3,5-difluorophenyl)pyrazolidine-3-carbonyl]-2-hydroxy-4-methoxy-3H-isoindol-1-one 4-chloro-N'-hydroxy-3-[(5-methyltetrazol-2-yl)methyl]benzenecarboximidamide 2-[3-(4-fluorophenyl)phenyl]acetaldehyde 4-[5-(2-methylpyrazol-3-yl)pentoxy]benzaldehyde 3-(2,4-dichlorophenyl)-N'-hydroxypyrazine-2-carboximidamide 1-cyclopropyl-3-[4-(2,6-dimethoxyphenyl)-5-(6-methoxypyridin-2-yl)-1,2,4-triazol-3-yl]pyrrolidine-3-carboxamide 4-[(3R)-3-azidopyrrolidine-1-carbonyl]-N,N-dibenzylbenzenesulfonamide 2-[4-(5,7-dimethylquinolin-8-yl)sulfanylpiperazin-1-yl]ethanol 1-[4-(hydroxyamino)naphthalen-1-yl]pyrrole-2,5-dione 4-[2-(4-ethylpiperazin-1-yl)-4,5-dimethoxyphenyl]-N,3-dimethylaniline 2-[(1S)-5,7-difluoro-6-hydroxy-4-oxo-3H-inden-1-yl]-N-[[6-fluoro-2-methoxy-4-(triazol-1-yl)phenyl]methyl]acetamide 4-[2-[2,6-dichloro-5-(2-fluoro-3-methylphenyl)pyridin-3-yl]ethynyl]benzaldehyde 2-[3-(N-cyclohexylcarbamimidoyl)indol-1-yl]acetic acid [2-methylsulfanyl-4-[(3R)-oxolan-3-yl]oxyphenyl]methylcarbamic acid 1-[2,6-di(propan-2-yl)phenyl]-2H-pyridine 2-methyl-N-[3-[(5R,7S)-9-oxo-6,10-diazatricyclo[9.4.0.02,7]pentadeca-1(15),11,13-trien-8-yl]phenyl]pyridine-4-carboxamide 2-[3,5-bis(3-methylphenoxy)phenyl]acetaldehyde 1-[(5-bromopyridin-2-yl)carbamoyl]pyrrolidine-3,4-dicarboxylic acid 2-(4-cyano-3-fluorophenyl)-5,6-diethyl-N-methylbenzamide;ethane 4-chloro-N-(1H-indol-2-yl)benzenesulfonamide 1-amino-3-methoxy-4,4-dimethyl-2H-pyrimido[5,4-c]quinoline-8-carbonitrile;N',N'-di(propan-2-yl)ethane-1,2-diamine (1S,2R)-2-[4-(1H-indol-3-ylmethylideneamino)phenyl]cyclohexan-1-amine N-[3-methylsulfanyl-4-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydroquinazoline-2-carboxamide (2E)-2-[(4-oxo-3H-quinazolin-6-yl)methylidene]thieno[2,3-b]pyrrole-5-carboxylic acid N-[2-(4-acetylpiperazin-1-yl)ethyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide N-[1-(diethylamino)propan-2-yl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 2-(4-ethoxyphenyl)sulfanyl-7H-purine 3-[1,4-bis(pyridin-2-ylmethoxy)naphthalen-2-yl]-3H-thiophene-2-thione 2-[(1Z)-buta-1,3-dienyl]-N-methyl-4-(1H-pyrazol-4-yl)-6-[4-(trifluoromethyl)phenyl]pyridine-3-carboxamide 2-(1H-pyrrol-2-yl)-4-[4-(trifluoromethoxy)phenyl]-1,3-oxazole 2-(6,7-dimethoxy-3-oxo-1H-isoindol-2-yl)acetamide 1-chloro-2-(3,5-dimethoxyphenyl)-4-ethenylbenzene 1-(2,3,4,5,6,7,8-heptafluoronaphthalen-1-yl)heptan-1-ol 5-chloro-N-[2,2-dimethyl-6-(1,3-thiazol-4-yl)-3H-1-benzofuran-5-yl]-2-fluorobenzenesulfinamide (2S,4R)-N'-[2,6-dichloro-4-(trifluoromethyl)phenyl]-2-(2,2,2-trifluoroethoxymethyl)piperidine-1-carboximidamide 2-[(4R)-3-(cyclopropylmethoxy)piperidin-4-yl]oxybenzoic acid N-[5,8-bis(methylsulfanyl)-6H-phenanthridin-3-yl]cyclopropanecarboxamide 1,5-dibromo-2-ethyl-3-fluorobenzene 4-[(3S)-1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one 1-[[4-amino-5-(2-methylpropanimidoyl)pyrimidin-2-yl]-methylamino]butan-2-one 2-bromo-3,4-dihydroacridine [3,3-bis(2H-pyran-4-yl)cyclobutylidene]methanol N-[(3R)-3-[2,4-dimethoxy-5-[3-oxo-3-[2-[2-(propylamino)ethyl]imidazol-1-yl]propyl]phenoxy]butanoyl]acetamide N-[3-chloro-1-(2,4-dimethylphenyl)-7-fluoro-5,6-dihydroxyisoquinolin-8-yl]cyclopropanecarboxamide;ethane N-(3-chloropropyl)-7-nitroquinazolin-4-amine N-[(1R)-5,7-difluoro-3,4-dihydro-2H-chromen-3-yl]-2-methoxyiminoacetamide 4-(2,5-dichlorophenyl)-3-methylbutanamide 1-azido-3,4-diethylbenzene (7S)-7-[2,5-dimethoxy-4-(methylamino)phenyl]-3-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-one 6-(2,3-dihydrothiophen-4-yl)-1-methylbenzimidazole;ethane 4-(2,5-difluorophenyl)-3-[2-[(4-ethoxycarbonylpiperidine-1-carbonyl)amino]imidazo[1,2-a]pyridin-6-yl]sulfonylpiperazine-1-carboxylic acid 1-[3,4-dihydroxy-5-(2H-tetrazol-5-yl)phenyl]hexa-3,5-diene-1,3-disulfonic acid 4-[[3-methoxy-5-(trifluoromethyl)pyridin-2-yl]amino]piperidine-1,4-dicarboxylic acid [4-(5,6-difluorobenzimidazol-1-yl)-2H-pyridin-1-yl]-(3,4-dimethoxyphenyl)methanone [3-(dimethylamino)phenyl]-[8-[2-(dipropylamino)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-2-yl]methanone 4-[(3E,5Z)-octa-1,3,5,7-tetraen-4-yl]oxyaniline 2-[6-(cyclohexen-1-yl)benzimidazol-1-yl]acetic acid 2-(9H-fluoren-1-yl)-4,5-dimethoxypyran (E)-2-[5-[(2,5-dimethylphenyl)sulfanylamino]pyridine-3-carbonyl]-4-methoxypent-1-en-3-one (2Z)-N-[5-(3,5-dimethylpiperidine-1-carbonyl)pyridin-2-yl]-4-methoxy-6-(trifluoromethoxy)hexa-2,4-dienamide 1-ethyl-4-[3-[(3S)-1-(3-propan-2-yloxybenzoyl)pyrrolidin-3-yl]-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl]pyridin-2-one 2-[3,5-bis(trifluoromethyl)phenyl]ethynamine 2-chloro-N-[4-chloro-3-(trifluoromethyl)phenyl]acetamide 5-(azetidine-1-carbonyl)-2,4-difluorobenzoic acid 1-[7-azido-6,8-dichloro-2-(trifluoromethyl)quinoline-3-carbonyl]azetidine-3-carboxylic acid 4-[3-chloro-6-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-8-yl]aniline 3,3-difluorohexanal;ethane;1'-[2-methyl-4-(trifluoromethoxy)benzoyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 2-(2,6-difluoro-4-propylphenyl)-7-[2-(4-ethoxy-2,3-difluorophenyl)ethynyl]-9,10-dihydrophenanthrene 1-(2,4-dichlorophenyl)-3-(4-methylpiperazin-1-yl)propan-1-one (Z)-2,3-diamino-4-[5-chloro-6-(methoxymethyl)pyridin-3-yl]but-2-enenitrile 2-bromo-4,5-ditert-butyl-1H-imidazole [(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-[5-[6-(2-methylanilino)pyridazin-3-yl]thiophen-2-yl]azanium 4-methyl-1H-pyrimido[5,4-d]pyrimidine-2,7-dione 3-[2-(azidomethyl)phenyl]pyrrolidine 5-azido-N,4-diphenyl-1H-pyrazole-3-carboxamide 1-(5-nitro-2H-pyrimidin-1-yl)-4-propan-2-ylpiperidine 2-(3,5-difluorophenyl)-2H-1,5-naphthyridine 5-[4-(2,5-difluorophenyl)piperazine-1-carbonyl]-1H-pyridin-2-one;ethane 2-(4-azidophenyl)-N,N-dimethylaniline N'-[1-(benzenesulfonyl)cyclopropyl]benzohydrazide 2-chloro-N-[1-[4,4-difluoro-3-(4H-pyrazin-5-ylmethyl)cyclohexanecarbonyl]piperidin-4-yl]-N-propan-2-ylbenzamide N-(1,2-diaminoethylidene)formamide;4-(3-hydroxypropylamino)-7-phenylmethoxyquinoline-6-carboxamide 5-[(Z)-(4,5-dichloropyrrolo[2,3-b]pyridin-3-ylidene)methyl]-2-[(4-hydroxypiperidin-1-yl)methyl]-1H-imidazole-4-carbonitrile N-benzyl-5,8-diethoxy-2,3-dihydro-1H-4,1,4,5-benzothiadiazol-7-imine 5-[1,3-dihydroxy-4-(4-methylsulfonylphenyl)butan-2-yl]oxycarbonyl-1,4-thiazepane-4-carboxylic acid 1-methyl-N',3-diphenyl-4H-pyridine-3-carboximidamide (2-ethylpyrazol-3-yl)-[(4S,5R)-1-methyl-4,5-diphenylimidazolidin-2-ylidene]azanium 3-[(4-ethoxy-2,4-dioxobutyl)-methylsulfonylamino]benzoic acid 3-[2-(2,4-dichlorophenyl)ethylamino]-N-oxopropanamide;5-methylcyclohepta-1,4,6-triene 2-(1,3-dihydroindol-2-ylidene)-5H-[1,3]dithiolo[4,5-b]pyrazine 2-(4-azido-3-tert-butylphenyl)-1,1,1,3,3,3-hexafluoropropan-2-ol 3-[(2S)-2-[[(2R,3R)-4-acetamido-3-hydroxy-1-phenylbutan-2-yl]amino]propyl]benzoic acid 4-[4-(2,3-difluorophenyl)phenyl]butanal 2-[2-chloro-4-(trifluoromethyl)phenoxy]-N-(5,6-dihydroisoquinolin-3-yl)acetamide N-[(4-bromophenyl)methyl]-5,6-dihydro-1H-triazolo[4,5-d]pyrimidin-7-imine 4-[(8-bromoquinoxalin-5-yl)-hexadecanoylamino]-2-hydroxybenzoic acid 1-(2,6-dichlorophenyl)-7H-cyclohepta[c]pyridine N-ethyl-4,5-difluoro-2-[(4R)-4-propan-2-yloxolan-3-yl]oxyaniline (3R)-1-[6-[(2Z,4E,7E)-8-aminoocta-2,4,7-trienyl]pyridin-2-yl]piperidine-3-carboxamide N-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-2-(1H-indol-3-yl)quinazolin-4-amine (4E)-2,3-bis[(Z)-1H-indol-3-ylmethylideneamino]-5-nitroiminocyclopent-2-en-1-one 2-[3-(4-cyanophenyl)propyl]isoindole-1,3-dione 3-(3,5-dibromo-4-phenylmethoxyphenyl)-2,2-dichlorocyclopropane-1,1-dicarbonitrile 2-chloro-6-(cyclobutylmethoxy)-4,8-dimethylpyrimido[5,4-d]pyrimidine;ethane (2R)-3-benzylsulfanyl-4-[(4-propan-2-ylphenyl)methylamino]butanenitrile 4-tert-butyl-2-(1,6-dimethoxycyclohexa-2,4-dien-1-yl)-3-hydroxybenzoic acid N-(2,3,4,5,6,7-hexahydroazepin-1-yl)-2-propan-2-ylbenzamide 4-fluoro-2-[3-(1H-imidazol-5-yl)-1,2,4-oxadiazol-5-yl]phenol 2-(3,4-dimethylphenoxy)-N-[3-(1H-imidazol-5-yl)phenyl]propanamide;hydrochloride 5-[5-(cyclopropylmethoxy)pyrazin-2-yl]-6-methylpyrimidine-2,4-diamine 6-(3,4-difluorophenyl)-N-ethyl-5-hydroxy-2-oxopiperidine-4-carboxamide 3-methyl-1-[2-methylidene-5-(1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]azepan-2-one 2-(6-chlorospiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carbonyl)furan-3-carboxylic acid (3R)-N'-hydroxy-2,2-dimethyl-4-[(2R,3S)-1-(3-phenylpropanoyl)-2-phenylpyrrolidine-3-carbonyl]octanediamide [1-ethylsulfanyl-5-(2-methoxypyridin-3-yl)sulfonylpenta-1,4-dienyl]carbamic acid 2-[5-chloro-3-(4,5-dihydro-1H-imidazol-2-yl)-2,6-dimethoxyphenyl]propanoic acid N-[2-[(4-cyanophenyl)sulfonylamino]ethyl]-5-(dimethoxyphosphorylmethyl)furan-3-carboxamide 2-[5,10-diphenyl-3,6-bis(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenanthro[9,10-d]imidazol-2-yl]-1H-quinolin-4-one 2-bromo-N-(1,3-thiazol-5-yl)-N-(4-sulfamoylphenyl)benzamide N-(2,3,4a,5-tetrahydro-1H-chromeno[4,3-c]pyrazol-7a-ylmethyl)-2-methoxybutanamide;hydrochloride 1-[2,3-bis(hydroxymethyl)phenyl]-N,N-diethylpropan-2-amine;chloromethane 2-[4-[1-(6-bromopyridin-3-yl)sulfonylpiperidine-4-carbonyl]piperazin-1-yl]ethanol 2-azidooxy-3-chloro-6,7-dimethylnaphthalene 1-azido-2,3,4-trimethoxy-9H-fluorene (2S)-1-methyl-N-[2-(7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl)ethyl]pyrrolidine-2-carboxamide 2,5-bis(1H-indol-4-yl)thiophene-3,4-dicarbonitrile 3-(4-benzylpiperazin-1-yl)-N'-[(2,6-difluorophenyl)methoxy]-2-[(2-ethylbutanoylamino)methyl]benzohydrazide 6-methoxy-2-(4-methylphenyl)imidazo[1,2-b]pyridazine 2-[2-(4-fluorophenyl)ethynyl]-5-methoxyaniline 2-[5-[4-(1H-benzimidazol-2-yl)phenyl]pent-4-ynoxymethyl]benzoic acid 2-[4,7-dimethyl-1-(2-phenylethyl)-6H-2,1-benzoxaborinin-3-yl]ethanol 5-chloro-2,3-dimethylbenzaldehyde;ethane 2-bromo-5,7-difluoroquinoline (2Z)-3-benzoyl-4,7-dihydroxyiminonaphthalene-1,6-disulfonic acid N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(6-methylpyridin-3-yl)benzimidazole-5-carboxamide (2R)-4,5-bis[(4-chlorophenyl)sulfanyl]pentane-2,3-diol N-[3-(1,2-dihydrotriazol-5-yl)phenyl]-3-methoxybenzamide N-[2-fluoro-4-(2,3,5,6-tetramethylphenyl)phenyl]-1H-imidazo[4,5-b]pyridin-7-amine 7-hydroxy-3-methyl-4,8-dioxospiro[2H-indeno[1,2-c]pyrazole-6,1'-cyclohexane]-5-carboxylic acid 6-(6,7-dihydro-4H-pyrano[2,3-c]pyrazol-2-yl)-5,8-difluoro-4-oxochromene-2-carboxylic acid [3-[(4R)-2,5-dioxoimidazolidin-4-yl]phenyl]urea 1-(5-ethylfuran-2-yl)sulfonyl-3-[4-methyl-6-oxo-2-propan-2-ylsulfanyl-1-[2-[2,3,5,6-tetrafluoro-4-(methanesulfonamido)phenyl]ethyl]pyrimidin-5-ylidene]urea 2-(cyclohexen-1-yloxymethyl)-4,5-dihydro-1H-indole 4-[(2,5-dimethoxyphenyl)sulfonylamino]-N-pyridin-3-ylbutanamide 2-[2,6-bis(methylamino)-4-(methylideneamino)phenoxy]acetic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-pyridin-4-ylpiperidine-1-carboxamide 3-[2-ethoxy-5-(methylamino)phenyl]oxirane-2,2-dicarbonitrile 2-[4-(benzylamino)phenyl]-1H-indole-7-carbonitrile 4-chloro-3-[(4-iodophenyl)methyl]-N,2-dimethylbutanamide N-[2,4,6-trichloro-3-(5-hydroxy-6-oxo-1H-pyrimidin-4-yl)phenyl]acetamide (3S,4R)-1-(7H-purin-6-yl)pyrrolidine-3,4-diol 2-(4-azidocyclohexyl)sulfanylethenylbenzene 3-(azidomethyl)-4-[2,6-dichloro-4-(trifluoromethoxy)phenoxy]-1H-pyrrole N-[3-[(7S,8aS)-2-[(4-fluorophenyl)methyl]-1,3,6,7,8,8a-hexahydropyrrolo[1,2-a]pyrazine-7-carbonyl]cyclobutyl]acetamide 4-[(2S)-3-(diethylaminomethyl)-2-(1,3-thiazol-2-yl)cyclopropanecarbonyl]-2-fluorobenzoic acid (2R)-4-hydroxy-N-[1,3]oxazolo[5,4-b]pyridine-2-carboxamide 3-amino-6-(2,4-dichlorophenyl)sulfanyl-9H-pyrido[3,4-b]indole-1-carboxylic acid 3-[3-[1-(2,4-dichlorobenzoyl)piperidin-4-yl]propoxymethyl]-6,7-dihydro-5H-cyclopenta[b]pyridine-2-carboxamide 2-(3,5-dimethoxy-4-phenylmethoxyphenyl)acetaldehyde;2-hydroxyethanol N-(1-methylpyrazol-4-yl)-2-[(4R)-3-oxo-1,2-oxazolidin-4-yl]-1,3-thiazole-5-carboxamide 4-(2,3-dimethylphenoxy)pentanoate (4-azidocyclohexyl)methoxymethylbenzene 1-(4-methylphenyl)sulfanylindole-3-carboxylic acid 3-[N-ethylsulfonyl-4-[(2-phenylpyrazol-3-yl)sulfamoyl]anilino]propanoic acid 3-bromo-5-methyl-2,4,6-tripropoxybenzaldehyde 3-azido-6,7-dimethoxy-2H-isoquinolin-1-one 7-[(2,6-dimethoxyphenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 2-[N-hexyl-4-(pyrimidin-2-ylamino)anilino]octanoic acid 3,7-diiodo-4-methyl-1H-quinolin-2-one ethane;1-[(3E)-hepta-1,3-dien-4-yl]-2-methoxynaphthalene 5-methyl-3-phenyl-2H-1,4-benzothiazepine;N'-[(E)-3-oxoprop-1-enyl]ethanimidamide 5-chloro-4-(trifluoromethyl)pyridine-3,8-diamine 2-[4-(N'-hydroxycarbamimidoyl)phenyl]-5-oxopyrrolidine-3-carboxylic acid ethane;3-fluoro-4-methoxy-N,5-dimethylbenzamide 4-[4-(2-cyanopropan-2-yl)pyridin-2-yl]-N,N-dimethylbenzamide;2,2,2-trifluoroacetic acid 3-[4-(5,6,7,8-tetrahydroquinazolin-4-yl)piperazin-1-yl]pyrazine-2-carbonitrile N'-[(2-hydroxyphenyl)methylideneamino]-N,N,3-trimethylbutanediamide 2-[(3,4-dimethylphenyl)sulfonylamino]-5-thiophen-2-ylbenzoic acid;2,2,2-trifluoroacetic acid 4-(4-chlorophenyl)-3,3a,4,5-tetrahydrobenzo[g]indazole 4-benzyl-5-propan-2-ylthiophene-3-carboxylic acid 3-[[5-bromo-4-(2,6-difluoroanilino)pyrimidin-2-yl]amino]propanamide 5-[3-(2,6-dichlorophenyl)-4-fluoropyrazolo[1,5-a]pyridin-7-yl]-N,4-dimethylpyridin-2-amine 3-[1,5-dimethyl-6-(propan-2-ylideneamino)cyclohexa-2,4-dien-1-yl]benzonitrile 5-[4-[(3R)-3-aminopyrrolidine-1-carbonyl]phenyl]sulfonyl-N-[4-chloro-2,6-dimethyl-4-(methylcarbamoyl)cyclohexa-1,5-dien-1-yl]-1H-pyrrole-3-carboxamide 1-[(E)-2-chlorobut-2-enyl]-2,4-difluorobenzene 1-butyl-2-methoxy-4-methylbenzene;5-[[(E,3Z)-3-ethylidenehept-4-enoyl]amino]-N,2-dimethylfuran-3-carboxamide 1-[5-chloro-6-(4,4-difluoropiperidin-1-yl)pyridine-3-carbonyl]azetidine-2-carboxamide 5-cyclopropyl-3-methoxy-2-[[4-(5-morpholin-4-ylquinoxalin-6-yl)phenyl]carbamoylamino]benzamide 5-(cyclopropylmethoxy)-2-fluoro-N-[6-[(3R,4S)-4-methylpiperidin-3-yl]pyridin-3-yl]benzamide N-butyl-2,3,5-triphenylaniline 2-(3,4,5-trimethoxyphenyl)propanamide 5-[1,2-diamino-3-(pyridine-4-carbonyl)propyl]pyrazine-2-carboxylic acid 2-methoxy-3,3-bis(4-methylphenyl)propanoic acid 2-[4-hydroxybutyl(phenacyl)amino]benzenesulfonic acid 1-(6,7-dimethylquinazolin-4-yl)-2H-pyridine-4-carboxylic acid (3R,4S)-3-[(2-cyclopentyloxyacetyl)amino]-N-[3-fluoro-5-methyl-1-(4-methylpiperidin-4-yl)pyrazol-4-yl]-4-propan-2-ylpyrrolidine-1-carboxamide 4-[8-[amino(2,3-dihydro-1H-inden-5-ylmethoxy)phosphoryl]oxy-5,6-dihydronaphthalen-2-yl]pyridine-2-carbonitrile 1-[2,5-dimethyl-4-(3-phenylpropyl)phenyl]ethanone N-[(E)-1-cyano-3,3-dimethylbutan-2-ylidene]-4-nitrobenzenesulfonamide N-[1-(4-chlorophenyl)ethenyl]-2-[3,5-dimethyl-4-(morpholine-4-carbonyl)pyrazol-1-yl]-3-(methylideneamino)propanamide;fluoromethane 6-(4-fluorophenyl)-3-[2-(1H-imidazol-5-ylmethoxy)ethyl]-8a-hydroxy-7,8,9,10-tetrahydrobenzo[f]chromen-1-one 2-[3,4-bis(methoxycarbonyl)anilino]propanoic acid 2-[1-(4-chlorophenyl)-2,6-dimethylpyrrolo[3,2-c]pyridin-5-yl]cyclobutan-1-amine (2-chloro-1,3,4-thiadiazol-5-yl)-(6-pyridin-2-yl-8-azabicyclo[3.2.0]heptan-8-yl)methanone [(2S)-2-amino-1,4-diphenylbutan-2-yl]carbamic acid (2R)-2-[3,5-dichloro-4-(1H-indol-3-ylmethoxy)phenyl]-2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-N-(4-fluorocyclohexa-2,4-dien-1-yl)acetamide 2-[4-(4,5-dimethylpyrimidin-2-yl)piperazin-1-yl]quinoline;formic acid [1-hydroxy-3-(4-methoxyphenyl)propan-2-yl]carbamic acid [3-amino-1-[6-methoxy-5,7-di(piperidin-4-yl)quinolin-4-yl]but-2-enylidene]azanide N-(4-bromophenyl)-N-(2,3-dihydroxypropyl)ethenesulfonamide N-(4,6-dimethoxypyrimidin-2-yl)-4-[5-iodo-3-methoxy-2-propanoyloxy-6-(trifluoromethyl)phenyl]-1H-imidazole-5-carboxamide N-[(3Z)-6-(4-cyclopropyloxypyridin-2-yl)-5,5-dimethylhepta-1,3,6-trien-2-yl]-3-(fluoromethyl)aniline 7-(1H-imidazol-5-yl)-4-(methoxymethoxy)chromen-2-one (2E)-3-[1,3-benzodioxol-5-ylmethoxy(hydroxy)phosphoryl]-N-ethyl-2-[(4-ethynylphenyl)hydrazinylidene]-3-oxopropanamide 3-azido-1,2-dimethylindole 2-amino-4,4-dimethoxy-6-[3-(trifluoromethyl)phenyl]-3-azabicyclo[3.1.0]hex-2-ene-1,5-dicarbonitrile 2-[[2,4-bis(trifluoromethyl)phenyl]methoxycarbonylamino]hexanoic acid 3-[4-[1,6,7,8-tetrahydropyrido[2,3-b]azepin-5-yl-(oxan-4-ylamino)phosphanylidene]phenyl]propanenitrile N-[3-hydroxy-4-(2H-pyridin-1-yl)phenyl]pyridine-4-carboxamide N-(2,3-dihydro-1H-inden-4-yl)-5-(6-fluoro-4-methoxypyridin-2-yl)-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-amine;ethane 1-(1,3-benzodioxol-5-yl)-2,3-dihydroindole 5-(1,3-benzodioxol-4-yl)pentane-2,5-dione (E)-N'-[3,5-bis(trifluoromethyl)phenyl]-2-(3-butylimidazol-4-yl)ethenol 5-(3,5-dimethyl-1,2-oxazol-4-yl)-N'-hydroxypyridine-2-carboximidamide 2-azidooxy-1-ethyl-3,4-diphenylbenzene 2-[[1,5-dimethyl-3-(trifluoromethyl)pyrazole-4-carbonyl]amino]-2-phenylpropanamide N-cyclohexyl-4-[4-(3-methoxyphenyl)piperazine-1-carbonyl]benzamide N-(4-azidooxypyridin-2-yl)-N',N'-dimethylethane-1,2-diamine 2-cyclopropyl-6-[[3-[(3,5-dichlorophenyl)methoxy]phenyl]methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-[3-fluoro-5-(2-pyrrolidin-1-ylethoxy)phenyl]-6,7-dihydroisoquinoline-8-carboxamide 3-[2,4,5-trichloro-6-(2,3-dimethylphenoxy)phenoxy]propan-1-ol N-[3-cyano-6-(2,5-dimethoxyphenyl)pyrido[3,4-b]pyrazin-8-yl]acetamide N-[(1R)-1-cyano-2,3-dihydro-1H-inden-4-yl]-2-ethynyl-5-methoxybenzamide 5-[(3R)-1-cyclobutylpiperidin-3-yl]oxy-7,8-dihydropyrido[4,3-d]pyrimidine;dihydrochloride 7-bromo-1-methyl-3,5-bis[4-(trifluoromethoxy)phenyl]pyrazolo[3,4-c]pyridine 4-[(2R,4R)-5-hydroxy-4-methyloxolan-2-yl]-1H-pyridin-2-one;propane (2-hydroxyphenyl)methanesulfonate (3-methylphenyl)-[(2S,4R)-2-methyl-4-[4-(1-propan-2-ylpyrazole-3-carbonyl)piperazin-1-yl]pyrrolidin-1-yl]methanone (7R)-5,9-dimethyl-2-[[1-[[6-(trifluoromethyl)pyridin-3-yl]methyl]pyrazol-4-yl]methylamino]-7H-pyrimido[4,5-b]azepine-8-carboxylic acid 2-[3-(4,5-dimethyl-1H-imidazol-2-yl)phenyl]propan-2-amine 7-azidooxyquinoline-2,3-dicarboxylic acid 7-[5-chloro-3-(2,6-dimethoxyphenyl)-1H-pyrazole-4-carbonyl]-1,4,8,10-tetrazacycloundecane-9-carboxylic acid 2-[5-(3,4-dimethoxyphenyl)thiophen-2-yl]pyridine 1-[[5-chloro-4-[1-(cyclopropylmethyl)-3,5-dimethylpyrazol-4-yl]pyrimidin-2-yl]amino]-7-(cyclohexylmethoxy)-N,N,4-trimethylphthalazine-6-carboxamide 2-(3,4-dimethoxyphenyl)cyclobutane-1-carboxylate 1-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]-6-fluoro-2H-quinoline 4-[1-[4-(dimethylamino)phenyl]pyrrol-3-yl]-N,5-dimethylcyclohexa-1,5-dien-1-amine 5-amino-2-(6,7-dimethoxyquinazolin-4-yl)oxyphenol 1,3-dibromo-2-(trichloromethoxy)benzene 3-[2,6-di(propan-2-yl)phenyl]iminopyrrolidine-1-carboxylic acid N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]ethanesulfonamide 5-azidonaphthalene-2,3-dithiol N-(2,4-difluorophenyl)-2-oxopentanamide N-[2,4-difluoro-3-[5-(1H-pyrrolo[2,3-b]pyridin-4-yl)-2H-pyrazolo[3,4-b]pyridine-3-carbonyl]phenyl]propane-1-sulfonamide (3S,4R)-2,2-dimethyl-4-[(1E)-1-(4-methylidene-2-oxo-1H-quinolin-7-yl)buta-1,3-dien-2-yl]-5-phenylpentanamide 2-(5-chloro-1H-indol-3-yl)-N-[2,6-di(propan-2-yl)phenyl]acetamide 2,4-dimethyl-5-phenylsulfanyl-1H-pyrimidin-6-one N'-[(Z)-N',N'-dimethylcarbamimidoyl]-4-[1-[3-(prop-2-enylamino)cyclobutyl]ethenyl]benzenecarboximidamide 2-methylsulfonylbenzenethiolate 4-[(3Z)-3,4-dihydroxyhexa-1,3,5-trien-2-yl]benzaldehyde 7-bromo-N-(4-chlorophenyl)-2-[5-chloro-3-methyl-6-(trifluoromethyl)pyridin-2-yl]oxy-1-cyclopropyl-9H-pyrido[3,4-b]indole-3-carboxamide 3-[3-(2,6-difluorophenyl)-1,2,4-oxadiazol-5-yl]hexanal N-[3-(6,7-dihydro-4H-pyrano[2,3-c]pyrazole-2-carbonyl)cyclopentyl]quinoline-5-carboxamide 2-[N-(2-hydroxyethyl)anilino]guanidine N-[1-[4-(difluoromethoxy)phenyl]ethyl]-2,6-dioxopiperidine-3-carboxamide 6-[4-(1H-indazol-5-yl)piperazine-1-carbonyl]pyridine-2-carbonitrile 4-bromobenzoate;nickel(2+) 2-(1H-imidazole-5-carbonyl)-3,4-dihydro-1H-isoquinoline-6-carboxylic acid 3-[[(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]benzoic acid 2-(4-aminopyridin-1-ium-3-yl)-5-tert-butylpyrazole-3-carboxylic acid (1R,2S)-1-[3-[3,5-bis[dideuterio-[(2-methylpropan-2-yl)oxycarbonylamino]methylideneamino]benzoyl]phenyl]-4-methyl-2-propan-2-ylcyclohexane-1-carboxylic acid 5-(3,5-difluoro-4-methoxyphenyl)imidazolidine-2,4-dione 4-(4,6-diiodocyclohexa-1,5-dien-1-yl)oxy-7-fluoro-2-methylquinazoline 3-[6-(1,2-dihydropyridin-5-yl)naphthalen-2-yl]phenol 2-(6,7,8,9-tetrahydro-5H-fluoren-3-yl)phenol 2-chloro-4-[2,5-dimethyl-3-(3-phenyl-1H-pyrazole-5-carbonyl)cyclohexa-1,5-dien-1-yl]benzonitrile 5-methyl-3-[5-[3-[(2S)-1,1,1-trifluoropropan-2-yl]oxyphenyl]pyridin-2-yl]-4H-1,2-oxazol-5-amine 2,4-diamino-6-[(2S)-4-azidobutan-2-yl]pyrimidine-5-carbonitrile 3-butyl-4-chloro-7H-purine-2,6-dione 1,3-bis[2,6-di(propan-2-yl)phenyl]-4,5-dihydroimidazol-1-ium;cyclopenta-2,4-dien-1-amine [3-cyclopropyl-1-(2,2-difluoroethyl)pyrazolo[4,3-c]pyridin-6-yl]azanium 4-[3-(2,5-dimethylimidazol-1-yl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine (2R,3S)-3-methyl-6-oxo-2-phenylheptanoic acid 6-(1,1-difluoroethyl)imidazo[2,1-b][1,3]thiazole ethane;1-[(3Z)-4-[2-methoxy-5-(trifluoromethyl)phenyl]hexa-1,3,5-trien-3-yl]-4-propan-2-ylpiperidine [(5Z)-3,7-dihydroxy-6-methoxycarbonyl-1,2,4,8,9-tetrahydrocycloocta[b]pyrrol-2-yl]boronic acid N-[(2R)-1-oxo-1-phenyl-3-[3-(trifluoromethyl)anilino]propan-2-yl]benzamide 3-amino-4-(methylamino)-5,6-dihydro-2H-benzo[f]quinazoline-1-thione 1-azido-4,5-dimethoxyindole 6-[(2,3-difluorophenoxy)methyl]-5H-pyrrolo[2,3-d]pyrimidine 6-[(2-phenyloxan-4-yl)methylamino]pyridazine-3-carbonitrile 1-[2,5-bis(trifluoromethyl)phenyl]sulfonylpyrrolidine N-[1-(3,5-difluorophenyl)-2-hydroxyethyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-6-carboxamide 3-(2,4-dichlorophenyl)-6-(3,5-difluorophenoxy)-1H-pyrazolo[4,3-c]pyridine 5-(1,3-benzothiazol-2-yl)-6-bromo-N-methylpyridin-2-amine 3-[(1R,2S)-4,6-difluoro-1-hydroxy-3,4-dihydro-1H-naphthalen-2-yl]benzonitrile 1-benzylsulfanyl-3,4-dimethoxydithiolane 1-[(2S)-2-aminopropanoyl]-N-(4-cyanophenyl)piperidine-3-carboxamide 2-[4-[6-(2,3-difluorophenyl)pyridazin-3-yl]piperazin-1-yl]-N-methylethanamine 6-[3-(dimethylamino)propoxy]quinoline-2,4-diamine 4-azidooxy-2,7-diethylfuro[3,2-c]pyridine 4-[2-methylsulfonyl-6-(trifluoromethoxy)pyridin-3-yl]oxybenzenesulfonate 2-[(2Z)-4,5-dimethylhepta-2,6-dienyl]sulfanylnaphthalene 6-[(3-methylphenyl)methyl]-2-propan-2-yl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one 1-[3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl]cyclobutane-1-carbonitrile 2,4-dinitro-3-(trifluoromethyl)phenol 4-benzyl-2-(6-bromoimidazo[1,2-a]pyridin-3-yl)morpholine 3,7-dichloro-1-(4-fluorophenyl)sulfonylquinolin-2-one 2-[[6-(6,7-dihydronaphthalene-1-carbonyl)-5H-pyrrolo[3,4-b]pyridin-5-yl]oxy]acetaldehyde 2-[3-chloro-4-(5-methyl-1H-pyrazol-4-yl)phenyl]-6-[(E)-methoxyiminomethyl]-7-propan-2-yl-4,5-dihydrothiepine-3-carboxylic acid N-[(Z)-1H-indol-3-ylmethylideneamino]-2-nitrobenzamide 5-[3-chloro-4-(trifluoromethyl)phenyl]imidazolidine-2,4-dione (2S,5R)-2-methyl-4-[3-methyl-6-[1-methyl-5-[(5-propan-2-ylpyridazin-3-yl)amino]triazol-4-yl]imidazo[1,2-a]pyridine-8-carbonyl]morpholin-3-one N-[2-(3-methoxyphenyl)ethyl]-4,5-dihydropyrene-1-carboxamide 2-chloro-5-N-(1,3,4-oxadiazol-2-ylmethyl)pyridine-3,5-dicarboxamide 4-(3,6-dimethylcarbazol-9-yl)-5-phenylpyridine-2-carbonitrile 1-(2,2-dichlorocyclopropyl)oxy-4-[3-(2,6-dichlorophenyl)pyrrol-1-yl]pyrazole 4-hydroxy-3,5-diphenyldiazenylthiophene-2-carboxylic acid 1-[(2S)-2-(5-azidooxyindol-1-yl)propanoyl]pyrrolidine-3-carbonitrile 2-[2,3-bis(trifluoromethyl)phenyl]-1-(4-chloro-3-hydroxy-5-propanoylphenoxy)propane-1,2,3-trione 2-[7-(4,6-diphenyl-1,3,5-triazin-2-yl)naphthalen-2-yl]-2-methoxypropanoic acid N-[(1S,2R)-3-amino-2-hydroxypropyl]benzamide 3-[(1,4-dichlorocyclohexa-2,4-dien-1-yl)methoxy]benzenethiol 4-azido-3,5-dimethyl-2H-quinoxaline 5-ethyl-N-[(Z)-1H-indol-3-ylmethylideneamino]-2-propan-2-yl-1,3-thiazole-4-carboxamide (5-methylpyridin-2-yl)-[4-(spiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,3'-azetidine]-1'-ylmethyl)piperidin-1-yl]methanone;2,2,2-trifluoroacetic acid 2-[(6S)-5,6-dihydrobenzo[b][1]benzoxepin-6-yl]acetic acid 2-amino-4-[(2,6-dimethylphenyl)methoxy]benzenecarboximidamide 7-(cyclohexylmethylamino)-3,4-dihydroisoquinoline-5-sulfinic acid 7-[2-(6-methylpyridin-3-yl)ethynyl]-1,4,5,6-tetrahydrotriazolo[4,5-c]pyridine;dihydrochloride 2-(2,4-dichlorophenyl)-3-[1-(3,5-difluorophenyl)cyclopropyl]-5-[methoxy(oxan-2-ylmethoxy)methyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one 5-[(2E,4Z)-3-chlorohepta-2,4,6-trien-2-yl]oxybenzo[b][1,4]benzoxathiine 2-(1,3-benzodioxol-5-yl)-N-[[4-(methoxymethyl)oxan-4-yl]methyl]cyclopropane-1-carboxamide 2-(N-(4-bromo-2,5-dimethylphenyl)-3-chloroanilino)acetonitrile [6-amino-1-[4-(2,5-difluorophenoxy)butyl]pyrazolo[3,4-d]pyrimidin-3-yl]methanol 1-[[3-fluoro-5-(trifluoromethyl)phenyl]sulfonylamino]-4-oxoazetidine-2-carboxylic acid [(1S)-1-azido-2,3-dihydro-1H-inden-4-yl]methanamine 6-[(4S)-4-benzyl-2-[1-(3,5-dimethoxyanilino)ethenyl]-3-oxo-1,4-oxazepan-7-yl]hexanamide 2-ethoxycarbonyl-6-phenylhexanoate N-(2,4-dimethylphenyl)-3-oxobutanamide 1-(2-methylpiperidin-4-yl)-N'-[4-[1-[(2R)-oxolan-2-yl]ethenylamino]phenyl]sulfonylpyrazolo[3,4-b]pyridine-5-carbohydrazide 4-(1,3-benzothiazol-2-yl)-5-imino-1-propan-2-yl-2H-pyrrol-3-ol 1-[3-(1,6-dihydropyrrolo[2,3-c]pyrazol-4-yl)phenyl]propan-2-amine 4-(2-azidoethyl)-3,5-dichlorophenol N-[(3,5-diethyl-1H-pyrazol-4-yl)methylideneamino]pyridazine-4-carboxamide 2-[4-(N,3-dimethylanilino)-7-(1-phenylbutoxy)quinolin-6-yl]acetonitrile [4-[2,5-bis(trifluoromethyl)phenyl]pyrazol-1-yl]methanamine 6-chloro-N-[1-(5-cyclopropylpyrimidin-2-yl)piperidin-4-ylidene]pyridine-3-carboxamide [7-(4,6-diphenyl-1,3,5-triazin-2-yl)-9H-xanthen-2-yl]boronic acid 4-methyl-3-[(E)-[2-(4-phenyl-1,3-thiazol-2-yl)phenyl]methylideneamino]oxybenzoic acid N-(2,3-dihydro-1H-inden-5-yl)-4-oxo-7-[[2,4,6-trimethoxy-4-(3-phenoxyprop-1-ynyl)cyclohexa-1,5-dien-1-yl]amino]-3H-pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide 7-cyclohexyl-5,6-dimethoxy-2H-chromene 1-[2-(dimethylamino)ethyl]indole-3,7-diol N-[1-(4-chlorophenyl)ethyl]-3,5-dimethyl-2H-pyrazolo[4,3-c]pyridine-7-carboxamide 3-(4-bromocyclohexyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine;2,2,2-trifluoroacetic acid 2-[3,5-dichloro-4-(1,1,2,2,2-pentafluoroethylsulfanyl)phenyl]-4-(hydroxymethyl)-5-methoxypyrazole-3-carboxylate 4-[2-(3,5-dimethylphenyl)ethynyl]benzonitrile N-azido-3,5-dibromobenzenesulfonamide 1-(benzenesulfonyl)pyrrolo[2,3-b]pyridin-6-ium 4-[3-hydroxy-6-(2-methyl-1H-imidazole-5-carbonyl)-1,5,7,8-tetrahydropyrazolo[4,3-g]quinolin-2-yl]benzonitrile [3-hydroxy-2,2-dimethyl-7-phenyl-6-(trifluoromethoxy)chromen-4-ylidene]oxidanium N-azido-2-[4-(3,4-dimethoxyphenyl)piperazin-1-yl]acetamide 2-[(1S)-1-azidoethyl]-6-fluorobenzonitrile N-(4,5-dimethylcyclohexa-1,3-dien-1-yl)-N'-[2-methoxy-4-(2-methylpiperidine-1-carbonyl)phenyl]methanimidamide 5-(cyclopropanecarbonyl)pyridine-2,3-dicarboxylic acid 2-(4,7-difluorobenzotriazol-2-yl)-5-(sulfanylmethoxy)phenol N-methyl-1-[2-(trifluoromethyl)phenyl]-5,6-dihydro-4H-cyclopenta[c]pyrazole-3-carboxamide [(3R,4S)-1-[2-(5,6-dimethylpyrazin-2-yl)ethyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methanol N-(2,4-dimethylpyridin-3-yl)sulfanylcyclobutanecarboxamide 5-(2,6-dimethylphenyl)imino-1-[3-nitro-4-[3-(trifluoromethoxy)phenoxy]phenyl]-4H-pyrazole-3-carboxamide 5-chloro-4,6-dinitrobenzene-1,2,3-triol N-(2,3-dihydro-1H-inden-5-yl)-3-fluoro-4-[2-hydroxyethyl-(4-methoxybutanoylamino)amino]benzamide;ethane N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-chloroacetamide N-[2,4-difluoro-3-(hydroxymethyl)phenyl]-7H-purin-6-amine (Z)-5-[3,4-bis(2,6-dimethylphenoxy)phenyl]sulfanyl-N-ethenyl-2-methoxy-1-N',3-N-dipropylpent-1-ene-1,3-diamine 2-[[6,7-difluoro-1-(2,3,4,5,6-pentafluorophenyl)sulfonyl-2H-indole-3-carbonyl]amino]acetic acid 2-(4-cyclobutylphenoxy)pyridine 6-chloro-3,4-dihydrodibenzofuran 4-[(E)-2-cyclohepta-1,3,5-trien-1-ylethenyl]-N-methylbenzamide;ethane 2-methyl-3-[2-(3,4,5-trifluorophenyl)imidazol-1-yl]propan-1-ol 2-[3,5-difluoro-4-[(2R)-6-methoxy-3-methyl-1,2-dihydroinden-2-yl]phenyl]-2-propyloxirane (4R)-7-[3-[2,6-dimethyl-4-[3-methyl-1-(oxan-2-yloxy)butyl]phenyl]azetidine-1-carbonyl]-4-hydroxy-4-methyl-N'-[[4-(trifluoromethyl)phenyl]methyl]heptanehydrazide 4-tert-butyl-N-[5-methoxy-2,6-dimethyl-3-[(Z)-pent-2-en-2-yl]cyclohexa-1,3-dien-1-yl]benzamide 1-[(1S)-1-hydroxybutyl]-3,6-dihydropyrrolo[2,3-c]carbazole (2R)-N-cyclopropyl-3,4-dioxo-2-[[4-(3-phenyl-1,2-oxazol-5-yl)benzoyl]amino]butanamide 3-[4,5-dimethoxy-2-(1-methylpyrrol-2-yl)phenyl]-N-formylpropanamide N-[2-amino-6-[1,5-bis(prop-2-enyl)pyrazole-3-carbonyl]phenyl]propanamide 1-[(3R)-2,6-dioxopiperidin-3-yl]-7-(4-ethenylphenoxy)heptan-3-one;5,7,7-trimethyl-1H-cyclohepta[b]pyrrol-6-one 3-[3-[4-(5,6-dimethylpyridin-2-yl)phenyl]cyclobuta-1,3-dien-1-yl]-9H-pyrido[2,3-b]indole 5-(5,8-dimethylquinoline-7-carbonyl)oxy-1,3,4-oxadiazol-2-olate 5-chloro-N-(3-chloro-2,6-difluorophenyl)-1H-indole-2-carboxamide 6-(2,3-dihydro-1H-inden-5-yl)-4-oxohexanoic acid 4-chloro-N-methyl-2,3-dihydro-1H-indene-5-sulfonamide (2S)-1-[2-[4-(diethoxyphosphorylmethylamino)piperidin-1-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethanone;2,2,2-trifluoroacetic acid 4-[6-(5,5-dimethylhexyl)pyrimidin-4-yl]-2-fluorobenzonitrile 3-[1-[5-[(2R)-2,6-diaminohexanoyl]pyridin-2-yl]triazol-4-yl]cyclobutane-1-carbonitrile;hydrochloride 1-[5,7-bis(trifluoromethyl)-3H-azepin-2-yl]-N-butyl-6-chlorobenzimidazole-2-carboxamide 1-(oxolan-2-yl)-4H-benzo[h]quinoxaline 2-(N-(4,5-dimethylpyrimidin-2-yl)-2-hydroxyanilino)decanoic acid 5-[4-(2,6-difluorophenyl)piperazine-1-carbonyl]pyridine-3-carboxylic acid;2,2,2-trifluoroacetic acid (5R)-5-[(1R,2S)-2-hydroxy-3-oxocyclohexyl]oxy-5,6-dihydroimidazo[2,1-b][1,3]thiazole-7-carboxylic acid 5-hydroxy-6-[3-(2-pyrrolidin-1-ylethoxy)phenyl]-7-[4-(trifluoromethyl)phenoxy]-9,10-dihydroanthracene-2-carbonitrile N-[2,4-dichloro-6-(1H-pyrazole-5-carbonyl)phenyl]hexanamide 1-(4-aminophenyl)-2-methylindole-6-carbonitrile 1-benzyl-5-(2,3-dihydroindole-1-carbonyl)piperidin-2-one (1S,3R)-N-(benzenesulfonylcarbamoyl)-2,2-dimethyl-6-propan-2-yl-3,4-dihydro-1H-naphthalene-1-carboxamide 2-methylsulfanyl-3-(2,4,6-trichlorophenyl)-N-[1-(1H-1,2,4-triazol-5-yl)cyclopropyl]propanamide 2-amino-7-[(4R,5S)-3,3,4,5-tetrahydroxyoxan-2-yl]oxychromen-4-one 4-[[(2S,3R)-2-(1H-pyrazol-5-yl)oxan-3-yl]methoxymethyl]pyridine 7-[3-[4-(7,8-dihydroisoquinolin-6-yloxy)butanoyl]azetidine-1-carbonyl]naphthalene-2-carbonitrile 3-[2-(4-ethoxyphenyl)ethyl]-1H-indole 4-(2,4,5-trimethoxyphenyl)pyridine (E)-2,3-dichlorobut-2-ene;5-[4-(2-methylpropanoylamino)phenyl]-N-pyridin-4-ylthiophene-2-sulfonamide 3-(4-methylpiperidine-1-carbonyl)-6,7-dihydropyrazolo[5,1-b][1,3]oxazine-2-carboxamide 6-chloro-3-methoxycarbonyl-1,4,9-triazatricyclo[8.4.0.02,7]tetradeca-2(7),10,12-triene-5-carboxylic acid 2-(3-cyanophenyl)-N,4-dimethyl-1H-imidazole-5-carboxamide 3-methyl-5-pyridin-4-yl-1H-indole 4-(2,4-dinitrophenoxy)-N'-hydroxypyridine-2-carboximidamide 2-(3-fluorophenyl)-N-methyl-4-oxochromene-7-carboxamide 6-bromo-3-ethylsulfanylpyrazolo[1,5-a]pyrimidine 6-chloro-2,3-bis(4-nitrophenyl)phenol 4-[(E)-[3,5-bis(trifluoromethyl)phenyl]methylideneamino]oxy-3-methoxypyridine-2-carboxylic acid 3-bromo-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine N-[1-(2,5-dimethoxyphenyl)pyrrolidin-3-yl]-3-thiophen-2-ylpropanamide N-benzyl-1-(5-bromothiophene-2-carbonyl)piperidine-4-carboxamide N-[[2-(azidomethyl)phenyl]methyl]-3,5-dichlorobenzamide 2-(3,4-dihydroxyphenyl)-N,6-diethylimidazo[1,2-a]pyrazine-8-carboxamide N-[2-methyl-4-[(2E,4Z)-hepta-2,4,6-trien-3-yl]phenyl]naphthalene-1-carboxamide 4-ethyl-N'-[[3-fluoro-5-(trifluoromethoxy)phenyl]methyl]-N-[2-(4-methylpiperazin-1-yl)ethyl]thiadiazole-5-carboximidamide [4-(3-acetylanilino)-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-2-yl]-ethylcarbamic acid 2-[(5-cyclobutyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-propanoyl-3H-quinazolin-4-one 2-[3-[methyl(propyl)amino]phenyl]-4H-1,3,4-oxadiazin-5-one 4-chloro-3,5-difluoroquinoline N-(2-methyl-3H-pyrrol-5-yl)-4-[1-methyl-7-[[(3S,4R)-3-methylpiperidin-4-yl]amino]pyrazolo[3,4-c]pyridin-5-yl]benzamide (Z)-2,3-difluoro-1-[4-[(E)-4,5,5-trimethylhept-2-enoxy]phenyl]hex-2-en-1-one N-(cyclopropylmethyl)-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-2-sulfonamide 4-(6,7-dihydrobenzo[c]carbazol-5-yl)-8-methoxycarbonylnaphthalene-1,3-disulfonic acid ethene;methanol;1-[3-(4-propyl-1,2,4-triazol-3-yl)phenyl]pyrazole (3S)-N,3-bis[2-(methylamino)ethyl]-1-sulfanylidene-2H-isoquinoline-7-carboxamide;dihydrochloride 2-[4-[(Z)-1-(3,5-dichlorophenyl)ethylideneamino]oxy-N-methylsulfonylanilino]acetamide 5-(5,7-difluoroquinolin-3-yl)furan-2-carboxylic acid 4-chloro-3,5-dimethyl-1H-pyrrolo[2,3-c]pyridine 2-[1-(3,5-ditert-butylphenyl)-4H-pyrano[4,3-c]pyrazol-6-yl]acetamide 1-[1-methyl-4,5-di(propan-2-yl)imidazol-2-yl]ethanol 4-(5,6,7-trimethyl-[1,2]oxazolo[3,4-b]pyridin-3-yl)aniline 2-N,7-diphenyl-1H-imidazo[4,5-f]quinoxaline 3-[3,4-bis(methylsulfanyl)phenyl]-5-prop-2-ynoxybenzoic acid 4-(9H-fluoren-1-yl)dodecanoic acid 5-[2,4-bis(phenylmethoxy)phenyl]-7-(4,6-dichlorocyclohexa-1,3-dien-1-yl)-N-(4-methylpiperazin-1-yl)-1,6-naphthyridine-2-carboxamide 2-[1-(4,5-dihydropyrrolo[3,2-d]pyrimidin-7-yl)ethoxy]-1,3-benzothiazole 3-[4-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)diazenyl]-N-ethylsulfonylanilino]propanoic acid 5-[1-(4-bromophenyl)pyrazol-4-yl]imidazolidine-2,4-dione 3-methyl-4-(2-oxopiperidin-1-yl)benzamide 3-(3,5-ditert-butyl-4-hydroxyphenyl)propanoyloxyazanium 2-[3-fluoro-5-(trifluoromethyl)phenyl]-1H-pyrrole 1-(3,5-dimethylpyrazol-1-yl)-2-[3-[(4-hydroxy-4-propan-2-ylpiperidin-1-yl)methyl]azetidin-1-yl]ethane-1,2-dione 2-bromo-5-methyl-1-[4-(trifluoromethoxy)phenyl]indole (5S)-2-anilino-N,N-bis[(4-methoxyphenyl)methyl]-3-methyl-2,7-diazaspiro[4.4]nonane-7-carboxamide 3-[[2-(2-hydroxyphenyl)-1,3-benzoxazol-5-yl]amino]propanal (E)-3-[2-[4-[[3,5-bis(trifluoromethyl)phenyl]methoxy]phenyl]-3H-benzimidazol-5-yl]prop-2-enoic acid;hydrochloride 4-azido-6,7-dimethoxyquinazolin-2-amine [1-(4-methylsulfanylphenyl)sulfonylpiperidin-3-yl]methanediol 2-[(4-chlorophenyl)methylsulfanyl]ethylboronic acid 2-[[4-[(6,7-dichloroquinazolin-4-yl)amino]benzoyl]-methylamino]acetic acid 4-hydroxy-2-[(1S)-3-oxocyclohexyl]isoindole-1,3-dione N-benzyl-6,7,8,9-tetrahydro-5H-tetrazolo[1,5-a]azepine-3-carboxamide 2-(3-aminophenyl)-4,5-dimethylphenol 4-[(2,2-difluorocyclopentyl)amino]pyrrolo[1,2-b]pyridazine-3-carboxamide 5-bromo-2,3-dimethoxy-4-methylbenzenesulfonic acid 1-[2-(3,4-difluorophenyl)morpholin-4-yl]-2-[5-methyl-2-(2-methylpropylamino)phenyl]ethanone [4-(3,4-dichlorophenyl)sulfanylphenyl]methanamine;ethane 1-cyclohexyl-3-(6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl)thiourea 2-azido-5-[4-(2-fluorophenyl)phenoxy]-1,3,4-thiadiazole (Z)-4,4,6-trimethyl-3-methylidene-N-[2-[1-(methylamino)ethyl]naphthalen-1-yl]hept-5-ene-1-sulfinamide 4-[5-(3,5-dimethylphenyl)thiophen-2-yl]phenol 1,3-dibromonaphthalene-2-carboxylic acid [1-(2,6-diphenylpyrimidin-4-yl)pyridin-1-ium-2-yl]-methylideneazanium N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-hexadecanoylbenzamide 1-(4-methylsulfonylphenyl)-3-[(2S)-2-(pyrrolidine-1-carbonyl)cyclopentyl]urea 1-[3-(2,5-dioxopyrrol-1-yl)phenyl]piperidine-4-carboxylic acid (2Z)-6-[[4-methoxy-3-[(E)-2-pyridin-2-ylethenyl]phenyl]methylidene]-7H-pyrrolo[3,4-b]pyrazin-5-one 2-(1,2,3,4,5-pentafluoronaphthalen-2-yl)phenol N-(2,6-dimethoxypyrimidin-4-yl)-4-[3,5-dioxo-1-[4-(trifluoromethyl)phenyl]pyrazolidin-4-ylidene]piperidine-1-carboxamide (3R)-N'-[5-chloro-4-fluoro-2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl)phenyl]-3-hydroxypyrrolidine-1-carboximidamide 4-(2,3-dichlorophenyl)sulfonyl-8-[1-(pyridin-4-ylmethoxy)ethyl]-1-oxa-4,8-diazaspiro[4.5]decane (3-methylphenyl)-piperidin-1-ium-2-ylidene-propanoylazanium 2-[3-(2,4-difluorophenyl)-1,2-oxazol-5-yl]acetamide 2-[1-(8,9-dihydrodibenzofuran-3-yl)-5-phenylpyrazol-4-yl]benzene-1,3-dicarbonitrile 2-[(Z)-1,2-difluoro-3-methylsulfanylbut-2-enoxy]-6-methylpyridine 3-ethoxy-2-(4-fluorophenyl)-4-methylsulfonylbenzenesulfonate (3S)-N-[(3-tert-butylphenyl)methyl]-1-[(4R)-1,8-dioxaspiro[4.5]decan-4-yl]pyrrolidine-3-carboxamide (2Z,5E)-1-acetyl-3,4-bis[(5-chloropyridin-2-yl)methylidene]-5-ethylidenepyrrolidine-2-carboxamide 3-[2,6-diethyl-4-(5-fluoro-1H-indole-7-carbonyl)phenyl]propanoic acid 6-[6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonyl(methyl)amino]hexanoic acid 2-[3-(7-methyl-6,8-dihydro-5H-pyrido[4,3-d]pyrimidine-2-carbonyl)phenyl]acetic acid 3-[6-methyl-5-(4-methylphenyl)-2,6-dihydro-1H-pyrimidine-4-carbonyl]benzamide 5-ethyl-3-(oxolan-2-ylamino)pyridine-2-carbonitrile N-[(1R)-2,3-dihydro-1H-inden-1-yl]-6-propan-2-ylpyrimidine-4-carboxamide N-azido-1-(1,3-benzodioxol-5-yl)-1-phenylethanamine N-[(6,8-dichloro-3,4-dihydro-2H-chromen-5-yl)methyl]-1H-pyrazolo[4,3-c]pyridine-7-carboxamide 1-[4-(5,6-dihydronaphthalene-2-carbonyl)phenyl]-3-[1-[4-(4-methylpiperazin-1-yl)-3-(trifluoromethyl)anilino]ethenylamino]thiourea 1-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]cyclohexan-1-ol 1-[(3S,4R)-1-(2,2-difluoroethyl)pyrrolidin-3-yl]-6-methoxyindole N-[(Z)-2-cyclopentyl-2-phenylethenyl]-3,4-dimethoxybenzamide 1-[4-chloro-3-(trifluoromethyl)phenyl]-N'-(2,6-diethylphenyl)sulfonylcyclopropane-1-carbohydrazide 1-[6-methyl-3,4-di(propan-2-yl)quinolin-8-yl]oxypentan-2-ol 2-(3-chlorophenyl)imino-5-[(1-methylindazol-6-yl)methylidene]-1,3-thiazolidin-4-one N'-(2,5-difluoro-3-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridine-4-carbohydrazide 1-[[(2R,3S)-5-azido-3-methylpentan-2-yl]oxymethyl]naphthalene 5-azido-2-(4,4-diethylpiperidin-1-yl)pyridine 4-[(5,7-dimethylquinolin-8-yl)amino]pyridine-2-carboxamide 1-[(4-methoxyphenyl)methyl]-2,3,6-trimethyl-2H-benzimidazole [2,3-bis(ethenyl)phenyl]methanamine N-[(1E)-1-[3-[4-(2-fluorophenyl)-1H-pyrrolo[3,2-c]pyridin-2-yl]-5,6-dihydro-1H-indazol-5-yl]buta-1,3-dienyl]ethanimine 4-(3-azidobutyl)-6-chloropyridazine 1-[2-azidooxy-3,4,5,6-tetrachloro-4-(phenylmethoxymethyl)heptanoyl]azetidine-2-carbonitrile 5-(3,4-dimethoxyphenyl)-2-oxopentanoic acid 1-cyclohexa-2,4-dien-1-yl-N-methyl-6,7-dihydro-5H-pyrazolo[3,4-d]pyrimidine-4-carboxamide 3-(6-butoxynaphthalen-2-yl)propanoic acid ethane;3-[4-(2-fluorophenyl)-1H-pyrrolo[3,2-c]pyridine-2-carboximidoyl]-5-methylaniline 1-amino-4-(3,4-dichlorophenoxy)butan-2-ol 4-[2-amino-6-(3-bromophenyl)pyrimidin-4-yl]piperazine-1-carboxylate 2-[(5S)-2-(cyclopropanecarbonylamino)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]acetic acid 2-hydroxy-N'-[2-(4-methylphenyl)ethyl]benzohydrazide N-azido-3,5-bis(ethenyl)benzenesulfonamide 4-[3,5-diethoxy-2-(2-hydroxyethyl)anilino]phenol 2-(3,4-difluorophenyl)-1H-indene 2-[(4,6-dimethoxy-1,3,5-triazin-2-yl)-ethylsulfonylamino]acetic acid 6-[2-(4-methylpyridin-3-yl)acetyl]oxyhexanoic acid 4-methyl-N-[(3R,5S)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]-2-(trifluoromethylsulfanyloxy)benzamide 3-ethyl-4-[(1Z)-2,2,5,6,6-pentamethylcycloocta-1,3-dien-4-yl]benzaldehyde 2-(7,8-difluoroquinolin-3-yl)benzonitrile;1-(3-hydroxyazetidin-1-yl)ethanone [6-methyl-3-(5,5,8,8-tetramethylnaphthalene-2-carbonyl)oxypyridin-2-yl]boronic acid N-[(2S)-3-methoxypropyl]-4-nitro-1H-pyrrolo[2,3-c]pyridine-7-carboxamide 3-[3-[2-(7,7-dimethylcycloocta-1,4,6-trien-1-yl)ethyl]-3-ethylazetidin-1-yl]-N-hydroxypropanamide 3-[4,6-bis(4-methylphenyl)pyrimidin-2-yl]pyridine;ethane 2-[6,6,8-trimethyl-7-(1H-pyrrole-3-carbonyl)-4-phenyl-5,7-dihydropyrazolo[3,4-b]pyridin-3-yl]acetamide 4-[2-azido-5-(trifluoromethyl)phenyl]butan-1-amine 2-[(2,6-dichloro-4-nitrophenyl)methyl]-5-(4-fluorophenyl)pentanenitrile N-[(1,1-dioxothiolan-3-yl)methyl]-N-ethyl-4-methoxypyrimidine-5-carboxamide 5-(2,3-dimethylimidazol-4-yl)-3-[4-(furan-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-2H-pyrazolo[3,4-b]pyridine 3-amino-5,6-difluoro-N-[4-[4-(1H-pyrazole-4-carbonyl)morpholin-2-yl]phenyl]pyridine-2-carboxamide [5-(7-methoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)pyrazin-2-yl]-[4-[2-phenylethyl(propan-2-yl)amino]piperidin-1-yl]methanone 1-methylsulfonyl-4-[(3E,5Z)-octa-1,3,5,7-tetraen-3-yl]benzene 1-(1,5-dimethylbenzimidazol-2-yl)-N-methylethenamine 2-(4,6-dimethoxypyrimidin-5-yl)-3,4-bis(ethenyl)-7,8-difluoropyrazolo[1,5-a]quinoline 4-[2-[(3-chlorophenoxy)methyl]phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 5-azidooxy-3,3-dimethyl-1,2-benzothiazol-4-amine 5-benzylsulfanyl-2,3,6,7-tetrahydroindole N-[(3,5-diethylphenyl)methylideneamino]formamide;4-[[[1-[(3R)-piperidine-3-carbonyl]azetidin-3-yl]-pyridin-2-ylcarbamoyl]oxymethyl]benzoic acid ethane;2-(3H-indol-4-yl)ethanamine;2-methoxyprop-1-ene;3-phenyl-6-(4-thiophen-2-ylphenyl)pyridazine (E)-3-[5-[6-amino-2-methyl-5-(1,4-oxazepan-4-yl)pyrimidin-4-yl]thiophen-2-yl]prop-2-enal 2-(2-bromo-N-butyl-4-fluoroanilino)ethanol [6-(2,4-dichlorophenyl)-1H-pyridazin-5-yl]methanol 7-[2-(3,4-dimethylphenyl)ethynyl]-2-methyl-5H-pyrrolo[1,2-a]quinoxalin-4-one 6-[3-(dimethylamino)prop-1-ynyl]-N'-hydroxy-5-nitropyridine-2-carboximidamide [2,6-di(propan-2-yl)phenyl]methylphosphane 1-bromo-3,5-bis(4-tert-butylphenyl)benzene;ethane N-[[1-benzyl-4-(5-methoxypyridin-3-yl)pyrrolidin-2-ylidene]amino]pyrimidin-2-amine 5-(N,2-dimethylanilino)isoindole-1,3-dione 2-[(3-bromophenyl)sulfanylmethyl]-4-[(3R,5S)-3,5-dihydroxypiperidin-1-yl]-6-oxopyran-3-carbonitrile (2S)-N-[4-[4-hydroxy-5-methoxy-3,6-dioxo-1-(2H-triazol-4-yl)pyridazin-4-yl]phenyl]pyrrolidine-2-carboxamide (E)-N'-[5-chloro-2-oxo-4-(trifluoromethylsulfanylamino)pyrimidin-1-yl]but-2-enimidamide;ethane 2-(7-aminopyrido[3,4-b]pyrazin-5-yl)oxy-N-methylbenzamide (2R,3S)-5,7-dihydroxy-N-propan-2-yl-8-(pyridine-4-carbonylamino)-6-[3-(trifluoromethyl)phenyl]iminooctanamide 4-[2-azidooxy-1,1-difluoro-2-(3-nitrophenyl)ethyl]benzenesulfonic acid 5-chloro-3,4-dihydroxy-N-[(E)-2-methoxybut-2-enoyl]naphthalene-1-carboxamide 2-(3,5-dimethylpiperidin-1-yl)-N'-hydroxypyridine-4-carboximidamide 3-[(4-tert-butylphenyl)sulfanylamino]oxane-2,5-dione N-[1-(2-methyl-6-oxopyran-4-carbonyl)pyrrolidin-3-yl]morpholine-4-carboxamide 2-hydroxy-5-[4-(3-hydroxyphenyl)but-1-enyl]benzoic acid 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]acetonitrile 5-methyl-N-[(4R,6S)-6-methyl-1-azabicyclo[3.2.0]heptan-7-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide ethane;1-methyl-4-[2-(6-phenylcyclohexa-1,5-dien-1-yl)propan-2-yl]benzene 4-[[5-bromo-1-(pyridin-3-ylmethyl)indole-2-carbonyl]amino]cyclohexane-1-carboxylic acid [6-(2,4-dimethoxyphenyl)-3-propan-2-ylthieno[2,3-b]pyridine-4-carbonyl]-methylideneazanium 2-[5,6-dimethoxy-1-[(4-nitrophenyl)carbamoyl]naphthalene-2-carbonyl]cyclopropane-1-carboxylic acid 3-(4,5-dihydro-1H-imidazol-2-yl)-N,N-dipropylbenzamide 5-(1-azidopiperidin-3-yl)oxypyridine-2-carboxylic acid 4-[[6-(2,2-difluoroethoxy)pyridin-3-yl]methylamino]-2-(oxan-4-ylsulfanylmethyl)-1H-pyrimidin-6-one 3-methyl-2-[(2Z)-2-[1-(4-octoxyphenyl)ethylidene]hydrazinyl]quinazolin-4-one 2-amino-6-[3,5-dimethoxy-4-(trifluoromethyl)phenyl]-4,4-dimethoxy-3-azabicyclo[3.1.0]hex-2-ene-1,5-dicarbonitrile 2-[4-(methyliodanuidylmethyl)phenyl]acetic acid 3-[4-chloro-2-(fluoromethyl)anilino]-2,2-dimethyl-N'-methylidenepropanimidamide 4-(2,3-dimethylphenyl)-N-[2-[1-[4-[[2-[6-(2-methoxyethylimino)piperidin-2-ylidene]hydrazinyl]methyl]naphthalen-1-yl]azetidin-3-yl]pyridin-3-yl]piperazine-1-carboxamide 4-(3-azidooxypropyl)-2,6-dimethylpyridine 3,6-ditert-butyl-10H-phenothiazine 2-(5-acetyl-6,7-dimethoxy-1H-indol-3-yl)acetate 4-[3,5-bis(methylamino)phenyl]-N-ethyl-2H-pyridine-1-carboxamide N-[4-(4-chlorophenoxy)phenyl]-2-methoxy-5-nitropyridine-3-carboxamide 1-(3-methoxyphenyl)sulfonyl-4-methylpyrrolo[2,3-b]pyridine 1-methylsulfonyl-3-propan-2-yl-6,7,8,9-tetrahydropyrrolo[3,2-c][1,7]naphthyridine 1-(4-propan-2-yloxy-3,5-dipropoxyphenyl)ethanesulfonic acid (3-azidopiperidin-1-yl)-[4-(2,3-dichlorophenyl)piperazin-1-yl]methanone 4-[5-(2,6-difluorophenyl)hexanoyl]morpholine-3-carbonitrile 3-(2-chlorophenyl)-N-[3-methoxy-4-(2,2,2-trifluoroethylsulfonylamino)phenyl]octanamide N-(4-bromophenyl)-4-(3,4-dimethylanilino)pyrrolo[1,2-b]pyridazine-2-carboxamide 4-[(1-phenylcyclopropyl)methylamino]piperidine-1-carboxylic acid 5-fluoro-1,3-diphenylbenzimidazol-2-imine N-[3-(difluoromethyl)phenyl]spiro[1,4-dihydroquinoline-3,1'-cyclohexane]-2-imine 2,6-dibromo-4-[(E)-[[6-(1H-indol-3-ylmethylideneamino)-1,3-benzothiazol-2-yl]hydrazinylidene]methyl]phenol 2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-3-ylmethyl)benzaldehyde 1-[4,6-dimethoxy-2-(7H-purin-6-ylamino)benzimidazol-1-yl]-3-phenylpropan-2-one N-[4-(4-fluoro-3-methoxyphenoxy)phenyl]-2,5-dimethylpyridine-3-carboxamide 4-[(2R)-2-amino-3,3,3-trifluoropropyl]sulfanyl-5-methoxy-1H-pyrimidin-6-one 3-(3,4-dimethylpiperazin-1-yl)-2-fluoro-N'-hydroxypyridine-4-carboximidamide (Z)-but-2-ene;N-ethyl-1,4,5-trimethoxy-6-oxopyridine-3-carboxamide 1-[4-(2,5-difluorophenyl)butyl]cyclohexane-1-carboxylic acid 4-[[2-chloro-3-(methoxymethyl)benzoyl]amino]oxolane-3-carboxamide 4-[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)phenyl]sulfonylmorpholine (1R,5S)-3-(2-diazohydrazinyl)-1-[4-(difluoromethoxy)phenyl]sulfonyl-3-azabicyclo[3.1.0]hexan-2-one 2-[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]phenol 5-amino-6-N-(1-aminocyclopentyl)-4-chloro-2-N-[2-(2,4-dimethoxyphenyl)ethyl]pyrimidine-2,4,6-triamine N-(3-azidopropyl)-4-oxochromene-2-carboxamide 5-fluoro-N-[(3R,4S)-1-methylsulfonyl-4-pyrazol-1-ylpyrrolidin-3-yl]pyrazine-2-carboxamide 1-[(3E)-4-[6-chloro-2-ethyl-8-fluoro-7-(2,2,2-trifluoroethoxy)quinazolin-4-yl]-3-methylpiperazin-1-yl]prop-2-en-1-one;methanol 6-(3-cyclobutylphenyl)hexanamide 2-azido-6-[3,5-bis(trifluoromethyl)phenyl]benzonitrile 3-amino-6-(3,4-dimethoxyphenyl)-N-[2-oxo-1-phenylpentan-3-yl]hexanamide N-[(3R,4S)-1-[2-(4,5-dimethylpyrazol-1-yl)ethyl]-4-propan-2-ylpyrrolidin-3-yl]morpholine-4-carboxamide;hydrochloride N-[3-[2-(4-amino-1,2,5-oxadiazol-3-yl)-3-propan-2-ylimidazo[1,2-a]pyridin-7-yl]phenyl]methanesulfonamide 4-[(E)-2-chlorobut-1-enyl]-N-[2,6-difluoro-3-[5-methoxy-4-oxo-3-[4-(trifluoromethylsulfonyl)phenyl]phthalazin-1-yl]phenyl]cyclohexane-1-carboxamide 1-[(4-ethylphenyl)methyl]-3-[(2S,6R)-5-hydroxy-6-propan-2-yloxepan-2-yl]urea N-(4-nitrophenyl)-5-propanoylcyclohexa-1,3-dien-1-amine 1,3-dimethyl-5-[2-(4-phenylpiperazin-1-yl)ethoxy]benzimidazol-2-one;hydrochloride 4-chloro-6-methylsulfanyloxynaphthalene-2,7-dithiol N-[4-(azidomethyl)cyclohexylidene]-3,5-bis(trifluoromethoxy)benzamide [2-(1,5-dimethylpyrazol-4-yl)pyridin-3-yl]oxyboronic acid (1Z)-1-[3-hydroxy-5-(2H-tetrazol-5-yl)-6,7-dihydrobenzo[f]benzimidazol-8-ylidene]guanidine [(2R,3S)-3-methoxypiperidin-2-yl]-phenylmethanone;hydrochloride 2-[4-bromobutan-2-yl(hexyl)amino]benzoic acid 6-[(Z)-2,3-dimethylbut-1-enyl]-1-propan-2-yl-5H-pyrazolo[4,3-c]pyridin-4-one;ethane 2-(4,5-dihydropyrrolo[3,2-d]pyrimidin-7-yl)-4-[(1S)-1-(2-methylpropylamino)ethyl]-6-thiophen-2-ylphenol 3-methyl-4-propan-2-ylidenethioxanthene-9,10-dione 3-(3,5-dichloro-4-fluorophenyl)oxirane-2,2-dicarbonitrile 4-(3,7-dimethoxyquinoxalin-2-yl)phenol 4-bromo-6-chloro-1-ethylpyrrolo[2,3-b]pyridine;ethane 2-amino-4,5,6-trichloropyridine-3-carboximidamide;cyclopropanol [6-(4-fluorophenyl)spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-yl]-(5H-pyrrolo[2,3-b]pyrazin-7-yl)methanone;formic acid 5-amino-N'-azido-1H-indole-2-carboximidamide 2-(4-ethylcyclohexyl)-5,6,7,8-tetrahydroquinoline ethene;4-(10,10,10-trifluorodecyl)pyridine N-benzyl-3,7-dimethoxy-5-(2-methylidenehydrazinyl)-6-oxocyclohepta-1,4,7-triene-1-carboxamide 4-[2,6-difluoro-3-(methyliminomethyl)phenyl]-1H-indole-7-carboxylic acid 1-(5-amino-4,4,7,6,10,11,12-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-8-yl)pyrrolidin-2-one 2-[4,6-bis(prop-1-en-2-yl)-3,5-dihydro-2H-pyrazin-1-ium-1-yl]aniline 4-(2,3-dimethylphenyl)sulfonylpyrrolidine-3,4-dione 6-bromo-2-tert-butyl-3H-quinazolin-4-one N-cyclohexyloxy-N,3-dimethylaniline (2R)-2-[(1,3-dioxoisoindol-2-yl)amino]butanoic acid N-azido-4,6-dichloro-5-[5-(3-ethynylphenyl)furan-2-yl]pyrimidin-1-ium-2-amine N-[5-(2,3-dichlorophenyl)sulfinyl-1H-indazol-3-yl]-4-piperidin-4-ylbenzamide 1-[(2S,4R)-2-methyloxan-4-yl]-N-[(1R,2R)-2-thiophen-3-ylcyclopropyl]piperidine-4-carboxamide 3-[(1S,2R)-2-[[4-[[cyclohexyl(propanoyl)amino]methyl]phenyl]sulfonylamino]cyclopentyl]pyridine-4-carboxylic acid 2-[4-ethyl-3-(trifluoromethoxy)phenyl]pyrimidine 2-[4-(3,4-difluorophenyl)-5-methylsulfonylthiophen-2-yl]-N-(4,6-dimethoxypyrimidin-2-yl)acetamide 2-benzamido-4,6-dihydropyrrolo[3,4-d][1,3]thiazole-5-carboxylic acid 1-azidooxy-3,4,5-trimethylnaphthalene 1-azidooxy-N-(cyclohexylcarbamoyl)isoquinoline-7-carboxamide 4-azido-N,5,6-trimethylpyridazin-3-amine N-[2-[(1Z,3E)-4-methylpenta-1,3-dienyl]-1-phenylcyclopropyl]thiophene-3-carboxamide 2-(4-fluorocyclohexa-1,5-dien-3-yn-1-yl)-5-[(1-methoxypyrrolidin-2-ylidene)amino]-1-methylbenzimidazole-4,6-dicarbonitrile 2-(4-tert-butylanilino)-5,7-dihydropyrrolo[3,4-d]pyrimidine-6,8-diol 4-(4-iodophenyl)-2H-chromene (Z)-2-[2,3-dihydroxypropyl-(4-morpholin-4-ylphenyl)iminomethyl]-1-hydroxypent-2-en-1-ol N-[5-(hydroxymethyl)oxolan-3-yl]-6,7-dihydro-4H-thieno[3,2-c]pyran-4-carboxamide 2-[3-methylbut-2-enyl(1,3-thiazol-5-yl)amino]acetonitrile 1-[4-(3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidine-3-carboxamide 2-(furan-3-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 2-ethyl-8-methoxy-3H-quinazolin-4-one 5-chloro-1-[4-(2,3-difluoro-2H-pyridin-1-yl)phenyl]-2,6-naphthyridine;3-methylmorpholine N-[(2S)-3-cyclohexyl-1-oxo-1-(2,4,5-trifluoroanilino)propan-2-yl]-2-methoxypyridine-3-carboxamide 4-azido-5,6-dibromospiro[2H-1-benzofuran-3,9'-xanthene] N-butyl-4-methoxy-3,5,8,10,14-pentazatetracyclo[7.6.0.02,6.011,15]pentadeca-1(9),2(6),4,7,11(15),12-hexaene-13-carboxamide;ethane [6-[(1R)-4,7-diamino-2-methyl-4,5,6,8-tetrahydroquinazolin-3-ium-6-yl]-4H-thiopyran-3-yl]methanol 5-[2-[(4S)-8,9-dimethyl-6-oxo-1,2,3,4-tetrahydroquinolizine-4-carbonyl]phenyl]pentanenitrile 3-[2-(4-phenylpiperazin-1-yl)ethoxy]benzamide 5-butyl-2-(2,6-difluoro-4-propoxyphenyl)thiophene 6-amino-1,3-bis(4-chlorobutyl)pyrimidine-2,4-dione N-[2-[3,5-difluoro-4-(trifluoromethyl)phenyl]propan-2-ylsulfanylmethyl]-1-[4-(trifluoromethoxy)phenyl]ethanamine N-[2-(4-methoxy-6,7-dihydrothieno[3,2-c]pyridine-5-carbonyl)cyclohexyl]-1H-pyrrole-3-carboxamide 2-[4-[3-(2,5-dimethylpyrazol-3-yl)propanoyl]morpholin-3-yl]benzoic acid 4-[1-(cyclohexylmethylamino)but-3-enyl]aniline 2,6-dimethyl-1-(3-thiophen-2-ylphenyl)-9H-fluorene N-(2,6-dimethylphenyl)-4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridine-2-carboxamide (E)-3-[5-methyl-2-(4-sulfophenyl)iminophenyl]prop-2-enoic acid [(2R,4S)-4-hydroxy-1-methylpyrrolidin-2-yl]-[4-[(3R,5R)-5-methoxyoxan-3-yl]piperidin-1-yl]methanone;formic acid 4-[[(3S)-3-fluoropyrrolidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine (2S)-N,1-dihydroxy-4-[2-[6-(4-methylphenyl)-3H-inden-5-yl]ethoxy]butan-2-imine 2-[4-cyano-N-(3,3,3-trifluoropropyl)anilino]-2-methyl-N-[6-oxo-1-(pyrimidin-5-ylamino)heptan-2-yl]propanamide;ethane 3-[1-(4-aminopiperidin-1-yl)ethoxy]-N-tert-butylbenzamide N-[[1-(6,7-dimethoxyquinazolin-4-yl)piperidin-3-yl]methyl]-1H-indazole-5-carboxamide 3-chloro-4-[2,6-dimethyl-4-(trifluoromethoxy)phenyl]-5-methoxybenzoic acid 4-[3-[6-methyl-1-oxo-5-(4,4,4-trifluorobutanoyl)isoquinolin-2-yl]phenyl]piperazine-1-carboxylic acid 1-cyclopropyl-6-fluoro-7,8-dimethoxy-4-oxoquinoline-3-carboxylic acid 2-(5,6-dichloro-1H-benzimidazol-2-yl)-4-(methoxymethoxycarbonyl)piperazine-1-carboxylic acid 2-benzyl-5-[[6-(ethenylamino)pyridine-3-carbonyl]amino]benzoic acid 3-(4-aminobenzoyl)oxypropanoic acid 2-[(5R,10bR)-7-methoxy-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 7-(2,4-diaminophenoxy)naphthalene-1,3,5,8,9-pentone 4-[2-(2,6-difluorophenyl)-1-fluoroethenyl]phenol [6-(1H-indazol-5-ylamino)pyrimidin-4-yl]oxyboronic acid (2S,4R)-N-[1-amino-3-(aziridin-2-ylmethylimino)prop-1-en-2-yl]-1-(cyclohexanecarbonyl)-4-phenylpiperidine-2-carboxamide 4-chloro-3-[2-hydroxy-5-(trifluoromethyl)phenyl]cyclobut-3-ene-1,2-dione N-[3-methoxypropyl(pyridin-3-yl)amino]formamide (2R)-4-[7-chloro-1-(4-fluorophenyl)indazol-3-yl]sulfonylmorpholine-2-carboxylic acid 2,4-dichloro-N-(1,2,3,3a,4,5,6,6a-octahydropentalen-2-yl)benzamide (4-chlorophenyl)methyl-diethoxyphosphane 1-(2-ethoxyphenyl)pentane-1,3-dione 1-butyl-3,5-bis(methoxymethoxy)benzene 3-[4-(2-morpholin-4-ylethoxy)phenyl]sulfonylchromen-4-one [3-(6-aminopyridazin-3-yl)piperidin-1-yl]-(2-methylthieno[3,4-b]pyrrol-5-yl)methanone 4-[4-(ethylamino)piperidine-1-carbonyl]benzenesulfonamide 2-[1-(azidomethyl)piperidin-3-yl]oxypyridine 4-(methoxymethyl)-N,N-diphenylaniline N-[(3R,4S)-1-[2-(difluoromethoxy)phenyl]sulfonyl-4-fluoropyrrolidin-3-yl]propane-2-sulfonamide 2-[2-[(1,5-dimethylpyrazol-3-yl)methoxy]phenyl]ethanol (E)-3-[2-(4,4-difluorocyclohexyl)oxyphenyl]-1-[4-[2-(oxan-2-yl)pyrazol-3-yl]-5-sulfamoylthiophen-2-yl]prop-2-en-1-one N-[2,3-difluoro-4-[1H-indol-3-yl(methylamino)methyl]phenyl]-2,6-difluorobenzenesulfonamide 2-bromo-4-tert-butylthiophene;5,7-dihydroxy-3-(4-methoxyphenyl)chromen-4-one (3R,4R)-4-[1-[4-cyano-3-(trifluoromethyl)phenyl]piperidin-4-yl]-N-cyclopropyl-1-(4,4-dimethoxybutyl)pyrrolidine-3-carboxamide (5Z)-2-(2,4-dimethylphenyl)imino-5-[(3-ethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 4-[6-(2-aminoethyl)pyrimidin-4-yl]oxy-N'-methanimidoylbenzohydrazide N-azido-4,5-diphenyl-1,3-thiazol-2-amine N-[(5S)-8-bromo-5,6,7,9-tetrahydropyrido[2,3-c]azepin-3-yl]-N-methylpropanamide 2-(3,4-dibromophenyl)-1,4,5,6-tetrahydropyrimidine 5-ethyl-6,8-dihydroxy-3H-quinazolin-4-one N-[(3S,4R)-1-[3-(azepan-1-yl)propanoyl]-4-methoxypyrrolidin-3-yl]-5-chlorothiophene-2-carboxamide 2-[5-carbamoyl-2-chloro-9-(furan-3-ylmethyl)carbazol-4-yl]oxyacetic acid 5-[2-(4,4-difluoroazepane-1-carbonyl)piperidine-1-carbonyl]-3-methyl-1H-benzimidazol-2-one 4-[[8,10-dichloro-7-(2-methoxyethyl)-1H-benzo[g]isoquinolin-3-yl]amino]pyridine-3-carbonitrile 1-butyl-3-(2,6-dimethoxyphenyl)imidazole-2-thione (2R)-N-[2,4-difluoro-3-[5-pyridin-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]phenyl]-2,3,6-trifluoro-5-methoxybenzenesulfonamide 2-methyl-6,7-dihydroquinoline-3,4,5,6-tetracarbonitrile (1R)-3,6-dimethyl-2-(prop-2-enoylamino)cyclohex-2-ene-1-carboxylic acid;ethane 2-(cyclopropylmethoxy)-5-fluoro-N'-hydroxypyrimidine-4-carboximidamide 2,2-dimethyl-N'-[(E)-2-phenylethenyl]pentane-1,5-diimine 4-[6-(2,3-difluorophenyl)pyridazin-3-yl]piperidine-1-carboxylic acid 2-[3,6-dihydroxy-5-(hydroxymethyl)-2-propanoylphenoxy]acetic acid 5-[6-methoxy-2,4-bis(phenylmethoxy)pyridin-3-yl]-1H-pyrazole-4-carboxamide (E)-N'-methyl-3-phenylprop-1-ene-2,3,4-triamine 4-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)imidazol-1-yl]pyridine-2-carboxylic acid;dihydrochloride N-[2,3-bis(4-methylphenyl)phenyl]dibenzofuran-1-amine;2-methylidenecyclopentane-1,3-dione 5-[1-(ethylsulfamoyl)pyrrolidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide 3-(4-fluorophenyl)-7-piperidin-1-yl-4H-pyrazolo[1,5-a]pyrimidine-5-thione 6-(2,2-dimethylhydrazinyl)-N-phenylpyridine-3-carboxamide 3-[2,4-bis(trifluoromethyl)phenyl]-5-bromopyridine N-azido-N-(pyrimidine-2,4-diyloxy)nitramide 4-chloro-2,5-diethylpyrazolo[3,4-b]pyridine N-[3-chloro-4-(pyridin-2-ylcarbamoyl)phenyl]piperidine-1-carboxamide N-(2,4-dichloropyrimidin-5-yl)-6-nitro-N-(3-methylbutyl)-1,3-benzothiazol-2-amine 4-(2,6-difluorophenyl)-5-methyl-1-[3-(trifluoromethoxy)phenyl]pyrazole 4-ethyl-6-methoxyspiro[chromene-2,1'-cyclopentane] 5-[1-(1,3-benzodioxol-4-yl)cyclopropanecarbonyl]-1-(1H-imidazol-2-ylmethyl)pyrimidine-2,4-dione 4-[2-hydroxy-3-[(E)-3-phenylprop-1-enyl]-5-propanoyloxyphenoxy]benzoic acid N-(4-hydroxycyclohexyl)-N-methyl-3-[5-(trifluoromethoxy)pyridin-2-yl]sulfanylpropanamide 2-[(3Z,6Z)-3-[4-(methylamino)anilino]octa-1,3,6-trien-4-yl]benzaldehyde;N,N,5-trimethylpyridin-2-amine 7-[3,5-difluoro-4-[3-(trifluoromethyl)phenyl]anilino]quinoxaline-2-carboxylic acid;ethane (2E)-N-[[4-[cyclopentyl(prop-1-en-2-ylamino)methyl]phenyl]methyl]-2-(hydroxymethylidene)hexanamide N-[4,6-bis(2-methylpyrazol-3-yl)pyridin-3-yl]sulfanyl-5-tert-butyl-2-fluoroaniline 2-fluoro-4-[1,3,3a,4,6,6a-hexahydrofuro[3,4-c]pyrrole-5-carbonyl(methyl)amino]benzoic acid (5R,7S)-N-(2,4-dichlorophenyl)-5-(furan-2-ylmethyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 5-[6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)naphthalen-2-yl]benzimidazolo[1,2-a]quinoline 1-(2,6-dichlorophenyl)-3-[5-(4-oxo-3H-quinazolin-2-yl)pentanoylamino]thiourea 2-methoxycarbonyl-3-(5,7,8,10-tetrazatricyclo[7.4.0.02,6]trideca-1(13),2,4,9,11-pentaen-12-yl)propanoic acid 4-[2,3-bis(ethenyl)phenyl]benzenesulfonate;1,3-dimethylpyrrolidine;yttrium 1-(4,5-dimethylcyclohexa-1,3-dien-1-yl)oxy-2-ethoxybenzene;methane 2-amino-7,8-dimethyl-3-[4-(trifluoromethyl)phenyl]purin-6-one 4-[2,6-dichloro-N-(3-methylbutyl)anilino]benzenesulfonamide 2-[[3-amino-5-(2,4-dimethoxypyrimidin-5-yl)-1H-pyrrole-2-carbonyl]amino]acetic acid 4-(2-propan-2-ylphenyl)morpholine 2-[1-(3,5-diethylcyclohexyl)piperidin-4-ylidene]butanal;3,6-dimethyl-N-propyl-N-[2-(trifluoromethoxy)phenyl]pyridine-2-carboxamide 1-[(2,3-difluorophenyl)methyl]-N-[(E)-4-(methylideneamino)pent-3-en-2-yl]indole-5-carboxamide N-[5-(3,4-dihydrocarbazol-9-yl)hexan-2-yl]acetamide 1-(4,5-dimethoxypyrimidin-2-yl)-3-(7H-purin-6-ylamino)urea 4-chloro-2-[(Z)-2-methoxycarbonyl-3,3-dimethylbut-1-enyl]benzoic acid (2-methylphenyl)-[4-(pyridine-4-carbonylamino)phenyl]azanium 5-(3-benzyl-1H-indol-2-yl)-3-phenylpenta-2,4-dienal 1-(4-methoxyphenyl)-N-[2-(3-methylimidazol-4-yl)ethyl]cyclopropane-1-carboxamide 4-[3-(dimethylamino)propoxy]-2,5,6-trimethylbenzene-1,3-diol 6-[(3aR,8aS)-3a-methyl-1,2,3,4,5,7,8,8a-octahydropyrrolo[3,4-d]azepine-6-carbonyl]pyridine-3-carbonitrile 3-methylsulfanyl-6-[3-(trifluoromethyl)phenyl]-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-1-one 3-(4-chlorophenyl)-1-methylpiperidine 1-[2,4,6-tris(phenylmethoxy)benzoyl]oxycyclohexane-1-carboxylic acid 5-[6-azido-2,3-di(propan-2-yl)phenyl]-1H-pyrazole 4-N-[(1E,3Z)-hexa-1,3,5-trienyl]benzene-1,4-diamine 4-[2-azidooxy-1,1-bis(phenylmethoxy)ethyl]phenol 2,4-diaminopyrimidine-5-carbonitrile;1-[(3S)-6-methoxy-3-methyl-3H-indol-2-yl]pentan-1-one 2-[(6S)-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]-N-(3,4,5-trifluorophenyl)acetamide 1-[[1-(6,7-dimethoxyquinolin-4-yl)piperidin-3-yl]methylamino]ethenethiol 5-[2-(4-amino-3,5-dichlorophenyl)ethyl]pyrimidine-2,4-diamine 1-(1,4-dihydroimidazo[4,5-c]pyrazol-6-yl)-3-(4-pyridin-2-yloxyphenyl)urea;ethane 4-amino-6-[(3,5-difluorophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-[2-azido-6-(trifluoromethyl)pyridin-3-yl]benzaldehyde 1-(azetidine-1-carbothioyl)pyrazole-4-carboxylic acid 4-(1H-imidazol-2-yl)-1,2,5,6-tetrahydrothieno[3,2-e]indole 2-azidooxy-3-(4-chlorophenyl)pyrazine 2-(4-methoxyphenyl)-7,8-dihydroquinazoline 4-amino-2,6-dinitro-N,N-bis(prop-2-enyl)benzenesulfonamide 2-bromo-6-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]phenol 3-(2,4-dichlorophenyl)-1-hydroxyazetidine;propanal 4-[(7-methoxy-1H-indol-3-yl)methyl]aniline 4-(azidomethyl)-2,3,5,6-tetrafluorophenol 3-(2,4,6-trichloro-N-ethylanilino)propane-1,2-diol 4-[(5-phenylpyridin-2-yl)amino]cyclohexan-1-one 1-[(3R,5S)-1,4-dihydroxy-5-propan-2-ylpyrrolidin-3-yl]-3-(1H-indol-4-ylmethylamino)thiourea 5-methyl-1-[4-(3,6,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,11-tetraen-4-ylsulfonyl)phenyl]pyrazole-4-carboxylic acid [5-(3,4-dichlorophenyl)-2H-benzotriazol-4-yl]boronic acid 2-amino-4-(3,5-dihydroxyphenyl)pyridine-3-carboxamide (4R,7S)-4-[1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl]oxy-6,8-difluoro-2,3,5,7-tetrahydrooxepine 4-[3-(3,5-dichlorophenyl)-1H-pyrazole-5-carbonyl]-N'-hydroxypiperidine-1-carboximidamide 2-bromo-7-methylquinoxaline N-[4,5-bis(4-methoxyphenyl)-1H-imidazol-2-yl]acetamide 2-(4,5-dimethylcyclohepta-1,3,6-trien-1-yl)oxy-N'-hydroxypyrimidine-4-carboximidamide 1-[4-chloro-2-fluoro-5-(trifluoromethyl)phenyl]pyrrolidine;3,6-dihydro-2H-pyran 1-[4-[(2,5-dimethylphenyl)sulfamoyl]-N-nonanoylanilino]propanoic acid N-[5-[3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]cyclohexanecarboxamide 2,4-dichloro-N-[2-(6-methylcyclohexa-1,3-dien-1-yl)phenyl]benzamide 2-[1-(3,5-difluorophenyl)sulfonylpiperidin-4-yl]benzoic acid 4-chloro-6,7-dimethoxy-3H-quinazolin-2-one 4-[[3-fluoro-5-(trifluoromethyl)phenoxy]methyl]piperidine 4-[3-[2-(3-methylthiophen-2-yl)pyridin-3-yl]propylamino]cyclohexan-1-ol (2E)-2-(1,3-benzodioxol-5-ylmethylidene)-5-(3,5-ditert-butylphenyl)-4-propan-2-ylfuran 1-methoxy-2-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethanol 4-[(3-azido-5,6-difluoropyridin-2-yl)methyl]morpholine 2-[4-chlorobutyl(methoxycarbonyl)amino]benzoic acid 5-(3,4-dichlorophenyl)imidazolidine-2,4-dione (5-azido-1,3-benzodioxol-4-yl)methanamine 5-azido-2,3-dihydro-1H-indole;hydrate [(2S,4R)-5-azido-1-benzyl-4-hydroxypyrrolidin-2-yl]methanol 4-(6-amino-7-methyl-2,3-dihydro-1H-inden-5-yl)-N-phenylpyridin-2-amine [4-amino-1-[5-(difluoromethyl)pyridin-3-yl]pyrrolidin-2-ylidene]cyanamide 3-[5-(4,5-difluoro-2-hydroxyphenyl)imidazo[1,2-a]pyrazin-8-yl]benzonitrile;ethane [(5R,7S)-2-ethyl-6-oxa-2-azaspiro[4.5]decan-7-yl]-(1H-indol-3-yl)methanone;2,2,2-trifluoroacetic acid 6-bromo-3H-pyrido[2,3-d]pyrimidin-4-one;ethane (E,2E)-2-ethylidene-N'-[(3-methylpyridin-2-yl)methyl]hex-4-enimidamide 2-[6-[4-(3,5-dimethylpyridine-4-carbonyl)piperazin-1-yl]-9H-xanthen-3-ylidene]acetic acid 4-[(1,3-benzodioxol-5-ylamino)-pyridin-2-ylmethylidene]cyclohexa-2,5-dien-1-one 3-(4-butylphenyl)-2,6-difluorophenol 2-[(5R,10bR)-7-methoxy-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-methoxyphenol 4-[3-(azidooxymethyl)-5-fluorophenoxy]-2,6-dichloropyridine 1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]ethanone N-(3,4-dimethoxyphenyl)-2-[7-(4-methylsulfanylphenyl)-6-oxo-2-thia-5,7,11-triazatricyclo[6.3.1.04,12]dodeca-1(11),3,8(12),9-tetraen-3-yl]acetamide (3S,4R)-4-[1-[[5-fluoro-6-[(2R)-2-methylmorpholine-4-carbonyl]pyridin-2-yl]amino]ethyl]-3-methoxypiperidine-1-carboxylic acid N'-(1,2-oxazol-3-ylmethoxy)quinoline-5-carboximidamide 1-[2,6-dichloro-4-(4-fluoropyrazol-1-yl)phenyl]ethanethiol 3-[4,5,6-trichloro-2-ethoxycarbonyl-1-(2H-tetrazol-5-yl)indol-3-yl]propanoic acid 4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxy-1H-triazole-5-carboxylic acid 2-[5-(aminomethyl)-4-(2-fluorophenyl)-1,3-thiazol-2-yl]-4-(trifluoromethoxy)phenol;ethane N-[2,6-difluoro-4-(2H-pyridine-1-carboximidoyl)phenyl]-3-methoxypropane-1-sulfonamide N-[4-hydroxy-2-[2-(5-methoxypyridin-3-yl)ethynyl]phenyl]propane-1-sulfonamide 2-[(Z)-1-aminoethylideneamino]-3-methylquinazolin-4-one;propane 2-[(1S)-2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclopentyl]acetic acid 6-(2-azidothiophen-3-yl)naphthalen-2-ol N-(2,2-difluoroethyl)-2-[4-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-yl)piperazin-1-yl]acetamide 1-[(2S,3R)-4-amino-3-cyclohexylbutan-2-yl]-N-(pyrazin-2-ylmethyl)triazole-4-carboxamide;hydrochloride 2-[1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]-7,8-dihydro-5H-pyrano[4,3-b]pyridine-3-carbonitrile N-[4-(5,6-dihydro-1H-indazol-3-yl)phenyl]cyclohexanecarboxamide N-[[(2S,4R)-1-ethyl-6-oxo-2-pyridin-3-ylpiperidin-4-yl]methyl]benzamide [4-(benzylcarbamoyl)phenyl]methoxyazanide [7-(3,5-dimethylbenzoyl)-3-morpholin-4-ylquinoxalin-2-yl]-phenylmethanone 2-chloro-N',4-dimethylpyridine-3-carboximidamide 2-[5-(cyclohexylmethylamino)pyridin-3-yl]-7-(4,6-difluoro-1H-indazol-5-yl)pyrido[1,2-a]pyrimidin-4-one 7-(dimethylamino)-1-ethoxy-5,6-difluoro-8-hydroxy-4-oxoquinoline-3-carboxylic acid 5-aminosulfanyl-4-hydroxynaphthalene-1,3-disulfonic acid;ethane N-[2-amino-5-(4-chlorophenyl)-3-fluorophenyl]-2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carboxamide [7-(cyclopentylamino)imidazo[1,2-a]pyridin-2-yl]-(4-methylpiperidin-1-yl)methanone N-(4-chlorobutyl)-N-[2-hydroxy-1-[6-(trifluoromethoxy)-1,3-benzothiazol-2-yl]ethyl]-2-methylpropanamide 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-N-[(4R)-8-methoxy-2,2-dimethyl-6-pyridin-4-yl-3,4-dihydrochromen-4-yl]acetamide 2-[1-(6-phenylpyridin-3-yl)ethenoxymethyl]benzonitrile [4-azido-1-(3,5-dichlorobenzoyl)piperidin-2-yl]urea N-[(2S)-1,1,1-trifluorobutan-2-yl]-4-(trifluoromethyl)benzamide 4-methyl-2-[N-(4-nitrobenzoyl)anilino]pentanoic acid [(3S,4R)-1-ethyl-3-fluoropiperidin-4-yl]-(7H-pyrrolo[2,3-d]pyrimidin-5-yl)methanone 5-ethyl-7-methoxypyrrolo[2,1-f][1,2,4]triazin-4-amine 5-[4-(2,6-difluorophenoxy)phenyl]-1H-pyrazol-3-amine 3-(furan-2-yl)-2-[4-(1H-indole-7-carbonylamino)phenyl]propanoic acid 5-[(3,4-dimethylphenyl)sulfonylamino]-2-[2-ethyl-4-(piperidine-1-carbonyl)anilino]benzoic acid;2,2,2-trifluoroacetic acid 2-[1,3-dimethyl-2-(4-methylphenyl)-5-(trifluoromethoxy)indol-6-yl]acetic acid N-(4-azidophenyl)-1H-indazol-5-amine N-[1-(2-phenylethyl)pyrazol-3-yl]-6,7-dihydro-4H-furo[3,2-c]pyran-4-carboxamide N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-N,5-diethylpyrimidin-2-amine 3-cyclohexyl-5,7,8,10-tetrazatricyclo[7.4.0.02,6]trideca-1(9),2,4,6-tetraene 3-[(2R)-1-(4,5-dimethylpyrazol-1-yl)propan-2-yl]-6-(1-methylimidazole-2-carbonyl)-1H-pyridin-2-one 2,3-dimethyl-N-[1-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)propan-2-yl]benzamide N-[(1R,2R)-4-(imidazol-1-ylmethyl)-2-propoxycyclohexyl]quinoline-3-carboxamide 6-[3,5-bis(trifluoromethyl)phenyl]-4,6-dioxocyclohexa-1,5-diene-1-carbonitrile 6-(4-methylcyclohexyl)oxypyridine-3-carboxylic acid N-[(1S)-1-[3-[5-chloro-2-[difluoro(iodo)methyl]phenyl]-4-fluorophenyl]ethyl]-1,2-oxazole-3-carboxamide 3-chloro-5,7-difluoro-N-(6-methyl-2-oxo-4-phenyl-1H-pyridin-3-yl)-1-benzothiophene-2-carboxamide N-[1,1-dihydroxy-3-(hydroxyamino)propan-2-yl]-4-methoxybenzenesulfonamide 2-(4-propan-2-ylsulfanylphenyl)butanenitrile N-[2,3-bis(difluoromethyl)phenyl]benzamide 2-[2-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-N,3-diethyl-7,8-dihydro-6H-cyclopenta[g]quinazolin-9-amine [1-(4-tert-butylphenyl)cyclopropanecarbonyl]carbamic acid 4-chloro-1,5-dimethyl-3-nitrosopyrazole;N,N-diethylethanamine 2-[[3-chloro-4-fluoro-5-(trifluoromethyl)phenyl]carbamoylamino]-N-cyclopentylacetamide 1-[3,5-bis(trifluoromethyl)phenyl]-2-pyridin-4-ylethanone 4-chloro-6,7,8,9-tetrahydronaphtho[2,1-g][1]benzofuran-10-one 2-chloro-3-(dimethoxyamino)naphthalene-1,4-dione 4-methylsulfanylspiro[3H-benzo[h]quinazoline-6,1'-cyclobutane] 1-[4-(4,4-dimethylpiperidine-1-carbonyl)phenyl]imidazolidin-2-one 1-[4-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidine-2-carboxamide 5-(4-azidopiperazin-1-yl)-2-[3-methoxy-4-(4-morpholin-4-ylpiperidine-1-carbonyl)phenyl]pyrimidin-4-amine 3-(2,4-diaminophenyl)propanoic acid 1-[2-(6,7-dimethoxyquinazolin-4-yl)ethynyl]cyclobutan-1-amine 3-hydroxy-N-[1-(2H-isoindol-1-yl)piperidin-4-yl]-N',N',2-trimethylbutanediamide 2-(2,6-difluorophenyl)-4H-[1,3]thiazolo[5,4-c]pyrazole N-(1-cyclopentylpyrazol-4-yl)-3,3a,5,6,7,7a-hexahydro-2H-pyrrolo[3,2-b]pyridine-1-carboxamide [2-(4-hydroxyphenyl)azetidin-1-yl]-[3-(methoxymethyl)furan-2-carbonyl]iodanuidylmethanethione (2S)-2-[[(E,3S)-6-cyclohexyloxy-5-phenylmethoxy-1-sulfanylidenepent-4-en-3-yl]carbamoylamino]propanoic acid 2-amino-4-(2,3-difluorophenyl)-6-methylbenzene-1,3-dicarbonitrile [5-(2,4-dimethylpiperazine-1-carbonyl)-2-nitrophenyl]thiourea 1-amino-5-(cyclohexylmethylamino)-6-nitronaphthalene-2-sulfonic acid 6-azidooxy-4,5-dimethylnaphthalene-2-carboxylic acid 2-(3,5-dimethylphenyl)-1,4-bis[4-(3-methoxypropoxy)phenyl]piperazine N-[4,5-difluoro-2-(hydroxymethyl)phenyl]-1,3-oxazole-4-carboxamide 2-azido-4,6-dimethoxy-3,5-bis(methylsulfanyl)benzonitrile 4-(5-ethylpyrimidin-2-yl)oxypiperidine-1,3-dicarboxylic acid [2-[(4S)-7,8-dihydro-6H-furo[3,2-e]indol-2-yl]phenyl]phosphane 2-amino-6-[1-[4-(3,5-difluorophenoxy)cyclohexyl]pyrazol-4-yl]-7H-pyrrolo[3,4-b]pyridin-5-one 3-(7-chloro-5-methylpyrrolo[2,1-f][1,2,4]triazin-2-yl)benzenethiol 2-(methylideneamino)-N-[1-[4-(methylsulfanylmethoxy)phenyl]butyl]propane-2-sulfinamide ethane;[4-[(1E)-4-methoxy-6,7-dimethylcycloocta-1,3,5,7-tetraen-1-yl]-3,6-dihydro-2H-pyridin-1-yl]-pyridin-4-ylmethanone 2-[4-[[3-(1H-imidazol-5-yl)phenyl]methoxy]-3,6-dihydro-2H-pyridin-1-yl]ethanamine 3-[2,5-diamino-4-(cyclohexylmethoxy)phenyl]propanenitrile;hydrochloride 2-amino-N'-(4-fluorophenyl)-1,3-thiazole-5-carboximidamide N-[2-(5,7-dichloro-2,4-dioxoquinazolin-1-yl)ethyl]benzenesulfonamide 2-(3-aminophenyl)-1,6,7,8-tetrahydroisoquinoline-5-carbonitrile 1-[2,4-difluoro-6-(triazol-1-yl)phenyl]-3-(5-methylpyrazin-2-yl)-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine 5-(3,4-difluorophenyl)-1H-indazole (3S,4S)-4-(5-bromothiophene-2-carbonyl)oxypiperidine-1,3-dicarboxylate 2-(3-fluoropyridin-4-yl)-N,3,3-trimethoxypropanamide 3,4-dimethoxy-N-[5-(2,4,6-trihydroxyphenyl)-1H-pyrazol-3-yl]benzamide N'-hydroxy-3-(4-phenylmethoxypiperidin-1-yl)pyrazine-2-carboximidamide 5-butoxycarbonylbenzoic acid 5-azidooxy-1,2,3-trimethoxy-4-methylbenzene (6R,9S)-6-methyl-2-methylsulfanyl-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 2-(7-benzyl-3,4-dihydro-1H-isoquinoline-2-carbonyl)quinoline-8-carbonitrile 7-bromo-2,4-diphenyl-1,10-phenanthroline 2-[4-(trifluoromethyl)phenyl]-3H-pyrido[2,3-d]pyrimidin-4-one 1-(1,3-benzodioxol-5-yl)-5-N-cyclohexylpyrazole-4,5-diamine 2-[1,4-dimethyl-3-(4-propan-2-yloxybutyl)-5H-pyrazolo[4,3-c]quinolin-7-yl]benzenesulfonamide 5-(3,4-difluorophenyl)sulfanyl-2,2-difluoro-1,3-benzodioxole 2-[4-ethoxycarbonyl-N-[(3-fluorophenyl)methyl]anilino]propanoic acid N-benzyl-N-butylethanesulfonamide 2-azido-N,N',3-trimethylbenzenecarboximidamide (3Z)-7,8-dimethyl-2-oxo-3-[(4-pyridin-3-ylpyrimidin-5-yl)methylidene]chromene-6-carbonitrile (1-aminoisoquinolin-5-yl)methylazanide 2-[(6-methyl-4-methylidenethieno[2,3-d]pyrimidine-3-carbonyl)amino]propanoic acid (Z)-1,2-dicyanoethene-1,2-dithiolate;iron(2+);4-[(2E,3Z,5Z)-4-methylhepta-2,5-dien-6-ynyl]pyridine 6-(2,4,5-trihydroxyphenyl)naphthalene-1-carboxylic acid 2-cyclohexa-1,5-dien-1-yl-N'-phenylethanimidamide 4-[2-(3,6-diphenylcarbazol-9-yl)pyrimidin-5-yl]pyridine-3,5-dicarbonitrile 3-[4,5-diamino-1-[2-(2-chlorophenyl)ethyl]imidazol-2-yl]propanal 2-[4-amino-3-chloro-5-fluoro-6-(2-methoxyethylsulfanyl)pyridin-2-yl]propanedinitrile 2-cyclohexyloxy-4,6-bis(5-methylhexoxy)benzaldehyde 2-[(3S)-7-nitro-3,4-dihydro-1H-isoquinoline-2-carbonyl]chromen-4-one 3,4-difluoro-5-iodobenzoic acid N-(cyclopropanecarbonyl)-N-ethyl-6-(trifluoromethoxy)pyridine-3-carboxamide (2S)-N,3-bis[2-(methyliminomethyl)phenyl]butan-2-amine 2-[2-(1-aminoethenyl)phenyl]-N,4-dimethoxyaniline N-[2-amino-1-[5-(3,4-dimethoxyphenyl)-1H-pyrrol-2-yl]ethenyl]pyridin-4-amine 2-chloro-N-(cyclopropylmethoxy)-6-fluoroaniline N-azido-2,5-dimethylthiophene-3-sulfonamide 4-[6-methoxy-5-(1,3-oxazol-2-yl)pyridin-3-yl]pyridine-3-thiol 4-hydroxy-3-[(6R)-7-methyl-8,9-dihydropyrimido[5,4-b]indolizin-6-yl]benzaldehyde (2S)-2-N-methyl-1-N,3-N-bis[(4-methylphenyl)methyl]pentane-1,2,3-triamine [1-[3,5-bis(trifluoromethyl)phenyl]-2H-pyridine-4-carboximidoyl]carbamic acid 2-[6-(4,5-dihydro-1H-imidazol-2-yl)indol-1-yl]acetic acid N-[(2-methoxyphenyl)carbamoyl]-1,3-benzoxazole-6-carboxamide N-(3,5-dichloropyridin-4-yl)-1,2-thiazol-5-amine N-[[4-[(3S)-2,5-dioxopyrrolidin-3-yl]oxyphenyl]methylidene]ethanesulfonamide 7-[3-(3,4-dihydro-2H-chromen-6-yl)-1,2,4-oxadiazol-5-yl]-5-pyridin-4-yloxypentanoic acid 1-azido-4-(4-fluorophenyl)sulfonylpiperazine (2-fluoropyridin-4-yl)-[(3S,4R)-3-methoxy-4-[(6-methylpyridazin-3-yl)amino]pyrrolidin-1-yl]methanone 6-chloro-4-(2,6-dichlorophenyl)-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 3-azidooxy-1,2,5-trimethylbenzene 4-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]isoindole-1,3-dione 3-[2-(6,7-dimethoxyquinolin-4-yl)ethynyl]-5-fluoroaniline;N'-methyl-N-propan-2-ylidenepyridine-3-carboximidamide 3-(4,5-dihydro-1H-imidazol-2-yl)-1-phenyl-N-[6-(trifluoromethyl)pyridin-3-yl]pyrazole-4-carboxamide 2-(4,7-dichloroindol-1-yl)ethanamine 1-ethyl-2,3-difluoro-4-[4-(4-methoxyphenyl)phenyl]benzene 2,6-dimethoxy-4-[5-(1H-pyrazol-5-yl)benzimidazol-2-ylidene]piperidine;hydrochloride 3-amino-5,8-dihydroxynaphthalene-1,2-disulfonic acid N-[3-[4-cyano-5-(1,2-oxazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]phenyl]prop-2-enamide 2-[(4-fluorophenyl)methylsulfanyl]-6,7-dihydro-5H-cyclopenta[d]pyrimidine 6-[(3aR,7aS)-1-(4-fluorophenyl)-2,2-dimethyl-3,3a,5,6,7,7a-hexahydropyrrolo[3,2-b]pyridin-4-yl]pyridine-3-carbonitrile (3S,4R)-3-(hydroxymethyl)-4-[[1-[4-isocyano-3-(trifluoromethyl)phenyl]piperidin-4-yl]amino]-5-(2-methoxyethylsulfonyl)-N'-methylpyrrolidine-1-carboximidamide (5S)-3-(4-fluorophenyl)sulfonyl-2,7-dimethyl-1-(trideuteriomethyl)-2H-pyrido[1,2-a]pyrazine 3-ethyl-2,5-difluoro-6-methylsulfanylbenzonitrile 2-amino-5-[4-(diethylamino)phenyl]-3,6-bis[4-fluoro-3-(trifluoromethyl)anilino]pyrimidin-4-one 4-[5-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-2-ethoxy-6-methylpyrimidin-4-yl]morpholine 1-azidooxy-6,7-diethoxyisoquinoline 6-(2,4-difluorophenyl)-3-fluoro-N-[5-methyl-1-[1-(trifluoromethoxy)ethyl]pyrazol-3-yl]pyridine-2-carboxamide 5-hydroxyimino-4,4-diphenyl-2H-thiophen-3-one 5-[3-[2,6-difluoro-4-(trifluoromethoxy)phenoxy]-5-oxopyrazolidin-1-yl]-2-fluorobenzoic acid 1-[(2-chloro-5-propan-2-yloxyphenyl)methyl]piperidine 1-azido-4-(3,4-dimethoxyphenyl)piperidine N-[(1S)-1-(5,6-dichlorocyclohexa-1,3-dien-1-yl)ethyl]-6-[4-ethoxy-7-(pyridin-4-ylmethylamino)imidazo[1,2-a]pyrimidin-2-yl]pyrimidin-4-amine N-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethyl)pyrazol-3-yl]butanamide;hydrochloride 5-[3,4-di(propan-2-yl)phenoxy]pentanenitrile (4E)-4-[[6-bromo-1-ethyl-3,8-bis(trifluoromethoxy)naphthalen-2-ylidene]hydrazinylidene]pentanoic acid 5-bromo-6-methyl-N-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]naphthalene-1-carboxamide 4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethylamino]-5-methoxy-1H-pyrimidin-6-one N'-[(1S,5R)-2,3,4,5-tetrahydro-1H-diazepino[6,7-b]indol-1-yl]propane-1,3-diamine;hydrobromide 2-(1,3-benzothiazol-6-yl)-N-[(2R)-1-hydroxy-5-(methanesulfonamido)pentan-2-yl]acetamide (E)-3-[5-bromo-2-[(3-fluorophenyl)methoxy]-4-methoxyphenyl]-2-sulfanylprop-2-enoic acid 2-[2-hydroxyethyl(3-morpholin-4-ylpropyl)amino]benzenesulfonic acid 4-[[4-(azetidin-1-yl)phenyl]methyl]morpholine N-[2-chloro-4-(trifluoromethyl)phenyl]-5-methoxy-8-piperidin-1-ylquinoline-3-carboxamide N-[(4R)-1-butan-2-ylpiperidin-4-yl]-6-(3-methoxyphenyl)imidazo[1,2-a]pyrazin-8-amine (4-benzoylphenyl)-[4-[2,6-di(propan-2-yloxy)phenyl]phenyl]methanone (E)-4-chloropent-3-enoic acid;1,2-difluorobenzene;[3-fluoro-5-[5-(methylamino)pyridin-2-yl]phenyl]methanol 3-[1-(cyclopropylmethylamino)-2,2,4-trifluoroethyl]benzenesulfonamide N-cyclohexyl-2,6-dioxo-3,4-dihydro-1H-1,3,5-triazine-5-carboxamide;ethane 7-(3-methoxyphenyl)imidazo[1,2-a]pyridine 2-chloro-4,5-dimethoxybenzenethiol 3-bromo-N'-[(E)-(3,4-dihydroxyphenyl)methylideneamino]-6-methylimidazo[1,2-a]pyridine-8-carboximidamide 1,2-diamino-4-(3-chloro-5-fluoro-2-hydroxyphenyl)-6-oxopyridine-3,5-dicarbonitrile 1-(6,7-dihydro-5H-[1,3]thiazolo[5,4-d]pyrimidin-2-yl)-N'-hydroxyimidazole-2-carboximidamide 4-N-[2-fluoro-5-(1H-pyrrolo[3,2-b]pyridine-6-carbonyl)phenyl]-5-methylfuran-2,4-dicarboxamide [1-azidooxy-4-(4-methylsulfanylphenyl)-3,5-dihydro-2H-1,4-benzodiazepin-8-yl]methanol N-(1,3-benzothiazol-5-yl)-2-methoxy-4-[7-(4-methylpiperazin-1-yl)quinazolin-4-yl]benzamide 2-[4-(3,5-dichlorophenyl)sulfanyl-N-methylanilino]ethanesulfonic acid 7-chloro-2-[2-(methylamino)-1,3-thiazol-5-yl]-3H-quinazolin-4-one;5-fluoro-2-piperidin-4-yl-3H-quinazolin-4-one 3-[[4-(2,5-dimethyl-1,3-thiazol-4-yl)phenyl]iminomethyl]-6-methoxy-1H-indol-2-ol 3-methyl-6,7,8,9-tetrahydropyrazino[1,2-a]pyrimidine-2,4-dione 4-[2-(3,5-dimethylpyrazol-1-yl)-6-propan-2-ylpyridin-3-yl]oxybenzoic acid 2-[4-(5-methoxycyclohepta-1,3,6-trien-1-yl)phenyl]acetonitrile [4-(6-chloropyridine-3-carbonyl)piperazin-1-yl]-phenylmethanone 1-[2,6-di(propan-2-yl)phenyl]-3-[N'-methyl-N-(3-methylpyridin-4-yl)carbamimidoyl]urea 2-[3,5-difluoro-4-(5-methylsulfanylpentyl)phenyl]pentanenitrile 4-[[5-[3-chloro-6-(2,2-difluoroethoxy)pyridin-2-yl]-1-methylimidazole-2-carbonyl]amino]-2-phenylbenzamide (4S,5R)-2,2-dimethyl-5-phenyl-1,3-dioxane-4-carboxylic acid 2-(6-tert-butylpyridin-3-yl)acetate [5-[(4-cyanophenyl)sulfonylamino]-6,7,8,9-tetrahydro-5H-carbazole-2-carbonyl]azanium 1-(4-chlorophenyl)sulfonyl-3,6-dimethylindole 6-(furan-3-ylmethyl)-2-thiophen-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-[1,6-dihydroxy-4-(trifluoromethyl)naphthalene-2-carbonyl]oxy-3-oxopropanoic acid 6-chloro-8-(4,5,7-trifluoro-1H-indol-2-yl)imidazo[1,2-b]pyridazine 3-[(6-butyl-2,3-dimethoxyphenyl)methylidene]azetidine 1-(2,4-dimethylphenyl)-4,5-bis[4-(N-propan-2-ylanilino)cyclohexa-2,4-dien-1-ylidene]pyrazole-3-carboxylic acid 2-azidosulfanyl-1,3,5-trifluorobenzene 2-amino-4-[1-(oxan-3-ylmethoxy)cyclobutyl]-6,7-dihydro-5H-pyrano[2,3-d]pyrimidine-8-carbonitrile 5-(2,3-dimethylbutyl)-4-(4-propanoylpiperazine-1-carbonyl)furan-2-carbonitrile (5-fluoro-2,3-dihydroindol-1-yl)-[5-(1H-pyrazol-4-yl)thiophen-3-yl]methanone 6-chloro-1,3-dimethylindole-2-carboxylic acid 4-[5-(9H-fluoren-9-ylmethoxycarbonylamino)pentanoyl-methylideneazaniumyl]butanoate 3-ethyl-8-fluoro-7-(4-pentylphenyl)naphthalene 4-amino-N,N'-diamino-6-methylpyrimidine-5-carboximidamide 2-(3-ethoxypyridin-4-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 3-[[(4S)-3,4-dihydro-2H-chromen-4-yl]methoxy]-5-(1H-pyrazol-4-yl)pyridine 2-[2-(1,3-diphenylpyrazol-4-yl)ethyl]-1H-benzimidazole 1-(2-ethoxy-4-fluorophenyl)-5,7-dihydrotriazolo[4,5-b]pyridin-6-one 3-[(E)-2-hydroxyethenyl]-5-methoxyquinoxaline-2,6-dicarbonitrile 1-[3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)piperidin-1-yl]-3-[4-(tetrazol-1-ylmethyl)phenyl]propan-1-one N-[2,6-dimethyl-4-(3-methylbutanoyl)phenyl]acetamide 2-[4,6-bis(trichloromethyl)pyrimidin-5-yl]oxyethanol 6-(3,4-dimethoxyphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 2-[1-(3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclopropyl]acetamide N-[3-[(5R)-3-amino-4-hydroxy-6,8-dimethyl-2H-pyrano[2,3-f]quinoline-9-carbonyl]phenyl]benzenesulfonamide 1-[(2S)-butan-2-yl]oxy-6,7-dimethoxynaphthalene;ethane 4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)-9-(1H-pyrrol-2-ylmethyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one 3-(5-methylpyridin-2-yl)-7H-purin-6-imine 1-(2,3-dihydropyridin-4-yl)-5-piperidin-3-ylindazole;dihydrochloride 4-fluoro-2-(1-methylpiperidine-3-carbonyl)-N-[5-(trifluoromethyl)pyrazin-2-yl]benzenesulfonamide (2S,4R)-4-amino-5-[4-(1H-indol-6-yloxy)phenyl]pentanoic acid 3-(4-methylphenyl)-2-oxo-N-phenylpyrrolidine-1-carboxamide N-(1H-benzimidazol-2-ylmethyl)-3-[4-(trifluoromethoxy)phenyl]aniline [7-[1-(4-fluorophenyl)ethyl]-2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl]methanol 1-[(E)-3-cyclopropylhex-2-enoxy]-4-[4-ethyl-3-(trifluoromethyl)phenyl]-2,5-difluorobenzene [2-(cyclopropylmethylamino)-5,6-dihydrobenzo[b][1]benzazepin-11-yl]methanol 2-[N-methylsulfonyl-4-(1,3,4-oxadiazol-2-yl)anilino]acetamide 4-[(2S)-1-(diethylamino)propan-2-yl]oxybenzoic acid 4-benzyl-1-methylpiperidine;3,3,5,5-tetramethylhexan-2-one 2-[4-azido-3-(pyridine-3-carbonyl)anilino]-1H-benzimidazole-5-carbonitrile 3-[(1R)-6-hydroxy-5,7-dimethoxy-2-methyl-4-oxochromen-8-yl]propanoic acid 2-(3,4-dihydroxyphenyl)-N-ethyl-2-hydroxyacetamide (2S)-2-[[4-cyclopropyl-5-(1H-indol-3-yl)-1,2,4-triazol-3-yl]sulfanyl]-N-methoxy-N-methyl-2-phenylacetamide 2-[[5-(2-aminoethyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-thieno[3,2-d]pyrimidin-4-one 4-ethyl-6-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]pyrimidine-2-carboxylic acid N-ethyl-2-hydroxy-N,3,4-trimethoxybenzamide (NE)-N-[(5Z,6Z)-4-fluoro-5-phenyl-1,3-diazocin-8-ylidene]hydroxylamine (3R,6'E)-1-[4-(4-methoxyphenyl)piperazin-1-yl]spiro[azepane-5,2'-3H-1H-benzofuran]-6'-ol 2-amino-4-(3,5-difluorophenyl)-6-ethoxy-4H-pyran-3,5-dicarbonitrile N-[(2S)-5-[(E)-[(6-aminopurin-9-yl)hydrazinylidene]methyl]-1-(4-nitrophenyl)sulfonylpiperidine-2-carbonyl]acetamide (6R)-3-[3-[(4-chlorophenyl)methoxy]phenyl]-8,8-diethyl-7,10-dihydro-2H-[1,2,4]triazino[5,6-c]quinazoline-1,5-dione N-(3,4-difluorophenyl)-2-(methylaminomethylideneamino)acetamide 4-[(2-methoxyphenyl)sulfanylamino]-5,6,7,8-tetrahydroquinoline-3-carboxamide 2-[5-(azetidin-1-yl)pyridin-3-yl]-N-azidoethanamine 3-[4-(3,4-dihydroxyphenyl)phenyl]prop-2-enoic acid N-[(Z)-(3-hydroxy-5-methoxyphenyl)methylideneamino]-1,2,3,4-tetrahydronaphthalene-1-carboxamide 1-[4-(6-methoxyquinolin-4-yl)cyclohexyl]-3-(2,2,2-trifluoroethanimidoyl)urea 2-[4-(3-chlorophenyl)-6-ethylpyrimidin-5-yl]oxy-1-[3,4-dimethyl-7-(1H-pyrrol-2-yl)pyrazolo[1,5-a]pyridin-5-yl]ethanone N-(8-aminooctyl)-4-[4-(1,2,4,5-tetrazin-3-yl)phenyl]piperazine-1-carboxamide (4E)-2-[(3,4-dimethoxyphenyl)methyl]-5-hydroxy-4-[(2Z)-penta-2,4-dienylidene]-1H-pyrimidin-6-one 3-amino-5,6,7,8-tetrahydronaphthalene-2-sulfonic acid 2-methyl-4-(6-piperidin-1-ylpyridin-3-yl)butan-2-amine N-(4-hydroxyphenyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole-6-carboxamide 2-[3,5-bis(trifluoromethyl)phenyl]cyclopropan-1-one 2-[2-chloro-4-(trifluoromethyl)phenyl]imino-5,6-diethoxy-N-phenylcyclohexa-1,3-dien-1-amine 2-[(3S)-1-(4,6-dimethylpyridine-3-carbonyl)piperidin-3-yl]oxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile [5-chloro-3-(methoxymethyl)pyrazol-1-yl]-(4-cyanophenyl)methanesulfonamide 4-(2,6-difluorophenyl)-3-methylsulfanylbenzoic acid 3-[6-(2,6-dichloro-4-methylphenoxy)hexoxy]benzenecarboximidamide 6-chloro-1,3-dimethylquinazoline-2,4-dione [2-[4-(1-methylazepan-3-yl)-1,2,5-oxadiazol-3-yl]thiophen-3-yl]-piperidin-1-ylmethanone 4-[3,5-dimethoxy-4-(trifluoromethyl)phenyl]sulfonyl-2-[(6R)-8-fluoro-1,4-oxazepan-6-yl]pyridine-3-carboxamide 2,3-diaminonaphthalene-1-carboxylic acid 4-[2,3-bis(ethenyl)-9H-fluoren-1-yl]benzenethiol 5-[2-(3,4-difluorophenyl)pyrrolidine-1-carbonyl]piperidin-2-one 1-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]imidazole N-[3-chloro-4-(5-methylpyridin-2-yl)oxyphenyl]-1H-indazole-5-carboxamide N-[3-(4-azidopiperazin-1-yl)phenyl]-2-[(Z)-2-methoxy-5-nitrohex-3-enoyl]-9,10-dihydroanthracene-1-carboxamide 4-(aminomethyl)-2-[1-[2,4-bis(trifluoromethyl)phenyl]ethyl]-5-methylphenol 1-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylamino)-4-[4-(3-ethoxyphenyl)piperazin-1-yl]butane-1,4-diol N-[2-(4-aminophenoxy)ethyl]-1,3-dimethoxypropan-2-amine N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxyiminoacetamide 3-chloro-N,5-dimethyl-4-(trifluoromethyl)benzamide;2,6-diaminopyridine-4-carbonitrile N-cyclobutyl-5-[3-(4,6-difluoro-1H-benzimidazol-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine 4-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N-[(3S)-1-hydroxypyrrolidin-3-ylidene]cyclohexane-1-carboxamide 4-(2,5-difluorophenyl)-3,6-dimethylheptane (2S)-2-[[3-bromo-1-(3,4-dimethylphenyl)propoxy]carbonylamino]pentanoic acid 2-[2,4-dinitro-N-(1,3-thiazol-5-yl)anilino]propanoic acid 4-(2,3-dimethylphenyl)-5,6-bis[2-(methylamino)ethyl]benzene-1,3-diol 4-(2-bromo-5-chloropyrimidin-4-yl)oxypiperidine-1-carboxylate N-[[3-amino-2,6-dimethyl-4-(4-methylpyridin-2-yl)phenyl]methyl]-1-ethylpyrazole-4-sulfonamide 3-[2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)phenyl]propanenitrile 2-[[2-(3-bromo-4-hydroxyphenyl)ethylamino]methyl]-8H-pyrano[3,2-g]quinolin-9-one ethane;1-[3-(2-methylphenyl)propoxy]azetidine 7-chloro-1,5,5a,6-tetrahydropyrido[2,3-f][1,4]benzoxazepine;hydrochloride N-[4-(2,6-dimethylanilino)-3-nitrophenyl]acetamide ethane;N-(2-fluoropropyl)formamide;methanamine;5,9,17-triphenylpentadeca-1,8-diene 6-(2,6-difluorophenyl)-2-[1-(3H-inden-4-yl)ethenyl]-5-methylpyrimidin-4-amine 2-bromo-N'-methoxy-6-(4-pyridin-3-ylsulfonylpiperazin-1-yl)pyrimidine-4-carboximidamide 1-[4-(trifluoromethyl)phenoxy]indole 2-[4-hydroxybutyl(pyridin-3-yl)amino]benzenesulfonic acid 5-[6-(2,3-dihydro-1H-inden-4-yl)pyridin-2-yl]pyrimidine (2R)-1-ethyl-N-[4-(2,2,3,3,5,5,6,7,8,8a-octahydroindolizin-5-yloxymethyl)phenyl]sulfonylpyrrolidine-2-carboxamide 2-ethoxy-3-[6-methyl-5-oxo-8-(trifluoromethyl)imidazo[1,2-a]pyrimidin-7-yl]benzonitrile 3-[4-azidooxy-1,6-bis(pyridin-2-ylmethyl)pyrazolo[3,4-d]pyrimidin-3-yl]benzoic acid [4-(3,5-dichloropyridin-2-yl)piperazin-1-yl]-phenylmethanone 2-[[4-(3,5-dichlorophenyl)piperazin-1-yl]sulfonylmethylideneamino]-N-hydroxy-4-phenylbutanamide 7-[(4-chlorophenyl)methyl]-8-hydroxy-3-propan-2-yl-1,3-diazaspiro[4.5]decane-2,4-dione 1-[3-(2,4-dihydroxyphenyl)propanoyl]piperidine-2-carboxylic acid (1E)-1-ethylidene-5,6-dihydroxyindene-2,3-dione N-[(2,3-dichlorophenyl)methyl]-6-oxo-1H-pyrimidine-4-carboxamide 2-methyl-3,4-bis(phenylmethoxy)-1H-indole N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-methoxy-N-prop-2-enylacetamide 5-(2,6-difluorophenyl)-4-methyliminoimidazolidin-2-one 2-[1-(2,3-dihydrothiophen-5-yl)propan-2-ylideneamino]-N-methyl-N'-phenylbenzenecarboximidamide 2-[(1-aminopiperidin-4-yl)methoxy]benzenethiol 3-(2,3,5,6-tetrafluorophenyl)benzamide 4-[3-amino-6-(2,5-dimethylphenyl)pyrazin-2-yl]benzenesulfonamide 3-azido-N-(2-chlorophenyl)-5,6-dimethyl-1H-pyrazolo[4,3-b]pyridine-7-carboxamide 3,5-bis(4-chlorophenyl)-2-[2-hydroxy-3-[methyl(2-morpholin-4-ylethyl)amino]propyl]cyclohexa-2,5-dien-1-one N-[(1R)-3-(4-chlorophenyl)-2-oxocyclopentyl]-7,8-dihydro-6H-thieno[3,2-c]azepine-5-carboxamide N-[4-(2,4-difluorophenoxy)-3-(7H-pyrrolo[2,3-d]pyrimidine-6-carbonylamino)phenyl]propanamide N-(4,5-dimethyl-2H-benzotriazol-7-yl)pyridine-3-carboxamide N-cyclopropyl-2-[4-(3,5-dimethoxyphenyl)pyrrolidin-3-yl]acetamide;N,N-dimethylformamide 5-methyl-4-(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)benzonitrile N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)isoquinoline-8-carboxamide N-[4-(2,6-dimethoxyphenyl)-5-(furan-2-yl)-1,2,4-triazol-3-yl]-7-fluoroquinoxaline-5-carboxamide 1-[3-(2,6-diphenylpyridin-4-yl)propyl]indole 2-(2,6-difluoro-4-methoxyphenyl)-5H-pyrimido[5,4-b]indole 3-[(2R)-2-cyclopropylbutyl]sulfanyl-4H-1,2,4-triazin-5-one 4-amino-6-[(3R,5S)-5-methylpiperazin-1-yl]pyrimidine-5-carbonitrile 3-azido-N-(4,5-dimethoxycyclohepta-1,3,6-trien-1-yl)pyridine-2-carboxamide 2-(4,4-dimethylpiperidine-1-carbonyl)benzoic acid (E)-1,2,3-triamino-4-[4-chloro-3-(5-oxopentylsulfanylmethyl)phenyl]-4-ethoxybut-2-en-1-one 1-(2,3-dichlorophenyl)sulfonyl-4-pyridin-3-ylpiperazine (2S,4R)-1-acetyl-N-[(3-chloro-6-methoxyquinolin-5-yl)methyl]-4-hydroxypyrrolidine-2-carboxamide 4-[(3S,4R)-1-tert-butyl-4-phenylpyrrolidine-3-carbonyl]-3,5-dihydro-2H-pyrido[3,4-f][1,4]oxazepine-9-carbonitrile 2-[[(5R,7S)-3-bromo-5-phenyl-6,7-dihydropyrazolo[1,5-a]pyrimidine-7-carbonyl]amino]acetic acid 4-cyclopropyl-3,5-dimethoxybenzoic acid 4-(1H-indazol-5-yl)aniline 1-(2,6-dioxopiperidine-3-carbonyl)indole-2,5-dicarboxylic acid N-[1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-4-yl]pyrimidine-5-carboxamide 2-[(3R,4S)-1-[(5-ethylfuran-2-yl)methyl]-4-methoxypyrrolidin-3-yl]-7-pyridin-3-yl-3H-imidazo[5,1-f][1,2,4]triazin-4-one 3-butyl-2-[(4-nitrophenyl)methylsulfanyl]quinoline 3-(2,4-difluorophenyl)-5-(3-methyltriazol-4-yl)isoquinoline 3-[6-(2,4,6-trimethylphenyl)pyridin-2-yl]benzamide 4-[3,5-dichloro-2-(hydroxymethyl)phenyl]benzoic acid 2-[4-(3,5-dimethylphenyl)-3-ethylcyclohexa-1,3-dien-1-yl]oxyacetic acid 3-[4-[1-(5,5,6,7-tetramethyl-2-oxoheptanoyl)piperidin-4-yl]oxyphenyl]propanoic acid 2-[5-fluoro-2,3-dimethyl-4-(pyrrolidine-1-carbonyl)phenyl]butanoic acid 6-[4-(oxetan-3-ylmethoxy)phenyl]-5,7-dihydropyrrolo[3,4-b]pyridine 3-bromoimidazo[1,2-a]pyrimidine-5-carboxylic acid N-[4-(dimethylamino)butyl]-3,7-dihydroxy-4H-1,2,4-benzotriazin-8-amine;hydrobromide N-[2-hydroxy-5-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isochromene-6-sulfonamide 2-[[(3R,4S)-1-(8,9-dimethoxy-2-oxobenzo[g]chromene-4-carbonyl)-4-hydroxypiperidin-3-yl]amino]-6,7-dihydro-5H-cyclopenta[b]pyridine-3-carbonitrile 2-chloro-1-(4-fluorophenyl)-3-[(Z)-(5-methyl-1H-pyrazol-4-yl)methylideneamino]guanidine;hydroiodide 3-[2,5-bis(methylsulfonyl)phenyl]-4H-pyridine N-[2-(5,5-dimethyl-4H-1,2-oxazol-3-yl)-6-hydroxyphenyl]-2-sulfanylacetamide 6-(3-amino-5-methylpyrazol-1-yl)-2,3-dihydroisoindol-1-one [(5E)-5-[(3,4-dimethoxyphenyl)methylidene]-2,2,8-trimethyl-3,4,10b-tetrahydroindeno[1,2-b]indol-6-yl]-(5-hydroxycyclohexa-1,3-dien-1-yl)methanone 3-fluoro-5-(2-methylphenyl)sulfanylphenol (3S,5R)-1-(4-fluorophenyl)sulfonyl-5-[(2-methoxy-6-propan-2-ylpyrimidin-4-yl)amino]piperidine-3-carboxylic acid 2-azido-3-[(2,4,6-trimethoxyphenyl)methyl]imidazo[1,2-a]pyridine 2-[4-[3-methyl-1-(2-phenylethynyl)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carbonyl]anilino]ethanol 6-[(E)-2-(5-methoxythiophen-2-yl)ethenyl]-3,4,5,7-tetrahydro-1H-1,3-diazepin-2-one 1-(1,3-benzodioxol-5-yl)-2-[2-methoxy-4-nitro-3-(trifluoromethyl)phenyl]ethanone 2-[[(1S)-2,3-dihydro-1H-inden-1-yl]oxy]ethanamine 4-cyclopropyl-3,5-dimethoxybenzenesulfonamide N-[2,2-dimethyl-3-[4-(trifluoromethoxy)phenyl]cyclopropyl]acetamide 5-azido-4,7-diphenyl-1H-indole 5-bromo-2,3-difluoro-N'-hydroxybenzenecarboximidamide 2,2-dimethyl-3-(3-pyrrolidin-1-ylphenyl)pentanoic acid [1-[2-[(3-chlorophenyl)methylamino]ethylcarbamoylamino]-3-iminoprop-1-enoxy]boronic acid (E)-3-[7,9-diethoxy-3-(4-ethylphenyl)benzo[f]chromen-2-ylidene]prop-1-en-1-olate N'-[1-benzyl-3-ethenyl-5-[2-fluoro-6-(trifluoromethoxy)phenyl]-4-hydroxy-2,6-dioxopyrimidin-5-yl]methanimidamide 3-[1-(3-hydroxypropyl)-7,8-dimethoxy-4-oxoquinoline-2-carbonyl]pyrrolidine-1-carboxylic acid N-(2,5-dimethylphenyl)sulfonyl-6-fluoropyridine-3-carboxamide 1-(3,4-dichlorophenyl)sulfonyl-N'-hydroxyimidazole-2-carboximidamide 2-azidooxy-6,8-dimethyl-7H-imidazo[1,2-a]pyridine 2-[5,6-difluoro-3-oxo-8-(triazol-1-yl)xanthen-9-yl]propanoic acid [4-(5,6-dihydro-1H-benzimidazol-2-yl)cyclohexylidene]methanamine 2-[1,3-bis(4-methylphenyl)indol-5-yl]oxyacetic acid;ethane 1-[3,5-dimethoxy-4-[2-(2-oxoimidazolidin-1-yl)ethoxy]phenyl]-N'-pyridin-4-ylethane-1,2-diamine 2-[(2Z)-4-oxo-2-[(Z)-[3,5,6-trifluoro-9-(2-hydroxyethyl)carbazol-1-yl]methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid [4-(4-cyclohexa-1,5-dien-1-ylphenyl)sulfanylpiperazin-1-yl]-[3-(trifluoromethoxy)phenyl]methanone 5-[3-[7-(4,6-dimethylpyrimidin-2-yl)imidazo[1,2-a]pyridin-3-yl]-8-fluoronaphthalen-2-yl]isoquinoline 1-(4-chlorophenyl)-N-[2,4-difluoro-3-[5-(furan-2-yl)-6-oxo-1H-pyridazine-3-carbonyl]phenyl]cyclopropane-1-carboxamide [5-(5,8-difluoroquinolin-3-yl)-4-methoxypyridin-2-yl]methanol 1-(2,6-dichlorophenyl)-3,5-dimethylpyrazole;N-[4-(dipropylamino)butyl]-4-formamidopentanamide N-(2,5-dichloropyrimidin-4-yl)-N'-ethoxybutanehydrazide 4-ethenyl-1,7-difluoro-2-phenylmethoxynaphthalene (5Z)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[[1,2,5]oxadiazolo[3,4-b]pyrazin-6-yl]imino]-3-[1-(4-ethoxyphenyl)ethylidene]-1,3-thiazolidin-4-one 2-(7-chloro-1H-indazol-5-yl)pyridine-3,4-diamine 3-(2,4-difluorophenyl)-5-[7-methoxy-8-(trifluoromethyl)imidazo[1,2-a]pyridine-6-carbonyl]benzoic acid N-(6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl)-3-pyridin-4-ylazetidine-1-carboxamide 3-(4-benzylsulfonylpiperazin-1-yl)cyclopentane-1,2-dione 4-(2,2-dihydroxypropoxymethyl)-8-ethyl-1,7-naphthyridine-2,3-dione 2-[4-(2,6-dichloro-4-methylphenoxy)phenyl]acetic acid N-ethyl-2,3-dimethoxybenzenesulfonamide [5-fluoro-1-(4-propan-2-ylsulfonylphenyl)indazol-6-yl]methanol N-[2,3-difluoro-4-(3-methylbutanoylamino)phenyl]-3-hydroxy-5-methoxypyridine-2-carboxamide N-[1-(8-oxo-7H-imidazo[2,1-c][1,4]oxazin-3-yl)ethyl]pyridine-3-carboxamide 3-(2,6-dimethylphenyl)imino-6-methoxy-1H-indol-2-one ethane;(5Z)-3-(4-fluorophenyl)-5-[[2,4,6-trimethyl-1-[(4-nitrophenyl)methoxy]indol-7-yl]methylidene]oxolane 2-[(2S)-4,6-dioxospiro[1,3-dihydroindene-2,5'-imidazolidine]-2'-yl]ethanesulfonic acid 4-(4-azidophenyl)-2-propan-2-yl-1,3-oxazole N-[(2S)-4,4-difluoropyrrolidin-2-yl]sulfonylbenzamide 3-[2-(4-chlorophenyl)-5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-ium-3-ylidene]propanal 5-(trifluoromethyl)benzene-1,3,4-triol;4H-pyrido[2,3-e][1,2,5]oxadiazepin-7-amine 1-benzyl-2-(3,4-dichlorophenyl)pyrazin-1-ium;tetrakis[(2,3,4,5,6-pentafluorophenyl)methoxy]boranuide 3-amino-5-chloro-2-methyl-N-[1-(6-oxo-1H-pyrimidin-4-yl)piperidin-4-yl]benzamide 5-bromo-2-(1H-indole-6-carbonyl)pyridine-3-carboxylic acid 5-[4-[[(3R)-1-azabicyclo[2.2.2]octan-3-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-(trifluoromethoxy)pyridine-2-carbonitrile 3-cyclopentyl-1-(2,4-dichlorophenyl)propan-1-ol 4-(dimethylamino)-N-[4-[[2-oxo-1-[5-(1H-pyrazol-4-ylamino)pyridin-3-yl]pyrrolidin-3-ylidene]amino]phenyl]benzamide (2R,5S)-4,7-dioxa-13-azatetracyclo[8.6.0.03,12.011,15]hexadeca-1(10),3,11,13-triene 6-(3-aminocyclobutyl)-2-cyclohexyl-N,N-dimethylpyrimidin-4-amine;dihydrochloride 2-chloro-4,5-difluoro-N'-methylbenzohydrazide 6-[(5-chloro-2-ethoxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (3R,4S)-3-amino-1-[(2-methyl-6-phenylpyrimidin-4-yl)methyl]piperidin-4-ol;dihydrochloride 6-methyl-1,3-diphenylpyrrolo[2,3-c]pyridine (E)-N-[4-chloro-3-(trifluoromethyl)phenyl]-3-hydroxy-2-[3-(hydroxymethyl)pyridin-1-ium-1-yl]-3-thiophen-2-ylprop-2-enethioamide N-[(2R,3S)-4,4-difluoro-1-(1H-imidazole-5-carbonylamino)-3-phenylbutan-2-yl]pyrazine-2-carboxamide (2R)-2-amino-4,4-dimethyl-6-phenylhexanoic acid 5-(4,6-difluorocyclohexa-2,4-dien-1-yl)-3-[4-methoxy-4-(pyrrolidine-1-carbonyl)piperidine-1-carboximidoyl]thiophene-2-carboxylic acid 4-bromo-2-[(E)-1H-indol-3-ylmethylideneamino]oxy-6-(morpholine-4-carbonyl)pyridazin-3-one N-[5-[3-(4,4-dimethylcyclohexen-1-yl)-5-propan-2-ylphenyl]pyrazin-2-yl]acetamide 3-benzylsulfanyl-5-(4,5-dimethoxy-2,6-dimethylcyclohexa-1,3-dien-1-yl)oxypyrazine-2-carbonitrile 1-[(2Z)-2-(aminomethylidene)butyl]-7-fluoroquinoxalin-4-one;ethane 3,9-dimethyl-2-(2-phenylpyrimidin-5-yl)-6H-furo[2,3-h]isoquinolin-8-one 1-(cyclopropylmethyl)-2-phenylpiperazine N-[3-(dimethylamino)cyclobutyl]benzamide 1-benzylsulfanyl-3-methoxybenzene;6,8-dibromo-2-(trifluoromethyl)-4H-imidazo[1,5-a]quinazolin-5-one 1-[4-(5-chloro-2,3-dimethoxyphenyl)piperidin-1-yl]propane-1-thione 6-azidooxy-3-(1H-benzimidazol-2-yl)quinoline (1R,3S)-3-[7-chloro-2-hydroxy-6-methyl-4-(trifluoromethoxy)benzoyl]oxycyclohexane-1-carboxylic acid 1-[5-fluoro-2,4-dimethoxy-3-(trifluoromethyl)phenyl]ethanone 3-methoxycarbonyl-2,4-diphenylcyclohexa-1,5-diene-1-carboxylic acid 1-[4-[(2S,3R)-3-methylmorpholin-2-yl]phenyl]ethanamine 5-[(3,5-dichlorophenyl)methylsulfanyl]-1-[2-hydroxy-3-(4,4,4-trifluorobutanoylamino)propyl]indole-3-carboxamide 3-fluoro-4,5-diiodobenzoic acid N-(6,7-dihydro-5H-cyclopenta[b]pyridin-2-ylmethylidene)-3-[4-(trifluoromethoxy)phenoxy]azetidine-1-carboxamide 3-cyclobutyl-2,5-dihydropyrrole;(4R)-7'-fluoro-1',6-dimethylspiro[1H-indole-3,3'-piperidine]-2-one N-[2-(1H-indol-3-yl)ethyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine;dihydrochloride 3-amino-N-(1-azidooxy-2,2,2-trifluoroethyl)benzenesulfonamide 2-azidooxy-4-propan-2-ylsulfonylaniline 5-(5-fluoropyridin-3-yl)-6,7-dimethoxyisoquinoline 2-cyclopropyl-4-[6-(methoxymethyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-yl]-1H-pyrimidin-6-one 2-(4-fluorophenyl)sulfinyl-3,3a,5,6,7,8-hexahydroquinazolin-4-one [2-(2,4-dihydroxyphenyl)cyclopropyl]-morpholin-4-ylmethanone (Z)-2,3-diamino-N'-[5-(4-fluorophenyl)-1,3-thiazol-2-yl]but-2-enimidamide N-azido-2,3,4,5,6-pentafluoroaniline 3-azido-7,8-dihydro-6H-furo[3,2-e]indole 4-[3,5-dichloro-2-(2,6-difluorophenyl)-1H-triazol-4-yl]aniline 3-amino-2,6-dichloro-N'-[5-methoxy-1-(4-pyridin-4-ylpiperazin-1-yl)sulfonylisoquinolin-8-yl]benzenecarboximidamide N-[4-(3,5-dichlorophenyl)sulfanylcyclohexa-2,4-dien-1-yl]acetamide (2Z)-1,3-dimethyl-4-pyridin-4-ylsulfanylpenta-2,4-dien-2-ol 4-(2,3-dichlorophenyl)butanal 3-[2,6-dichloro-4-nitro-N-(4-nitrobenzoyl)anilino]butanoic acid N-butyl-2,4-dichloro-N-(5-nitro-1,3-thiazol-2-yl)pyrimidine-5-sulfonamide 2,2,4-trimethyl-3-oxobutanoate 2-[4-[(2,3-dimethyl-1H-indol-6-yl)amino]quinazolin-7-yl]oxyethanol N-(2,4-dimethoxyphenyl)-2-(4-ethylpiperidin-1-yl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-[(5S,7R)-3,7-dimethyl-5-thiophen-2-yl-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazol-2-yl]benzenesulfonamide 2-[3,5-bis(trifluoromethyl)phenyl]sulfanyl-N'-[2-(4-bromo-3-hydroxyphenyl)ethylamino]-N-prop-2-enoyl-1H-benzimidazole-5-carbohydrazide 4-[1-[4-(2,5-dimethylphenyl)phenyl]benzimidazol-5-yl]butanamide;ethane 2-[3-[3-(8-chloroquinolin-6-yl)oxypyrrolidine-1-carbonyl]phenyl]propanamide (E)-2-[[3,5-bis(trifluoromethyl)phenyl]iminomethylamino]-1-(4-pyrimidin-2-ylamino)prop-1-ene-1,3-diol;ethane N-[(5-cyclobutyl-4-methyl-1,2,4-triazol-3-yl)methyl]-3-(tetrazol-1-yl)benzamide 4-[6-(2,2,3,3,5,5,8b-hexadeuterio-7aH-furo[2,3-b]pyridin-4-yl)pyridazin-3-yl]morpholine 1-[5,6-dichloro-3-(methylamino)-2-(2-pyridin-4-ylethylamino)benzimidazol-7-yl]ethanone N-[(Z)-1-amino-3-hydroxyprop-2-enylidene]-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamide (3S,4R)-3-azido-1-phenylmethoxycarbonylpiperidine-4-carboxylic acid N-(2,3-difluorophenyl)-6-ethyl-1-oxothieno[3,2-e]thiazine-4-carboxamide 2-[4-(methylaminomethyl)phenyl]sulfonyl-1,3,6,7-tetrahydropyrazolo[1,5-a]pyrazine-4-thione 1-[(3Z,5E)-4-bromohexa-1,3,5-trien-2-yl]oxyethoxymethane;formaldehyde 6-[4-(4-propan-2-ylphenyl)sulfonylpiperazine-1-carbonyl]-3,4-dihydroisochromen-1-one 6-chloro-7-[(2S,3R)-4-[(6-fluoro-5-methoxypyridin-2-yl)methyl]-3-hydroxy-4-(1,3,4-oxadiazol-2-yl)butan-2-yl]oxy-4H-chromene-2-carboxylic acid 1-[7-(2,3-dihydropyrrol-1-yl)heptanoylamino]-N-[2-(4-ethoxyphenyl)-2-methylpropyl]cyclohexane-1-carboxamide 2-[8-chloro-6-fluoro-4-hydroxy-5-(methoxyiminomethyl)chromen-7-ylidene]propanedinitrile 4-(azidomethyl)-2-chloro-N-[2,4-difluoro-3-[5-[(4-methoxyphenyl)methylamino]-1,3,4-oxadiazol-2-yl]phenyl]benzamide 2-[4-[(4R,5S)-3,4-dihydroxy-5-methyloxolan-2-yl]oxyphenyl]acetonitrile N-(1,3-benzothiazol-2-ylmethylidene)hydroxylamine 3-[2-(dimethylamino)phenyl]propyliminoazanium (4S)-N-[2-cyano-5-(oxan-4-yloxy)phenyl]-1,3-dimethyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridine-4-carboxamide N-[1-(2-oxopyrrolidin-1-yl)propan-2-yl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-2-carboxamide N-(2,3-dihydro-1H-inden-5-yl)-2-methoxy-5-[[(1R,4S)-2,2,4-trifluorocyclopentanecarbonyl]amino]benzamide N-[1-(3,4,5-trimethoxyphenyl)ethyl]-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide N-(5-aminopentan-2-yl)-7-fluoroquinoline-3-carboxamide (4S)-1,3-dimethyl-4-[4-[2-(6-methylpyridin-3-yl)ethynyl]phenyl]-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 2-(1H-benzimidazol-4-yloxy)-5-[3-(trifluoromethyl)phenyl]pyridine-3-carboxamide 2-(3,6-dihydro-2H-pyridin-1-yl)-N-[4-fluoro-3-(trifluoromethyl)phenyl]pyrimidine-5-carboxamide 4-(6,11a-dihydrobenzo[b]quinolizin-2-yloxy)-N-diazobenzenesulfonamide 4-tert-butyl-2-(1H-indol-3-yl)morpholine 4-[5-methyl-2-(trifluoromethoxy)phenyl]pyrimidine N-ethyl-2,5-difluoro-4-phenylmethoxy-N-(2H-tetrazol-5-yl)aniline N-[[2-chloro-6-(1,5-dimethylimidazole-4-carbonyl)phenyl]carbamoyl]-2-hydroxybenzamide 4-chloro-2-N,5-N-bis(3-methylphenyl)pyridine-2,5-diamine (4-aminopiperidin-1-yl)-[5-chloro-6-(2,3-difluorophenyl)pyridin-3-yl]methanone 4-[3,5-bis(trifluoromethyl)phenyl]-2,6-dichloro-N-diazobenzenesulfonamide 4-hydroxy-1-[5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one 3-chloro-2,4-bis(9H-fluoren-1-yl)benzoic acid N-[1-(4-bromophenyl)-2,3-dimethylpropan-2-yl]formamide 4-[2-hydroxy-5-(2-methoxypyridin-3-yl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 1-N,3-N,5-N-tricyclopropylpyrazole-1,3,5-triamine 4-[2-(cyclopropylmethoxy)anilino]-5,8-dimethylquinoline-3-carboxylic acid;4,7-difluoronaphthalene-1-sulfinate (3S,4R)-N-[(2S)-1-(4-bromoanilino)-3-methylbutan-2-yl]-1-oxo-2,7-diazaspiro[4.4]nonane-4-carboxamide 2-methyl-4-(5,6,7,8-tetrahydronaphthalen-1-yloxy)pyrimidine ethane;N-ethyl-3-[4-(methylamino)-1H-indol-2-yl]imidazo[1,2-a]pyridine-7-carboxamide 1-(2-azido-6-methoxypyridin-3-yl)azepane (2Z)-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]penta-2,4-dienimidate 4-methoxy-6-(2-morpholin-4-ylethoxy)indazole-1-carboxylic acid 6-(3,4-difluorophenyl)-2-[5-(methylaminomethyl)pyrazin-2-yl]pyridine-3-carbonitrile 1,3-dibromo-5-(2,4,6-trimethylphenyl)sulfonyl-9H-fluorene 3-[(Z)-[4-(2,3-dihydro-1H-imidazole-5-carbonylamino)phenyl]methylideneamino]oxybenzoic acid 2-azidooxy-5,7-difluoroquinoline 1-(4-bromophenyl)-3,4-dihydronaphthalene 5-[4-(1H-indol-2-yl)cyclohexyl]pyridine-3-carboxamide 2-ethoxy-3,5,6-trimethylpyridine-4-carboxylic acid 2-amino-N'-[(1S)-1-cyclohexylethyl]benzenecarboximidamide 1-[2,3-bis(methylideneamino)phenyl]ethanol;formaldehyde 3-[3,5-dichloro-4-(1H-pyrazol-4-yl)phenyl]-2-oxopropanoic acid 2-(3,5-diethyl-1H-pyrazol-4-yl)-4-methoxy-6-[1-(oxan-4-yl)piperidin-4-yl]pyrimidine 2,4-dimethyl-N-(1H-1,2,4-triazol-5-yl)thiophene-3-carboxamide 5-[2,4-dichloro-3-(phenylmethoxymethyl)pyrrol-1-yl]-1H-pyrazole 1-[4,5-difluoro-2-(2-methylbenzoyl)phenyl]propan-2-one N-(4-bromophenyl)-2,3-dihydro-1,4-benzothiazine-6-sulfonamide;propane N-[5,6-bis(4-chlorophenyl)pyridazin-3-yl]propanamide 3-fluoro-4-(1,3,5-trimethylpyrazole-4-carbonyl)piperazin-2-one N-(2,3-dihydroxypropyl)-2-methoxy-N-[4-(thiophen-2-ylsulfamoyl)phenyl]acetamide (2R,3S)-3-methyl-4-oxo-1-[(3S)-3-phenylpyrrolidine-1-carbonyl]azetidine-2-carboxylic acid 2-[4-(difluoromethoxy)phenyl]-6,7-dihydrocyclopenta[b]pyridine 2-[3-(1H-indol-2-yl)phenyl]aniline 3-[1-(2,5-dimethylphenyl)triazol-4-yl]propane-1-sulfonamide 2-amino-1,4,5,6,7,8-hexahydrocyclohepta[b]pyrrole-3-carbonitrile;N-[(1R)-1-phenylethyl]acetamide 6-butoxy-3-(1-methylpyrazol-4-yl)pyrazolo[1,5-a]pyridine 1-[(4R)-3,3-difluoro-1-methylpiperidin-4-yl]-2H-pyrimidine 6-[4-bromobutan-2-yl(2,3-dihydroxypropyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 3-[2,4-difluoro-N-(3-methylbutyl)anilino]propane-1,2-diol 5-[2,3-dichloro-4-(trifluoromethyl)phenoxy]carbonyl-1,3,6,6a-tetrahydrocyclopenta[c]furan-3a-carboxylic acid N-[6,7-dichloro-2-hydroxy-1-(4-methoxyphenyl)sulfonylindol-3-yl]iminonaphthalene-1-carboxamide 7-chloro-3-ethylimidazo[4,5-c][1,8]naphthyridine 2-(hydroxymethyl)-5,7,8-trimethyl-1H-imidazo[4,5-g]quinoxaline-6,9-dione 4-(3,5-dimethoxyphenyl)sulfanyl-6-[4-methyl-6-(4-prop-2-ynoylpiperazin-1-yl)pyridin-2-yl]-1H-pyrrolo[2,3-c]pyridine-7-carbonitrile 1-(2,4-difluorophenyl)-N'-ethylmethanediamine;(E)-N-[4-[6-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]-4-oxobut-2-enimidamide 4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]cyclohexan-1-amine 6-[(3,5-diethoxy-4-hydroxyphenyl)methyl]-2-cyclohexa-1,5-dien-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one ethane;5-(4-fluorophenyl)-2-[3-methoxypropyl(methylsulfonyl)amino]-N-methyl-1-benzofuran-3-carboxamide 4-chloro-N-cyclohexyl-3-(2H-triazol-4-yl)benzamide 4-[2,5-dimethyl-1-(oxan-2-yl)imidazol-4-yl]pyridine N-(4,5-dihydroimidazol-1-yl)-2,7-dimethylindazole-3-carboxamide 2-(5-chloro-6H-benzo[b][1]benzazepin-11-yl)-N,N-dimethylethanamine (2E,4Z)-5-bromohepta-2,4-dienal;3-fluoro-N-methylaniline;N-[[1-(3-fluoroazetidin-3-yl)piperidin-4-yl]methyl]acetamide 5-[[3,4-bis(difluoromethoxy)benzoyl]amino]-2-(4-ethyl-1,4-diazepane-1-carbonyl)benzamide N-[2-(methylamino)ethyl]quinoline-3-carboxamide (2-benzamido-3,3-dimethylbutanoyl)phosphonic acid 5-[(1E,3Z)-4-aminopenta-1,3-dienyl]-N-methyl-1H-imidazole-2-carboxamide [(Z)-2-(2,6-difluorophenyl)-1-[4-(1H-1,2,4-triazol-5-ylsulfanylmethyl)anilino]ethenyl]-(pyridin-3-ylmethyl)azanide ethane;1-(4-ethoxyphenyl)-2,3-difluorobenzene (2R)-3,7-dihydroxy-1'-[(3S,4R)-3-phenylmethoxycarbonyl-1,2,3,4-tetrahydroisoquinoline-4-carbonyl]spiro[indene-2,4'-piperidine]-1-one 1-[[2,4-bis(methoxycarbonyl)phenyl]sulfonylamino]cyclopropane-1-sulfonic acid 2-amino-5,6-bis(4-hydroxyphenyl)pyrazine-3-carbonitrile 4-hydroxy-5-(4-methoxycarbonylphenyl)furan-2-carboxylic acid (3R)-4-(1,1-dioxothiazinan-2-yl)-N-[4-[(3S)-3-ethynylpyrrolidine-1-carbonyl]phenyl]-3-methylpiperazine-1-carboxamide;hydrochloride 5-[[1-(2,3-dihydro-1H-indene-4-carbonyl)piperidin-4-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one 1-[(2S)-3,3-dimethylbutan-2-yl]oxy-4-prop-1-en-2-ylbenzene [4-amino-3,5-dibromo-2-(trifluoromethyl)phenyl]methanethiol;butanoic acid 3-chloro-N-[1-[2,6-dichloro-4-(trifluoromethyl)phenoxy]propan-2-yl]aniline 5-[(4-ethylsulfanylpiperazin-1-yl)methyl]-2-methoxypyridine 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[[3-[4-methoxy-3-(trifluoromethoxy)phenyl]phenyl]methylsulfonylamino]urea 3-[4-(1,2-dihydronaphthalen-2-yl)phenyl]-5-(4-propoxyphenyl)-1H-pyrazole 4-[5-(3,3-dimethylbutoxy)pyridin-2-yl]oxy-6,7-dihydroquinoline (E)-4,4-difluoro-N-[5-(4-hydroxypiperidine-1-carbonyl)-2-methylphenyl]but-2-enamide 4-[6-(cyclobutylamino)pyridazin-3-yl]phenol (NZ)-N-[2-isoquinolin-3-ylchromen-4-ylidene]hydroxylamine 1-ethenylsulfonyl-4-[(3E)-hexa-1,3,5-trien-3-yl]benzene 4-[6-[(2E,3Z)-2-ethylidenehexa-3,5-dienyl]pyridin-1-ium-3-yl]benzoic acid (1S,2R)-2-fluoro-N-[6-methyl-4-oxo-3-phenyl-5-(trideuteriomethoxy)-7H-pyrazolo[4,3-d]pyrimidin-1-yl]cyclopropane-1-carboxamide 3,4-dibromo-N-[1-(4-ethylsulfonylphenyl)pyrrolidin-3-yl]benzamide 6-azido-5,8-dihydro-1H-pyrazolo[3,4-g]quinoline [3-(2,4-dichlorophenyl)imidazo[1,5-a]pyridin-1-yl]-cyclopropylidenemethanol 6-benzylsulfanylcyclohexen-1-ol 1-cyclopropyl-N,2-dimethyl-5-pyridin-3-ylimidazole-4-carboxamide 1-azido-3,3-difluoro-4-(3,4,5-trichlorophenyl)butan-2-one N-(2-hydroxyethyl)-4-[4-[3-methoxy-4-[5-methyl-1-[2-[(1-propan-2-ylpyrazol-3-yl)amino]pyrimidin-4-yl]imidazol-2-yl]phenyl]piperazin-1-yl]benzamide (5E)-5-[[2,3-bis(trifluoromethyl)phenyl]methylidene]-4-hydroxy-2-sulfanylidene-1,3-thiazolidin-3-ium-3-carboxamide 5-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-ethoxy-4-[6-methyl-3-[(2-morpholin-4-ylacetyl)amino]cyclohexa-1,3-dien-1-yl]-1,2-oxazole-3-carboxamide N-[(4-chlorophenyl)methyl]-2-cyano-N,3-dimethylbenzimidazole-5-carboxamide N-benzyl-3-(dimethylamino)-5-nitrocyclohexa-1,4-diene-1-carboxamide 1-cyclobutyl-N-[2-(7-methoxyquinolin-4-yl)ethyl]formamide 5-[2-[7-(4,6-dimethoxypyrimidin-5-yl)thieno[3,2-b]pyridin-2-yl]-1-phenylethylidene]-1,3-thiazolidine [3,4-bis(phenylmethoxy)phenyl]methanimine 3-[2-(4-ethylphenyl)phenyl]-5-methoxyphenol 7-(2,6-difluoro-3,5-dimethoxyphenyl)-1H-pyrido[2,3-d]pyrimidine-2,4-dione N-(5-chloro-2,3-dihydro-1H-inden-4-yl)formamide;1-[5-[methylamino-(2,2,6,6-tetramethylpiperidin-4-yl)oxyphosphinothioyl]oxypyridin-2-yl]ethanone 1-cyclopropyloxyethanol;1-[2,3-dihydroxy-6-(piperidine-1-carbonyl)naphthalen-1-yl]propan-1-one 3-azido-2,4-dihydroindeno[1,2-b]pyridine 5-N-[(3R)-1-methylsulfonylpiperidin-3-yl]-1,2-dihydroquinoline-4,7-diamine 6-methyl-N-(3-phenylpropyl)nonan-1-amine 2-(7,8-difluoro-3,4-dihydro-1H-pyrano[4,3-c]pyridin-5-yl)acetamide;ethane 4-[(3E,5Z)-6,7-difluorohepta-1,3,5-trien-3-yl]-N-[3-(5-pyridin-2-yl-1H-pyrazolo[3,4-c]pyridin-3-yl)phenyl]piperazine-1-carboxamide [2-(1,3-benzothiazol-2-yl)phenyl]-dimethoxyphosphane 2-chloro-5,6-dideuterio-N-[3-(4-fluorophenyl)-1-hydroxypropan-2-yl]-3-hydroxybenzamide 2-azido-N-(1,3-benzothiazol-2-ylmethyl)-5-[(4,4-difluorocyclohexyl)amino]pyrrolo[2,3-d]pyrimidine-7-carboxamide 5-(2,4,6-trihydroxyphenyl)-1H-pyrazole-3-carboxylic acid (2-hydroxynaphthalene-1,4-diyl)phosphonic acid 1-[5-(3,4-dihydroxyphenyl)-6-methyl-7-pyridin-4-ylpyrazolo[1,5-a]pyrimidine-2-carbonyl]pyrrolidine-2-carboxylic acid 2-[(2,4-dichloropyrimidin-5-yl)-pyridin-3-ylamino]decanoic acid 2-[4-(1H-indole-5-carbonyl)piperazin-1-yl]-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one N-methyl-2-[[5-(1H-pyrrole-3-carboximidoyl)pyrimidin-4-yl]amino]ethanimidate 2-(dimethylamino)-7,9-bis(3-hydroxypropyl)purine-6,8-dione N-[(3S)-6-chloro-1'-(2,2-dimethylpropanoyl)spiro[1H-indole-3,4'-5,7-dihydropyrazolo[3,4-b]pyridine]-2'-yl]benzamide 2-[5-(4,6-dimethoxypyrimidin-2-yl)-2,3-dihydrothieno[3,4-b][1,4]dioxin-7-yl]ethanamine;hydrochloride N-cyclohexyl-1,3-dihydroisoindole-2-carboxamide 5-amino-2,4,6,7-tetrahydrotriazolo[4,5-c]pyridine-3-thione (E)-N-[3-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]phenyl]but-2-enehydrazide N-[(4-cyanophenyl)methyl]-1,3-dimethyl-4H-pyrido[2,3-d]pyrimidine-6-carboxamide 6-[4-(1,3-thiazol-2-ylmethoxy)phenyl]hexanoic acid 3-[(6-bromopyridin-2-yl)amino]sulfanylbenzoic acid 3-[4-(cyclohexylamino)-6-[3-methyl-4-[[2-(methylamino)acetyl]amino]phenyl]-5H-pyrido[3,2-d]pyrimidin-8-yl]propanamide (2E)-2-[1-(4-methylphenyl)sulfanylpyrrol-3-ylidene]-N-phenyl-3H-thieno[3,2-b]thiopyran-6-amine 2-[5-(2,6-difluorophenyl)-1H-pyrazol-4-yl]-8-methoxypyrido[3,2-d]pyrimidine 3-methylsulfonyl-N-[3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)phenyl]propanamide 5-(cyclohexanecarbonylamino)-3-methylthiophene-2-carboxylic acid 4-[6-(4,4-dimethylpiperidine-1-carbonyl)pyridin-3-yl]-2-methoxyphenol 2-azido-N-[2-(3,4,5-trimethoxyphenyl)ethyl]acetamide 2-[(4-methylphenyl)iminomethyl]pyridin-1-ium-3,4-diamine;bromide 5-methyl-2-(5-oxopyrrolidin-2-ylidene)tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaene-7,12,14-tricarboxylic acid 5-phenylcyclohepta-1,3,6-triene-1-carboxylic acid N-[4-(difluoromethylsulfanylamino)cyclohexyl]-2-[2-[(E,3S)-7-hydroxyhept-1-enyl]-5,6-dihydrobenzimidazol-1-yl]acetamide 1-[2-(3,5-dimethoxyphenyl)ethynyl]pyrazole 4-N,6-N-bis[(2E)-4-hydroxypenta-2,4-dienyl]quinoline-2,7-disulfonamide (E)-N-[4-chloro-3-[(2,3-dimethylphenyl)carbamoyl]phenyl]-3-(4-hydroxy-1H-indol-6-yl)prop-2-enamide (5S,6R)-7-acetyl-3-butylsulfanyl-2,6-diphenyl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 6-methyl-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-10H-benzo[b]carbazole 2-amino-4-(4-ethoxy-3-methylphenyl)-1,5-dihydropyrrolo[3,2-d]pyrimidine-2-carbonitrile 6-[[4-(diethylamino)phenyl]methyl]-2,5-bis(methylideneamino)pyrimidine-4-carbonitrile;hexane 2-(2,4-dimethoxyphenyl)-3-[7-(trifluoromethyl)-1H-indol-5-yl]-1H-pyrido[4,3-b]azepine N-[1-(3,4-dimethoxyphenyl)-2-[6-ethyl-5-[methyl-(2,2,6,6-tetrafluorooxan-4-yl)amino]pyridazin-3-yl]ethylidene]hydroxylamine 2-(4-ethylsulfonylphenyl)-5-(1,1,1,3,3,3-hexafluoropropan-2-ylideneamino)-6H-phenanthridine 5-chloro-2-[3-[(4,6-dioxo-1H-1,3,5-triazin-2-yl)sulfanyl]propoxycarbonylamino]benzoic acid 5-cyclobutyl-3-[2-hydroxy-4-(propanoylamino)phenyl]-N-[2-(trifluoromethoxy)ethyl]pyrazole-1-carboxamide 3-(2,6-dimethyl-4-oxo-5H-thieno[2,3-d]pyrimidin-3-yl)piperidine-1-carboxylic acid 5-chloro-2-[3-(4-methyl-1,3-thiazol-2-yl)phenoxy]benzonitrile 5-(2-bromophenoxy)-1,3-thiazolidine 2-[[3-amino-6-(4-methylcyclohexen-1-yl)pyrazine-2-carbonyl]amino]acetic acid N-[(2R)-2-amino-1-[3-(trifluoromethyl)phenyl]sulfonylpropan-2-yl]acetamide N-(2,3-dihydro-1H-inden-5-yl)-4-[[1-ethyl-6-methoxy-7-(2-pyrrolidin-1-ylethoxy)quinazoline-2,4-diylidene]amino]aniline 4-[[3,5-bis(trifluoromethyl)phenyl]iminomethyl]-2-iodo-6-nitrophenol 1,2-dimethyl-N-(5-methyl-1,3-thiazol-2-yl)-6-oxopyridine-3-carboxamide [(3R,4S)-3-amino-4-hydroxypiperidin-1-yl]-[2-methyl-5-(trifluoromethoxy)phenyl]methanone;hydrochloride 4-N-[(2S)-1-aminopropan-2-yl]-6-N,3-dimethyl-5-N-[(4-phenyl-1H-pyrazol-5-yl)methyl]-3,6-dihydro-2H-pyridine-4,5-dicarboxamide 4-chloro-N'-(2,3-dihydroindole-1-carbonyl)pyridine-2-carbohydrazide [4-hydroxy-2-(hydroxymethyl)pyrrolidin-1-yl]-(5,6,7,8-tetrahydroquinolin-6-yl)methanone 3,5-diethyl-4-methoxypyridine-2-carboximidamide 1-(2-tert-butylpyridin-4-yl)-6-[[7-methoxy-2,3-dihydro-1H-cyclopenta[b]quinolin-9-ylidene]amino]hexan-2-one 1-(2-azidophenyl)-9H-fluorene 1-[2,4-bis(phenylmethoxy)phenyl]-N-[6-(4-fluoroanilino)purin-9-yl]ethanimine 4-[(1S)-5-methylcyclohex-2-en-1-yl]benzoic acid 1-(3,4-dichlorophenyl)sulfonyl-N-ethyl-N-methylpiperidin-4-amine 4-[6,7,8,9,10,11-hexahydroazecin-3-yl(difluoro)methoxy]aniline 2-[(4-acetylphenoxy)methyl]-3H-quinazolin-4-one 3-(difluoromethoxy)benzenethiol (E)-N-[2-hydroxy-2,3-bis[(Z)-prop-1-enyl]cyclobutyl]-4-pyridin-4-ylbut-3-enethioamide 1-azidooxy-3,5-dichloro-2-methylbenzene 4-[(3R)-6-[cyclopropylsulfonyl-[(2S)-2-hydroxy-3-phenylpropanoyl]amino]spiro[3.5]nonan-3-yl]oxypyridine-2-carboxamide 3-(2,4-dihydroxyphenyl)-6-methylsulfanyl-2-(1H-pyrazol-5-yl)phenol 6-[(1,3-dioxoisoindol-2-yl)methyl]quinoline-8-sulfonic acid N'-(4,6-dimethylpyrimidin-2-yl)-4-(trifluoromethoxy)benzenecarboximidamide (Z)-3,7,11-trihydroxynaphtho[1,2-b][1]benzofuran-6,11-dione [(3aR,7aS)-1-(4-fluorophenyl)sulfonyl-2,2-dimethyl-3a,5,6,7,7a-hexahydropyrrolo[3,2-b]pyridin-3-yl]-cyclopropylmethanone N-(2,2-dimethylpropyl)-1'-[2-(trifluoromethyl)benzoyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 1-amino-2,3-diethylanthracene-9,10-dione 6-[5-(cyclopentylmethoxy)pyridin-3-yl]isoquinolin-2-ium 3-butyl-1,5,6,7,8,9-hexahydrocyclohepta[b]pyrrole 4-chloro-6,8-difluoroquinoline-3-carboxylic acid 2-[(2E,4Z)-hexa-2,4-dien-3-yl]oxy-1H-indole 1-azido-3-[5-ethyl-6-methoxy-2-(trifluoromethyl)indol-1-yl]propan-2-ol 5-(2-methylpropoxy)-N-[5-(4-oxo-2,3,5,7,8,10-hexazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,9-tetraen-11-yl)pyrazin-2-yl]pyridine-2-carboxamide N-(2,3-dimethylphenyl)-4-hydroxy-5-oxothieno[3,2-b]pyran-7-carboximidate 4-(3-ethoxyphenoxy)-N'-[2-(3-methylfuran-2-yl)-2,3-dihydro-1H-benzimidazole-5-carboximidoyl]cyclohexane-1-carboximidamide 4-(1H-pyrrol-2-yl)benzaldehyde;N,3,3-trimethylbutanamide 2-[5-azido-1-(furan-3-yl)pentan-3-yl]thiophene 1-(4,6-dimethoxypyrimidin-2-yl)-3-(furan-2-yl)sulfonylurea 6-(4-fluorophenyl)-1-[(E,3R)-5-methoxy-2-methylidenehex-4-enyl]indazole 2-methyl-4-phenyl-1,3-dihydroisoindole 1-(4-bromo-3-chlorophenyl)-2,6-dimethylheptan-3-one 2-(4,6-dimethylpyrimidin-5-yl)cyclohepta-1,3,5-triene-1-carbonitrile 2,6-dichloro-4-(methylcarbamoyl)benzoic acid;ethane [4-[2-(2,6-diethylanilino)-1-methylbenzimidazole-5-carbonyl]piperazin-1-yl]-[4-(3H-pyrrolo[2,3-c]pyridin-2-yl)phenyl]methanone [(3R)-1-azido-4,5-dimethoxypentan-2-yl]benzene [5-[3-fluoro-5-(3-methoxyazetidine-1-carbonyl)phenyl]-3-methylpyridin-2-yl]-morpholin-4-ylmethanone N-[4-[[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]carbamoyl]phenyl]pyridine-4-carboxamide 4-ethyl-2,6-dipyridin-3-ylpyridine 6-azidooxy-2,4-dichloroquinoline N-[4,6-dichloro-2-(methylamino)pyrimidin-5-yl]hydroxylamine [2-(5-bromopyrimidin-4-yl)oxyphenyl]methanamine;hydrochloride 6-[3-(4,7-diazaspiro[2.5]octan-7-yl)propylamino]pyridine-3-carboxylic acid 2-[[4,5-dimethyl-3-(1H-pyrrole-2-carbonyl)furan-2-yl]methoxy]-5-fluorobenzamide [1-cyclopropyl-4-[6-(5-methoxypyridin-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]pyrrolidin-3-yl]methanol 2-[1,3-bis(sulfanyl)propoxy]isoindole-1,3-dione (1R)-2,2-dichloro-N-[4-fluoro-3-[6-(1H-indazol-5-ylamino)-5-methanimidoylpyrimidin-4-yl]phenyl]cyclopropane-1-carboxamide 1-(2,3-dihydro-1H-inden-5-yl)-3,4-dimethylpiperazine 1-(5,6,7,8-tetrahydroisoquinolin-3-yl)butan-2-one 3-(2-phenylmethoxyethyl)oxetan-3-ol N-[(1R,2S)-2-hydroxycyclohexyl]-7-(methylamino)-5-[[6-(morpholin-4-ylmethyl)pyridin-3-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carboxamide 4-azido-N,N-diethyl-1H-indazole-5-sulfonamide (E)-3-[4-[2-(2,5-dimethylphenyl)ethoxy]-3-iodophenyl]prop-2-enoic acid 1-azidooxy-4-methylsulfonylbenzene 6-methyl-N-[1-(2-pyrazol-1-ylethyl)piperidin-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 1-(4-benzylpiperazin-1-yl)ethanethiol;4-(dimethylamino)-N-[[2-fluoro-5-[3-(morpholin-4-ylmethyl)phenoxy]phenyl]methylideneamino]benzamide N-[3-[(2S)-morpholin-2-yl]propyl]-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamide 1-[2-ethyl-5,6-bis(trifluoromethoxy)benzimidazol-1-yl]-3-(4-isocyanophenyl)propan-1-one 3,4-difluoro-5-[7-methoxy-6-(4-pyrrolidin-1-ylpiperidin-1-yl)quinoline-2-carbonyl]benzamide 7-[(E)-2-(4-methoxyphenyl)ethenyl]-3H-benzimidazol-5-ol 1-[2,4,6-trimethyl-N-(1-phenylpropyl)anilino]propan-2-one 6-N,2-bis(4-tert-butylphenyl)-4-N-[1-(4-chlorophenyl)ethylideneamino]pyrimidine-4,6-diamine 1-[2-methyl-1-oxo-1-[(2S)-pyrrolidin-2-yl]propan-2-yl]-3,5-bis(trifluoromethyl)pyrazole-4-carboxylic acid N-[5,6-difluoro-4-(2-fluorophenoxy)pyridine-3-carbonyl]acetamide 2-(2,5-dimethylpyrazol-3-yl)-N-[1-(2-hydroxyethylamino)propan-2-yl]thieno[2,3-b]pyridine-4-carboxamide;ethane 2-[2,6-dichloro-N-(4-hydroxybutyl)-3-nitroanilino]propanoic acid 3-fluoro-4-[(2R)-2-methoxypropyl]benzenecarboximidamide 2-amino-5,6-difluoro-1-phenylmethoxycarbonylindole-3-carboxylate 1-[3-[4-(2-methoxypyridin-4-yl)imidazol-1-yl]phenyl]pyrrolidine-3-carboxamide [(3R)-4-[(5-methylpyrido[2,3-b]indole-9-carbonyl)amino]oxolan-3-yl]carbamic acid 3-[4-(1,1-difluoropropyl)phenyl]azetidine;ethane (1S,2R)-N-[8-amino-6-(5-chloropyridin-3-yl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide (E)-N-[1-[5-ethyl-4-[2-(4-hydroxy-3,5-dimethoxyphenyl)-6-methoxyquinolin-4-yl]-2-methoxyphenyl]ethenyl]propanamide 4-[2,6-dibromo-3-(cyclopropylmethoxy)phenyl]pyridine N-methyl-3,5-di(propanoyl)benzamide N-cyclohexyl-2-[[5-(1H-pyrrol-3-yl)thiophen-2-yl]sulfonylamino]acetamide 1-[3-(3,4-dihydroquinoxalin-2-yl)propyl]-3-phenylurea;ethane 2-[(2,4-dioxo-1H-pyrimidin-5-yl)-propylamino]-2-methylpropanoic acid N-[5-(4,5-dimethoxycyclohexa-1,3-dien-1-yl)sulfonyl-2-fluorophenyl]propanamide N-[2,5-dichloro-3-[3-cyano-6-(2-fluorophenyl)pyridin-2-yl]phenyl]carbamate 3-[1-azido-3,5-bis(trifluoromethyl)pyrazol-4-yl]-4-ethoxypyridine 1-(4-azidophenyl)-3,5,5,8,8-pentamethyloctane-2,7-dione 1-(3,4-dihydroxyphenyl)hexan-2-one 4-(2,6-ditert-butylphenyl)sulfonylbenzenethiol;titanium 1-[2,4,6-tris(trifluoromethyl)phenyl]piperazine N-(1H-benzimidazol-2-ylmethyl)-5,6-dihydroisoquinoline-3-carboxamide 1-(4-chlorophenyl)sulfonyl-7-ethenyl-5-methoxyindole 1-[2-chloro-3-(methoxymethyl)phenyl]sulfonyl-4,5-dihydroimidazole 4-[5-(3,4-dihydropyrazole-2-carbonyl)-1H-pyrrol-3-yl]benzonitrile 6-[[5-amino-3-[4-(1H-indol-2-yl)phenyl]pyrazol-1-yl]methylidene]cyclohexa-2,4-dien-1-one N-[3-(4-methoxyphenyl)sulfanylpropyl]-1-[[1-[2-(3-methylphenoxy)acetyl]piperidin-4-yl]methylsulfonyl]-6-(trifluoromethyl)-2,3-dihydroindole-2-carboxamide (2R)-2-[(5,6-dimethylpyrimidine-4-carbonyl)amino]-4-methoxybutanoic acid 1-amino-1-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]pentane-1,5-diol (1R)-2-[5-fluoro-2,3-bis(trifluoromethyl)phenoxy]-N-methoxy-1-pyrimidin-2-ylethanamine 5-[(E)-[2-hydroxy-3-methoxy-4-[[3-(trifluoromethyl)phenyl]iminomethyl]phenyl]methylideneamino]-1,3-dimethylbenzimidazol-2-one 5-(4-fluorophenyl)sulfonyl-N,2,3-trimethylbenzamide 1-(2,3,5,6-tetradeuteriophenyl)decan-1-one 2-[(5Z)-4-oxo-5-[[3-[(E)-2-phenylethenyl]furan-2-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid 5-[[(1S)-3,4-dichlorocyclohexa-2,4-dien-1-yl]methoxy]-N-ethylthiophene-2-carboxamide 3-[3-bromopropyl(cyclohexylmethyl)amino]phenol 3-[[4-azidooxy-1-(2,6-difluorophenyl)butyl]amino]propanenitrile 6-[2-[3,5-dimethyl-1-(methylsulfonylmethyl)pyrazol-4-yl]pyridin-3-yl]-N-[4-methoxy-5-(trifluoromethyl)pyrimidin-2-yl]-8-methylquinazolin-4-amine [3-(4-hydroxyphenyl)azetidin-1-yl]-[2-(thiophen-3-ylmethoxy)naphthalen-1-yl]methanone 2-[1-(3-chlorophenyl)piperidin-4-yl]oxyquinoline 2-[4,5-difluoro-6-(4-fluorophenyl)-1H-indol-3-yl]acetic acid (E)-3-[4-(2,5-dioxopyrrol-1-yl)phenyl]prop-2-enoic acid 4-[2,3-bis(ethenyl)-5H-1,4-benzodiazepine-1-carbonyl]-N,N-dipropylbenzamide 2,5-bis(4-methylphenyl)-N,N'-dipentylpropanediamide 3-[1-(2,4,6-trimethylphenyl)imidazol-2-yl]benzene-1,2-diol;zinc (2S)-3-(1H-indol-5-yl)propane-1,2-diol;(E)-N'-(6,7,8,9-tetrahydrobenzo[g]quinazolin-4-yl)but-2-enehydrazide 4-azido-2,3-dichlorobenzoic acid 1-[(2S)-3-cyclohexyloxy-1-methoxypropan-2-yl]-N,2-diphenylindole-6-carboxamide 2-[(Z)-[3,5-dimethyl-1-(6-oxohexyl)pyridin-4-ylidene]methyl]isoindole-1,3-dione 4-[[(3R)-1-methyl-5-oxopyrrolidin-3-yl]amino]benzamide (2S)-N-[1,3-dihydroxy-1-[4-(7-methylcyclohepta-1,4,6-trien-1-yl)phenoxy]propan-2-yl]-5-oxopyrrolidine-2-carboxamide (2-methyl-4-phenylthiophen-3-yl)-[3-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone 6-methyl-3-[(5-methylthiophen-2-yl)methyl]-1,4-dihydroquinazolin-2-one [2-(4-methoxyphenyl)sulfanylphenyl]boronic acid 1-[3-(oxolan-2-ylmethoxy)-5-[[3,4,7-trihydroxy-6-(hydroxymethyl)naphthalen-2-yl]methylideneamino]phenyl]ethanone (2S)-2-[4-[5-(1,3-benzoxazol-2-ylmethoxy)pyridin-2-yl]piperidine-1-carbonyl]pyrrolidine-1-carboxylic acid 4-[[6-bromo-1,8-dimethyl-7-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]amino]-N'-hydroxybenzenecarboximidamide 1-(4,5-dichlorothiophene-2-carbonyl)-2-methylpyrrolidine-2-carboxamide 5-fluoro-1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethyl)indazole 2,6-bis(2,4,4-trimethylpentan-2-yl)benzene-1,4-diol [(Z)-[4-ethyl-2,3-bis(hydroxymethyl)phenyl]methylideneamino]thiourea (1S,3R)-5-(2-azidocyclopropyl)oxy-N'-[(4-chlorophenyl)methyl]-3-(methanesulfonamido)-1-methyl-2,3,4,9-tetrahydrocarbazole-1-carbohydrazide 1-[4-(4,5-dihydro-3H-1-benzazepine-2-carbonyl)phenyl]imidazolidin-2-one 4-[2-[4-[(1R)-3,5-bis(trifluoromethyl)cyclohexa-2,4-dien-1-yl]phenyl]ethynyl]-N-(1,4,5,6-tetrahydropyrimidin-2-yl)benzamide 2-methyl-N-(1,3-thiazol-4-yl)oxane-3-carboxamide 4-[7-cyclopentyloxy-6-methyl-8-(2,3,5,6-tetradeuteriopyridin-3-yl)oxyoctyl]benzaldehyde (4-dibenzofuran-3-ylphenyl)-[2,6-di(propan-2-yl)phenyl]azanide;hafnium 3-[(4-methoxyphenyl)sulfonylamino]-N-phenylpyrrolidine-1-carboxamide N-methyl-6-[4-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]pyridine-3-carboxamide 5-azidooxy-1H-benzo[c]chromene (1R,2S)-2-N-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]-2-N-[5-(trifluoromethoxy)pyridin-2-yl]cyclohexane-1,2-diamine 4-[2,3-dihydroxypropyl(ethyl)amino]benzenesulfonamide 2-chloro-N-[[3-(2-methylpyrazol-3-yl)phenyl]methoxy]acetamide (4-butylphenyl)-oxo-[(2-phenylacetyl)amino]azanium 3-[[(5Z)-3-benzyl-5-[[4-bromo-2-(trifluoromethoxy)phenyl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoic acid 2-(2,6-diethylphenyl)-N-[4-fluoro-3-[7-(2-methoxyethylamino)pyrido[1,2-a]pyrimidin-4-ium-4-yl]oxyphenyl]-5-oxopyrrolidine-1-carboxamide 2-[1-(1H-indol-5-yl)ethenoxy]aniline 5-[4-[(2,3,6-trifluorophenyl)methoxy]phenoxy]pentanoic acid 1-[4,6-di(propan-2-yl)pyrimidin-5-yl]but-3-en-1-one 3-[2-(1-aminocyclobutyl)phenyl]pyrrolidine-2,5-dione;hydrochloride 2-[4-(2,3-dichlorophenyl)piperazin-1-yl]benzoic acid 2-amino-4-[3,5-bis(ethenyl)phenyl]-6-methylbenzene-1,3-dicarbonitrile 2-[4-(2,5-dimethylpyrrol-1-yl)phenyl]-6-[3-methoxy-4-[(4-nitropyrazol-1-yl)methoxy]phenyl]oxan-4-ol 4-(3,5-dimethylphenoxy)-2-ethenyl-1-prop-1-ynylbenzene;ethane 2,3-bis(propan-2-ylsulfanylmethoxy)quinoline 4-[5-(3,7-dimethylimidazo[1,2-a]pyridin-6-yl)-1,2-oxazol-3-yl]phenol [2-[(2,6-difluorophenyl)methoxy]pyridin-3-yl]-(2-ethylmorpholin-4-yl)methanone 2-(dimethylamino)-1'-[(3,5-dimethylphenyl)methyl]spiro[4H-isoquinoline-3,4'-piperidine]-1-one;2,2,2-trifluoroacetic acid (3Z,5E)-N,N,3-trimethyl-7-[[2-[4-(2H-tetrazol-5-yl)phenyl]ethylamino]sulfanylamino]hepta-3,5-dienamide N-[1-(5,6-dihydrothieno[2,3-b]pyrrole-4-carbonyl)piperidin-4-yl]-4-ethoxybenzamide 6-fluoro-3-(1H-pyrazol-5-yl)indole-2,7-dione 2-[(4-ethylpiperazin-1-yl)methyl]-7,8-dihydro-6H-furo[3,2-e]benzimidazole;hydrochloride (1S,5R)-1-(2,4,6-trimethylphenyl)bicyclo[3.1.0]hexane 2,3-dimethylpentane;6-ethenyl-N'-propanoylpyridine-3-carbohydrazide 4-[[4,5-dimethyl-2-(sulfanyloxymethyl)thiophen-3-yl]methylideneamino]benzonitrile 6-methylsulfanyl-4-(phenylsulfamoyl)naphthalene-2-carboxylic acid N-(4-bromobutan-2-yl)-2,4-dichloro-N-(1H-imidazol-5-ylmethyl)pyrimidin-5-amine 1-[2,3-difluoro-4-(trifluoromethoxy)phenyl]pentan-2-one 4-[2,6-difluoro-3-[(5R)-3-[3-methoxycarbonyl-1-methylsulfonylazetidin-3-yl]-5-propanoyl-1,4-oxazepane-4-carbonyl]phenyl]benzoic acid [(4R,5S)-3,6-dimethyl-7-azabicyclo[2.2.1]heptan-4-yl]-(8-fluoroquinolin-5-yl)methanone 3-(N-benzyl-2,4-dinitroanilino)propanoic acid 3-[(3R)-2,6-dioxopiperidin-3-yl]-5-[2-(methylamino)ethylcarbamoylamino]thiophene-2-carboxamide N-benzyl-N-methyl-1H-imidazole-2-sulfonamide 2-(5,6-diaminopyridin-3-yl)-N-[4-[2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxyethyl]phenyl]acetamide N-[4,4-dimethyl-1-(1H-pyrrolo[3,2-b]pyridin-6-yl)piperidin-3-yl]-2-(1-methoxyindol-7-yl)acetamide [4-(4-methoxyphenyl)piperazin-1-yl]-(3-methylsulfinylquinolin-6-yl)methanone 1-[4-[3-(3,5-dimethyltriazol-4-yl)-6-[1-(oxetan-3-yl)pyrazol-4-yl]imidazo[4,5-b]pyridin-2-yl]-3-fluorophenyl]pyrrolidine-2,3-dione 4-azido-5-ethylnaphthalene-2-thiol 3-[[2-fluoro-4-(trifluoromethyl)phenyl]carbamoylamino]propanoic acid 1-[4-(5-ethoxypyridin-3-yl)phenyl]-2,6-dimethyl-7H-purine 4-(N-azidosulfonylanilino)benzenecarboximidamide N-[[4-(5,6-dimethylpyridin-3-yl)phenyl]methyl]formamide;3-fluorobenzaldehyde 1-(2,4-dichlorophenyl)-N-[4-methyl-3-(1-oxo-6H-pyrrolo[3,4-c]pyrrole-5-carbonyl)phenyl]cyclopropane-1-carboxamide (2R)-1-[3,4-bis(phenylmethoxy)phenyl]propan-2-amine;hydrochloride 2-[3-aminopropyl(propan-2-yl)amino]acetaldehyde;4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)benzenesulfinamide 4-N,6-N-bis(2-phenylmethoxyethyl)pyrimidine-4,6-diamine N-(7,8-dimethyl-5,6-dihydroimidazo[1,2-a]pyridin-3-yl)cyclopropanecarboxamide 5-chloro-N-[(3,4-dimethoxyphenyl)methyl]-2-[[4-(hydroxyamino)cyclohexylidene]amino]benzamide 2-[(5R)-4,7-dioxo-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]-N-(1-phenylethyl)acetamide 1,2-diphenyl-5-(trifluoromethyl)cyclohexa-3,5-diene-1,3-dicarboxylic acid [4-amino-2-(3,6-dimethylimidazo[1,5-a]pyridine-7-carbonyl)thieno[2,3-d]pyrimidin-5-yl]-cyclohexylmethanone N-[(2S)-3-(4-methoxyphenyl)-1-oxo-1-[3-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]azetidin-1-yl]propan-2-yl]furan-2-carboxamide N-[2-methyl-4-(3,4,5-trimethoxyphenyl)pyridin-3-yl]acetamide N-[(4S)-1,2,3,4-tetrahydroisoquinoline-7-carbonyl]-3H-benzimidazole-5-carboxamide N-[(1R,2S)-3-chloro-1-hydroxy-1-[4-(4-morpholin-4-ylphenyl)phenyl]propan-2-yl]carbamate 5-(3,4-dimethylphenyl)-4-[(2-ethoxyphenyl)iminomethyl]-1,2-dihydropyrazol-3-one N-[2-[3-(4-chlorophenyl)pyrrolidin-1-yl]ethyl]spiro[5,6-dihydrocyclopenta[b]pyridine-7,3'-azetidine]-1'-carboxamide (2R)-N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-1-[6-(trifluoromethoxy)pyridine-3-carbonyl]pyrrolidine-2-carboxamide 1-[4-(aminomethyl)phenyl]propane-2,2-diol;ethane 4-[(3,5-dichlorophenoxy)methyl]-1-ethoxypiperidine;propan-2-ol 1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethanone 4-tert-butyl-1-chloro-2-methoxybenzene;ethane 1-[(E)-3,4-dimethylpent-2-en-2-yl]-3-fluoro-5-iodobenzene 2-[4-fluoro-3-(2,2,2-trifluoroethyl)phenyl]acetamide 6-(4,8-diazaspiro[2.5]octane-8-carbonyl)-1H-quinolin-2-one 2-[(Z)-benzylideneamino]oxyethanol N-ethyl-4-(4-methoxyphenyl)-2,3,7,11-tetrazatricyclo[7.3.0.02,6]dodeca-1(12),4,6,8,10-pentaen-5-amine 2-(3,5-difluorophenyl)-4H-pyrrolo[3,4-c]pyrazol-6-ium 2-[[4,5-bis(ethenyl)imidazol-1-yl]methoxy]-3H-quinazolin-4-one (3-methylcyclobutyl)-[3-[4-[2-(5H-pyrrolo[1,2-a]imidazol-7-ylidenemethylamino)ethyl]pyridin-2-yl]sulfanyl-2-(trifluoromethoxy)phenyl]diazene 3-[2,6-dichloro-4-(trifluoromethyl)phenoxy]pyridine 1-(1,3-benzodioxol-5-ylmethoxy)-N'-hydroxypyrazole-4-carboximidamide 2-[(4S,7R)-7-methyl-5-phenyl-3-thiophen-2-yl-6,7,8,9-tetrahydro-4H-pyrazolo[3,4-b]quinolin-1-yl]phenol 6-methoxy-2,3-dipropylnaphthalene-1,4-dione 3-[(4-chlorophenyl)methyl]-N-cyclohexa-1,5-dien-1-ylazetidine-1-carboxamide 1-[4-(dimethylamino)phenyl]-3,3-dimethylbutan-2-one N-[(2S,3R)-1-oxo-7-pyrrolidin-1-yl-6-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-5-yl]cyclopropanesulfonamide 4-[2,2-diethoxyethyl([1,2,4]triazolo[4,3-a]pyrazin-5-yl)amino]benzoic acid 3-[3,5-dihydroxy-7-(hydroxymethyl)oxepan-2-yl]benzonitrile 5-(1,3-benzoxazol-6-yl)-3-[4-[3-fluoro-5-(2-pyrrolidin-1-ylethoxy)phenyl]-1H-benzimidazol-2-yl]-1H-pyrazolo[4,3-b]pyridine 6-(2-methylsulfanylnaphthalen-1-yl)-5,7-dihydropyrrolo[3,4-b]pyridine 3-(1H-benzimidazol-2-yl)propanamide (2E)-N'-[(Z)-4-aminobut-2-en-2-yl]-N,N-dimethyl-3-propan-2-ylidene-2-pyridin-2-yliminobut-4-enimidamide 2-(4-fluorophenyl)-3-[methyl(2,2,2-trichloroethoxycarbonyl)amino]propanoate 2-[4,5-bis(4-tert-butylphenyl)imidazol-1-id-2-yl]ethanol 1,5-dichloro-4-methyl-2-nitrobenzene;formic acid [1-azido-3-(4-fluorophenyl)propan-2-yl]oxymethanedithiol 4-azidooxy-2,3-dimethylbenzoic acid 4-(azidomethyl)-1,3,7-trimethoxynaphthalene N-[2,6-dimethyl-4-(1,3-oxazol-5-yl)phenyl]acetamide 1-[4,6-bis(ethenyl)-3,5-dihydro-2H-pyrazin-2-yl]-N-[(E)-1H-indol-3-ylmethylideneamino]oxymethanamine 4-(2,3,5,6,7,8-hexafluoronaphthalen-1-yl)-N,N-diphenylaniline ethane;1-(2-methoxy-5-propylphenyl)pyrazole N-(4-fluorophenyl)-N'-[3-(2H-triazol-4-ylmethoxymethyl)pyridin-4-yl]pentanediamide 6-hydroxy-5-[(2R)-3-phenyl-2-pyridin-4-ylpropanoyl]piperidin-2-one N-[5-[3-(4-thiophen-2-yl-1H-imidazo[4,5-c]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclohexanecarboxamide (4-azidooxyphenyl)methanamine 3-[(2R)-1-butanoylpyrrolidin-2-yl]-1,4-dihydro-1,2,4-triazol-5-one 1-[(4-phenylmethoxyphenyl)methyl]benzotriazole 4-[2,3-dihydroxypropyl(2-methylpropanoyl)amino]benzenesulfonic acid 2-[4-(6,7-dihydro-1H-indol-5-yl)-3,5-dimethylphenyl]acetic acid N-[(2S)-6,7-difluoro-1-phenylheptan-2-yl]-4-methylpyridine-3-carboxamide 5-[1-(3,4,5-trimethoxyphenyl)propan-2-yl]-1H-pyrazole (2-methoxy-1H-pyrrol-3-yl)-[7-[5-[5-(trifluoromethyl)pyridin-2-yl]hexanoylamino]heptyl]carbamic acid (3R)-1-[1-[4-fluoro-2-[5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]phenyl]ethenylamino]-N-methylsulfinylpiperidine-3-carboxamide 2-[(3aR,6aS)-5-(4-chlorophenyl)sulfonyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]pyrimidine 3-(3,5-ditert-butyl-4-hydroxyphenyl)benzonitrile 1-azido-2,4-bis(2-chlorophenyl)piperazine 3-(4-bromophenyl)-1,2-oxazole 3-[3-[4-[(1E)-buta-1,3-dienyl]-5-ethenyl-1H-pyrrol-2-yl]phenyl]-3-[3-oxo-4-(2-propoxyethyl)piperazin-1-yl]propanenitrile;propane 4-hydroxy-N-[[(2S,3R)-1-methyl-5-oxo-2-pyridin-3-ylpyrrolidin-3-yl]methyl]benzamide N-[1,3-dihydroxypropan-2-yl(ethoxy)phosphoryl]-3-phenylpropanamide 3-[6-[(2R)-4-benzylmorpholin-2-yl]pyridin-2-yl]pyridine-2,5-diamine 2-[(4,5-dimethyl-1H-pyrazol-3-yl)methylidene]propanedioic acid 2,5-dimethyl-4-[3-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-5-yl]phenol (2E)-1-amino-3-ethyl-6,10-dimethoxy-7-phenylmethoxy-3,4-dihydroazepino[2,1-b]quinazolin-2-one 2-[1,3-dioxo-7-(pyridin-4-ylmethoxy)isoindol-2-yl]acetic acid N-[2-(4-amino-6,7-dimethoxyquinazolin-3-ium-2-yl)ethyl]-3H-isoindole-1-carboxamide N-[1-(cyclopropanecarbonyl)azetidin-3-yl]-7-hydroxy-2,4-dimethylpyrrolo[2,3-d]pyrimidine-5-carboxamide 6-(3,5-dimethylphenyl)-1H-pyrrolo[2,3-b]pyridine (E,3R)-N-ethylsulfonyl-2-methoxy-5,5,8,8-tetramethyl-6-methylidenenon-8-enamide;1-[1-(methylamino)propyl]pyridin-4-one 4-[(4-aminophenyl)diazenyl]-2,5-diethyl-3-hydroxybenzaldehyde [7-(4,6-diphenyl-1,3,5-triazin-2-yl)-9a-methyl-2,5,8-triaza-3-azanidabicyclo[3.3.0]heptan-3-yl]boronic acid 1-[4,5-bis(ethenyl)triazolo[4,5-f][1]benzothiole-7-carbonyl]piperidine-3-carboxylic acid 1-(3,5-difluorophenyl)-4-[(Z)-2-phenylethenyl]cyclohexane-1-carboxylic acid (2S)-6-methyl-4,5-dihydro-1H-thieno[3,2-g]indazole 2,5-bis(phenylmethoxy)-N-[1-(4-pyridin-2-ylpiperazin-1-yl)propan-2-yl]benzamide 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-(1-phenylethyl)amino]benzenesulfonic acid 1-[[4-(4-methoxypyrimidin-2-yl)phenyl]methyl]piperazine 1-azidooxy-2,3,4,5,6-pentachlorobenzene 2-[[2-(dimethylamino)propanoylamino]methyl]-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-ylmethyl)benzamide;hydrochloride [1-[6-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]indol-3-yl]-[4-[2-(sulfinoamino)ethoxy]cyclohexyl]methanone [2-methoxy-5-[2-(4-morpholin-4-ylphenyl)ethenyl]benzenecarbothioyl]azanium 1-[5-(dimethylamino)-2,3,4a,10a-tetrahydroindeno[1,2-b]pyridin-2-yl]-3-(4-methoxyphenyl)propan-1-one 2,4-dichloropyrimidine-5-carboxamide;ethane 3,5-ditert-butyl-4-hydroxy-2,3,6-trimethylbenzonitrile 1-butanoyl-4-[3-(dimethylamino)propyl]-N,N-bis(2-ethoxyethyl)-2-methyl-5-naphthalen-2-ylpyrrole-3-carboxamide [4-(cyclohexylmethoxy)phenyl]-(3,6-dimethylpyrazin-2-yl)methanol 2-[(4-ethylpiperidin-1-yl)methyl]pyridine;formic acid 2-[6-[(E)-prop-1-enyl]pyridin-3-yl]oxyethanamine (3,4-dihydroxyphenyl)-(3,3,4-trimethylpiperazin-1-yl)methanone 4-(4,5-difluoro-1H-indole-2-carbonyl)-N'-hydroxypiperidine-3-carboximidamide;hydrochloride N-(2-azidoethyl)-4-[3,5-dichloro-4-[1-(4-propan-2-ylsulfonylphenyl)ethoxy]phenoxy]benzamide 5-[1-(2,6-dioxopiperidin-3-yl)-3-methylideneisoindole-4-carbonyl]hexanal;ethane 4-amino-5-methylsulfanyl-1-phenylpyrazole-3-carbonitrile;ethane (2R)-N'-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-2-hydroxy-2-tritylsulfanylbutanediamide 5-(3,4-dimethoxyphenyl)-6-[ethyl(propan-2-yl)amino]-N'-hydroxypyridine-3-carboximidamide 2-[2,4,6-tribromo-3-(3-methylbutoxy)phenyl]benzoic acid (5R)-2-(4-chloroanilino)-N-[(Z)-1H-indol-3-ylmethylideneamino]-5-phenyl-1,3-thiazole-4-carboxamide 1-[4-(3,6-dichlorocarbazol-9-yl)phenyl]-2-hydroxy-2,3-dihydropyrrol-5-amine 5-[[(2S)-1-fluoropropan-2-yl]amino]-N'-hydroxypyrazolo[1,5-a]pyrimidine-3-carboximidamide 1-(3,5-dichloro-4-methylphenyl)sulfonyl-2-ethylazetidine 2-(diaminomethylideneamino)-5-(4-methylanilino)pentanoic acid 2-[(1S)-6-chloro-3,4-dihydro-1H-isoquinoline-2-carbonyl]-8-hydroxy-9-methyl-5,7-dihydropyrido[2,3-c]azepine-6-carboxamide (2S)-N'-hydroxy-3-[[2-(1,2,4-triazol-1-ylmethoxy)phenyl]sulfonylamino]-5-(5,6,7,8-tetrahydroquinolin-4-ylsulfanyl)pentanediamide 2-[4-(1-ethylpyridin-1-ium-3-carbonyl)cyclohexa-1,5-dien-1-yl]propanedinitrile 2-(1,2,4-oxadiazol-3-yl)-6-propan-2-yloxyquinoline-5-carbonitrile (2R,3S,4R)-6-[4-chloro-3-(5-methyl-1H-pyrazol-4-yl)phenyl]-2-(hydroxymethyl)oxane-3,4-diol 6-(2,5-dimethylphenoxy)pyridine-3-sulfonamide 4-[2,6-difluoro-3-(pentylamino)benzoyl]oxybutanoic acid 4-(6,8,10-trioxodecyl)benzoic acid 3-[2,6-di(propan-2-yl)phenyl]iminopentanenitrile 1-cyclopentyl-N,5-dimethylpyrrole-3-carboxamide;2-(3,4-dimethoxyphenyl)acetamide N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-fluoro-6-(1-morpholin-4-ylethylsulfanylamino)-1-benzofuran-2-carboxamide 3,5-dichloro-2-[(3Z)-penta-1,3-dien-2-yl]pyridine (2S)-1,1,1-trifluoro-3-(5-iodoindol-1-yl)propan-2-ol N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]-5H-cyclopenta[b]pyridine-7-carboxamide 2-[(1-aminocyclohexyl)methylamino]-6,7,8-trihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxylic acid;dihydrochloride 2-chloro-5-[(1-methylcyclohexanecarbonyl)amino]-N-pyridin-3-ylbenzamide 1-phenylmethoxy-2,3-dihydroindole;hydrochloride 1-ethyl-2,6-dimethoxy-4-(3-methoxyphenyl)sulfanylbenzene 5-[(3S)-4-azidobutyl]-3-tert-butylsulfonyl-2,6,7,11b-tetrahydropyrazolo[1,5-d][1,4]benzoxazepine [4-(aminomethyl)phenyl]-[(2R,3S)-2-benzyl-3-methylpiperidin-1-yl]methanone N-cyclohexyl-2-[4-(3-methoxyphenyl)piperazine-1-carbonyl]iminochromene-6-sulfonamide 2-(1,3,4,5,6,7,8a-octahydroisoquinoline-2-carbonyl)-4-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carboxylic acid 6-(4-azidooxyphenoxy)-N,2,3-trimethylaniline 2-[3,4,5-trifluoro-6-(3-fluorophenyl)pyridin-2-yl]phenol 3-butyl-4,6-dimethoxypyridine-2-carboxylic acid 6-methoxy-N'-phenylmethoxypyridine-2-carboximidamide 3-methyl-1-[4-[(2R)-6-(oxan-4-ylsulfonyl)hexan-2-yl]phenyl]butan-1-one N-[3-(diethylamino)-2,4-difluorophenyl]-3-(1,3-dioxoisoindol-2-yl)piperidine-2-carboxamide 5-[3,4-bis(ethenyl)phenyl]pentaleno[2,1-b]thiophene ethane;1-[4-(3-ethylsulfonyl-5-fluorophenyl)-2-methoxyphenyl]-N'-methylpropane-1,3-diamine 1-[5-(3-azidooxyphenyl)furan-2-yl]-N,N',N'-trimethylethane-1,2-diamine 3-[(1Z)-buta-1,3-dienyl]-6-methylidenecyclohexa-2,4-diene-1-carboximidamide;[(E)-2-phenylethenyl]benzene 1-[3-[2-(5,6-dimethylpyrimidin-4-yl)hydrazinyl]propyl]indole 2-[(4Z,6E)-7-(4-methylphenyl)hepta-1,4,6-trien-3-yl]-5-phenylthiophene 1-[6-ethyl-5-(2,4,6-trifluoroanilino)pyridine-3-carbonyl]piperidine-4-carboxylic acid 4-N,4-N-diethylquinazoline-2,4-diamine 2-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]-N,2-dimethylpropanamide 3-amino-4-cyano-5-[1-(2,4-dichlorophenyl)pyrazol-4-yl]-1H-pyrrole-2-carboxamide 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxy-1H-indole 2-[3,5-dichloro-N-(3-methylbut-2-enyl)anilino]acetic acid 2-[4-[6-(1H-indazole-3-carbonyl)pyrimidin-4-yl]piperazin-1-yl]pyridine-3-carboxylic acid 4-chloro-5-[2-(1,3-dioxoisoindol-2-yl)ethoxy]pyrimidine-2-carboxylic acid 2-[7,8-dimethyl-5-[(E)-2-pyridin-3-ylethenyl]quinolin-6-yl]propan-2-ol 4-(2,4-difluoro-3-propan-2-ylphenyl)butan-1-ol 2-(4-butylphenyl)-1,3,5-trifluorobenzene;ethane 3-fluoro-5-methylbenzenesulfonic acid;4-[(Z)-1-iminobut-2-en-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 2-[[5,6-bis(4-chlorophenyl)pyridazine-3-carbonyl]amino]acetic acid 7-fluoro-6,12-dithiapentacyclo[11.8.0.02,11.05,10.016,21]henicosa-1(13),3,5(10),7,14,16(21),17,19-octaene (1S,2R)-N-[[6-(diethylaminomethylsulfanyl)pyridin-3-yl]methoxymethyl]-2-phenylcyclopropane-1-carboxamide N-(6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl)-5-methoxypyridine-2-carboxamide ethane;2-(4-propylphenyl)-5,6-dihydro-1H-indole 2-[(3S,4R)-4-azido-3-methoxypiperidin-1-yl]-5-chloropyrimidine 2-amino-4-[(1R)-1-(7H-pyrrolo[3,2-d]pyrimidin-4-ylamino)ethyl]benzenethiol [5-(2,3-difluorophenyl)sulfanyl-2H-triazol-4-yl]methylhydrazine 2-[4-azido-3-(4-chlorophenyl)pyrazol-1-yl]ethanol (3R)-4,4,4-trifluoro-N'-[7-(methylamino)-8-oxooctyl]-2,3-diphenylbutanimidamide 3-[(4-chlorophenyl)methyl]-5-propan-2-yl-1,3,4-thiadiazol-2-one 2-cyclopropyl-N-[4-(4-ethoxyphenoxy)butyl]pyrimidine-5-carboxamide N-(2,3-dihydro-1H-inden-5-yl)-4-[(9S)-7-(4-methoxyphenyl)-6,6a-dihydrothieno[3,2-d]pyrimidin-4-yl]piperazine-1-carboxamide 2-benzylsulfanyl-4-(trifluoromethoxy)benzoic acid (Z)-2-[(Z,1E)-1-[3-(dimethylamino)propoxyimino]but-2-en-2-yl]-4-methylidene-N-[4-[6-methyl-5-(morpholine-4-carbonyl)pyridin-3-yl]-5-(trifluoromethyl)pyrimidin-2-yl]hexa-2,5-dienamide 6-fluoro-N-[1-methyl-5-(2,4,6-trifluoroanilino)pyrazol-3-yl]sulfonyl-1H-benzimidazole-2-carboxamide 4-ethoxy-3,5-difluoro-N'-hydroxypyridine-2-carboximidamide N-[5-(methoxyamino)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]-3-phenylpropanamide N-[2-(2,5-dimethylphenoxy)ethyl]pyridine-4-carboxamide 2-(1,3-benzodioxol-5-ylmethylamino)-4-[5-(1H-pyrazol-4-yl)furan-2-yl]-1H-pyrimidin-6-one N-(4,4-difluorocyclohexyl)-2-methoxypyridine-3-sulfonamide 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]acetamide 4-hydroxy-3-methoxy-N-[(2S)-6-oxopiperidin-2-yl]benzamide 2-methylsulfanyl-4-[3-(thiophen-2-ylmethylidene)cyclohexyl]furan N-[(1R)-3-[5-(2,6-difluoro-4-iodobenzoyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-3-yl]cyclohexyl]acetamide 2-(5,6-diethoxypyridin-3-yl)-7-fluoro-1-[2-(4-fluorophenyl)ethyl]pyrrolo[3,2-c]pyridine 1-[3-(6,7-dihydropyrrolo[2,3-d]pyrimidine-5-carbonyl)pyridin-2-yl]ethanesulfonic acid (NZ)-N-[1-amino-2-[[5-methyl-6-(6-methylpyridazin-3-yl)pyridin-3-yl]oxymethyl]piperidin-4-ylidene]hydroxylamine 2-amino-3-(4-bromophenyl)propanamide;1-(2,5-difluoro-4-methylsulfanylphenyl)piperazine 2-[4-(dimethylamino)phenyl]-7-fluoro-3H-quinazolin-4-one 2-(4,6-dimethoxypyrimidin-5-yl)-N-[2-(3-fluorophenyl)ethyl]sulfonylacetamide [2-amino-5-fluoro-6-[(4-fluorophenyl)methyl]pyrimidin-4-yl]azanium (NE)-N-[1-amino-3,5-bis(4-methylphenyl)-7H-pyrrolo[2,3-b]pyrazin-2-ylidene]hydroxylamine 3-[5,7-dichloro-2-(4-propan-2-ylsulfanylphenyl)benzimidazol-1-yl]-N'-hydroxypropanehydrazide 3,5-dichloro-6-(trifluoromethyl)pyridine-2-carboxylic acid 2-fluoro-1-(4,5,6,7-tetrahydro-2H-[1]benzothiolo[2,3-d]pyrimidin-1-yl)ethanone 3,4-bis(methylsulfanyl)benzenesulfonate 4-N-[2-[2,6-difluoro-3-(1-piperidin-4-ylethenoxy)anilino]pyrimidin-5-yl]-2-N-(oxan-4-yl)quinazoline-2,4-diamine 1,2-difluoro-4-isothiocyanatoiodanuidylbenzene 2-[3-[4,5-bis(ethenyl)imidazol-1-yl]phenyl]-1H-benzimidazole N-[2-[4-(hydroxycarbamoyl)phenyl]ethyl]-2,3-dihydro-1H-indene-5-carboxamide 2-methyl-2,3-dihydrothiopyrano[2,3-b]quinoline 2-tert-butyl-N-[1-(4-fluorophenyl)-3-[2-methoxy-4-[3-[methyl(methylamino)amino]propoxy]phenyl]imidazo[1,5-a]pyrazin-8-yl]-N-methylsulfanylpyridine-4-carboxamide 6-[4-bromo-2,5-dimethyl-N-(1-phenylethyl)anilino]-4-hydroxynaphthalene-2-sulfonic acid (2S)-6-azido-4,7-dimethyl-2H-chromene 4-amino-N',1-dimethylindole-6-carboximidamide [4-[3-[2,6-dichloro-4-(1,1,2,2-tetrafluoroethoxy)benzoyl]indole-1-carbonyl]piperazin-1-yl]-(2H-triazol-4-yl)methanone 1-[4-[4-[2-(3,4-difluorophenyl)cyclopropyl]-6-hydroxyquinolin-7-yl]-2-methoxyphenyl]-3-ethylurea 4-(3,5-dimethylphenyl)-1H-1,2,4-triazol-5-one 2-[5-methoxycarbonyl-1-(6-oxo-4,5-dihydro-3H-pyridazin-3-yl)indol-3-yl]acetic acid (6-chloropyridazin-4-yl)-[4-fluoro-3,5-bis(trifluoromethoxy)phenyl]methanone 1,3-dimethoxy-2-[(4E)-5,5,8,8-tetramethylundeca-1,4-dien-3-yl]benzene 2-[4-(3,6-dimethylpyrazine-2-carbonyl)-1,4-diazepan-1-yl]-N-phenylpropanamide 3-methylsulfonylnaphthalene-2,7-diamine (2S)-2-[3,5-difluoro-4-[6-[2-(5,6,7-trifluoronaphthalen-2-yl)ethynyl]naphthalen-2-yl]phenyl]-4,5-dimethoxyoxane N-[(E)-1-[5-(4,6-diphenyl-1,3,5-triazin-2-yl)cyclohexa-2,4-dien-1-yl]ethylideneamino]-N'-methylbenzenecarboximidamide N-[2,6-difluoro-3-(methylcarbamoyl)phenyl]piperidine-4-carboxamide ethane;7-methyl-1,9-dihydroindeno[2,3-c]pyridine (4Z)-2,3-diphenyl-5-propan-2-yliminohepta-4,6-dienoic acid 4-[(1S)-6-fluoro-2,3-dihydro-1H-inden-1-yl]-5-hydroxy-7,8-dimethoxychromen-2-one N-[2,3,6-trifluoro-4-(3-pyridin-3-ylimidazo[1,5-a]pyrazin-8-yl)phenoxy]acetamide (4-methoxyphenyl)-[5-[3-(1H-pyrrol-2-yl)propanoyl]-1,3,6,6a-tetrahydrocyclopenta[c]furan-3a-yl]methanone 3-ethenyl-N'-(7-methoxyquinazolin-4-yl)-1-phenylbut-2-ene-1,4-diimine (4R)-3,4-dichloro-6-fluoro-5-iodo-7,8-dihydropyrimido[5,4-b]pyrrolizine N-(6-ethenyl-1H-imidazo[4,5-b]pyridin-2-yl)formamide 7-[4,4-bis(methoxycarbonyl)piperazine-1-carbonyl]naphthalene-2-carboxylic acid 6-[(4aS,7R,8aR)-6-methyl-2-oxo-1-phenyl-4,5,7,8,8a-hexahydroimidazo[1,5-a]pyrazin-3-yl]-N-ethylpyridine-3-sulfonamide 5-[4-(2,6-difluorophenyl)cyclohexyl]-1,3,4-oxadiazol-2-amine 3-[2,6-difluoro-4-(2H-tetrazol-5-yl)phenyl]-N-(2,6-dimethoxypyridin-3-yl)quinoline-7-carboxamide 3-[4,6-bis(trichloromethyl)pyrimidin-2-yl]sulfanylpropanenitrile 2-chloro-3-(4-phenylmethoxybutyl)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-one 1-azidooxy-2,4-dichloro-3-(2,6-dimethylphenoxy)benzene (5Z)-3-[2-(dimethylamino)ethyl]-5-[(7,8-dimethyl-1,4-dihydroquinoxalin-5-yl)methylidene]-1,3-thiazolidine-2,4-dione (E)-N-[[4-chloro-3-[6-oxo-1-(2,4,6-trimethylphenyl)pyridazin-3-yl]phenyl]methyl]but-2-enamide 2-amino-4,5-bis(ethenyl)naphthalene-1,3,6-tricarbonitrile 2-(4-amino-5-fluoropyridin-3-yl)-1,6-naphthyridine-8-carboxamide 6-methyliodanuidyl-3H-1,3-benzoxazol-2-one 5-(2,3-dihydro-1H-inden-2-yl)-3-(4-propan-2-yloxyphenyl)-6,7,8,9-tetrahydroimidazo[1,2-a]quinazoline 2-(1,3-benzoxazol-4-yloxy)acetate 2-[4-(1-azidoethyl)phenoxy]ethanol 1-cyclopropyl-2-fluoro-4-[4-(trifluoromethyl)phenyl]benzene N-(3,4-difluorophenyl)-2-hydroxyethanesulfonamide 4-(3-azido-2,6-difluorophenyl)pyridine 1-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]ethanamine [1-(2,4-dichlorophenyl)-2-oxopiperidin-3-yl]urea 3-chloro-6,7-dimethoxy-5-nitroquinoline N'-[(E)-1,3-bis(4-methoxyphenyl)propylideneamino]ethane-1,2-diamine 6-(2-cyanopropan-2-yl)-4H-1,3-benzodioxine-8-carboxylic acid N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-(2,3-dimethoxyphenyl)-5-oxopyrrolidine-2-carboxamide 2,3-difluoro-1H-anthracene-9,10-dione 2-[3-methylbutyl(nonanoyl)amino]benzoic acid (7R)-N,4,8-trimethyl-2-[[1-[3-(trifluoromethoxy)phenyl]pyrazol-4-yl]amino]-5,7-dihydropteridin-6-imine (2S,4R)-1-[[2-(3-chlorophenoxy)acetyl]amino]-N-[(6-methoxypyridin-2-yl)methyl]-N,2-dimethylpiperidine-4-carboxamide 4-[[3-[(2-bromophenyl)methoxy]phenyl]methyl]morpholine 4-(aminomethyl)-2-[1-methoxypropan-2-yl(methyl)amino]-1H-pyrimidin-6-one 6-methyl-1,5-diphenylspiro[2H-indole-3,4'-cyclohexa-2,5-diene] 1-[3-fluoro-4-(trifluoromethyl)phenyl]-N,2,5-trimethylpyrazole-3-carboxamide (E)-2-cyclohexa-1,5-dien-3-yn-1-ylsulfanyl-N-[4-fluoro-3-(trifluoromethoxy)phenyl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide 1-methylsulfonyl-5-(trifluoromethyl)indole 5-[2,3-dihydrofuran-2-ylmethoxy(phenyl)methyl]tetrazolo[1,5-a]pyridine (2S)-5-[benzyl(propanoyl)amino]-N-[(2R,3S)-1-methoxy-4-oxo-3-phenylbutan-2-yl]-N'-methylidenepyrrolidine-2-carboximidamide 1,2-dihydroxy-5-methoxyxanthen-9-one ethane;2-methyl-5,7-dihydrofuro[3,4-d]pyrimidine;N-methyl-1-(1H-pyrazol-5-yl)cyclopentan-1-amine N-[1-(1,3,4-thiadiazol-2-yl)piperidin-3-yl]spiro[3.3]heptane-6-carboxamide (1R)-1,2,3,4-tetrahydroisoquinoline;dihydrochloride 2-[5,6-bis(ethenyl)pyridin-3-yl]-N-[5-tert-butyl-2-methoxy-3-(methanesulfonamido)phenyl]acetamide 2-(1,2-dihydronaphthalen-1-yl)-6-methoxybenzene-1,4-dicarbonitrile N-[1-(4-fluorophenyl)sulfonyl-3,3a,5,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-7-yl]-4-methoxybenzamide 5-methyl-3-[1-(oxan-4-yl)piperidin-4-yl]-1,2,4-oxadiazole 5-[2-(3,4-dichlorophenyl)ethyl]-N'-hydroxypyridine-2-carboximidamide N-[1-cyclohexyl-2-(2,4-difluorophenyl)ethyl]-3-[6-methoxy-5-(trifluoromethyl)pyridin-3-yl]sulfanyl-N-methylpropanamide N-(2,6-dichloro-4-nitrophenyl)-3-pyridin-3-ylbutanamide 1-(2-chloroethyl)-3,5-bis[(4-fluorophenyl)methoxy]benzene 1-(diethoxyphosphorylmethyl)triazole 5-ethenyl-3-(1,1,2,3,3-pentafluoropropoxy)pyridin-2-amine 4-[[2,5-difluoro-3-(1-methylsulfonylpiperidin-4-yl)oxyphenyl]methylamino]quinazoline-8-carboxylic acid 6-chloro-2-[(2,4-dichlorophenyl)methyl]-4-fluoro-3H-isoindol-1-one (4E,5Z)-6-[3-chloro-2-(3-chlorophenyl)-1-hydroxypropyl]imino-4-ethenyl-8-hydroxy-9,9-dimethoxy-3H-azocine-2,7-dione 2,3-bis(ethenyl)-1-methylideneindene;ethane 7-(3,4-dichlorophenyl)-N-(2-fluoro-5-methoxyphenyl)-5-methyl-2-[(1S)-1-methyl-2,3-dihydro-1H-inden-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine (1R)-2,3,4,5-tetrahydro-1H-3-benzazepine-7-carboxylic acid 2-[[1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]pyrrolidin-2-yl]methoxy]pyrazine (2S,3R)-N-[4-[3-(acetamidomethyl)phenyl]butyl]-1-cyclohexa-1,5-dien-1-yl-2-methoxypiperidine-3-carboxamide N'-(3,5-difluoro-4-isothiocyanatophenyl)-N,N-diethylmethanimidamide (1R)-N,3,6-trimethyl-2-propan-2-yloxy-1H-inden-1-amine 1-[(3R,5S)-4-benzyl-3-propan-2-yl-3,5-dihydro-2H-1,4-oxazepine-5-carbonyl]pyrazole-4-carboxylic acid 6-[(4-azidophenyl)methylamino]-5-bromo-2H-1,8-naphthyridine-3-carboxylic acid 1-[(4-ethenyl-2,3,5,6-tetrafluorophenyl)methoxy]-4-fluoro-2,3-dihydro-1H-indene 2-[4-(1,3-benzodioxol-5-yl)butanoylamino]acetic acid 1-(6,7,8,9-tetrahydrodibenzofuran-3-yl)-9H-fluorene 4-(2-azidoethyl)-5,6,7-trimethoxychromen-2-one (2S)-1-[4-[(3,5-dichloropyridine-4-carbonyl)amino]benzoyl]pyrrolidine-2-carboxylic acid N-azido-5-methyl-4,6-diphenylpyrimidine-2-carboxamide 4-[[1-amino-2-oxo-3-(3,5,6,7-tetrahydropyrrolo[3,4-d]pyrimidin-4-yloxy)propylidene]amino]benzoic acid 5-[5-azido-2-(4,6-dimethylpyrimidin-2-yl)phenyl]-1,3-oxazole 2-methyl-1-[(2Z,4E)-3,5,7,9,10-pentamethylideneundeca-2,4-dienoxy]naphthalene 2-[3,5-bis(trifluoromethyl)phenyl]-N-[7-[1-(cyanoamino)cyclopropyl]quinolin-4-yl]acetamide 5-cyclopropyl-3-fluoro-N-[(2R,4S)-2-methylpiperidin-4-yl]pyridine-2-carboxamide N-methyl-N-[1-(4-phenylsulfanyloxyphenyl)ethylideneamino]benzenesulfonamide N-[4-chloro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-2-cyclopentylacetamide 1-benzyl-6-(cyclopropylmethyl)-5,8-dihydroxy-4H-3,1-benzothiazin-2-one 6-butyl-1,2,3-trimethoxynaphthalene 2-[(2E)-2-[(E,3Z)-3-ethylidenehepta-4,6-dien-1-ynyl]penta-2,4-dienoxy]-5-propan-2-yl-3H-pyrano[2,3-d]pyrimidine-4,7-dione 3-[(4S)-4-methoxy-6-oxopiperidine-2-carbonyl]benzonitrile 3-(5,6-dihydrophenanthridin-9-yl)phenol 3-[4-(5-methylpyridin-2-yl)oxyphenoxy]azetidine;pentane 1-[4,6-bis(2-chlorophenyl)-3-cyano-5-(trifluoromethyl)pyridin-2-yl]-3-diazourea N-(3-hydroxypropyl)-2,4,6-trimethyl-N-(3-nitrophenyl)benzenesulfonamide 3,4-difluoro-N-[(1S)-2-oxocyclohexyl]benzenesulfonamide 4-[(3-ethynylphenyl)methylamino]thieno[2,3-d]pyrimidine-6-carboxylic acid 6-[2,4-bis(trifluoromethyl)phenyl]-5-(3,4-dichlorophenyl)spiro[3,4-dihydropyrrolo[1,2-a]pyrazine-1,4'-piperidine] ethane;5-methyl-1H-indole;N-(3-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 3-[[2,5-dioxopyrrol-1-yl(phenyl)methylidene]amino]oxypropanamide 2-(4-methylpyrimidin-5-yl)-6-oxo-1H-pyrimidine-4-carboxylic acid 4-[2,3-dihydroxypropyl(ethenylsulfonyl)amino]benzenesulfonic acid 1-azido-2,3,5,6-tetramethylindole 2-(3,5-dimethylpyrazol-1-yl)-N-[[6-(trifluoromethyl)pyridine-3-carbonyl]amino]acetamide 2-[(1S)-6-chloro-4-fluoro-1H-inden-1-yl]quinoline 4-[1,3-bis(2,6-dimethylphenyl)imidazol-1-ium-2-yl]benzene-1,2,3-triol N-[2-[7-(1-aminopropyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl]ethyl]-3-[2-chloro-4-fluoro-5-methoxy-3-(trifluoromethyl)phenyl]propanamide 3-methyl-2,4,9,10-tetrahydro-1H-pyrimido[4,5-c]isoquinoline 2-ethylsulfonyl-5,6-dihydroimidazo[2,1-b][1,3]thiazole N'-[3-[(4-methyl-1,2,5-oxadiazol-3-yl)methoxy]phenyl]-N-(oxolan-2-ylmethyl)oxamide 2,3-dichloroanthracene 2-(2,4-difluorophenyl)-1-[4-(4-fluorophenoxy)piperidin-1-yl]ethanone 2-cycloheptyloxybenzoate 3-[3-(2,5-difluorophenyl)phenyl]-7-N-pyridin-4-yl-9H-carbazole-1,7-dicarboximidamide 6-fluoro-2-[4-[(3S)-3,5,7,8-tetrahydroxyoctoxy]phenyl]indazole-3-carboxylic acid 7-[2-(cyclohexylmethoxy)phenyl]-5-methylidenehepta-1,6-diene-3-thione 3-[(1-benzylpiperidin-4-yl)methoxy]-N-[(E)-(2,5-dichlorophenyl)methylideneamino]pyrazine-2-carboxamide;2,2,2-trifluoroacetic acid N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-6-pyrrolidin-1-ylpyrimidine-4-carboxamide;2,2,2-trifluoroacetic acid 2-(diethylamino)-7-methyl-3-(2,4,6-trifluorophenyl)pyrido[1,2-a]pyrimidin-4-one 1-[3,4,5-trimethoxy-N-(2,2,6,6-tetramethylpiperidin-4-yl)anilino]-3H-2,1-benzoxaborole 2-chloro-4,5,6-trifluoro-3-(1-methylindol-3-yl)phenol 1-[(5E)-1,2-difluoro-4-methylidenenona-1,5-dien-3-yl]sulfonyl-4-(trifluoromethoxy)benzene [7-(4-chlorophenyl)-5-methyl-2-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-6-yl]-[4-[(5R)-5-hydroxycyclohepta-1,3-dien-1-yl]piperidin-1-yl]methanone 1-[(4R)-4,7-dimethoxy-3-oxoheptyl]indole-2-carboxylic acid 2-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)piperidin-2-yl]acetic acid 5-[(6,7-dimethoxyquinolin-4-yl)amino]-N-[1-(6-methylpyridazin-3-yl)azetidin-3-yl]pyridine-2-carboxamide N-[3-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]oxolane-3-carboxamide 5-methyl-3-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)imidazol-2-yl]pyridin-2-amine 4-[(2S)-6-amino-1,2,3,5-tetrahydropyrido[3,2-b]indole-8-carbonyl]benzonitrile N-[[4-(6,7-dimethoxyquinolin-4-yl)oxycyclohexa-2,4-dien-1-ylidene]amino]-3-fluorobenzamide N-cyclohexyl-2,6-dioxo-3H-purine-9-carboxamide 2-azido-4-chloro-5-(2,6-dimethoxyphenyl)pyrimidine (5Z)-2-cyclohexylimino-5-[(3,4-dichlorophenyl)methylidene]imidazolidin-4-one N-[4-(2,3-dichlorophenyl)-5-(4-methoxyphenyl)-1,3-thiazol-2-yl]acetamide 6-azidooxy-2,3-dichlorophenol 4-(2-aminoethyl)-N,3,5-triphenylaniline [2-amino-5-[6-(trifluoromethyl)pyridin-3-yl]phenyl]-oxoazanium 5-[2,6-dimethyl-4-(trifluoromethoxy)phenyl]-N-[3-(2-oxopropanoylamino)cyclohexyl]-1,3,4-oxadiazole-2-carboxamide 1-[3-(difluoromethyl)phenyl]-2,5-bis(trifluoromethyl)benzene 3-[(2R)-2,6-dimethylmorpholine-4-carbonyl]-7-fluoro-1H-quinolin-2-one 1-methyl-3-[2-(4-nitrophenyl)ethyl]benzene ethane;(E)-3-methyl-N'-[2-methyl-5-(methylideneamino)phenyl]but-1-ene-1,4-diamine 2-[N-(4-chlorobutyl)-4-sulfamoylanilino]acetic acid (1S)-3-methoxyiminocyclopentane-1,2-diolate;4-pyridin-2-ylpyridine;ruthenium(2+);triphenylphosphanium 6-methyl-N-(4-methylphenyl)-7,8a-dihydroquinoline-3-carboxamide 1-(2-methoxyphenyl)pentane-1,3-diol 5-butyl-3,6-difluoro-2-[4-(4-propylcyclohexyl)phenyl]naphthalene 1-(3,5-dimethylpiperidin-4-yl)-2-[5-(1H-indol-2-yl)imidazo[1,2-a]pyridin-6-yl]ethanone;3-methylsulfanylpropanoic acid 1-[(Z)-3-cyclopropyl-2-fluoro-4-oxopent-2-enoyl]-N-phenylpiperidine-4-carboxamide N-[4-amino-6-methyl-2-(1,3-thiazole-5-carbonyl)pyrimidin-5-yl]formamide 5-[3-(benzenesulfonyl)phenyl]sulfanylpyrimidine-2,4-diamine 2,3-dimethoxybenzo[h]quinazolin-4-one 6-[[4-fluoro-1-(4-methylsulfonylphenyl)-2H-pyridin-3-yl]sulfanyl]isoquinoline 3-azido-N,N-dimethyl-6,7-dihydropyrrolo[2,1-c][1,4]oxazine-1-carboxamide 1-azido-2-hexylanthracene 2-[5-amino-1-(6-methoxypyridin-3-yl)triazol-4-yl]propan-2-ol 2-N-cyclopropyl-4-N-[1-(5-fluoropyrimidin-2-yl)azetidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-2,4-diamine (3R)-1,4-dimethyl-3-[7-(oxan-2-yloxymethyl)-9H-pyrido[2,3-b]indole-5-carbonyl]piperazin-2-one (2R)-1-[2-acetyl-3-[3,5-dimethoxy-4-(7-methyl-6-oxoheptoxy)phenyl]benzimidazol-5-yl]-N,2-diethylpiperidine-2-carboxamide (E,5R)-N-ethenyl-5-[7-methoxy-2-oxo-3-[4-(trifluoromethoxy)phenyl]benzimidazol-1-yl]-6-iminohex-2-ene-2-sulfonamide 4-[6-[3,5-bis(trifluoromethyl)phenyl]-8-chloroimidazo[1,2-b]pyridazin-2-yl]piperazine-1-carboxylate 2-[1-[(4R)-2,5-dioxoimidazolidin-4-yl]piperidin-3-yl]isoindole-1,3-dione N-[5-(4-methoxyphenyl)-1,3,4-thiadiazol-2-yl]imidazo[1,2-b]pyridazine-6-carboxamide 4-[5,6-diamino-4-(3,4-difluorophenyl)pyrimidin-2-yl]benzene-1,2-diol 2-[6-(diethylamino)pyridin-3-yl]-4,5-dihydro-1H-imidazole-4-carboxylic acid 2-[2,3,4,5-tetrafluoro-6-(1H-indol-3-yl)anilino]ethanol (E)-3-[5-methoxycarbonyl-1-(pyridine-4-carbonyl)pyrrol-2-yl]prop-2-enoic acid (7-methylbenzo[g][1,3]benzoxazol-2-yl)methanol 6-(dimethylamino)-4-N,5-N,8-triethyl-3H-phenazine-2,4-diamine 6-[(3R)-1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl]oxy-2,3-dihydrofuro[3,2-b]pyridine;2,2,2-trifluoroacetic acid N-[4-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazole-2-carbonyl)phenyl]cyclopropanecarboxamide (2S,5R)-N-[3-fluoro-4-[6-methoxy-7-(piperidine-1-carbonyl)quinolin-4-yl]oxyphenyl]-2-nitro-3-oxo-4-sulfanylidenemorpholine-5-carboxamide 1-[(2R)-3-(3,4-dihydro-1H-isoquinolin-2-yl)-2-hydroxypropyl]-3-(2-ethoxypyridin-3-yl)sulfonylurea 3-[1,2-bis(4-chlorophenyl)ethyl]imidazole-4-carboxylic acid [4-(dimethylamino)phenyl]-[3-[2-ethoxyethyl(ethyl)carbamoyl]phenyl]azanium 4-(5-pyridin-2-ylthiophen-3-yl)benzenesulfonamide 2-cyclopentyl-N-[5-[3-(4-piperidin-1-yl-1H-pyrrolo[2,3-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]acetamide 2-[N-(1,3-thiazol-5-yl)anilino]acetonitrile N-[2-chloro-4-fluoro-5-(1,3,5-trimethylpyrazol-4-yl)phenyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboxamide N-(2,3-dihydroxypropyl)-2-methoxy-6-methyl-4-[5-(1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]benzamide 5-bromo-3-(1H-indol-2-yl)-4-methoxy-6-nitropyridine-2-carboxamide N-[4-[4-(3,5-dichlorophenyl)-2H-pyridin-1-yl]butyl]-2-[2-(hydroxymethyl)piperidine-1-carbonyl]benzamide 1-[6-(2,4-dimethylpentanoyl)pyridin-2-yl]prop-2-en-1-one 4-(3-azidopropyl)-2,5-dimethoxypyridine 2-[(4R,7S)-3-methyl-5-oxo-1-pyridin-3-yl-6,7,8,9-tetrahydro-4H-pyrazolo[3,4-b]quinolin-4-yl]benzoic acid 2-[(3R)-1-[5-bromo-6-(3-fluorophenyl)pyridine-2-carbonyl]pyrrolidin-3-yl]-4-cyclopropyl-1H-pyrimidin-6-one 3-chloro-N,N-dimethylbutanamide;ethane N-[[1-(4-ethylphenyl)cyclopentanecarbonyl]carbamoyl]acetamide 4-[1-[(E)-2-methylpent-3-enoyl]piperidin-4-yl]-2H-phthalazin-1-one 1-[4-(2-hydroxyethyl)phenyl]-3,3-dimethylazetidine-2,5-dione [(2S,4R)-2-(5-carboxyfuran-3-yl)-4-methoxypyrrolidin-1-yl]oxidanium 3-chloro-2-[3-(difluoromethoxy)phenyl]-4H-thieno[3,2-b]pyrrole;N-hydroxyformamide 4-(5,7-dihydrocyclopenta[d]pyrimidin-6-yl)aniline N-[5-(2,4-dimethylphenyl)pyridin-3-yl]-1H-indole-6-carboxamide N-azido-2,2,6,7-tetramethyl-4H-3,1-benzothiazin-8-amine 2-[4-bromo-N-(3,5-dichlorophenyl)anilino]acetonitrile 2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)oxyethanesulfonic acid 2-(7-bromospiro[1H-indole-3,4'-piperidine]-5-yl)ethanol 4-(2-chlorophenyl)-1,3-dimethyl-5-oxo-7H-pyrazolo[3,4-b]pyridine-6-carboxylic acid 4-amino-2-(trifluoromethyl)chromene-6-carboxylic acid;ethane 1-[3,5-bis(trifluoromethyl)phenyl]-N-(cyclopenten-1-yloxy)propan-2-imine 3-(1-cycloheptylethoxy)benzenethiol (2R)-3-[5-amino-1-(4-fluorophenyl)triazol-4-yl]propane-1,2-diol 1,3-dimethyl-2H-pyridine;ethane;4-[4-(2-hydroxyphenyl)-6-morpholin-4-ylpyridin-3-yl]benzonitrile 2-[5-carbamoyl-9-[(3-phenylphenyl)methyl]carbazol-4-yl]oxyacetic acid [4-amino-2-(cyclopentylcarbamoyl)pyridin-3-yl]-[5-(aminomethyl)-1H-pyrrol-3-yl]azanium 2-amino-9-[(4-methylphenyl)methyl]-7,8-dihydropyrimido[1,2-a]pyrimidin-6-one 4-[5-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl)pyridin-2-yl]benzoic acid;dihydrochloride N-[6-(diethylamino)pyridin-3-yl]-2-methoxyquinoline-8-carboxamide 3-[2-hydroxyethyl(methyl)amino]-1,5-diphenylpentan-3-ol N-(2,3-dioxopiperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidine-5-carboxamide 1-[(E)-2,3-dimethylbut-1-enoxy]-4-[[4-[(2E,6Z)-octa-2,6-dien-3-yl]cyclohexyl]methoxy]benzene 1-[(3,4-difluorophenyl)methylamino]-3-propan-2-ylthiourea [(E)-3-cyclohexa-1,5-dien-1-ylprop-2-enoyl]-(4-hydroxyphenyl)azanium [3-(4,5-dihydrobenzotriazol-2-yl)naphthalen-1-yl]-[4-(2,6-diphenylpyrimidin-4-yl)phenyl]methanone 2-(2-bromoethenyl)-4,5-ditert-butyl-1H-pyrrole 2-(4-methylpiperazin-1-ium-1-ylidene)-3H-benzo[g]quinazoline 2-(3,5-dichlorophenyl)-1-(4-methylpyrrolidin-3-yl)ethanone 5-[4-[6-ethyl-8-fluoro-7-(2-fluorophenyl)naphthalene-1-carbonyl]-3,3-dimethylpiperazin-1-yl]pyridine-2-carbonitrile 4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-ethylhexane-2-sulfinamide 4-[5-methyl-3,6-bis(2-oxobutanoyl)naphthalen-1-yl]oxybenzonitrile N-[2,6-di(propan-2-yl)phenyl]-4-methylpentanamide N-cyclohexyl-4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-6-[(2E,4Z)-5-ethoxypenta-2,4-dien-2-yl]pyrimidine-2-carboxamide 6-(2,4-dimethylpentan-3-ylamino)pyridine-3-carbonitrile 3-[2-(4,5-dimethylcyclohexa-1,5-dien-1-yl)oxyethyl]pyridine 2-[N-(3-methylbutyl)-2,4,6-trinitroanilino]acetamide N-(3-methoxyphenyl)-4,6-dinitrodibenzofuran-1-carboxamide 2-(5,7-difluoroquinolin-3-yl)aniline 1-[(2R)-2-azidopyrrolidin-1-yl]-3-[4-methoxy-7-propan-2-yl-5-(trifluoromethyl)-1H-indol-3-yl]propan-1-one 2-[5-chloro-3,4-dimethyl-1-(methylideneamino)naphthalen-2-yl]acetic acid N-[4-methyl-3-(propylamino)phenyl]propanamide N-[4-[3-(cyclopropanecarbonylamino)anilino]quinolin-6-yl]-2,2-difluoroacetamide 2-[1-(5,6-dimethoxy-7-phenylmethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)piperidin-4-yl]benzonitrile 2-[5-(2,4,6-trimethylphenyl)imidazol-1-id-2-ylidene]indene-1,3-dione (3S,4R)-N'-tert-butyl-2-[1-[(5,7-difluoroquinolin-6-yl)methyl]piperidin-4-yl]-4-phenylpyrrolidine-3-carbohydrazide 4-[2,3,5-trichloro-N-(4-hydroxybutyl)anilino]butanoic acid 2-[[5-(1H-indol-3-yl)-4-(oxolan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]benzonitrile 1-methoxycarbonyl-2,3-dihydropyrrolo[2,3-c]pyridine-7-carboxylic acid 3-(1,2,5-thiadiazol-3-yl)benzoic acid 1-azidooxy-2,3,4-trimethyl-5-phenoxybenzene 1-chloro-3-(difluoromethyl)benzene;N-[2,4-difluoro-5-[5-methoxy-7-methyl-6-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]phenyl]formamide 7-[4-(5-cyclohexylpentanoyl)piperazine-1-carbonyl]chromen-2-one N-(2,3,4,5,6-pentafluorophenyl)azetidine-1-carboxamide 2-(4,5-diphenyl-1H-imidazol-2-yl)phenol N-butyl-3,6-dichloropyrazin-2-amine 2-[[[(2R)-1-aminohexan-2-yl]amino]methyl]-3H-thieno[3,2-d]pyrimidin-4-one 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-3-morpholin-4-ylpropanamide 7-(8,10-dimethylundecyl)naphtho[2,3-c]isochromene 2,3-dimethylbutane;3,5-dimethoxybenzonitrile (1R)-N-[3-(6,7-dihydroquinolin-5-yl)propyl]-1-pyridin-4-ylethanamine;hydrochloride 2-(4-cyclobutyl-1,3-thiazol-2-yl)phenol 1-(6-fluoroquinolin-4-yl)-2,3-dihydropyrrolo[2,3-b]pyridine;2-methylcyclobutane-1-thiol 2-[2-[2,5-difluoro-4-(trifluoromethyl)phenoxy]ethoxy]-7-fluoroquinoline N-[1-(4-benzylsulfanylpiperidin-1-yl)propan-2-yl]acetamide;hydrochloride 2-[6-(4-bromoanilino)-3,5-dicyano-4-ethylpyridin-2-yl]sulfanylacetamide 5-(6-aminopyridine-3-carbonyl)-3-benzylsulfanyl-N'-hydroxy-1,2,4-triazole-1-carboximidamide;2-tert-butylpyridine 5-[3,3-dimethylbutanoyl(methyl)amino]naphthalene-2-carboxylic acid N-(7,8-dihydronaphthalen-1-ylmethoxy)formamide 2-benzyl-N-[4-(4-chlorophenyl)sulfonyl-1,3-thiazol-2-yl]-6-methoxybenzamide 1-[4-(3,5-dimethylbenzene-6-id-1-yl)but-3-yn-2-ylideneamino]-N,N'-diphenylmethanediamine;osmium(1+) (3S)-N-cyclopentyl-6-[2-hydroxyethyl(methylsulfonyl)amino]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1-(3,4-dimethoxyphenyl)-3-[4-(2,6-dioxopiperidin-3-yl)phenyl]urea 2-azido-5,8-dimethylquinoline 2-(2,6-difluorophenyl)-7-[3-hydroxypropyl(methylsulfanyl)amino]-5-iodo-3H-pyrido[2,3-d]pyrimidin-4-one 2,2-difluoro-N-[3-[4-[4-(4-morpholin-4-ylbenzoyl)-1,3-oxazol-5-yl]phenyl]pentyl]acetamide (7S)-N-benzyl-5-methyl-7-phenyl-2-piperidin-1-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 1-azidooxy-2-phenylethanesulfonic acid 5-(3,4-dichlorophenyl)-2-[[4-methyl-6-oxo-1-(2,4,6-trichlorophenyl)pyridazin-3-ylidene]methyl]pyrazole-3-carboxylic acid 4-chloro-1,2,6,8a-tetrahydrocyclopenta[c]chromene (2R)-2-[4-oxo-5-[[4-oxo-6-propan-2-yloxy-3-(2,2,2-trifluoroethylcarbamoylamino)quinazolin-7-yl]methylidene]-1,3-thiazolidin-2-yl]propanenitrile 1-(4-aminocyclohexyl)-2,5-dimethoxypyridin-4-one 2-[(3R,4S)-3-fluoro-1-[2-(1H-indol-3-yl)ethyl]piperidin-4-yl]propan-2-ol 5-azidooxy-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione 5-azido-N,6,7-trimethoxynaphthalen-2-amine 3,4-dimethyl-1-[5-(2-pyridin-2-ylethynyl)pyrimidine-2-carbonyl]imidazolidin-2-one 1-bromoimidazo[5,1-b][1,3]benzothiazol-6-amine;ethane (2R,6S)-N-[3-[1-(4-chlorophenyl)cyclopentyl]prop-1-en-2-yl]-4,7-dioxo-2-phenyl-8-(phenylmethoxymethyl)-6-pyridin-2-yloctanamide 1,2-diamino-4-[5-bromo-2-(3,5-dimethylphenoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile 5-(3,4-difluorophenyl)-2-fluoro-N'-methylsulfanylbenzohydrazide (6R)-N,2-dimethyl-4,5,6,7-tetrahydro-1,3-benzothiazole-6-sulfonamide;hydrochloride 1-[2,6-bis(trifluoromethyl)phenyl]ethanesulfonate 4-N-azido-5,6-dihydrocyclohepta[d]pyrimidine-2,4-diamine 2-(1,3-dihydroxy-4H-thieno[3,4-c]pyran-2-yl)acetic acid 7-[[(2S,4R)-1-acetyl-3,4-dihydroxypyrrolidin-2-yl]methoxy]chromen-2-one 2-[4-[(1,3-dioxoisoindol-2-yl)methyl]pyrazol-1-yl]cyclopentan-1-one ethane;3-(trifluoromethyl)imidazo[1,2-b]pyridazine N-[(1R,5S)-3-[(Z)-(4-hydroxyphenyl)methylideneamino]-6-bicyclo[3.1.0]hexanyl]pyridine-4-carboxamide 4-amino-N'-[2-(dimethylamino)ethyl]thieno[3,2-c]quinoline-7-carboximidamide N-[4-[(Z)-1-iminobut-2-en-2-yl]phenyl]prop-2-ynamide 1-[(5S,7R)-2-methyl-5-phenyl-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazol-7-yl]ethanone 3-[4-amino-3-(methyliminomethyl)phenyl]-1-azidopropan-2-ol (5R)-3,5-diethyl-1-[4-methoxy-3-(trifluoromethyl)phenyl]piperidine ethane;(5E)-2-methylidene-5-[(3-phenylphenyl)methylidene]cyclohexan-1-one 1-amino-5-cyclohexyl-6,7-difluoropyrido[2,3-d]pyrimidine-2,4-dione 2-amino-4-(3,5-dimethoxyphenyl)-6-[2-oxo-1-(piperidine-1-carbonyl)piperidin-3-yl]pyridine-3-carbonitrile 2-[4-(2,5-dioxopyrrolidine-1-carbonyl)phenyl]sulfanylbenzoic acid 6-[3-(2-methylphenyl)sulfonylpropanoyl]-3-nitro-1H-quinolin-4-one 4-[5-fluoro-2,4-dimethyl-3-(1H-pyrazol-5-yl)phenyl]morpholine 4-hydroxy-3-[(4-phenyltriazol-2-yl)methyl]benzoic acid 2,4-dinitrobenzamide;ethane 6,8-dimethoxy-4-methyl-2-[(E)-pent-3-enyl]pyrido[2,3-b]pyrazin-5-one;ethane 2-[4-[(5Z)-6,7-dihydroindol-1-yl]butyl]guanidine (E)-3-[5-tert-butyl-2-[4-(trifluoromethoxy)phenyl]pyrazol-3-yl]prop-1-en-1-ol;(3Z,4Z,5E)-4-ethenylocta-1,3,5-triene 3-chloro-5,5-dimethylcyclohexa-1,4-diene;2-[(2S)-4-(2-chlorophenyl)sulfonylmorpholin-2-yl]acetaldehyde 2-[4-(diethylamino)-2-oxo-1H-pyridine-3-carbonyl]-N-oxidobenzamide 4-(6,7-dimethylquinolin-1-ium-8-yl)oxyaniline 2-chloro-4-[6-(cyclohexylamino)imidazo[1,2-b]pyridazin-3-yl]-N-ethylaniline 3-(6-aminopurin-9-yl)-N-[5,8-bis(ethenyl)naphthalen-1-yl]propanenitrilium 1-[4-[(2S)-3,3-dimethylbutan-2-yl]phenoxy]ethanamine 2-[5-[1,3-benzoxazol-7-yl(hydroxy)methyl]pyridin-2-yl]-4-(4-cyclopropylpiperazin-1-yl)benzonitrile 1-[3-(2,2-diethoxyethyl)-5-methylfuran-2-carbonyl]piperidine-4-carboxylic acid 4-[2,3,5-tris(trifluoromethyl)phenyl]butanamide (2-butoxycarbonyl-4-chlorophenyl)-(oxan-3-ylmethyl)carbamic acid 3-[(2E)-2-ethenylpenta-2,4-dienoxy]-N'-hydroxypyrazine-2-carboximidamide (Z)-1-[(6S,11R)-11-methoxycarbonyl-7,9,12-trioxo-4-oxa-1,8-diazatricyclo[8.4.0.03,8]tetradeca-10,13-dien-13-yl]but-2-ene-1,5-disulfonic acid N-[3-[(E)-3,5-dimethylhex-2-en-2-yl]cyclopenta-1,4-dien-1-yl]-4-methoxyaniline 4-[(7S)-2,6-dimethyl-8-phenyl-5H-imidazo[1,2-a]pyrazin-3-yl]-3,5-dimethoxyphenol N-(3,4-difluorophenyl)-2,7-diazaspiro[3.5]nonane-7-sulfonamide;hydrochloride 1-[4-[(E)-2-chloro-3-[[(E,3R)-3-ethylnon-5-enoyl]amino]prop-2-enoxy]phenyl]piperidine-2-carboxylic acid 3-(5,7-difluoro-1H-indole-2-carbonyl)-4-hydroxypyrrolidine-1-carboxylic acid 2-[4,6-bis(4-methoxyphenyl)-1,3,5-triazin-2-yl]naphthalen-1-ol (6S)-10-bromo-3-ethylsulfanyl-6-thiophen-2-yl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-1-one 2-[[4-[(2,3,4,5,6-pentafluorophenyl)methyl]phenoxy]methyl]oxirane N-[(E)-(3,5-dibromo-2,4-dihydroxyphenyl)methylideneamino]benzamide 4-[3-(benzenesulfonyl)propyl]piperazine-1-carboxylic acid 1-(2,6-diethylphenyl)propane-1,3-diimine (1R)-2-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]-1-ethoxy-N-oxocyclopentane-1-carboxamide 2-methyl-3-(4-pyrrolidin-1-ylphenyl)aniline 2-[N-(2,3-dihydroxypropyl)-4-nitroanilino]octanoic acid 2-[3,5-bis(trifluoromethyl)phenyl]-N,2-dimethoxy-1-phenylethanimine 3-(2,3-dihydroxypropyl)-9H-fluoren-1-amine N-[3-[(2,4-dichlorophenyl)methylsulfonylamino]-1-bicyclo[1.1.1]pentanyl]-3-fluoro-6-(propoxymethyl)pyridine-2-carboxamide 4-[2-azido-4,6-difluoro-3-(2H-tetrazol-5-yl)phenyl]morpholine ethane;6-ethyl-2,7-dimethylthieno[3,2-f]quinoline N-(2,6-dichlorophenyl)-2-[(E)-pent-1-enyl]sulfanylacetamide 3-azido-6-methyl-2-(trifluoromethoxy)pyridine 3-methyl-5-[4-(6-pyrrolidin-1-ylpyridin-2-yl)phenyl]-2H-triazolo[4,5-b]pyrazine 6-amino-9,10-dioxoanthracene-2-sulfonic acid 5-[4,6-diamino-1-(4-fluorophenyl)pyrazolo[3,4-d]pyrimidine-3-carbonyl]pentanamide N-[3,4-bis(methoxymethoxy)phenyl]-2,3-dihydroxybenzamide (3-cyclohexyl-1,2,4-oxadiazol-5-yl)-[(7S)-2,7-dimethylazepan-1-yl]methanone N-(7,8-dihydro-5H-pyrano[3,4-b]pyridin-9-yl)-2-methoxybenzamide (2E)-4,5,6-trimethyl-2-[(4-phenylphenyl)methylidene]-1-benzofuran 1-(2,3-dihydro-1H-inden-5-yl)piperazine;hydrochloride N-[3-(4-methoxyphenyl)sulfonylpropyl]isoquinoline-5-sulfonamide ethane;6-[3-(1H-pyrrole-2-carbonylamino)azetidin-1-yl]pyridine-3-carboxylic acid [1-[3-(azidomethyl)phenyl]sulfonylpiperidin-4-yl]methanol 4-bromo-N-[(2,6-dichlorophenyl)methyl]aniline;N-[[3,5-bis(trifluoromethyl)benzenecarbothioyl]amino]propanamide 3-[3,5-bis(trifluoromethyl)phenyl]-2-cyano-2-fluoropropanamide 1,2-diamino-4-(3-fluoro-5-methoxyphenyl)-6-oxopyridine-3,5-dicarbonitrile 2-azido-4-(2,6-ditert-butylphenoxy)pyridine 2-[3,4-dimethyl-6-(5-pyrimidin-5-ylpyridin-3-yl)-2H-pyridin-1-yl]ethanol [3-(4-azidophenoxy)propyl]benzene 2-(4-tert-butylphenyl)sulfinylethanol 6-[(3,5-dichlorophenyl)methyl]-2-(trifluoromethyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-[3-(dimethylamino)propyl]formamide;methane;4-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl]morpholine N-[(Z)-4-amino-3-cyclopropylimino-1-(5-hydroxypyridin-2-yl)but-1-enyl]pyridine-3-carboxamide 2-azido-3,4,5,6-tetraethyl-1H-indole N-[2-(2,3-dihydroindol-1-yl)ethoxy]-1H-indole-2-carboxamide 3-[2-(4-benzylpiperidine-1-carbonyl)-6-chlorocyclohexa-2,4-dien-1-ylidene]propanoic acid 2-(N-ethylsulfonyl-4-methoxycarbonylanilino)propanoic acid ethane;3-methylpentane;1,2-xylene 1-[2-[4-(dimethylamino)phenyl]ethynyl]-5,7-dihydroxynaphthalene-2,3-disulfonic acid;ethane 2-methyl-1',1'-dioxospiro[7H-benzo[f]isoindole-6,3'-indole]-5-carbonitrile 3-[4,5-bis(methoxycarbonyl)piperazin-1-yl]sulfonylbenzoic acid 2-(6,7,8a,9,10,11-hexahydrobenzo[b][1]benzazepine-5-carbonyl)benzoic acid N-[4-[(2E,4Z)-hepta-2,4,6-trien-3-yl]phenyl]dibenzofuran-2-amine 4-[4-(1,3-benzodioxol-5-yl)piperazin-1-yl]-6-phenylpyrimidine N-cyclohexyl-1,5-bis[4-(dimethylamino)phenyl]pyrazole-3-carboxamide (2S)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-ethoxy-5-(2-morpholin-4-ylethylamino)-2-propan-2-yl-2,3-dihydro-1-benzofuran-7-carboxamide 1-[3,5-dichloro-4-(2-sulfanylpropoxy)phenyl]ethanol 1-[3-amino-4-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione 3-N,4-diphenyl-2H-benzotriazol-1-ium-1,3-diamine (3S,5R)-1,6-dimethyl-2-oxo-4-[4-(1,3-thiazol-2-ylamino)phenyl]-N-(4-thiophen-2-ylphenyl)piperidine-3-carboxamide 1-(1,2,3,4-tetrahydroisoquinolin-7-yl)pyrrolidine-2-carbonitrile 3-[2,3-dihydroxypropyl(3-methylbut-2-enyl)amino]phenol N-[4-(2,6-dimethylmorpholine-4-carbonyl)cyclohexa-1,5-dien-1-yl]sulfonylfuran-3-carboxamide N-[3-[(2R)-6-benzoyl-1,2,3,4-tetrahydroquinolin-2-yl]propyl]-5-bromofuran-3-carboxamide 6-(5,6,7,8-tetrahydronaphthalen-1-yloxy)pyrazine-2-carboxylic acid 2-[6-(6,7-dimethoxyquinolin-4-yl)oxypyridin-3-yl]-3H-benzimidazole-5-carboxamide (3R,5S)-7-[3-cyclopentyloxy-4-(difluoromethoxy)phenyl]sulfonyl-N-hydroxy-1-oxa-7-azaspiro[4.4]nonane-3-carboxamide 2,3-dichloropyridine;ethane 3-[4-bromo-N-(2,2-dimethoxyethyl)-2,5-dimethylanilino]-2-sulfanylidene-1,3-thiazolidin-4-one 2-benzylsulfanyl-5,6-bis(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine 1-azidooxy-2,3,4-trimethylanthracene 3-methyl-4,5,6,7,8,9-hexahydrothieno[2,3-b]quinoline 2-(4-bromophenoxy)-1,3-diphenylbenzene 6-(5-methylpyrimidin-2-yl)oxy-3,4-dihydro-1H-quinoxalin-2-one [2-hydroxy-3-[4-(6-pyridin-3-yl-2,3,4a,5-tetrahydro-1H-pyrimido[4,5-b]indol-4-yl)piperazin-1-yl]propoxy]methanol 3-[[1-(4-chlorophenyl)cyclobutyl]methyl]-2,5,6-triethoxypyrimidin-4-one 1-azidooxynaphthalene;3,7-bis(methylamino)chromen-2-one (E)-3-[4,5-bis(ethenyl)thiophen-2-yl]-N-hydroxyprop-2-enamide 1-[(3,5-difluorophenyl)methylamino]-3-(2-naphthalen-2-ylethyl)thiourea 4-azidooxy-5-fluoro-2-(trifluoromethyl)pyrimidine 4-fluoro-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]benzoic acid 1-[1-(4-amino-2,3-dichlorophenyl)ethyl]pyrrolidine-3-carboxamide 5-[(5-amino-3,6-dihydro-2H-pyridine-1-carbonyl)amino]-N-ethylnaphthalene-1-carboxamide (4S,5R)-4-phenylmethoxy-2,3,6,7-tetrahydroazepine 1-(2,2-dichlorocyclopropyl)oxyethenylbenzene 3-[(4-fluorophenyl)methyl]-1,2-benzothiazole 4-ethoxycarbonylnaphthalene-1,6-disulfonic acid N'-[3-(5-chloro-2-fluorophenyl)-1H-indazol-6-yl]thiophene-2-carboximidamide;ethane 6-bromo-7-hydroxy-2,2-dimethylchromene-3-carboxylic acid 3-(1,2-diethylbenzimidazol-5-yl)oxy-N'-hydroxypyrazine-2-carboximidamide (5S)-2-[(4-chlorophenyl)methylsulfanyl]-N-naphthalen-1-yl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 2-[4-(1H-imidazol-2-yl)phenyl]-5-methyl-N-[3-methyl-3,4-di(propan-2-yloxy)cyclohexa-1,3-dien-1-yl]pyrimidin-4-amine (5-azidopyridin-2-yl)oxy-oxidoazanium N-[2-(4,7-dihydroxy-6,8,9,10-tetrahydro-5H-cyclohepta[b]pyridin-3-yl)-1,3-benzoxazol-5-yl]acetamide 2-[(1E,3Z)-1-amino-4-methylpenta-1,3-dien-2-yl]-5-[5-bromo-6-(4-methoxyphenyl)pyridazin-3-yl]phenol N-ethylsulfonyl-4-nitro-N-(4-sulfamoylphenyl)benzamide (2R)-4,4-difluoro-N-[1-(hydroxymethyl)cyclopropyl]-7-phenylmethoxy-2-[5-[4-(trifluoromethyl)phenoxy]pentanoylamino]heptanamide 3-[3-hydroxy-4,6-bis(methoxymethyl)oxan-2-yl]oxyphenol 4-[(2S)-5-(1,3-benzothiazol-6-ylamino)-1,2,3,6,7,8-hexahydropyrrolizin-2-yl]pyridine-2-carboxamide 2-[1-[6-(1H-benzimidazol-2-yl)-9H-fluoren-4-yl]-3,5-diphenylpyrazol-4-yl]propanamide N-(4,6-dimethylpyrimidin-2-yl)-3,5-dihydroxybenzamide 2-(3,5-difluorophenyl)-5-ethylfuran (3E)-3-[[4-fluoro-2,6-di(propan-2-yl)phenyl]methylidene]piperidine (2R)-2-[3-chloro-4-fluoro-9-oxo-6-propan-2-ylacridin-10-yl]butanediamide 5-hydroxy-1'-methylspiro[2H-indole-3,4'-pyrrolidine]-7-carboxylic acid N-[2,3-bis(ethenyl)phenyl]-N-[3-fluoro-4-[(E)-hydrazinylidenemethyl]phenyl]-1H-indole-3-carboxamide 6-[(3R,5S)-3,4,5-trimethylpiperazin-1-yl]pyrazine-2-carbonitrile 2-[3-[5-[(4-phenyl-3,6-dihydro-2H-pyridine-1-carbonyl)oxymethyl]furan-2-yl]phenoxy]acetic acid 4-[1-(3-fluoro-5-pyrimidin-2-ylpyridin-2-yl)pyrazol-4-yl]oxypiperidine-1-carboxylic acid 5-[1-(3,4-difluorobenzoyl)piperidin-4-yl]sulfanylthiophene-2-carboxylic acid 2-cyclohexyloxy-1-methylidenefluorene 4-[(2S)-5-[4-[[3-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)propanoylamino]methyl]phenyl]pentan-2-yl]oxybutanoic acid [(3aR,7aS)-5-pyrimidin-2-yl-3a-(pyridin-4-ylmethoxymethyl)-1,3,4,6,7,7a-hexahydropyrrolo[3,4-c]pyridin-2-yl]-cyclopropylmethanone;2,2,2-trifluoroacetic acid 5-azido-4,6-dichloro-2-(2,3,5-trifluorophenyl)pyrimidine 4-[azido-(2,4-difluorophenyl)methyl]-5-fluorobenzonitrile 3-[2-(4-fluorophenyl)-6-methylphenyl]iminobutan-1-ol N-cyclobutyl-4-(3-fluorophenyl)-N'-[[1-[(2R,4R)-2-methyloxane-4-carbonyl]azetidin-3-yl]methyl]butanehydrazide N-[2-(azepan-1-ylmethoxy)phenyl]-3,4-dihydro-1H-isochromene-7-carboxamide 5-[2,6-difluoro-4-(trifluoromethyl)phenyl]spiro[1H-indole-3,1'-cyclopentane]-2-one N-[(2,4-dimethoxyphenyl)methyl]-7,8-dimethoxy-1-pyridin-3-yl-5H-chromeno[4,3-c]pyrazole-3-carboxamide 5-methyl-N-(2-methylphenyl)sulfanylpyrimidin-2-amine 2-[4-[(2,6-dichlorophenyl)methyl]morpholin-3-yl]ethanol 3-(2,4-dimethylphenyl)-5-[(3R)-1-propanoylpiperidin-3-yl]oxypyrazin-2-amine 5-(5-azidopyridin-2-yl)oxyisoquinoline (2Z,4E)-N,5-dimethyl-3-[1-methylidene-4-(N-phenylanilino)naphthalene-2-carbonyl]hexa-2,4-dienamide N-[2,4-difluoro-3-[1-(2-methoxypyridin-3-yl)pyrazolo[4,3-c]pyridin-5-yl]phenyl]ethanesulfonamide 1-[3-(2,6-difluorophenyl)oxetan-3-yl]-N,N-bis(prop-2-ynyl)methanamine N-benzylsulfanyl-N-[(2E,4Z)-hexa-2,4-dien-3-yl]ethanamine 7-[(2R)-2,3-dihydroxypropoxy]-4H-1,4-benzoxazin-3-one 1-(3,5-dichlorophenyl)-5-(2,4-dimethyl-6-oxocyclohexen-1-yl)pentan-1-one;ethane 5-(4-azidobutyl)benzotriazole N-benzyl-4-(2,3-dihydro-1H-indole-5-carbonyl)piperazine-1-carboxamide 2-[(3R,5S)-3-amino-5-methylpiperidin-1-yl]quinoline-7-carboxylic acid;dihydrochloride 2-chloro-4,5,6-trifluoro-3-methylbenzenesulfonamide 2-[2,3-difluoro-4-(2-methoxyethylcarbamoyl)phenyl]sulfonyl-N-hydroxy-1,4-dihydroquinoline-6-carboxamide 2-[4-chlorobutyl(ethyl)amino]benzenesulfonic acid N'-[(2S,3R)-3-hydroxybutan-2-yl]-N-(2-methoxyphenyl)methanimidamide (2S)-N-[3-ethoxy-4-[6-methyl-7-[(1-propanoylpiperidin-4-yl)amino]quinolin-4-yl]phenyl]pyrrolidine-2-carboxamide 4-(3,5-dichlorophenyl)-N-(6-methyl-2-oxo-1H-quinolin-7-yl)piperazine-1-carboxamide N-[1-(6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-2-yl)piperidin-3-yl]pyrimidin-2-amine 1-(4-propylsulfanylphenyl)but-3-ene-2,2-diol 6-(2,4-dimethylphenyl)spiro[3H-furo[3,4-c]pyridine-1,4'-piperidine] [3-(cyclopropylmethoxy)-4,5,6,7-tetrahydro-1H-indazol-5-yl]methanol 4-fluoro-2-methylsulfanylbenzenethiol;7-(furan-3-yl)-N,N-dimethylthieno[3,2-d]pyrimidin-2-amine 4-[(2-azidoacetyl)amino]benzenecarboximidamide [(3R)-1-(1,2,4-triazin-3-yl)piperidin-3-yl]methanol N-ethyl-1-[4-(3-methoxyprop-2-enoyl)cyclohexyl]-7H-cyclopenta[c]pyridine-6-carboxamide N-[5-(2,3-dichlorophenyl)sulfonyl-1H-indazol-3-yl]benzamide 7-methoxy-6-[3-(methylamino)pyrrolidine-1-carbonyl]-4H-chromen-3-one 4-methyl-N-[(2S)-1,1,1-trifluoropropan-2-yl]benzamide (E)-1-[4-(benzylamino)butyl]-3-(5-bromothiophen-2-yl)oct-1-en-3-ol 2-[2-(4-fluorophenyl)ethyl]-4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-N-[2-(methylamino)ethyl]benzamide (2R,4S)-N-[1-(benzenesulfonyl)-3,6-dihydro-2H-pyridin-4-yl]-4-fluoro-1-(6-methoxynaphthalen-2-yl)pyrrolidine-2-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-2,6-dimethoxybenzenesulfonamide 4-[4-(1H-indazole-3-carbonyl)piperazin-1-yl]sulfonylbenzonitrile 2-tert-butyl-5-fluoro-4-(3-methoxypyridin-2-yl)sulfanylpyridine 4-[7-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[3.5]nonan-2-yl]phenol 6-(4-methylphenyl)-9H-carbazole-3,5-diamine 4-[7-(1H-indol-6-ylmethylamino)quinazolin-2-yl]-N,N'-diphenylbutanehydrazide 3-[2-(3,4-dimethoxyphenyl)ethyl]-1-oxa-8-azaspiro[4.5]decane 1-[(1Z,3E)-5-methoxyhexa-1,3-dienyl]sulfanyl-4-propan-2-ylbenzene [(5R,7S)-4-azido-3-methyl-5,6,7,8-tetrahydronaphthalen-2-yl]urea 6-amino-9-[(2R,3R,4S,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-purin-2-one;ethane N-(4,6-dimethylpyrimidin-2-yl)-4-[propyl([1,2,4]triazolo[4,3-a]pyrazin-5-yl)amino]benzenesulfonamide 2-[3,5-dichloro-4-(7-hydroxy-6-methyl-4-oxoquinazolin-3-yl)phenyl]acetamide 1-[(3-bromophenyl)methyl]-5,6,7,8-tetrahydro-4H-pyrazolo[3,4-d]azepine;2,2,2-trifluoroacetic acid 6-[(4-fluorophenyl)methyl]-1',2,3,8-tetrahydroxyspiro[anthracene-9,3'-indole]-7-carbonitrile 2-[(Z)-2-cyano-3,3,3-trifluoroprop-1-enyl]-N-(4-iodopyridin-2-yl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 2-(6-hydroxy-3,4-dihydronaphthalen-1-yl)benzoic acid (E)-1-[2-butyl-5-methoxy-4-[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]phenyl]pent-3-en-1-one 1-[6-(azidomethyl)pyridin-2-yl]-2,4-difluorobenzene N-[1-[1-[(2S)-butan-2-yl]piperidin-4-ylidene]benzimidazol-5-yl]-2,6-difluoro-3-methoxybenzamide (4aS)-5-acetyloxy-7-acetamido-8-(5,6-dichloropyrazine-2-carbonyl)-N,2,4,4a,9,9a-hexahydroxanthene-1-carboxamide (4R)-1-[2-fluoro-5-(trifluoromethyl)pyridin-3-yl]-N,8-dimethyl-N-phenyl-3,6,9,10-tetrazatetracyclo[7.7.0.02,6.011,16]hexadeca-2,4,10,12,14-pentaen-12-amine N-[3-[(1Z)-buta-1,3-dienyl]phenyl]acetamide;ethane N-[1,2-difluoro-5-(2-phenylethyl)cyclohepta-2,4,6-trien-1-yl]hydroxylamine 2-methoxy-4-[4-[(1S)-2,2,2-trifluoro-1-hydroxyethyl]phenyl]phenol 6-methyl-7-[2-(4-phenylpiperazin-1-yl)ethoxy]-4H-pyrido[3,2-b][1,4]oxazin-3-one;hydrochloride 3-[3,5-difluoro-4-(2-phenylethynyl)phenoxy]cyclobutan-1-ol N-[(1R)-1-(2,4-dichlorophenyl)ethyl]-6-[3-methoxy-4-(trifluoromethyl)pyridin-2-yl]sulfanyl-8-nitroquinolin-4-amine 2-[(5S)-4,6-dioxo-1-(4-phenoxyphenyl)-5H-pyrazolo[3,4-d]pyrimidin-5-yl]acetic acid 2-hydroxy-3,4-dimethoxybenzenecarboximidamide 4-N-(3-bromo-5-fluorophenyl)-6-N,7-dimethylquinazoline-2,4,6-triamine 2-methylsulfanyl-N-[3-(1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carbonyl)phenyl]acetamide 1-(3,4-dichlorophenyl)-5-[2-(ethylamino)ethyliminomethyl]-6-hydroxypyrimidine-2,4-dione N-(3,5-dichlorophenyl)-3-methyl-4,7-dioxo-2-sulfanylidene-1H-thieno[3,2-d]pyrimidine-6-carboxamide 2-[(6E)-8-cyclopentylimino-7,9-dihydro-5H-pyrido[3,4-b]indol-6-yl]benzonitrile (E)-3-[2,3-difluoro-4-[1-methyl-3-(4-pentanoyloxyphenyl)cyclohexen-1-yl]phenyl]prop-2-enoic acid (2R)-2-amino-N'-[4-methyl-3-[6-methyl-7-(pyridin-3-ylmethoxy)quinolin-4-yl]phenyl]propanediamide 2-(4-fluoro-N-phenacylanilino)octanoic acid (E)-4-[diethylamino-[2-methyl-6-(trifluoromethoxy)benzimidazol-1-yl]methylidene]-N,2-dimethylpent-2-enamide 2-bromo-5-[4,7-dimethyl-6-(1-pyridin-3-ylpropoxy)-3,4-dihydro-2H-quinoline-1-carboximidoyl]benzonitrile 2-(2,6-dichloro-N-methylsulfonyl-4-nitroanilino)octanoic acid N-[3,5-dichloro-4-(trifluoromethyl)phenyl]-2,6-dihydroxybenzamide 6-ethenyl-5-[(1R)-1-[(3S,4S)-4-methoxy-3,4-dihydro-2H-chromen-3-yl]ethyl]pyrimidine-2,4-diamine (3S)-1-[5-[2-(3,4-dimethoxyphenyl)propan-2-yl]-4H-pyrrolo[3,2-d][1,3]thiazole-6-carbonyl]pyrrolidine-3-carboxamide 3-(1,2,3,6-tetrahydropyridine-4-carbonyl)naphthalen-1-ol 2-(2,6-dimethylpyridin-4-yl)-5-methyl-1H-indole;ethane 5-chloro-2-(cyclobutylmethoxy)-4-fluoropyrimidine [3-(2-hydroxyethyl)morpholin-4-yl]-(6,7,8,9-tetrahydrothieno[3,2-c]oxepin-4-yl)methanone 1-[3-fluoro-4-[5-fluoro-6-(hydroxymethyl)pyridin-2-yl]phenyl]-2-[5-(trifluoromethoxy)pyridin-3-yl]ethanone 5-[2-[4-(methanesulfonamido)phenyl]ethyl]-N-methylthiophene-3-carboxamide (Z,2S)-4-[4-methoxy-3-(5-methyl-1H-pyrazol-3-yl)phenyl]-2-[2-(trifluoromethyl)ethylimino]pentanal N-[(2-hydroxy-5-iodophenyl)methylideneamino]-2-(3,4,5-trimethylphenoxy)acetamide 4-[2-(N-formylanilino)ethylamino]butanamide (3,5-dichloropyridin-4-yl)methanesulfonamide N-(3,5-dichlorophenyl)-2-[1-[4-(hydroxymethyl)oxane-4-carbonyl]piperidin-4-yl]oxyacetamide N-benzyl-1-oxo-4H-thieno[2,3-c]thiazine-7-carboxamide 1-cyclopentyl-N-[(4-ethoxyphenyl)methyl]piperidin-3-amine (3Z,5E)-7-amino-N-[[4-[2-fluoro-3-methyl-4-(2,2,2-trifluoroethoxy)phenyl]cyclohexyl]methyl]hepta-1,3,5-triene-2-sulfonamide ethane;N-[(2E,4Z)-hexa-2,4-dien-3-yl]aniline 1-phenyl-2-[(1-propylindol-3-yl)methylideneamino]guanidine 2-[3-[4-(benzenesulfonyl)morpholin-2-yl]propanoylamino]thiophene-3-carboxamide (3R)-1-acetyl-N-[5-methoxy-2-methyl-4-(trifluoromethyl)phenyl]piperidine-3-carboxamide 3-(2,4,5-trifluorophenyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine (7S)-N,4,8-trimethyl-2-[[1-[(3R,5R)-3,4,5-tris(phenylmethoxy)piperidine-1-carbonyl]cyclopropyl]amino]-6-oxononanamide (1R)-2,3-bis(phenylmethoxy)cyclopentan-1-ol 6-[2,3-difluoro-4-(4-pentylphenyl)phenyl]-1,8-difluoronaphthalene-2-carbonitrile 2-[4-(benzenesulfonyl)piperidin-1-yl]-5,7-dihydropyrrolo[3,4-d]pyrimidine N-azido-4,5-dichloro-2-(dimethylamino)benzenesulfonamide 2-amino-3-(1H-imidazol-5-ylmethylidene)quinazolin-4-one 4-[(E)-3,5-dihydroxypent-1-enyl]benzonitrile N-[2,4-difluoro-3-[(E)-5-methyliminohex-1-enyl]phenyl]formamide;5-cyclopentylpyridine-3-carbonitrile (E)-N,3-dimethyl-1-(1H-pyrrol-2-yl)pent-1-en-3-amine [4-(1H-indol-3-yl)piperidin-1-yl]-[5-(trifluoromethyl)furan-2-yl]methanone 3-[4-hydroxy-3,5-di(propanoyl)phenyl]-1H-indole-2-carboxylic acid (1S,3R)-4-[7-chloro-1-cyclopropyl-6-fluoro-8-[2-methoxyethyl(methyl)amino]isoquinoline-5-carbonyl]-N',3-dihydroxy-3-phenylmethoxycyclohexane-1-carbohydrazide 2-[(4-chlorophenyl)methyl]-8-methoxy-1,7-dihydropurin-6-one 4-[5,6-bis(ethenyl)-3a,7a-dihydro-1H-indol-2-yl]benzaldehyde 4-[1-(benzylsulfonylamino)ethyl]benzoic acid 2-[6-chloro-1-(1,3-dimethylindazole-7-carbonyl)piperidin-4-yl]acetic acid N-[(4,5-dimethylcyclohexa-1,3-dien-1-yl)methyl]-2-[(5-ethoxy-6-oxo-7H-imidazo[4,5-f]quinolin-9-yl)amino]propanamide 4-[2,5-bis(trifluoromethyl)phenyl]pyridine-3-carboxylic acid N-[1,3-di(propan-2-yl)pyrazol-4-yl]-6-fluoroquinoline-7-carboxamide (2S,3S)-6-[(1R)-5-fluoro-2-hydroxy-2-methylcyclohexyl]-3-phenyl-2-propan-2-yloxycarbonylheptanoate 5-(4-cyclopropyl-6,7,8,9-tetrahydropyrido[3,2-b]indolizine-6-carbonyl)pyridine-3-carbonitrile N-(3-hydroxysulfanylphenyl)-1H-pyrrolo[2,3-b]pyridine-4-carboxamide (2S)-2-[5-chloro-4-oxo-3-phenylquinazolin-7-yl]oxy-N-(6,7-dihydro-4H-thieno[3,2-c]pyran-4-ylmethyl)-N'-hydroxy-N'-propan-2-ylbutanediamide 5-tert-butyl-2,6-dimethoxy-1H-indole (2S)-N,4-dibenzyl-6,7,8,9-tetrahydropyrido[3,2-c]azepine-2-carboxamide 4-[1-(3-bromophenyl)ethyl]-5-methoxycarbonyl-2,6-dimethyl-1,4-dihydropyridine-3-carboxylic acid 7-[1-(2,6-dichloro-3,5-dimethoxyphenyl)ethyl]-2-pyridin-4-ylpyrazolo[3,4-d]pyrimidine 2-[5-carbamoyl-9-(cyclopropylmethoxy)-4-oxoquinolizin-3-yl]oxyacetic acid 4-[[5-chloro-2-(4-fluoropiperidin-1-yl)pyrimidin-4-yl]amino]-N,3-dimethoxybenzenesulfonamide [4-(aminomethyl)phenyl]-[4-[(1S)-1-azidoethyl]piperazin-1-yl]methanone 1-[6-(4-bromophenyl)-5,7-dihydro-4H-thieno[2,3-c]pyridin-2-yl]ethanone 5-chloro-N,N'-bis(pyridin-2-ylmethyl)-1,2,4-triazol-3-amine 4-chlorobenzene-1,3-disulfonate;dichlorotitanium (2S)-N,3-dimethyl-1-[2-methyl-4-[2-[5-[2-[2-oxo-3-(propanoylamino)pyridin-1-ium-1-yl]ethoxy]-2,3-dihydroindol-1-yl]phenyl]phenyl]but-3-en-2-amine 7-[(2-chlorophenyl)methyl]-4-hydroxy-3,5-dihydropurine-2,6,8-trione N-[2,6-difluoro-4-(3-methylbut-1-en-2-yl)phenyl]-2-methoxyethanimidate N-[3-(benzimidazol-1-yl)propyl]-3,4,5,6,7,8a,9-octahydroquinoline-8-carboxamide;dihydrochloride [4-amino-2-chloro-3,6-di(propan-2-yl)phenyl]urea 3-[4-(5,6-dimethylpyrimidin-4-yl)oxyphenyl]cyclopropane-1,1,2,2-tetracarbonitrile [6-(3-fluoroanilino)pyridin-2-yl]-[(2S,4R)-4-methoxy-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-2-yl]methanone N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-5-(dimethylcarbamoylamino)-6-fluoropyridine-3-carboxamide 4-[3-fluoro-6-(2-methylpropoxy)pyridine-2-carbonyl]piperazine-1-carboxylic acid 2,3-bis(4-bromophenyl)butanedioate 4-(diethylamino)-2-[2,6-dimethoxy-4-(methylaminomethyl)phenyl]-1H-pyrimidin-6-one N-(5-chloropyridin-2-yl)-4-[2-(oxan-3-ylmethoxy)ethyl]piperidine-1-carboxamide 5-[4-(2-fluorophenyl)-6,7-dihydro-1H-benzimidazol-2-yl]-N-(5-methoxypyridin-3-yl)-1H-pyrrole-3-carboxamide N-[(1S)-1-cyclohexylethenyl]-4-[2-[3-(methoxyamino)piperidin-1-yl]pyridin-4-yl]cyclohexane-1-carboxamide 3-chloro-1,2-bis(4-hydroxyphenyl)propane-1,2-dione N-[(3S,4R)-1-[2-(dimethylamino)ethyl]-4-propan-2-ylpyrrolidin-3-yl]furan-2-carboxamide;hydrochloride 2-[4-(3,5-dimethylpyrazol-1-yl)piperidin-1-yl]-5-methylpyridine 2-[(3,4-difluorophenyl)methyl]-3-[4-(3,5-difluoropyridin-4-yl)piperazine-1-carbonyl]cyclopentan-1-one 2-azido-1,4-dichloro-3,5-dimethylbenzene 1-[(6S,11R)-10-bromo-8-oxa-2,13-diazatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-12-yl]pyrrolidin-3-ol 2,4-diamino-5-[(3R)-1-ethylsulfonylpiperidin-3-yl]-1H-pyrimidin-6-one 4-[2,6-difluoro-3-(methylcarbamoyl)phenyl]pyridine-3-carboxylic acid N-benzyl-4-[5-methoxy-6-(3,4,4,5,6,7-hexahydro-2H-1-benzofuran-2-carbonylamino)pyridin-3-yl]piperidine-1-carboxamide 4-[(3-ethyl-1,3-benzothiazol-3-ium-2-yl)methylidene]-6-methoxyquinoline 1-[(2R,4S)-1,4-dimethoxypentan-2-yl]oxyethylbenzene 3-azidooxy-1H-pyrrolo[2,3-b]pyridine [2-(oxan-4-yl)pyrazol-3-yl]methanamine;hydrochloride [6-(2,4-dichlorophenyl)imidazo[1,2-a]pyridine-8-carbonyl]azanium 2-fluoro-5-(5-piperidin-4-yloxypyridin-3-yl)aniline 5-amino-7-(2,6-dichlorophenyl)sulfanylpyrrolo[1,2-b]pyridazine-3-carbonitrile;ethane 4-amino-3-chloro-1-methyl-5,6,7,8-tetrahydroquinolin-2-one 6-(2,3-dihydro-1H-inden-5-yloxy)pyridine-3-carbonitrile 3-ethyl-2-(4-pyridin-2-ylpiperidin-1-yl)pyrimidin-4-one 5-(4-azido-3-cyclopropylphenyl)-2-[(2S)-1-methoxypentan-2-yl]pyridine N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-prop-2-ynylethenesulfonamide 4-(azidomethyl)-3-cyclopentyloxybenzonitrile 1-azidooxy-3-(1,2,4-triazol-1-yl)propan-2-ol 1-(4-tert-butylcyclohexyl)-N,2-dimethylnaphthalene-2-carboxamide;methanamine (5Z)-2-cyclopropylimino-5-[(3,4-dichlorophenyl)methylidene]imidazolidin-4-one 4-[5-(2,3-dihydro-1H-inden-2-ylamino)-1,3,4-thiadiazol-2-yl]-2,6-dimethoxyphenol N-(6,7-dihydro-4H-pyrano[3,2-d][1,2]oxazol-3-ylmethyl)-5-methoxypyrazine-2-carboxamide 1-cyclopentyl-N-[[5-[3-[4-(2-fluorophenyl)-1H-indol-2-yl]-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]methyl]methanamine (7Z)-7-[(2-fluorophenyl)methylidene]-4,8-dioxo-3,6-dihydropteridine N-methyl-1,3-diphenylpropan-2-amine 2-[(Z)-1-anilinoprop-1-enyl]-3,5,6-trimethoxy-4-(2-phenoxyethoxy)benzamide 3-[4-(2,6-difluorophenyl)phenyl]-1-(5-methyl-1H-pyrazol-4-yl)imidazolidine 3-amino-N-[(2S,4R)-2-methyloxan-4-yl]thieno[2,3-b]pyrazine-6-carboxamide 7-(2,4,6-trimethylphenyl)heptanehydrazide 3-[(4,5-dimethyl-6,7-dihydro-5H-[1,3]thiazolo[5,4-b]pyridine-2-carbonyl)amino]cyclobutane-1-carboxylic acid 3-(1H-imidazol-5-yl)-N-[6-methoxy-2,4-di(propan-2-yl)pyridin-3-yl]propanamide 3-[5-chloro-4-(trifluoromethyl)pyrimidin-2-yl]aniline 3-methyl-5-[(1E,4Z,6Z)-5-methylidene-8,9-dihydrocycloocta[b]pyridin-2-yl]benzonitrile N-(3,4-dihydronaphthalen-2-ylsulfonyl)pyridine-4-carboxamide N'-[2,4-dichloro-3-[(3S)-3,5-dimethylpiperazine-1-carbonyl]phenyl]-2,3-dihydroindole-1-carboximidamide N-[2,4-di(propan-2-yl)phenyl]-6-methoxy-3H-indole-5-carboxamide 1-[(Z)-3,4-dimethylhex-2-enyl]-1-(4-fluorophenyl)hydrazine 2,4-bis(2-chlorophenyl)-5-[(3-fluoropyridin-4-yl)methoxy]cyclohexa-1,3-diene-1,3-dicarboxamide 2-(4,5-dimethyl-1H-imidazol-2-yl)phenol 5-[[(4S,9aR)-4-methyl-8-propanoyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-8-yl]sulfonyl]-4-ethoxy-N-(2-fluorophenyl)pentanamide (6E)-7-[2-chloro-3-(trifluoromethyl)phenyl]hepta-1,4,6-trien-3-one 2-[(4-hydroxy-5,6,7,8-tetrahydronaphthalene-1-carbonyl)amino]propanoic acid N-[(Z)-3-amino-2-fluoroprop-2-enyl]-1-[6-[(E)-hept-4-enyl]pyridine-3-carbonyl]piperidine-4-carboxamide 7-[(4R,5S)-2,6-dioxo-1,3-oxazinan-4-yl]pyrido[1,2-a]pyrimidin-4-one N-(1-phenylmethoxyethyl)-3,4-dihydrochromen-2-imine 1-cyclopropyl-N-[(Z)-3-methyl-6-oxoheptan-2-ylidene]-5-phenylpyrazole-4-carboxamide 2-[(2Z,5S)-2-[(Z)-[4-(4-tert-butylphenoxy)-3-chlorophenyl]methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 3-(1,3,5-triazin-2-yl)benzonitrile 4-[(Z)-2-amino-1-[3-chloro-5-methyl-N-[(6-methylsulfonylpyridin-2-yl)methyl]anilino]ethenyl]benzoic acid N-[5-(4,4-difluoropiperidin-1-yl)pyrazin-2-yl]benzamide 1-[(E)-6,7-difluorohept-5-enoxy]-2,3-difluorobenzene;ethane 4-[5-(2,2-difluoroethoxy)pyridine-2-carbonyl]piperidine-1-carboxylic acid 7-(benzenesulfonyl)-1-phenylindole 3-(4-propan-2-ylphenyl)quinoline 2-methyl-4,6-diphenyl-1H-benzimidazole N-[(3R,4S)-1-[2-(azetidin-1-ylmethyl)pyridine-4-carbonyl]-4-fluoropyrrolidin-3-yl]methanesulfonamide;hydrochloride (2R)-1-[(2S,3R)-3-[(5-chloro-4-oxoquinazolin-3-yl)methyl]-2-hydroxypentanoyl]pyrrolidine-2-carboxamide 3-(2-ethylmorpholine-4-carbonyl)furan-2-sulfonamide 6-(azetidine-1-carbonyl)-4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3H-pyrrolo[2,1-f][1,2,4]triazin-4-ol 3-[(E)-2-cyclohexylprop-1-enyl]-N-(pyridin-4-ylmethyl)quinoline-8-carboxamide N-(8,11-dichloro-4a,12b-dihydroindolo[3,2-b]carbazol-6-yl)-3-pyridin-3-yl-1H-indazol-5-amine 1-[(6R,11S)-7-hydroxy-2,10-diazabicyclo[10.4.0]hexadeca-1(12),13,15-trien-2-yl]ethanone 3-azido-4,5-ditert-butylphenol 1-(3,4-dihydro-2H-chromen-7-yl)-1-(2-phenylethyl)urea 7-[(4E)-2,6-dimethylnona-4,7-dien-3-yl]naphthalene-1,8-disulfonic acid 1-azidooxybenzo[h]isoquinoline 4-tert-butyl-2,6-dimethoxybenzaldehyde 3-cyclohexyl-5-(4-phenylphenyl)pyridine 2-[(E)-hexan-3-ylideneamino]oxy-N-methyl-6-piperidin-1-ylaniline 5-[(3,4-dimethoxyphenyl)methylidene]-2-imino-1,3-thiazolidin-4-one (2S)-1,1-diphenylethanol;[3-(methylamino)phenyl]-piperazin-1-ylmethanone 5-methoxycarbonyl-2-thiophen-3-ylthiophene-3-carboxylic acid 4-(2,4,6-trimethylphenoxy)carbonylbenzenesulfonic acid 2-[(Z)-[(2,4-dimethylphenyl)hydrazinylidene]methyl]-6-ethoxyphenol 2-[(3S)-1-methylpyrrolidin-3-yl]oxy-4,5-dihydrobenzo[g][1]benzothiole 4-[(3,5-dimethoxyphenyl)diazenyl]-2-[(E)-(4-hydroxyphenyl)methylideneamino]-1H-pyrazole-3-thione 2-[5-bromo-2-[(4-ethylphenyl)methoxy]phenyl]ethanamine [2-chloro-6-(trifluoromethyl)phenyl]-[4,5-dihydroxy-6-[4-(propanoylamino)butoxy]naphthalen-1-yl]azanium 1-azido-5,6-difluorobenzotriazole 3-[4-(difluoromethoxy)phenyl]-5-[4-[(Z)-2-pyridin-3-ylethenyl]cyclohexyl]-1,2,4-oxadiazole (4-aminophenyl)-[4-(4-ethylphenyl)piperazin-1-yl]methanone 2-(1,5-dimethylpyrazol-4-yl)-N-[(E)-(3-hydroxyphenyl)methylideneamino]quinoline-4-carboxamide 6-[(2Z,4E)-5-dimethoxyphosphanylocta-2,4-dien-4-yl]-3-(2-ethylphenyl)-1H-thieno[3,2-d]pyrimidine-2,4-dione ethane;N-methylsulfanyl-1,3-benzothiazol-2-amine 1-[3-(azepan-4-yl)phenyl]ethanone [2-(3-methoxyphenyl)piperazin-1-yl]-(2-methylpyrazol-3-yl)methanone 4-[3-(1H-imidazol-5-yl)propanoyl]-12a-methyl-2,3,6,7,8,9,10,11a,12b-decahydro-1H-pyrido[1,2-b]isoquinoline (2S)-1-[2-chloro-4-[[6-(2,3-dihydroxypropoxy)quinazolin-2-yl]amino]phenyl]sulfanylpyrrolidine-2-carboxamide N-[(1S)-4,6-dimethylcyclohex-3-en-1-yl]-5-nitrofuran-2-carboxamide 4-[(2S,5R)-2,5-bis(phenylmethoxy)cyclohexyl]oxybenzenesulfonamide 2-(4,5-dimethylpyrazol-1-yl)-N-[6-fluoro-3-(2H-tetrazol-5-yl)-2,3-dihydro-1H-inden-1-yl]acetamide 7-bromo-8-(4,6-diphenylpyridin-2-yl)-6H-benzo[c]chromene N-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-6,11-dioxobenzo[b][1,4]benzoxazepine-7-carboxamide 4-[(5Z)-5-[[1-[2,6-dichloro-4-(trifluoromethyl)phenyl]pyrrol-2-yl]methylidene]-3-(2-fluoropyridin-4-yl)pyrazol-1-yl]butanenitrile 6-(azetidin-3-ylmethoxy)-N-[[2-chloro-4-(cyclohexa-1,5-dien-1-ylamino)phenyl]methyl]pyridine-3-carboxamide (4S)-4,5-bis[4-(difluoromethoxy)phenyl]imidazolidine 2,6-dimethyl-7-(trifluoromethoxy)imidazo[1,2-a]pyridine 2-[(4S)-3-methylpiperidin-1-yl]-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-4-one 2-(3,4-dihydro-1H-isoquinolin-2-yl)pyrimidine-5-carbohydrazide;hydrochloride 1-[(3R)-3-azidopyrrolidin-1-yl]-2-(4-chlorophenyl)ethanone (E)-3-amino-1-[5-bromo-4-[(1Z,6E)-1,7-difluorohepta-1,4,6-trienyl]pyridin-2-yl]prop-2-en-1-one 4-[(2-azidophenoxy)methyl]pyridine 1-[5-chloro-4-(cyclohexylamino)pyridin-2-yl]ethanone 2-(3,4-dimethoxyphenyl)-1-(2-fluoro-6-hydroxycyclohexa-2,4-dien-1-yl)ethanone 1-[2,3-bis(4-chlorophenyl)phenyl]-3-[3-[3-(dimethylamino)propoxy]piperidin-4-yl]urea 5-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine 2-[(E)-1,3-benzodioxol-5-ylmethylidenehydrazinylidene]-5-[(4-ethoxyphenyl)methyl]-5-methyl-1,3-thiazolidin-4-one (3R)-3-[2,5-difluoro-4-[5-[[(4-methylcyclohexa-1,5-dien-1-yl)sulfonylamino]methyl]furan-2-carbonyl]phenyl]pentanoic acid 3-[1,4-diethyl-2-hydroxy-6-methoxy-5-(2-phenylethenyl)cyclohexa-2,4-dien-1-yl]propanal 3-[5-cyano-1-(4-methylphenyl)sulfonyl-2,3-dihydroindole-2-carbonyl]benzoic acid 4-methoxy-2,3-dinitronaphthalen-1-amine 2-(diethylamino)-N-[(E)-1-[6-methylidenecyclohexa-2,4-bis(4-methylphenyl))-3-oxocyclohepta-1,5-dien-1-yl]ethylideneamino]acetamide (3S,5R)-2-[4-chloro-5-(difluoromethyl)pyridin-2-yl]oxy-N'-hydroxy-5-propan-2-ylpyrrolidine-1-carboximidamide 4-[2-(2,5-dimethylpyrazol-3-yl)phenyl]pyridine 1-chloro-2,3-dimethylbenzene;N'-hydrazinylidene-5-[(Z)-prop-1-enyl]thiophene-3-carboximidamide 2-(1H-indol-3-yl)-N-methyl-N-[(4-oxo-3H-quinazolin-2-yl)methyl]acetamide 2-(1,3-benzoxazol-2-ylamino)-N'-hydroxypyridine-4-carboximidamide 4-[1-methyl-7-(propylamino)pyrazolo[3,4-c]pyridazin-5-ium-6-yl]phenol N-[5-[3-(4-pyridin-2-yl-1H-indol-2-yl)-1H-indazol-5-yl]pyridin-3-yl]pentanamide (5Z)-5-[[4-methyl-3-[4-(N-phenylanilino)phenyl]cyclohexa-1,5-dien-1-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one N-[[(2R,3S)-1-ethyl-2-pyridin-4-ylpiperidin-3-yl]methyl]-2-phenoxyacetamide 2-[(1S)-6-methoxy-3,4-dihydro-1H-isochromen-1-yl]propan-2-ol N-[3-amino-2,4-bis(methylperoxy)phenyl]acetamide N-[(2,6-dimethylimidazo[1,2-a]pyridin-3-yl)methylidene]hydroxylamine N-[[(2S,3S)-1-ethyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]methyl]-3-hydroxypyridine-4-carboxamide 4-(3,5-dimethylphenyl)-N-[4-hydroxy-4-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]-2-(hydroxymethylideneamino)butanamide (2S)-1,4,4-trifluoro-3-oxobutan-2-olate;triphenylphosphane [[4-hydroxy-3,5-di(propan-2-yl)phenyl]methylideneamino]urea 4-[2-azido-1,1-bis(methoxymethyl)indene-5-carbonyl]oxybenzoic acid (2R,5S)-4-[3-chloro-4-cyano-5-fluoro-6-(4-methoxyanilino)pyridin-2-yl]-2,5-dimethylpiperazine-1-carboxylate 4-N,8-dimethyl-6H-benzo[b][1]benzoxepine-2,4-dicarboxamide 6-(trifluoromethyl)imidazo[1,2-a]pyridine-3-sulfonamide 6-(cyclohexylmethoxy)-1,2,3,4-tetrahydroquinoline N-[3,5-dimethoxy-4-(1-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-1H-imidazole-2-carboxamide 4-[4-(2,3-difluorophenyl)phenyl]sulfanylbenzonitrile N-[(3R)-1-[2-fluoro-5-(methylcarbamoyl)phenyl]pyrrolidin-3-yl]pyridine-4-carboxamide N-cyclopentyl-5-(1H-imidazo[4,5-b]pyridin-2-yl)-7-methoxyimidazo[1,2-a]quinoxalin-4-amine 6-[(2-hydroxyphenyl)methyl]-1,3-benzodioxol-5-ol 4-[1-(azidomethyl)piperidin-2-yl]phenol (2R)-2-hydroxy-N,3-dimethyl-N-[4-[[3-[3-(trifluoromethoxy)phenyl]-1H-pyrazol-5-yl]amino]quinazolin-7-yl]butanamide 2-cyclohexyl-N-[5-[3-(4-pyridin-4-yl-1H-indol-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]acetamide (4-aminopiperazin-1-yl)-[4,6-bis[5-chloro-2-(tetrazol-1-yl)phenyl]pyridin-3-yl]methanone (1-ethyl-4,6-dimethoxypyrazolo[3,4-d]pyrimidin-5-yl)-(4-hydroxypiperidin-1-yl)methanone 1-[2,6-diethyl-4-(3-methylpyridin-2-yl)phenyl]-5-[(E)-prop-1-enyl]sulfanylpentane-1,7-dione (3R)-3,4-dimethyl-1-[5-(2-phenylethynyl)pyridin-2-yl]sulfonylpiperazine N-[4-(cyclopropylsulfonylamino)butyl]pyridine-2-carboxamide N-(4,5-dihydroimidazol-1-yl)-4-[1-(3-methylphenyl)benzimidazol-2-yl]aniline 4-(dimethylamino)-N'-(2,3-dihydro-1H-inden-1-yl)-5-propan-2-yl-1,2,3,6-tetrahydropyridine-2-carboximidamide (1Z)-1-[5-bromo-2-methyl-3-[4-(5-nitropyridin-2-yl)piperazine-1-carbonyl]phenyl]propan-1-olate (5S)-1,3-diethyl-5-[4-[2-(methylideneamino)ethoxy]phenyl]imidazolidine-2,4-dione (2R,4R)-N,3-dihydroxy-1-[6-(trifluoromethyl)pyridine-2-carbonyl]piperidine-2-carboxamide 3-azidooxy-1,2-difluoronaphthalene 5-(1-hydroxyethyl)-4,5-dihydrothieno[3,2-g]chromen-7-one 1-(4-benzylsulfanylphenyl)imidazole 2-fluoro-4-(7,8,9,10-tetrahydropyrido[1,2-a]indol-6-yl)benzamide (3R)-N',3-dimethylpentanehydrazide;1-fluoro-4-[4-methanimidoyl-5-(methylideneamino)thiophen-2-yl]cyclohexa-2,4-dien-1-amine 3-chloro-4-[4-(trifluoromethyl)phenyl]cyclohexa-2,4-diene-1-sulfonamide 3-hydroxy-5,6-dimethoxy-4,8-dimethylnaphthalene-1,2-disulfonic acid 1-(4,6-dichloropyrimidin-5-yl)oxypiperidine-2-carboxylic acid N-[5-fluoro-4-(8-fluoro-2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-7-yl)pyrimidin-2-yl]-6-methoxy-1H-indazol-5-amine 6-tert-butylsulfanyl-3,5,7-trimethoxy-2H-benzo[f]isoindol-1-one 6-(N-naphthalen-2-ylsulfonylanilino)hexanoic acid N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]benzamide 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N'-hydroxypyrimidine-4-carboximidamide 4-[2-[(Z)-1,3-diaminoprop-2-enylidene]hydrazinyl]-6-methoxyquinoline-7-carboxamide (E,2Z)-2-ethylidene-6-[4-methoxy-3-[(5-methylpyrazin-2-yl)sulfamoyl]phenyl]hex-3-enamide;1-ethylpyrrolidine 4-[4-(diethylamino)phenyl]-2,5-dimethoxyphenol 7-N,7-N-bis(4-methoxyphenyl)-2,3-dihydroimidazo[1,2-a]pyridine-3,7-disulfonamide 6,7-dimethyl-1H-quinolin-4-one;1-ethoxy-3,5,10,13-tetrazatricyclo[7.4.0.02,7]trideca-2(7),8,11-triene 1-[(6R)-4-benzoyl-3,3a,5,6,7,7a-hexahydro-2H-pyrrolo[3,2-b]pyridin-1-yl]-2-[4-(1H-imidazole-2-carbonyl)piperazin-1-yl]ethane-1,2-dione (5S)-1-[4-methoxy-3-(trifluoromethylsulfonyl)phenyl]-2,5,6,7-tetrahydropyrrolo[2,3-f]benzimidazole 3-methyl-1,4-dihydropyrazino[2,3-b]quinoxaline 4-benzyl-2-chloro-3-ethoxybenzoic acid 5-[(2,4-dichloropyrimidin-5-yl)-prop-2-enylamino]naphthalene-2-sulfonic acid 2-bromo-5,6,7,8-tetrahydroquinoline 3-[8-(1,2-dihydropyridin-4-yl)dibenzofuran-2-yl]pyrido[2,3-b]indole 1,4-dioxane;5-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-N-(4-methylcyclohexyl)-6-propan-2-ylpyrimidin-4-amine N-[3-(4-fluorophenyl)-5,6,7,8-tetrahydrocinnolin-4-yl]methanesulfonamide 1-bromo-6-chloro-4H-naphtho[2,3-b][1]benzothiole 1-[(2S,3S)-4-acetyl-N-[3-amino-5-(trifluoromethyl)phenyl]-3-fluoroanilino]-2-cyclopropylethanone 5-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,3-diol 2-[[1-methyl-4-[4-(oxan-3-yl)piperazine-1-carbonyl]pyrazol-3-yl]oxymethyl]-3H-quinazolin-4-one 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfanylpropane-1-thiol 2-azido-4,7-diphenyl-1H-benzimidazole 6-amino-3-ethyl-5-methyl-1H-pyrazolo[4,3-c]pyridin-7-one 5-[4-(2,6-difluorophenoxy)piperidin-1-yl]-8-[(E)-methoxyiminomethyl]-N-(1H-pyrazol-5-yl)quinazolin-4-amine 2-[1,4-bis(3,5-dimethylphenyl)-2-oxoimidazo[4,5-h]quinazolin-3-yl]acetamide 5-methyl-1-(4-propanoylphenyl)hexane-2,3-dione N-[5,6-dichloro-3-(hydroxymethyl)cyclohepta-1,4,6-trien-1-yl]naphthalene-2-carboxamide 5-[3-(ethylsulfinylmethoxy)phenyl]imidazolidine-2,4-dione N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-3-oxocyclobutane-1-carboxamide 5-[2-methylbutanoyl(1,3-thiazol-5-yl)amino]naphthalene-2-sulfonic acid 2-[(3,5-dichloro-4-hydroxyphenyl)methyl]propanedinitrile 2-(2,6-difluorophenyl)-1-(3-methylpyrrolidin-1-yl)ethanone N-[1-(2-azidooxyethyl)piperidin-4-yl]-3,5-dinitroaniline 5-amino-4-(7-fluoro-2-methylindazol-5-yl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 2-chloro-4-(ethylamino)naphthalene-1,5-dicarboxylic acid 1-[[5,6-dichloro-3-(2H-tetrazol-5-yl)indol-1-yl]methoxy]cyclohexan-1-amine 7-fluoro-4-[(2-methoxypyridin-3-yl)methyl]-2,3-dihydroquinoxaline 3-(2,4-dimethylcyclopenta-1,3-dien-1-yl)-5,7-bis[ethynyl(propan-2-yl)amino]naphthalene-2-carboxylic acid 1,2,3-trifluoro-5-[2-(4-methylcyclohexa-1,3-dien-1-yl)ethynyl]benzene [2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazole-2-carbonyl)phenyl]-methoxycarbamic acid N-(2,4-dimethylphenyl)-1-methylideneindazol-1-ium-3-carboxamide (4E)-2,5-bis[(3,4-difluorophenyl)methyl]-4-(furan-2-ylmethylidene)pyrazol-3-one [3-amino-4-(cyclopropylmethylamino)phenyl]carbamic acid N-[3-(2,6-dichloropyridine-4-carbonyl)-4,5-difluorophenyl]acetamide 3-amino-N-(2,5-dioxopyrrolidin-1-yl)benzenesulfonamide 1-[4-(2,3,6-trimethylphenyl)pyrazol-1-yl]propan-2-one N-(furan-2-ylmethyl)-4-[[1H-indazole-3-carbonyl(propanoyl)amino]methyl]benzamide (2R)-5,6-difluoro-1,4-bis[(3-methylphenyl)sulfonyl]-2-piperidin-1-ylbenzimidazole 2-[(1S)-1-aminoethyl]-5-bromo-3H-quinazolin-4-one 4-(2,5-dihydroxybenzenecarboximidoyl)benzaldehyde 2-(4-methylpiperazin-1-ium-1-ylidene)ethanamine;3,3,3-trifluoroprop-1-ene N-[(1R)-3-amino-2,4-dioxocycloheptyl]-5-methoxyquinoxaline-2-carboxamide 6-tert-butyl-N-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)piperidin-3-yl]pyridine-3-carboxamide 1-(1-tert-butyltriazol-4-yl)decan-2-ol N-[1-(2,4-difluorophenyl)pyrrolidin-3-yl]-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide 5-(1,3-benzodioxol-4-yl)-1-methylcyclohexa-3,5-diene-1,3-dicarboxylic acid 5-[4-[2,6-di(propan-2-yl)phenyl]-1,2,4-triazol-3-yl]-1,2,4,5-tetrazine;iridium (3S,7R,8aS)-2-(6-methylpyridine-3-carbonyl)-N-pyrimidin-4-yl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-amine 5-[(6R)-8-oxo-6,7-dihydro-5H-naphthalen-2-yl]-N-phenylfuran-3-carboxamide 4-(6,7-dihydrothieno[3,2-d]pyrimidin-4-yl)morpholine 5-[4-[2-(1,3-benzodioxol-4-yl)acetyl]piperazine-1-carbonyl]pyrrolidin-2-one 6-amino-4-[3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 6-(4-fluorophenyl)-N-methyl-5-(4-oxo-3H-phthalazine-1-carbonyl)-1-benzofuran-2-carboxamide 1-[(E)-2-ethenylbut-2-enoxy]-4-fluorobenzene 3-(6-cyano-4,5-dihydro-1H-indazol-7-yl)-2-methoxybenzoic acid 2-(2,4-dimethoxyphenyl)-6-hydroxy-1-[3-(trifluoromethyl)-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine-6-carbonyl]indole-3-carbonitrile 2-[(1E)-3-methylbuta-1,3-dienyl]-5-propan-2-ylbenzenesulfonamide ethane;N-[[4-(2-methylpropoxy)phenyl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide N-[4-(methylsulfamoyl)phenyl]-2-pyridin-3-ylacetamide 2-[(4-azidophenyl)methylamino]ethanol (2R)-N-[3-[4-[(Z)-but-1-enyl]phenoxy]phenyl]pyrrolidine-2-carboxamide 5-[3-(4-methylcyclohexa-1,3-dien-1-yl)oxyphenyl]penta-2,4-dienoic acid (Z)-N'-[2-[[5-chloro-6-[4-[2-(dimethylamino)ethoxy]anilino]pyrimidin-4-yl]amino]phenyl]but-2-enimidamide 2-[5-(2,4-difluorophenoxy)-2-ethylphenyl]-5-[1-(4-methoxybutanoyl)piperidin-3-yl]pyrazole-3-carboxylic acid ethane;1-[[6-fluoro-3-(5-methylcyclohexa-2,4-dien-1-yl)quinoline-7-carbonyl]amino]-3-(3-nitrophenyl)urea 2-(6-butoxynaphthalen-2-yl)acetamide 3-ethyl-7-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]-6,11-dihydro-5H-benzo[b][1,4]benzodiazepine 1-[3-(trifluoromethoxy)phenyl]pyrazole-3-carboxylic acid 2-(N-octylanilino)decanoic acid N-(2,6-difluorophenyl)sulfonyl-4-[3-oxo-7-(triazol-1-yl)-1H-isoindol-2-yl]pentanamide N-[3,4-bis(ethenyl)pyridin-2-yl]-5-cyano-1H-imidazole-2-carboxamide 2-(azidomethyl)-5-ethoxy-1,4-dimethylimidazole N-[(4E,6Z)-6-fluorooctaa-2,4,6-trien-3-yl]-1-methoxy-5-propan-2-ylidenepyrazole-3-carboxamide N-[[1-methyl-5-(piperidine-4-carbonyl)pyrrol-2-yl]methyl]formamide 4-[5,6-bis(2,3-dihydropyridin-4-yl)pyrazin-2-yl]-2H-thieno[3,2-b]pyridine 2-amino-4-[5-(3,4-dichlorophenyl)-1,2,4-oxadiazol-3-yl]phenol (2S)-N'-[1-(4-cyanophenyl)cyclopropyl]-3,3-dimethyl-2-phenylbutanimidamide [4-(1,3-dioxoisoindol-2-yl)phenyl]phosphonic acid (1R,4S)-N-[1-(2-methoxyethylamino)-2-naphthalen-2-yl-3,4-dihydroisoquinolin-5-yl]-4-propan-2-ylcycloheptane-1-carboxamide N-[2,6-difluoro-3-(propanoylamino)phenyl]sulfonyl-5-methylpyrazine-2-carboxamide N-[[2-(1,3-benzothiazol-2-yl)-5-(4-chloro-1H-pyrazol-5-yl)phenyl]methyl]-3-ethylcyclobutan-1-amine 2-ethylsulfonylnaphthalene-1,4-dione 2-[1-(2-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one 2-[[5-(3,4-dichlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[2,4-dimethyl-6-(piperidine-1-carbonyl)cyclohexa-1,3-dien-1-yl]acetamide 2,3-diphenylhept-2-enoate 2-N,3-N-dimethyl-4-[4-(1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl]butane-2,3-diimine 3-chloro-N-[4-[2-(4,5-dimethylimidazol-1-yl)ethoxy]cyclohexyl]-7H-pyrrolo[2,3-d]pyrimidin-4-imine 6-(3-bromophenyl)cyclohexa-2,4-diene-1,1-diamine 2-[4-(hydroxymethyl)-5-methoxy-1-(4-methoxyphenyl)sulfonylindol-3-yl]acetamide N-[(E)-(4-fluorophenyl)methylideneamino]-2-propoxybenzamide (5E)-2-imino-3-methyl-1-[(4-phenylpyridin-2-yl)amino]octa-3,6-dien-1-ol 4-(1H-inden-2-yl)-1,3,5-triazin-2-amine N-[2,6-dichloro-4-(trifluoromethoxy)phenyl]-5-fluoropyridine-3-sulfinamide 3-[2-(5,6-dihydronaphthalen-2-ylmethoxy)phenyl]hex-4-enoic acid 5-(5-fluoropyridin-3-yl)sulfonyl-2,3-dihydro-1H-indene-4-carbonitrile 6-(3,4-dimethylphenyl)-2-pyridin-4-yl-N-[3-(trifluoromethyl)phenyl]pyrimidin-4-amine 3-[[2-(1H-indol-4-yl)-7H-purin-6-yl]amino]propane-1,2-diol N-[(1E,3Z)-2,4-dimethylhexa-1,3,5-trienyl]-5-(3-ethylphenyl)thiophen-2-amine;2-ethylidenebut-3-enenitrile 1-(2,3-dimethylphenyl)-6-hydroxy-5-[[5-(4-iodopiperazin-1-yl)pyridin-2-yl]iminomethyl]pyrimidine-2,4-dione 5-[[[2,2,3,3,4,4,5,5-nonadeuterio-1,4-bis(trifluoromethyl)cyclohexyl]amino]methyl]-1H-quinolin-2-one 6-(3,4-dimethylphenyl)pyrazolo[1,5-a]pyrimidine (2R)-N-[4-[3-amino-5-(trifluoromethyl)pyridin-2-yl]oxyphenyl]-3,6-diazabicyclo[3.1.0]hexane-2-carboxamide N-[1-(4-azidophenoxy)-2,3-dihydroinden-5-yl]butane-2-sulfonamide 3-(5-propyltriazol-1-yl)pyridine 3-[1-(2,6-difluorophenyl)piperidin-4-yl]-5-ethoxy-2H-benzimidazole 3-(1H-indol-2-yl)-4-phenylmethoxybutanoic acid N-[5-[7-fluoro-3-[4-(5-methylthiophen-2-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-2H-indazol-5-yl]pyridin-3-yl]cyclobutanecarboxamide [3-(benzylamino)-2,6-difluorophenyl]methanol 4-(1-methylimidazo[4,5-c]pyridin-6-yl)-3H-pyrrol-2-one [2-(3,5-dichlorophenyl)-2-hydroxyethyl]azanium [1-[4-(difluoromethyl)phenyl]pyrazol-4-yl]boronic acid 1-[4-(cyclopropylmethoxy)-3-fluorophenyl]ethanol 1-(4-methylpentanoyl)-4-phenylpiperidine-2-carboxamide N'-(1,4-dimethylcyclohexa-2,4-dien-1-yl)-N'-[2-[ethyl(methyl)amino]pyridine-3-carbonyl]benzohydrazide (E)-N-ethoxy-1-[6-(2,3,4,5,6-pentachlorophenyl)pyridin-2-yl]methanimine 4-(2,6-dimethylphenyl)imino-1-ethoxy-7-methylidene-5H-[1,3]thiazolo[5,4-d]pyrimidine-2-thione 3-(4-methoxyphenyl)-7-methyloctanal 5-(2,4,6-trimethylphenyl)-3H-quinazolin-4-one 3-(4-carbamimidoylphenyl)-1H-indazole-5-carboxamide;ethane 4-(1,3-benzothiazol-2-ylamino)phenol N-[[4-amino-6-(4,5-difluorocyclohexa-1,3-dien-1-yl)-5-hydroxypyridine-2-carbonyl]carbamothioyl]-2,3-dihydroindole-1-carboxamide 2-[(3S)-1-[5-(4-methoxyphenyl)pyrimidin-2-yl]pyrrolidin-3-yl]acetic acid N-[3,5-bis(4-chlorophenyl)-2H-pyridin-1-yl]piperidine-2-carboxamide 4-[2,3-dihydroxypropyl(2H-tetrazol-5-yl)amino]butan-1-ol 5-[3-chloro-4-(trifluoromethyl)phenyl]-2,7-diethyl-N-[1-(2-hydroxypropan-2-ylamino)ethenyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide (4aR,9aS)-6-methylsulfonyl-N-[2-(3-oxo-1H-isoindol-2-yl)ethyl]-2,3,4a,5,7,8,9,9a-octahydrobenzo[g][1,4]benzoxazine-8-carboxamide 2-(4-methylphenyl)sulfonyloxy-3-phenoxypropanoic acid 2,3-dimethyl-4-[(2E)-5-[1-(6-methylcyclohexa-2,4-dien-1-yl)ethenoxy]penta-2,4-dien-2-yl]pyridine (1Z,3E)-3-[2-(5-methylthiophen-2-yl)ethynyl]hexa-1,3,5-trien-1-amine 2-[3-ethoxy-5-(trifluoromethyl)phenyl]benzo[g][1,3]benzothiazole N-(7-amino-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-3-yl)-N-methylacetamide [4-[[5,7-difluoro-2-(4-fluorophenyl)-1H-indole-3-carbonyl]amino]cyclohexyl]carbamic acid 3-[[2,5-dimethyl-1'-(1,3,4-oxadiazol-2-ylmethyl)spiro[indole-3,4'-piperidine]-6-yl]amino]cyclobutan-1-one;hydrochloride 1-(1,2-benzothiazol-3-yl)cyclohexa-2,4-dien-1-ol N-butyl-2,4-dichloro-N-[(3,5-difluorophenyl)methyl]pyrimidin-5-amine 1-(5,6-dimethoxypyridine-3-carbonyl)-4-hydroxypiperidine-4-carboxamide 1-[4-azidooxy-3-(2,3-dichlorophenyl)-5-methylphenyl]ethanone 3-fluoro-N-[4-methoxy-6-(pyrazol-1-ylmethyl)-1,2-benzoxazol-3-yl]benzamide N-(4-chlorophenyl)sulfanyl-2,3-dihydropyrrolo[2,1-b][1,3]benzothiazol-7-amine;ethane N-[4-[1,1,2,3,3,3-heptafluoropropan-2-yl(methoxy)amino]phenyl]sulfonylbenzamide (3R)-3-azido-6,7-dimethoxy-1H-quinoxaline-2,5-dione 1-[5-cyclohexa-2,4-dien-1-yl-7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-6-yl]pyrrolidine-3-carbonitrile (Z)-4-bromo-2,3-dihydroinden-1-one N-[2-(2-ethylbutoxy)phenyl]formamide 4-[2-chloro-6-(1,3-thiazol-5-yl)pyridin-3-yl]morpholine 2-[4-(3,5-difluorophenyl)triazol-1-yl]benzoic acid (1S)-N,2-diphenylcyclopentan-1-amine 1-[6-(2,3-dimethylphenoxy)pyrimidin-4-yl]-7,7-dimethyl-3-phenyl-6,8-dihydroquinoline-5,5-dione 4-(6,7,8-trifluoroquinazolin-2-yl)benzenesulfonamide 1-[4-(4-fluorophenyl)cyclohexyl]propan-2-amine 4-[2-(dimethylamino)ethylcarbamoyl]-2,3,5,6-tetrafluorobenzenesulfonic acid 4-[(4S)-3-methyl-6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl]benzonitrile 2-[4-(azetidine-1-carbonyl)piperidin-1-yl]-N,N-dimethylbenzamide 6-bromo-2-butylsulfanylquinazoline (2Z,4E)-1-phenyl-5-(4-sulfanylanilino)penta-2,4-dien-1-one 2-(N,2-dimethoxyanilino)ethanol 5-cyclohexyl-6-(9,9-dimethylfluoren-4-yl)-2-pyridin-4-ylpyrimidine-4-carboxylic acid N-methylsulfanyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide;methylsulfanylcyclohexane 1-[6-(5-cyclopentyloxypentanoyl)-2,3-dihydroindol-1-yl]ethanone 5-bromo-2,4-difluoro-N-(3-methylbutan-2-ylideneamino)benzenesulfonamide 1-[2-hydroxy-4-methylsulfanyl-3-(trifluoromethoxy)phenyl]-N,N-dimethylmethanesulfonamide (3E)-N'-[2,6-dimethyl-4-[5-[(4R)-4-methylazepan-1-yl]pyrrolo[3,2-b]pyridine-1-carbonyl]phenyl]-3-[(5Z)-5-ethylidene-3-oxopyrrol-2-ylidene]benzohydrazide 2-[4-(6-aminopyridin-3-yl)phenoxy]acetaldehyde;7,8-difluoro-1-methoxynaphthalene;N,5-dimethyl-1,2,4-thiadiazol-3-amine 4-(aminomethyl)-5-(2,3-dihydro-1H-inden-1-yl)-N-[3-hydroxy-2-(hydroxymethyl)butanoyl]thiophene-3-carboxamide;hydrochloride 2-amino-5-[3,4-dimethoxy-5-(propylamino)phenyl]-5-[4-(4-fluorobut-1-ynyl)phenyl]-3,6-dimethylpyrimidin-4-one (4S)-N-(2,5-dimethoxyphenyl)-6-oxo-3,4,7,8-tetrahydropyrimido[1,2-a]pyrimidine-4-carboxamide N-[(E)-3,7-dihydroxyhept-5-enyl]-5-methylthiophene-2-carboxamide 1-[(2R)-2,3-dihydroxypropyl]-4,5-bis(phenylmethoxy)piperidine-3-carboxylic acid 3-[4-(azidomethyl)phenyl]benzenecarboximidamide 4-(methylamino)-N-[1-(2,4,5-trichlorophenyl)sulfonylpiperidin-3-yl]pyrimidine-5-carboxamide N-[2,6-dimethyl-4-(methylsulfamoyl)phenyl]pyridine-3-carboxamide 2-(dimethylamino)-5,6,7,8-tetrahydroquinazoline-4-carboxamide;hydrochloride 5-fluoro-2-(4,4,5,5-tetramethyloxaborolan-2-yl)benzonitrile (1R,3S)-2,2-dichloro-3-[4-fluoro-5-(trifluoromethyl)pyridin-2-yl]cyclopropane-1-carbonitrile 2,5-dimethyl-N'-(7-morpholin-4-ylquinazolin-4-yl)benzenecarboximidamide 2-(3,4-dichlorophenoxy)acetaldehyde;6-[5-[(3R)-1-propanoylpiperidin-3-yl]pyridin-3-yl]oxynaphthalen-2-ol 5-azidooxy-N,6-diphenylpyrimidin-4-amine 2-amino-8-[5,6-difluoro-1-(4-methylphenyl)sulfonyl-3,4-dihydro-2H-quinolin-7-yl]-N,N-dipropyl-3H-1-benzazepine-4-carboxamide (6-chloropyridin-3-yl)methanesulfonate (2E)-2,3,4-trifluoro-7-methylocta-2,6-dienal (6aR,12bR)-10-methyl-N-phenyl-1,2,3,4,5,6a,11b-octahydroindolo[2,3-b]quinoline-7-carboxamide 4-[5-(2,5-difluorophenyl)-1H-imidazol-2-yl]-N-(3,4,5-trimethoxyphenyl)-1,8-naphthyridin-2-amine 4-[1-(2,3-dihydro-1H-inden-5-yl)propan-2-yl]morpholine 3-[2-(1-phenylethyl)pyridin-4-yl]-6,7-dihydro-5H-cyclopenta[c]pyridazine 3-(2,6-dichlorophenyl)-7H-thieno[3,4-b]pyrazin-5-one;N-(oxolan-3-yl)formamide (4-azidomorpholin-2-yl)-[4-[2-(hydroxymethylamino)pyridin-3-yl]phenyl]methanone 3-cyclobutyl-2,6-dimethoxybenzamide N-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-2-propan-2-yloxybenzamide (Z)-3-[4-(2-methoxyethylsulfanylamino)phenyl]prop-2-enamide N-methyl-N'-[(5Z)-2-[2-(trifluoromethoxy)phenyl]imino-4,6-dihydro-1H-pyrimidin-3-ium-3-ylidene]ethanimidamide 3-ethyl-N-methyl-1,2-benzothiazol-6-amine;5-[3-fluoro-4-(1,3-oxazol-5-yl)phenyl]pyrimidin-2-amine N-[3-(5,6-dimethoxy-1H-benzimidazol-2-yl)phenyl]-1,3-dioxo-4H-naphthalene-2-carboxamide 2-(benzylsulfanylmethyl)-4,6-ditert-butylpyridine;ethane 3-[4-(2,6-dimethylcyclohexen-1-yl)-N-ethylanilino]propanenitrile (E)-3-[4-[6-ethyl-7-oxo-5-[2-[(1S)-1,2,2-triphenylcyclopropyl]phenyl]octyl]phenyl]prop-2-enoic acid 3-[3,4-bis(ethoxymethyl)-5-hydroxyphenyl]benzoic acid 6-chloro-4-(3,5-dimethylphenyl)cyclohexa-2,4-diene-1-carboxylic acid N-[(5-ethoxy-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6,8-bis(trifluoromethyl)imidazo[1,2-a]pyridine-2-carboxamide 3-amino-1-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-one;1,1-difluoroethane N-[(1R)-1-(4-methoxyphenyl)propyl]pyridine-3-sulfonamide 2-[2,6-dichloro-N-(2-methylpropanoyl)-4-nitroanilino]decanoic acid ethane;4-[1-(3-methoxyphenyl)ethenyl]pyridine N-ethenylmethanimine;4,6-diphenyltriazolo[2,1-a]isoquinoline 2-[[4-[3,6-dimethyl-1-(oxan-4-yl)indol-5-yl]-6-phenylpyridine-2-carbonyl]amino]-2-[2-fluoro-4-(trifluoromethyl)phenyl]acetic acid 2-amino-6-methyl-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carbonitrile 1,4-difluorobenzene;(2S)-2-[[4-[2-[(2-fluorophenyl)methoxy]ethyl]piperidine-1-carbonyl]amino]-3,3-dimethylbutanoic acid 4-(1,3,4-oxadiazol-2-yl)-N-phenylnaphthalene-1-sulfonamide 2-[[(4S)-1,3,4-trimethylpyrrolidine-3-carbonyl]amino]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide N-[2-(2,3-dihydroindole-1-carbonyl)phenyl]benzamide 2-[3,4-dichloro-5-(trifluoromethyl)phenyl]acetonitrile 4-N,6-bis(2,3-dihydronaphthalen-1-yl)pyrimidine-4,5-diamine 1-azidooxy-3-phenoxyphenanthrene (2S)-2-(9H-fluoren-1-yl)-5,7-dihydroxyheptanoic acid 3-N-[2-(4-aminophenyl)ethyl]pyridine-3,4-diamine;1-benzyl-4-(4-methyl-5-sulfanylidene-1H-pyrazol-2-yl)pyridin-2-one N-(4-aminophenyl)-2-chloro-N-[3-methyl-4-[3-[5-(trifluoromethyl)pyridin-2-yl]propoxy]phenyl]acetamide 5-bromo-N-[[1,3-bis(4-chlorophenyl)pyrazol-4-yl]methylideneamino]-2-hydroxybenzamide N-[(6-aminopyridin-2-yl)methyl]-2-ethoxyacetamide 2-[3,5-difluoro-4-(methylamino)phenyl]-1,1,1-trifluoropropan-2-ol;formic acid 5-(4,6-dimethylpyrimidin-2-yl)oxy-6-ethylpyridine-3-carboxylic acid 2-methylpropane;(3Z)-5'-phenylspiro[cyclohepta-1,3,6-triene-4,9'-thioxanthene] 3-(3,5-difluorophenoxy)-N'-hydroxypyridine-2-carboximidamide 2-[(5-fluoropyridin-3-yl)amino]-4,7-dioxo-N-phenyl-6H-pyrimido[1,2-a]pyrimidine-9-carboxamide 7-methoxy-2-[4-[5-(2,3,4-trifluorophenyl)pyrimidin-1-ium-2-yl]oxycyclohexylidene]acetamide (NE)-N-[1-[4-bromo-2-[(3-chlorophenyl)methylamino]phenyl]ethylidene]hydroxylamine 1-[[2-fluoro-5-methyl-4-(3,4,5-trichlorophenyl)phenyl]methylsulfonyl]-N-[1-(trifluoromethoxy)piperidin-3-yl]piperidine-4-carboxamide N-cyclohexyl-2-(1,3-dimethylpiperidin-4-yl)-5,6,7,8-tetrahydroquinazolin-4-amine 1,2-difluoro-3-[(E)-4-methylpent-3-enyl]benzene;2-ethylpyrrolidine 2-[2,5-difluoro-4-(3-methylphenyl)sulfanylphenoxy]acetic acid 2-[3-chloro-4-(furan-2-ylmethoxy)phenyl]-6,7-dihydro-5H-imidazo[1,2-a]imidazole [2-cyclopropylimino-3-(2,6-dichlorophenyl)-1,3-thiazol-4-ylidene]methanol N'-[(E)-3-fluorobut-2-enyl]-4,7-dimethoxy-N,N-dipropylisoquinoline-1-carboximidamide 7,10-dibromo-2-phenyl-2H-benzo[c]chromene N'-methyl-3-[4-(5-methylidenepyridin-2-yl)pyrazol-1-yl]propanimidamide N-[3-(1H-imidazol-5-yl)propyl]-N',4-dimethylpiperidine-4-carbohydrazide 3-[6-(2,5-dimethylthiophen-3-yl)imidazo[1,2-b]pyridazin-2-yl]-2-oxopropanoic acid [(Z)-1-[2-[2,5-bis(trifluoromethyl)phenyl]propanoylamino]-3-hydroxyprop-2-enylidene]azanium 2-[4-(4-methylpyrimidine-5-carbonyl)morpholin-3-yl]benzoic acid 4-[(1R)-1-aminoethyl]-N'-hydroxypyridine-2-carboximidamide (3S)-1-benzylsulfanyl-N,N'-dimethyl-2-oxopyrrolidine-3-carboximidamide 1-[(2S)-2-amino-5-azidopentyl]-3-phenylurea 2-chloro-N,N'-dimethyl-1H-indole-6-carboximidamide 6-[(Z)-1,2-difluoroprop-1-enyl]-7H-purine 3,3-difluoro-N'-methyl-2-[(E)-2-(4-methylphenyl)ethenyl]propanimidamide 5-methyl-2-(3,4,5-trifluorophenyl)benzonitrile 6-bromo-N-diazo-1,3-benzothiazole-2-sulfonamide 1-(4-chlorophenyl)-2-(disulfanylmethoxy)propane-1,3-dione (2S)-2-[9H-fluoren-1-ylmethoxycarbonyl(methyl)amino]-4-oxobutanoic acid [2-amino-1-(4-aminophenyl)ethylidene]-phenylazanium 2-(5-azido-2,4-dimethylphenyl)pyridine 6-[(2S)-1,4-dioxan-2-yl]-3H-pyrido[3,2-d]pyrimidine-4,7-dione 2-(1-benzylpiperidin-4-ylidene)-7,8-dihydroimidazo[2,1-b][1,3]benzothiazol-1-one 2-[4-[2-[1-[5,6-bis(ethylamino)naphthalen-2-yl]sulfonyl-3-chloroindole-2-carbonyl]cyclopenten-1-yl]phenyl]acetic acid 1-[(2,6-dimethylphenyl)methoxy]-2-fluoro-4-propan-2-ylbenzene;N-methylethanesulfonamide 2-[(4S)-5,7-difluoro-3,4-dihydro-1H-isoquinoline-2-carbonyl]pyridine-4-carbonitrile 2-amino-6-ethoxy-4-(4-methylsulfanylphenyl)-4H-pyran-3,5-dicarbonitrile 2-[[(3R,4R)-4-(1H-indol-5-ylamino)oxolan-3-yl]oxymethyl]phenol 2-[[4-(trifluoromethoxy)phenyl]sulfanylamino]propanedioic acid N-(2,6-difluorophenyl)-5-fluoro-4-[3-methylbutyl(pentan-3-yl)amino]pyridine-3-carboxamide 4-[3-(1H-imidazol-2-yl)-1,2,4-oxadiazol-5-yl]phenol 1-[4-(3-azidophenyl)thiophene-2-carbonyl]azetidine-3-carbonitrile 4-methyl-2-[(5E,7Z)-9-propan-2-ylidene-1H-purin-6-yl]phenol 1-methylsulfinyl-5-[3-(trifluoromethoxy)phenyl]pyrrolidine-2,4-dione 2-[5-carbamoyl-9-[(3,4-difluorophenyl)methyl]-2-propan-2-ylcarbazol-4-yl]-2-hydroxyacetic acid 2-[3-(3-fluoropyridin-4-yl)oxypyrrolidin-1-yl]sulfonylthiophen-3-ol [4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]-(2-phenoxyphenyl)methanone 2-[3-(4,5-difluoro-1H-indole-2-carbonyl)phenyl]acetic acid (2S)-1-[5-[5,6-difluoro-1-[3-(4-methoxyphenyl)propanoyl]indol-2-yl]pyridine-3-carbonyl]pyrrolidine-2-carboxamide 3-(ethylamino)-N-[5-(methylsulfonylcarbamoyl)-1H-pyrazol-4-yl]benzamide 7-benzyl-4-(methylamino)-3-(1,2,3,6-tetrahydropyridine-4-carboximidoyl)-1H-quinolin-2-one 2-[2-(aminomethyl)morpholin-4-yl]-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-4-one;dihydrochloride 5-(2,6-dichlorophenyl)-4-ethyl-N-[3-(3-fluorophenoxy)phenyl]-1,2-oxazole-3-carboxamide (5Z)-3-ethyl-5-[[4-[4-methoxy-2-(trifluoromethyl)phenyl]phenyl]methylidene]imidazolidine-2,4-dione N-(2-methylphenyl)-N',3,4-trinitrobenzenecarboximidamide 6-[[4-(4-methylcyclohexyl)phenoxy]methyl]bicyclo[3.1.0]hexane 2-bromo-1,3,5,6-tetradeuterio-4-fluorobenzene (1R,2S)-N-[(2R)-1-amino-1-oxopropan-2-yl]-6-cyano-2-methoxy-3-naphthalen-2-ylcyclohexa-2,4-diene-1-carboxamide 2-[4-chloro-3-(pyridin-2-ylsulfanylmethyl)anilino]-N'-[(Z)-1,3-diaminoprop-2-enylidene]-6-(trifluoromethoxy)benzenecarboximidamide 4-[3-methylbutyl(prop-2-enyl)amino]benzenesulfonic acid 2-(5-bromonaphthalen-1-yl)-2H-chromene (3S,4R)-1-[6-chloro-8-(trifluoromethyl)imidazo[1,2-a]pyridine-7-carbonyl]-3-(5-methoxypyrazin-2-yl)piperidin-4-ol N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-ethanimidoyl-5-[(E)-1-[(1-hydroxycyclobutyl)amino]prop-1-enyl]-6-(1-methylpiperidin-4-yl)oxypyrazine-2-carboxamide N'-[[2,4-dichloro-3-[(4-phenylcyclohexyl)amino]benzoyl]amino]piperidine-1-carboximidamide (3S)-1-[4-[[2,6-difluoro-4-[(3R)-3-hydroxypyrrolidine-1-carbonyl]phenyl]methyl]-5H-cyclopenta[b]pyridin-7-yl]piperidine-3-carboxylic acid ethane;1-[3-methyl-4-(2-phenylethenyl)thiophen-2-yl]propan-2-one 4-azidooxy-6,7-dimethoxy-2H-benzotriazole N'-cyclohexyl-N-[6-(3,5-dimethoxyphenyl)pyridin-3-yl]-4-(4-propanoylpiperazin-1-yl)piperidine-1-carboximidamide 4-[(1R,3E)-3-azido-2-fluorohexa-1,3,5-trienyl]pyridine N-[[1-(2,6-dimethylpyrimidine-4-carbonyl)pyrrolidin-3-yl]methyl]-5-ethylthiophene-2-carboxamide (2R)-N-[5-[[1-[4-[bis(prop-1-en-2-yloxy)phosphoryl]butanoylamino]piperidin-4-ylidene]methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]azetidine-2-carboxamide 5-[2-(difluoromethyl)pyridin-4-yl]pyridine-3-carbonitrile 5-butanoyl-1-phenylindazole-3-carboxylic acid 3-chloro-4-[[(E)-2,6,10,11-tetramethoxy-8,9-dimethyl-5-oxa-1-azatricyclo[7.3.0.02,6]dodeca-2,7,9,11-tetraen-12-yl]amino]sulfanylbenzoic acid N-[(3S,7R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]benzamide 1-[5-chloro-2-(4,4-difluoropiperidin-1-yl)pyrimidin-4-yl]ethanol;5-(dimethylaminosulfanyl)-3-methylimidazo[4,5-c]pyridine-6-carbonitrile 5-[(1S)-2-[[5-(3-cyanophenyl)pyridine-2-carbonyl]amino]cyclohexyl]pentanoic acid (Z)-1-N-benzyl-3-hydroxyimino-2,5,6,7,8,8a-hexahydrocyclopenta[b]naphthalene-1,6-dicarboxamide;ethane 1-[3-cyclopropyl-4-(pyridine-2-carbonyl)piperazin-1-yl]-2-(4,5-difluorothiophen-2-yl)ethanone (3S)-3-[2-oxo-2-[4-(trifluoromethoxy)phenyl]ethyl]pyrrolidine-1-carboxylic acid 4-(1H-indol-5-ylmethyl)quinazoline N-[(3,5-dibromopyridin-4-yl)methylideneamino]acetamide 2-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]-5,7-difluoro-6-pentoxy-1,4-dihydronaphthalene 2-[3,4-difluoro-5-(trifluoromethyl)phenyl]-5,7-diethoxynaphthalene N'-[amino(methyl)amino]-2-(trifluoromethyl)benzenecarboximidamide 2-[N-(carboxymethyl)anilino]benzenesulfonic acid 5-(1H-indazol-4-yl)-N-methoxythiophene-2-sulfonamide 4-(4,6-diamino-1,3,5-triazin-2-yl)naphthalene-1-sulfonic acid 4-tert-butyl-2,5-dimethoxy-N-(3-pyridin-2-yl-1H-indazol-6-yl)benzamide N-[(Z)-1H-indol-3-ylmethylideneamino]-2-phenylmorpholine-4-carboxamide 2-(3,4-dimethylcyclohexa-1,5-dien-1-yl)oxy-N-[6-(piperidine-1-carbonyl)pyridin-2-yl]acetamide 4-[(2E,3S)-6-aminohepta-2,5-dien-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-amine 4-azidosulfanyl-2-chloro-6-methoxyphenol 3-azido-5-bromo-2-(4-methylsulfonylpiperazin-1-yl)pyridine 4-[2-[[(5S)-9-fluoro-3-methyl-6,7-dihydro-5H-pyrimido[5,4-d][2]benzazepin-2-ylidene]amino]ethyl]phenol 3-(2,4-dihydroxyphenyl)-4-[4-(4-fluoroanilino)-1-(oxan-2-yl)pyrazolo[3,4-b]pyridin-5-yl]butanoic acid N-[5-(aminomethyl)-1,3-thiazol-2-yl]-4-(4-hydroxyphenyl)benzamide N-[3-(1,2,4-triazol-1-yl)phenyl]prop-2-enamide 2-[4-(3,4-dihydronaphthalene-1-carbonyl)piperazine-1-carbonyl]-1-methylquinolin-4-one 2-[4-chlorobutyl(naphthalen-1-yl)amino]acetamide 1-[3,5-difluoro-2-(4-nitrophenyl)phenoxy]propan-2-one [5-fluoro-3-methyl-6-(2H-pyrazolo[1,5-a]pyrimidin-7-yl)cyclohexa-1,5-dien-1-yl]-[4-(3-hydroxypiperidine-1-carbonyl)piperazin-1-yl]methanone 4-[1-(4,5-dimethylcyclohexa-2,4-dien-1-yl)buta-1,3-diynyl]naphthalene 1-(2-bromoethyl)naphthalene 1-[1-(3-chloro-4-fluorophenyl)-5-hydroxypyrazole-4-carbonyl]piperidine-2,6-dione 1-[2,3-difluoro-4-(4-methylcyclohexyl)phenyl]ethanone 3-[(2,3-dihydroxyphenyl)methylidene]-5-ethyliminocyclohexan-1-ol 1-azidooxy-2,3,4,5-tetrabromobenzene 2-chloro-N,3,6-trimethylimidazo[1,2-a]pyrazin-8-amine N-[3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-6-propan-2-ylidenecyclohexa-2,4-dien-1-imine [(4aS)-3,4a,5,6,7,8,8a-octahydro-2H-benzo[b][1]benzofuran-4-yl]methanamine;hydrochloride 2-methyl-6,12,12a,14a-tetrahydroindolo[3,2-d][1]benzazepine (2R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-pyridin-4-ylsulfonylpyrrolidine-2-carboxamide [4-[(2S)-1,1-dioxothiazetidine-2-carbonyl]piperazin-1-yl]-[4-fluoro-3-methoxy-5-[6-[2-(methylamino)pyrimidin-5-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]methanone 6-(2,3-dihydroindole-1-carbonyl)-5H-pyrrolo[3,4-b]pyridin-7-one 7-methyl-N-propanoyl-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamide N-[5-(1H-indole-3-carbonyl)pyridin-2-yl]spiro[3.4]octane-6-carboxamide 4-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethynyl]-N-[(4S)-5-(hydroxymethyl)-6-oxo-8,9-dihydro-7H-pyrido[3,2-c]azepin-10-yl]pyridine-2-carboxamide 2-[[2-(4-oxo-3H-quinazolin-2-yl)spiro[3.5]nonan-7-yl]amino]ethanesulfonic acid 1-(2,6-dimethylphenyl)-3-(N'-hexanoylcarbamimidoyl)urea 5-(1,3-benzothiazol-2-yl)-4-[[5-[3-ethoxypropyl(methylsulfonyl)amino]naphthalen-1-yl]diazenyl]-2-hydroxybenzenesulfonic acid 2-[4-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]pyrazol-1-yl]ethanamine;hydrochloride 2-[(4-chlorophenyl)methylsulfanyl]-N'-hydroxypyrimidine-4-carboximidamide 1-(4-methylphenyl)sulfonylpyrrole-2,5-dione 3-(2,2,4,5-tetrafluorocyclopenta-1,3-dien-1-yl)oxyphenol 5-[6-(aminomethyl)pyridin-2-yl]sulfonyl-3,4-dihydro-1H-isoquinoline-2-carboxylic acid;hydrochloride 3-chloro-N-[(3S,4R)-1-methylsulfonyl-4-phenylpyrrolidin-3-yl]-4-[[5-(trifluoromethyl)pyridine-2-carbonyl]amino]benzamide N-(1,3-benzodioxol-5-yl)-4-[[2-(2,4-dichlorophenoxy)acetyl]amino]piperidine-1-carboxamide N-[(3S)-2,5-dioxopyrrolidin-3-yl]-5-(4,6-dimethoxypyridin-2-yl)thiophene-2-carboxamide 2-amino-4,6-di(propan-2-yl)benzenesulfinic acid;ethane (3S)-5-hydroxy-1',6-dimethylspiro[3H-chromene-2,4'-piperidine]-4-one 2,3-dimethyl-N-[1-(trifluoromethyl)cyclopropyl]thiophene-4-carboxamide (E)-1-[4-hydroxy-6,7-dimethyl-2-[4-[3-oxo-5-(trifluoromethyl)-1H-isoindol-2-yl]phenyl]-1-benzofuran-3-yl]-3-(4-propan-2-yloxyphenyl)prop-2-en-1-one 2-(3,5-dibromophenyl)-4,6-dimethylpyridine 2-(2,6-dioxopiperidin-3-yl)-5-[[1-methyl-2-(methylaminomethyl)indol-4-yl]methoxy]isoindole-1,3-dione;dihydrochloride 2-(4-fluorophenyl)sulfanylethanethiol;2-methoxyethanol 4-[3-(2-azidoethoxy)phenoxy]aniline 2-methyl-1-[5-(6-phenylimidazo[1,5-b]pyridazin-3-yl)pyridin-2-yl]propan-1-one 2-[(E)-1H-indol-3-ylmethylidenehydrazinylidene]-4,5-dihydro-1,3-thiazol-4-ol 2-[3,5-dichloro-4-(hydroxymethyl)phenyl]acetonitrile 2-[(5-chloropyridin-3-yl)methoxy]-1,7-dihydropurin-6-one N-[1-(3,4-dimethoxyphenyl)piperidin-4-yl]-5-(2,6-dioxopiperidin-3-yl)pentane-1-sulfonamide 2-[4-(6,7-dichloroquinoxalin-2-yl)piperazin-1-yl]ethanol (3S)-2',7-difluorospiro[1,3-dihydroindene-2,3'-5H-pyrazolo[1,5-a]pyrimidine]-4'-one 2-chloro-5-[4-[[(1S)-3,3-difluorocyclopentyl]amino]-2-methoxyphenyl]-N-pyridin-3-ylpyrimidine-4-carboxamide 2,7-diazaspiro[4.5]decan-3-yl-(2-imidazo[1,2-a]pyridin-6-ylpyridin-3-yl)methanone [5-[5-[[1-(4-chlorophenyl)cyclopropyl]sulfamoylmethyl]-2,3-dihydroindole-1-carbonyl]thiophen-2-yl]chloranium N-[1-[3,5-bis(trifluoromethyl)phenyl]ethenyl]-4-chlorocycloheptan-1-amine;4-piperidin-1-ylbutanenitrile 6-(4-methylphenyl)imidazo[2,1-b][1,3]benzothiazole 5-N-[2,4-dichloro-3-(1H-indole-2-carbonyl)phenyl]-7-ethoxyquinazoline-2,5-diamine 2-[1-(4,5-dimethylpyrimidine-2-carbonyl)piperidin-3-yl]sulfanylpyridine-4-carbonitrile (6R)-4-[2-hydroxyethyl-(1-methoxycyclohexanecarbonyl)amino]-3,8-dioxo-7-thiatricyclo[5.3.0.02,6]deca-1(10),2,4,12-tetraene-9-carboxylic acid 2-(3,5-dimethylphenyl)sulfanylacetic acid N-[2,4,7-tris(sulfanylidene)-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidin-3-yl]acetamide (5S)-N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2,6-dimethoxybenzoyl)-2-methylidene-4,5-dihydrocyclopenta[b]pyridine-5-carboxamide [5-chloro-6-(2,3,4a,8a-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carbonylamino)cyclohexa-1,3-dien-1-yl]carbamic acid 1,2-diethylpyrene [4-amino-2-(3-chloropyridin-2-yl)imino-5,6,7,8-tetrahydronaphthalen-1-ylidene]-oxoazanium 2-[5-chloro-3-methyl-4-(2,4,6-trifluorophenyl)-1H-pyrrol-2-yl]pyridine 5-chloro-N',6-dihydroxy-2-(3-methylbutanoyl)pyridine-3-carboximidamide 2,3-diethyl-1H-benzimidazole-2-sulfonate 2-[[(Z)-3,4-dioxopent-1-enyl]carbamoyloxymethyl]benzoic acid 1-(3,4-difluorophenyl)-2-(6-propylimidazo[1,2-b]pyridazin-3-yl)hydrazine 4-fluoro-N-[(E)-(2-hydroxyphenyl)methylideneamino]benzamide 1-(1-cyclohexylbenzimidazol-2-yl)-N,2-dimethylpiperidine-4-carboxamide N-[(Z)-2-aminoethenyl]formamide;2,3-dichloro-5-cyclopropylpyrazine 7-(2,3-dihydrothiophen-4-yl)-N-methoxyimidazo[1,2-a]pyridine-2-carboxamide 1-chloro-4-methylbenzene;N,N',4-triaminoquinazoline-7-carboximidamide 2-[4-(6,7-dihydro-1H-indazol-5-yl)phenyl]-N'-[4-(methoxysulfanylamino)butanoyl]-2-prop-2-ynylbutanehydrazide 2-(1,5-dimethylpyrazol-3-yl)-7-[(4-fluorophenyl)methyl]-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one (4R)-4-[2-(3,5-dimethylanilino)-1H-benzimidazol-4-yl]-6-methoxy-2,2-dimethylhexanamide N-[4-(diethylamino)phenyl]-3-nitroquinoxalin-2-amine 1-[4-(3-acetylphenoxy)pyridin-2-yl]cyclobutane-1-carbonitrile 5-[(E)-1,2-bis(4-hydroxyphenyl)ethenyl]-N-[5-(1,1-difluoropropoxy)pentyl]-1H-imidazole-4-carboxamide 1-(2,3-dihydroindol-1-yl)-4-[[5-(1H-imidazol-2-yl)pyridin-2-yl]amino]butan-1-one;dihydrochloride 2-azidooxy-1,3,5-trichloro-4-(2-ethylphenoxy)benzene N-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-9H-pyrido[2,3-b]indole-3-carboxamide 1-(1,3-benzodioxol-5-yl)-N'-tert-butyl-4-ethoxycyclohexa-2,4-diene-1-carbohydrazide 6-[3-[4-(2,6-difluorophenyl)piperazin-1-yl]propoxy]pyridine-2-carboxamide (5Z)-2-[4-chloro-3-fluoro-2-methyl-6-(trifluoromethyl)phenyl]imino-5-[[3-ethoxy-4-hydroxy-5-(1,1,2,2,2-pentafluoroethyl)phenyl]methylidene]-1,3-thiazolidin-4-one 4-[1-(2,6-dimethylphenyl)imidazole-2-carbonyl]-1H-pyrrole-2-carbonitrile 2-[4-methyl-6-[(4-pentan-3-ylphenyl)methoxy]cyclohexa-1,3-dien-1-yl]acetic acid 1-[(E)-2,3-difluorobut-2-enyl]-3-[4-[[4-(5,6-dihydronaphthalen-1-ylmethoxy)phenyl]sulfonylamino]butyl]urea 3-amino-N'-(4-chlorophenyl)-6-methylsulfanylpyridazine-4-carboximidamide 1-[3,4-dimethoxy-5-(2-phenylethynyl)phenyl]ethanol (3S,4R)-N-[2-methyl-5-(1-methylpyrazol-4-yl)phenyl]-4-oxopyrrolidine-3-carboxamide ethane;2-methylpropyl-(4-piperidin-1-ylpyridin-3-yl)phosphane (3R,4S)-1-[2-(1H-benzimidazol-2-ylmethoxy)ethyl]-4-(quinoline-2-carbonylamino)piperidine-3-carboxylic acid 2-amino-6-[(E)-3-methoxyprop-1-enyl]pyridine-4-carboxylic acid 2-[[5-(5-methylthiophen-2-yl)thiophen-2-yl]sulfonylamino]-3,4-diphenylbutanoic acid 3-(1-methylpiperidin-4-ylidene)-N-propan-2-ylnaphthalene-2-carboxamide 1-(2,5-dimethylcyclohexa-1,3-dien-1-yl)butan-2-ol;[2-methoxy-4-[6-(trifluoromethyl)pyridin-3-yl]phenyl]urea 1-chloro-3-(5,6,7,8-tetrahydronaphthalen-2-yl)propan-2-ol 4-[5-chloro-2-(difluoromethoxy)phenyl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 2,6-ditert-butyl-4-[(2S)-1-hydroxypropan-2-yl]phenol (3Z,5E)-N-[2-chloro-4-(1H-indol-4-yloxy)phenyl]-4-ethenylhepta-1,3,5-trien-2-amine;(Z)-but-2-ene 1-(4-propan-2-ylphenyl)sulfonylpiperidine-3-carboxylic acid (2R)-4-[7-chloro-1,3-benzodioxol-5-ylmethylsulfanyl]-2-propan-2-yl-2H-chromene 1-[2,6-difluoro-4-(3-methylbutanoyl)phenyl]-3-methylidenepiperidine-4-carbonitrile 3-[4-methoxy-3-(3-phenylprop-1-ynyl)phenyl]-5-(trifluoromethyl)-2,3-dihydro-1H-pyrazole 5-[4-fluoro-3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]-N,N-dimethylpyridin-3-amine 2-methyl-1,3-dihydroisoindole;4-(2,2,2-trifluoroethyl)benzaldehyde 3-[2,4-dichloro-5-(4-hydroxyoxan-4-yl)phenyl]-1-methyl-6-(trifluoromethyl)pyrimidine-2,4-dione ethane;3-[[3-(2-ethenylphenyl)cyclohepta-1,4,6-triene-1-carbonyl]amino]pentanoic acid 3-[5-(2,3-dihydro-1H-inden-4-yl)-6,7-dimethoxy-1,3-benzoxazol-2-yl]cyclohexa-1,5-dien-1-amine N-[2,6-diamino-3-(4-methylphenyl)sulfinylphenoxy]benzamide 4-fluoro-2-(1H-indol-5-yliminomethyl)phenol 1-cyclopropyl-3,4-dimethylbenzene;N,N-diethyl-5-fluoro-4-([1]benzofuro[2,3-d]pyrimidin-7-ylamino)piperidine-1-carboxamide 6-[(1R,3S)-3-hydroxycyclopentyl]-2-methoxy-5H-pyrrolo[3,4-b]pyridin-7-one 3-[2-hydroxyethyl(methylamino)amino]naphthalene-1,4-dione 2-bromo-4-methoxy-3,5-dimethylbenzoate 3-[4-(3,5-difluoroanilino)phenyl]-2-hydrazinylpropanoic acid N-(2,4-dimethylphenyl)-3,5-bis[(4-fluorophenyl)sulfanyl]-1,4-dihydroxynaphthalene-2-carboxamide 4-azido-5-ethyl-3-phenylpyridazine 2-[5-(4,7-dimethylcycloocta-1,3,6-trien-1-yl)thiophen-2-yl]-N-(1H-indol-6-yl)butanamide 6-[2,6-difluoro-4-(hydroxymethyl)phenyl]-1,3-benzothiazole-2-carbonitrile 2-N,4-N-bis[(2S)-butan-2-yl]quinoline-2,4-dicarboxamide 2-ethylsulfanyl-7,8-dihydro-6H-thiopyrano[3,2-d]pyrimidine 1-phenyl-2,5-dihydropyrrole;1-(4-pyridin-3-yl-1H-indazol-7-yl)ethanone N-[(1R,2S)-2-hydroxycyclohexyl]-7-[(6-methoxypyridin-3-yl)amino]-5H-pyrimido[4,5-b][1,4]oxazepine-2-carboxamide N-azido-2,4-dichloro-5-(dimethoxyphosphorylcarbamoyl)benzamide 4-azido-2,6-dibromopyrimidine 3-(4-benzylsulfonylphenyl)cycloheptan-1-one 6-[4,5-bis(trifluoromethyl)pyridin-2-yl]oxyhexanoate 3-(4,5-diethylpyridin-2-yl)-7-oxa-1,10-phenanthroline N-azido-6,7-dichloro-2-methylquinoline-3-carboxamide [6-(3,4-dimethoxyphenyl)pyrazin-2-yl]-piperidin-1-ylmethanone 1-[3-(3-chloro-4-fluorophenyl)-2H-tetrazol-3-ium-5-yl]pentan-3-one 4-fluoro-2-methyl-N-[1-oxo-6-(trifluoromethyl)phthalazin-2-ium-2-yl]benzamide 6-(N-[2-methylpropanoylamino)phenyl]-7-phenylmethoxy-1H-indole-2-carboxylic acid N-[1-(2,3-dihydroindol-1-yl)ethylidene]-4-iodobenzamide 2,2-dichloro-3-[4-(2,6-dichlorophenyl)phenyl]cyclopropane-1,1-dicarbonitrile 5-bromo-2-[3,3-bis(4-methylphenyl)-2-oxopyrrolidin-1-yl]benzoic acid 2-[(4-fluorophenyl)methylimino]-5-[(4-hydroxy-3,5-diiodophenyl)methylideneamino]-1,3-thiazolidin-4-one 1-N,3-N,6-trimethylpyrazolo[3,4-d]pyrimidine-1,3-diamine (2S)-1,1,1-trifluoro-3-(methylamino)-4-[6-(3H-pyrrol-5-yl)imidazo[1,2-a]pyridin-8-yl]butan-2-ol 1-[7-(azidomethyl)naphthalen-2-yl]-1,1-difluoropropan-2-one 5-azidooxy-3,4-dimethyl-6-(2H-triazol-4-yl)pyridine 1,5-dibromopentylbenzene 2-(2,6-dioxopiperidin-3-yl)-5-[4-[1-[(Z)-N'-ethenoxycarbamimidoyl]cyclopropanecarbonyl]piperazin-1-yl]isoindole-1,3-dione 3-azidosulfanyl-4-ethenoxypyridine N-ethenyl-1,6-diphenylpiperidine-2-carboxamide 4-[6-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)pyrrolo[2,3-b]pyridin-1-yl]benzoic acid 4-amino-3,5,6-trifluorophthalic acid 6-ethyl-1,3-dimethoxynaphthalene 1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxycarbonylnaphthalene-2-carboxylic acid 2-methylsulfanyl-3,4-dihydroisoquinolin-1-one;(2S)-N-[2-[(5-phenyl-1H-1,2,4-triazol-3-yl)amino]ethyl]propane-2-sulfonamide (2S)-2-azido-N-[1-[4-[(4-methylphenyl)sulfamoyl]benzoyl]piperidin-3-yl]-3-phenylpropanamide 2,4-difluoro-6-[(3S)-1-(triazol-1-ylmethylsulfonyl)pyrrolidin-3-yl]oxybenzoic acid ethane;6-[(5S)-2,7,11-trimethyldodeca-2,9,12-trienoxy]quinoline 2-(4-azidophenyl)-1-benzothiophene 4-[3,5-bis(trifluoromethyl)phenyl]-6-chloro-2-sulfanylidene-1H-pyrimidine-5-carbonitrile [5-[1,3-bis(ethenyl)-2-methylidenebenzimidazole-5-carbonyl]-2-[methanimidoyl(propyl)amino]phenyl]azanide 4-hydroxy-6-[2,3,5,7-tetrafluoro-9H-fluoren-1-yl]pyridine-3-carboxylic acid 2-(2,6-dimethylanilino)-4-propan-2-yl-1H-pyrimidin-6-one 2-(azidomethyl)-N,3-diethylaniline 2-(3,4-difluorophenyl)acetate N-[2,4,6-trimethyl-3-(1H-pyrazol-5-yl)phenyl]methanesulfonamide (Z)-N'-amino-2-[5-methyl-3,4-dioxo-6-[(E)-propan-2-ylideneamino]pyrazin-2-yl]pent-4-enimidamide 3-(1,2,4-triazol-1-yl)isoquinoline 2-amino-4-[3-(dimethylamino)phenyl]-6,8-bis(2-morpholin-4-ylethoxy)pyrimido[5,4-f]quinoxaline-9,10-dione 1,4-difluorobenzene;2,3,6,7-tetramethylimidazo[2,1-b][1,3]thiazole 2-methyl-N-[5-[3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]propanamide 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonylamino)butanoic acid [(1S,5R)-8-amino-4-azabicyclo[3.2.1]octan-4-yl]-[2-fluoro-6-(1,3-thiazol-5-yl)phenyl]methanone 2-(cyclopropylmethoxy)-N-[6-[4-(1,3-dihydroxy-3,4-dihydroisoquinoline-2-carbonyl)piperidin-1-yl]pyridin-3-yl]benzenesulfonamide 2-azidosulfanyl-5,6-dimethoxy-1H-benzimidazole (5R)-3-amino-N-[(1S)-1-(4-fluorophenyl)ethyl]-5-methoxyhexanamide;hydrochloride 1-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-2,6-dihydropyridine-4-carboxylic acid 2-cyclohexyl-4,6-bis[(2E)-3,7-dimethylocta-2,6-dienoxy]-1,3,5-triazine 2-(3-methylbutanoyl)oxybenzoic acid 1-[4-(5-chloropyridine-3-carbonyl)piperazin-1-yl]-2-pyridin-4-ylethane-1,2-dione (2S)-1,5-bis[3-(cyclopropylmethoxy)phenyl]pentan-2-ol 2-benzylsulfanyl-6,7-dimethoxy-1H-phenanthro[9,10-d]imidazole 2-[3-(1,4-dioxaspiro[4.5]decan-8-yl)phenyl]pyridine 1-[[4-[(3Z)-2,5-dimethylhexa-1,3,5-trien-3-yl]phenyl]methyl]piperidine 3-(6,7-dimethoxyquinolin-4-yl)oxy-N'-hydroxybenzenecarboximidamide 2-[5-azido-6-(4-chlorophenoxy)pyridin-3-yl]-1,3-thiazole 1-methyl-4-[4-[(6-methylidenecyclohexa-2,4-dien-1-yl)oxymethyl]phenyl]benzene 1-(3-chlorophenyl)-4,5-dimethylpyridin-2-one 2-methylpropan-1-ol;3-(5,6,7,8-tetrahydronaphthalene-2-carbonylamino)benzoic acid 1-[2-fluoro-4-(trifluoromethyl)phenyl]sulfonyl-5,5-diphenylpiperidine 1-methoxy-3-[3-[4-(pyridine-2-carbonyl)phenyl]propylamino]propan-2-one N-[2,4,6-trimethyl-3-(1-phenylbutan-2-yl)cyclohexa-1,5-dien-1-yl]-2H-benzotriazole-4-carboxamide 2-[4-(dimethylamino)pyrimidin-5-yl]oxyacetate 4-methyl-3-[(5-oxo-6,7,8,9-tetrahydroimidazo[1,2-a]quinazoline-3-carbonyl)amino]butanoic acid N-[4-[2-[(5-chloropyridine-3-carbonyl)amino]ethylcarbamoyl]-1,3-thiazol-5-yl]-6-fluoro-2-methylpyridine-3-carboxamide 5-(2-azidopropan-2-yl)-3-chlorothiophene 1,3-bis(2-iodophenyl)urea 1-ethenyl-3-[(4-methoxyphenyl)methyl]-6,7-dihydronaphthalene 2-[(2R)-1-methoxycarbonylpyrrolidine-2-carbonyl]benzenesulfonic acid 4-(3,5-dimethylphenyl)-7-[4-(trifluoromethoxy)phenyl]-2,1,3-benzothiadiazole 3-bromo-4-[2-(3,5-ditert-butyl-4-hydroxyphenyl)ethyl]-1H-indole-7-carboxamide 4-[(2R)-3-azidobutan-2-yl]-1,2-bis(phenylmethoxy)benzene 5-methyl-3-(trifluoromethyl)-N-[5-[6-(trifluoromethyl)pyridazin-4-yl]pyridin-2-yl]-1,2-oxazole-4-carboxamide ethane;methanamine;1-(5,6,7,8-tetrahydroisoquinolin-1-yl)piperidine 2-[[4-(3,4-dichlorophenyl)-5-propan-2-ylsulfanylpyridin-3-yl]amino]butanedioic acid 2-[4,5-bis(ethenyl)-1H-pyrazol-3-yl]phenol ethane;2-[3-(methylamino)phenyl]imidazo[1,2-a]pyrimidine-7-carboximidamide 1,5-dimethyl-2-(2-propan-2-ylphenyl)imidazole N-[6-(2,4-dichloro-3-methylphenoxy)hexan-3-yl]acetamide N-(2-hydroxyethyl)-3-[4-[1-[4-(2,2,2-trifluoroethoxy)phenyl]-1,2,4-triazol-3-yl]phenoxy]pyrrolidine-1-carboxamide (2R,3S)-4-[(1-benzylpiperidine-2-carbonyl)amino]-5-methoxy-3-methyl-N-[(4-methylphenyl)methyl]-2-propan-2-ylhexanamide 2-[4-(6-methoxy-1H-benzimidazol-2-yl)phenoxy]ethanol 1-[4-[2-(azepan-1-yl)ethoxy]phenyl]-3-(2-methylphenyl)urea 7-[(4-aminophenyl)methyl]-2-methylsulfinyl-8H-pyrimido[5,4-b][1,4]oxazin-6-one 5-(3,4-dimethylphenyl)-2-[4-(7-fluoroquinolin-6-yl)butyl]-4H-1,2,4-triazol-3-one 4-[[2,6-dichloro-3-(ethoxymethyl)phenyl]methylideneamino]aniline [5-(3,5-dimethoxyphenyl)-2,2,4-trimethylpentanoyl]phosphonamidous acid 4-hydroxy-3,5,6-trimethyl-N-(2-morpholin-4-ylethyl)-1,4-dihydroquinoline-2-carboxamide 3-[(2S)-1-hydroxypropan-2-yl]-7-methoxy-6H-quinoline-5,8-dione 2-(1H-benzimidazol-2-ylmethylcarbamoyl)azetidine-3-carboxylic acid 4-[6,7-dimethoxy-2-(1H-pyrazol-5-yl)quinoline-3-carbonyl]piperazine-1-carboxylic acid 2-[6-[5-(hydroxymethyl)-1,3,4-oxadiazol-2-yl]pyrazolo[3,4-b]pyridin-1-yl]-N-[2-hydroxy-5-(trifluoromethoxy)phenyl]acetamide 1-(3,4-dimethoxyphenyl)heptane-3,5-dione [3-cyclopropyl-3-(5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-3-carbonylamino)azetidin-1-yl]oxyboronic acid (1R)-2,2-dimethyl-N-[6-[5-[(5-phenyl-1,3,4-oxadiazol-2-yl)amino]-1,3,4-thiadiazol-2-yl]pyridin-2-yl]cyclopropane-1-carboxamide 6-[4,6-difluoro-2-(1-fluoroethoxy)phenyl]-3-[4-ethyl-5-oxo-3-(trideuteriomethyl)-1H-pyrazol-2-ium-2-yl]-5-fluoro-1-methylpyridin-2-one N-cyclopropylformamide;1-(2,5-dimethoxyphenyl)azetidine N-[[(3S,4S)-1-methyl-4-phenylpyrrolidin-3-yl]methyl]spiro[2.5]octane-6-carboxamide N-[(3-azidocyclohexyl)methoxy]pyridine-2-carboxamide 2-[4-ethyl-5-(3-phenyl-1H-pyrazole-5-carbonyl)-6,7-dihydronaphthalen-1-yl]acetic acid 2-[[4-[4-(trifluoromethoxy)phenyl]phenoxy]methyl]oxirane 3-ethoxy-N',2-dihydroxy-5-(4-pyridin-4-ylphenyl)benzenecarboximidamide 2-amino-1,3-dimethyl-4-[(Z)-prop-1-enyl]quinolin-1-ium-6-ol 1-[6-(4-fluorophenyl)-8-methyl-7H-carbazole-3-carbonyl]piperidin-2-one N-[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]formamide;6-[4-chloro-3-[methyl(propan-2-ylsulfonyl)amino]phenyl]quinazoline-8-carboxylic acid N-ethylsulfonyl-2,4,6-trimethyl-N-(3-nitrophenyl)benzenesulfonamide 2-amino-9-(2,5-dimethyloxolan-3-yl)-1H-purin-6-one;methanamine (5R)-3-(4-methoxyphenyl)-2,7,7-trimethyl-1-[4-(4-methylphenyl)butyl]-6,8-dihydroquinoline-4,5-dione 2-[(E)-1,1-bis[4-(dimethylamino)phenyl]but-1-enyl]-6-tert-butylphenol 4-azidooxy-1H-indazole 4-[3-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)phenyl]benzonitrile 6-methylsulfonyl-2-phenyl-3,4-dihydro-1H-isoquinoline (1S)-N-[(Z,4R)-6-amino-7-ethoxy-2-hydroxy-8-oxooct-7-enyl]-3,5-diphenylcyclohexa-2,4-diene-1-carboxamide 5-chloro-2-[(1R)-3,3-dimethylcyclohexyl]oxypyridine;hydrochloride 3-[4-(cyclopentylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile 6-azidooxy-1H-indole-2,3-dicarboxylic acid (2-benzyl-2-methoxyheptyl)benzene 5-[(4S)-5-ethoxy-4-hydroxypentyl]sulfanyl-1,2-dimethylnaphthalene-6,7-diol 2-cyclopropyl-1',4-dimethoxyspiro[chromeno[3,4-d]imidazole-7,4'-piperidine] N-(4-hydroxybutyl)-6-nitro-N-octyl-1,3-benzothiazol-2-amine [1-[[(2S)-1-[3,3,3-trifluoro-2-methoxy-2-phenylpropanoyl]pyrrolidin-2-yl]methylcarbamoylamino]cyclopentyl]urea 3-[4-(3,6-diamino-2H-1,4-thiazin-5-yl)phenyl]propanoic acid N-[2-[(5R)-2-(1,3-benzothiazol-6-ylimino)-4-oxo-1,3-thiazolidin-5-yl]ethyl]thiophene-3-carboxamide (6-ethoxy-3,4,5-trimethoxycyclohexa-2,4-dien-1-yl)-phenylmethanone [(3R)-1,2,3,4,6,7,8,9-octahydropyrimido[1,2-a]indol-3-yl]-(6-propan-2-yloxypyridin-2-yl)methanol N-(2-phenylethyl)-3,7,11,16-tetrazatetracyclo[8.6.0.02,7.012,15]hexadeca-1,9,11(15),13-tetraene-14-carboxamide N-[(1R,2S)-2-aminocyclohexyl]-5-chloro-2-oxo-3H-benzimidazole-1-carboxamide;hydrochloride 6-(4,5-difluoro-1H-pyrazol-3-yl)-2-[(3R,4S)-3-hydroxypiperidine-4-carbonyl]-3-phenyl-7,8-dihydroquinolin-5-one (3aR,6aS)-5-[2-(5-methylthiophen-2-yl)acetyl]-1-(pyridin-4-ylmethyl)-3,3a,4,6a-tetrahydropyrrolo[3,4-c]pyrrole-2,6-dione;2,2,2-trifluoroacetic acid 4-[4-(oxiran-2-ylmethoxy)phenyl]-6,8-dihydro-5H-thiopyrano[3,4-d]pyrimidine N-[5,8-dimethoxy-2-(3-phenylpropyl)quinolin-7-yl]-4,6-difluoronaphthalene-1-carboxamide 2-(cyclohexylmethyl)-6,7-difluoroquinoxaline [5-hydroxy-8-(hydroxymethyl)quinolin-7-yl]iodanium 1-[3-(6-chloro-2,7,8,9-tetrahydro-1H-pyrano[2,3-d]azepine-4-carbonyl)phenyl]ethanone N-[(Z)-1-(1,3-benzodioxol-5-yl)ethylideneamino]-7-iodoquinoline-3-carboxamide 1-[4-(4,5-dimethylpyrimidin-2-yl)piperazin-1-yl]-3-quinolin-8-yloxypropan-2-ol (2S)-3,3-dimethyl-1-[4-[[6-(2H-tetrazol-5-yl)pyridin-3-yl]oxymethyl]piperidin-1-yl]butan-2-ol 2,4-dichloro-N-[(3R)-1-methylpyrrolidin-3-yl]benzenesulfonamide 2-(4,6-dimethylpyrimidin-5-yl)acetic acid;3,3a,7a-trimethyl-1-[(E)-prop-1-enoxy]azetidine N-(6-chloropyridin-3-yl)-2,4,6-trimethyl-N-phenacylbenzenesulfonamide 5-(2-diazohydrazinyl)-6-oxo-1H-pyrimidine-4-carboxylic acid 1-ethyl-3,5-difluorobenzene;2-(4-methylpiperazin-1-ium-1-ylidene)-6-oxohexanal 4-[(4-bromo-2,3-dihydroxyphenyl)methyl]piperazine-1-carboxylic acid (E)-2-benzylsulfanyl-3-[(E)-2,4,8-trimethylnon-5-en-6-ylideneamino]prop-2-enenitrile;cyclopentanol;ethane 1-(2,4-dimethyl-6-oxo-1H-pyrimidine-5-carbonyl)-N,N-diethylazetidine-3-sulfonamide 2,6-dimethyl-4-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrazine;ethane (E)-N'-[(2,6-dimethoxyphenyl)-[4-[4-(trifluoromethyl)anilino]pyridin-1-ium-1-yl]methylidene]ethanimidamide 3-[[2,6-bis(ethenyl)pyridin-4-yl]methoxy]-N-cyclohexa-1,5-dien-1-yl-4-[(E)-4-fluorohept-2-en-3-yl]benzamide 3-[4-(azidomethyl)phenyl]-5-[4-chloro-2,6-difluoro-3-(phenylsulfanylamino)phenoxy]benzonitrile 3-N,3-N-diethyl-1H-indazole-3,6-dicarboximidamide 5-[4-(2,3-difluoro-4-propoxyphenyl)cyclohexyl]-1,3-difluoro-2-(trifluoromethyl)benzene 2-amino-6-chloro-8,9,10-trihydroxy-1H-tetracene-5,12-dione 4-N,8-bis[(2E)-2-ethenylpenta-2,4-dienyl]-2-N-methylpyrimido[5,4-d]pyrimidine-2,4-diamine N-[4-[1-aminoethenyl(methyl)amino]phenyl]sulfanyl-2,6-difluoroaniline N-[1-(furan-2-ylmethylamino)propan-2-ylidene]-4-methoxybenzenecarboximidamide (2S,3R)-3-hydroxy-5-[(4-nitrophenyl)methyl]-2-[5-(4-nitrophenyl)sulfonyl-2H-tetrazol-1-ium-1-yl]pentanoic acid N-cyclohexyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide 3,4-diethyl-1-methylidene-2H-benzo[e]indole;formaldehyde 5-[5-[(4,6-dichloropyridin-2-yl)methoxy]indole-1-carbonyl]spiro[3H-chromene-2,3'-oxetane]-4'-one N-[2-(5,6-difluoro-1H-indol-3-yl)ethyl]-2,4,8,9-tetrahydro-3H-pyrimido[4,5-b]azepine-7-carboxamide N-[(Z)-1-(5,5-dimethyl-2-phenylcyclopenten-1-yl)propylideneamino]-4-methylbenzenesulfonamide 2-[4-(4,4,5,5-tetramethyloxaborolan-2-yl)phenoxy]ethanol 6-azidooxy-N,2-dimethyl-3H-quinazolin-4-one 1-[4-(2-aminoethoxy)phenyl]sulfonylpyrrolidine-3,4-diol 3-(2,5-dimethylpyrrol-1-yl)sulfonyl-N-[(Z)-1H-indol-3-ylmethylideneamino]benzamide 2-fluoroethanamine;3-methylbutane-1,2-diol;1-[(E)-1-phenylprop-1-en-2-yl]-3-(trifluoromethoxy)benzene 4-fluoro-2,5-dimethyl-3-[(6-propan-2-ylpyridin-2-yl)carbamoylamino]benzoic acid (3S)-1,2-dioxospiro[6H-benzo[b][1]benzazepine-5,4'-cyclohexane]-3,8-diol N-(3,5-dichlorophenyl)-N-(4-nitrobenzoyl)butanamide 1,1-dimethyl-3-[4-[[3-[(2-phenylacetyl)amino]propanoylamino]methyl]pyridin-2-yl]thiourea 6-[2-[4-(trifluoromethyl)phenyl]ethynyl]pyridine-3-carboxylic acid 1-azidooxy-4-(3,4,5-trimethylphenoxy)benzene 1,2-dibenzyl-4-cyclohexa-1,3-dien-5-yn-1-ylpyridin-1-ium;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide 1-chloro-2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)hydrazine 1-(3,4-dimethoxyphenyl)sulfonylpiperazine 5-(3-bromophenyl)-7H-[1,2,4]triazolo[1,5-c]quinazoline 6-chloro-4-[2,3-difluoro-5-(trifluoromethyl)phenyl]-2-sulfanylidene-1H-pyrimidine-5-carbonitrile ethane;5-(1,2-oxazol-3-yl)-4,8-dioxonaphthalene-2-sulfonic acid 3-[(2-fluorophenyl)methoxy]-5-(1H-pyrazol-4-ylamino)benzoic acid 1-[4-hydroxy-3,5-bis(2-methylpropoxy)phenyl]propan-1-one 3-[1-(2,5-dimethylphenyl)ethenyl]-5,6-bis(4-fluorophenyl)pyrimidine-4-thione 4-(3,5-dichloropyridin-2-yl)pyridine;methanamine 7-chloro-4-[(2S)-6,8-difluoro-2-methyl-3,4-dihydro-2H-quinoline-1-carbonyl]-1-[4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]phenyl]pyrido[2,3-d]pyrimidin-2-one (2R)-1-amino-3-[4-(2,6-dimethoxyphenyl)phenyl]sulfanylpropan-2-ol N-[4-(2,6-dimethylanilino)pyridin-3-yl]benzamide 2-[[(1S,5R)-8,9-diazatricyclo[4.3.0.02,4]nona-7,9,11-trien-7-yl]methoxy]-N-(3-fluoropyridin-4-yl)benzamide 2-(5,6-dihydronaphthalene-1-carbonyl)-4,7-dimethoxyisoquinolin-2-ium-1-one 5-[(2R)-5-hydroxy-4,6-dimethyloxan-2-yl]-1H-pyrimidine-2,4-dione ethane;3-(3-fluorophenyl)propylboronic acid N-benzyl-6-[(1S)-1-(2,3-dihydro-1H-inden-4-ylamino)ethyl]pyrazin-2-amine N-[4-amino-3,4-dioxo-1-(1H-pyrrol-2-yl)butan-2-yl]-4-thiophen-2-yl-1,2,5-thiadiazole-3-carboxamide 2-[(E)-3-azidoprop-1-enyl]-5,6-dimethoxy-3H-quinazolin-4-one (5Z)-2-cyclohexylimino-5-[[5-methoxy-2,4-bis(phenylmethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one (2E,5S)-5-methyl-3-oxo-2-[(Z)-1-thiophen-2-ylethylidenehydrazinylidene]cyclohexan-1-olate 3-[4-(trifluoromethyl)phenyl]imino-5,6-dihydro-1H-indol-2-one 1-amino-3-(benzylamino)thiourea [1-[[4-(ethoxymethyl)phenyl]methyl]piperidin-3-yl]-pyrrolidin-1-ylmethanone 4-[2-[3-[(1S)-6-chloro-8-fluoro-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenoxy]ethoxy]butan-1-ol N-azido-1,3-dimethoxy-6-naphthalen-2-ylnaphthalene-2-carboxamide 4-fluoro-2,5-dimethyl-N-[4-(4-morpholin-4-ylcyclohexa-1,3-diene-1-carbonyl)phenyl]benzamide 2-[4-[1,1,1,3,3,3-hexafluoro-2-(4-methoxyphenyl)propan-2-yl]phenoxy]ethanamine N-[6-[(3S)-4,5-dioxooxolan-3-yl]oxynaphthalene-2-carbonyl]cyclohexanecarboxamide 2,6-dichloro-4-[8-(3-methylbutyl)quinazolin-4-yl]phenol 1-azidooxy-2,3-dimethylpyrrolo[2,3-b]pyridine 1-[6-(3,5-dimethylpyrazol-1-yl)pyrimidin-4-yl]indole 4-azido-5,6-dimethoxychromen-2-one 1-[4-(3,5-dichlorophenyl)piperazin-1-yl]propan-2-one 2-(5-methylsulfanylfuran-3-carbonyl)cyclohexane-1-carboxylic acid N-[[2-(dimethylamino)pyridin-4-yl]methylideneamino]pyrimidin-5-amine 6-hydroxy-5-(3-methylcyclohexen-1-yl)naphthalene-2-carboxylic acid 7-aminopyrazolo[1,5-c]quinazoline-3-carboxylic acid 4-(cyclopropanecarbonylamino)-2,6-dimethylbenzoic acid 1-methyl-2-propan-2-ylsulfanyl-3-[4-(trifluoromethoxy)phenyl]benzene (2S)-2-[[2,6-dimethoxy-4-(3-phenylmethoxypropylcarbamoyl)benzoyl]amino]propanoic acid 2-chloro-N-[4-(1H-indol-3-yl)butanoyl]propane-1-sulfonamide 3-azido-N-[2,5-difluoro-4-(2H-tetrazol-5-yl)phenyl]imidazo[1,2-a]pyrazin-8-amine 2-[3,5-dichloro-4-(1H-indol-3-yl)phenyl]acetaldehyde N-(2,4-dinitrophenyl)-3-fluoro-5-hydroxybenzamide 3-benzylsulfanyl-6,7,8,8a-tetrahydroquinazoline-2-thione 2-bromo-3-ethylbenzonitrile;chlorobenzene 2-[4,6-bis(dimethylamino)-1H-imidazo[4,5-c]pyridin-2-yl]-N-[3-(2-phenylpyrazol-3-yl)phenyl]cyclopentane-1-carboxamide 2-(4-cyclohexylphenyl)-N-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide 5-azidooxy-2-(trifluoromethyl)pyrimidine 5-[2-(4-fluorophenyl)ethynyl]-1,3-dihydrobenzimidazol-2-one 5-[4-[2-(dimethylamino)ethoxy]phenyl]-7,8-dihydro-6H-1,6-naphthyridine-3-carbonitrile 2-[3-methyl-2,5-bis(oxiran-2-ylmethoxy)phenyl]ethanol 3-(1,2,5-trichloropentyl)benzenethiol (4-bromophenyl)methyl-ethynylcarbamic acid 4-(4-hydroxyphenyl)sulfinylphenol 2,5-dimethoxy-N'-[4-(morpholine-4-carbonyl)anilino]benzenecarboximidamide 2-(benzenesulfonamido)-3,4,5,6-tetradeuteriobenzoic acid 1-(6,7-dimethoxy-3,4-dihydro-2H-quinolin-1-yl)propan-1-one 4-(2,5-dimethylthiophene-3-carbonyl)morpholine-2-carboxamide 3-[2-(1,3-benzothiazol-2-yl)-5-tert-butylpyrazol-3-yl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridine N-[[1-(cyclohexylmethyl)pyrrolidin-3-yl]methyl]-6,7-dihydro-4H-pyrano[4,3-d][1,3]thiazole-2-carboxamide 1-[3-bromo-4-(trifluoromethyl)phenyl]-5-(trifluoromethyl)pyrazole [(1S,3R)-3-methoxycyclohexyl]-[4-[6-(trifluoromethyl)pyridazin-3-yl]piperazin-1-yl]methanone 3,8-diaminonaphthalene-2,7-disulfonate N-[(2R)-1-amino-4-methylsulfanylbutan-2-yl]-2-phenylbenzamide 6-chloro-5,8-dimethyl-1-(2,4,6-trifluorophenyl)imidazo[1,5-a]pyridine 4-[(3,5-dimethylphenyl)-phenylmethylidene]cyclohexa-2,5-dien-1-one 4-[2-(3,5-ditert-butyl-2-hydroxyphenyl)propan-2-yl]-2-methoxyphenol 2-N-(3-chlorophenyl)-5-methyl-4-N-[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazol-4-yl]pyrimidine-2,4-diamine 2,3-difluoro-1-(4-methylphenyl)sulfonyloxynaphthalene N-(4-chloro-2,6-difluorophenyl)-1,1-bis[3-(trifluoromethyl)phenyl]methanesulfonamide 1-azidooxy-2,3-diethylnaphthalene 4-(cyclopropylamino)-N'-[4-methyl-3-[1-[[7-methylideneazepine-5-carbonyl-2-(1,2,3,6-tetrahydropyridin-4-yl)benzimidazol-1-yl]methyl]cyclopropyl]phenyl]thieno[2,3-d]pyrimidine-6-carboximidamide 4-hydroxysulfanyl-1-[2-(3,6,6-trimethyl-4-oxo-7H-pyrazolo[5,1-c][1,2,4]triazin-2-yl)ethyl]piperidine 2-[3-[1-(2,4-dichlorophenyl)sulfonylindol-5-yl]pyrazol-1-yl]acetaldehyde 4-(2,6-dimethylphenyl)but-3-en-1-amine;ethane 3-N,5-N,7-N,5-tetramethylpyrazolo[1,5-a]pyrimidine-3,7-diamine 2-(1,3-benzodioxol-5-yl)-N'-hydroxy-6-[methyl(methylsulfonyl)amino]benzenecarboximidamide 4-azidooxy-5,6-diphenyl-2,3-dihydrofuro[2,3-d]pyrimidine 1-[7-chloro-4-hydroxy-3-(2H-tetrazol-5-yl)-1,2,4-benzotriazin-6-yl]ethanone 6-fluoro-7-[4-[2-(oxan-2-yloxy)ethyl]piperazin-1-yl]-8H-imidazo[1,5-a]quinazolin-5-one 3-[3-(cyclopropylmethoxy)phenyl]pyrrolidine;ethane 1-[5-tert-butyl-2-(3,4,5-trimethoxyphenyl)pyrazol-3-yl]-3-diazourea 4-[5-fluoro-2-(trifluoromethyl)pyrimidin-4-yl]oxypiperidine-1-carboxylic acid 1-[5-(2,4-dimethylphenoxy)pentyl]-N-[3-(5-ethylimidazol-1-yl)propyl]triazole-4-carboxamide N-[(3S)-1-[5-(difluoromethyl)-4H-pyrazol-3-yl]pyrrolidin-3-yl]-6,7,8,9-tetrahydro-5H-pyrimido[5,4-b]azepin-2-amine 5-[3-methoxy-4-[6-(trifluoromethyl)pyridin-2-yl]phenyl]-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidine-2,4,7-trithione 3,6-dihydroxy-2,4,9-tris(phenylmethoxy)nonanal 1-cyclohexyl-4-fluoro-2,3-dimethoxybenzene [(Z,2E)-2-ethylidene-4-(1H-indol-7-ylmethyl)pent-3-enoyl]oxidanium (3S)-1-(6-chloropyridin-2-yl)piperidine-3,4-diamine;hydrochloride 5-methyl-6-(4-pyrrolidin-1-ylphenoxy)pyridine-3-carbonitrile N-[4-(5-methoxybenzimidazol-1-yl)phenyl]furan-3-carboxamide (Z)-2,3-dichloroprop-1-en-1-amine;N'-[5-methyl-4-[4-[1-methyl-5-[[3-methylidenepentanoyl(propan-2-yl)amino]methyl]pyrazol-3-yl]phenyl]pyrimidin-2-yl]cycloheptanecarboximidamide (2S)-2-[4-chloro-3-(trifluoromethyl)phenyl]-1-N-(3,5-dihydroxy-6-oxopiperidin-1-yl)pyrrolidine-1,2-dicarboxamide 2-[(3-nitrophenyl)methyl]-1,4-dihydroquinazoline 2-[N-(4-bromobutan-2-yl)-4-chloroanilino]benzoic acid N-(2,6-dimethylphenyl)-4-[3-ethoxy-1-(3-fluoropyridin-2-yl)azetidine-3-carbonyl]piperazine-1-carboxamide 3-[4-chloro-6-[4-(2,3-dihydro-1H-tetrazol-5-yl)piperazin-1-yl]pyrimidin-2-yl]oxycyclobutan-1-amine 2-[1-(4,6-dimethylpyrimidin-5-yl)sulfonylpiperidin-3-yl]ethanol 7-chloro-4-methyl-1H-quinoline-2-thione 6-(2-chlorophenoxy)-1,3-benzoxazol-2-amine;methanamine N-(2,5-dimethylpyrazol-3-yl)oxane-4-carboxamide 6-methyl-N'-[2-(1,3,5-triazin-2-yl)acetyl]spiro[4H-quinoxaline-3,4'-piperidine]-2-carbohydrazide [3-fluoro-5-(trifluoromethyl)phenyl]methanamine;hydrochloride 2-methylsulfanyl-6-[(4-methylsulfonylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 1-chloro-6-[5-fluoro-2,3,6-trimethyl-4-(5-methylpyridin-3-yl)phenyl]pyrido[3,4-d]pyridazine 2-azido-5-cyclopropyl-4-ethoxy-1,3-thiazole 4-bromo-2-(2,5-dihydrofuran-3-yl)pyrazolo[1,5-a]pyridine;(Z)-but-2-ene;cyclohexane 4-chloro-5-[3,6-dimethyl-2-oxo-1-(trifluoromethyl)pyridin-4-yl]oxyindole-1-carboxylic acid 4-bromo-2-[(E)-[[5-chloro-1-[[2,4-bis(trifluoromethyl)phenyl]methyl]indazole-3-carbonyl]hydrazinylidene]methyl]phenolate 4-[3-[7-(5,6-didehydropyridine-2-carbonyl)naphthalen-1-yl]propyl]benzonitrile 5-methoxy-2-[4-(morpholine-4-carbonyl)phenyl]-3H-isoindol-1-one 7-[(E)-4-cyclopropylbut-3-enyl]-2,3-dihydrothieno[3,4-b][1,4]dioxine (1S)-1,2-dimethylcyclopropane;1-ethoxy-4-(5-phenylpentyl)benzene N-cyclohexyl-3-(4-morpholin-4-ylsulfonylphenyl)quinoxalin-2-amine N-[3-(2,5-dimethylpiperazine-1-carbonyl)phenyl]-4-propan-2-ylbenzamide;hydrochloride 5-bromo-4-fluoro-1H-imidazo[4,5-c]pyridine 3-[(5R)-5-(aminomethyl)-2-oxooxolan-3-yl]benzoic acid 5-(8-cyanoindolizine-2-carbonyl)oxycyclohexa-1,3-diene-1-carboxylic acid N-[(5R)-4,7-dioxo-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]benzamide 3-(5-bromofuran-2-yl)-N-[(2,4-dihydroxyphenyl)methylideneamino]propanamide N-[4-(3,5-dimethylpyridin-2-yl)oxyphenyl]pyrazine-2-carboxamide 4-[8a-(methylamino)-3a,7,8,8a,9-tetrahydrothieno[2,3-b]chromene-2-carbonyl]-N-[5-chloro-6-[1-(difluoromethyl)cyclopropanecarbonyl]pyridin-3-yl]benzamide N-(3,5-dimethylphenyl)-2-[1-[2-(4-methoxyphenoxy)acetyl]piperidin-4-ylidene]butanamide N-[2-oxo-1,6-diphenylhexan-3-yl]benzamide 4-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]benzonitrile 2-[3,5-bis(4-cyanophenyl)phenyl]-4,6-diphenylbenzene-1,3-dicarbonitrile 3-azido-2,4,6-trichloroaniline 1-chlorobuta-1,3-diene;4-[(2E)-4-methylhexa-2,5-dien-3-yl]benzonitrile 1-(2-bromophenyl)sulfonyl-5,6-dihydrobenzo[f]chromene 4-amino-2-(2,6-dibromophenyl)-5-propyl-1H-pyrimidin-6-one 2-chloro-N-(4,6-dimethylpyrimidin-2-yl)-5-[2-(ethylideneamino)phenyl]sulfonylbenzamide N-[4,6-bis(2,3-difluorophenyl)-5-[2-oxo-2-[2-[2-(propylaminomethoxy)ethoxy]ethylamino]ethyl]pyridin-2-yl]cyclobutanecarboxamide N-butyl-5,6-bis(4-methoxyphenyl)spiro[2.4]heptane-5-carboxamide (2E,4Z)-5-[1-(3-methoxyphenyl)ethenylamino]penta-2,4-dienal 2-[4-(4-aminopiperidin-1-yl)pyridin-3-yl]-5,7-dimethoxyquinazoline-4,6-diamine (1S)-3-[2,6-dichloro-4-[5-methylsulfonyl-6-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyridazine-2-carbonyl]phenyl]oxycyclopentane-1-carboxylic acid 1-[5-(4-methoxyphenoxy)pentyl]pyrazolidin-3-one 4-[2-(2,3-dimethylphenyl)ethenyl]-7,8-dihydro-6H-cyclopenta[e]indene (4-chlorophenyl)-(3-phenylmethoxypropylsulfanyl)methanesulfonate 4-[(Z)-1,2-difluoropent-1-enyl]-2-methoxy-1,3-bis(trifluoromethyl)benzene 3-[4,6-bis(3,5-dimethylpyrazol-1-yl)pyrimidin-2-yl]aniline;ethane 2-chloro-N-[6-chloro-2,4-dimethyl-3-(6-methylsulfonyl-1H-benzimidazol-2-yl)phenyl]acetamide 3-[1-(4-chlorophenyl)sulfonylpiperidine-2-carbonyl]benzoic acid 2-(4-aminobutyl)-5-methyl-N'-[4-(propanoylamino)phenyl]benzenecarboximidamide (4R)-3-(2-hydroxyphenyl)-5-[(E,3S)-3-hydroxyoct-1-enyl]-4-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-6-one (3S)-N-[1-[4-methoxy-3-(4-oxohexanoyl)phenyl]propyl]-5,7-dioxo-2,3,6,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide 1-butyl-4-[(E)-3,7-dimethyloct-5-enoxy]-2-ethynylbenzene;(E)-1,1-difluoropropane 2-chloro-N-(6-methoxypyridin-3-yl)pyrimidine-4-carboxamide;ethane N'-[(3Z)-4,5-dimethylhepta-1,3,6-trien-2-yl]benzohydrazide 2-[(3S)-4,5-dimethoxy-1,2,3-tris(phenylmethoxy)pentan-2-yl]-2H-pyran 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2]oxazolo[5,4-b]pyridine N-(3,4-dichlorophenyl)-3-[2-methoxyethyl(methyl)amino]azetidine-1-carboxamide 4-(1,3-benzodioxol-5-yl)-2-(4-cyclopropylphenyl)piperidine 4-[6-(4-methoxyphenyl)pyridazin-3-yl]-N,N,2,5-tetramethylpyrazole-3-carboxamide 3-[(5Z)-4-oxo-2-sulfanylidene-5-[(E,3R,5S)-6,7,8-trihydroxy-1-methyl-5-oxonon-8-en-3-ylidene]imidazol-1-yl]benzoic acid (2S,4R)-N'-[6-[(2-aminopyridin-3-yl)methoxy]spiro[3.4]octan-8-yl]-4-benzoyl-1-(3,4,5-trifluorophenyl)pyrrolidine-2-carbohydrazide 2-[3-[(4S)-4,6,7,8-tetrahydrothieno[3,2-c]oxepine-4-carbonyl]thiophen-2-yl]acetic acid [2,4-dihydroxy-6-(2-methylpropyl)phenyl]-[3-hydroxy-5-(hydroxymethoxy)-7-methylnaphthalen-1-yl]methanone 2-(4,6-dimethoxypyrimidin-5-yl)propanedioic acid 1-(2,3,4,5-tetramethoxyphenyl)octane-2,3-diol (5R,7S)-2-chloro-N-[2-(3-methylphenyl)ethyl]-N-propan-2-yl-5-(trifluoromethyl)-5,6,7,8-tetrahydroquinolin-8-amine 2-[5-bromo-4-(2-hydroxyethyl)-3-methoxy-2,6-dioxopyrimidin-1-yl]acetic acid 3-azido-N,N-dimethylacridine-9-carboxamide 3-[(1R)-1,2-dihydroxyethyl]-6-fluoro-7-methoxy-2H-isoquinolin-1-one 2,3-dichloro-N-diazo-6-[4-(trifluoromethyl)anilino]benzenesulfonamide (1S,2R)-2-[[2,3-dihydro-1H-indene-5-carbonyl-(4-phenylcyclohexyl)amino]methyl]cyclopentane-1-carboxylic acid 5-(N-cyclohexyl-2-methoxyanilino)-3H-1,3,4-thiadiazole-2-thione 3-[4,6-dimethyl-5-(2,2,2-trifluoroethoxy)pyridin-2-yl]-1-(1H-indazol-6-yl)pyridin-2-one N-(2-methylpropyl)-4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-ylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide 4-hydroxy-2,6-dimethoxynaphthalene-1,3,5-trisulfonic acid 2-(2,6-difluorophenyl)-N-[(4S)-7-hydroxy-3,4-dihydro-2H-chromen-4-yl]acetamide 2-[(4S)-5,8-dimethoxy-2,2-bis(trifluoromethyl)-3,4-dihydrochromen-4-yl]guanidine (4aS,8aR)-6-[3-[2-methyl-5-(1-propan-2-ylpiperidin-4-yl)phenyl]azetidine-1-carbonyl]-4,4a,5,7,8,8a-hexahydropyrido[4,3-b][1,4]oxazin-3-one 3-[1-[5-amino-6-(2,4,6-trifluorophenyl)pyrazine-2-carbonyl]piperidin-4-yl]-1H-benzimidazol-2-one N-[3,5-bis(trifluoromethyl)phenyl]-2-bromoaniline 2-methylsulfanyl-6-pyridin-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 5-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]pyridine-3-carboxylic acid [6-[4-(1,3-benzodioxol-5-yl)phenyl]-5-hydroxypyrazin-2-yl]urea 3-[(2R)-1,2-diaminopropan-2-yl]oxybenzenesulfonamide 2-[4-[(dibutylamino)methyl]phenyl]sulfonylethanamine 2-chloro-5-(4-fluorophenyl)pyridine [3-amino-4-methylsulfonyl-2-(phenylsulfanylcarbonylamino)but-2-enylidene]azanium (2S)-N'-[4-(dimethylamino)phenyl]-N-[(1R,2R)-2-ethenylcyclohexyl]-2-phenylmorpholine-3-carboximidamide 2-[(2,5-diaminophenyl)methylamino]benzoic acid 4-[(2S)-5-chloro-4,6,11-triazatetracyclo[8.7.0.03,8.012,16]heptadeca-1(10),2,3(8),11,13,15-hexaen-9-yl]-3-fluoroaniline 1-[3-(cyclohexylamino)pyrrolidin-1-yl]-2-phenylethanone (2R,3S)-1-azido-4-(benzylamino)butan-2-ol 2-[4-(1,3-benzothiazol-2-ylsulfanyl)butyl]isoindole-1,3-dione N-benzylsulfanylformamide;methane 6-bromospiro[2H-1,4-benzodioxine-3,4'-piperidine];ethane 4-(2,6-dihydroxyphenyl)-5,6,7,8-tetrahydroisoquinoline-1,3-dione 6-benzyl-3-methoxy-4-methylchromen-2-one 4-[2-(4-azidophenoxy)ethyl]quinazoline 2-fluoro-N-[(5E)-5-[(4-methylphenyl)methylidene]-1,3-thiazolidin-2-ylidene]benzenesulfonamide 2-[(1S)-2-methylcyclopentyl]oxybenzenesulfonic acid 4-[[2-cyclopropyl-6-(trifluoromethoxy)phenyl]methylamino]-5,8-dihydropyrimido[4,5-d]pyrimidine-6,7-dione (2R,4S)-2-[4-chloro-3-[(4-cyclopropyloxyphenyl)methyl]phenyl]oxane [3-(trifluoromethyl)quinoxalin-2-yl]methanol 3-bromo-5,6-dimethyl-1,4-benzothiazepine 1-(4-ethoxyphenyl)-3,8-dimethyl-7H-purine-2,6-dione 5-amino-4-[2-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 2-[4-(2,6-difluorophenyl)sulfonylpiperazin-1-yl]pyrimidine 5-ethyl-2-(4-methylcyclohexen-1-yl)benzene-1,3-diol (7S)-7-(4-bromophenyl)-2,5-dimethyl-N-naphthalen-1-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 2-[4-[4-chloro-3-[(5,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-7-yl)oxy]phenyl]triazol-1-yl]ethanol 2-(cyclopentylmethoxy)-N'-hydroxypyrimidine-4-carboximidamide (1-butylpyridin-4-ylidene)-ethoxymethanol 3-[(3S)-2,6-dioxopiperidin-3-yl]oxycarbonyloxybenzoate 5-(1-hydroxypyridin-2-ylidene)-4,6-dimethylcyclohexa-1,3-dien-1-ol 2-(5,6-dichloropyridin-3-yl)oxyphenol 3-(2-amino-5,6-dihydroquinazolin-7-yl)benzonitrile 2-[2-hydroxy-4-(1H-indazol-5-ylamino)phenyl]acetamide 1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]-1-(pyridine-3-carbonyl)thiourea N-[(4-fluorophenyl)methyl]-6-[5-morpholin-4-yl-2-(3-oxo-1H-isoindol-2-yl)benzoyl]-7,8-dihydro-5H-2,6-naphthyridine-3-carboxamide 2,7-dibromofluoren-9-one 3-[4-[4-(2,4-dichlorophenyl)piperidine-1-carbonyl]-3-methylpyrazol-1-yl]benzoic acid [(E)-2-[4-(1,3-benzodioxol-5-yloxy)phenyl]-3-ethylpent-2-enyl]azanium 4-(azidomethyl)-6,7-dimethoxyquinoline 5-[3-(4,4-difluoropiperidine-1-carbonyl)phenyl]-2H-isoquinolin-1-one 3-(7,8-dihydronaphthalen-2-yl)propanamide 3-[[(2S)-3,7-dioxo-6H-1,4-oxazepine-5-carbonyl]amino]-4-fluorobenzoic acid 2-(4,5-diphenyl-1H-imidazol-2-yl)phenol N-methyl-4-(trifluoromethoxy)aniline [1-(2,3-dimethoxyphenyl)-6-methylsulfanylbenzimidazol-2-yl]thiourea 2-[(3S,4R)-4-azidopyrrolidin-3-yl]oxypyrimidine 1-[4-[(2R)-2-[3-chloro-5-fluoro-6-[(4-fluorophenyl)methoxy]pyridin-2-yl]-4,4-difluoropyrrolidin-1-yl]benzoyl]-N'-hydroxyazetidine-3-carboximidamide N-[2-(3-bromopyridin-4-yl)ethyl]-5-chlorospiro[1H-indene-3,4'-piperidine]-1'-amine 2-amino-6-(2,3-difluorophenyl)benzoic acid 3-[[5-[2-(dimethylamino)ethoxy]pyridine-3-carbonyl]amino]propanoic acid 1-[2-(3,5-dimethylphenyl)pyrrolidin-1-yl]-2-(4-iodopiperidin-4-yl)ethanone [6-(3,4-difluorophenyl)benzotriazol-1-yl]oxymethanol (1-azidooxycyclohexyl)oxybenzene 2-(3,5-difluorophenyl)-N-methyl-1H-pyridazine-4-carboxamide 4-chloro-2-[6-(3,5-ditert-butylphenyl)-1-methylpyridin-1-ium-2-yl]phenol N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-(4-ethylsulfanylphenyl)-6-methyl-1-[[1-(oxetan-3-yl)piperidin-4-yl]methoxy]indole-3-carboxamide (5R)-2-[(Z,3E)-4-fluoropent-1-enyl]-6,11-dihydrobenzo[c][1]benzoxepine 5-(4-chlorophenyl)-4-(2,3-dihydro-1H-indene-2-carbonyl)-6-ethyl-1,4-dihydropyridine-3-carboxylic acid 4-azidooxy-1H-pyrrolo[2,3-b]pyridine 3-methyl-4-[6-(methylamino)pyridazin-3-yl]phenol 2-[(3S,4R)-1-benzylpiperidin-3-yl]-4H-1,4-benzothiazin-7-ol 4-(3-chlorophenyl)-6,7,8-trimethoxyquinazoline (4-methylphenyl)-[3-(oxan-2-yloxycarbonylamino)phenyl]sulfamic acid 4-[6-(difluoromethyl)pyridin-3-yl]oxy-1-propan-2-ylpyrrolidine-2-carboxylic acid 3-azido-5-[1-(1,2,4-triazol-4-yl)propan-2-yl]-1H-indole 1-(2,4-difluorophenyl)-5H-pyrazolo[3,4-d]pyrimidin-4-one N-[5-(4-fluorophenyl)thiophen-2-yl]-5,7-dimethoxyquinazolin-4-amine N'-(3,4-dimethylphenyl)-2-phenylethanimidamide 1-(2,4-difluorophenyl)sulfonyl-3-[(3S)-5-methylsulfanyloxolan-3-yl]-6-propan-2-yloxyindole 4-[4-methyl-6-(3-propan-2-ylphenyl)cyclohexa-1,5-dien-1-yl]oxy-N-[(4R)-3-methylideneoxolan-2-yl]pyrimidin-2-amine N-[3-[(5S)-2-amino-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]-4-fluorophenyl]methanesulfonamide ethane;5-[4-(3-ethoxy-1,2,4-triazin-6-yl)piperazin-1-yl]sulfanylpyridine-2-carbonitrile 2-[(3S)-1-benzylpyrrolidin-3-yl]propanoic acid 2-[3-(cyclohexyloxymethyl)azetidin-1-yl]pyridine 4-chloro-N,5-diethyl-3H-1,2,4-benzotriazin-7-amine (E)-1-[4-[(Z)-3-cyclopropylpent-2-enyl]phenyl]but-1-en-3-one N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1-propan-2-ylpiperidine-3-carboxamide 3-(azidomethyl)-2,5-diphenyl-1,4-dioxane 2-(5-chloro-3,4-dihydro-1H-isoquinoline-2-carbonyl)pentanal 2-[6-chloro-3-(dimethylamino)-4-oxoquinazolin-2-yl]sulfanyl-N-phenylacetamide 6-[2,2-dimethoxyethyl(hexadecanoyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 5-[3-fluoro-4-(7-methoxy-2,6-dimethylheptoxy)phenyl]-2-pyridin-4-ylpyridine 3-azido-2-[(4-methoxyphenyl)methyl]-1H-indole 6-(1,2-diethoxybutan-2-yl)-3-[4-(trifluoromethyl)phenyl]chromen-4-one 2-hydroxy-6,8a-dihydronaphthalene-1-sulfonic acid 2-(4,4-diethoxybutyliminomethyl)-6-[3-(trifluoromethyl)phenyl]phenol 2-[5-(methoxymethyl)-1,3-thiazol-4-yl]-N-[2-(6-oxocyclohexa-2,4-dien-1-ylidene)hydrazinyl]acetamide 3-methyl-5,6-dihydroindole;2-[1-(4-methylphenyl)propan-2-yl]-N,7-dioxooctanamide (4-azidopiperidin-1-yl)-[2,4-dimethoxy-6-[2-(trifluoromethoxy)phenoxy]phenyl]methanone N'-hydroxy-3-(2,5,8-trimethyl-2,4-dihydro-1H-pyrido[4,3-d]pyrimidin-3-yl)benzenecarboximidamide 2-chloro-5-[(4-chlorobenzoyl)amino]-N-[2-[3,3-dimethylbutanoyl(2-phenylethyl)amino]ethyl]benzamide 5-[3-chloro-4-(2,3-dihydroxypropoxy)phenyl]hexanoic acid 2-[4-fluoro-2-[1,3-thiazol-5-yl(quinolin-6-yl)amino]phenyl]sulfonylacetic acid 3-amino-6-cyclopropyl-N'-hydroxypyridazine-4-carboximidamide 2,4-ditert-butyl-6-[[1-[(3-hydroxyphenyl)methoxy]pyridin-1-ium-3-yl]iminomethyl]phenol;bromide (2S)-5,6-diamino-2-[[(3R)-4-methylpentanoyl]amino]-N-[[2-oxo-4-phenyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl]hexanamide [(1S,2R)-2-aminocyclohexyl]-[4-[(2-methoxypyrimidin-5-yl)methyl]piperidin-1-yl]methanone;dihydrochloride 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]oxetan-3-amine 4-[3-(1,2-dihydropyridazin-6-yl)phenyl]butanoic acid 1-[4-(3,6-dihydro-2H-pyran-5-yl)phenyl]-N-methylpyrrolidin-3-amine (3S)-2,5,7-trimethyl-6-phenyl-N'-propan-2-yloxyoctanediamide N-[4-[4-[(2R)-2,3-dimethylbutoxy]phenyl]-1,3-thiazol-2-yl]-5-ethylpyridine-3-carboxamide N-[(4,5-dichloro-2-ethylsulfonylphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine 2-[(4-acetylphenyl)methoxy]-1-chloropropan-2-ol 6-(3,3,4,4,5,5-hexamethylpiperazine-1-carbonyl)pyrimidine-2-carboxylic acid 5-[(Z)-1,2-dihydroindol-3-ylidenemethyl]-N-pyridin-4-ylfuran-2-carboxamide 2,3-dimethyl-4,9-dihydrobenzo[h]quinoline N-[(Z)-1H-indol-3-ylmethylideneamino]-2-(N-methylsulfonylanilino)acetamide 2-[(3-butoxyphenyl)sulfonylamino]acetic acid 2-(3-methoxyphenyl)-1,4-dihydropyrimidine 2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-[2-[(2S)-3-fluorobutan-2-yl]oxyethyl]acetamide (5R,8aS)-7-[4-(difluoromethoxy)benzoyl]-2,3,6,7,8,8a-hexahydropyrrolo[1,2-a]pyrazine-1,5-dione 2-[1,3-benzodioxol-5-yl(hydroxy)methylidene]-4,4,5,6-tetramethylcyclohexane-1,3-dione N-[6-[4-(1,1-difluoroethyl)phenyl]pyridin-3-yl]formamide (2R)-2-amino-4-[(5S,7R)-7-methyl-1,3-oxazepane-5-carbonyl]-N-[[3-methyl-6-oxo-8-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-benzo[b][1,4]benzoxazepin-9-ylidene]amino]pentanamide N-(2,4-dinitrophenyl)-2-methyl-5-nitro-N-propan-2-ylaniline 3-[(4S)-1-methyl-6-oxo-2,4-dihydropyrazolo[3,4-b][1,4]oxazepin-8-yl]benzamide 3-[2-chloro-4-[(4R)-4,5,5-trifluoropentoxy]phenyl]-1H-pyrrole N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-ethyl-2-[ethyl-[(2S)-4,4,4-trifluorobutan-2-yl]amino]-7-[3-[(4-morpholin-4-ylpiperidin-1-yl)methyl]phenyl]-3H-benzimidazole-5-carboxamide 2-[8-(1,3-benzodioxol-5-ylmethyl)-8-azabicyclo[3.2.1]octan-3-yl]-N-(4-chlorophenyl)acetamide (2S,4S)-N-[[5-chloro-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methyl]-6-oxopiperidine-2-carboxamide 1-ethyl-2-(6-phenylheptoxy)benzene 7-(methylamino)-5-[(3-propan-2-ylcyclobutyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile 3-[5-fluoro-2-hydroxy-4-[3-(oxan-2-yloxy)propoxy]phenyl]-N,7-dimethylpyrazolo[1,5-a]pyrimidine-6-carboxamide N-(2,6-dibromopyridin-4-yl)-N-methoxybenzamide N-[(2S)-1-oxo-1-(3,4,5-trifluoroanilino)propan-2-yl]butane-2-sulfonamide 3-(5,6-dihydroxynaphthalene-2-carbonyl)oxybutanoic acid 3-[8-(3,4-dichlorophenyl)-9-oxo-6H-[1,2]thiazolo[5,4-b]quinolin-7-yl]-1-methylsulfanylcyclobutane-1-carboxylic acid 4-[2-(methylamino)phenyl]-N-propan-2-ylaniline 7-(2,6-dichlorophenyl)-12-[2-[4-(4-ethylpiperazine-1-carbonyl)piperidin-1-yl]pyridin-3-yl]-2,5,11,13-tetrazatricyclo[7.4.0.02,6]trideca-1(13),3,5,9,11-pentaen-8-one 3-(3,4-dimethoxyphenyl)-5-[1-(6-ethylpyridin-2-yl)cyclobutyl]-1,2,4-oxadiazole 1-[(5R)-2-methyl-5,6-dihydrobenzo[h]quinolin-4-yl]hexan-1-one (2S,6R)-4-[5-[(4-cyanophenyl)methyl]-1,3-thiazole-2-carbonyl]-N-cyclopropyl-12-hydroxy-7-oxo-9-oxa-3,5,6,10-tetrazatricyclo[8.4.0.02,6]tetradeca-1(14),2,4,10,12-pentaene-15-carboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]-2,5-dimethoxybenzenesulfinamide 4-(3,5-dimethylbenzene-6-id-1-yl)sulfonyl-N-propan-2-ylbenzenesulfonamide;uranium(2+) 1-[(2S)-2-[3,5-dimethoxy-4-(methylsulfanylamino)phenyl]piperidin-1-yl]-3-(2-ethylsulfonylpyridin-4-yl)propan-1-one 2-methyl-3-(3-phenylphenyl)pyridine 3-(4-tert-butylphenyl)-2,5-difluoroaniline 1-(3,5-difluorophenyl)pentan-2-amine;5-[4-(3,5-difluorophenyl)phenyl]pentane-2,4-dione 3-[(4aR,8aS)-2,3,4a,5,7,8,8a-octahydropyrano[3,2-c]pyridine-4-carbonyl]benzoic acid;cyclohexanol 3-[(2,6-dimethoxyphenyl)methylidene]-1H-indol-2-one 4-[[6-(4,5-dimethylcyclohexa-1,3-dien-1-yl)pyridine-2-carbonyl]amino]thiophene-2-carboxylic acid 5-[6-(4,7-difluoro-1H-indole-2-carbonyl)-6-azaspiro[3.4]octan-8-yl]-N-ethylpyridine-2-carboxamide 2-cyclopropyloxy-6-[4-(3,5-dimethylpyridin-2-yl)piperidine-1-carbonyl]benzamide 2-[4-(3,4-dichlorophenyl)sulfonylpiperazine-1-carbonyl]-1H-quinolin-4-one 2-[2-(4,6-difluorocyclohexa-1,3-dien-1-yl)-4-methoxyphenyl]pyrrolidine 4-(2,3-dihydro-1H-imidazol-2-yl)phenol 2-[(1S)-7-nitro-3,4-dihydro-1H-isoquinoline-2-carbonyl]chromen-4-one 2-[5,6-di(propan-2-yl)pyridin-3-yl]acetamide 1-(4-fluorophenyl)-3-[3-hydroxy-2-methyl-5-oxo-4,4-bis(prop-2-ynylamino)pentanoyl]-6-(trifluoromethoxy)pyridine-2,4-dione (5R)-5-(3,4-dihydro-2H-chromen-8-yl)-6,7-bis(sulfanylidene)octanal 2-(5-chloro-3,4-dimethoxyphenyl)ethanamine;hydrochloride 1-[3-(dimethylamino)phenyl]-4-pyrrolidin-1-ylcyclohexane-1,4-diol N-[3-[[(Z)-1H-indol-3-ylmethylideneamino]carbamoyl]phenyl]-4,5,6,7-tetrahydro-2,1-benzoxazole-3-carboxamide (3S)-N'-[2,4-bis(ethylsulfonyl)phenyl]-5,6-dimethyl-1-(4-methylbenzoyl)piperidine-3-carbohydrazide 2-(1-hydroxycyclobutyl)-N-methyl-N-[6-[4-(2,2,2-trifluoroethanimidoyl)phenoxy]hexyl]acetamide 2-[4-(dipropylamino)phenyl]-1,2,3,3a-tetrahydropyren-5-one N-methyl-1-[2,3,4,5-tetrafluoro-6-(trifluoromethyl)phenyl]-1-benzothiophen-5-amine 3-(2-chlorophenyl)-5,6-diethylchromen-4-one 1-[4-(methoxymethyl)triazolo[4,5-c]pyridin-2-yl]butan-1-one 3-[3,4-bis(phenylmethoxy)-1H-pyridin-2-ylidene]propanenitrile N-[3-[4-[4-[2-(3,6-dihydro-2H-pyran-4-yl)ethynyl]pyridin-3-yl]phenyl]prop-1-en-2-yl]cyclohexanamine (6-aminopyrimidin-4-yl)-(3,7-difluorocycloocta-2,4-dien-1-ylidene)azanium (Z)-2-cyano-3-cyclopropyl-N-[4-(trifluoromethoxy)phenyl]prop-2-enamide 7-(methoxymethyl)benzo[c][2,6]naphthyridine N-[4,5-dimethyl-2-(6-oxo-4-propan-2-yl-1H-pyrimidin-2-yl)pyrazol-3-yl]benzamide 2,6-diaminopyridine-4-carboxylic acid;dihydrochloride 2-(azidomethyl)-1-chloro-3-ethenylbenzene 4-fluoro-2-[7-(3-hydroxyazetidine-1-carbonyl)-9-methoxypyrido[3,4-b]indol-3-yl]benzenesulfonamide 1-[(4S)-4-azidopentyl]-3,7-dimethoxy-6-methylquinolin-2-one 1-[(4R,5S)-5-(2,6-difluorophenyl)-3,8-dimethyl-2,3,4,7-tetrahydropyrazolo[3,4-b]quinolin-4-yl]ethenamine 6-benzylsulfanyl-4,5,7-trifluoroquinoline 2,4-difluorobenzaldehyde;4-(1-methylpyrazol-3-yl)oxy-N-propan-2-ylaniline 3-[2,2-dimethoxyethyl(hexadecanoyl)amino]phenol 2-(4-fluorophenyl)-4-phenylbutanoic acid 2-chloro-N-[3-[[(4,5-dimethyl-1H-imidazole-2-carbonyl)amino]methyl]phenyl]pyridine-4-carboxamide 2-[3,6-difluoro-4-(2-methylsulfanyloxyethyl)cyclohexa-1,5-dien-1-yl]pyridine 4-[4-azidooxy-6-(3,5-difluorophenoxy)-2H-pyran-3-yl]pyrimidine (3,4-dimethylphenoxy)-oxidoborane 5-bromo-3,6-bis[(4-methoxyphenyl)methoxy]benzimidazole-2-carboxylic acid 3-[1-(2,6-dichlorophenyl)triazol-4-yl]propane-1,1-diol N-[1-(2,6-difluorophenyl)-3-methylbut-2-enyl]cyclopropanamine 1-[(3Z,5E)-6,7-dimethylnona-3,5-dien-4-yl]-2-methoxybenzene 3,5-dichlorophenol;5-[(4-fluorophenyl)sulfanylmethyl]thiophene-2-carboxamide N-azido-6-[2,3-difluoro-4-(trifluoromethoxy)phenyl]pyridazin-3-amine N-[2-fluoro-4-methylsulfonyl-3-(trifluoromethoxy)phenyl]-3,5-dimethylpyrazole-1-carboxamide 3,5-ditert-butyl-2-(diphenylphosphorylmethoxy)benzenesulfonamide N-[4-(1H-pyrazol-5-yl)phenyl]cyclohexanecarboxamide 1-(3-chlorophenyl)-4-[2-methyl-6-oxo-5-[[4-(trifluoromethyl)phenoxy]methyl]-1H-pyrimidin-4-yl]piperazine-2-carbothioamide (E,3S)-2-[5-[4-(trifluoromethoxy)phenyl]-1H-pyrrole-3-carbonyl]hex-4-enediamide N-[5-fluoro-6-(4-methylpyridin-3-yl)pyridin-2-yl]formamide 1-[4-[3-(4,5-dihydro-1H-imidazol-2-yl)propoxy]phenyl]ethenamine N-[(4-chlorophenyl)methyl]-4-(pyridine-3-carbonyl)piperazine-1-carboxamide 5-bromo-2,3,7,8-tetrahydro-1H-[1]benzothiolo[2,3-e]indole 4-[(E)-5-[4-(methoxymethyl)phenyl]pent-1-enyl]pyridine N-[4-chloro-2-(2-cyclopropyloxyethoxy)phenyl]sulfanyl-5-methylpyridin-2-amine 2-[(3,4-dichlorophenyl)methyl]-1H-triazole-5-thione N-(3,5-dimethylphenyl)-2-[3-fluoro-6-[hydroxy(methoxy)methyl]pyrazolo[4,3-b]pyridin-1-yl]acetamide 3-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]oxybenzonitrile 2,6-bis[4-(diethylamino)phenyl]benzene-1,3,5-triol [3-[(3,4-dichlorophenyl)sulfonylamino]oxolan-3-yl]carbamic acid N-[(E)-N'-[amino-(4-chlorophenyl)methyl]carbamimidoyl]cyclohexanecarboxamide 2-[(E)-2-aminoethenyl]-4-methoxyaniline;3-(1H-indazol-5-yl)pyridin-2-amine (4Z)-2-methyl-4-[1-(1H-pyrrol-3-yl)propylidene]-1,2,5-oxadiazolidine N-(4,5-dimethyl-1H-pyrazol-3-yl)-2-[6-fluoro-8-(trifluoromethoxy)isoquinolin-3-yl]acetamide 2-(3-methoxyphenyl)-1,4,5,8,12-pentazatricyclo[7.3.0.03,7]dodeca-3(7),9,11-trien-6-one N-[(4R)-1-amino-6-bromo-4,5,7,8-tetrahydrocyclohepta[c]pyrazol-4-yl]pyrazolo[3,4-b]pyridine-1-carboxamide N'-hydroxy-6-[methyl(oxan-4-yl)amino]pyridine-2-carboximidamide [(1-ethylcyclopentanecarbonyl)amino]carbamodithioic acid;N,N,3-trimethyl-4-pyrazol-1-ylbenzamide 2,3-dihydroxypropyl-[[4-(2H-tetrazol-5-yl)phenyl]methyl]azanium 2-hydroxy-4-[N-methylsulfonyl-4-(pyridin-3-ylsulfamoyl)anilino]benzoic acid 4-[(1,1,2,2,3,3,4,4,5,5,6,8,8a-undecadeuterio-7-methoxyoctyl)amino]benzoic acid 1-[2-(1,3-benzodioxol-5-yl)ethyl]-6-[3-methoxy-4-[6-[methyl(pyrrolidine-2-carbonyl)amino]hexanoylamino]phenyl]piperidine-3-carboxylic acid 1-[2,4-difluoro-3-(2,2,2-trifluoroethoxy)phenyl]-2-methylbutan-1-one 3-[(2,6-difluorophenyl)methyl]-5-(4-piperidin-1-ylcyclohexa-1,5-dien-1-yl)triazolo[4,5-d]pyrimidine 5-(dimethylamino)-3-[4-fluoro-1-(2,2,6,6-tetramethylpiperidin-4-yl)piperidin-4-yl]thieno[3,2-b]pyran-7-one;ethane 2-(2-bromophenyl)-4,5-difluoropyrimidine 4-[6,6-difluoro-3-(2H-tetrazol-5-yl)cyclohexa-1,3-dien-1-yl]aniline 5-(3,4-dimethoxyphenyl)-2,6-diethyl-9H-pyrido[2,3-b]indole 5-(2,3-dihydrothiophen-4-yl)-3-ethyl-6-[(E)-prop-1-enoxy]imidazo[2,1-b][1,3]thiazole [4-(4-hydroxyphenoxy)phenyl]methanesulfonate 4-[2,2-dimethoxyethyl(3-methylbutyl)amino]-N-pyrimidin-2-ylbenzenesulfonamide 1-(3,4-difluorophenyl)-5-[[2,4-bis(trifluoromethyl)phenyl]sulfanylamino]pentan-3-ol;ethane 5-(4-ethoxyphenyl)-2,6-dimethylpyrimidin-4-amine N'-(3,4-dichlorophenyl)propanediamide 3-[5-[(2,6-difluorophenyl)methyl]tetrazol-1-ium-1-ylidene]-6-methoxyindole 1-(4,6-dimethoxypyrimidin-2-yl)sulfonylnaphthalene-2-sulfonamide 6-(3,4-dihydro-2H-quinoline-1-carbonyl)pyridine-3-carboxylic acid 2-[(3R)-1-benzylpiperidin-3-yl]oxy-5-chloro-3-hydroxy-8-methylidene-9,10-dioxoanthracene-1-sulfonic acid 5-(3,4-difluorophenyl)sulfanyl-2-ethyl-6H-1,3,4-thiadiazine 2-(2,3,5,6-tetrachlorophenyl)phenol (2R)-N-[[4-(2-hydroxyethylcarbamoyl)phenyl]methyl]-1-(6,7,8,9-tetrahydrothieno[3,2-b]azepine-2-carbonyl)pyrrolidine-2-carboxamide 2-[2,6-difluoro-N-(3-methylbut-2-enyl)anilino]acetic acid N-[1-(4-fluorophenyl)ethyl]-2,6-dimethoxybenzamide 6-[1-azido-3-(5-chloropyrimidin-2-yl)oxypropan-2-yl]quinoline N'-[5-chloro-3-methyl-2-(5-methylsulfonyl-1,2,4-triazol-1-yl)phenyl]-N-ethylpropane-1,3-diamine 4-cyclohepta-1,3,5-trien-1-yl-N'-[3-(4-ethoxyphenyl)-2H-furo[3,2-c]quinolin-8-yl]piperidine-1-carboximidamide [(3S,4R)-1-benzyl-3-(dimethylamino)piperidin-4-yl]carbamic acid 2-ethoxy-5-[(2R,3S)-3-[1-(4-phenylmethoxyphenyl)propan-2-yloxy]butan-2-yl]phenol 5-[3-(azepan-1-yl)butanoyl]-N,2-dimethoxybenzenesulfonamide (3R,4S)-3-[(2Z)-2-[(Z)-1-chloroprop-1-enyl]penta-2,4-dienoyl]-N'-(5-cyano-2,6-difluorophenyl)pyrrolidine-1-carboximidamide N-(2,4-dimethylpentan-3-yl)-3-propan-2-ylbenzenesulfonamide 1-(3,4-dihydronaphthalen-2-yl)-3-[(6R)-1-methoxy-6-methylcyclohexa-2,4-dien-1-yl]prop-2-yn-1-one 6-[(4,7-difluoro-2,3-dihydroindole-1-carbonyl)amino]imidazo[1,2-a]pyridine-2-carboxylic acid 5-[1-(4,4a,5,6,7,8,8a-octahydroquinazolin-4-yl)cyclopropanecarbonyl]imidazolidine-2,4-dione 5-chloro-2,3,4-trihydroisoquinolin-1-one 2-[[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfinylamino]benzoic acid 1-[2,3,5-trifluoro-4-[2-(methylideneamino)ethoxy]phenyl]indole-7-carboxylic acid 1-[2-fluoro-5-(trifluoromethyl)phenyl]-3,4-dihydronaphthalene 5-[4-(2,3-dihydroindole-1-carbonyl)phenyl]-6-fluoro-N-methyl-N'-pentan-2-ylidene-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboximidamide 7-tert-butyl-N-ethanimidoylisoquinoline-1-carboxamide;(E)-1,3-dichloroprop-1-ene 2-aminooxy-6-[(3-nitrophenyl)diazenyl]benzenesulfonic acid 2-(5-aminopyridin-3-yl)quinoline-8-carboxylic acid 3-(4-phenylbutyl)pyridine-2,5-dicarboxamide [1-azidooxy-2,3-bis(phenylmethoxy)propan-2-yl]oxybenzene 4-amino-6-[(5-hydroxy-2,3-diiodophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 3-(5,7,10,11-tetrazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-ylsulfanylamino)benzonitrile 1-phenyl-3,6,7-triazabicyclo[3.2.0]hept-6-ene 5-[(2,6-dimethoxypyrimidin-4-yl)-(4-ethoxy-4-oxobutyl)amino]naphthalene-2-sulfonic acid 3-[(E)-2,4-difluoropent-1-enyl]-N-ethylaniline 3-[[4-cyclohexyl-N-(2-methoxyethyl)anilino]methylidene]-1H-indol-2-one 4-[[(Z)-1-amino-3-sulfanylprop-2-enylidene]amino]benzoic acid 3-[1,4-bis(phenylmethoxy)cyclohexa-2,4-dien-1-yl]propanoic acid 2-(4,5-diaminothiophen-3-yl)-1H-indol-6-ol 2-[4-[1-aminoethyl(methyl)amino]-5,6-difluoro-8-[(2S)-oxolan-2-yl]oxyquinazolin-7-yl]phenol N-[1,3-bis(triazol-2-yl)propan-2-ylidene]hydroxylamine 3-(6-ethyl-2,4-dioxospiro[1H-quinazoline-8,4'-piperidine]-1'-carbonyl)benzoic acid 5-cyclobutyl-N-[(2S)-1-hydroxy-3,4-dihydro-2H-naphthalen-2-yl]-4-(2-methoxyethyl)-1,2-oxazole-3-carboxamide 1-(2-methoxyphenyl)pentan-2-one 3-[3-[1-(2,6-dichlorophenyl)triazol-4-yl]phenyl]-5-phenyl-1,2,4-oxadiazole 2-(2-methylphenyl)-1H-benzimidazole 2-[[4-(cyclohexyloxymethyl)-3-(trifluoromethyl)phenyl]carbamoylamino]-N,5-dimethylbenzamide N-azido-6-chloro-2,3-dihydroinden-1-imine 2-(1,3-dioxolan-2-yl)benzenesulfonic acid 5-[3-[4,5-bis(ethenyl)furan-2-carbonyl]-1H-indol-7-yl]-2,3-dimethoxybenzoic acid N-(2,6-dichlorophenyl)-7-hydroxy-5H-pyrrolo[3,4-b]pyridine-6-carboxamide 1,3-bis(2,5-difluorophenyl)benzene;ethane 4-(4-fluorophenyl)-2-iodo-5,6,7,8-tetrahydroquinazoline (2S)-3-(4,5-dihydropyrimidin-2-yloxy)-N-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-2-[[6-(trifluoromethyl)quinazolin-2-yl]amino]propanamide 6-[[4-chloro-2-(propylaminomethyl)benzoyl]amino]-N-(cyclohexylmethyl)imidazo[1,5-a]pyridine-7-carboxamide N-(5-azidopyridin-3-yl)acetamide 4-(3,5-dichlorophenyl)sulfanylbutanenitrile (4R)-2'-amino-1-methylspiro[5,6-dihydropyrazolo[3,4-d]pyrimidine-7,3'-indole]-2'-one 3-azido-4,5-difluoro-2-phenylaniline 5-[(5E)-7,8-dimethyl-4-[3-(trifluoromethoxy)phenyl]-2H-pyrano[2,3-c]pyrazole-1-carbonyl]thiophene-3-carboxylic acid 2-(1H-imidazol-5-yl)-7-methylbenzimidazolo[1,2-a]quinazolin-6-one 5-[3-[4-(3-fluorophenyl)-1H-pyrrolo[2,3-c]pyridin-2-yl]-1H-pyrazolo[4,3-b]pyridin-5-yl]-N,N-dimethylpyridin-3-amine [(2S,3R)-4-methyl-1-oxo-5-sulfanylidene-2H-3-benzazepin-2-yl]-phenoxyphosphinous acid 7-chloro-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]quinolin-4-amine N-[5-[3-(1H-pyrrolo[2,3-b]pyridine-2-carbonyl)phenyl]-2-bicyclo[4.2.0]octa-1,3,5-trienyl]methanesulfonamide N-(4-chlorophenyl)-3,5-dimethyltriazole-4-carboxamide [3-(2-methoxyethyl)phenyl]-piperidin-1-ylmethanone 5-(4-fluorophenyl)-1-(pyridin-2-ylmethylsulfonyl)-3a,7a-dihydroindole-2,3-dicarboximidamide 2,6-dibromo-4-[[3-(hydroxymethyl)pyrrolidin-1-yl]methyl]phenol 2-amino-5,6,7-trimethyl-N-(1H-pyrrolo[3,2-c]pyridin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 2-methyliminospiro[4,5-dihydro-1H-1,4-benzodiazepine-3,4'-piperidine]-8-carbonitrile N-[4-(2,6-dimethylmorpholin-4-yl)pyridin-3-yl]benzamide (2S)-N-[2,6-difluoro-4-(5-oxo-1,4-oxazepane-4-carbonyl)phenyl]pyrrolidine-2-carboxamide 4-N-[(4Z)-5,7-dimethylcycloocta-1,3,6-trien-1-yl]pyridine-2,4-diamine (6-diphenylphosphanyl-2,4-dimethoxycyclohexa-1,3-dien-1-yl)-diphenylphosphane 3-[2-[5-(4,6-dimethylpyridin-3-yl)furan-2-yl]piperidin-1-yl]cyclobutan-1-amine 2-[[(5R)-1,4-dioxaspiro[4.6]undecan-8-yl]sulfamoyl]-N-(3,4,5-trifluorophenyl)benzamide N-[2-(1-benzofuran-5-ylmethylamino)pyrimidin-4-yl]cyclopropanecarboxamide 4-(difluoromethyl)-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]aniline 1-[(2R,4S)-4-hydroxy-2-phenyl-6-oxa-9-azaspiro[4.5]decan-9-yl]propan-1-one 2-[(1S,3R)-3-[4-(5-fluoro-6-methylpyridin-3-yl)phenyl]sulfonylcyclopentyl]propanamide 4-[1-(3,5-dimethoxyphenyl)piperidin-4-yl]-2-phenyl-1H-pyrimidin-6-one 7-(2,3-dimethoxyphenyl)-5-fluorospiro[1H-indole-3,4'-piperidine]-2-one 4-[(2E,3Z)-2-ethylidenehexa-3,5-dienoyl]oxybenzenesulfonate 5-methyl-2-[3-(6,7,8,9-tetrahydro-5H-carbazol-3-yl)-1,2,4-oxadiazol-5-yl]phenol 2-(5,6,7-trimethoxynaphthalene-2-carbonyl)cyclopentane-1-carboxylate (1S,3R)-N-[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]-3-N-hydroxy-1,3-dihydroisoindole-1,3-dicarboxamide 5-(2,3-dihydroindol-1-ylmethyl)pyrimidine 4-(aminomethyl)-2-[2-(3,5-dichloropyridin-4-yl)ethynyl]-1H-pyrimidin-6-one (2S)-4,5,5-triethyl-1-[3-(4-fluorophenyl)sulfanylpropyl]pyrrolidine-2,3-dicarboxylic acid 1-[4-[3-(2,5-difluorophenyl)-3,4-dihydropyrazole-2-carbonyl]pent-4-enyl]-N-(2-methoxyethyl)pyrazole-4-sulfonamide 2-[1-(3,5-dimethylbenzoyl)-4-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]piperidin-4-yl]acetic acid 2-(2,5-dichloropyridin-3-yl)oxy-N'-hydroxypyrimidine-4-carboximidamide 1-(2,6-dimethylphenyl)sulfonyl-N-(2H-pyrazolo[3,4-b]pyrazin-5-yloxy)indazol-3-amine N-(4-ethylphenyl)-N',N'-dimethylheptanediamide 3-(1,2,4-triazol-1-ylmethyl)oxane-2,5-dione 5-[4-methoxy-3-(trifluoromethyl)phenyl]hexa-2,4-dienamide [[(3S)-3-methylcyclopenten-1-yl]amino]methoxy-[4-phenylsulfanylbut-2-ynoxy-[6-(trifluoromethoxy)pyridine-3-carbonyl]amino]phosphinic acid 4-(4-methoxy-1H-indol-3-yl)aniline 2-cyclobutylsulfanyl-4,5,7-trimethyl-1,3-benzothiazole 2-fluoro-5-[[3-(oxolan-3-yl)benzoyl]amino]benzoic acid 4-(2,5-dihydroxyphenyl)-6-(3,4-dimethoxyanilino)quinoline-3-carbonitrile 2,3-bis(ethenyl)-5,6-difluoroquinoxaline N-[2-(4-fluorophenyl)ethyl]-3-(6-methoxypyridin-3-yl)piperidine-1-carboxamide 2-[3,5-dichloro-4-(4-propan-2-yloxyphenoxy)phenyl]ethanethioamide N-(4,5-dichlorothiophen-2-yl)sulfanyl-3-fluoro-4-[(Z)-1-methoxyprop-1-enyl]pyridin-2-amine;ethane (3S,5R)-3-azido-5-phenylpiperidine 2-(4,5-dimethyl-2-phenyldiazenyl-N-prop-2-enylanilino)octanoic acid 4-methoxy-2,3-bis(4-propan-2-ylsulfanylbutyl)pyridine 4-(aminomethyl)-3-azidobenzenesulfonamide N-[3,5-bis(2-methylpropoxy)phenyl]-2-iodopyridine-4-carboxamide (5S)-3,4-dimethyl-6,7-dihydro-5H-1-benzothiophene-2-carboxylic acid 4-[[(2S,3R)-2,3-dihydroxypropoxy]methyl]-N'-hydroxypyridine-2-carboximidamide 1-[2-bromoethyl(ethyl)amino]-4-methylanthracene-9,10-dione 2,4-bis(9H-fluoren-1-yl)thiophene (2R)-1-(4-fluorophenyl)sulfinyl-N,N'-dimethylpyrrolidine-2-carbohydrazide 2-[(4S)-6,9-dimethyl-3,4-dihydrocarbazol-1-yl]acetic acid (2Z,4E)-N-[3-(difluoromethyl)phenyl]-5-ethoxypenta-2,4-dienamide 2-(3,5-ditert-butylphenyl)-1-benzofuran (4-cyclohexylpiperazin-1-yl)-[2-(hydroxymethylamino)pyridin-4-yl]methanone 2-[4-chlorobutyl(2H-tetrazol-5-yl)amino]propanoic acid 2-[3-[[2-methylpropyl(4,5,6,7-tetrahydroindazol-1-yl)amino]methyl]phenoxy]-2-thiophen-3-ylacetic acid 4-[5-fluoro-6-(3,5,5,8,8-pentamethylnaphthalen-2-ylidene)cyclohexa-1,3-dien-1-yl]benzenethiol N-methyl-N-[4-(2,3,6,7-tetrahydro-1H-pyrrolo[2,3-d]pyrimidin-5-yl)cyclohexa-1,5-dien-1-yl]hydroxylamine 1-(2,5-dioxopyrrolidin-1-yl)-N'-[5-methoxy-6-[3-(trifluoromethyl)phenyl]pyridin-3-yl]cyclopropane-1-carbohydrazide N-(3-chlorophenyl)sulfonyl-2-[2-(2,6-dimethylphenyl)ethynyl]-1-[2-methoxy-4-(trifluoromethyl)phenyl]imidazole-4-carboxamide 2-[2,4-bis(trifluoromethyl)phenyl]-1H-imidazole-5-carboxylic acid 4-chloro-2,5-dimethylbenzonitrile;N-(1H-pyrazol-5-yl)-2,3,4,9-tetrahydro-1H-carbazole-3-carboxamide 1-azidooxy-N,N-dimethylindole-3-carboxamide N-[2,3-dihydroxypropyl(1,5-naphthyridin-4-yl)amino]acetamide 5-(2,4-dichloropyrimidin-5-yl)-N-ethyl-6-fluoro-1H-benzimidazole-2-carboxamide N-(4,5-dimethylpyridin-2-yl)-N',N'-bis[3-(2H-tetrazol-5-yl)propyl]ethane-1,2-diamine;trihydrochloride (6R)-4-ethyl-11-hydroxy-8,12-dioxo-N-[[2-(trifluoromethoxy)phenyl]methyl]-1,4,8-triazatricyclo[7.3.0.02,6]dodeca-9,11-diene-10-carboxamide (3E,5Z)-4-[2-chloro-6-[[5-methoxycarbonyl-7-[3-[(2R)-pyrrolidine-2-carbonyl]piperazin-1-yl]pyrazolo[4,3-d]pyrimidin-1-yl]methyl]phenoxy]-2,5-dimethylidenehepta-3,5-dienoic acid (1R,2S)-2-azido-4-(3-chlorophenyl)cyclopentan-1-ol 3-ethyl-2,4-dioxo-1H-quinazoline-7-carboxamide 6-chloro-4,7-dihydrotetrazolo[1,5-a]pyrimidine-5-carboxylic acid 6,8-dimethoxy-2-methylquinoline N-[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1H-thieno[3,4-d]pyrimidin-7-yl]azetidine-1-sulfonamide N-[5,6-dimethyl-3-(2,4,7-trimethylquinolin-6-yl)oxypyrazin-2-yl]cyclopropanesulfonamide N-[2-methyl-5-(2-morpholin-4-ylpyrimidin-4-yl)-1H-pyrrol-3-yl]thiophene-2-carboxamide N-[2-aminoethyl(propan-2-yl)carbamothioyl]benzamide 3-[(4,7-dimethyl-1H-benzimidazole-2-carbonyl)amino]-N-phenylcyclobutane-1-carboxamide (3S,4R)-1-[3-(3-cyanopyridin-2-yl)propanoyl]-4-hydroxypiperidine-3-carboxamide [3-methyl-2,4-bis(phenylmethoxy)phenyl]methanol 2,4-bis[(3R)-pyrrolidine-3-carbonyl]thiophene-3-sulfonamide;hydrochloride [3-(chloromethyl)-4,5-dihydrothieno[2,3-g]indazol-7-yl]methanamine 1-(4-chlorobutoxy)-2,3,5-trimethylbenzene 2-[4-[2-(2,6-difluorophenyl)-5-methyl-6H-pyrrolo[3,2-d]pyrimidine-7-carbonyl]piperazin-1-yl]-N,N-dimethylacetamide 2-tert-butyl-6-chloropyrrolo[3,4-b]pyridine-5,7-dione 3-[2-(2-methoxyethyl)-3-oxo-5-phenyl-1H-pyrazol-4-yl]propanoic acid N-[(1E)-1-(3,4-dichlorophenyl)buta-1,3-dienyl]propan-2-imine N-(6-oxo-4H-thieno[3,2-c]pyrazol-5-yl)benzamide 4-amino-6-[(5-bromo-2,3-diiodophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-methyl-N,7-diphenylpyrazolo[1,5-a]pyrimidine-3-carboxamide 5-(8,9a-dihydrodibenzofuran-3-yl)benzene-1,3-dicarbonitrile 5-[4-amino-3-(methylamino)phenoxy]carbonylfuran-2-carboxylic acid 4-(1H-indol-3-yl)-5-[5-phenylmethoxy-6-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-amine [1-azido-5-(9H-fluoren-1-yl)-2,3-dihydro-1,4-benzodiazepin-8-yl]hydrazine 6-(4-chlorophenyl)-7-hydroxy-2,4-dimethyl-5H-pyrazolo[1,5-a]pyrimidine 4-(1,3-benzothiazol-2-yl)-N-(2-chloropyridin-3-yl)piperidine-1-carboxamide 4-(2,5-dibromophenyl)pyrimidine-2-carboxamide 3-fluoro-2,6-diiodopyridine 4-(difluoromethoxy)-1,3-bis[2-methyl-5-(trifluoromethyl)phenyl]pyrazole 5-chloro-4-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrimidin-6-one 5-cyclopentyloxy-2-(3,4-dimethoxyphenyl)pyridine N'-(cyclopropanecarboximidoyl)-N-(4-phenoxyphenyl)carbamimidate N-[3,6-dimethyl-5-[2-(1H-pyrazol-4-yl)ethynyl]pyridin-2-yl]-4-iodo-2,5-dimethylbenzenesulfonamide 4-chloro-N'-[5-(2,6-dimethylphenyl)pyrimidin-1-ium-4-yl]butanimidamide 1-[2,4-bis(phenylmethoxy)phenyl]pentane-3,4-dione 1,3-diphenylpropylhydrazine 5-(4,5-dimethylcyclohexa-1,3-dien-1-yl)furo[3,2-c]pyridine (E)-1-[4-[2-(9,10-dihydroanthracen-1-yloxy)ethyl]piperazin-1-yl]-3-(3-methoxyphenyl)prop-2-en-1-one 3-[(4-azido-5-methylpyrazol-1-yl)methyl]-5-chloropyridine 6-[(5-methylthiophene-2-carbonyl)amino]hexanoic acid N-[6-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2H-pyridin-5-ylidene]hydroxylamine 6-[[2-(1,3-benzodioxol-5-yl)ethylamino]methyl]-2-cyclopropyl-N,4-dihydroxybenzamide 1-[(5R,7S)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]pyrazole-3-carboxylic acid 2-[4-amino-3-(methoxymethyl)phenyl]sulfanyl-4-propyl-1H-pyrimidin-6-one N-methyl-1,2-diphenylcyclopropane-1-carboxamide ethane;2-(4-fluorophenyl)-N-methyl-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide (1R,2S)-N-[4-[(2S)-3-cyano-6-ethoxy-2-methyl-4-oxo-2H-pyrido[2,3-d]pyrimidin-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide 4-[4-hydroxy-3,5-di(propan-2-yl)phenyl]-6-methoxy-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]pyridine-2-carboxamide 4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-pyridin-2-one N-[[3-(difluoromethoxy)phenyl]methyl]spiro[1,4,5,6-tetrahydroindazole-7,4'-piperidine]-2-carboxamide 1-azidooxy-4-butan-2-yloxybenzene 2,5-dimethyl-4,6-bis[2-(2-propan-2-ylimidazol-1-yl)ethoxy]pyrimidine;uranium(2+) 2-[4-(aminomethyl)phenoxy]-3H-pyrido[2,3-d]pyrimidin-4-one (5-bromothiophen-3-yl)-[(2R,6S)-2,6-dimethylmorpholin-4-yl]methanone 1-[(E)-but-2-enyl]-4-[1-(3,5-dichlorophenyl)ethoxy]benzene;propane N-(3-chlorophenyl)-2,4,6-trimethyl-3-[2-oxopropanoyl-[[5-[2-(2H-tetrazol-5-yl)phenyl]furan-2-yl]methyl]amino]benzamide (3E)-4-amino-3-[(5-butylthiophen-2-yl)methylidene]azete-2-thione 4-[3-[1,3-dioxo-2-(pyridin-2-ylmethyl)isoindol-5-yl]piperidine-1-carbonyl]benzonitrile 2-[2-(4-azidophenyl)ethyl]cyclohexan-1-one ethene;6-methyl-2-(2,3,4,5-tetrachlorophenyl)sulfanylnaphthalene 6-(dimethylamino)-4-hydroxynaphthalene-2-sulfonic acid (1S)-2-[4,5-bis(ethenyl)furan-3-carbonyl]cyclohexan-1-one N-[[5,6-bis(ethenyl)pyridin-2-yl]methylideneamino]-2-pyridin-4-ylbutanamide (NZ)-N-[1-(4-methylsulfonylphenyl)-2-(2-pyridin-3-ylethylamino)-2H-pyrrolo[2,3-d]pyrimidin-5-ylidene]hydroxylamine 3-chloro-4,5-difluoro-N-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzenesulfonamide 2-(4-azidophenyl)-1,3-dioxane N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-methoxyacetamide 4-(methoxymethyl)-6-(oxan-2-yloxymethyl)-7-[3-oxo-3-(2,2,2-trifluoroethylamino)propyl]-1H-quinoxaline-2,3-dione N-(5-chloropyridin-2-yl)-N-cyclohexylnonanamide 3-(2,4-difluorophenyl)-1-methyl-5-propan-2-yl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine (E)-1-[4,5-bis(prop-2-ynoxy)-3H-indol-6-yl]-3-thiophen-2-ylprop-2-en-1-one 1-methyl-4,5-dioxo-2,3-bis[(4-phenylcyclohexa-1,3-dien-1-yl)sulfonyl]isoindole-6-carboxylic acid [3-[4,6-bis(2-methoxyphenyl)pyridin-2-yl]oxybenzene-2-id-1-ylidene]azanide;zirconium(4+) 2-[3-(4-cyclohexa-1,5-dien-1-ylphenyl)propoxy]carbonylbenzoate 6-[(3,4-dimethoxyphenyl)methyl]-2-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-ethyl-N-[(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)methyl]-5-phenylpyrazole-1-carboxamide 2-methyl-6-[(4-phenoxyphenoxy)methylidene]piperidine N-(cyclohexylmethyl)-3-[5-ethenyl-4-(5-fluoropyridin-2-yl)-1,2,4-triazol-3-yl]aniline N-[3-(4,5-dichloroimidazol-1-yl)propyl]decanamide 1-azido-2,3,4-trichloro-5-methylbenzene 1-[3-(2,2,2-trifluoroethoxy)phenyl]ethanone 1-cyclopropyl-6-fluoro-7-[4-(5-hydroxy-1,3-dihydroisoindole-2-carbonyl)piperazin-1-yl]pyrido[2,3-d]pyrimidine-2,4-dione 1-[3-bromo-5-(trifluoromethyl)phenyl]-2,2,2-trichloroethanone 1-[(4-fluorophenyl)methyl]-3,5-dimethoxybenzene;toluene 4-[1,3-dimethyl-7-[(Z)-prop-2-enylideneamino]pyrazolo[3,4-c]pyridin-5-yl]phenol 2-(6,8-dimethoxy-3-methylimidazo[1,5-a]pyridin-7-yl)-4-methylmorpholine N-ethyl-4-[3-fluoro-5-(methylideneamino)phenyl]-1H-pyrrole-2-carboxamide 2-[N-(1,3-thiazol-5-yl)anilino]decanedioic acid ethane;3-methoxypyridine-2,6-diamine;N-(3-methylcyclobutyl)-3-propan-2-ylbenzamide 1-methyl-3-[5-(3-methylphenyl)pentyl]benzene 3-(2,6-dichlorophenyl)-7-[4-ethyl-4-(pyridin-4-ylmethyl)piperidin-1-yl]sulfanyl-5H-[1,3]oxazolo[4,5-d]pyrimidin-2-one 1,2-diamino-4-[4-(4-phenylmethoxyphenoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile 5-(methoxyiminomethyl)naphthalene-1,7-diol 1-chloro-2-[3-(3,5-dimethoxyphenyl)phenoxy]benzene;ethane 5-chloro-N,2-dimethyl-4-[(Z)-1H-pyrrol-2-ylmethylideneamino]oxyaniline 3-[2-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]phenyl]-5,6-dihydrobenzo[b][1]benzazepine 2-[4-(2-chloro-5,6-dihydroquinolin-3-yl)phenoxy]ethanol [4-(aminomethyl)piperidin-1-yl]-[2-cyclopropyl-6-[[5-(4-propan-2-ylpiperazin-1-yl)pyridin-2-yl]amino]pyrazolo[1,5-a]pyrimidin-3-yl]methanone 2-azidooxy-5,6-difluorobenzenesulfonic acid 1-azido-3,6-dichloro-2-methylindole N-[(3E)-hexa-1,3,5-trien-3-yl]-2-propan-2-ylidene-3H-1-benzofuran-4-amine 3-[[4-(cyclohexanecarbonyl)phenyl]iminomethyl]-7-fluoro-1H-indol-2-ol N-methyl-N-[1-(3-methylimidazo[4,5-b]pyridin-2-yl)piperidin-3-yl]ethenesulfonamide 2-(2-azidooxyphenoxy)-4,6-dimethylpyridine 2-[4-(1,3-diazepane-4-carbonyl)piperazin-1-yl]-N'-[3-methoxy-5-[(Z)-(2-oxo-2-propan-2-yliminoethylidene)amino]phenyl]ethanimidamide 4-[2,4,6-trimethyl-N-(1-phenylethyl)anilino]benzenesulfonic acid 2-(1-benzothiophen-5-ylsulfonylamino)-3-phenylpropanoic acid 1-ethyl-4-[(3S,4S)-4-methoxypyrrolidine-3-carbonyl]piperazine-2-carboxylic acid;hydrochloride 1-[4-[3-(2,5-dioxopyrrolidin-1-yl)propanoyl]piperazin-1-yl]-4,8-dimethoxyisoquinoline-6-carboxamide N-[1-(2-bromophenyl)propan-2-yl]-3-hydroxybutanamide 1,3-diethyl-2-phenyl-5H-indene 5-azido-2-butyl-1H-benzimidazole 4-[(Z)-2-amino-1,3-dicyanoprop-2-enyl]-N-methylbenzenesulfonamide 2-amino-5-[4-(4-fluorophenyl)phenyl]pentanoic acid 4-(7,8-dimethoxy-4H-[1,3]thiazolo[5,4-b]quinolin-2-yl)phenol 4-[3-(dimethylcarbamoyl)phenyl]-1H-pyrazole-5-carboxylic acid 2-bromo-N-[(3S)-7-fluoro-4,4-dimethyl-1,3-dihydroisoquinolin-2-yl]benzamide;(1S)-2-hydroxy-5,6-dimethoxy-1-methyl-1,2-dihydrobenzo[f]isoindole-3,9-dione (5S)-2-[(2-fluorophenyl)methylsulfanyl]-N-(2,4,6-trimethoxyphenyl)-7-(trifluoromethyl)-4,5,6,8-tetrahydropyrazolo[1,5-a][1,3]diazepine-5-carboxamide (7R)-7-azido-2-[3,5-difluoro-4-[6-methyl-8-(oxetan-3-ylamino)imidazo[1,2-a]pyridin-2-yl]anilino]-4,8-dimethyl-5H-pteridine-6-carboxylic acid N'-[6-(3,4-dimethoxyphenyl)-5-ethylpyridin-2-yl]propanimidamide 3-[(2R)-1-[[4-[2-fluoro-4-[4-(3-methylbutoxy)phenyl]phenoxy]oxan-2-yl]amino]propan-2-yl]oxy-5-propan-2-ylbenzonitrile N-[(1R)-1-phenylethyl]-2,3-dihydro-1H-indene-4-carboxamide (3R)-2,4,5-trimethyl-3-[4-(1-propan-2-ylazetidin-3-yl)oxybenzoyl]cyclohexane-1,2-dione 4-hydroxy-1-(2-methyl-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-ylidene)piperidine-4-carboxamide N-[(Z)-(5-bromo-2-hydroxyphenyl)methylideneamino]-1,3-benzodioxole-5-carboxamide N-cycloheptyl-5-(methoxyiminomethyl)-1H-indole-7-carboxamide 5-[2,3-difluoro-4-(trifluoromethoxy)phenyl]-1,3,6-trifluoro-2-(3,3,3-trifluoroprop-1-ynyl)naphthalene 5-[3-ethylsulfonyl-7-(trifluoromethoxy)imidazo[1,2-a]pyridin-2-yl]-2-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine 5-[2-(1H-indol-4-ylmethylamino)pyridin-3-yl]imidazolidine-2,4-dione 4-bromo-1-[(5S)-3,3,5-trimethylcyclohexyl]indole 1-[(3R,4S)-4-hydroxy-3-propan-2-ylpyrrolidin-1-yl]-5-phenylpentane-1-thione 5-[4-fluoro-2-[(3-methyloxetan-3-yl)oxycarbonylamino]phenyl]furan-3-carboxylic acid 2-[4-(4,5-dimethyl-1H-pyrazole-3-carbonyl)morpholin-3-yl]-N-ethylacetamide (NZ)-N-[5-cyclopropyl-3-[2,6-dichloro-4-(trifluoromethoxy)phenyl]-3H-1-benzothiophen-2-ylidene]hydroxylamine 1-[5-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonylamino)pentyl]cyclohexane-1-carboxylic acid N-[(3R)-1-[6-(2,5-dimethylpyrrol-1-yl)pyridine-3-carbonyl]pyrrolidin-3-yl]-2-fluorobenzamide 4-[(2S)-6-(6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-2-carbonylamino)-4,8-difluoro-9-methoxy-2,3-dihydro-1H-pyrrolo[3,4-c]isoquinolin-5-yl]benzoic acid 4-[3-fluoro-5-(trifluoromethyl)phenyl]-1H-tetrazol-5-one 4-[2,5-dichloro-N-(4-hydroxybutyl)anilino]benzenesulfonamide 3-[(2,4-dioxoimidazolidin-1-yl)methyl]-N'-hydroxypyridine-2-carboximidamide N-[[(2R,4S)-1-acetyl-4-fluoropyrrolidin-2-yl]methyl]-4-chlorobenzamide 2-azido-N-[(3R)-1-[4-[ethyl-[2-(methylamino)acetyl]carbamoyl]benzoyl]pyrrolidin-3-yl]imidazo[1,5-a]pyridine-7-carboxamide 2-[(3E)-4-methoxyhexa-1,3,5-trien-3-yl]-5-(1H-pyrrolo[3,2-b]pyridin-6-yl)pyrimidin-4-amine 2-amino-4-(4-hydroxyphenyl)-5-oxo-6H-pyrrolo[3,4-d]pyrimidine-7-carbonitrile 2-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]acetate N-[(E)-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)-2-hydroxybut-2-enoxy]-5-(trifluoromethyl)pyrazine-2-carboxamide 4-[(E)-[(6R)-6-ethyl-5,6,7,8-tetrahydroquinazolin-2-yl]iminomethyl]phenol N-(4-methoxybutyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidine-7-carboxamide 2-[4,7-difluoro-3-(1H-indole-6-carbonyl)quinoxalin-2-yl]acetonitrile 2-(1-cyclopropylethylamino)-3H-quinazolin-4-one 1-(4-fluorophenyl)-N'-[5-methyl-6-oxo-4,7-bis(phenylsulfanyl)pyrrolo[3,4-d]pyrimidin-3-yl]piperidine-4-carboximidamide 2-(aminomethyl)-6-[(1E,3Z)-2-(trifluoromethoxy)hexa-1,3,5-trienyl]aniline N'-(benzenecarbonothioyl)-N,2-dimethylpropanehydrazide 2-[3-(4-propan-2-yloxybenzoyl)benzimidazol-5-yl]acetic acid N-[(1R,2S)-1-amino-1,3-dimethoxy-4,4-dioxo-5-phenylpentan-2-yl]piperidine-2-carboxamide;hydrochloride 4-[(4-aminoquinolin-2-yl)methylamino]benzamide 1-cyclopentyl-4-[3-(3,5-difluorophenyl)-3,4-dihydropyrazole-2-carbonyl]piperidine-4-carboxamide 1-methyl-6-[[5-(4-nitrophenyl)thiophen-2-yl]sulfanylamino]indole-2,3-dione [(4S)-3,9-dimethyl-5-thia-1-azatricyclo[6.2.0.02,6]decan-7-yl]-[6-(pyridin-2-ylsulfanylamino)pyridin-3-yl]methanone 2-(6-aminopyridin-3-yl)-N,N,5-trimethylpyrimidine-4-carboxamide N-butyl-5,5,6-trifluoro-4-(7-methoxynaphthalene-2-carbonyl)cyclohexa-1,3-diene-1-sulfonamide N-[(E)-3-[4-hydroxy-5-(piperidin-1-ylmethyl)thiophen-2-yl]pent-2-en-2-yl]-4,5-dihydro-1H-imidazole-2-carboxamide 1-(2,6-dimethylphenyl)-4-[5-(trifluoromethoxy)pyridin-3-yl]triazole 4-[2-(dimethylamino)ethoxy]-1,10-dihydroanthracene-9,10-dione 3-(6,7-difluoro-3,4-dihydroisoquinolin-2-ium-2-yl)-1H-pyrrolo[2,3-b]pyridine 1-[4-(6,7-dimethoxyquinolin-4-yl)oxy-2-fluorophenyl]-3-propan-2-ylurea N-(4-chloro-3,5-dimethylphenyl)-2-[(6S)-2-ethyl-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 2-(4-bromophenyl)-N-phenylmethoxyacetamide 2-[4-(azidomethyl)phenyl]-N'-hydroxy-3,5-dioxo-6H-imidazo[1,5-c]imidazole-7-carboximidamide 2-azido-3,4,5-trifluorophenol 3-[(2S)-2,4-dimethylpiperazine-1-carbonyl]benzamide 4-[3-[4-(N'-methanimidoylcarbamimidoyl)anilino]-1,2-oxazol-5-yl]-3-(trifluoromethoxy)benzonitrile 2-chloro-4,5,6-tris(3,5-ditert-butylphenyl)pyrimidine 5-amino-3-(4,6-diethoxy-2-oxochromen-3-yl)-1H-pyrazole-4-carbonitrile (2-azidophenyl)methoxy-[dimethylphosphoryl(methyl)amino]methanol 2-(4-methylpiperazin-1-yl)-5H-pyrido[3,2-b]indole;4-(2-pyrrolidin-1-ylpyridine-4-carboximidoyl)benzenethiol 4-[3-(benzenesulfonamido)propyl]piperazine-1-carboxylic acid 4-[[[5-chloro-2-(trifluoromethyl)phenyl]sulfanylamino]methyl]-3-hydroxy-N-[3-(1,1,2,2-tetradeuteriopropyl)phenyl]thiophene-2-carboxamide N-[1-(4-azidophenyl)pyrazol-3-yl]pyrimidin-2-amine 6-bromo-3-[(4-propan-2-ylphenyl)methylimino]spiro[1,4-dihydroquinoxaline-2,4'-piperidine]-5-carboxamide N-[4-chloro-3-(5-hydroxy-1,3-dihydroisoindole-2-carbonyl)phenyl]acetamide (Z)-3-amino-2-[5,8-dimethyl-9-(6-piperidin-1-ylpyridine-3-carbonyl)oxy-1,2,3,4-tetrahydrocarbazol-3-yl]but-2-enimidamide 3-[4-(2,6-dimethylphenyl)-1,2,4-triazol-3-yl]-N-phenylaniline 2-[(2R)-1,4-dioxaspiro[4.5]decan-2-yl]-6-ethoxy-N-[(3S)-5,7-dimethyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]pyrimidine-4-carboxamide 3-(4,6-diphenylpyrimidin-2-yl)pyridine-2-carboxamide N-(4-chlorophenyl)-2-[[4,7-dioxo-3-propan-2-yl-2-sulfanylidene-6-[[3-(trifluoromethyl)phenyl]methylsulfanyl]-1H-thieno[3,2-d]pyrimidin-5-yl]sulfanyl]acetamide 5-[[4-cyclopropylimino-2-[(3,4-dimethoxyphenyl)methylamino]pyrazolo[1,5-a][1,3,5]triazin-8-ylidene]methyl]-1,3-diethylbenzimidazol-2-ol (3E)-6,10-bis[2,4,7-tris(sulfanylidene)-1H-pyrimido[1,2-a]benzimidazol-3-yl]deca-1,3-dien-4-one 6-[(4-hydroxyphenyl)methyl]-2-pyridin-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-(1H-imidazo[4,5-b]pyridin-2-yl)-N-phenylmethoxyazetidine-1-carboxamide 2-(2,6-dimethylpyrimidine-4-carbonyl)-9-phenyl-6-oxa-2,9-diazaspiro[4.5]decan-8-one 3-[N-(4-hydroxybutyl)-2,6-dimethoxyanilino]propane-1,2-diol 3-methyl-2-[4-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)methoxy]phenyl]butanoic acid N-[(2,6-dichlorophenyl)methyl]-3-methoxynaphthalene-2-carboxamide 2-[4,7-dimethyl-1-(oxan-4-yl)indazol-3-yl]oxy-N-pyridin-2-ylsulfonylacetamide N-(6-azaspiro[2.5]octan-2-yl)-4-chlorobenzenesulfonamide 5-[2,6-dimethoxy-4-(2-phenoxyethyl)phenyl]imidazolidine-2,4-dione [2,3-bis(methylsulfanyl)phenyl]-hydroxyazanium 4-(2,3-dihydropyrrol-1-ylsulfonyl)benzenesulfinic acid 2,7-dibromonaphthalene-1,8-disulfonic acid 2-[2-(4-methylpiperazin-1-yl)ethoxy]-9,15-diazatetracyclo[8.6.0.03,8.011,15]hexadeca-1,3,5,7,9,11,13-heptaene 2-azidooxy-N-methylpyridine-3-carboxamide 6,7-dihydroxynaphthalene-1,2-disulfonic acid 1-[2,6-dichloro-4-(2-cyclohexylethoxy)phenyl]piperazine 1-[(4R)-6,7-diethoxy-3,4-dihydro-2H-chromene-4-carbonyl]piperidine-4-carboxylic acid (2E)-4,5-dimethoxyhexa-2,4-diene;5-(3,4-dihydro-1H-isoquinolin-2-ylsulfinyl)quinoline 1-(3,4-difluoro-5-methylphenyl)ethanone;2-methylbutane;6-methyl-3,3a,4,8b-tetrahydroindeno[1,2-c]pyrrole N'-[1-(3-cyanophenyl)pyrrolidin-3-yl]methanimidamide 1-[6-(2,2-difluoroethyl)thieno[3,2-d]pyrimidine-4-carbonyl]azetidine-3-carboxamide (Z)-3-[4-tert-butyl-5-ethoxy-2-(trifluoromethyl)phenyl]-N-ethyl-1,2-diphenylprop-2-en-1-imine 2-(4,6-dichloropyrimidin-5-yl)oxybenzonitrile 4-chloro-2,3-dinitrophenol 2-[3-[[5-chloro-4-(methylamino)pyrimidin-2-yl]amino]phenyl]ethanol 2-amino-N'-[[5-(6,7-dihydroquinolin-4-yl)pyridin-3-yl]methyl]-5-fluoropyridine-3-carboximidamide N-[1-(3,4-dimethoxyphenyl)ethyl]formamide;2,6-dimethyl-5-[4-(1H-pyrazol-5-ylsulfanyl)anilino]hexanenitrile 2-(3,4-dichlorophenyl)-6-[(4-methylpyrazol-1-yl)methyl]pyridine 2-chloro-5-[4,7-dihydroxy-6-(hydroxymethyl)-9,9-dimethoxyxanthen-3-yl]phenol (2Z)-4-[3,5-bis(trifluoromethyl)phenyl]-N-ethoxy-6-fluoro-3-[(E)-prop-1-enyl]hexa-2,4-dienamide N-butyl-4-(2,3-dihydro-1H-indazol-5-ylmethyl)aniline N-(1,3-benzodioxol-5-ylmethyl)-2-(cyclobutanecarbonylamino)pyrimidine-4-carboxamide 1-[6-(aminomethyl)pyrazin-2-yl]-3-azidoindazole-7-carboxamide 4-(2-acetamidoimidazo[1,2-b]pyridazin-6-yl)oxy-N-cyclopropyl-3-methylbenzamide N-(3,5-dimethylpyridin-4-yl)-6-fluoroquinoxaline-2-carboxamide 2-[6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-9H-xanthen-3-yl]pyridine 4-(1,3,2-dioxathiolan-4-yl)benzenesulfinate N-(3,4-dihydronaphthalen-2-yl)-2-[(1Z,3E,5Z)-hepta-1,3,5-trienyl]-N'-methylbenzenecarboximidamide 2-[N-(carboxymethyl)-3-hydroxyanilino]octanoic acid 2-[3-chloro-5-(trifluoromethyl)phenyl]-N,N'-diphenylethanimidamide 3-amino-5-(3,4-dimethoxyphenyl)-6-[(2E,4Z)-6-ethenylhepta-2,4-dien-2-yl]-N-[1-(3-fluorophenyl)ethyl]pyrazine-2-carboxamide 2,6-ditert-butyl-4-(cyclohexa-1,5-dien-1-ylmethylamino)phenol 2-(1,3-benzothiazol-2-ylsulfanyl)-N'-[(2-ethoxyphenyl)methylideneamino]acetohydrazide (5E)-2-(4-chlorophenyl)imino-5-[[4-[(3,4-difluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-1,3-thiazolidin-4-one 5-chloro-4-[4-(2,3,5-trifluorophenyl)piperidin-1-yl]sulfonyl-1H-pyrazole 1-N',2-N',3-trimethyl-2-N-(5-phenylsulfanyl-1,3-thiazol-2-yl)butane-1,1,3-triamine 2-(4-bromophenyl)-7-[1-[(4-chlorophenyl)methyl]piperidin-4-yl]oxyimidazo[2,1-f][1,2,4]triazin-4-amine 1-cyclopropyl-3-[6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonylamino)-1H-benzimidazol-2-yl]urea 2-[(E)-1-bromoprop-1-enyl]-3-chloro-6-(difluoromethoxy)-4-(4-methoxyphenyl)quinoline 4-[2-ethoxyethyl(methyl)amino]-1H-pyrimidin-6-one (2S)-3-[4-(cyclopropylmethoxy)phenyl]-1-N-[(6,7-dichloroquinolin-4-yl)methyl]propane-1,2-diamine (4Z)-2-methyl-6-phenylhepta-1,3-diene-3-thiol (2S,4R)-1-azido-4-phenylsulfanylpyrrolidine 4-(2,5-dimethyl-1H-imidazol-3-ium-4-yl)-N-methoxy-2-(trifluoromethyl)aniline;chloride 6-(cyclopentylamino)pyridine-3-carboxamide N-[5-tert-butyl-3-(4,5-dimethylpyrimidine-2-carbonyl)pyrazin-2-yl]acetamide 4-[[(2Z)-2-[6-(cyclopropylmethoxy)pyridin-3-ylidene]ethyl]amino]benzoic acid;ethane 1-[(6-methoxypyridin-2-yl)methyl]-3-(piperidin-4-ylamino)thiourea 1-azidooxy-4,5-dimethyl-2-propan-2-ylidenetriazolidine 2-(1,3-dioxol-2-yl)benzo[g]indazole N-[1,3-bis(2,6-dichlorophenyl)-3-oxopropylidene]hydroxylamine 1-[3-(4-ethylphenyl)sulfonyloxy-5-(2-methoxyphenoxy)phenyl]-N,N-dimethylmethanamine 4-[[2-(cyclohexylamino)-3,5,6-trimethylpyridine-4-carbonyl]amino]bicyclo[2.1.0]pentane-1-carboxylic acid 1-chloro-3,5-dimethylbenzene;formaldehyde;3-[4-[[(3S)-6-hydroxy-7-(3-piperidin-1-ylpropoxy)-2,3-dihydro-1H-inden-4-yl]oxy]phenyl]hex-4-ynoic acid 1-(cyclopropylmethylamino)-3-[(4-fluorophenyl)methyl]urea 6-(2,5-dimethylpyrrol-1-yl)-3-(4,4,5,5-tetramethyloxaborolan-2-yl)quinoline 1-[(4-methoxyphenyl)methyl]piperidine-3-carboxamide (4-aminocyclohexa-1,3-dien-5-yn-1-yl)-(2-butan-2-ylidene-7,8-dihydro-4H-pyrazolo[4,3-b]azepin-5-yl)methanone 1-chloro-4-[(3S,5S)-5-ethyl-2,3,4,5-tetramethylhexan-2-yl]benzene (E)-3-[1-aminoethylidene-[5-(2,4-difluorophenyl)thiophen-2-yl]azaniumyl]-N'-[6-chloro-2-(3,4-dihydropyridin-5-yloxy)pyrimidin-4-yl]prop-2-enimidamide 3-azido-1,2-dinitronaphthalene N-(4,5-dimethyl-1H-pyrazol-3-yl)pyrazine-2-carboxamide (5E)-2,4,6-trioxo-5-[[3-(1H-pyrrol-2-yl)phenyl]methylidene]piperidine-3-carbonitrile 6-cyclohexyloxy-N-(2,4-difluorophenyl)pyridine-3-carboxamide (E)-1-[3-[5,7-difluoro-2-[4-(1,2,2-trifluoroethenoxy)phenyl]quinolin-4-yl]sulfanylpyrrolidin-1-yl]but-2-en-1-one 2,3-bis(ethenyl)-5-propan-2-ylidene-1H-indeno[4,5-f]indole 6-methyl-3-[(2E)-2-[1-(4-nitrophenyl)ethylidenehydrazinylidene]-2-oxoacetyl]-1,5-dihydro-1,2,4-triazin-4-one 6-(2,5-dichlorophenoxy)-2,3-dihydrothiochromen-4-one N-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-6-[6-(methoxymethyl)pyridin-2-yl]sulfonyl-1H-benzimidazole-2-carboxamide 5-(2,3-dichlorophenyl)imidazolidine-2,4-dione N-(3,4-dimethylphenyl)-2-oxo-4-(2,3,4,5-tetrahydropyridin-6-yl)pentanamide 7-(3,4-dichlorobenzoyl)-2-[4-(1,3-oxazole-5-carbonyl)piperazin-1-yl]-3-propanoyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-one 2-[(Z)-2-aminoprop-1-enyl]-3,5-dichloroaniline 2-(2-ethylbutanoylamino)-2-[4-methoxycarbonyl-6-phenylmethoxycarbonyl-1,3-dihydrobenzimidazol-2-ylidene]acetate 1-(5-bromopentoxy)-4-methylnaphthalene N-methyl-4-[(5-nitroindazol-2-yl)oxymethyl]aniline 3-[1,2-dihydroxy-2-(4-iodophenyl)ethenyl]cyclohexan-1-one (E)-2-cyano-3-[4-[1-(cyclopropylmethoxymethyl)-7-methoxyindol-5-yl]pyridin-3-yl]prop-2-enamide 2-(3,5-dimethylphenyl)-6-[1-(2,4,6-trifluorophenyl)ethylidene]cyclohexane-1,3-dione 2-tert-butyl-N-[6-(4,4-difluoroazepan-1-yl)-2-phenylmethoxypyridin-3-yl]benzenesulfonamide 5-(3,4-dichlorophenyl)-N'-hydroxypyridine-2-carboximidamide (E)-1-[2-chloro-5-methyl-4-[1-[[2,2,2-trifluoro-1-[3-[4-[2-[(2-methylpropan-2-yl)oxy]ethoxy]ethoxy]phenyl]ethylideneamino]amino]ethenylamino]phenyl]-N-ethyl-3-[2-(trifluoromethyl)pyridin-4-yl]prop-2-en-1-imine 1-(azidomethyl)-4-(1,3-benzodioxol-5-ylmethoxy)piperidine 2-[6-[5-(hydroxymethyl)-1-methylpyrazol-4-yl]isoquinolin-3-yl]-N-[(3S,5R)-5-methylpiperidin-3-yl]pyridine-4-carboxamide N-[6-(4-fluorophenyl)pyrimidin-4-yl]-5,6,7,8-tetrahydronaphthalene-2-sulfonamide 4-hydroxy-6-[propyl(2,3,4,5,6-pentafluorophenyl)sulfonylamino]naphthalene-2-sulfonic acid N-cyclopropyl-2,6-difluoro-4-[4-(1H-indazole-3-carbonyl)piperazin-1-yl]benzamide 1-[2,4-dichloro-3-[(7H-purin-6-ylamino)methyl]benzoyl]pyrrolidine-2-carbonitrile;2,2,2-trifluoroacetic acid (5R)-N'-[(Z)-1H-indol-3-ylmethylideneamino]-5-phenylpyrrolidine-2-carboximidamide 1-cyclopropyloxycarbonyl-4-phenylmethoxycyclohexane-1-carboxylic acid 1-[4,6-bis(1-methoxybutyl)pyrimidin-2-yl]-N-ethyl-N-propylpiperidin-4-amine [7-(4-chlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-ylidene]methanol 1-[2,6-di(propan-2-yl)phenyl]-3-[(E)-[2-[4-(tetrazol-1-yl)anilino]pyrimidin-5-yl]methylideneamino]urea 6-[4-[2-[1-[(E)-but-2-enyl]piperidin-4-ylidene]ethylamino]piperazine-1-carbonyl]-7,8-difluoro-4H-1,4-benzoxazin-3-one 2-[4-(1,3-benzodioxol-5-ylsulfonyl)piperazin-1-yl]-1H-indole (3S,6aS)-3,6a-dimethyl-5-phenyl-2,3,5,6,7-hexahydropyrrolo[2,1-c][1,4]oxazol-4-one 4-(7-ethylquinolin-4-yl)oxy-N,2-dimethylbenzamide 1-[2,3-dihydroxypropyl(ethenylsulfonyl)amino]-N-(4-phenyl-1,3-thiazol-2-yl)pyrrolidine-2-carboxamide [(2S,4R)-3,3-dimethyl-1,4-bis(phenylmethoxy)pentan-2-yl]phosphane 7-chloro-6,8,13,16,17-pentazatetracyclo[8.7.0.02,7.012,15]heptadeca-1(10),2(7),3,5,11(15),14-hexaene 5-fluoro-3,8-bis(trifluoromethyl)quinoxaline 1-(4-methoxyphenyl)-3-(2H-pyran-6-ylsulfonylamino)thiourea 2-(1,4-dioxan-2-yl)-N-[1-(3-hydroxy-6-methylpyridin-2-yl)ethylidene]acetamide 5-bromo-4-N,6-dimethyl-2-N-[4-(2H-triazol-4-yl)phenyl]pyrimidine-2,4-diamine N-butyl-6,7-dimethoxyquinazolin-4-amine 2-(1,3-benzothiazol-2-yl)-4-[6-(2-bromoethoxy)pyridin-3-yl]pyrazolidine-3,5-dione (1R)-2,2,2-trifluoro-N'-[3-fluoro-4-[[5-methylsulfonyl-1-[4-(trifluoromethoxy)phenyl]imidazole-4-carbonyl]amino]benzoyl]-1-methylcyclopropane-1-carbohydrazide 2-(3-aminophenyl)-N'-[(1S,2R)-2-hydroxycyclohexyl]-5H-pyrrolo[2,3-b]pyrazine-7-carboximidamide 7-methyl-3,5-bis(4-methylphenyl)-3aH-pyrrolo[2,3-b]pyrazine 1-[4-(2,6-dichlorophenyl)piperazin-1-yl]propan-2-ol N-(2-methoxy-4-nitrophenyl)-5-methylpyrimidine-4-carboxamide 2-[3,5-dimethoxy-4-(2-methylpyrazol-3-yl)phenyl]-7-(5-fluoropyridin-3-yl)imidazo[1,2-a]pyrimidine 4-(4-azidophenyl)-2-fluorophenol N-(3-fluorophenyl)-2,4,5-trimethylfuran-3-carboxamide 2-[3-(cyclohexylmethoxy)-5-(2,4-diaminophenoxy)phenyl]acetic acid N-[6-(3,5-dichlorophenyl)sulfanylpyridin-2-yl]-1H-indazole-6-carboxamide;ethane N-methyl-1,3-bis(4-phenoxyphenyl)propan-2-imine 4-bromo-2-[2,2-difluoroethoxy(methyl)amino]-1H-pyrimidin-6-one 1-(4-bromophenyl)-3-(2,4-dimethylphenoxy)piperidine 2-[4-(diethylamino)phenyl]-3-[(Z)-octadec-9-enyl]chromen-4-one 4-(4-chlorophenyl)-6,7-dimethoxy-2-[4-(1,3-oxazol-5-yl)phenyl]quinazoline N-(5,6-dimethylpyridin-3-yl)pyrimidine-4-carboxamide 1-(2,6-dimethoxyphenyl)-N-[5-ethylsulfonyl-4-(trifluoromethyl)pyridin-2-yl]-3-methylsulfanyl-2H-indol-7-amine 2-ethylsulfanyl-6,7-dimethyl-5-propan-2-ylpyrrolo[3,4-d]pyrimidine 4-[3,5-dibromo-2-hydroxy-6-(trifluoromethyl)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile [(4Z,6E)-4-ethoxydeca-1,9-dienyl]benzene 1-methyl-2,3-bis(2-methylphenyl)pyrazine [4-(3,3a,4,5,6,6a-hexahydro-2H-pyrrolo[2,3-c]pyrrole-1-carbonyl)-2,3,4,5-tetrafluorophenyl]azanide 4-[2,6-dichloro-3-fluoro-4-(oxetan-3-yloxymethyl)phenyl]piperidine 6-hydroxy-2,8-dimethyl-1H-quinazoline-4-thione [5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]urea 1-butanoyl-N-cyclopropyl-4-hydroxybenzenesulfonamide;4-[2-(4-methoxyphenyl)ethynyl]-3,5-dimethylpyridine N-[[(6S)-2-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl]methyl]-3-phenylpyrrolidine-1-carboxamide 4-methyl-2-[3-(trifluoromethoxy)phenyl]-5,6,7,8-tetrahydroquinazoline 1,3-bis(2-methylprop-2-enoyloxy)naphthalene-2-sulfonic acid 2-[[6-(2,3-dihydropyrrol-1-yl)pyridine-3-carbonyl]amino]acetic acid 5-butyl-7-[4-(diethylamino)phenyl]-2,3,9-trimethylpyrido[1,2-a]pyrimidin-8-one 3-[5-[(2S)-2-[4-(N,3-dimethylanilino)piperidine-1-carbonyl]pyrrolidine-1-carbonyl]pyridin-2-yl]benzonitrile 2-chloro-1,3-bis(ethenyl)-9H-fluorene 3-(4-cyanophenyl)sulfanyl-N,N-dimethylprop-2-enimidamide 4-(4-propanoylphenyl)-1,3-thiazole-2-carboxylic acid 2-[(4-chloro-3,5-dimethylphenoxy)methoxy]-N-ethylethanamine 4-cyclopropyl-3-[2-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]morpholine 3-amino-N',5,7-trimethyl-6-(1-methylindol-4-yl)oxypyridine-2-carboximidamide 3-[(2,3-diethoxy-4-methylphenyl)methylidene]-6-ethoxy-5-propanoylcyclohexa-1,4-diene-1-carboxylic acid 1-cyclopropyl-2,3-dimethoxybenzene;3-[5-fluoro-1-(4-phenoxybenzoyl)pyrrolidin-3-yl]oxybenzaldehyde N-[1-(dimethylamino)propan-2-yl]-3-nitrobenzenesulfonamide 2-(7,8-dihydronaphthalen-1-yl)-6-fluoro-N-methylidenebenzamide;methane 5-benzyl-N,2,4-trimethylaniline 2-amino-4,5-bis(prop-1-enyl)benzenesulfonic acid N-[1-(2,3-dimethoxyphenyl)ethyl]-7H-purin-6-amine 1-methylsulfonyl-3-[2,4,6-tri(propan-2-yl)phenyl]urea 3,5-ditert-butylaniline;ethane (1S)-4,4,8-trimethyl-5H-[1,3]dioxolo[4,5-g]chromene 1-[6-(4,5,6,7,8,9-hexahydro-2H-carbazol-1-yl)-1,3-benzothiazol-2-yl]pyrrolidin-2-one 2-(azidosulfanylmethyl)-5-ethoxyphenol N-[3-(6-azidopyridin-2-yl)phenyl]-5,8-diazaspiro[3.4]octane-8-carboxamide 2-amino-4-(1,5-dimethylpyrazol-3-yl)benzenecarboximidamide 1-[(4-cyclopentylphenyl)methoxy]-3-fluoro-5,6-dihydrobenzo[b]carbazole 6-bromo-2-[(E)-1,3-diaminoprop-2-enylidene]-1H-indole-7-carboxamide 3-azido-4-chloronaphthalene-1,5-disulfonic acid 4-[[3-(1,3-thiazol-2-yl)phenoxy]methyl]aniline N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N'-(4-ethoxyphenyl)butanediamide (5R)-3,8-diethyl-2-phenyl-7-phenylmethoxy-5H-1,3-benzothiazol-6-one N-[2-(4,4-difluoropiperidin-1-yl)ethyl]-5-methylfuran-3-carboxamide 1-azido-3-benzyl-4-chloro-5-(trifluoromethyl)pyrazole 3,4-difluoro-N'-hydroxy-5-[(2-methoxyethylamino)methyl]benzenecarboximidamide 4-[2-(1,3-benzothiazol-2-yl)-2H-quinolin-6-ylidene]butanoic acid 6-[(2,3-difluorophenyl)methyl]-1H-indazole 2-[4,5-dimethoxy-6-(2-methylpropanimidoyl)pyridin-3-yl]acetaldehyde 4-[(E)-2-cyanoethenyl]-3-methoxycarbonylbenzoic acid (4R)-1-[(2S,3S)-3-amino-3-methyl-2-phenylbutanoyl]-N,N-diethyl-6-phenyl-3,4-dihydro-2H-quinoline-4-carboxamide 1-[2,3-dihydroindol-1-yl(phenyl)methyl]-4-[(5R,7S)-5-pyridin-3-yl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]pyrrole-2-carboxylic acid (1S)-1-(3,4-dimethoxyphenyl)sulfonyl-N-[1-(2H-triazol-4-yl)ethyl]propane-1,3-diamine 3-(2,6-dichlorophenoxy)-N'-hydroxypyridine-4-carboximidamide 5-[2-(3,4-difluorophenyl)pyrrolidin-1-yl]sulfonyl-N-[4-methoxy-6-(pyrazol-1-ylmethyl)pyridin-2-yl]furan-2-carboxamide 4-amino-2-hydroxy-6-(2-hydroxy-3,5,5-trimethylhexyl)benzoic acid 1-[(3R,4S)-4-(4-cyclopropylimidazol-1-yl)-3-hydroxypiperidin-1-yl]-2-(tetrazol-1-yl)ethanone 1-(4,5-ditert-butyl-1H-pyrazole-3-carbonyl)pyrrolidine-2-carboxylic acid 4-fluoro-N-[2-methyl-3-[[(1S)-1-[5-(trifluoromethyl)pyrimidin-2-yl]ethyl]carbamoyl]phenyl]benzamide N-methylformamide;2-[3-(4-propan-2-ylphenyl)phenyl]-1,10-phenanthroline 3-(4,6-dimorpholin-4-yl-1H-benzimidazol-2-yl)propanoic acid [3-(1H-imidazol-5-yl)morpholin-4-yl]-(2-methoxy-4,6-dimethylpyridin-3-yl)methanone 2-[2,6-difluoro-N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)anilino]acetic acid 4-(2-chlorophenyl)sulfanylaniline N-(3,5-dichlorophenyl)sulfanyl-2,4,6-trimethylaniline N-(3,4-dimethylphenyl)-5-fluoro-6-methoxypyrazine-2-carboxamide 2-[4-(benzylamino)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-b]azepin-2-yl]phenol 6-[1,3-benzodioxol-5-ylsulfonyl(methyl)amino]-2-(4-phenylpiperazine-1-carbonyl)-1H-indole-3-carboxylate 1-(5,7-difluoro-2,3-dihydroindole-1-carbonyl)pyrazole-4-carboxylic acid 1-[3-(4-ethylphenyl)hexan-2-yl]imidazole 2-(3,4-diethoxyphenyl)-N-[5-(1H-pyrrol-2-ylmethylideneamino)pentyl]benzamide 6,8-dimethoxy-1,2-benzothiazine N-[4-[(E)-2-cyclopropyloxyethenyl]phenyl]-1,3-dimethylpyrazole-4-carboxamide (2R)-N-[3,5-dichloro-4-(1H-indole-6-carbonylamino)phenyl]-1-phenylsulfonylpyrrolidine-2-carboxamide (2S)-3-[4-(1,2,4-triazol-4-yl)phenyl]propane-1,2-diamine;hydrochloride 5-[2-ethoxyethyl-[6-(4-methylphenyl)pyridazin-3-yl]amino]pyridine-2-carboxylic acid (2-azidooxycyclohexa-1,3-dien-1-yl)benzene (3aR,6aR)-5-[6-methyl-4-(trifluoromethyl)pyridine-2-carbonyl]-1,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-2-one 2,4-dichloro-N-(1-phenylethyl)aniline (2R)-1-N-[4-methoxy-6-(2,2,2-trifluoroethylamino)-1,3,5-triazin-2-yl]-3-(methylsulfanylamino)propane-1,2-diamine 4-[2,5-difluoro-3-methyl-3-(2H-pyrazolo[3,4-b]pyridin-5-yl)indol-1-yl]benzoic acid N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-[4-hydroxy-1-(2-methoxyethyl)piperidin-4-yl]acetamide N'-(3,4,5-trifluorophenyl)benzohydrazide 2-azido-5-bromo-N,3-dimethylbenzenesulfonamide N'-[(Z)-2,3-dihydroxyprop-2-enimidoyl]-6-ethyl-3-methoxy-N-phenylpyridine-4-carboximidamide N-[3-(1,2,5-oxadiazol-3-yl)oxolan-3-yl]butanamide 2-(2,3-difluorophenyl)imidazo[1,2-a]pyridine;ethane N-[4-(5,7-dimethyl-1,3-benzothiazol-2-yl)phenyl]sulfanylpropan-2-amine 5-[3-[7-(4,6-diphenylpyrimidin-2-yl)-3H-imidazo[4,5-c]pyridin-2-yl]-1H-isoindol-5-yl]-N,N-dimethylpyridin-3-amine 4-(dimethoxyphosphorylmethyl)-2,6-bis[4-fluoro-3-(trifluoromethyl)phenyl]pyrimidine N-[(4R)-7-ethyl-2,2-dimethyl-3,4-dihydrochromen-4-yl]propanamide 3-(1,3-benzodioxol-5-yl)-6,7-bis[(4-bromophenyl)methoxy]quinazolin-4-one (4Z)-5,6-dimethyl-2-oxo-N-[(2S)-1-phenylethoxy]hepta-4,6-dienamide 4-[(2S,3R)-1-butanoyl-2-methylpiperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one 2-azidooxy-4,6,7-trimethyl-1H-benzimidazole 3-[4-[2-(6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl)ethylsulfanyl]phenyl]-N-propan-2-ylidenepropanamide 1-(5-chloropyridine-2-carbonyl)-N-(2,6-diethylphenyl)piperidine-3-carboxamide 4-hydroxy-5,7-dimethyl-3-(2-nitrophenyl)sulfanylnaphthalene-2-carboxamide 4-[(1R)-2-(3,5-dimethyl-4-propan-2-yloxyphenyl)-6-fluoro-1-hydroxy-8,9-dimethyl-5H-pyrimido[5,4-d]azepin-7-yl]piperidine-1-carboxylate 4-(2,1,3-benzothiadiazol-4-yl)benzonitrile;iridium;2-phenylpyridine 6-(aminomethyl)-N,2,3,4-tetrahydrochromene-8-sulfonamide;(4S,5R)-1-[5-chloro-4-(cyclohexa-1,5-dien-1-ylamino)pyridin-2-yl]-3-sulfanylidene-2-azabicyclo[4.1.0]heptane-2-carboxamide (1S)-2,2,3,3a,4,5-hexahydro-[1]benzothiolo[6,5-c]chromene 2-[4-[5-(azidomethyl)cyclohexen-1-yl]phenyl]ethanamine N-(6,6a-dihydro-5aH-benzo[b][1]benzoxepin-11-yl)-4,5,7-trioxo-2-propan-2-ylidene-1,3-thiazolidine-3-carboxamide 2-[4-(3-ethoxyphenyl)piperazin-1-yl]-N-propan-2-ylacetamide [2-fluoro-3,5-bis(trifluoromethyl)phenyl]phosphane 2-[3-(5-methyltriazol-1-yl)azetidin-1-yl]pyrimidine 3-methoxy-4-(2,5,7-trimethyl-6,8-dihydropyrazolo[1,5-a][1,3]diazepine-3-carbonyl)benzonitrile N-(1,3-benzothiazol-2-ylmethyl)pyridine-4-carboxamide 2,6-diamino-3-hydroxyimino-5H-phenanthridine-7,8-dione 5-[6-[2,4-dimethyl-3-(methylideneamino)phenyl]-3-fluoropyridin-2-yl]-N-ethylpyrimidin-2-amine (2S)-2-[(4-hydroxypiperidine-1-carbonyl)amino]-3-naphthalen-2-ylpropanoic acid;hydrochloride (4aS)-8a-methyl-7-[5-(trifluoromethylsulfanyloxy)pyridine-3-carbonyl]-1,5,6,8-tetrahydro-[1,3]oxazolo[3,4-a]pyrazin-3-one 2-bromo-6-[(3E)-penta-1,3-dien-3-yl]phenol [4-(2,3,5,6-tetramethyl-1H-indole-7-carbonyl)piperazin-1-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone 4-[(Z)-[3,5-dichloro-2-(6-methylpyridin-2-yl)phenyl]methylideneamino]oxy-N-methylaniline 3-(1,2-dimethylbenzimidazol-5-yl)cyclopropane-1,1,2,2-tetracarbonitrile 3-(2,4-difluorophenyl)-1-[4-(1H-indazol-5-yloxy)cyclohexyl]pyrazolo[3,4-d]pyrimidine N-[(5-cyanopyrazin-2-yl)methyl]-3-(tetrazol-1-yl)benzamide 3-methylspiro[3,4-dihydrochromene-2,1'-cyclopentane] 3-(1H-indol-6-yl)-2-oxopropanoic acid 3-[[(2E,4Z)-5-amino-6-chlorohexa-2,4-dienoyl]amino]-N-(1H-indazol-5-yl)benzamide N-azido-2,6-dimethylaniline N-azido-5,6-dimethyl-N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyrimidin-4-amine 1-[(3,5-dichlorophenyl)methyl]-3-ethynylpyrazole 3-hydroxy-4-[(5-nitro-1,2,4-triazol-1-yl)iminomethyl]naphthalene-2-carboxylic acid N-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]benzamide N-[(2R)-4,6-dioxooxan-2-yl]-1-(3-oxocyclohexen-1-yl)benzimidazole-5-carboxamide 4-[(3,5-difluorophenyl)methyl]piperazine-1-carboxylic acid 5-bromo-2,3-difluoro-N-(4-methylsulfinylphenyl)benzamide 3-[3,4-dihydro-2H-pyran-5-ylsulfonyl(oxolan-2-ylmethyl)amino]benzamide [2-(dimethylamino)ethylamino]-phenylphosphonamidic acid N-[4-fluoro-5-(6-fluoroquinolin-4-yl)-2,3-dihydroinden-1-ylidene]hydroxylamine 5-[4-fluoro-3-(2,4,6-trimethylphenyl)-1,2-oxazol-5-yl]benzene-1,3-diol (5S)-2-[2,6-dichloro-4-[3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]anilino]-N-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxamide 3-(4-benzyl-2,5-diphenylpyrazol-3-yl)propanoate 4-[5-(3,4-dimethoxyphenyl)pyridine-2-carbonyl]morpholine-3-carboxylic acid (2E,3E)-6-(5-methylpyridin-3-yl)sulfanyl-3-propylidenedeca-1,4,7,9-tetraen-5-amine 2-[3,5-bis(trifluoromethyl)phenyl]-N-(4-ethylpiperidin-1-yl)acetamide;N',N'-dimethylethane-1,2-diamine;ethene N-[4-[2-(butylamino)ethylsulfanyl]phenyl]acetamide 5-fluoro-2,3-dimethylquinoline-6-carboxylic acid 5-tert-butyl-N'-methylsulfanyl-2,3,4,9-tetrahydro-1H-carbazole-3-carbohydrazide 4-amino-6,8-dichloroquinoline-5,7-disulfonic acid 6-[[5-chloro-2-(3,4-dimethylphenyl)-1H-indol-3-yl]methyl]-2-propan-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-methyl-2-naphthalen-1-ylsulfanylpropanenitrile (2R,3S)-2-(1,5-dimethylpyrazol-4-yl)oxane-3-carboxylic acid N-(2,6-dioxopiperidin-3-yl)-1-fluoro-4H-indeno[1,2-c]pyrazole-3-carboxamide 3-azido-5-bromo-1H-pyrrolo[2,3-b]pyridine 2-[4-amino-6-(methylamino)pyrimidine-5-carboximidoyl]phenol 2-fluoro-6-phenylmethoxybenzenecarboximidate 2,4-dichloro-5-(1,1,1,3,3,3-hexafluoropropan-2-ylsulfamoyl)benzoic acid 3-[4-(4,4-dimethylpiperidin-1-yl)-5-(4-methoxyphenyl)-2-nitrophenoxy]propan-1-amine 2-methylsulfonyloxy-6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazole-3-carboxylic acid 1-(4,5-dimethoxy-2-nitrophenyl)triazole 4-[6-[5-[2-(diethylamino)ethyl]-3,6-dihydro-2H-pyridine-1-carbonyl]naphthalen-2-yl]benzonitrile 3-(4-bromobutoxy)-7,8-dimethyl-2H-1,6-naphthyridine 4-(5,6-dihydroimidazo[2,1-b][1,3]thiazol-3-yl)-N,6-dimethylpyrimidin-2-amine 3-amino-1-methoxy-6,8,11b-trimethyl-4,5,6a,7,8b,9,10,12,12a-octahydronaphtho[2,3-g]quinoline-7,11-diol 2-chloro-N-(4,5-dimethyl-1,3-thiazol-2-yl)quinoline-6-carboxamide (4aS,7S,7aR)-N-[2-(dimethylamino)ethyl]-6-pyrimidin-5-yl-3,4a,5,7,7a-hexahydro-2H-pyrrolo[3,4-b][1,4]oxazine-4-carboxamide;2,2,2-trifluoroacetic acid 2,3-bis(4-chlorophenyl)-4-cyclopentyl-1H-pyrrole 2-[1,3-benzoxazol-2-yl(ethyl)amino]-4-fluorophenol 2-[1,4-bis(2-methylbutan-2-yl)cyclohexa-2,4-dien-1-yl]-4-fluorophenol 6-butyl-N,3-diphenyldibenzothiophen-4-amine 4-(1,3-benzothiazol-2-yl)benzene-1,3-diamine 6-(2,5-dichlorophenyl)sulfanyl-1H-benzimidazole 2-[4,7-di(cyclobutadienyl)heptanoylamino]benzoic acid 4-chloro-3-ethyl-N,6-dimethylquinolin-2-amine;propane 4-[5-(2,6-dichlorophenyl)sulfanylpyrazin-2-yl]morpholine 5-chloro-N-methylsulfanyl-2,3-dihydro-1H-indene-2-carboxamide;fluorocyclopentane N-[(2R)-4-aminobutan-2-yl]-3-phenylmethoxybenzamide 4-azido-1,2,3,5-tetramethyl-6-(4-phenylmethoxyphenoxy)cyclohexa-2,4-diene-1-carbonitrile 5-(aminomethyl)-2-[3-(cyclopropylmethoxy)phenyl]-N-[(4-ethylsulfonylphenyl)methyl]triazole-4-carboxamide;hydrochloride 2-[1-(6,7-dihydro-5H-cyclopenta[d]pyrimidine-4-carbonyl)pyrrolidin-3-yl]-3H-quinazolin-4-one 3-[1,2-bis(4-methylphenyl)ethenyl]-5-(4-chlorophenyl)sulfonylaniline 2-[4-azido-5-(difluoromethyl)pyrazol-1-yl]pyridine 5-[4-(2-hydroxyethylcarbamoyl)-6-(trifluoromethoxy)cyclohexa-1,3-dien-1-yl]oxypyridine-3-carboxylic acid 2-(3,4-dimethoxyphenyl)-1H-[1]benzothiolo[2,3-d]imidazole (2S,4R)-4-hydroxy-1-methylsulfonyl-N-[4-(trifluoromethyl)phenyl]pyrrolidine-2-carboxamide 5-[3-[(2-methylpyridin-4-yl)amino]-1H-pyrazol-5-yl]oxolan-2-one 1-benzyl-N-[2,3-dihydroxy-4-(trifluoromethoxy)phenyl]pyrrolidine-2-carboxamide 1-cyclohexyl-4,5-dimethoxyindazole 2-[(1Z,3E)-4,5-difluorohexa-1,3,5-trienyl]sulfanyl-3-pyridin-3-ylquinoxaline 1-(5,7-dimethylpyrrolo[2,3-d]pyrimidin-4-yl)-6-methoxyspiro[2H-indole-3,2'-pyrrolidine] (3S,4R)-1-[2-(6-fluoropyridin-3-yl)ethyl]-4-propan-2-ylpiperidine-3-carboxylic acid 5-chloro-2-fluoro-4-[(2Z,3E)-2-ethylidene-1-methylsulfanylhexa-3,5-dienoxy]benzoic acid 2-[7-(3,4-dichlorophenyl)-5-methyl-2-(trifluoromethyl)-1H-imidazo[4,5-b]pyridin-6-yl]-2-oxoacetaldehyde;N'-propan-2-ylidenemethanimidamide 2-[4-(methanesulfonamido)phenyl]-N-quinolin-8-ylbenzamide (3R,4R)-N-[6-(3-fluorophenyl)pyridazin-3-yl]-1-methylsulfonylpiperidine-4-carboxamide 2-[[4-[2-(trifluoromethyl)phenyl]piperazine-1-carbonyl]amino]-3,4-dihydro-1H-isoquinoline-6-carboxamide;hydrochloride 2-[7-methoxy-8-(4-oxocyclohexyl)oxychromen-2-ylidene]propanedinitrile 2-(5-tert-butyl-1H-imidazole-4-carbonyl)-N,N-diethylmorpholine-4-carboxamide N-[(2S)-1-aminopropan-2-yl]-6,7-difluoroquinoxaline-5-carboxamide (3R)-4,4,5-trihydroxy-3-[[2-methylpropanoyl(phenylmethoxycarbonyl)amino]methyl]pentanoic acid N-[4-(4-acetylpiperazine-1-carbonyl)-3-chlorophenyl]-2,6-difluorobenzamide 2-[4-(cyclopropylmethoxy)phenyl]-N-[3-ethynyl-5-fluoro-4-(1H-pyrazol-4-yl)phenyl]propanethioamide 1-(2-chloroethyl)-7-methylsulfonylquinolin-4-one 1-(5-azidopyridin-3-yl)piperidin-4-ol 2-tert-butyl-4-methylcyclohepta[d]triazole 3-[(2E)-4-oxo-2-[(Z)-(3,5,8-trihydroxynaphthalen-1-yl)methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]propanoic acid N-(1,3-dimethylpyrazolo[3,4-b]pyridin-5-yl)-2-fluoro-5-nitrobenzamide 2-cyclopropyloxy-1,3-difluoro-5-(4-iodophenyl)benzene 5-(4-fluorophenyl)-N-[1-(methoxymethyl)cyclopentyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide;hydrochloride 6-(1,2-difluoropentan-3-yl)-5H-pyrrolo[3,4-b]pyridine N-[2-(2,5-difluorophenyl)-3H-benzimidazol-5-yl]furan-2-carboxamide 2-hydroxy-N,3-dimethylbutanamide;5-[(Z)-(4-oxo-1-phenylpyridazin-6-ylidene)methyl]thiophene-3-carbonitrile (3Z)-4-amino-3-[2-(1H-benzimidazol-5-yloxy)ethylidene]azete-2-thione [4-hydroxy-3,5-di(propan-2-yl)phenyl]iminourea 2-methyl-1,3-thiazol-4-ol;N'-[6-(1H-pyrazole-5-carbonyl)isoquinolin-3-yl]piperidine-1-carboximidamide N-[[(3R,4S)-1-[2-[2-(aminomethyl)piperidin-1-yl]-2-oxoethoxy]-4-phenylpyrrolidin-3-yl]methyl]acetamide;dihydrochloride 2-[(4,5-dimethyl-1H-pyrazol-3-yl)amino]-8-[(4-ethoxyphenyl)methyl]pyrido[2,3-d]pyrimidin-7-one 2-[(4-fluorophenyl)methyl]pentanal (E)-3-[4-[2,6-difluoro-4-[[[hydroxy(phenyl)methyl]-methoxycarbonylamino]methyl]phenoxy]thieno[3,2-d]pyrimidin-7-yl]prop-1-enolate 4-[(4R)-5,8-dichloro-3-cyclohexyl-1,2,3,4-tetrahydroquinolin-4-yl]morpholine (2-chlorophenyl)-[3-[5-[6-(1,1-difluoroethoxy)pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-carbonyl]-2-(methoxymethoxy)-5-methylsulfonylphenyl]carbamic acid 7-bromo-1,2,3-trimethyl-5H-pyrazolo[4,3-c]quinolin-4-one;ethane 3-(cyclohexen-1-yl)-4,5-dihydroxybenzaldehyde (E)-1,3-bis[2-(ethylaminooxymethyl)phenyl]prop-2-en-1-one (5E)-2-[4-(dimethylamino)phenyl]imino-5-[[1-(3,4,5-trimethoxyphenyl)pyrrol-2-yl]methylidene]-1,3-thiazolidin-4-one N-[4-[(7R)-5-[4-chloro-3-(trifluoromethyl)phenyl]-7-methyl-6-oxo-8H-imidazo[1,2-b]pyridazin-7-yl]pyridin-2-yl]acetamide 1-[5-chloro-4-(trifluoromethyl)pyrimidin-2-yl]indole 1,6-dimethyl-3-[(E)-2-(4-phenoxyphenyl)ethenyl]pyrazolo[3,4-b]pyridine 3-[(4Z,5E)-5-ethylidene-4-prop-2-enylidenefuran-2-yl]propanoic acid 1-ethyl-2,5-difluoro-4-(2-methoxyethynyl)benzene 2-[1-(4-methoxyphenyl)cyclobutyl]ethanamine 6-(trifluoromethyl)-2-[4-[2-(trifluoromethoxy)phenyl]piperazine-1-carbonyl]-3,5-dihydropyrano[3,2-d]pyrimidin-4-one 3-azido-N',2-dihydroxybenzenecarboximidamide 7-[(3,4-dichlorophenyl)methyl]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 2-[(4-acetamidobenzoyl)amino]-3,4-dimethoxybenzamide 1-[4-(1-cyclopropylcyclobutanecarbonyl)piperazin-1-yl]-2-phenylethanone (NZ)-4-chloro-2,5-difluoro-N-[(5R,6S)-8-thiatricyclo[7.3.0.03,5]dodeca-1(9),10-dien-12-ylidene]benzenesulfonamide 4-(3-aminophenyl)sulfanyl-N'-hydroxypyridine-2-carboximidamide N-(1H-benzimidazol-2-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 4-[3-methylbut-2-enyl(octyl)amino]benzenesulfonamide 2-[4-(3,4-dichlorobenzoyl)piperazin-1-yl]-N-(3,5-dimethylphenyl)acetamide 5-[2-(4,4-difluorocyclohexyl)ethyl]-N-methoxyimidazo[1,5-a]pyridine-6-carboxamide 3-[2-(4-propan-2-ylphenoxy)phenyl]oxirane-2,2-dicarbonitrile [3-(2,4-difluorophenyl)azetidin-1-yl]-(3-methoxyquinoxalin-6-yl)methanone ethane;2-[(5-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)sulfinyl]benzonitrile 1-(5-ethoxypyridine-3-carbonyl)-7-methylazecan-4-one 5-[3,6-dioxo-2-(1H-pyrrol-2-ylmethylidene)-1-benzofuran-5-yl]pyridine-2-carboxylic acid 7-methoxy-2-(4-prop-1-en-2-yl-3,5-dihydro-2H-pyrazin-6-yl)quinoline (6R,9S)-2,3,4,5,6-pentadeuterio-6-[7-[[2-fluoro-4-(morpholin-4-ylmethyl)phenyl]methoxy]-3,4-dihydro-1H-isochromen-5-yl]-4,8-dimethyl-7-oxa-10-azatricyclo[6.4.0.02,6]dodeca-1(12),9,11-triene 2-(1,5-dimethyl-4H-pyridin-3-yl)-5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-6-hydroxy-3H-isoindol-1-one 5-(2,3,4a,5,6,7,8,8a-octahydroquinoxaline-1-carbonyl)-N-methylpyridine-3-carboxamide 2-(4-ethoxyphenyl)-3H-thieno[3,2-d]pyrimidin-4-one 3-[[1,4-dimethyl-5-(trifluoromethoxy)indole-2-carbonyl]amino]benzoic acid [3-azidooxy-1,2-bis(phenylmethoxy)propan-2-yl]benzene 6-[[5-(4,6-dimorpholin-4-ylpyrimidin-2-yl)imidazol-1-yl]methyl]quinoline 5-bromo-2-(1H-pyrrol-3-ylmethylidene)-3,4-dihydronaphthalen-1-one [2-[2,4-dihydroxy-3-(4-methoxyphenyl)-6-pentylbenzoyl]oxyacetyl]azanium 1-(2,4-dichlorophenyl)-3-[1-hydroxy-3-methyl-6-oxo-7-(trifluoromethoxy)pyridazin-4-yl]urea [2-[(4,5-difluoro-1H-benzimidazol-2-yl)methyl]pyrazolo[3,4-c]pyridin-6-yl]-(6-fluorospiro[3.3]heptan-2-yl)carbamic acid N-[2,3-dioxo-1-(propylcarbamoyl)-4H-quinoxalin-6-yl]acetamide (2S)-2-amino-N'-[(3Z,5E,7Z)-cycloocta-1,3,5,7-tetraen-1-yl]-N-[(E)-3-pyridin-4-ylprop-2-enylideneamino]butanediamide 4-[4,6-bis(3-methoxyphenyl)-1,3,5-triazin-2-yl]morpholine [(2S,5R)-5-hydroxy-2-methylpiperidin-1-yl]-(1H-indol-3-yl)methanone 2-(3,4,5-trimethoxyphenyl)cyclohexa-1,3-diene N-[5-tert-butyl-2-methoxy-4-(trifluoromethyl)phenyl]pyridine-3-carboxamide (3S)-1'-benzylspiro[1,2-dihydroindole-3,4'-piperidine] (2R)-2-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-1-phenylpropan-1-one 4-[2-chloro-5-(3,6-dihydro-2H-1,4-oxazin-5-yl)pyridine-3-carbonyl]benzonitrile 4-chloro-2,6-difluoro-N-(4-nitrobutyl)aniline 2-(3,4-dimethoxyphenyl)-1,1-dioxo-N-(4-propanoylpyridin-3-yl)-1,2,6-thiadiazine-5-carboxamide N-azido-2,3-dihydro-1,4-benzodioxin-5-amine 2-[3,5-dichloro-4-[3-(trifluoromethyl)phenyl]sulfanylphenyl]-6-[[1-(hydroxyamino)-1,3-thiazol-5-yl]methoxy]oxane-2,4-diol N-[3,5-bis(4-methylphenyl)pyrazol-1-yl]benzamide 1-amino-3-[2-(bromomethyl)phenoxy]propan-2-ol 4-(1H-benzimidazol-2-yl)-N-[(3R,5S)-5-methylpyrrolidin-3-yl]piperidine-1-carboxamide [3-[3-[5,6-bis(4-methylphenyl)pyrazin-2-yl]oxyphenoxy]phenyl]hydrazine N-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-formylcyclopropane-1-carboxamide 4-chloro-2-[5-(dimethylamino)-3-ethoxy-1,4-benzothiazepine-7-carbonyl]cyclohexa-1,3-diene-1-carbonitrile (5Z)-5-[(2,5-dichloro-3-methylsulfonylphenyl)methylidene]imidazolidine-2,4-dione 3-[(5,6-dichloropyridine-2-carbonyl)amino]azetidine-1-carboxylic acid 1-ethyl-3-[6-(2,3,4-trifluorophenyl)quinolin-8-yl]urea 2-[(3S)-1-[2-oxo-6-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyrimidin-4-yl]pyrrolidin-3-yl]acetic acid 1-[(3R)-3,4-dimethylpiperazin-1-yl]-2-(2-ethylimidazo[1,2-a]pyridin-6-yl)ethanone 5-bromo-1,3-dichloro-2-[3-fluoro-4-(trifluoromethoxy)phenyl]benzene 1-(4-amino-3,5-dimethoxyphenyl)-2H-pyrazine-6-carboxylic acid 1-(1,3-benzodioxol-5-ylmethyl)-8-pyridin-4-yloxy-2,4-dihydro-1H-pyrazino[1,2-b]indazole (E)-N'-[2-methyl-4,6-di(propan-2-yl)phenyl]but-1-ene-1,4-diamine 6-hydroxysulfanyl-3-methoxy-1,2,4,5-tetrahydroazepino[3,4-b]indole 4-chloro-N-(2,6-dimethylphenyl)-3-[5-oxo-7-[[(2R)-oxolan-2-yl]methoxy]thieno[3,2-b]pyran-2-yl]benzenesulfonamide (1S,2S)-N'-[2-[(4-cyclopropyloxyphenyl)methylamino]ethyl]-2,3-dihydro-1H-indene-1-carboximidamide 1-(2-chloro-3,4-dimethoxyphenyl)-N-(4,5-dichlorocyclohepta-1,4,6-trien-1-yl)sulfonylimidazole-4-carboxamide 4-cyclohepta-1,3-dien-1-yloxypyridine (4E,5Z)-3-methyl-1-(pyridine-4-carbonyl)hepta-4,6-dien-2-one ethane;5-methyl-2,3,4,6-tetrahydro-1H-1,5-benzodiazocine (E)-3-[4-hydroxy-5-(indol-6-ylidenemethyl)-2-sulfanylidene-1,3-thiazol-3-yl]prop-2-enoic acid N-[3-[6-(1,2,4-triazol-1-yl)pyridin-3-yl]propyl]isoquinoline-7-carboxamide (3R)-N'-[(4-chlorophenyl)methyl]-3-methoxy-2,6-dihydroazepino[4,5-b]indole-1-carboximidamide (E)-3-[4-chloro-2-fluoro-5-methoxy-3-(trifluoromethyl)phenyl]-2-sulfanylprop-2-enoic acid 1-(3-bromophenyl)-N',N'-dimethylbutane-1,4-diamine 3-[4-(1,2-dihydropyridine-5-carboximidoyl)pyridin-2-yl]-N-methylbenzenecarboximidate 1-[3,4-bis(ethenyl)-6-hydroxycyclohexa-2,4-dien-1-ylidene]-5-phenylsulfanylindene-2-carboxamide (2S)-2-[5-azido-4-[3-bromo-5-methyl-4-(trifluoromethoxy)phenyl]-1H-imidazol-2-yl]pyrrolidine (E)-3,4-dihydroxybut-2-enoic acid;1-[[5-methoxy-7-(2-methylpyridin-4-yl)-1-benzofuran-2-yl]methyl]pyrrolidine 2-amino-3-azidooxy-6-[(4-chlorophenyl)methyl]benzamide 5-[2-(4,6-dioxo-1H-pyrimidin-3-yl)acetyl]benzene-1,3-disulfonic acid N-(1,2-benzoxazol-3-ylmethyl)-7-fluoroquinoline-3-carboxamide 2-methoxy-4-[3-(1H-pyrrol-2-yl)pyrazole-1-carbonyl]benzoic acid 6-(1,3-benzodioxol-5-ylmethyl)-3-[1-(2-fluorophenyl)pyrazol-4-yl]-7H-imidazo[1,2-b][1,2,4]triazin-8-one 1-(3,3a,4,5,6,7a-hexahydro-2H-indol-1-yl)-2-[[6-methoxy-2-(4-piperazin-1-ylanilino)pyrimidin-4-yl]amino]ethanone N'-(2,4-difluorobenzenecarboximidoyl)-3,3-dimethylbutanimidamide 1-[3-(4-propanoylphenyl)phenyl]ethanethione (Z,2S)-1-(2,5-dimethylphenyl)-2-(4-fluorophenyl)pent-3-en-1-one;1-propoxypentan-1-ol 5-chloro-4-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-ylmethoxy)pyridin-2-amine N-[4,6-bis(ethenyl)-5-methanimidoylpyrimidin-2-yl]-N-phenylhydroxylamine N-(3-bromopropyl)-N-(2,4-difluorophenyl)benzamide 4-chloro-2-[[3-[(4-ethylphenyl)carbamoyl]-5-methoxyphenyl]-phenylmethylidene]piperidine-1-carboxylate 5-[3-methyl-4-(2,2,2-trifluoroethoxy)phenyl]imidazolidine-2,4-dione 2-[1,3-benzodioxol-5-ylmethyl(cyclopropanecarbonyl)amino]-N-(4,6-dimethoxypyrimidin-2-yl)acetamide 3-[(E)-2-(4,5-dimethoxycyclohepta-1,3,6-trien-1-yl)ethenyl]-1H-pyridazin-6-one N-[4-(azepan-1-ylmethyl)phenyl]-4-oxo-2,3-dihydrochromene-8-carboxamide [3-(4,5-dihydropyrazolo[1,5-a]pyrimidine-7-carbonylamino)phenyl]boronic acid (7S)-N-benzyl-9-[2-(diethylamino)ethoxy]-5,7-bis(phenylmethoxy)-8-(trifluoromethyl)-6H-pyrimido[4,5-b][1,3]oxazin-2-amine [(4R,5S)-3-hydroxy-8-thiatricyclo[12.4.0.02,7]octadeca-1(18),2(7),3,5,14,16-hexaen-12-yl]-(2-phenylphenyl)methanone 4-[4-(2-amino-5-bromophenyl)butan-2-yloxy]-3-methylbutanoate 2-(3,5-dichloropyridin-4-yl)benzaldehyde 5-azidosulfanyl-2-methoxypyrimidine 3-azido-5-(2,6-dimethylphenyl)-1H-pyridine-4-thione 4-(4,5-dihydrobenzo[g]quinoline-3-carbonylamino)thiophene-2-carboxylic acid 6-[4-(2,6-difluorophenyl)-5-oxotetrazol-1-yl]hexanamide 1-[4-[[(3S)-6,7-dimethoxy-2,3-dihydro-1-benzofuran-3-yl]amino]piperidin-1-yl]ethanone N-[1-(cyclopentanecarbonyl)azetidin-3-yl]-2-methoxy-5-(1,2,4-triazol-1-yl)benzamide (3S,4R)-N'-[4-cyano-2-(trifluoromethyl)phenyl]-1-(4-hydroxybutanoyl)-N-propylpyrrolidine-3-carbohydrazide 2-[6,6-dimethyl-3-(trifluoromethyl)cyclohexa-1,4-dien-1-yl]-N-(7H-purin-6-yl)acetamide 2-[(5E)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-yl]-N-phenylacetamide 2-[4-[[6,7-dimethoxy-1-[4-(trifluoromethyl)phenyl]sulfonylbenzimidazol-2-yl]methoxymethyl]cyclohexa-2,4-dien-1-yl]ethanamine 6-[2-[3-(4,5-dihydro-1H-imidazol-2-ylamino)anilino]pyrimidin-4-yl]-2,3-dihydroisoindol-1-one 3-(2,4-dichlorophenyl)-1-[1-(1H-imidazol-5-ylmethoxy)isoquinolin-6-yl]urea (3,5-dimethylphenoxy)-(4-hydroxy-2-propanoyloxyphenyl)borinic acid 4-(5,6-dihydroxypyrimidine-4-carbonyl)oxybenzoic acid 4-(2,5-dihydroxyphenyl)-1,3-oxazole-5-carboxylic acid 2-tert-butyl-5-(4,5-dihydro-1H-imidazol-2-yl)quinolin-8-ol 2-[4,6-bis(2-methylbutan-2-yl)pyrimidin-5-yl]ethanesulfonate [(2Z,4Z)-hepta-2,4-dienyl]-[1-(4-methoxyphenyl)cyclopropyl]sulfanium 4-[(5S)-1-amino-2,3-dimethyl-6-oxo-5-phenylpiperidin-2-yl]-N-tert-butylbenzenesulfonamide 3-[4-(1,2,5-oxadiazol-3-yl)piperidin-1-yl]cyclobutane-1-carbonitrile 1-(2,4-difluorophenyl)piperazine;1-[4-methyl-5-(oxolan-3-yloxymethyl)-1,3-thiazol-2-yl]ethanone (3-iodophenyl)methanesulfinamide 4-amino-N'-(aminomethyl)benzimidazole-1-carboximidamide 5-[4-(4-fluorophenoxy)phenyl]-3-(1-methylpyrazol-3-yl)pyrazine 2-[3,5-bis(trifluoromethyl)phenyl]-4,6-dipyridin-3-yl-1,3,5-triazine 4-azido-1,3-dibutoxy-5-methylbenzene 1-azido-3-propan-2-yloxynaphthalene 1-[4-fluoro-3-(trifluoromethyl)phenyl]-N,N,6-trimethylpyrazolo[3,4-d]pyrimidin-4-amine 2-[4-[4-(cyclopropanecarbonylamino)phenoxy]phenyl]acetate 4-[2-chloro-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalene-1-carbonyl)phenyl]benzoic acid 4-[(6E)-8,11-dihydro-5H-imidazo[1,2-b]thiocin-9-yl]-2,3,3a,4,5,6,7,7a-octahydro-1H-isoindole N-[6-[2-(4-cyanoanilino)pyrimidin-4-yl]-1H-benzimidazol-2-yl]-3,5-difluoropyridine-4-carboxamide 3-[4-(2,6-dimethylpyridin-3-yl)phenyl]-N,2-dihydroxy-4H-chromene-8-carboxamide (4-chlorophenyl)methanol;3,5-dihydroxynaphthalene-2,7-disulfonic acid 4-(4,5-dimethoxy-2-sulfanylphenyl)benzene-1,3-disulfonic acid 3-[1-azido-3,4-dioxo-2-(trifluoromethyl)thieno[3,4-d]pyridazin-7-yl]benzonitrile N-[[5-(3,4-difluorophenyl)-1H-pyrazol-4-yl]methylideneamino]-6-morpholin-4-ylpyridine-2-carboxamide N-[4-(2,5-dichlorophenyl)-3-(1H-imidazole-5-carbonylamino)phenyl]-7-phenyl-6-azaspiro[3.4]octane-6-carboxamide N-[3-amino-6-(5-ethylsulfonylpyridin-2-yl)pyrazin-2-yl]-1H-pyrrole-3-carboxamide 6-chloro-N-[2-(difluoromethoxy)-5-morpholin-4-ylphenyl]imidazo[1,2-b]pyridazine-3-carboxamide 2-(1,3-benzodioxol-5-yl)-N'-hydroxypyrimidine-4-carboximidamide N-butyl-4,5-dimethyl-N-(1,2,3,6-tetrahydropyridin-4-yl)thiophene-2-carboxamide 7-[(4R)-3,4-dihydro-2H-chromene-4-carbonyl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-one 1,4-bis[(3,4-difluorophenyl)sulfanyl]-2-ethoxybenzene 2-[(Z)-[[1,3-dimethyl-5-[(1E,3Z)-penta-1,3-dienyl]benzimidazol-1-ium-2-yl]hydrazinylidene]methyl]-4-nitrophenol 3-[(4-benzylpiperazin-1-yl)methyl]-2H-isoquinolin-1-one 2-(1,3-benzodioxol-5-yl)-N-[4-fluoro-5-[5-(piperidine-1-carbonyl)pyridin-3-yl]oxy-2-(propanoylamino)phenyl]-3H-benzimidazole-5-carboxamide 2-[3-(dipropylamino)propyl]-5,6-bis(4-fluorophenyl)isoindole-1,3-dione 2-[4,6-dichloro-1-(trifluoromethyl)cyclohexa-2,4-dien-1-yl]acetic acid (E)-1,2,3-trimethyl-4-[1-methyl-4-[(5-phenylpyridin-3-yl)methyl]pyrazol-3-yl]pent-1-en-3-amine 2-[4-(difluoromethoxy)phenyl]-1-[3,5-dimethyl-4-(pyridin-3-ylmethylamino)phenyl]ethanone N-(5-azidooxy-2,4-dichlorophenyl)benzamide (2S)-1-azido-3,4-dichloro-2-[3-fluoro-4-methyl-5-[3-(trifluoromethylsulfanylamino)phenoxy]phenyl]butan-2-ol 5-(2,3-dihydro-1H-indene-4-carbonyl)-N-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide N-[1-(4-chlorophenyl)-2,5-dimethylpyrazol-3-yl]-2-ethoxyethanimidate (7-chloro-1,3-dimethylindol-5-yl)-[4-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperazin-1-yl]methanone 6-[(2,5-dimethoxyphenyl)carbamoyl]-1H-indole-4-carboxylic acid 7-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-2-methyl-3H-thieno[3,2-d]pyrimidin-4-one 4-(6,7-dimethoxyquinolin-3-yl)piperazine-1-carboxylate (5-bromopyridin-3-yl)-[5-fluoro-2,4-dihydroxy-6-[6-(triazol-1-ylmethyl)pyrrolo[3,2-b]pyridin-1-yl]phenyl]methanone N-[(2R,3S)-2-azido-4-bromobutyl]benzenesulfonamide N-[4-(2,6-dimethoxyphenyl)-5-pyridin-3-ylsulfanyl-1,2,4-triazol-3-yl]-1H-pyrrole-2-carboxamide 3-(5,6-dihydroquinolin-4-yl)-2H-1,3-benzothiazole N-[(2,4-dimethylphenyl)carbamothioyl]benzamide 1-[3,5-bis(4-fluorophenyl)phenyl]-2,3-dihydro-1H-indene 4-bromospiro[1,2-dihydroindene-3,5'-imidazolidine]-2'-one 2-[6-(9H-fluoren-1-yl)hexoxycarbonyl]benzoic acid 3-[[5,6-dichloro-1-(4-fluorophenyl)benzimidazol-2-yl]methoxy]-N-hydroxycyclobutane-1-carboxamide N-[4,5-diamino-1-(benzylamino)-3-butylnaphthalen-2-yl]acetamide (3S)-1-[6-ethyl-4-methylidene-2-[2-(2,3,4,5-tetrafluorophenyl)-3H-benzimidazol-5-yl]pyrido[2,3-d]pyrimidin-3-yl]-N,N',3-trimethylbutane-1,3-diamine (4E)-N,N-dimethyl-5-phenyl-2-propan-2-ylidenehexa-3,5-dienamide 1-[4-[5-[(7S)-4,7-dimethylocta-2,6-dienoxy]pentoxy]phenyl]ethanone 2-(4-cyclobutylphenyl)quinoline N'-[2-methyl-5-(1H-pyrrolo[2,3-b]pyridine-4-carbonyl)phenyl]-N-phenyloxamide 6-chloro-4-(4-cyclopropylphenyl)quinoline [4-hydroxy-3-[4-(2-phenylethenyl)phenoxy]-1H-indol-7-yl]-phenylmethanone N'-hydroxy-2-methyl-4,6-bis(3-nitrophenyl)benzenecarboximidamide 5-bromo-2-[[4-(methylamino)phenyl]diazenyl]phenol (2S)-5-amino-2,4-dimethyl-6-phenylhexanoic acid 1-(3,5-dimethylphenyl)sulfonyl-N-[(2-ethoxypyridin-4-yl)methyl]pyrrolidine-2-carboxamide 3,6-dimethoxy-9-(4-oxooxan-2-yl)fluoren-1-ol 4-(3,5-dichlorophenyl)-3-methyl-1,2-oxazol-5-amine 2-tert-butyl-6,7-dihydroxy-3H-benzo[g]quinazolin-4-one 2-[3,4-diamino-5-(methoxymethyl)phenyl]ethanol 2-amino-5,6-dimethylcyclohexa-1,3-diene;5-ethynyl-13,20-bis(hydroxyimino)-8-oxa-15,16,18,20,22-pentazatricyclo[16.4.0.02,7]docosa-1(18),2,4,7,9,11,19-heptaen-10-one (2R)-3-[4-[7-benzyl-5-(methoxymethyl)pyrrolo[2,3-d]pyrimidin-4-yl]pyrazol-1-yl]propane-1,2-diol 2-benzylsulfanyl-4,5,6,7-tetrahydro-1H-indene;N-[(1E)-1,3-diaminobuta-1,3-dienyl]formamide N-[2,2-dimethyl-1-(2-methylphenyl)propyl]acetamide 4-[2-[(E)-2-nitroethenyl]imidazol-1-yl]benzonitrile 3-[(7S,8aS)-1-[2-(4-hydroxyphenyl)acetyl]-7-methyl-3,4,6,7,8,8a-hexahydro-2H-pyrrolo[1,2-a]pyrazin-3-yl]propanoic acid 4-chloro-5-[(3,4-difluorophenyl)methylamino]dithiol-3-one 2-[(3R)-1-acetylpyrrolidin-3-yl]-6-phenylpyridazin-3-one 4-hydroxy-7,10-dimethylanthracene-9,10-dione N-benzyl-2-[[[(E,3S)-6-[ethoxycarbonyl(methyl)amino]-3-methylhept-4-en-2-yl]amino]methyl]-1H-benzimidazole-4-carboxamide (2S,4R)-1-[4-cyano-3-(trifluoromethyl)phenyl]-N-cyclopropyl-4-(1H-imidazol-5-ylsulfonylamino)pyrrolidine-2-carboxamide 2-(1-benzylsulfonylpiperidin-4-yl)-5-(cyclopropanecarbonylamino)benzoic acid;2,2,2-trifluoroacetic acid (2R,3S)-N-[5-(cyclohexylmethoxy)pyridin-2-yl]-2-methylpiperidine-3-carboxamide 2-[4-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-ylmethoxy)phenyl]-N-hydroxyacetamide 6-chloro-2,5-dimethylindazole 2-[(4S)-4-[3,5-bis(trifluoromethyl)phenyl]-2,4-dihydroimidazo[1,5-a]indol-4-yl]acetamide N-(4-bromophenyl)-2,6-dimethyl-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]aniline 3-(4-chlorophenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidine 2-[(1R)-1-[5-chloro-3-[[3,4-difluoro-2-(trifluoromethyl)phenyl]methylamino]pyridine-4-carbonyl]-4-cyclopropylpiperidin-4-yl]acetic acid 5-[3-(1H-indol-4-yl)-2,2-dimethylpropanoyl]-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 3-fluoro-2-(4-methoxyphenyl)pyridine 2-methoxy-1-[6-(4-phenylbenzoyl)-9H-xanthen-3-yl]ethanone N-[2-fluoro-4-methyl-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-3-sulfanylidene-6-(trifluoromethyl)-1H-isoindole-2-carboxamide 1-[2,3-diamino-4-(3-methoxypropyl)phenyl]ethanone 6-[2-ethoxy-4-(4-hydroxyphenyl)phenyl]-4,8-dimethyl-3,7-dihydropyrimido[5,4-e][1,4]oxazin-2-one 4-[2-azido-5-(methylamino)phenyl]butanal N-(7-fluoro-4-oxo-2,3-dihydrochromen-6-yl)-1-hydroxy-N',2,2,6,6-pentamethylpiperidine-4-carboximidamide 6-[4-[(4,5-dichloropyridin-2-yl)carbamoyl]phenoxy]pyridine-3-carboxamide;ethane 2-[azido(phenyl)methyl]-1,3,5-trifluorobenzene 3-[2,5-difluoro-4-(propylsulfanylamino)phenyl]-7-methoxy-1H-quinoxalin-2-one 2-(3-azidopropyl)-6-chloro-5,7,8-trimethoxynaphthalene-1,4-dione 1-azidooxy-2,3,4,5,6-pentafluorobenzene (3S,4R)-1-[1-(2-methoxyacetyl)piperidin-4-yl]-N-propan-2-yl-4-pyrazol-1-ylpyrrolidine-3-carboxamide 3-[6-oxo-7-(phenylmethoxymethyl)-1H-purin-8-yl]benzonitrile N-[(1S)-2-[6-(2,3-dichlorophenyl)spiro[4H-1,3-benzodioxine-2,4'-piperidine]-1'-carbonyl]cyclohexyl]-5-methoxythiophene-2-sulfonamide 2-(1H-benzimidazole-4-carbonyl)-4-[(4-methylphenyl)diazenyl]naphthalene-1,3-disulfonic acid 4-[(5S)-2,3-dimethoxypyrrolidine-1-carbonyl]-6-ethyl-3H-1,3-benzoxazol-2-one N'-[3,5-diethyl-2-(hydroxymethyl)phenyl]methanimidamide 3-(4-phenoxyphenyl)cyclohexan-1-ol N-[5-(3,4-dichlorophenyl)sulfonyl-1H-indazol-3-yl]-2-(2,4,6-trifluorophenyl)acetamide [4-[4-(2,3-dichlorophenyl)piperazin-1-yl]oxan-4-yl]methanamine 6-amino-9-[(3R)-1-[2-[4-(5-azidothiophen-2-yl)phenyl]ethyl]piperidin-3-yl]purine-8-carboxamide 5-bromo-N-[4-chloro-2-(1,3-dioxan-2-yl)phenyl]-6-fluoro-N'-hydroxypyridine-3-carboximidamide [(3S)-4-(7,8-dichloroquinoline-2-carbonyl)-3-methylpiperazin-1-yl]-(1-cyclopentylpiperidin-4-yl)methanone N-[1,2-diamino-3-(2-methylphenyl)propylidene]-6-methoxypyridine-3-carboxamide 2-[4-(3,5-dimethylbenzoyl)piperazin-1-yl]-6,7-dihydrothieno[3,2-d]pyrimidine-4-carboxylic acid 3-fluoro-2-[[1-(2,4,6-trimethylphenyl)sulfonylpiperidin-3-yl]methoxy]pyridine 3-[2-chloro-4-(trifluoromethyl)phenyl]-5,6-diethyl-1H-pyrimidine-2,4-dione 4-(4,6-dimethylpyrimidine-2-carbonyl)-3,5-dihydro-1H-imidazo[1,5-a]quinazolin-9-one 3-[4-(4-chlorophenyl)piperazine-1-carbonyl]-5,7-dimethyl-2H-pyrazolo[4,3-c]pyridine-6-carboxylic acid (2R,3S)-N-[[1-(2,5-dimethylphenyl)piperidin-4-yl]methyl]-2-ethenyloxolane-3-carboxamide [(E)-3-amino-2-[4-[1-[1-[2-chloro-5-(trifluoromethyl)phenyl]ethyl]-2,6-dioxo-1,3-diazinan-5-yl]pyrazol-1-yl]prop-2-enylidene]azanium 1-benzylsulfanyl-3-(methylamino)pyrrolidine-2,5-dione (Z,3E)-4-[6-[3-(dimethylamino)phenyl]-8-fluoroimidazo[1,2-a]pyridin-3-yl]-1-N'-propan-2-ylidenebut-1-ene-1,1-diamine;ethane [(5-chloro-2,3-dihydro-1H-inden-4-yl)oxycarbonylamino]carbamodithioic acid 2-[(3Z,6E)-6-(4-ethoxyphenyl)sulfonyliminohepta-1,3,6-trien-2-yl]phenol (3-bromo-4,6-dihydropyrrolo[3,4-d]imidazol-5-yl)-phenylmethanone 1-[6-(3,4-dimethoxyphenyl)pyrimidine-4-carbonyl]imidazolidine-2-sulfonamide 1-[2-(3,4-dichlorophenyl)ethylamino]-3-[(5-nitrothiophen-2-yl)methyl]thiourea 2-[4,6-bis(4-fluorophenyl)pyridin-2-yl]pyridine;dibromomethane;N,N-di(propan-2-yl)propan-1-amine 4-(2,6-difluorophenyl)-N-[5-(furan-2-yl)-1H-pyrazol-3-yl]piperazine-1-carboxamide N'-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)-4,10,11-triazatricyclo[6.3.0.02,6]undeca-1(12),2,4,13-tetraene-3-carbohydrazide 4-azidosulfanyl-N,N'-dimethoxybenzenecarboximidamide 2-(3,4-dichlorophenyl)-5-[(E)-1H-indol-3-ylmethylideneamino]-1,3-oxazole-4-thione 2-[2,4,6-tri(propan-2-yl)phenyl]hydrazine 4-ethylsulfanyl-1,2,3,7-tetrahydro-[1]benzofuro[3,2-e]indole 2-[(4S)-4-aminopentyl]-1,6-dichloro-5-methanimidoylindole-3-carbonitrile (7-methyl-1H-indol-2-yl)-[3-(pyridin-4-yloxymethyl)piperidin-1-yl]methanone 1-(2,3-difluorophenyl)-4-[2-hydroxyethyl(methylsulfonyl)amino]pyrrolidine-2-carboxamide 4-hydroxy-3,6-diphenyl-1H-pyridin-2-one 7-[(4-chlorophenyl)methyl]-2-propan-2-ylidene-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 2-amino-N'-(2-hydroxyethyl)-4-imino-3-phenylmethoxybenzenecarboximidamide [4-(2,6-dimethoxybenzoyl)-1H-pyrrol-3-yl]carbamic acid 4-(2,5-difluorophenyl)-3-methylbutanal 1-N-ethenyl-2-methylidenebutane;4-[(4Z,8E)-9-methoxy-2,3,5-trimethylideneundeca-4,6,8,10-tetraen-4-yl]phenol N-(2-bromophenyl)-5-[2-(dimethylamino)ethoxy]-3,4,6-trihydroxyoxane-2-carboxamide 4-methyl-2-(8-nitroquinolin-6-yl)-1,3-thiazole 5-chloro-6-[[2,3-dihydrothiophene-4-carbonyl(methyl)amino]methyl]pyridine-3-carboxylic acid N-(2,2-diethoxyethyl)-N-[4-(pyridin-2-ylsulfamoyl)phenyl]hexadecanamide (1-benzyltriazol-4-yl)-[6-bromo-3-(cyclopropanecarboximidoyl)indol-1-yl]methanone (2S,4R)-N'-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-4-(2-bromophenyl)-2-hydroxy-6-[[(1R,2S)-2-methoxycyclohexyl]amino]-N-methylideneoctanediamide N'-hydroxy-4-(1H-indol-3-yl)benzenecarboximidamide (2S)-N-[6-(3,5-dimethylpyrazol-1-yl)pyridin-3-yl]azetidine-2-carboxamide 2-hydroxy-N'-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]propanediamide 5-[4-chlorobutyl(2,3-dihydroxypropyl)amino]naphthalene-2-sulfonic acid (3R,4S)-1-[2-methoxy-5-[3-methyl-2-[[7-methyl-6-(trifluoromethyl)imidazo[1,2-a]pyridine-2-carbonyl]amino]butanoyl]benzoyl]piperidine-4-carboxylic acid N-[(2S)-1,5-dicyclopropylpentan-2-yl]-5,6-dimethoxy-1H-indole-2-carboxamide 5-azido-3-(trifluoromethyl)pyridine-2-carboxamide 2-[(5S)-3-[4-(dimethylamino)phenyl]-6-ethoxy-5,10b-dihydro-1H-pyrazolo[1,5-c]quinazolin-5-yl]phenol 2-[(E)-4,4-dimethylpent-1-enyl]-N-[6-[(5R)-3,8-diazabicyclo[3.2.0]heptan-3-yl]pyridin-3-yl]benzamide 3-[4-(2,4-dichlorophenyl)sulfanyl-3-prop-1-en-2-ylsulfonylphenyl]pyridine 6-chloro-2-[4-(3,5-difluorophenyl)cyclohexyl]-1H-benzimidazole 2-(3-azidophenyl)-5-methylfuran 2-[(5R)-3,4,7,8-tetrahydro-2H-azocin-6-yl]-1H-benzimidazole ethane;3-[4-(6-methoxypyridin-2-yl)cyclohexyl]propanamide 1,4-bis(4-tert-butylphenyl)piperazine;ethane [3-(dimethylsulfamoyl)naphthalen-1-yl]sulfamic acid 3,5-bis(hydroxymethyl)naphthalene-1,2-disulfonic acid 4-[azido(pyridin-3-yl)methoxy]butanoic acid (3S)-N-benzyl-1,5-dimethylpyrrolidine-3-carboxamide;hydrochloride 2-(azidomethyl)-6,7-dimethoxynaphthalene 3-[(2,6-dimethylphenyl)sulfinyl-methylamino]-N-(pyridin-4-ylmethoxy)thiophene-2-carboxamide 6-amino-2,5-diphenylhexanoic acid N-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-4,6-dioxo-1H-thieno[3,4-d]pyrimidine-5-carboxamide (3R,4S)-1-[2,6-dimethyl-4-[(5-methyl-3-phenyl-1H-pyrazole-4-carbonyl)amino]benzoyl]-3-methylpiperidine-4-carboxylic acid N-[[2,6-dimethyl-4-(2-phenylethynyl)anilino]carbamothioyl]benzamide 4-azido-5-chloro-2-methoxybenzoic acid 3-N-[[6-amino-5-(4-methylphenyl)pyrimidin-4-yl]methyl]-3-N,2-dimethylbenzene-1,3-dicarboxamide 3-(2,5-dimethoxyphenyl)sulfanyl-1-[(4-methoxyphenyl)methyl]pyridin-2-one 2-[4-(1,3-benzodioxol-5-yl)phenyl]-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidine N-[2-[(3S)-5-cyano-7-ethylsulfanyl-1,2,3,4-tetrahydroisoquinolin-3-yl]phenyl]methanesulfonamide (3S)-1-benzyl-N-[5,7-bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]piperidine-3-carboxamide [(2S)-1-methoxypentan-2-yl]oxybenzene (2R)-N-[6-[2-[2,4-bis(trifluoromethyl)phenyl]ethylsulfamoyl]pyridin-3-yl]pyrrolidine-2-carboxamide 2-cyclopropyl-1,3-diethylpyrrolo[2,3-b]pyridine 2-[4-(1H-pyrrolo[3,2-b]pyridine-5-carbonyl)morpholin-2-yl]ethanesulfonic acid 3-[7-(5-methylthiophen-2-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-pyrazin-2-yl-1H-pyrazolo[4,3-b]pyridine 1-[3-(2,4-dihydroxyphenyl)quinoxaline-6-carbonyl]piperidine-3-carboxylic acid (2E)-N-benzyl-6,7-dichloro-N-methylhepta-2,4-dien-3-amine 2-[[5-(1H-benzimidazol-2-yl)pyridin-3-yl]iminomethyl]-4,6-ditert-butylphenol;dichlorozirconium 4-[1-(2,3,6,7-tetrahydro-1H-inden-1-yl)ethyl]benzoic acid 2-(1-azidonaphthalen-2-yl)acetaldehyde (5R,7S)-5-phenylmethoxycarbonyl-9-oxa-2,5-diazatricyclo[8.4.0.03,8]tetradeca-1(10),11,13-triene-13-carboxylate 5-(4-azidooxyphenyl)-3H-1,3,4-oxadiazol-2-one 4-[4-(4-amino-2,7-dimethylpyrimido[5,4-b][1,4]oxazin-6-yl)phenyl]piperazine-1-carboxylic acid 4-[3,5-bis(trifluoromethyl)anilino]-7-methoxyquinoline-6-carbonitrile N-(2,3-dihydro-1H-inden-5-ylsulfamoyl)-3-fluoro-4-hydroxybenzamide 3-(aminomethyl)-5,6-dichloro-N-[2-[2-(5-cyanopyrazin-2-yl)ethynyl]pyridin-4-yl]pyridine-2-carboxamide 4-(4,5-dimethyl-1H-pyrazole-3-carbonyl)-6-[2-(pyridin-3-ylmethoxy)ethyl]piperazin-2-one 6-bromo-N-(4,5-dihydropyrimidin-2-yl)pyridine-3-carboxamide 5-benzyl-2-[(4,6-dimethylpyridine-3-carbonyl)amino]benzoic acid (2S)-3,3,4,5-tetradeuterio-2-[1,1-dideuterio-7-[[dideuterio-[5-[trideuterio(difluoromethyl)methoxy]pyridin-2-yl]methyl]amino]-3-oxoisoindol-2-yl]piperidine-2-carboxylic acid N-[6-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-ylmethylideneamino)hexan-2-yl]-2,4,5-trifluoroaniline 1-methyl-3-[4,5,6-tris(difluoromethoxy)pyridin-2-yl]imidazolidine 5-methyl-3-[(E)-2-[4-[2-[methyl(pentanoyl)amino]ethoxy]phenyl]ethenyl]-N-propylfuran-2-carboxamide N-[5-[(2R,3S)-4-(cyclopropylamino)-3-hydroxy-1-phenylbutan-2-yl]pyridin-2-yl]acetamide 3-(2,6-dichlorophenyl)-7-[(4-methoxypyridin-2-yl)amino]-N-(trideuteriomethyl)-2H-pyrimido[5,4-e][1,3]oxazin-8-amine 2-ethyl-4-(3,7,11-trithia-9,16-diazatetracyclo[8.6.0.02,7.012,17]hexadeca-1,5,8,10,12,14-hexaen-8-yl)aniline 3-[1-[(2S)-5,7-dimethyl-2-propyloctoxy]-4-(trifluoromethyl)naphthalene-2-carbonyl]-5-ethyl-4-hydroxypyran-2-one 2-[[3,5-bis(trifluoromethyl)phenyl]methylamino]-6-[[5-(difluoromethoxy)pyridine-2-carbonyl]amino]-1-(2-hydroxyethyl)benzimidazole-4-carboxamide 7-ethylsulfonyl-3-[(4-fluorophenyl)methyl]-8,9-dihydro-5H-pyrrolo[2,1-d][1,2,6]triazepine (3R,4S)-1-[2-methyl-6-(4-propan-2-ylpiperazine-1-carbonyl)pyrimidin-4-yl]-4-pyrazol-1-ylpyrrolidin-3-ol 6-(4-methoxyphenyl)spiro[3,4-dihydropyrano[2,3-b]pyridine-2,1'-cyclohexane] 4-(4-chlorophenyl)-3-[6-[(2-methylpropan-2-yl)oxycarbonylamino]pyridin-3-yl]butanoic acid (3-ethylimidazol-4-yl)-[(2S,6R)-2-phenyl-6-propan-2-ylmorpholin-4-yl]methanone 4-(6,7-dihydrocyclopenta[b]pyridine-5-carbonyl)-3-methylpiperazin-2-one N-(cyclohexylmethylidene)-4-(2,3-dichlorophenyl)piperazine-1-carboxamide N-[(Z)-1H-indol-3-ylmethylideneamino]-5-iodonaphthalene-2-carboxamide 4-[(2,3-dimethylimidazol-4-yl)sulfonylamino]thiophene-3-carboxylic acid 5-methoxy-2-[4-(4-propylcyclohexa-1,3-dien-1-yl)phenyl]benzaldehyde N-[4-(1,3-benzodioxol-5-yloxy)phenyl]acetamide 7-[(6-aminopyridine-3-carbonyl)amino]thieno[2,3-b]pyrazine-5-carboxylic acid 2-methyl-3-(4-methylsulfanylphenyl)quinoline N-[1-(6-bromopyridin-2-yl)ethenyl]-3-methoxycyclobutan-1-amine 2-[6-[(4-methylsulfonylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridin-3-yl]quinoline 1-N'-[[4,5-dichloro-2-(2H-tetrazol-5-yl)phenyl]methoxy]-1-N-(2,6-difluorophenyl)cyclopropane-1,1-dicarboxamide 1-(3,4-dimethoxyphenyl)ethanamine;[2-fluoro-5-(trifluoromethyl)-3H-pyridazin-6-yl]urea (2S,3R)-4,4-dimethyl-3-[2-[1-[(4-methylpyridine-2-carbonyl)amino]cyclobutyl]acetyl]oxy-5-oxopentanoic acid (1S,3R)-4,4-difluoro-3-[1-hydroxyethyl-[[5-methoxy-2-[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]-3H-inden-1-yl]amino]methyl]cyclohexane-1-carboxylic acid N-[4-(3,5-dimethylpyrazin-2-yl)butan-2-ylidene]hydroxylamine N-[1-(2,3-dichlorobenzoyl)piperidin-4-yl]-4H-thiopyran-2-carboxamide N-[1,3-dihydroxy-4-(4-methoxyphenyl)pentan-2-yl]acetamide 3-ethoxy-5-(trifluoromethyl)benzoate ethane;7-[(5-methyl-1,3,4-oxadiazol-2-yl)amino]-1-phenyl-2H-pyrido[3,4-b]pyrazine-3,6-dione [3-(hydroxymethyl)-2,6-dimethoxyphenyl]boronic acid 3-(3,5-dichlorophenyl)butyl-[2-[ethenyl(ethylidene)amino]oxypropyl]carbamic acid 7-(3,4-difluorophenyl)-2,5-dimethylpyrido[3,4-b]pyrazine 1-[3,5-bis(trifluoromethyl)benzoyl]-2-(2H-triazol-4-yl)pyrrolidine-2-carboxylic acid 4-[(2R)-1-methoxy-5-phenylpentan-2-yl]sulfanylbutanoic acid 3-(3,5-dichlorophenyl)-1-[3-methyl-2-(pyrrolidine-1-carbonyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-yl]propan-1-one 1-[2,6-di(propan-2-yl)phenyl]-3-[1-[(4-methoxyphenyl)methylamino]piperidin-4-yl]urea 2-[(5,7-dichloro-1H-indole-2-carbonyl)amino]acetic acid N-[3,5-bis(trifluoromethyl)phenyl]-2-cyanopropanamide 2-methylsulfonylpyrazolo[1,5-a]pyrazine 3-[(2,3,4,5-tetramethoxyphenyl)methyl]pyridine N-[4-(5-aminopentoxy)phenyl]sulfanyl-1,3-thiazol-2-amine 2-hydroxyethylimino(oxo)azanium;4-[5-[3-oxo-1,5-diphenylpentyl]thiophen-2-yl]benzoate [(2S,3R)-1-ethyl-5-oxo-3-phenylpyrrolidin-2-yl]-morpholin-4-ylmethanone 4-ethenylsulfanyl-N,N-bis(3-nitrophenyl)benzenecarboximidamide 3-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)-N-ethyl-2-hydroxybenzamide 2-[4-[[(Z)-(3-aminophenyl)methylideneamino]carbamoyl]phenoxy]acetate N-(1,3-dimethylpyrazolo[3,4-b]pyridin-5-yl)oxane-2-carboxamide N-[4-(3,3a,4,5,6,7,7a-octahydro-1H-isoindol-2-yl)pyrimidin-2-yl]benzamide (3R)-4,4,6-trimethyl-2-[6-methylidene-5-(1H-pyrazole-4-carbonylamino)pyrimidin-1-yl]heptanoic acid 3-[6-(1,3-benzodioxol-4-yl)pyridin-2-yl]propanoate 3-fluoro-2-[6-(4-methylphenyl)sulfonyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-yl]phenol 2-[(3,5-dichloropyridine-4-carbonyl)amino]hexanoic acid 5-[2,4-dimethyl-6-[3-oxo-3-(6,7,8,9-tetrahydropyrido[1,2-a]indol-10-ylidene)prop-1-enyl]phenoxy]carbonylthiophene-2-carboxylic acid N-[1-[(3R,4S)-3,4-dimethylpiperidin-1-yl]-1-oxo-3-phenylpropan-2-ylidene]hydroxylamine N-(3,5-dimethoxyphenyl)-1H-indole-2-sulfonamide 3-(2,6-dichlorophenyl)-7-[4-(4-propan-2-ylpiperazin-1-yl)anilino]pyrimido[5,4-e]thiazin-4-one 6-methyl-2-[(3R)-1-(thiophene-2-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 1-[(4S)-3,4-dimethylhexan-2-yl]sulfonyl-4-propan-2-ylbenzene ethane;(Z)-3-[4-(10-methylundecoxy)phenyl]prop-2-enenitrile 5-(2,3-dichlorophenyl)sulfanyl-4,6-diethoxypyridine-2,3,7-triamine 3-(6,8-dichloro-2H-chromene-3-carbonyl)-5-methyl-1,2-oxazole-4-carboxylic acid 1-[3-(4-hydroxypiperidine-4-carbonyl)phenyl]pyrrolidin-2-one 2-N,3-N-bis(3-pyridin-4-ylprop-1-enyl)pyrrolidine-2,3-dicarboxamide 2-[(E)-3-methylsulfonylprop-1-enyl]naphthalene N-(2,4-difluorophenyl)-2-[4-oxo-5-[(6R)-6-phenyloxan-3-yl]pentyl]benzamide 2-(4-oxo-3H-quinazolin-6-yl)benzenesulfonamide 2-(benzylamino)propanoic acid;ethane;4-(3H-pyrrol-5-yl)-2-[3-(trifluoromethoxy)phenyl]quinazoline 2-methyl-3-phenylbenzenesulfonamide 2,4-dichloro-3-ethylsulfonylbenzoate 5-amino-4-(3,7-dimethyl-1H-indol-2-yl)penta-1,4-dien-2-ol 2-methylsulfonyl-N-[4-(1,3-thiazol-2-yl)phenyl]propanamide N-[6-(4-fluorophenyl)cyclohexa-1,5-dien-3-yn-1-yl]propanamide 2-[(2E,5S)-2-[(Z)-1-(4-methoxyphenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid (1S,2S)-N-[3-(4-methylpiperazin-1-yl)cyclobutyl]-2-phenylcyclopropane-1-carboxamide [(2R,4S)-4-hydroxy-2-phenylpyrrolidin-1-yl]-(5-methoxypyridin-3-yl)methanone 2,6-dimethyl-N-(5-pyridin-3-ylpyrimidin-4-yl)morpholine-4-carboxamide 5-bromo-6-(dimethoxyphosphorylmethyl)pyrimidine-2,4-diamine 3-[4-chloro-2-(cyclobutylmethylamino)phenyl]sulfanyl-N,5-dimethoxy-2H-1,3-thiazole-2-carboxamide [(2R,4S)-3-tert-butylsulfanyl-1-[(5-cyanopyridin-2-yl)methyl]piperidine-2-carbonyl]azanium N-[(1S)-2,3-dihydro-1H-inden-1-yl]benzamide [2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]sulfonylphenyl]methanamine 2-[4-[6-(2,3-difluorophenyl)pyridin-2-yl]-1H-pyrazol-5-yl]-N-propan-2-ylacetamide 4-amino-6-[(3-chloro-2-fluorophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-N-(cyclopropylmethoxy)-6-methanimidoylpyrimidine-2,4-diamine 4-N,6-dimethylpyrimidine-2,4,5-triamine;1-ethoxy-3-(5-fluoropyridin-2-yl)propan-2-ol 1-ethenyl-5-methoxy-3-(methoxysulfanylamino)-7,8,9,10-tetrahydrophenanthridine-6,12-dione (2R)-N-[3-cyano-6-ethyl-5-(2,4,6-trimethoxyphenyl)pyridin-2-yl]-1-(4-fluoro-3-methoxybenzoyl)piperidine-2-carboxamide (2S)-6-methyliodanuidyl-2,3,5,7-tetrahydro-1H-furo[3,4-e]indole 2-[1-[(4-methoxybenzoyl)amino]cyclopropanecarbonyl]pyrrolidine-1-carboxylic acid (5-methoxycarbonylfuran-3-yl)boronic acid 2-[4,5-bis(3-aminophenyl)-1,3-thiazol-2-yl]benzene-1,3-diamine N-methyl-2-(3-piperidin-1-ylpropoxy)-4,5-dihydro-1H-benzo[g]quinoline-8-carboxamide 2,3-difluoro-1-[4-(3,4,5-trifluorophenyl)cyclohexyl]oxy-4-(trifluoromethyl)benzene 2-(1H-indol-5-yl)-N-[4-[5-methyl-6-(trifluoromethyl)pyridin-3-yl]butyl]-1,3-thiazole-5-carboxamide (3R)-3-azido-1-[2-[methyl(2-phenylethyl)amino]propanoyl]pyrrolidine-3-carboxylic acid 2-(1-cyclohexylethylamino)-4-phenylbenzonitrile;2-(5-nitroindol-1-id-3-yl)acetaldehyde (3S)-4-[2-[4-chloro-2-[[1-(cyclopropylmethyl)pyrazole-4-carbonyl]amino]phenoxy]ethoxycarbonyl]morpholine-3-carboxylate 4-[(Z)-3-amino-2,3-dimethylbut-1-enyl]-N-[(E)-pent-1-enoxy]benzamide 2-(1,3-benzothiazol-2-yl)phenol;cyclohexa-3,5-diene-1,2-diimine;1-phenylnaphthalene;platinum(2+) 1-[2-hydroxy-3,5-bis(phenylmethoxy)benzoyl]piperidine-4-carboxylic acid 1-methyl-2-[3-(1H-pyrazol-4-yl)phenyl]pyrazine 2-[6-amino-5-(methylamino)pyridazin-3-yl]phenol (6R,11bS)-9-[4-bromo-3-(trifluoromethoxy)phenyl]-6-(3,4-dichlorophenyl)-5,6,7,11b-tetrahydro-2H-[1,3]thiazolo[5,4-a]quinolizine 4-[2-(difluoromethyl)benzimidazol-1-yl]-5-iodo-1H-pyrimidin-6-one N-[2,6-dichloro-3-(3-oxo-5H-imidazo[1,5-a]isoindol-5-yl)phenyl]-5-fluoro-4-(1,3-thiazol-4-yl)thiophene-2-carboxamide 1-[(2S)-4-acetyl-7-fluoro-6,8-dimethoxy-3,4-dihydro-2H-naphthalen-2-yl]ethanone 2-[(1E,3Z)-5-bromopenta-1,4-dienyl]sulfanyl-5-chloro-N'-methyl-1H-benzimidazole-4-carboximidamide N-[3-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)phenyl]-6-pyrrolidin-1-ylpyridine-2-carboxamide 5-[(3,4-dichlorophenyl)methyl]-3-propanoyl-1H-indole-7-carboxylic acid 4-(3,4-difluorophenyl)-N-[2-[(1S)-3-hydroxycyclohexyl]indazol-6-yl]piperazine-1-carboxamide ethane;5-methyl-6-oxo-3-phenylpiperidine-2,4-dione 2-ethyl-3,5-dimethoxy-6-(phenyliminomethyl)phenol 2-[[4-(5-aminopyridin-3-yl)-1H-indazol-6-yl]oxy]acetic acid 4-[3-[(2,6-dichlorobenzoyl)amino]pyrazol-1-yl]benzamide 2-[(3Z)-4-(trifluoromethoxy)hexa-1,3,5-trien-3-yl]oxypyridine (4aS)-7-methylsulfonyl-1,2,3,4,4a,5-hexahydropyrazino[1,2-a]quinoline;hydrochloride (E)-3-[4-[4-[[4-butyl-2-cyclopentyl-1-[1-(2,4-dichlorophenyl)ethyl]-6-oxopyrimidine-5-carbonyl]amino]phenoxy]phenyl]-2-methylprop-2-enoic acid 2-[6,8-dideuterio-4-methyl-5-(trifluoromethoxy)naphthalen-2-yl]-1,3-thiazole 3-bromo-2,5-dimethylimidazo[1,2-a]pyridine;ethane N-[(1S,2R)-4-fluoro-5-(methylaminosulfanylmethyl)-2,3-dihydro-1H-inden-2-yl]acetamide N-[1,3-benzothiazol-2-yl(diphenyl)methyl]-4-ethylaniline (5Z)-2-methylsulfanyl-5-[(3,4,5-trimethoxyphenyl)methylidene]imidazolidin-4-one 5-[6-(trifluoromethyl)pyridin-3-yl]-1,2-dihydro-3,1-benzoxazin-4-one 1-[(Z)-3-methylsulfanylprop-2-enyl]-4-oxoquinoline-3-carboxamide 4-[6-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]pyrimidine-5-carbonitrile 3-ethylsulfonylbenzene-1,2-diamine 2,6-diiodo-N-[(Z)-1H-indol-3-ylmethylideneamino]benzamide N-[[1-(3,4-difluorophenyl)cyclobutyl]methyl]-5-[2-hydroxy-4-[3-[4-[4-(4-propan-2-ylpiperazine-1-carbonyl)piperidin-1-yl]but-1-ynyl]anilino]pyrimidin-5-yl]pentane-1-sulfonamide 2-[3-(4-methoxyphenyl)-1-[[(3R,5S)-5-methylpiperidin-3-yl]methylamino]-1,7-naphthyridin-6-yl]phenol 6-bromo-3,4-dimethoxypyridine-2-carboximidamide 2-[(2,4-dichlorophenyl)methyl]-5-hydroxy-7-oxabicyclo[4.1.0]hepta-1,3,5-trien-8-one N-[6-(3,5-dimethylpyrazol-1-yl)pyridin-2-yl]-2-(7H-purin-6-ylamino)acetamide 3-chloro-2-methoxynaphthalene;4-(3-ethylphenyl)morpholine (4E)-2-[2-chloro-5-(trifluoromethyl)phenyl]-3,7-dihydro-2H-1-benzoxocine;ethane 2-[(2R)-1-hydroxypropan-2-yl]oxybenzamide (3R)-5-ethyl-4-hydroxy-7-iodo-3-[(2E,5Z)-2-methoxyhepta-2,5-dienoyl]-1-pentyl-3H-1,4-benzodiazepin-2-one 3-(5-cyclopropylthiophen-2-yl)imino-2H-1,2-benzothiazole-7-carboxamide 5-[(2Z,4E)-hepta-2,4,6-trien-2-yl]oxy-6-propan-2-ylidene-1-[4-(pyridin-2-ylmethyl)phenyl]hexane-3,4-dione 2-[5-(1-ethoxypropyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-2-yl]-7-methylidene-8H-[1,2,4]triazolo[1,5-a]pyrazine 1-[(2R,3S)-5-azido-4-hydroxypentan-2-yl]pyrimidine-2,4-dione 2-methylsulfonyl-6-(thiophen-3-ylmethoxy)pyrimidine-4-carbonitrile 3-(1,2-dihydropyrrolo[2,3-b]pyridin-5-yl)-5-ethylpyrazolo[1,5-a]pyrimidine N-[4-(2,3-dihydrothiophen-5-yl)phenyl]-3-fluoroaniline 7-(6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl)-3,4,5,6-tetrahydro-1H-1,4-benzodiazepin-2-one 3-(2,6-dibromophenyl)butanamide 2-[(E)-3-(5-fluoropyridin-1-ium-4-yl)prop-2-enyl]-3,7a-dihydroisoindole-1,3'-dione N-[5-(furan-2-yl)pyridin-3-yl]-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-4-carboxamide 1-[4-[(3E,7Z)-3,5,6-trimethyldeca-3,7,9-trienoxy]phenyl]cyclopropane-1-carboxylic acid 4-(5-methyl-1,3-thiazol-2-yl)-N-[6-(trifluoromethoxy)pyridin-3-yl]thiophene-2-carboxamide 5-fluoro-3,7-dihydroxy-2-(4-nitrophenyl)-4H-chromene-6-carboxamide 2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1]benzofuro[3,2-d]pyrimidine 4-[[5-(2-fluorophenyl)-3-[6-[4-(trifluoromethyl)phenoxy]hexanoyl]pyrazol-1-yl]methoxycarbonylamino]pyridine-2-carboxylic acid 2-[N-(5,6,7,8-tetrahydronaphthalen-1-yl)anilino]benzoic acid ethane;4-methyl-2,2-diphenyl-3H-1-benzofuran 4-[4-(azidomethyl)phenyl]-1-(3,4,5-trifluorophenyl)cyclohexan-1-ol 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-N-pyridin-2-ylazetidine-3-carboxamide ethane;3-[1-[2-(5-methylfuran-2-yl)imidazol-1-yl]propan-2-ylamino]cyclohex-2-en-1-one 4-[2-chloro-5-(trifluoromethyl)phenyl]-3,6-dihydro-2H-pyridine-1-carboxylic acid 2-(4,5-dimethyl-3H-azepine-6-carbonyl)benzoic acid 2-(4,5-dihydro-1,3-thiazol-2-yl)-3H-imidazo[4,5-c]pyridine 2-[3-(4,5-dihydrothieno[3,2-b]pyrrole-2-carbonyl)phenoxy]acetamide 4-(3-azidopropylamino)pyrimidine-5-carbonitrile 2-[1,4-dimethyl-7-(trifluoromethyl)-3H-furo[2,3-c]pyridine-5-carbonyl]-6-oxa-2,9-diazaspiro[4.5]decan-8-one N-[(E)-2-methyl-1,1-diphenylpentan-3-ylideneamino]-4-morpholin-4-ylphthalazin-1-amine 2-[3-(dipropylamino)phenyl]-4-pyridin-1-ium-1-yl-6-(trifluoromethyl)phenol 1-[3,4-di(propan-2-yl)phenoxy]-N-propan-2-ylideneisoquinoline-7-sulfonamide 3-[2-(1-methylcyclohexa-2,4-dien-1-yl)ethynyl]aniline (3-aminosulfanylphenyl)methanesulfonic acid [5-chloro-2-fluoro-4-(hydroxymethyl)phenyl]-[4-[5,7-difluoro-6-(3,3,3-trifluoropropoxy)pyridin-2-yl]piperazin-1-yl]methanone;(2S)-N-ethylsulfanylhexan-2-amine (3S,6R)-3-[2-hydroxyethyl(methylsulfonyl)amino]-4-(3-phenylpropanoyl)-8-oxa-4-azabicyclo[5.2.0]nonane-9-carboxylic acid 6-[4-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]pyridine-3-carboxamide 4-[4-amino-7-methyl-6-(2-phenoxyphenyl)pyrrolo[3,4-d]pyrimidin-5-ylidene]-N-propan-2-ylcyclohexane-1-carboxamide (2S,4S)-4-hydroxy-1-[2-(3-methyltriazol-4-yl)acetyl]pyrrolidine-2-carboxylic acid 1-[5-(4-azido-2,6-dimethoxyphenoxy)pyridin-3-yl]-N-ethylmethanimine (E)-N-[2,5-dimethoxy-4-(1H-pyrrol-3-yl)phenyl]but-2-enamide 1-[4-[3-(4,5-dihydro-1H-imidazol-2-ylamino)pyridin-2-yl]oxycyclohexa-2,4-dien-1-ylidene]-N'-methylmethanediamine 2-[6-fluoro-5-(4-methylpyridin-3-yl)-1H-indazol-3-yl]-7-thiophen-3-yl-4,5-dihydro-3aH-cyclopenta[c]pyrazole 4-cyclohexyl-2-phenylcyclohexa-1,5-dien-3-yn-1-amine N-[(2,5-dichlorophenyl)methyl]formamide;1,3-difluoro-2-methoxybenzene 6-methoxy-N-(1-methylsulfonylpiperidin-4-yl)spiro[3,4-dihydrochromene-2,4'-piperidine]-4-carboxamide [4-(1,3-benzodioxol-5-yl)-6-hydroxy-2H-chromen-3-yl]-cyclopropylmethanone (2R,4S)-N-(benzenesulfonylcarbamoyl)-1,9-dioxa-3-azaspiro[5.5]undecane-2-carboxamide 4-azidooxy-2,6-dichloro-5,7-dimethylquinazoline 3,4-dimethylbenzaldehyde;ethane;1-[(2E)-2-ethenylpenta-2,4-dienyl]-6-[2-[5-[3-(oxolan-2-ylmethoxy)propoxy]-6H-naphthalen-2-yl]ethynyl]naphthalene 1-(5-bromopyridin-2-yl)propan-1-imine;ethane 1-[4-(6,7-dimethoxyquinolin-4-yl)oxy-2-fluorophenyl]-3-[5-(1H-indole-2-carbonyl)-2-methoxyphenyl]urea 4-chloro-6-[2-(1,5-dimethylpyrazol-3-yl)ethynyl]quinazoline 6-[(Z,3E)-1-amino-3-(pyridin-2-ylhydrazinylidene)prop-1-en-2-yl]-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide 2-methylsulfanyl-6,7,8,9-tetrahydropyrimido[4,5-b][1,5]diazepine (3R)-N'-[2-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]ethyl]-3-hydroxybutanehydrazide;6-methoxy-1,2-benzoxazol-3-amine 1-[2,4-dichloro-3-[(6-morpholin-4-ylpyridin-3-yl)methyl]quinolin-7-yl]ethanone 6-bromo-2-[5-(4,4-dimethylcyclohexen-1-yl)pyridin-3-yl]-7-fluoroquinoline [(1R)-2,3-dihydro-1H-inden-1-yl]urea ethane;1-[2-methoxy-3,5-di(propan-2-yl)phenyl]-N-methylmethanimine 3-amino-N-(2,6-dichlorophenyl)-2-hydroxypropanamide;ethane 5-[(4-methoxyphenyl)sulfonylamino]-2-morpholin-4-ylbenzoic acid;2,2,2-trifluoroacetic acid (1R)-N,N-dimethyl-3-phenyl-1-[4-(trifluoromethoxy)phenyl]propan-1-amine 6-[(1,1-dioxothiolan-3-yl)amino]-8-[[(2S)-2-methylpiperidin-4-yl]amino]-7-nitro-3H-quinazolin-4-one 2-[3-(2,4,6-trimethylphenyl)propanoylamino]propanedioic acid 3-amino-N',2-bis(4-bromophenyl)-5-(2-methyltetrazol-5-yl)benzenecarboximidamide 6-methyl-2-[(1S)-1-(1,5,7-trimethylpyrrolo[3,2-b]pyridin-4-ium-3-yl)ethoxy]quinoline 3,4-dimethoxy-N-[(2E,4Z)-5-phenylhepta-2,4,6-trien-2-yl]benzamide (E)-N-[2-(4-methylphenyl)phenyl]-3-pyridin-2-ylprop-2-enamide (2R,4S)-1-acetyl-4-methoxyimino-N-[[5-(4-methylphenyl)furan-2-carbonyl]amino]pyrrolidine-2-carboxamide 2-[(1S,3R)-3-[(6-chloro-8-fluoroquinazolin-4-yl)amino]cyclopentanecarbonyl]prop-2-enenitrile 2-(4-bromophenyl)sulfonylbenzonitrile 1-[5-methoxy-2,2-dimethyl-4-(3-oxo-1H-isoindol-2-yl)-3,4-dihydrochromen-6-yl]-5-pyrrolidin-3-ylpyrazole-3-carboxylic acid 2-chloro-4,6-dimethoxypyrimidine;ethane N-[1,2-diamino-3-(4-aminobutyl)-5,6-dimethoxybenzimidazol-1-ium-4-yl]-N-phenylcarbamate 4-tert-butyl-2-(2,6-difluorophenyl)quinoline N-[[3-(4,5-dimethyl-1H-imidazole-2-carbonyl)phenyl]methyl]-5-[(2R)-1,1-dioxothiolan-2-yl]-1,3,4-thiadiazol-2-amine 1-[4-(1H-indol-6-yl)-2,5-dimethylphenyl]ethanone 1-[(5,6-diamino-2-methylpyrimidin-4-yl)amino]propan-2-one 4-azido-2,6-difluoro-N-methyl-3-[(2-oxopyrrolidin-1-yl)methyl]benzamide 2,4-dimethyl-6-(3-nitrosophenyl)pyrimidine N-(3,5-dimethoxyphenyl)-3-[2-[4-methyl-6-oxo-1-[4-[2-(trifluoromethyl)pyridin-4-yl]piperazin-1-yl]pyridazin-3-yl]ethynyl]benzamide (2R)-N-(6-benzylsulfonyliminopyridin-3-yl)-2-[7,8-difluoro-2-methoxy-4-oxo-5-[4-(trideuteriomethyl)phenyl]quinazolin-1-yl]propanamide 1-[(1S,2R)-1-azido-5-methyl-3,4-dihydro-2H-naphthalen-1-yl]ethanone 5-methylspiro[2H-1,4-benzoxazine-3,1'-cyclopentane]-7-sulfonamide 2-[1'-(cyclopropanecarbonyl)-7,9-dioxospiro[4H-pyrido[1,2-a]pyrimidine-3,4'-piperidine]-2-yl]acetonitrile 4-[5-(2,3-dihydro-1H-inden-4-yl)-1,3-thiazol-2-yl]piperidine-1-carboxylic acid N-[2-[4-(dimethylamino)phenyl]ethyl]-2,3-bis(ethenyl)aniline [7-(4,6-diphenyl-1,3,5-triazin-2-yl)naphthalen-1-yl]boronic acid 1-[(2R)-3-acetylsulfanyl-2-methoxypropyl]indole-6-carboxylic acid 1-cyclopentyl-4-(3,5-dimethylphenyl)piperidine 3-(2,6-difluorophenyl)cyclopropane-1,1,2,2-tetracarbonitrile 1-(4-chlorophenoxy)butan-2-one;propane 2-amino-N-(3-methoxypropyl)pyridine-4-carboxamide;8-[2-chloro-5-(1,2,4-triazol-1-ylmethyl)phenyl]-3-ethyl-2-phenylisoquinolin-1-one 2-(cyclopentylmethyl)-7-(thiophene-3-carbonylamino)heptanoic acid 2-[(1R,3S)-3-[[7-(carboxymethoxy)-6-methylquinazolin-4-yl]amino]cyclopentyl]acetic acid 1-[3-(2,4-dichlorophenyl)prop-2-enyl]piperidine 5-chloro-N-[(3R,4S)-1-methylsulfonyl-4-phenylpyrrolidin-3-yl]pyrimidine-2-carboxamide 3-[(4-phenylphenyl)methyl]benzamide (6-phenyl-2,4-diazatricyclo[5.2.1.02,7]deca-3,5,7,9-tetraen-3-yl)methanol 5-(bromomethyl)-3-(4-ethenoxyphenyl)-1,2,4-oxadiazole 2-(2,6-dioxopiperidin-3-yl)-5-[(1R,3S,4S)-3-hydroxy-4-methylcyclopentyl]isoindole-1,3-dione N-[4-chloro-2-(2,3-dihydropyridin-5-yl)phenyl]propanamide 2-[(3S)-7-[(2,6-dichlorophenyl)methoxy]-1,2,3,4-tetrahydroisoquinolin-3-yl]-5-ethynylphenol N-[5-[(Z,1E)-2-hydrazinylidenebut-3-enoxy]pyrazin-2-yl]acetamide (4S)-3,7,7-trimethyl-N-[[2-(methylamino)pyridin-1-ium-4-yl]methyl]-1-oxo-6,8-dihydro-5H-pyrrolizine-4-carboxamide 2-amino-6-ethoxy-4-[3-nitro-5-(trifluoromethyl)phenyl]-4H-pyran-3,5-dicarbonitrile 5-[(2Z)-2-[4-chloro-2-methyl-3-(trifluoromethyl)phenyl]-2-methoxyiminoethyl]-N,2,3-trimethylimidazole-4-carboxamide 4-(3,5-dichlorophenyl)sulfanylmorpholine 3-[5-fluoro-2-(3-hydroxyphenyl)phenyl]phenol 5-[5-(2-fluorophenyl)-1H-pyrazol-3-yl]pyridine-2-carboxamide N-ethyl-2,4-difluoro-5-[3-[(1S)-3-hydroxycyclopentyl]-6-oxopyridazin-1-yl]benzenesulfonamide 2-[2-(4,5-dimethoxycyclohexa-1,5-dien-1-yl)cyclopropyl]-N-methylaniline 2-fluoro-4-[3-(N'-hydroxycarbamimidoyl)phenyl]benzoic acid 3-(4-chlorophenoxy)-N'-hydroxy-5,6-dimethylpyridazine-4-carboximidamide ethane;3-ethyl-8,9-dimethoxy-6-methylidene-5H-benzo[b][1]benzazepine 3-[(5-cyclohexyloxy-2,3-dihydro-1H-inden-4-yl)methyl]piperidine 1-[5-chloro-2-(3,4-dihydropyrazol-2-yl)phenyl]piperidine 3-cyclobutyl-N,5-diphenylpyrazolo[1,5-a]pyrimidine-6-carboxamide N-[2-fluoro-4-(trifluoromethyl)phenyl]-3,5-diiodobenzamide (E)-N-[2-(4-cyclohexylphenyl)propan-2-yl]but-1-ene-1,3-diamine 3-methyl-6,7-bis[4-(2-oxopyrrolidin-1-yl)phenyl]pyrido[2,3-d]pyrimidin-3-ium-4-one 3-(2,6-dichloroanilino)-N-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide 1-[5-(3,4-dichlorophenyl)-4-[[4-(hydroxymethyl)cyclohexyl]amino]-2-propan-2-yloxybenzoyl]piperidine-2-carboxylic acid 1-benzyl-4-[4-(hydroxymethyl)cyclohexa-2,4-dien-1-yl]piperazine-2,6-dione N-(4,4,4-trifluorobutyl)-1H-indole-2-carboxamide (5-benzylsulfanyl-4,6,7-trihydroxy-2,3-dihydroinden-1-ylidene)azanium (E,2S)-N-[(1R)-1-(4-chloro-3-fluorophenyl)ethyl]-2-formyl-6,7-dimethoxy-5-methylidenehept-3-enamide 3-[4-[(1S)-1-aminoethyl]phenyl]sulfanyloxyaniline;hydrochloride 2-[[6-(3,5-dimethylpyrazol-1-yl)pyridine-3-carbonyl]amino]acetic acid 2,5-dimethylbenzene-1,3-disulfonate 3-[(4E,7Z)-5-chlorononaa-2,4,7-trienyl]phenol 1-(2-benzylphenyl)propane-2,2,3-triol 1-(1,2-oxazol-5-ylmethylamino)-3-[(4-phenylphenyl)methoxy]urea 4-cyclopropyl-6-(5,7-dimethoxy-3-oxo-1H-isoindol-2-yl)-N-(1H-pyrrolo[2,3-b]pyridin-4-yl)cyclohexa-2,4-diene-1-sulfonamide 5-[3-(2,6-difluorophenyl)imidazol-4-yl]-2-propan-2-yltetrazole 2-[(6-chloropyridazine-3-carbonyl)amino]ethyl-dimethylsulfanium 2-[(3S)-5,5-difluoropiperidin-3-yl]-N-pyrazin-2-ylsulfanylethanamine (5S,7R)-5-(3,4-dichlorophenyl)-N-[3-(2,5-dimethoxyphenyl)butyl]-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide N-[5-tert-butyl-2-(3-methylphenyl)pyrazol-3-yl]-4,5-dihydropyrimidin-2-amine N-[(5Z)-5-[[4-(2,3-dihydro-1,4-benzodioxin-6-yloxymethyl)phenyl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]benzamide ethane;2-[1-[4-methyl-6-(2,3,5-trifluorophenyl)pyridine-2-carbonyl]azetidin-3-yl]acetonitrile N-[(2S,4S)-5-cyclopropyl-1-ethanimidoylpiperidin-2-yl]pyrimidine-5-carboxamide N-[(3S,4R)-1-cyclopentylsulfonyl-4-(5-methoxypyridin-2-yl)pyrrolidin-3-yl]ethanesulfonamide;hydrochloride 2-[6-[(E)-1,2-bis(4-chlorophenyl)ethenyl]-3H-imidazo[1,5-a]pyrazin-4-ylidene]ethanamine;fluoromethane 3-N,3-N-dimethyl-5-[4-(trifluoromethoxy)phenyl]-2H-furo[2,3-e]indole-7,8-diamine 3,4-dichloro-5-[1-[6-methyl-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-4-yl]-1,2-thiazole N-[(3R)-1-benzylpiperidin-3-yl]-2-chloro-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carboxamide (3R)-N-[(1S)-5-aminocyclohepta-2,4-dien-1-yl]-1-[7-[(2-oxopyrrolidin-1-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]piperidine-3-carboxamide 2-(2,4-difluoro-3-iodophenyl)acetic acid (3-chlorophenyl)-[4-(thiophene-2-carbonylamino)phenyl]carbamic acid N-azido-2-chloro-4-methylsulfanylbenzohydrazide 2,6-difluoro-N-(3-methylbutyl)aniline N-cyclopropylsulfanyl-2,5-difluoro-4-[(1R)-2-oxo-1-phenyl-8-pyridin-3-yloxyoctyl]benzamide 3-ethyl-N,5-dimethoxy-4-[(Z)-2-[5-(4-methoxyphenyl)-1H-imidazol-2-yl]-3-phosphanylideneprop-1-enyl]-N-[[(E)-oxolan-2-ylidenemethyl]amino]benzamide 3-azido-4,6-bis(3-methylbutoxy)pyran-2-one 3-(3,4-dimethoxyphenyl)sulfinylpropylhydrazine 1-(3-chloro-4-methoxyphenyl)-4-[2-(difluoromethyl)pyrimidin-5-yl]butane-1,4-dione N-[1-(3,4,5-trimethoxyphenyl)imidazol-4-yl]-2H-[1,2,4]triazolo[4,3-a]pyridine-1-carboxamide (1-hydroxy-3,4-dihydro-2H-quinolin-8-yl)-(3-pyridin-4-yl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl)methanone;2,2,2-trifluoroacetic acid 5-(2,3-dihydropyrrole-1-carbonyl)-2-(propanoylamino)benzamide 2-(1,3-dimethylpyrazolo[4,3-d]pyrimidin-7-yl)sulfanylpyridine-3-carboxylic acid 2-[(3,4-difluorophenyl)methyl]piperidine;hydrochloride 2-(1H-imidazole-5-carbonylamino)benzenesulfonate 7-butyl-3-chloro-4H-quinoxaline 2-[4-[6,7-dimethoxy-2-(trifluoromethyl)-1H-indole-3-carbonyl]piperazin-1-yl]-N,N-dimethylacetamide 4-(1,1,1-trifluoropropan-2-yl)pyridine-3-carboxylic acid 4-[(1S)-2,3,5,6-tetrahydro-1H-1-benzazocin-9-yl]butanal 2-amino-N,6-dimethyl-1H-benzimidazole-5-carboxamide;N'-[4-(3,5-difluorophenyl)pyridin-2-yl]ethanimidamide 2-(4-ethylsulfonylphenyl)benzonitrile N-(2,6-dimethylphenyl)-4-ethoxyiminobutanamide N-(cyclohexylmethyl)-2,5-difluoro-3,4-dihydro-1H-pyrido[4,3-b]indole-8-carboxamide 1-[(4-fluorophenyl)methyl]-5-hydroxy-3H-indol-2-one N-(6-aminopyridin-3-yl)-2-[2,4-dioxo-1-(thietan-3-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]acetamide [(2R,3S)-3-[1-[4-[4-[[(E)-N'-hydroxycarbamimidoyl]phenyl]methyl]pyridine-2-carbonyl]piperidin-4-yl]oxiran-2-yl]carbamic acid 2-methyl-N-(3,3,4,5,6-pentadeuterio-7-hydroxyheptan-2-yl)benzamide 1-(2-fluorophenyl)-4,5,6,7-tetrahydroindazole 4-(6-propanoylpyrimidin-4-yl)oxypiperidine-1-carboxylic acid 4-(aminomethyl)-1-[5-(3,3-dimethylbutoxy)-6-ethylpyridine-2-carbonyl]piperidine-4-carbonitrile 2-cyclopropyl-1'-[(6-methylpyridin-3-yl)methyl]spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,4'-piperidine]-4-one N-azido-5,6-dihydroxynaphthalene-2-carboxamide N-[[2-(3,5-dimethyl-1H-pyrazol-4-yl)phenyl]methyl]-1H-pyrrolo[2,3-b]pyridine-6-carboxamide N-(1,3-benzothiazol-5-yl)-2-(4-methoxypiperidin-1-yl)-5-(trifluoromethyl)pyridine-3-sulfonamide N-[3-(4-aminophenyl)-2,6-difluorophenyl]-2,6-bis(trideuteriomethoxy)benzamide 3-[3,4-difluoro-2-(trifluoromethyl)phenoxy]azetidine 3-bromo-1,5-bis[2-(3-fluorophenyl)ethyl]pyrazole (3-cyclopropylpiperidin-1-yl)-[5-ethylsulfonyl-6-[7-methoxy-2,2,4-trioxo-8-(trifluoromethyl)-3H-chromen-3-yl]-1-benzofuran-2-yl]methanone (2S)-1,3-dimethyl-N-[6-[4-[5-(trifluoromethyl)pyridin-3-yl]oxycyclohexyl]pyridazin-3-yl]azetidine-2-carboxamide 2-amino-4-(3,5-difluoro-1H-pyrrolo[2,3-b]pyridin-7-yl)-N,6-dimethoxypyrimidine-5-carboxamide 3-(2,2-difluoropropyl)-2,4,6-trimethylaniline;ethane [2-methyl-3-(2-methyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-yl)-3,5,6,8-tetrahydro-1H-pyrrolizin-7-yl]urea 1-[(2R,3S)-2-hydroxy-3-(tetrazol-1-yl)butanoyl]-N-phenylpyrrolidine-2-carboxamide 2-amino-N',5-dihydroxybenzenecarboximidamide 1-(2,4-dimethylphenoxy)-3-[2-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]piperidin-1-yl]propan-2-ol 7-(2,4-difluorophenyl)-3-[(1S)-6-methoxy-5-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]heptanoic acid (3E)-4-amino-3-[[2,6-difluoro-4-(trifluoromethyl)phenyl]methylidene]azete-2-thione 2-[3-(1,2-dihydroisoquinolin-6-yl)pyrazol-1-yl]-N-ethylacetamide 6-[5-(aminomethyl)thiophen-2-yl]quinoxaline-2,3-diamine N-[(5R,7S)-2-methyl-9-oxo-11-oxa-1,3-diazatricyclo[8.4.0.03,8]tetradeca-10,13-dien-12-yl]furan-2-carboxamide 3-[(2,5-difluorophenyl)methoxy]thiophene 2-(4-benzylpiperazin-1-yl)-N'-hydroxypyrimidine-5-carboximidamide 2-[6-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-3-ylamino)imidazo[1,2-b]pyridazin-3-yl]-4-fluorophenol 4-bromo-2,3-difluoro-6-[(E)-1-hydroxybut-1-enyl]phenol;4-chloroaniline 4-methoxy-N-[5-[2-(1-methylpyrazol-3-yl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]benzamide 5-[3,4-dimethyl-1-(2H-tetrazol-5-yl)cyclohexa-2,4-dien-1-yl]sulfanylpentanoic acid 2-azido-3,4,5,6-tetrafluorobenzoic acid 2-bromo-5,6-dihydroisoquinolino[1,2-b]isoquinoline 3-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl)-1H-pyridazin-6-one [2-methyl-4-(pyridin-3-yldiazenyl)phenoxy]boronic acid 4-[4-[(3Z,5Z)-hepta-1,3,5-trien-2-yl]pyridin-3-yl]benzoic acid 6-[(1R,2R)-2-acetylcyclopropanecarbonyl]oxy-N-phenylpyridine-3-sulfonamide N-(2,2-diethoxyethyl)-N-[(3R,4S)-4-(dimethylamino)pyrrolidin-3-yl]thiophene-2-carboxamide;hydrochloride 3-[2,4-dimethyl-1-(5-phenyl-1H-imidazole-2-carbonyl)pyrrolidin-2-yl]propanoic acid 2-methylsulfanyl-4-(1,3-thiazol-5-yl)-6H-thieno[2,3-b]pyrrole-5-carboxamide 1-[4-[2-(2-fluorophenyl)-5-methylpyrrolidine-1-carbonyl]-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]ethanone N-[3,5-bis(trifluoromethyl)phenyl]-2-chloro-N-ethylacetamide 2-bromo-4,6-bis(propan-2-yloxymethyl)aniline (2S,4R)-1-[(5,6-diphenyl-[1,2]thiazolo[3,4-b]pyridin-7-yl)oxymethyl]-N-hydroxy-4-(pyrrolidine-1-carbonyl)piperidine-2-carboxamide [4-(cyclopropylmethoxy)-1,2-dihydroquinolin-6-yl]-[2,4-dihydroxy-3-(3-methylbut-2-enoxy)phenyl]methanone 4-[2,4,6-trichloro-N-(2-methylpropanoyl)anilino]benzenesulfonic acid 1-(2,3-dichlorophenyl)-N-[(Z)-(4-hydroxy-3-nitrophenyl)methylideneamino]-5-pyrrolidin-1-ylpyrazole-4-carboxamide 3-(2,6-dichlorophenyl)-7-[4-(1H-pyrazol-5-ylmethyl)piperazin-1-yl]-2H-pyrimido[5,4-e][1,3]oxazin-4-one 2-[2-(4,4-difluoropiperidine-1-carbonyl)imidazo[1,2-a]pyridin-6-yl]chromen-4-one;ethane 7-(4,6-dimethoxypyrimidin-5-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-4H-pyrrolo[2,1-c][1,2,4]triazole-6-carboxamide 2-(5,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl)benzoic acid 4-[2-(2,6-dioxopiperidin-3-yl)hydrazinyl]-N-(4-methoxyphenyl)butanamide 2-[4-(2,2-dimethylpropoxy)-3,5-difluorophenyl]benzotriazole (2S)-1-ethoxycarbonyl-6-methyl-3,4-dihydro-2H-quinoline-2-carboxylic acid 2-azido-4,6-dimethyl-N-propan-2-ylbenzamide (4-benzyl-1,3-oxazol-2-yl)methanesulfonate N-[1-(2,4-difluorophenyl)ethyl]-3-methylbenzamide 4-[2-(diethylamino)anilino]benzenesulfonic acid 2-[1-(3,4-dimethoxyphenyl)-6-hydroxy-2H-quinazolin-7-yl]acetamide 1,7-dimethoxy-2-[(E)-3-[4-[1-(3-propylphenyl)ethylideneamino]oxyphenoxy]prop-1-enyl]naphthalene-6-sulfonic acid 3-[2-[(2,4-difluorobenzoyl)amino]anilino]benzoic acid 4-[4-(6,7-dimethoxyquinolin-4-yl)oxyanilino]cyclohexan-1-ol 2-chloro-4-methyl-6-[(E)-[1-(3,4,5-trimethoxyphenyl)imidazol-2-yl]iminomethyl]phenol [3-chloro-2-(5,6-dihydronaphthalen-1-yl)phenyl]phosphane 2-[(5-amino-1,3,4-thiadiazol-2-yl)diazenyl]phenol 4-[1,3-bis(2-bromoethyl)imidazol-1-ium-2-yl]butanoate 4-(azidomethyl)-6-[2-(4-fluorophenyl)ethynyl]-1H-indazole 1-cyclopentyl-N-[(1S)-1-pyridin-2-ylethyl]pyrazole-4-sulfonamide N-[4-(2,6-dimethylmorpholine-4-carbonyl)pyridin-3-yl]cyclopropanecarboxamide 1-[(4-chlorophenyl)methyl]spiro[2H-indole-3,8'-6H-furo[2,3-e]indole] 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-1H-pyrazole 2-bromo-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N-ethylbenzamide ethane;3-[4-(4-ethenylphenoxy)butoxy]propanal 2-methoxy-4-[(E)-(1,3,3,5-tetraethylindol-2-ylidene)methyl]phenol 5-[2,6-dichloro-4-(trifluoromethyl)phenoxy]-1H-pyrazole N-[6,7-diamino-2,5-bis(hydroxymethyl)cycloocta-1,4,6-trien-1-ylidene]benzamide (5E)-2-(2,3-dichlorophenyl)imino-5-[[4-(naphthalen-1-ylmethoxy)naphthalen-1-yl]methylidene]-1,3-thiazolidin-4-one 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonylamino)cyclobutane-1-carboxylic acid N-[2,6-dichloro-4-(cyclohexylcarbamoyl)phenyl]-4-(methoxyiminomethylamino)-3-(methylamino)thiophene-2-carboxamide 2-[5-chloro-3-(4-hydroxyphenyl)-1H-pyrazol-4-yl]cyclohexan-1-one 1-[2,4-dichloro-3-[(4-methoxyphenyl)-phenylphosphanyl]phenyl]ethanethione 2,4-bis[(Z)-(phenylhydrazinylidene)methyl]phenol ethane;2-[4-methoxy-6-(propan-2-ylamino)pyridin-3-yl]acetaldehyde (2R)-1-[4-(1,3-oxazol-5-ylmethyl)piperidin-1-yl]sulfonylpyrrolidine-2-carboxylic acid 6-[4-(aziridin-1-yl)-3-fluorophenyl]-2H-pyrazolo[3,4-c]pyrazol-3-amine N-[2-[1'-(cyclopropanecarbonyl)spiro[3,5-dihydrochromeno[4,3-d]pyrimidine-2,4'-piperidine]-4-yl]ethyl]acetamide;hydrochloride 1,3-bis(ethylamino)-3,4-diphenylbutan-2-one 2-(2,4-dimethoxyphenyl)-6-propylbenzenesulfonamide (5-fluoropyridin-2-yl)-[4-[3-(triazol-1-ylmethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperazin-1-yl]methanone N-[1-(3,4-dichlorobenzoyl)piperidin-4-yl]-2-methoxybenzamide 3-[2-chloro-5-(trifluoromethyl)phenyl]propanoic acid 5-butylsulfanylthiophene-2,3,4-triamine 4-(4-fluorophenyl)-1-[2-methoxy-6-[3-(trifluoromethyl)piperidin-1-yl]pyrimidin-4-yl]pyrrolidin-2-one (2S)-2-[4-(2,5-difluorophenyl)-3H-1,3-thiazol-2-ylidene]cyclopentan-1-one 5-hydroxy-1-phenyl-N-[(Z)-pyridin-2-ylmethylideneamino]pyrazole-4-carboxamide 7-[(3-chlorothiophen-2-yl)methyl]-1',3-dimethylspiro[5,6,8,8a-tetrahydro-[1,3]oxazolo[3,4-a]pyrazine-1,4'-piperidine] N-[(1S,2R)-2-hydroxycyclopentyl]-7-(methoxyamino)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide 1-(2,5-difluorophenyl)-3-[4-methyl-6-oxo-2-(pyridin-2-ylmethoxy)pyrimidin-1-yl]urea (2R)-1,1,1-trifluoro-3-[4-(5-methylsulfonylindazol-1-yl)pyrimidin-2-yl]propan-2-ol 1-[(2,5-dimethylfuran-3-carbonyl)amino]-N-[1-(3,4-dihydro-2H-chromene-2-carbonylamino)cyclohexanecarbonyl]cyclopropane-1-carboxamide 5-(1,3-benzodioxol-5-yloxymethyl)-4-ethyl-1,2-oxazole 2-[6-(4-fluorophenyl)-7-methylsulfonylimidazo[1,2-b]pyridazin-3-yl]-5-methylphenol 6-chloro-N-methyl-2-propan-2-ylpyridine-3-carboxamide 6-(2,3-dihydroxypropyl)-4,5,7,8-tetrahydrothieno[2,3-d]azepine-2-carboxylic acid 2,2-bis[3-chloro-4-(trifluoromethoxy)phenyl]butanedioic acid 2-methoxy-6-[[2-(4,5,6,7-tetrahydroindazol-1-yl)pyridin-3-yl]sulfamoyl]benzoic acid (1R)-2,2,2-trifluoro-1-[2-methoxy-4-(4-propan-2-ylphenyl)phenyl]ethanamine 6-[(3S)-3-aminopiperidine-1-carbonyl]-4H-1,4-benzoxazin-3-one 4-[3,5-bis(trifluoromethyl)anilino]-6-oxo-2-pyrrolidin-1-yl-1H-pyrimidine-5-carbonitrile 5-(2,6-dichlorophenyl)pyridine-3-thiol;methanol (4aR)-9a-methyl-2,3,4,9-tetrahydropyrido[3,2-b]indole N-(4-azidosulfonylphenyl)propane-1-sulfonamide 5-chloro-4-[(2,6-difluoro-3-methoxyphenyl)methylamino]-1H-pyrimidin-6-one 2-[1-[1-(4-methylphenyl)ethenyl]azetidine-3-carbonyl]benzonitrile 4-(2,3-dihydroindol-1-yl)-7H-pyrrolo[2,3-d]pyrimidine 2-chloro-4,5-difluoro-N,N-dimethylbenzamide N-[2-(dimethylamino)ethyl]-6,7-difluoro-4,5-dioxobenzo[b][1,8]naphthyridine-3-carboxamide 7-(1,3,4-oxadiazol-2-yl)chromene-4,6-dione [4-[1-(2,3,5,6-tetrafluorophenyl)ethoxy]phenyl]urea 1-[2-(3,4-difluorophenyl)morpholine-4-carbonyl]cyclopropane-1-carbonitrile N-[5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1,7-naphthyridin-8-yl]azetidine-3-carboxamide 2-[(3R)-2,6-dioxopiperidin-3-yl]-5-[(E)-1-morpholin-4-ylbut-2-en-2-yl]isoindole-1,3-dione 2-[N-(2,6-dibromopyridin-4-yl)-4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]anilino]phenol 6-chloro-7-[5-fluoro-2,3-di(propan-2-yl)phenoxy]-2-methyl-2H-chromene 1-[6-[(4aS,8aR)-2,3,4a,5,7,8,8a-octahydropyrano[3,4-b]pyrazine-1-carbonyl]-9H-fluoren-2-yl]pyrazole-3-carboxamide;formic acid (1S)-2-[(5R,6S)-3-fluoro-6-[4-[(4-methylphenyl)methoxy]phenyl]-7-oxo-2,6-diazaspiro[3.4]octan-2-yl]cyclopentane-1-carboxamide N-[5-(6,7-dihydroquinoline-3-carbonyl)pyridin-2-yl]cyclohexanecarboxamide (Z)-4-[[5-tert-butyl-2-[4-[(E,3R)-1-(4-ethoxyphenyl)sulfanylpent-1-enyl]phenoxy]phenyl]methylideneamino]oxycarbonyl-2,3-dihydropyrano[3,2-b]pyridine-4-carboxylic acid 1-(2,4-dichloro-3-methylphenyl)-N-[2-oxo-5-(pyridine-3-carbonylamino)pentanoyl]cyclopropane-1-carboxamide N-[(2R)-1,3-dihydroxypropan-2-yl]-7-fluoro-4-oxo-5H-pyrazolo[4,3-c]quinoline-2-carboxamide N-[1-(4-oxobutyl)-2,3-dihydroinden-1-yl]methanesulfonamide N-(3-methylbutyl)-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-4-carboxamide 6-[(1S)-2-ethylsulfonylcyclopentanecarbonyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-benzyl-6,7-dimethyl-1,2,3,4-tetrahydroquinoxaline-5-carboxamide N-(2,4-dichlorophenyl)-5-[1-[[6-oxo-4-(trifluoromethyl)-1H-pyrimidin-2-yl]sulfanylmethyl]pyrazol-4-yl]furan-2-carboxamide [(4S)-4-azido-3,7-diazabicyclo[2.2.1]heptan-7-yl]-phenylmethanone N-(3-nitrophenyl)-N-(1,2,4-triazol-4-yl)ethenesulfonamide 5-amino-3-(1,3-benzothiazol-2-yl)chromene-4-thione 2-[4-[3-(1H-imidazol-5-yl)piperidin-1-yl]pyrimidin-2-yl]-5,6-dihydro-4H-thieno[2,3-c]pyrrole 5-bromo-4-ethyl-2-(1H-imidazol-2-yl)-1H-pyrimidin-6-one 1-[4-[1-(2,6-dimethylphenyl)imidazol-4-yl]pyrazol-1-yl]ethanone;hydrochloride 2-[3,5-dichloro-N-[(4-nitrophenyl)methyl]anilino]acetonitrile 7-chloro-1,4-dioxospiro[3H-pyrimido[5,4-e][1,2,4]triazine-2,1'-cyclohexane]-8-one 2-[(1S)-1-[(3R)-piperidin-3-yl]ethoxy]benzaldehyde (3S,4R)-1-[2-(3,4-dimethoxyphenyl)-5-methyl-7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-hydroxypiperidine-3-carboxamide 4-(1,3,2-benzodioxaborol-6-yl)aniline 2-[4,5-dimethyl-1-(4-nitrophenyl)imidazol-2-yl]-N,N-dipropylethanamine 4-(1,5-dimethylpyrazole-3-carbonyl)spiro[1H-quinoxaline-2,4'-piperidine]-6-carboxamide 3-hydroxy-1-[4-(2-phenylethyl)piperidine-4-carbonyl]pyrrolidine-3-carboxamide;dihydrochloride N-[2-methylsulfonyl-6-(trifluoromethoxy)phenyl]formamide 7,8-dichloro-2H-thiochromene-3-carboxylic acid 2-tert-butyl-6-[(4,5-dimethylfuran-2-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-(dimethylamino)-N-[2-fluoro-5-[3-(piperidin-1-ylmethyl)phenoxy]phenyl]butanamide 5-(2,5-dimethoxyphenyl)sulfonyl-2-[4-(pyridine-3-carbonyl)piperazin-1-yl]-N-(2-thiophen-2-ylethyl)benzamide 1-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-3-phenylthiourea 2-azido-N,N-diethylpyridine-4-carboxamide 2,4-dimethyl-5-propan-2-yl-1,3-thiazole;ethane 2-(1,3-benzothiazol-2-yl)-N-[4-(5-tert-butylthiophen-2-yl)-2-methoxyphenyl]benzamide N-(2,3-dihydro-1H-inden-4-yl)-6-methoxy-2-phenylquinoline-7-carboxamide 2-bromo-5-[[(2S)-1,4-dioxan-2-yl]methoxy]benzaldehyde 1-[3-(5,6-dimethylimidazo[2,1-b][1,3]thiazol-2-yl)phenyl]ethanone 3-(2,5-dimethylphenyl)pentane-1,4-diol (1-azidosulfanyl-2,3,4,5-tetramethoxycyclopenta-2,4-dien-1-yl)benzene 4-[6-(1-aminocyclopropyl)pyridin-2-yl]oxybenzenethiol 1-azidooxy-2,4,5,6-tetrachloronaphthalene 1-[(3S,4R)-2-oxo-4-(2-phenylethylamino)piperidin-1-yl]-4-[4-(trifluoromethoxy)phenoxy]butan-2-one 1-[(4R)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-yl]-3-(1,3-thiazol-2-yl)propan-1-one 1-[(2R,5S)-3-hydroxy-4,5-dimethylheptan-2-yl]pyridin-2-one (3R,4S)-1-[[1-(3,5-difluorophenyl)pyrazol-4-yl]methyl]-N,N-bis(pyridin-2-ylmethyl)-3-(quinolin-3-ylmethoxymethyl)piperidine-4-carboxamide 2-[(Z)-3,5-dimethylhex-2-enyl]quinoxaline (1R)-3,7-bis[2-(diethylaminomethylideneamino)ethoxy]-8-oxocyclooctane-1-carboxylic acid 1,1-bis(3,4-dihydronaphthalen-2-yl)propan-2-one (5R,6S)-3-methyl-1-[4-[[(3S)-oxolan-3-yl]oxymethyl]phenyl]-5-pyridin-2-yl-5,6-dihydro-2H-azepino[4,5-b]indole 6-[(2R)-2,4-dimethylpentoxy]-3-methylquinazolin-4-one (2S)-4-phenylmethoxybutan-2-amine N-[(4,5-dimethoxycyclohexa-1,3-dien-1-yl)methyl]naphthalene-2-carboxamide 2-[(3R)-3-methoxypyrrolidin-1-yl]-4-(1,1,1-trifluorobutan-2-ylamino)pyrimidine-5-carboxamide 4-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-6-one 1-[2,3-bis(ethenyl)phenyl]butan-1-one 2-tert-butyl-3,5-diphenylfluoren-1-one 2-[4,5-bis(chloromethyl)imidazol-1-yl]benzoic acid [(2S,4R)-1-(cyclohexanecarbonyl)-4-methoxypyrrolidin-2-yl]-morpholin-4-ylmethanone 7-[(2S,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-purin-6-one 3-[4-(2-methyl-5,6,7,8-tetrahydroquinolin-3-yl)-1H-benzimidazol-2-yl]-5-pyrimidin-5-yl-1H-pyrazolo[3,4-c]pyridine 3-[(4S,5R)-2-amino-1-ethyl-3-methylidene-6-oxo-4-phenylpiperidin-4-yl]-N-butan-2-ylpropanehydrazide 4-[5-(aminomethyl)pyridin-3-yl]-2,6-difluorobenzoic acid [2-[5-(3,4-dihydro-1H-isoquinoline-2-carbonyl)thiophen-2-yl]phenyl]urea 2-(3-hydroxypropyl)-6,8-dimethoxypyrimido[4,5-c]isoquinolin-5-one [3-(1,1-dioxo-3a,4,5,6,7,7a-hexahydroinden-2-yl)-1H-indol-5-yl]methanol 1-azidooxy-2,3-dibromobenzene (Z)-3-amino-N'-[(5,6-dichloro-2,1,3-benzothiadiazol-4-yl)methyl]-N'-ethylbut-2-enimidamide 2-[5-(4,5-dihydropyrimidin-4-yl)pyridin-3-yl]-6-methylpyridine N-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-methoxy-1,2,4-thiadiazol-3-amine N-[4-[2-(cyclohexylamino)ethyl]phenyl]acetamide 2-chloro-N-(4-fluorophenyl)-1,3-dioxoisoindole-5-carboxamide;ethane 3-(furan-2-yl)-1-phenyl-5H-pyrazolo[4,3-c]quinolin-4-one 3-(4,5-dihydro-1H-imidazol-2-yl)-1-benzofuran-7-amine 3-(2-aminoethyl)-1H-indole-5-carbonitrile;6-methoxy-3,4-dihydro-2H-chromene 2-(4-phenoxypyridine-3-carbonyl)-1,3-thiazole-5-carboxylic acid 1-[6-(methoxymethyl)-3,5-dihydro-2H-4,1-benzoxazepin-7-yl]ethanone 2-(hydroxymethyl)pyrrolidine-1,3-dicarboxylic acid;N-[5-[4-fluoro-2-(trifluoromethoxy)phenyl]-6-methanimidoylpyridin-3-yl]methanesulfinamide 2-aminooxy-3-[2-(1,1-difluoroethyl)phenyl]propanoic acid 2-[5-bromo-3-(difluoromethyl)pyrazol-1-yl]-5-nitrobenzoic acid 2-hydroxy-N'-[(E)-1H-indol-6-ylmethylideneamino]benzohydrazide 2-[3-aminopropyl(ethyl)carbamoyl]benzenesulfonic acid 1-(4-aminophenyl)-3,5-dimethylhexan-1-one 2-amino-6,7-dimethoxyquinoline-3-carbonitrile;ethane 4-amino-6-[(4-methoxyphenyl)methyl]-1H-1,3,5-triazin-2-one 3-(5-methyl-4H-1,2,4-triazin-3-yl)pyridine N-[(1S)-1-[5-fluoro-2,3-dihydroindol-1-yl-8-methoxy-4-(trideuteriomethyl)quinolin-6-yl]ethyl]pyrimidine-5-carboxamide 2-(4-but-3-enylphenyl)benzonitrile 5-N,1,3-trimethyl-2-N-phenylimidazo[4,5-b]pyridine-2,5-diamine (3Z,4E)-4-ethylidene-5-methoxycarbonyl-2-[methyl(propan-2-ylsulfonyl)amino]-6-oxo-1H-pyridine-3-carboxylic acid 3-(1H-indol-5-yl)-N-[(4-methoxyphenyl)methyl]-2-[4-[2-(oxan-4-ylamino)pyridin-3-yl]-2,6-di(propan-2-ylidene)cyclohexa-1,3-dien-1-yl]prop-2-enamide 2-[5-(3,4-difluorophenyl)-1H-pyrrol-3-yl]acetic acid N-(1-benzofuran-3-yl)-3-[5-ethoxy-2-[[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]amino]phenyl]pentanamide 4-[2-azido-1-(diethylamino)propyl]phenol N-[5-tert-butyl-2-(5,6,7,8-tetrahydronaphthalen-1-yl)pyrazol-3-yl]-4-methoxybenzamide 1-[4-(3-methylcyclopenten-1-yl)phenyl]pyrazole 5-[1-(2,6-difluorophenyl)piperidin-4-yl]oxyspiro[2H-indole-3,3'-pyrrolidine] 5-[2,4-bis(phenylmethoxy)phenyl]imidazolidine-2,4-dione 4-[(3-aminopyridin-2-yl)amino]-6-[[[2-(dimethylamino)acetyl]amino]methyl]pyridazine-3-carboxamide 2-N,4-dimethyl-1-N-(3-naphthalen-2-ylpropyl)pentane-1,2-diamine 4-[(E)-1,2-diphenylethenyl]pyrimidin-5-ol 2,5-difluoro-4-[2-(1H-indol-3-yl)ethyl]phenol 4-[3,5-bis(2,6-dioxopiperidin-3-yl)-1,2,4-triazol-1-yl]butanoic acid 3-[3-[4-methoxy-2-[(3E,5Z)-6-morpholin-4-ylhepta-1,3,5-trien-3-yl]phenyl]-4-oxochromen-7-yl]sulfanylpropanenitrile 7-[3-(4,5-dihydro-1H-imidazol-2-ylsulfanyl)propyl]pyrido[2,3-b]pyrazine 6-[(3E,5Z)-hepta-1,3,5-trien-4-yl]pyridine-2-carbonitrile 5-(2,4-difluorophenyl)-N-[3-methoxy-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)pyrrolidin-3-yl]furan-2-carboxamide 5-hydroxy-6-[1-(4-methylpiperazine-1-carbonyl)cyclopentyl]oxyisoindole-1,3-dione 2-[2,6-di(propan-2-yl)phenyl]-1-propan-2-ylisoquinolin-2-ium 3-ethyl-2-methylhexane;4-[(4-fluorophenyl)carbamothioylamino]cyclohepta-1,3-diene-1-carboxylic acid 2-methyl-1-(3,4,5-trimethoxyphenyl)imidazole 4-benzyl-1,3-bis[2-(methylamino)ethyl]imidazolidin-2-one;ethane 5-bromo-2,4-ditert-butyl-6-chloropyrimidine 5-[2-(3,4-dichlorophenyl)ethylamino]sulfanyl-3-methylpyridine-2-carboxylic acid N-[(1R,2S)-2-hydroxycyclohexyl]-4,6-dimethoxypyrimidine-5-carboxamide N-[1-(2,4-dihydroxyphenyl)ethylideneamino]pyridine-3-carboxamide N-[3-(2,4-difluorophenyl)propyl]-5-(6-methylpyrazolo[1,5-a]pyrimidin-3-yl)thiophene-2-carboxamide 4-methyl-N-[(Z)-1-[2-[2-(trifluoromethoxy)phenyl]cyclopropen-1-yl]propylideneamino]aniline 4-[(2,3-difluorophenyl)methoxy]-N'-hydroxypyridine-2-carboximidamide ethane;2-[[4-(4-propylcyclohexyl)phenyl]methoxy]guanidine N-(4,6-dimethylpyrimidin-2-yl)sulfanylhexanamide 2-[6,8-dichloro-4-(4-chlorophenyl)-3-methyl-1-propanoyl-7-nitronaphthalen-2-yl]acetic acid N-[(5R)-3,4-dihydroxycyclohexyl]-2-(5-methoxy-3-oxo-1H-isoindol-2-yl)acetamide [4-[(E)-3,3,3-trifluoroprop-1-enyl]phenyl]methanamine 4-chloro-7-(1H-pyrazol-5-yl)benzo[g]isoquinoline 3-(5-bromopyridine-2-carbonyl)imidazolidine-1,4-dione 6-chloro-2-[1-(3-ethylphenyl)-2,2,4-trimethylpentyl]-3-methoxyaniline N-[(E)-1H-indol-6-ylmethylideneamino]-2-(5-oxotetrazol-1-ium-1-yl)acetamide N-[5-(4,6-dimethoxypyrimidin-2-yl)oxypyridin-2-yl]-2-(difluoromethoxy)-3-(1,1-dioxothiolan-3-yl)benzamide 1-[4-(4-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole ethane;2-ethenylcyclohexane-1,3-diamine;N-(2-methoxyethyl)-4-[3-(trifluoromethyl)pyridin-2-yl]aniline 1-[(2R,3S)-2-[4-methyl-6-(1H-pyrazol-5-ylamino)pyrimidin-2-yl]oxan-3-yl]ethanol 4-[2-(6,7-dimethoxyquinolin-4-yl)oxyethyl]piperidine-1-carboxylic acid 1-[2-methyl-4-[(3E)-5,6,7-trimethoxy-3-methylidenehepta-1,4,6-trien-2-yl]phenyl]ethanone (2-methyl-1,3-benzothiazol-5-yl)-[4-(pyridin-4-ylmethoxy)piperidin-1-yl]methanone 5-chloro-6-(4-chlorophenyl)pyridine-2,3-diamine;hydrochloride 4-[3-bromo-1,2-bis(ethenyl)pyrrol-3-yl]pyrimidin-5-ol 5-[1-cyclopropyl-2-(7H-purin-6-ylamino)ethyl]-3H-1,3,4-oxadiazole-2-thione 6-[5-(4,4-difluoropiperidine-1-carbonyl)pyridin-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one 1-[(2S)-butan-2-yl]pyrazolo[3,4-c]quinolin-4-amine 3-[1-methyl-2-oxo-3-[4-(2,2,2-trifluoroethoxy)phenyl]imidazolidin-4-yl]benzoic acid 2-benzylsulfanyl-N'-hydroxy-6,7-dihydro-4H-thieno[3,2-c]pyran-5-carboximidamide 2-(1,3-dioxoisoindol-2-yl)-N-[5-[4-[(2S)-1-hydroxypropan-2-yl]oxyphenyl]sulfanyl-3H-1,3-thiazol-2-ylidene]acetamide N-[2,6-bis(2,3,4,5,6-pentamethylphenyl)-5H-benzimidazol-5-id-7-yl]acetamide;chloroform;platinum 2-[4-(6,7-dihydrothieno[3,2-c]pyridin-5-yl)piperidin-1-yl]-N-[3-methoxy-4-(4-morpholin-4-ylbutanoylamino)phenyl]acetamide;2,2,2-trifluoroacetic acid 4-(4-aminophenyl)-N-[2,5-dimethyl-3-oxo-1-propan-2-yl-6-(trifluoromethyl)pyridazin-4-yl]piperazine-1-carboxamide 4-[[2-(3,5-dimethoxy-2-methylphenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]cyclohexan-1-ol N-[5-(2-cyclobutyloxypyridin-4-yl)-4-methyl-1,3-thiazol-2-yl]acetamide [2-(oxolan-3-yloxy)phenyl]phosphane 1-(5-bromo-4-fluoropyridin-2-yl)-6-methylsulfonyl-7,8-dihydro-6H-quinazoline-2,4-dione 6-ethyl-3-[6-(4-piperidin-1-ylpiperazine-1-carbonyl)-1H-benzimidazol-2-yl]-1H-quinolin-2-one 3-fluoro-5-(1-methylpyrrole-2-carbonyl)benzonitrile (E)-2,6-dimethyl-N-[(3S)-5-methyl-4-oxohexan-3-yl]-7-phenylhept-5-enamide;2,4-dimethylpenta-1,3-diene 6-[(E)-1-bromobut-2-enyl]-8-chloro-2,3-dihydrochromen-4-one [3-(3,4-dimethoxyphenyl)-1H-pyrazol-5-yl]urea 7-(4,5-dihydrothieno[2,3-d][1]benzoxepine-2-carbonyl)-2-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-one 5-[3-(2,6-dimethylmorpholine-4-carbonyl)anilino]-1,7-naphthyridine-8-carbonitrile N-[1-(5-fluoropyridine-2-carbonyl)piperidin-3-yl]-N-[2-(1,2,4-triazol-1-yl)ethyl]methanesulfonamide 2-[(1R)-1-amino-3,4-dihydro-1H-naphthalen-2-ylidene]propanedinitrile 4-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-6,11-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene 2,6-diethyl-4-[3-fluoro-5-(trifluoromethoxy)phenyl]-1H-imidazo[4,5-c]pyridine 5-amino-7-[(2,3,4-trifluorophenyl)methyl]-9H-pyrrolo[3,4-b]quinoline-1,8-diol N-[(2E)-4-[bis(4-methoxyphenyl)-phenylmethoxy]penta-2,4-dienyl]methanimine 3-methylsulfonyl-5,6,7,8-tetrahydroquinoline 4-fluoro-N-methylnaphthalene-2-sulfinamide 2-(4-chlorophenyl)-N-[4-(3,4-dihydroquinoline-8-carbonylamino)phenyl]benzamide N-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-7-yl)pyridine-4-carboxamide 2-[5-(4-chlorophenyl)-3-[hydroxy-(1-methylcyclopentyl)methylidene]piperidin-1-yl]sulfonylbenzonitrile 4-[3-(dimethylamino)propoxy]-1,2,5,6-tetrahydropyrrolo[2,1-c][1,4]benzothiazepine-9-carboxamide 1-(6-chloronaphthalene-2-carbonyl)azetidine-3-carboxylic acid 2-[4-amino-6-(3,5-difluoroanilino)pyrimidine-5-carboximidoyl]phenol 4-[3-(3,4-dichlorophenyl)-3-hydroxypropyl]pyrrolidine-2,3-dione [4-[3-[6-(hydroxymethyl)pyridin-2-yl]-1,2,4-oxadiazol-5-yl]cyclohexyl]azanide 5-[4,6-bis(trichloromethyl)-1,3,5-triazin-2-yl]-2H-tetrazole N-(2,4-dimethoxyphenyl)-5-[3-[4-(trifluoromethyl)benzoyl]azetidine-1-carbonyl]thiophene-2-sulfonamide 1-[2,3-dimethoxy-4-(trifluoromethyl)phenyl]sulfonylpyrrolidine 2-[5-(1,3-benzodioxol-4-yl)pyridin-3-yl]-4,4-dimethyl-5H-1,3-oxazole N-[2-(N-hexadecylanilino)ethyl]acetamide 6-methoxycarbonyl-3,4,5,7-tetrahydro-1H-[1,2]thiazolo[5,4-b]pyridine-8-carboxylic acid 5-[3,5-bis(trifluoromethyl)phenyl]-4,6-dimethylbenzene-1,2,3-triol 3-[6-azidooxy-2,3-dichloro-4-(1-hydroxybutan-2-yl)phenoxy]propanenitrile 1-(3-ethoxyphenyl)-2,4,6-trimethylpyridine-3-carbonitrile 2-[azido(nitro)methyl]pyridine N'-[4,5-bis(4-fluorophenyl)imidazol-1-yl]-4,4-dimethylhexanehydrazide 1-[(3R)-5,6-dichloro-3-(4-fluorophenyl)-2-methyl-2H-1,3-benzothiazol-4-yl]ethanone N-ethyl-3-fluoro-2,5-dimethoxy-6-[3-[(E)-N'-nitrocarbamimidoyl]phenyl]sulfanylbenzamide 4-(2-ethylbutyl)-N,2,6-trimethylaniline 2-[(3R)-piperidin-3-yl]-3,5-bis[4-(trifluoromethoxy)phenyl]benzamide 2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)phenol 3-azidosulfanyl-1-(benzylamino)propane-2,2-diol (Z)-3-amino-2-[6-methoxy-5-(5-methylpyridine-2-carbonyl)pyrimidin-4-yl]prop-2-enamide N-(2-tert-butylphenyl)benzenesulfonamide 4-amino-N'-[[1-(2,5-dichlorophenyl)sulfonylazepan-3-yl]methyl]benzenecarboximidamide;hydrochloride 3-benzyl-N,N-dimethyl-2-propanoylaniline 2,7-dimethyl-5-(thiophen-2-ylmethyl)-5,8-dihydroimidazo[1,2-a]pyrimidine;2,2,2-trifluoroacetic acid 1-[3-(4-chlorophenyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carbonyl]cyclopentane-1-carboxylic acid [4-methyl-1-(3-methylbutyl)cyclohepta-2,4,6-trien-1-yl]-phenylmethanone 1-(5,7,12,20,23,26-hexaoxaheptacyclo[11.10.0.02,10.03,8.04,22.014,22.016,21]tricosa-1(13),2(10),3(8),6,9,11,14,16(24)-octaen-19-yl)ethanone 3-(4-chlorophenyl)sulfanyl-6-(6-methyl-1H-indol-2-yl)pyrazin-2-amine (E)-3-cyclopentyl-N-[[6-[1-[[4-fluoro-5-methoxy-2-[2-(methylamino)ethoxy]phenyl]methylcarbamoyl]cyclopropyl]pyridazin-3-yl]methyl]-N,3-dimethylbut-2-enamide 2-amino-6-[(3R)-1-(4-fluorobenzoyl)piperidin-3-yl]-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one [(1R)-3,4-dihydro-2H-naphthalen-1-yl]-[(5S)-7-methyl-5-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methanone 5-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-2-[(E)-2-phenylethenyl]pyran-4-one 2-[(E)-(4,5-dihydro-1H-imidazol-2-ylhydrazinylidene)methyl]-6-ethoxyphenol 2-[(Z)-3-methyliminopent-1-enyl]benzenethiol 4-[4,6-bis(2-methoxyphenyl)-1,3,5-triazin-2-yl]-2H-naphthalen-2-ide;uranium(2+) 4-[[2,3-dihydro-1H-inden-5-yl(methyl)amino]methyl]cyclohexan-1-amine (5E)-2-(4-ethoxyphenyl)imino-5-[(1,3,2,4,7-pentamethylquinolin-6-yl)methylidene]-1,3-thiazolidin-4-one N-(4,5-dimethylpyridazin-3-yl)-2-[4-[1H-indol-2-yl(sulfanyl)methoxy]phenyl]acetamide N-(5-bromo-1H-pyrrolo[2,3-b]pyridin-4-yl)carbamate 1-methyl-3-(3-prop-2-ynoxyphenyl)pyrazole (2Z,4E)-4-amino-2-[5-(methoxymethyl)pyridin-3-yl]hexa-2,4-dienamide 4-[1,3-bis(2-chlorophenyl)propan-2-yloxy]-3-propan-2-ylideneoxolane 1-(4-bromophenyl)ethyl-dimethylsulfanium 3-[3-(2,6-dichloroanilino)-4-oxocyclohexa-1,5-dien-1-yl]-7-fluoro-1H-indole-2-carboxamide 4-[3-[(3,5-difluorophenyl)methyl]-1H-indol-2-yl]-N-(pyridin-3-ylmethyl)benzenesulfonamide 2-[4-chloro-3,5-difluoro-7-(trifluoromethyl)dibenzothiophen-1-yl]-1-cyclopropylidenebutan-2-ol 5-[2,3-dihydroxypropyl(propanoyl)amino]naphthalene-2-sulfonic acid N-ethenyl-3,5-difluorobenzamide 1-[1,3-bis(2-ethoxyphenyl)propan-2-yl]imidazole;dihydrobromide 2-azido-N,N-dimethylquinoline-4-carboxamide (5S,7R)-N-[2-(3,4-dimethoxyphenyl)ethyl]-7-(trifluoromethyl)-5-(3,4,5-trimethoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide N-[6-(4-propan-2-ylpiperazine-1-carbonyl)pyridin-3-yl]acetamide [(4aS,8R)-4-hydroxy-2-[6-(trifluoromethyl)pyrimidin-4-yl]-1,3,4a,5,7,8,8a-octahydropyrrolo[3,4-d]azepin-6-yl]-(5-methylthiophen-2-yl)methanone 1-[2-(5-chloro-4H-cyclopenta[d]imidazol-2-yl)pyrrolidin-1-yl]butan-1-one 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidin-2-ide;palladium(2+) 2-[6-[3,4-dihydro-1H-isoquinolin-2-yl(methyl)amino]pyrazin-2-yl]-5-(2-fluoropropan-2-yloxy)phenol [(2R,3S)-4-hydroxy-2-phenyloxolan-3-yl]oxymethylphosphonic acid 2-chloro-N,3-dimethyl-4-(1-phenylethyl)aniline;ethane (1-methyl-9-oxa-2,3,4,5-tetrahydropyrido[2,3-f][1,8]naphthyridin-7-yl)-morpholin-4-ylmethanone;2,2,2-trifluoroacetic acid [2-(4-methoxyphenyl)-3,5-dihydropyrido[3,2-e][1,2,4]triazin-4-yl]hydrazine N-methyl-2,2-diphenyl-N-(2-pyridin-4-ylethyl)propanamide 7-bromo-N,2-dimethylthieno[3,2-b]pyridine-4-carboxamide N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-N'-(N'-propanoylcarbamimidoyl)methanimidamide 6-[(4,5-dichloro-2-hydroxyphenyl)methyl]-2-(trifluoromethyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 1-[(2-methoxyphenyl)methyl]indole-7-carboxamide N-[5-cyano-4-(2,4-difluorophenyl)pyridin-2-yl]acetamide N-[(3,5-difluorophenyl)methyl]-2-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-ylidene]acetamide 3-(2,3,5,6-tetrafluorophenoxy)pentanal N-(4,5-dimethyl-2-phenyldiazenylphenyl)-2-methoxy-N-prop-2-enylacetamide 2-[[1-(4-bromobenzoyl)piperidin-3-yl]methoxy]-6-ethylpyridine-3-carbonitrile 2-hydroxy-5,6-di(propan-2-yloxy)-3H-isoindol-1-one 4-[3-(1,2,3,6-tetrahydropyridin-4-yl)pyrazol-1-yl]piperidine N'-[(1R)-5,7-difluorospiro[1H-2-benzofuran-3,4'-piperidine]-1'-yl]methanediamine 2-[2-(furan-2-yl)ethylamino]-4,8-dimethoxypyrido[3,4-d]pyrimidine-6-carboxylic acid 1-[4-(6,11-dihydropyrido[3,2-c][1]benzazepine-5-carbonyl)-2,3-dimethylphenyl]ethanone 2-[5-chloro-1-(4-methylpentan-3-yl)-6-oxopyrimidin-2-yl]sulfanyl-N-(2,4-dimethoxyphenyl)acetamide 1-(4-azidobutan-2-yl)-N,N-diphenylpiperidin-4-amine 3-bromo-6-methoxy-2-(4-pyridin-3-ylphenyl)quinoxaline 2-[[4-chloro-3,5-bis(trifluoromethyl)phenyl]carbamothioylamino]-N-ethoxy-3-(trifluoromethyl)benzamide 2-amino-4,6-dimethoxybenzimidazole-1-carboxylate 3,5-diamino-2-[[6-(3-chlorophenyl)pyridin-3-yl]methyl]benzoic acid 6-chloro-N-[(4R)-3-cyano-1-methyl-4H-pyrazolo[3,4-b]indol-5-ylidene]-2-(trifluoromethoxy)cyclohexa-2,4-diene-1-carboxamide N-[6,8-bis(4-methylphenyl)-2-oxo-1H-purin-9-ium-9-ylidene]acetamide [(1E,3Z)-1-aminohexa-1,3,5-trien-2-yl]sulfonylbenzene N-benzyl-2-(hydroxyiminomethyl)prop-1-en-1-amine 2-fluoro-N-[(4R)-2,5,6-trimethyl-4-propan-2-ylideneheptan-3-yl]benzenesulfonamide 4-cyclobutyl-1-[(2,5-difluorophenyl)methoxy]-6-[3-(trifluoromethyl)pyrrolidin-1-yl]isoquinoline N-[1,2,3,5]tetrahydro-[1,3]thiazolo[5,4-c][1,4]benzoxazin-7-yl(1H-pyrrolo[2,3-b]pyridin-4-yl)methanimine 2-[4-(5-bromo-1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-1H-pyridin-4-one 6-(4-chlorophenyl)-9-methoxybenzo[h][1,2]benzoxaphosphinine 2-[6-(methoxymethyl)pyrimidin-4-yl]-5,7-dihydropyrrolo[3,4-b]pyridine N-[(2S)-1-amino-4-methylsulfanylbutan-2-yl]-1,3-dioxoisoindole-5-carboxamide (3R)-N-[4-cyano-2-(4,5-dihydro-1H-imidazol-2-ylsulfanylmethyl)phenyl]-1-[1-(cyclopropanecarbonylamino)ethenyl]pyrrolidine-3-carboxamide 5-bromo-2-methylimino-1-oxo-4,7-diphenyl-3H-s-indacene-3a-carbonitrile N-(furan-2-ylmethyl)-4,7-dioxo-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 2-chloro-4-methyl-3,5-bis(methylperoxy)benzonitrile 3-[1-aminoethyl(methyl)carbamoyl]-6-chloro-N,2-dimethoxybenzamide 2-[2-(1,3-thiazol-4-yl)butylsulfanyl]pyrimidine-5-carboxamide 5-[4-[(1S)-1-(2-fluoro-5-methoxyphenyl)ethyl]piperazin-1-yl]-3,4-dihydro-1H-quinolin-2-one 1-benzyl-4-(pyridin-3-ylamino)-7H-pyrazolo[3,4-b]pyridin-6-one 1-azido-4,5-dichloro-2-methoxy-3-(trifluoromethyl)benzene N-azido-3-(trifluoromethoxy)benzamide 3-[2-methoxyethyl(propan-2-yl)amino]-N'-methylpyridine-4-carboximidamide 6-[(3,4-dichlorophenyl)methyl]-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile 4-[5-[4-(6-hydroxyheptoxy)phenyl]thiophen-2-yl]phenol N-(2,4-dimethylphenyl)-3H-benzimidazole-5-carboxamide [(2E,4Z)-3-bromohepta-2,4,6-trien-2-yl]oxybenzene N-[(4S,6R)-6-[1-(4-fluorophenyl)indazol-5-yl]-2-methoxycarbonyl-5-oxo-1-phenyloctanoyl]piperazine-2-carboxamide 4-[2,3-bis(methoxycarbonyl)phenyl]benzoic acid 2-[(2-butanoyl-5-methylsulfonylindol-1-yl)amino]propanal;ethane 5-[1-azido-3,4-bis(difluoromethyl)cyclohexa-2,4-dien-1-yl]-1H-indole N-[4-(6,7-dimethoxyquinolin-4-yl)oxy-2-fluorophenyl]-1-(3-fluorophenyl)-2-oxo-5-pyridin-3-ylpyrrolidine-3-carboxamide N-(3,4,6,7,8,8a-hexahydro-2H-pyrrolo[1,2-a]pyrazin-1-yl)-1,7-naphthyridine-6-carboxamide;dihydrochloride 1-[4-(3,6-diazabicyclo[3.2.0]heptan-6-yl)phenyl]-N-[3-[3-fluoro-5-methoxy-4-(1H-imidazole-5-carbonylamino)phenoxy]propyl]piperidine-4-carboxamide [(3E,5Z)-6-fluorohexa-1,3,5-trien-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]methanone 3-[[4,5-bis(4-chlorophenyl)-1H-imidazole-2-carbonyl]amino]propanoic acid 3-ethyl-6-[[2-(3-fluorophenyl)sulfonylpyrrolidine-1-carbonyl]amino]pyridine-2-carboxylic acid N-[(4-nitrophenyl)methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 3-(1-hydroxyhexyl)-2,3-dihydrochromen-4-one 2-[4-amino-3,5-dichloro-N-(2-ethylhexyl)anilino]acetic acid;hydrochloride 2-(N-butyl-4-chloroanilino)acetic acid 5-[6-methoxy-3-(1H-pyrazol-4-yl)quinolin-4-yl]oxypyridine-2-carboxamide 4-[3-(1,3-benzoxazol-2-yl)phenyl]-5H-benzo[c]phenanthridine 5-[1-(3,4-difluorophenyl)ethyl]-2H-tetrazole N-[(5E)-2-methyl-4-oxo-5-[(Z,3Z)-3-propylidenehept-1-enyl]iminothiophen-2-yl]acetamide N-[4,5-diethoxy-2-(methylamino)phenyl]acetamide 1-(6-bromo-3,4-dihydro-2H-chromen-8-yl)piperidine 3-(methoxyamino)-4,7-dioxo-1H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid N-butyl-5,7-dimethoxyquinazolin-2-amine 3-[4-(2,6-dimethylpyrimidin-4-yl)piperazin-1-yl]oxolan-2-one N-[(4E,5Z)-4-ethylidenehepta-1,5-dien-2-yl]-3-methoxybenzamide 1-[4,6-bis(2,2-dimethylpropoxy)pyrimidin-5-yl]ethanone 4-[(8aS)-1,3-dioxo-6-pyrazol-1-yl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-2-yl]benzonitrile 4-[2-(1,3-benzoxazol-2-yl)benzoyl]oxy-2,5,6-trimethylbenzenesulfonic acid N-(4-chlorophenyl)sulfanyl-2,6-dimethoxybenzamide 4-[1-aminobutyl(propan-2-yl)carbamoyl]-N-phenylcyclohexane-1-carboxamide;methanamine 5-(methanesulfonamido)-4-oxochromene-2-carboxylic acid 1-[5-methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]butan-1-one 1-(2,3-dihydro-1H-inden-2-yl)-5-fluoronaphthalene (E)-N-[1-[(4-fluorophenyl)methyl]pyrazol-3-yl]-3-(furan-2-yl)prop-2-enamide 3-(1,3-benzothiazol-2-yl)-5-(oxan-4-ylamino)piperidine-2,6-dione (6R,11bS)-7-acetyl-3-ethenylsulfanyl-6-methoxy-6,10b-dihydro-2H-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 2-(methoxymethyl)-1,3-dioxoisoindole-5-carboxylic acid 3-(4,6-diphenyl-1H-1,3,5-triazin-2-yl)aniline 1-[(4-methylcyclohexyl)methoxy]ethenylbenzene;3,7,11-trithiatetracyclo[6.3.0.02,6.010,15]undeca-1(8),2(6),9-trien-4-amine N-[2-(2,6-dichloroanilino)ethyl]-5-oxopentanamide 1-[3,5-bis(trifluoromethyl)phenyl]propan-2-one;4-(2-oxopyrrolidin-1-yl)benzonitrile N-[3-chloro-4-[(E)-2-cyclopentylethenyl]phenyl]cyclohexanimine;ethane (Z)-3-hydroxy-N-methyl-2-[3-[4-[3-(4-octoxyphenyl)propyl]piperazine-1-carbonyl]phenoxy]but-2-enamide [5-chloro-6-[(4,4,4-trifluorobutylamino)methyl]pyridin-3-yl]oxyboronic acid 5-[2-(4-cyclopropylpiperazine-1-carbonyl)thieno[3,2-b]pyridin-7-yl]oxy-N'-hydroxy-6-methylidenecyclohexa-2,4-diene-1-carboximidamide 3-(4-ethoxyphenyl)-6-(2-pyrrolidin-1-ylethylamino)-2,5-dihydropyrazolo[3,4-d]pyrimidin-4-one 4-[5-cyano-1,3-dimethyl-6-(trifluoromethoxy)benzimidazol-1-ium-2-yl]butanethioate 2-methoxy-5,7-dimethyl-N'-(1-pyridin-3-ylethenyl)pyrrolo[2,3-b]pyrazine-6-carboximidamide 2-(1,4-diazepan-1-yl)-6-(quinoline-3-carbonylamino)imidazo[1,2-a]pyridine-8-carboxamide 2-[5-bromo-1-(4-methylsulfonylphenyl)sulfonylpyrrolo[2,3-b]pyridin-3-yl]acetamide (3-azidoazetidin-1-yl)-[4-(5-chloropyridin-2-yl)phenyl]methanone 2-[5-(1,3-dioxolan-2-yl)pyridin-2-yl]pyrimidine 4-[[5-[(3,5-dimethoxyphenyl)methylsulfanyl]pyrimidin-2-yl]amino]-N-hydrazinylidenebenzenecarboximidamide 2-[[5-(1,3-benzothiazol-6-yl)-4-chlorothiophen-2-yl]sulfonylamino]acetic acid N-(diaminomethylidene)-2,3,4-trimethylbenzenesulfonamide N'-(3,4-dimethylphenyl)-2,6-dihydroxybenzenecarboximidamide 1-(2,3-dihydroindol-1-yl)-2-[2-(3-fluorophenyl)-5-(trifluoromethoxy)indol-1-yl]ethanone 3-[4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]-N-octylanilino]propanoic acid 1-[5,7-difluoro-2-(4-fluorophenyl)-3H-benzotriazol-4-yl]ethenamine N-(2,4-dimethylphenyl)-1H-indole-6-carboxamide (2Z,5R)-2-[(E)-1-(4-ethoxyphenyl)propylidenehydrazinylidene]-5-[(4-fluorophenyl)methyl]-1,3-thiazolidin-4-one (E)-N,2-dimethyl-3-[2-[4-(6-methylidenecyclohexa-1,3-dien-1-yl)phenoxy]ethoxy]prop-2-enamide N-(cyclopropylmethyl)-4-methoxy-2,5-dioxoimidazolidine-1-carboxamide;5-[(E)-3-(6-fluoroquinolin-7-yl)prop-2-enimidoyl]-4H-pyrazol-3-amine N-(4,6-dimethyl-2H-pyrazolo[3,4-c]pyrazol-3-yl)-4-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]benzamide (E)-N-tert-butylsulfanyl-1-[3-chloro-5-(trifluoromethoxy)phenyl]methanimine (Z)-[2,4-difluoro-6-methyl-3-[1-(oxan-4-yl)piperidin-4-ylidene]cyclohexa-1,5-dien-1-yl]methoxyiminomethanediol 2-amino-4,5-dichlorobenzenesulfonamide [2-(4-amino-1H-pyrrolo[3,2-c]pyridine-7-carbonyl)oxycyclopropyl]methanesulfonate N-[2-(aminomethyl)pyrimidin-5-yl]-3-chloropropanamide 2-(4-fluorophenyl)-5,6,7,8-tetrahydropyrazolo[1,5-a][1,3]diazepine;hydrochloride 3-(2,6-diphenylpyrimidin-4-yl)oxypropanoic acid 2-(N-(3-ethoxy-3-oxopropanoyl)anilino)-2-methylpropanoic acid 1-(4,5-dimethyl-6-oxo-2-pyridin-3-yl-1H-pyrimidin-5-yl)propane-1,3-dione N-[2-(3-chlorophenyl)ethyl]-2,4-dimethylidenepyrrolidine-1-sulfonamide N-[(Z)-(4-hydroxyphenyl)methylideneamino]-2-morpholin-4-yl-6,7-dihydroquinazoline-8-carboxamide 1-(3,5-ditert-butylphenyl)propan-2-one (5S)-2,3,4-trideuterio-5-[7-[[2-fluoro-6-hydroxy-4-(2,2,3,3,3-pentadeuteriopropoxy)phenyl]methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione 1-[2-(3,4-dichlorophenyl)ethyl]pyrrolidine (3S)-1-[4-(2,6-difluorophenyl)phenyl]sulfonyl-N-[(1R)-6-oxocyclohexa-2,4-dien-1-yl]pyrrolidine-3-carboxamide N-(3,5-dichlorophenyl)-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]acetamide 2-methyl-3,4-dihydro-1H-isoquinoline;6-(5-methylidene-1,4,6,7-tetrahydroindazol-3-yl)pyridine-3-carboxamide N-[(2S)-2-hydroxycyclohexylidene]quinoline-2-carboxamide (5Z)-5-[2-(dimethylamino)ethylimino]-3-methyl-1,4-thiazepane-7,8-dione 4-(1H-indol-2-yl)-3-methylidenepiperazine-1-carboxylate [3-amino-4,4-difluoro-2-(2H-tetrazol-5-yl)pyrrolidin-1-yl]-(3,4-dimethoxyphenyl)methanone 1-(2,3-dimethylphenyl)-5-iodopyrrole-2-carboxylic acid ethane;1-[2-(4-fluorophenyl)propanoyl]pyrrolidine-3-carboxylic acid 6,7-dimethoxy-4-[1-(2H-quinolin-3-yl)ethenyl]quinazolin-2-amine 3-(1H-indol-2-yl)-4,5-dihydrothieno[3,4-b][1]benzoxepine 2-[4-(1H-indole-6-carbonyl)piperazin-1-yl]benzonitrile 2-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]oxyethanol 2-(2,4-dimethylphenyl)sulfonylsulfanyl-N'-hydroxybenzenecarboximidamide 4-(5-methylpyridin-2-yl)-N'-[(6R,9S)-6-thiophen-3-yl-8-azaspiro[4.5]decan-9-yl]benzenecarboximidamide N-(4,6-dichloropyrimidin-2-yl)-3-fluorobenzamide N-[(E)-(4-hydroxyphenyl)methylideneamino]-2-[4-(2H-tetrazol-5-yl)phenoxy]acetamide 4-(4-azidophenyl)-N-[2-methoxy-3-[1,3-dioxo-6-(1H-pyrazol-5-ylamino)isoindol-2-yl]phenyl]benzenesulfonamide 4-[[(2S)-3-cyclohexyl-1-oxo-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)amino]propan-2-yl]carbamoyl]piperidine-1-carboxylic acid 4-amino-6-(1H-indol-3-yl)-2-(1H-pyrazol-5-ylmethoxy)pyrimidine-5-carbonitrile 3-bromo-N-[1,2,4-triazol-3-yl(thiophen-3-yl)methylidene]benzenesulfonamide (4-chlorophenyl)-[2,3-dichloro-6-methyl-5-(trifluoromethoxy)phenyl]methanol 2-[(3E)-4,5-dimethylhexa-1,3,5-trien-3-yl]-N-[2-hydroxy-6-(pyrrolidin-1-ylmethyl)phenyl]pyridine-4-carboxamide 7-phenyl-6H-phenanthridine 4-(3,5-dimethoxyanilino)quinoline-7-carbonitrile N-(3,5-difluorophenyl)-N'-[4-[2-(dimethylamino)ethoxy]-2-fluorophenyl]oxamide;ethane N-[1-(2,4-difluorophenyl)pyrrolidin-3-yl]-1-methyl-4,5,6,7-tetrahydroindazole-6-carboxamide 1-[6-(2,5-dimethylphenoxy)pyrimidin-4-yl]-3-ethylurea;5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]thiophene-3-sulfinate 1-[(3S,7R,8aS)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-N-methylimidazole-4-carboxamide 3-(2,4,6-trifluorophenyl)dithiolane 5-(4,6-dimethoxypyrimidin-2-yl)sulfanyl-1-[(3R,4S)-4-methoxypyrrolidin-3-yl]triazole N-cyclobutyl-2,4-dihydroxy-3-(5-methoxy-1H-indole-3-carbonyl)-N-[[2-[3-(trifluoromethoxy)phenyl]acetyl]amino]benzamide 5-(3,4-dimethoxyphenyl)hex-1-en-2-yloxymethanamine 5-bromo-N-[[3,5-dibromo-2-(4-fluorophenyl)sulfonyl-1-benzofuran-6-yl]methyl]pyridine-3-carboxamide [(3R)-5-amino-1-oxo-2,3-dihydroinden-4-yl]carbamic acid (1S,3R)-N-[2,4-difluoro-5-(2H-tetrazol-5-yl)phenyl]-3-methoxycyclohexane-1-carboxamide 2-(N-acridin-9-ylanilino)acetonitrile 2-(3-fluoropyridin-4-yl)oxyacetate 4-(2,5-dimethoxyphenyl)sulfanyl-3-iodobenzoic acid 2-[4-[(2Z,3E)-1-chloro-3-ethylidenehepta-2,5-dienyl]phenyl]acetic acid N-[(2S,3R)-6-oxo-1-phenyl-2-(4-pyridin-3-ylcyclohexa-2,4-dien-1-yl)piperidin-3-yl]methanesulfonamide 5-tert-butyl-2,4-dihydroxy-N'-(3-morpholin-4-ylpropyl)benzenecarboximidamide 5-[[2-(1H-benzimidazol-4-yl)ethynyl]methyl]imidazolidine-2,4-dione 3-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]-7,8-dihydro-1H-quinolin-2-one 4-chloro-2-[(3,5-difluorophenyl)methyl]-8-fluoroquinazoline 2-[2-methyl-3-oxo-4-[(2,3,5,6-tetrachlorophenoxy)methoxy]oxan-2-yl]acetic acid (5R)-N-(3,4-dichlorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-cyclobutylimino-5-(7-methoxyimidazo[1,2-a]pyridin-3-yl)-1-phenylimidazolidin-2-one 1-(4,5-dihydro-1H-imidazol-2-ylmethyl)pyrazole-3-sulfonamide 4-azido-1-methyl-2,3,5,6-tetraphenylbenzene 6-methyl-N-(1H-pyrazolo[4,3-b]pyridin-5-yl)thieno[2,3-d]pyrimidin-4-amine 2-methylsulfanyl-5H-1,3-diazepine;4-[(E)-prop-1-enoxy]benzaldehyde 2,4-dimethyl-N'-phenylbenzenecarboximidamide (2S)-N-[3,5-difluoro-4-methyl-6-(2,4,6-trimethylphenyl)pyridin-2-yl]-1-methylpyrrolidine-2-carboxamide (1S,3R)-3-[4-[5-[(2-bromoanilino)methyl]-1-(oxan-4-yl)triazol-4-yl]phenoxy]cyclohexane-1-carboxylic acid 4-[(5R)-3-methyl-5,6-dihydrobenzo[b][1]benzoxepin-11-yl]benzenesulfonamide (5-tert-butyl-1,3-oxazol-4-yl)-[2-[(Z)-prop-1-enoxy]phenyl]methanone 5-[(2E,4Z)-hexa-2,4-dien-3-yl]benzo[b]carbazole;propane 4-[(3R)-1-benzylpyrrolidin-3-yl]-2H-phthalazin-1-one;hydrochloride 5-(2,3,4-trichlorophenyl)sulfanyloxypyrimidine 4-azido-5-ethyl-2,3,6-trifluoroaniline 5-chloro-4-[2,6-difluoro-3-[methyl-(1-prop-2-enoylazetidine-3-carbonyl)amino]phenyl]-N-ethylpyridine-2-carboxamide N-[(2R)-3,3,4,5,6-pentadeuterio-1-hydroxyhexan-2-yl]-5-(trifluoromethoxy)pyrimidine-2-carboxamide 2-[3,5-dibromo-4-(methoxycarbonylamino)anilino]acetic acid N-(azidomethyl)-3,4,5-trimethoxyaniline 2-(3,4-difluorophenyl)-1-[3-(5-methylpyridazin-3-yl)pyrrolidin-1-yl]ethanone 4-[3-(2-propylphenoxy)propoxy]benzenecarboximidamide N-(2,3-difluorophenyl)-1-methyl-5-[4-methyl-6-[2-oxo-2-(propylamino)ethoxy]pyridin-3-yl]pyrazole-4-carboxamide;ethane 4-(1H-pyrazol-5-yl)-N-[[3-(pyridin-2-ylmethoxy)phenyl]methyl]piperidine-1-carboxamide 4-[2-(2,3-dihydrothiophen-2-yl)ethynyl]pyridine 4-(2,3-dihydropyrrol-1-yl)-N'-hydroxypyridine-2-carboximidamide 4-(3,5-dichlorophenyl)sulfonyl-6-hydroxycyclohex-2-en-1-one N-[1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonyl)piperidin-4-yl]benzamide 6-cyclopropyl-3,4-difluoro-5-(2-methylhydrazinyl)benzene-1,2-diol 1-[(6S)-8-benzyl-11-hydroxy-2,9-diazaspiro[5.5]undecan-2-yl]ethanone;2,2,2-trifluoroacetic acid 4-methyl-2-N,7-N-dipropylpyrazolo[1,5-a]pyrimidine-2,7-diamine 2-[(4Z)-5-[(3,4-dimethoxyphenyl)methyl]-4-[[5-(trifluoromethyl)furan-2-yl]methylidene]pyrazol-1-yl]-N-propan-2-ylacetamide N-ethyl-2,3-difluoro-N-[(4-oxo-3H-quinazolin-2-yl)methyl]benzamide 3-azidooxy-5,7-dimethyl-1H-indole (3R,5S)-3,4,5-trihydroxy-6-oxo-7-[4-(trifluoromethyl)phenoxy]heptanoic acid 1-(4,5-dimethylthiophen-2-yl)sulfonylpyrrolidine N-(1,3-benzodioxol-5-ylmethylideneamino)-4-[2-[5-(piperidin-1-ylmethyl)-1H-indol-2-yl]pyridine-4-carbonyl]piperazine-1-carbothioamide 1-N',3,5,6-tetraphenylcyclohexa-2,4-diene-1,1-dicarboximidamide (4E)-2,3-bis[(Z)-but-1-enyl]-N-methoxy-6-phenylhepta-2,4-dienamide 1-[4-[1,3-bis(4-chlorophenyl)pyrazole-4-carbonyl]piperazin-1-yl]propan-1-one (Z)-N'-[4-[3,6-dihydro-2H-pyran-5-ylmethoxycarbonyl]phenyl]-4-imino-N,4-dimethyl-2-methyliminobut-2-enimidamide N-(2,3-dichlorophenyl)-1-oxothiane-4-carboxamide (4aR,8aS)-6-[3-[4-(azidomethyl)phenyl]azetidine-1-carbonyl]-4a-methyl-3,4,5,7,8,8a-hexahydro-2H-pyrano[3,2-c]pyridine-2-carboxylic acid 4-[(2R)-1-hydroxy-3,3-dimethylbutan-2-yl]oxycarbonylbenzoate ethane;5-methylcyclohepta-1,3,6-triene;(2R)-N-[2-oxo-3-phenyl-4-[[(2R)-4-sulfanylidenebutan-2-yl]amino]butyl]azetidine-2-carboxamide 4-amino-3,5,6-trifluorobenzenesulfonic acid;2-[(2,3-dichlorophenoxy)methyl]-1,3,5-trifluorobenzene N-(2,4-difluorophenyl)sulfanyl-6-methoxyisoquinolin-8-amine 5-[(2,4-dihydroxyphenyl)methylideneamino]-2-sulfanylidene-1H-pyrimidin-6-one 6-[(2,5-difluoro-3-methoxyphenyl)methyl]-4-hydroxypiperidine-1-carboxylic acid 4-[(2R)-2-[3-fluoro-5-[6-methyl-7-oxo-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-8-yl]phenyl]propanoyl]piperazine-1-carboxylic acid 1,4-diamino-2-[(3,5-dichloropyridin-2-yl)methylsulfanyl]anthracene-9,10-dione (6-propan-2-ylpyridin-3-yl)-[4-(pyrazin-2-ylamino)piperidin-1-yl]methanone 5-chloro-N-[(1R,3S)-3-ethylcyclopentyl]-1H-indole-2-carboxamide 2-[3-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]-N-[(3R)-3,5-dimethylcyclohexa-1,5-dien-1-yl]acetamide 2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[1-(4-hydroxyphenyl)ethyl]acetamide 2-[1-[(2,4-dichlorophenyl)methyl]piperidin-3-yl]acetic acid 2-[(3S,5R)-3-amino-5-methylpiperidin-1-yl]-4-ethanimidoylquinolin-7-ol 6-tert-butyl-2-ethyl-N-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-fluorobenzamide;ethane N-(3,4-dimethoxyphenyl)-1H-pyrrole-2-carboxamide 4-(1,3-benzodioxol-5-yl)-1H-[1]benzoxepino[2,3-c]pyrrole;ethane 2-(4-chlorophenyl)sulfanyl-1-[4-(2,3-difluoro-4-methoxybenzoyl)piperazin-1-yl]ethane-1,2-dione 2-[[2-methyl-6-(4-piperazin-1-ylphenyl)-7H-imidazo[1,2-a]azepin-5-yl]oxy]propanoic acid [(2S,4R)-2-ethyl-1,3-dimethylpiperidin-4-yl]-[4-hydroxy-4-[[4-phenyl-6-(trifluoromethyl)pyrimidin-5-yl]oxymethyl]piperidin-1-yl]methanone 2-(7-methoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)-N'-[1-(3-methylphenyl)propyl]piperidine-1-carboximidamide 2-[[3,5-diamino-4-(3-chloropropyl)-1H-pyrrol-2-yl]methylidene]cyclohexan-1-ol [3-fluoro-4-[6-(4-hydroxyphenyl)pyridazin-3-yl]oxyphenyl]azanide N-(2-amino-5-methylhexanoyl)-4-benzylpiperazine-1-carboxamide [4-amino-3,5-bis(trifluoromethyl)phenyl]-[2,6-dibromo-4-(1H-pyrazol-5-yloxymethyl)phenoxy]borinic acid N-[(3S,4R)-1-cyclohexyl-4-(5-methoxypyrazin-2-yl)pyrrolidin-3-yl]propanamide 4-(6-chloronaphthalene-2-carbonyl)-N,8-dimethylquinoline-3-carboxamide 4-[(2,5-dioxopyrrolidin-3-yl)amino]benzenesulfonic acid 3-[(5R)-1,8-diazaspiro[4.5]decane-8-carbonyl]-1H-pyridin-2-one N-[2-(1H-indol-3-yl)ethyl]-4-nitro-N-prop-2-enylbenzamide 5-[1,3-benzodioxol-5-yl-[[2-(2-chloro-4-fluorophenyl)cyclopropanecarbonyl]amino]methyl]furan-3-carboxylic acid (2S)-2-(8-bromodibenzofuran-1-yl)-2,3-bis(4-tert-butylphenyl)propanenitrile 5-chloro-2,3-dihydropyrrolo[2,1-b][1,3]benzothiazole 3-[2-(4-cyclopropylphenyl)ethynyl]-5,6-dihydrobenzimidazolo[1,2-a]isoquinoline 1-[(E)-3-azidoprop-2-enyl]naphthalene 4-(7-fluoroimidazo[1,2-a]pyridin-3-yl)-7-[[5-[1-methyl-6-oxo-5-[4-(trideuteriomethoxycarbonyl)piperazine-1-carbonyl]pyridin-3-yl]thiophen-2-yl]amino]-2,3-dihydroisoindol-1-one N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-ylmethyl)piperidine-3-carboxamide 1-(2,6-difluorophenyl)-4-[3-(2-methylpyrimidin-5-yl)benzoyl]piperazin-2-one 5-[2-(4,6-dimethylpyridin-3-yl)-1H-indol-7-yl]-N-methylpentanamide 2,5-dimethyl-4-(3-methylideneoxan-3-yl)pyrimidine 4-(3,5-dimethyl-1H-pyrazol-4-yl)-N'-(4-fluorophenyl)pyridine-2-carboximidamide 2-[(2Z)-2-[(3-bromophenyl)methylidene]hydrazinyl]-5-propan-2-yl-4H-1,3-thiazol-4-ol N-(2,3-dihydro-1H-inden-5-yl)-4-methyl-5-[(E)-(5-oxoimidazolidin-4-ylidene)methyl]furan-2-carboxamide (E,3S)-4,7-dihydroxy-6-methyl-1-phenyldec-5-en-3-one N-azido-2,3-dihydrobenzo[g][1]benzothiole-4-sulfonamide 2-ethyl-4-iodo-3-methylthiophene 2-[N-(benzenesulfonyl)-3,5-dibromoanilino]propanoic acid [3-(hydroxymethyl)-4,5,7,8-tetrahydro-1H-pyrazolo[3,4-d]azepin-6-yl]-[3-(2-propan-2-ylimidazol-1-yl)phenyl]methanone 2-[(2R)-1,4-dibenzyl-5,7-dioxo-3,6-dihydro-2H-pyrrolo[2,3-d]pyrimidin-2-yl]acetamide ethane;[2-(methylamino)phenyl]-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)methanone N'-[(5R)-3-[3,4-bis(phenylmethoxy)phenyl]-1-[2-(4-chlorophenyl)ethyl]-2-oxopyrrolidin-3-yl]heptanediamide 2-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-4,6,7-trimethoxypyrrolo[3,4-c]pyridin-5-ol 1-(2,3-dihydro-[1]benzothiolo[2,3-c]pyridin-4-yl)-3-methoxypropan-2-one 4-[[5-(2,3-dihydro-1H-inden-5-yloxymethyl)benzimidazol-1-yl]methyl]-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide 2-N-[3-[1,4-bis(benzenesulfonyl)pyrrol-2-yl]phenyl]-2-N-ethyl-2H-pyrimidine-2,5-diamine (4R)-N-butyl-N,5-diethyl-3,3-dimethyl-1,2-dihydrothieno[3,2-f]quinoline-7-sulfonamide 6-ethyl-2-fluoro-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methoxy]benzenecarboximidamide;hydrochloride (6-cyano-3,4,5,7-tetrahydro-2H-azepin-1-yl)-[3-(difluoromethoxy)pyridin-4-yl]borinic acid 4-[(3-chlorophenyl)methyl]-2,5,6-triethoxypyrimidine 4-[2-(3-tert-butylpyrazol-1-yl)ethoxy]piperidine;1,5,7-trimethylimidazo[4,5-b]pyridine N-[2-(5-fluoropyridin-3-yl)ethyl]-4,6-dimethoxypyrimidine-5-carboxamide 5-(9H-fluoren-2-yl)naphthalene-1,4-dicarboxylic acid N-benzyl-2-bromo-6-nitroaniline (3E,5E)-6-[2-methyl-4-(trifluoromethyl)phenoxy]hepta-1,3,5-triene-3,4-diol 4-N-[2-chloro-3-(trifluoromethyl)phenyl]-6,7-dihydropyrrolo[2,1-f][1,2,4]triazine-2,4-diamine;ethane 6-[5,5-dimethylhex-1-en-2-yl(propanoyl)amino]oxypyridine-3-carboxylic acid 4-hydroxy-3-(2-hydroxypropan-2-yl)benzenesulfinic acid N-[(3S,7R,8aS)-3-propan-2-yl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-3-methoxy-1-benzothiophene-2-carboxamide N-[(Z)-(4-hydroxy-3,5-diiodophenyl)methylideneamino]-3-methyl-1H-indole-2-carboxamide 4-fluoro-1'-(2-phenylethyl)-N-propan-2-ylspiro[7,8-dihydro-5H-naphthalene-6,3'-azetidine]-2-carboxamide N-cyclopropyl-5,7-dimethoxy-4H-1,8-naphthyridine-3-carboxamide 2-[6-fluoro-1'-[4-(trifluoromethyl)benzoyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-4-yl]oxy-N-propan-2-ylsulfonylacetamide 6-butyl-3-[4-(oxiran-2-ylmethoxy)phenyl]triazolo[1,5-a]pyridine 3-(3,5-difluorophenyl)-2-(4-fluorophenoxy)propanoic acid (2S)-1-[6-(2-propan-2-ylpyridin-3-yl)-8,9-dihydropurin-9-id-4-yl]propan-2-amine N-[4-[2,2-diethoxyethyl(propan-2-yl)amino]phenyl]sulfonylbenzamide 5-(4-cyanophenyl)pentylazanium 2,4-bis(3-fluoro-2H-indazol-5-yl)pyridine-3-carboxylic acid N-[(Z)-1-aminoethylidenecarbamothioyl]benzamide 1-[4-[[5-fluoro-2-(iodomethoxy)phenyl]methylamino]oxan-4-yl]propan-2-one 2-benzamido-N-cyclohexyl-6-[[(Z)-N'-diazenylcarbamimidoyl]amino]benzamide 2-(4-bromophenyl)-3,6-dimethyl-1H-pyrazin-4-ium 2-(2,4-difluorophenyl)-1H-pyrimidine-2,4-diamine 2-(3,4-dimethoxyphenyl)sulfonyl-N-hydroxypropanamide 1-[2-methylsulfonyl-4-(trifluoromethoxy)phenyl]piperidine 2-cyclopropyl-4,5-diphenylimidazole N-(cyclohexylmethoxy)-2,4-dioxo-1H-quinoline-3-carboxamide 6-tert-butylsulfanyl-1,3-dihydroindol-2-one ethane;3-[3-(4-methylphenyl)-2-propoxypentyl]piperidine N-[2-[(5Z)-5-benzylidene-4-oxo-1,3-thiazolidin-2-yl]ethyl]acetamide [(5R,7S)-1-methyl-2-oxo-7-phenyl-3-(pyridin-4-ylcarbamoylamino)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]diazepine-5-carbonyl]oxidanium 4-(6,7-dimethoxyquinolin-4-yl)oxyaniline 6-(2-hydroxyethyl)-N,4-dimethyl-1-[5-[3-oxobutanoyl(propyl)amino]pentyl]-2-oxopyridine-3-carboxamide 3-[[2-(methoxymethyl)pyrimidin-5-yl]methyl]-2,8-dioxaspiro[4.5]decane 3-[(2,6-dichlorobenzoyl)amino]-N-(2H-triazol-4-yl)propanamide 1-[5-fluoro-6-(3,4,5-trifluorophenyl)pyridine-2-carbonyl]-N-(5-nitrothiophen-2-yl)azetidine-2-carboxamide 4-chloro-6,7-difluoro-2H-benzotriazolo[1,5-a]pyridine 1,3-dibenzylbenzo[e]indole N-(2-benzylsulfanylethyl)-N-(4-methoxyphenyl)hydroxylamine 3,4-dichloro-N-[[(2S)-oxan-2-yl]methylideneamino]aniline 2-(3,4-dichlorophenyl)imidazo[1,2-a]pyridine 4-[5-(1,3-benzodioxol-5-yl)-2-propanoyloxypentyl]piperazine-1-carboxylic acid 2-[[4-(benzenesulfonyl)-3,5-dihydro-1H-cyclopenta[c]pyridin-6-yl]amino]-1,3-thiazole-5-carboxamide 2-(2,6-diethylphenyl)-5-methylsulfanylphenol N-[3-[4-(2-chlorophenyl)piperazin-1-yl]propyl]-5-methoxy-1H-indole-2-carboxamide (2S)-2-[[5-(1,3-benzothiazol-2-ylmethylsulfanylmethyl)furan-2-carbonyl]amino]hexanoic acid (3aR,6aS)-2-[4-chloro-5-(trifluoromethyl)pyridin-3-yl]-1-methylsulfonyl-3,3a,4,5,6,6a-hexahydro-2H-pyrrolo[2,3-c]pyrrole 5-[7,7-dimethyl-8-oxo-2-(3-phenylpropanoylamino)-6,9-dihydropyrido[1,2-a]indole-10-carbonyl]pyridine-3-carboxylic acid 5-[3-fluoro-4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl]imidazolidine-2,4-dione 2-(5-bromothiophen-3-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine 2-[(1R,3S)-3-aminocyclopentyl]oxy-5-fluoroaniline [1-(1,5-dimethyl-3-propanoylpyrazol-4-yl)cyclopentanecarbonyl]carbamic acid 2,4-dimethyl-1'-(5-methylsulfonylpyrimidin-2-yl)spiro[5H-cyclopenta[c]pyridine-7,3'-azetidine] N-[5,6-dimethyl-2-(1-pyrimidin-4-ylethenoxy)pyridin-3-yl]benzenesulfonamide (5E)-2-imino-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 2-(1H-benzimidazol-2-ylsulfanyl)-N-[(Z)-(5-bromo-3,4-dihydroxyphenyl)methylideneamino]acetamide (Z)-3-amino-2-[amino-[[6-[5-chloro-3-ethyl-2-fluoro-4-(1-methylpiperidin-4-yl)oxyphenyl]pyrido[2,3-d]pyrimidin-2-yl]methyl]amino]prop-2-enamide 4-[(3R)-1-[2-fluoro-6-methoxy-4-(trifluoromethyl)phenyl]-5-oxopyrrolidine-3-carbonyl]-N,N-dimethylpiperazine-1-sulfonamide N'-(4-methylphenyl)sulfonyl-2,3-dihydro-1H-indene-2-carbohydrazide (4S)-3,8-diazatricyclo[9.4.0.02,7]pentadeca-1(15),11,13-triene;4-methylphenol 5-[4-(1,3-dioxolan-2-yl)butanoyl]-4-methoxy-6-oxopyran-2-carboxylic acid 2-[(4-methylphenyl)sulfonylamino]-N-[2-oxo-3-[[(3S,5R)-5-(trifluoromethoxy)piperidin-3-yl]amino]pyridin-1-yl]acetamide 4-(2-bromophenoxy)pentanoic acid 2-[4-(2,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-5,6-dihydroquinoline (2S)-2-[5-(4-cyanophenyl)pyridin-2-yl]-1,3-thiazolidine-4-carboxamide 2-[4-(3,5-dimethylphenyl)-6-(3-naphthalen-1-yloxyprop-1-en-2-ylsulfanyl)-1,3,5-triazin-2-yl]-5-propoxyphenol (4-fluorophenyl)methyl-[3-(2H-pyrazolo[3,4-b]pyridin-3-ylamino)piperidin-1-yl]iodanium 2,6-bis(methoxycarbonyl)pyridine-4-carboxylic acid 5-fluoro-7-[1-(2,2,2-trifluoroacetyl)piperidine-4-carbonyl]-N-[1-(trideuteriomethyl)cyclopropyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide 3-[4-[(5R)-5-amino-2,2-dimethylpentoxy]-3-(trifluoromethyl)phenyl]-7-[3-hydroxyprop-1-ynyl(piperidin-4-ylmethyl)sulfamoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide 1,2-diamino-4-(2,6-dimethoxyphenyl)-6-oxopyridine-3,5-dicarbonitrile 4-methyl-6-[3-[(1R,2S)-2-thiophen-2-ylcyclopropanecarbonyl]azetidin-1-yl]pyrimidine-5-carbonitrile N-cyclohexyl-2-(1H-imidazol-5-ylmethylidene)butanamide N-[4,6-dimethyl-3-(trifluoromethyl)cyclohexa-1,3-dien-1-yl]-5-methylpyridine-2-carboxamide 1-[5-(3,4-dichlorophenyl)-2,8-dimethylimidazo[1,2-a]pyrazin-6-yl]propan-1-one N-[4-(4,4-dimethylpent-1-enyl)cyclohexa-2,5-dien-1-ylidene]pyridine-3-carboxamide N-[(4,5-dihydro-1H-imidazol-2-ylhydrazinylidene)methyl]thiophene-3-carboxamide 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-phenacylamino]benzoic acid N-cyclopropyl-2,4,6-trimethoxypyridine-3-carboxamide 2-[2,4-bis(trifluoromethyl)phenyl]-5-(4-methylpiperazin-1-ium-1-ylidene)-6H-[1,3]thiazolo[5,4-d]pyrimidin-7-one 5-[(4-aminophenyl)diazenyl]-1-tert-butylpyrazole-3-carboxylic acid 4-[3-(2,5-difluorophenoxy)propyl]-1H-pyrazole 4-chloro-6-[2-(2,2-difluoroethoxy)-3-methoxyphenyl]-2-sulfanylidene-5,6-dihydro-1H-pyrimidine-5-carbonitrile 1-bromo-3-chloro-5,6-diphenylcyclohexa-2,4-dien-1-amine [3-[4-(1,3-benzodioxol-5-yl)piperidine-1-carbonyl]cyclopenten-1-yl]methanesulfonamide 2-[4-[(3R)-5-amino-2,6-dimethylheptan-3-yl]phenyl]ethanamine 6,7-dihydroxy-2-(3,4,5-trimethoxyphenyl)chromen-4-one 2-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]acetic acid 2-[(2R)-1,4-dibenzylpiperazin-2-yl]ethanol 2-[6-[(E)-[4-phenyl-5-(1H-pyrrole-2-carbonylhydrazinylidene)pyrazolidin-3-ylidene]methyl]pyridin-2-yl]propanoic acid 2-(2,3-dichlorophenyl)acetonitrile;5-[4-methyl-5-[1-methyl-5-(trifluoromethyl)pyrazol-4-yl]-1H-imidazol-2-yl]imidazolidine-2,4-dione 2-[1-(4-azidobenzoyl)azetidin-3-yl]oxyacetonitrile 1-[[(3S,4R)-1-cyclohexylpiperidin-3-yl]methyl]-5-phenylimidazole 1-(azidomethyl)anthracene N-[(1S)-2-azidocyclopropyl]-2,4-dichlorobenzenesulfonamide 2-[4-[5-(3,5-dichlorophenyl)-5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]phenyl]-N'-hydroxypropanehydrazide 4-(2,5-difluorophenyl)thiophene-3-carboxamide (5Z)-5-[[4-[2-[cyclopropylmethyl-[(2,6-difluorophenyl)carbamoyl]amino]ethoxy]phenyl]methylidene]imidazolidine-2,4-dione 2-[2-hydroxypropyl-(6-nitro-1,3-benzothiazol-2-yl)amino]acetamide N-(4-ethoxyphenyl)-N-[2-methyl-5-(1,3,4-oxadiazol-2-yl)phenyl]acetamide N-[(4-aminophenyl)methyl]-3,3,4,5,6-pentamethylcyclohexa-1,5-diene-1-carboxamide 2-[(2Z)-4-oxo-2-[[3,4,5-triethoxy-6-(3-methylbutoxy)naphthalen-1-yl]methylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 5-hydroxy-N'-(4-nitrophenyl)-2-[4-(trifluoromethyl)anilino]-1H-imidazole-4-carboximidamide 1-[4-[3-(azidomethyl)phenyl]piperidin-1-yl]ethanone 3-(1H-indol-2-yl)-4-methylpentan-1-amine;4-phenyl-1,3-thiazol-2-amine N-(5-chloropyridin-2-yl)-2,4,6-trimethyl-N-(3-methylbut-2-enyl)benzenesulfonamide 3-[4-(cyclopropylmethylamino)butanoylamino]-2,6-difluorobenzamide (E)-3-[4-amino-2-fluoro-5-(trifluoromethylsulfanyloxy)phenyl]-N-cyclopropyl-3-phenylprop-2-enamide N-[1-(2-chloroethyl)cyclohexyl]quinoline-3-carboxamide 3-[4-(2,5-dioxopyrrolidin-1-yl)piperidin-1-yl]benzonitrile 2-methyl-N'-(6-phenyl-7H-purin-8-yl)pyridine-3-carboximidamide 1-azidooxy-2,3,4-trichloronaphthalene 1-azidooxy-4-phenoxybenzotriazole (5R,7S)-2-benzylsulfanyl-N-ethyl-5-methyl-7-phenyl-4,5,6,8-tetrahydropyrazolo[1,5-a][1,3]diazepine-3-carboxamide [(2R,6S)-4-[2-chloro-3-[[5-cyclopropyl-3-(2,6-dichlorophenyl)pyridine-2-carbonyl]amino]phenyl]-2,6-dimethylmorpholin-4-ium-2-carbonyl]oxidanium 2-[[3,5-bis(trifluoromethyl)phenyl]sulfonylamino]-4-(3,6-dihydro-2H-pyran-5-yloxycarbonyl)benzoic acid 1-(4,5-difluoro-2-propylphenyl)-3-methylbenzene;N-[6-[(3S)-3-ethylpiperazin-1-yl]pyridin-3-yl]formamide 3-chloro-4-[(E)-2-hydroxypropanoyl]pyridine-2,6-dicarboxylic acid 4-[(1R)-2,5-dimethylcyclohexyl]oxybenzonitrile 7-cyclopentyl-2-[[5-(N'-piperidin-3-ylcarbamimidoyl)pyridin-2-yl]amino]pyrrolo[2,1-f][1,2,4]triazine-6-carboxylic acid 2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]thiophene-3-carbonitrile N-[3-(2,4,6-trimethylphenyl)-2H-imidazol-1-ium-2-id-1-yl]pyridine-2-carbothioamide 2-[4-chloro-N-(6-hydroxy-1H-benzimidazol-2-yl)anilino]acetamide 4-[(5-aminotetrazol-1-yl)methyl]-6,7-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine 5-[2,6-dichloro-4-(1H-imidazol-2-yl)phenoxy]-3-ethylsulfonylpyridine (2S)-N,3-dimethyl-2-[(4-morpholin-4-ylphenyl)sulfonylamino]butanamide 2-[3,5-difluoro-4-(triazol-1-yl)anilino]pyrimidine-5-carbohydrazide 1-[(4aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1]benzoxepin-10-yl]-N-methylethenamine (E)-N-[(4-methoxyphenyl)methyl]-N',2-dimethylprop-1-ene-1,3-diamine (4-hydroxyphenyl)-[(3R,5S)-1-[2-methyl-6-(1H-pyrazol-4-yl)pyrimidin-4-yl]-5-(pyridin-3-ylmethoxy)piperidin-3-yl]methanone N-benzyl-N-methyl-1,2-oxazole-5-carboxamide;ethane 2-[[4-[(Z)-2-aminoethenyl]triazol-1-yl]methoxymethyl]-6-fluorobenzaldehyde N-ethyl-4-[2,3,4,5-tetrafluoro-6-methoxycarbonyl-N-(methylcarbamoyl)anilino]butanoic acid 4-methyl-3,5-di(propanoyl)benzenesulfonic acid (3R,4R)-3-phenylsulfanyl-1-(thiophen-2-ylmethyl)piperidine 2-[2-chloro-4-(trifluoromethyl)phenyl]sulfonyl-N,1-dimethylcyclopentane-1-carboxamide (4-azidopyridin-2-yl)-[3-cyclopropylidene-6-hydroxy-1-(oxan-4-yl)-5-pentoxyisoindol-2-yl]methanone 6-cyclohexyl-1-[(4S)-2,2,4-trimethylpiperidin-4-yl]indazole 4-amino-1-tert-butyl-3,3a,4,5,7a-hexahydroimidazo[2,1-c][1,4]benzoxazin-8-ol 1-[3-methylbut-2-enyl(phenacyl)amino]propan-2-one 4-(2,6-dichloro-3-fluorophenyl)-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 6-[(3,4-dimethylphenyl)sulfamoyl]-1H-indole-2-carboxylate 3-[N-(2,4-difluorophenyl)sulfonyl-3-(trifluoromethyl)anilino]propanamide N-[4-amino-3,4-dioxo-1-(1,2,3,4-tetrahydroquinolin-6-yl)butan-2-yl]-3-pyridin-3-ylimidazole-4-carboxamide 3-[2,6-di(propan-2-yl)phenyl]-5-iodobenzonitrile 3-(difluoromethyl)-1,4-benzothiazine 2-(1-methylpyrazol-4-yl)-6,7,8,9-tetrahydro-5H-pyrrolo[3,2-b]azepine 2-[2,6-bis(1-pyridin-3-ylethoxy)phenyl]acetamide 6-chloro-2,3,4,5-tetrahydroazepino[1,7-a]indole 6-[(3,4-dichlorophenyl)methyl]-2-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-[5,6-difluoro-1-(1H-pyrazole-4-carbonyl)benzimidazol-2-yl]acetonitrile 6-amino-3,4-difluoro-5-nitro-2-propanoylbenzonitrile 3-[[2,6-dichloro-4-(3-chloropropoxy)phenyl]sulfonylamino]propanoic acid 4-methyl-7-(1H-pyrazole-5-carbonyl)-3,5-dihydro-2H-pyrido[3,4-f][1,4]oxazepin-6-one 2-(1H-indol-3-ylmethylidene)-1,4-dimorpholin-4-ylbutane-1-thione 5-[2-(3,5-dimethylphenyl)-1H-indol-4-yl]-1,2-oxazol-3-one;ethane 6-[(2R)-1-hydroxypropan-2-yl]oxy-N,N-dimethylpyridine-3-sulfonamide N-[4-(7,8-difluoroimidazo[1,2-a]pyridin-3-yl)-5-methylpyrimidin-2-yl]cyclopropanecarboxamide 2-[2-[[4-(butylcarbamoyl)-5,6,7,8-tetrahydronaphthalen-1-yl]oxymethyl]phenyl]benzamide N-[(2E,3Z)-2-ethylidenehexa-3,5-dienyl]-4,6-dimethylpyridin-2-amine N-(4,5-dimethyl-2-phenyldiazenylphenyl)-1H-pyrrolo[3,2-c]pyridine-3-carboxamide 2-(3-bromophenyl)-1,2-dihydrobenzo[e]benzimidazole 3-(1H-benzimidazole-2-carbonyl)benzoic acid N-[1-(1H-indole-2-carbonyl)piperidin-3-yl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-6-carboxamide 4-(5,6,7,8-tetrahydroquinoline-3-carbonylamino)butanoic acid N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2-oxoazetidine-3-carboxamide N-[5-(3,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-2-piperazin-1-ylbenzamide (5Z)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[(2-fluoro-6-hydroxyphenyl)methylidene]-1,3-thiazolidin-4-one 2,6-diamino-4-(3-bromo-4-fluorophenyl)-4H-pyran-3,5-dicarbonitrile 6-methyl-3,4-diphenyl-9H-fluorene 1-(2-amino-4,5-dihydro-3H-azepin-6-yl)-4-[3-[6-methoxy-5-(1-methylpyrazol-4-yl)pyrazolo[1,5-a]pyridin-2-yl]piperidine-1-carbonyl]piperazin-2-one 4-[(3S)-4-benzylpiperazin-1-ium-2-yl]oxyaniline N-[3,5-bis(2-chlorophenyl)pyrazol-1-yl]benzenesulfonamide 1-[3-(5-methyl-2,4-dioxopyrimidin-1-yl)propanoyl]pyrrolidine-3-carboxamide N'-(4-bromo-2,5-dimethylphenyl)-N'-naphthalen-1-ylethane-1,2-diamine (Z)-2-methylimino-5-[6-phenyl-3-(trifluoromethyl)imidazo[1,2-b]pyridazin-7-yl]pent-3-en-1-amine 2-(2-fluoropyridin-4-yl)-7-([1,3]oxazolo[5,4-b]pyridin-2-ylamino)imidazo[1,2-a]pyridine-6-carbonitrile N-(1,3-benzodioxol-5-ylmethyl)-3-butanoyl-2H-[1]benzofuro[3,2-b]pyridine-4-carboxamide N-[2,6-difluoro-3-(1H-indole-4-carbonyl)phenyl]piperidine-4-sulfonamide N-[3-methyl-4-(1,2-oxazol-5-yl)phenyl]-5-pyrrolidin-2-ylthiophene-2-carboxamide 1-[5-(3,4-dichlorophenyl)sulfanyl-2-hydroxyphenyl]ethane-1,1,2,2-tetracarbonitrile 4-methoxy-2,6-dimethylbenzenesulfonic acid;4-[2-[2-(3,4,5-trimethoxyphenyl)ethylidene]hydrazinyl]benzenesulfonamide 2-chloro-N-[(6S)-5,6-dihydro-4H-1,3-thiazin-2-yl]benzamide N-(2,6-dioxopiperidin-3-yl)-4-[3-[(3E)-hexa-1,3,5-trien-3-yl]oxyphenyl]benzenesulfinamide 2-(3,5-dimethylpyrazol-1-yl)-N-[2-(3-fluoro-4-hydroxyphenyl)ethyl]acetamide 2-azidooxy-5-[2,4-dichloro-3-[(2,6-difluorophenyl)methyl]phenoxy]pyridine N-methyl-2-[4-methylidene-3-(5-methylthiophen-3-yl)-1,3-thiazinan-2-ylidene]ethanamine N-[[6-fluoro-5-(7-pyridin-2-yl-1,3-benzothiazol-2-yl)pyridin-3-yl]methyl]-3-oxocyclobutane-1-carboxamide N-[(2S)-4-azidobutan-2-yl]-3-cyclohexyloxybenzamide 3-azidosulfanyl-1,2-difluoro-4-phenylbenzene 1-N,6-N-bis[(4-methoxyphenyl)methyl]heptane-1,6-diamine N-(diaminomethylidene)-3,5-diphenylbenzenecarboximidamide 6-(4-methylpiperazin-1-yl)-2,3-dihydrochromen-4-one 3-[3-[(Z)-2-aminobut-1-enyl]phenyl]sulfanylpropanenitrile 1-(1,2-dihydroisoquinolin-7-yl)-3-[(3S)-1-methylpyrrolidin-3-yl]urea (2S)-2-[[[6-chloro-5-(4-ethylcyclohexanecarbonyl)pyridazin-3-yl]amino]methyl]pyrrolidine-1-carboxylic acid (4E,5Z)-N-ethenyl-N-[3-[2-(1H-indol-2-yl)ethynyl]phenyl]hepta-4,6-dienamide 5-azido-3-methylsulfanyl-N-[4-(trifluoromethoxy)phenyl]-1,2-thiazol-4-amine 1-(azetidine-3-carbonyl)-N-[2-(1,3,4-trimethylpyrazol-3-yl)ethyl]pyrrolidine-2-carboxamide [2-cyclopropyl-6-(trifluoromethoxy)phenyl]thiourea 5-(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-3-yl)-N-propan-2-yl-6-[(1S,4R)-2,2,4-trifluorocyclopentyl]pyrazin-2-amine [1-(4-chlorophenyl)cyclopropyl]-(3-imidazol-1-ylpyrrolidin-1-yl)methanone N-[(E)-2-aminoprop-1-enyl]-4-[3-(4-ethanimidoylcyclohexa-1,5-dien-1-yl)oxyphenoxy]-6-methylpyridine-2-carboxamide N-[3,4-bis(ethenyl)phenyl]-2-methoxy-1-(3-morpholin-4-yl-1H-1,2,4-triazol-5-yl)ethanimine 2-[1,1,1,3,3,3-hexafluoro-2-(3,4,5-trimethoxyphenyl)propan-2-yl]phenol 4-[4-[2-(cyclopropylmethylamino)ethoxy]phenyl]aniline 2-methyl-N,4-diphenylaniline;5-(4-methylcyclohexa-1,3-dien-1-yl)-6a,7a-dihydro-[1]benzofuro[2,3-c]carbazole (Z)-2-amino-3-[amino(cyclopropylmethylsulfanylmethyl)amino]-N-[1-(4,6-dichloropyridin-2-yl)ethenoxy]-N'-prop-1-en-2-ylbut-2-enimidamide 6-[(E)-(cyclobutylidenehydrazinylidene)methyl]pyridine-2,5-dicarboxylic acid 2-[4-[[1-(cyclohexylmethoxy)pentan-3-ylamino]methyl]phenyl]acetic acid (1S,3R)-3-[6-[5-[[dideuterio-[4-[dideuterio(methyl)carbamoyl]oxyphenyl]methylideneamino]carbonyl]thiophen-2-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid 5-[[6-chloro-3-(difluoromethoxy)pyridin-2-yl]carbamoyl]pyridine-2-carboxylic acid 4-[3-ethylsulfonyl-5-(trifluoromethoxy)pyridin-2-yl]-6-[1,2,4]triazolo[1,5-a]pyridine-8-carbonitrile 3-(1H-imidazol-2-yl)naphthalene-2-carboxamide 2-[4-(aminomethyl)phenyl]sulfanyl-3H-pyrido[3,2-d]pyrimidin-4-one 1-[(6S)-2,6-dimethylmorpholin-4-yl]-7-methyl-5H-imidazo[1,2-a]quinoxalin-4-imine 2-(1H-benzimidazole-2-carbonyl)-6,7,9,9a-tetrahydro-5H-imidazo[1,5-a][1,4]diazepine-1,3-dione N-[5-(hydroxymethyl)-2-propan-2-yloxyphenyl]-4-(3,7,11-triazaspiro[5.6]dodecane-10-carbonyl)benzamide 4-(2,3-dimethylphenyl)-6-oxo-2-propan-2-ylsulfanyl-1H-pyrimidine-5-carbonitrile 4-(6-chloropyridazin-3-yl)-6-[1,1-difluoro-2-methoxyethyl(sulfino)amino]pyrimidine 2-[3-hydroxy-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-N,N-dimethylacetamide 1-(4-methoxyphenyl)-N,2-dimethylcycloheptane-1-carboxamide 5-(2,6-difluorophenyl)-N-methyl-3-[3-[2-(6-pyridin-4-ylimidazo[1,2-a]pyrazin-8-yl)acetyl]phenyl]imidazole-4-carboxamide 2-(3,5-ditert-butyl-4-methoxyphenyl)propanoic acid N-[(4,5-dimethoxy-2-nitrophenyl)carbamothioyl]benzamide 4-(3-azidopropyl)-1,2,3,5,6,7-hexamethoxynaphthalene 5-(2,6-dichlorophenyl)sulfanyl-4H-1,3-thiazol-2-amine 5-(2-cyclohexylethenylamino)-N'-methylidenebenzenecarboximidamide 1-(3,5-dimethylphenyl)sulfanylpiperidine N-ethyl-2-[3-[2-(4-ethylphenyl)phenyl]propanoylamino]-1,3-thiazole-5-carboxamide 4-[[4-(2,3-dimethoxyphenyl)imino-1,3-thiazolidin-5-ylidene]methyl]benzene-1,3-disulfonamide N-[(1S,3R)-3-[[2-[2-(4-methylpiperazin-1-yl)ethoxy]quinazolin-4-yl]amino]cyclohexyl]propane-2-sulfonamide 4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylamino)phenol 2-[4-(4,4-dimethylpiperidin-1-yl)-5-[4-[2-(6-fluoro-4-oxochromen-3-yl)ethoxy]phenyl]-2-methylpyridin-3-yl]acetic acid 4-[2-(dimethylamino)ethyl]-N-(3-hydroxyphenyl)piperazine-1-carboxamide N-(3,4-difluorophenyl)-3-[2-hydroxy-5-methyl-1-(1,3-thiazol-5-yl)pyrrol-3-yl]propanamide 4-[8-amino-6-(2-hydroxyethyl)imidazo[1,5-a]pyrazin-3-yl]benzaldehyde 2-[6-(2,4-difluorophenyl)-3-iodo-5H-pyrazolo[1,5-b][1,2,4]triazol-7-yl]ethanol 1-[4,5-diamino-3-(ethoxymethyl)thiophen-2-yl]ethanone N-[2-[6-fluoro-3-(2H-tetrazol-5-yl)indole-1-carbonyl]-4,5-dihydrothieno[2,3-g]indazol-7-yl]benzenesulfonamide 7-[6-[(E)-2-methylhept-3-en-4-yl]oxypyridin-3-yl]-1,5-naphthyridine 2-(4-fluorophenoxy)-5-hydroxycyclohepta-2,4-dien-1-one 3-azidooxy-4-(2,5-difluorophenyl)furan N-cyclohexyl-2,4-dimethoxy-5-nitrobenzenesulfonamide N-[3-fluoro-5-[2-[7-(4-methylimidazol-1-yl)-3H-imidazo[4,5-c]pyridin-2-yl]-1H-imidazo[4,5-b]pyridin-7-yl]phenyl]-N',N'-dimethylethane-1,2-diamine N-[(6S)-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazol-6-yl]-2-methoxybenzamide 6-(4,5-dimethylfuran-2-carbonyl)-3a-phenyl-5,7,8,9-tetrahydroimidazo[1,2-a]pyrimidine-1,3-dione 3-amino-N-[(E)-1-(2-fluorophenyl)butylideneamino]benzamide (2R)-3-[6-(4,4-dimethylpiperidin-1-yl)-5-fluoropyridin-3-yl]-2-[(3S)-3-[formyl(hydroxy)amino]pyrrolidin-1-yl]propanoic acid 1-(4-methylpiperazin-2-ylidene)but-3-en-2-one;N-[5-[5-[[2-[[2-(trifluoromethoxy)phenyl]carbamoylamino]cyclohexa-2,4-diene-1-carbonyl]amino]indazol-2-yl]pyridin-3-yl]acetamide 2-amino-4,6-dichlorobenzenesulfonic acid 1-[4-amino-5-methyl-6,7-bis(quinolin-3-ylmethoxy)quinazolin-2-yl]propan-2-one 4-chloro-6,7-dimethoxy-1H-quinoline-2,8-dione [(5S)-4-hydroxy-7,8-dihydro-6H-pyrazolo[1,5-a][1,3]diazepine-5-carbonyl]carbamic acid 2-(3,4-dimethoxyphenyl)-5-fluoroquinazoline;hydrochloride ethane;methanol;5-[4-(3-oxohexyl)phenyl]pentanenitrile 1-(azidomethyl)-3-(3,4-dichlorophenyl)benzene 5-bromo-2-(2,3-dihydroindol-1-yl)benzoic acid 3-[4,5-bis(ethenyl)cyclohepta-1,4,6-triene-1-carbonyl]benzoic acid 4-[(2S)-2-[4-(4,6-dichlorocyclohexa-1,5-dien-1-yl)phenoxy]-3-methoxypropanoyl]piperazine-1-carbothioamide 2-amino-6,9-dimethyl-3H-pyrido[3,4-b]indol-1-one;(2R)-4-methoxybutan-2-ol 2-[3,4-dichloro-5-methyl-1-(3-methylphenyl)pyrazol-4-yl]acetonitrile 5-(5-azidofuran-2-yl)-3-methoxypyridine 7-N,1-dimethyl-5-N,3-diphenylpyrazolo[4,3-d]pyrimidine-5,7-diamine [2-amino-4-(pyrrolidine-1-carbonyl)phenyl]-diethoxyazanium;chloride 1-[(2S,3R)-2,4-dimethylpent-4-enoxy]-4-ethylbenzene;5-methyl-N-[4-methylidene-6-(propanoylamino)hexyl]thiophene-2-carboxamide 2-methoxy-5-[(5S)-4,7,7-trimethyl-1-(3-nitrophenyl)-2,6-dioxo-5,8-dihydropteridin-9-ium-3-carbonyl]benzonitrile 4-methylspiro[1,2-dihydropyrido[3,4-d]pyridazine-8,4'-piperidine] 3,5-dichloro-2-[1-(oxan-4-yl)ethenoxy]pyridine 4-chloro-5-[3-[(2R)-2-ethoxypropyl]phenyl]-N-(oxan-3-ylmethyl)-1H-indazole-6-carboxamide 4-(2,3-dihydropyrazin-5-yl)-7H-purine 2-[6-fluoro-5-(4-methylpyridin-3-yl)-1H-indazol-3-yl]-4-thiophen-3-yl-1,8-dihydrocyclohepta[b]pyrrole 3-azidosulfanyl-2,4,5,6-tetrafluorobenzenethiol 2-(diethoxyphosphorylmethyl)isoindole 1-[3-ethoxypropyl(2-hydroxyethyl)amino]-2,3-dihydroindene-4-carboxylic acid 2-[3,4-dichloro-N-(1H-indol-5-yl)anilino]benzenesulfonic acid 5-chloro-6,8-difluoro-2H-pyrrolo[1,3-a]quinoxaline 2-[(7-methyl-1H-indol-5-yl)methoxy]pyrimidine [4-(2,6-dichlorophenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-fluorocyclobutyl)methanone 4-[1-[(2-ethylphenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one 4-bromo-N-[2,6-dimethyl-5-[methyl(2-pyridin-3-ylethyl)carbamoyl]phenyl]-1H-pyrrole-2-carboxamide (3-bromo-4,6-dihydropyrrolo[1,2-c]triazol-5-yl)-[6-[[1-(cyclopropylmethyl)pyrazol-3-yl]amino]pyrazin-2-yl]methanone 2-methyl-2-[1,3]thiazolo[5,4-f][1,3]benzoxazole 1-N,2-N-dimethylbenzene-1,2-disulfonamide (Z)-N'-[5-[2-[4-[1-(5-cyclopropylpyrimidin-2-yl)piperidin-4-yl]oxyphenyl]ethynyl]pyridin-2-yl]-1,3-thiazole-4-carboximidamide 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-4-[6-methoxy-7-(piperidin-1-ium-4-ylamino)imidazo[1,2-a]pyridin-3-yl]-1H-1,2,4-triazol-5-one (4S)-3,7,11-trioxatetracyclo[8.7.0.02,6.012,16]heptadeca-1(10),2(6),4,8,12(16),13-hexaen-14-amine 3-[4-[(E)-2-cyclohexylethenoxy]phenyl]propanoic acid;5-methyl-1,3-benzodioxole (1E,3Z)-1-N'-[4-(2-azidoethynyl)phenyl]-1-N'-ethylbuta-1,3-diene-1,1,2-triamine 4-chloro-N-[(Z)-2-iodoethenyl]pyridine-3-carboxamide 2-[(2S)-4-bromo-3,6-dimethyloxan-2-yl]oxy-N'-hydroxypyridine-4-carboximidamide 3-[(3R)-3-methylpiperidine-1-carbonyl]-4H-1,2,4-benzotriazin-5-one 2-[2-(3,4-dimethoxyphenyl)ethyl]-6-N,7H-purine-9,12,14-tetramine N-[(2R)-3-hydroxy-3-methylbutan-2-yl]formamide;[4-(4-pyrrolidin-1-ylanilino)thieno[3,2-d]pyrimidin-6-yl]methylazanium N-[(4Z,6E)-10-chloro-9-(diethylamino)-1-methoxydeca-2,4,6-trienylidene]-3,5-bis(trifluoromethyl)benzenesulfonamide 4-[2,3-dihydroxypropyl([1,2,4]triazolo[4,3-a]pyrazin-5-yl)amino]benzoic acid ethane;1-(4,5,6,7-tetrahydrothieno[3,2-b]pyridine-3-carbonyl)piperidine-4-carboxylic acid [2-chloro-4-(3-nitrophenyl)sulfonylphenyl]methanamine (5S)-N-methyl-5-[4-[[3-oxo-2-(trifluoromethyl)pyridazin-1-ium-1-ylidene]amino]phenyl]pyrrolidine-2-carboxamide (4S)-1,3-diphenyl-3a,6a-dihydro-[1,2]oxazolo[5,4-c]pyrrole 2-(dimethylamino)-N-[5,6-dimethoxy-1-[2-[2-(2,3,4,5-tetrahydro-1H-inden-2-yl)ethyl]-9H-fluoren-1-yl]benzimidazol-2-yl]acetamide 4-(3,5-dimethylpiperidin-1-yl)-N-(6-iminocyclohexa-2,4-dien-1-ylidene)benzamide (5S)-5,7-dimethyl-3-propan-2-yl-2,6-dihydropyrazolo[4,3-e][1,4]oxazepine 3-[2,4-dichloro-N-(1,3-thiazol-5-yl)anilino]propanoic acid 3-azido-4,5-difluoro-2-methylbenzamide N-ethylsulfonyl-N-[2-(2H-tetrazol-5-yl)phenyl]benzamide 3-(2,4-dimethylphenyl)sulfanyl-7H-pyrrolo[2,3-d]pyrimidin-6-amine 1-[4-(4-iodoanilino)piperidin-1-yl]-3,3-dimethylbutan-2-one 5-fluoro-2,4-bis(trideuteriomethyl)-6-[5-(1H-pyrazol-5-yl)benzotriazol-2-yl]pyridine-3-carbonitrile 2-amino-3,4-bis[(2-bromophenyl)sulfonyl]benzoic acid 2-fluoro-5-(3,3,4,4,5,5-hexadeuteriooxolan-2-yl)benzonitrile 1-(5,7-dichloroquinolin-4-yl)-2,3,6,7,8,9-hexahydro-1H-azepino[4,5-b]indole 4-[3-(4-oxopentoxy)propyl]benzoic acid 2-azidooxyquinoline-6-carbonitrile 3-cyclopropyl-7,8-difluoroisoquinoline 3,8-dimethoxy-1-(4-phenylbutyl)-7H-purine-2,6-dione N-[3-(2,5-dimethylphenyl)phenyl]-4-(4-propoxybenzoyl)piperidine-1-carboxamide 1-[5-(ethoxymethyl)-2,4-dimethylpyridin-3-yl]ethenamine 2-[1,3-dihydroxy-5-(3-propan-2-yloxyphenoxy)isoindol-2-yl]acetamide 2-amino-4,5-dichloro-N'-[1-(2-hydroxyphenyl)ethylideneamino]benzenecarboximidamide N-[(1S)-3,5,7a-trimethyl-2,4,9b-tetrahydro-1H-cyclopenta[c]quinolin-8-yl]-2-phenylacetamide 2-[3-(trifluoromethyl)phenoxy]cyclohexane-1,3-diamine 4-tert-butyl-2-[1-(cyclopentanecarbonyl)piperidin-3-yl]-1H-pyrimidin-6-one 1-azidooxy-2,4,5-trichloronaphthalene 1-[4-chloro-3-(trifluoromethyl)phenyl]-2,3-dihydro-1H-indene 2-[4-(1-benzothiophen-3-yl)piperazin-1-yl]-N-[(E)-but-2-enyl]-N',N'-dimethylethanimidamide 1,3-dimethylbenzo[g]quinoxaline-2,4,5,6-tetrone 2-(3-ethylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine 1-(5,6-dimethylpyrimidin-4-yl)piperidine-2-carboxylic acid [2-(5-chloropyridin-2-yl)cyclopropyl]-[4-(oxetan-3-ylmethoxymethyl)piperidin-1-yl]methanone ethane;2-(9-methylpurin-6-yl)guanidine 5-[2,3,6-trichloro-4-(1H-indol-4-yloxy)phenyl]thiadiazole 2-(3,4-dimethylphenyl)sulfonyl-N-[1-(1H-indazol-6-yl)ethylideneamino]acetamide 2-(6-methoxypyridin-2-yl)-3H-benzimidazole-5,7-diol 2-ethylsulfanyloxy-3H-benzimidazole 2-methyl-N,6-bis(4-nitrophenyl)pyridin-3-amine 1-[5-chloro-2-(difluoromethoxy)phenyl]-3-[(E)-N',N'-bis(4-methylpyrimidin-2-yl)carbamimidoyl]urea (5S)-2-[(3R,4R)-3-fluoropiperidin-4-yl]oxy-1-[4-(triazol-1-yl)piperidin-1-yl]ethanone;hydrochloride 1-[2-chloro-5-(trifluoromethyl)phenyl]hexan-1-one 1-[2-(3,4-dimethoxyphenyl)ethyl]benzimidazole N-(3,3-difluorocyclobutyl)-2-[6-fluoro-5-[(4S)-4-methyl-1,4-oxazepane-4-carbonyl]naphthalen-2-yl]acetamide 3-butylsulfanyl-2-(diethylamino)quinoline-5,8-dione [6-(cyclopropylmethylamino)pyridine-3-carboximidoyl]urea [1-(azidomethyl)piperidin-4-yl]-phenylmethanone N-[5-fluoro-3,4-dimethyl-7-(6-phenylheptoxy)naphthalen-2-yl]-1,3-thiazol-2-amine 2-chloro-N',3,4,5-tetramethylbenzohydrazide 2-[[5-chloro-3-(2,6-dioxopiperidin-3-yl)indol-1-yl]methyl]isoindole-1,3-dione 1-[4-[3,5-difluoro-2-(3-methyl-4H-azepin-7-yl)phenyl]piperazine-1-carbonyl]piperidin-4-one (3-fluorophenyl)methyl-[4-[1-hydroxy-2-[6-hydroxy-7-(methoxyamino)-2,3-dihydro-1H-inden-5-yl]ethyl]phenyl]sulfamic acid 4-[5-(1,3-benzodioxol-5-yl)-1H-pyrazole-3-carbonyl]piperazin-2-one 4-[2-(5,6-dichloro-1H-benzimidazol-2-yl)phenyl]piperazine-1-carboxylate [(E)-3-amino-2,5-bis[4-[difluoro(iodo)methyl]anilino]-1-hydroxypent-2-enylidene]azanium 4-(3-fluoropyridin-2-yl)-1,4-diazepane 4-[3-azidopropyl-(1,3-benzodioxol-5-ylmethyl)amino]butanamide 1-[3-[7-[(3,5-dichlorophenyl)methylamino]-2-oxo-4H-3,1-benzoxazin-1-yl]phenyl]-3-ethoxyurea 3-[2-(7-bromoimidazo[1,5-a]pyridin-1-yl)ethynyl]-N'-hydroxybenzenecarboximidamide 7-(2,5-dimethylphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine (2S)-4-[(1,5-dimethyl-3-oxopyrazol-4-yl)sulfonylamino]-2-hydroxybutanoic acid 5-cyclopropyl-3-[4-[(4-oxo-1-phenylpiperidine-2-carbonyl)amino]-1,3-thiazol-2-yl]pyrazine-2-carboxylic acid 1-amino-3,4-bis[(4-methoxyphenyl)sulfanyl]butan-2-one 2-chloro-4,7-dimethyl-1H-[1,3]thiazolo[5,4-b]pyridine 2-(cyclopropylmethoxy)-4-[6-[3-[(2R,5S)-2,5-dimethylpiperazine-1-carbonyl]anilino]pyrimidin-4-yl]benzoic acid 2-(3,5-difluorophenyl)-1-[3-hydroxy-3-(triazol-1-ylmethyl)piperidin-1-yl]ethanone 1-[(3R)-3-azidopyrrolidin-1-yl]-2,2,2-trifluoro-N-[[4-(1-methylpyrazol-3-yl)phenyl]methyl]ethanimine (E)-1-[2-(4,6-dimethylpyrimidin-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-7-yl]pent-1-en-3-one 4-amino-5-hydroxynaphthalene-2,7-disulfonic acid 3-(4-bromophenyl)-1-[7-fluoro-6-(hydroxymethyl)-2,3-dihydropyrido[3,2-b][1,4]oxazin-1-yl]propan-1-one N-[(1S,2R)-1,3-dihydroxypropan-2-yl]-4-propan-2-yl-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide 2-(8-iodoquinazolin-4-yl)phenol 2-bromo-6-[(4-nitrophenyl)iminomethyl]phenol 5-(methoxycarbonylamino)pyridine-3-carboxylic acid N-(2,4-dichloropyrimidin-5-yl)-4-nitro-N-[4-(thiophen-2-ylsulfamoyl)phenyl]benzamide N-[4-(methylamino)phenyl]sulfanyl-1,3-thiazol-5-amine;propane N-[3-(1,2-dihydroimidazol-5-yl)phenyl]-4-fluorobenzamide 2-[[3-cyano-5,7-diethyl-6-methoxy-4-(3-nitrophenyl)-1H-indol-2-yl]methylidene]propanedinitrile 1-[(3R,4S)-3-[5-chloro-2-[6-fluoro-4-(1H-pyrazol-5-ylamino)quinazolin-7-yl]oxyethyl]-4-hydroxypiperidin-1-yl]ethanone (3E)-2,2-dimethyl-4-[1-[(4-pyrazol-1-ylphenyl)methyl]imidazol-2-yl]penta-3,5-dienoic acid N-[1-(2,4-dichlorophenyl)ethyl]-6-fluoroquinoline-3-carboxamide 1-[3-(2,4-difluorophenyl)cyclobutyl]pyrrolidine;N-(4-methoxyphenyl)formamide 7-methyl-3,4-dihydro-2H-thiochromene-5-thiol N-[(2S)-1-amino-3,3,3-trifluoropropan-2-yl]-4-cyclohexa-1,5-dien-1-ylbenzamide (2S)-4,6-difluoro-7-[1-[3-(5-methylpyrimidin-2-yl)propanoyl]azetidin-3-yl]oxy-2-(phenylmethoxycarbonylamino)heptanoate 3-chloro-2-[3-(4-ethylanilino)propoxy]phenol;hydrochloride 2-[4-(cyclohexylmethylamino)phenoxy]acetamide 6-chloro-1,2-dihydronaphthalene;4-chloro-3-fluorobenzenesulfonic acid 5-azido-3,4-dihydro-1H-pyrido[2,3-b]pyrazine-2,7-dione 4-[3-amino-6-(1,2-dimethylpyridin-1-ium-3-yl)pyrazin-2-yl]benzonitrile 3-(3,5-dichlorophenyl)-N-[(4S)-7-methoxy-2,2-dimethylheptan-3-yl]prop-1-enamide 2-chloro-N-[1-(3,5-dimethylpyridin-2-yl)piperidin-4-yl]acetamide 1-(5-ethyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-3-yl)-N',N'-dimethyl-N-[2-oxo-2-[(3E)-penta-1,3-dien-3-yl]oxyethyl]methanediamine 1-chloro-4-[(5E)-3,3-dimethylhepta-1,5-dien-2-yl]benzene;4-ethyl-1-(3-methoxyphenyl)piperidine 3-[2,6-dichloro-4-nitro-N-(1-phenylpropyl)anilino]butanoic acid 3-azido-6-methylacridine N-[(1R,2S)-2-methyl-1H-inden-1-yl]dibenzofuran-3-amine 2-(9H-fluoren-9-ylmethoxycarbonylamino)-5-(propanoylamino)pentanoic acid 5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)thiophen-2-amine 6,7-dimethoxy-2,3-dihydroindene;3-phenylcyclopropane-1-carbonitrile 2,4-dichloro-5-fluoro-6-[(3R)-3-methylpyrrolidin-1-yl]pyrimidine 6-bromo-1,3-dimethylindole 2-(5,8-dichloro-3,4-dihydro-1H-isoquinoline-2-carbonyl)benzenesulfonamide 5-[(3-bromophenyl)methyl]-2,3,6-trimethoxyphenol 4-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxybenzaldehyde;chloromethane [5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]urea 5-[2-amino-4-[(E)-1-amino-3-iminoprop-1-en-2-yl]phenyl]sulfanyl-3H-triazin-4-one N-[1-[3,5-bis(trifluoromethyl)phenyl]ethylsulfanyl]-2,6,6-trichlorohexa-1,3-dien-1-amine 5-N-cyclopentyl-1H-pyrimidine-2,4-dione N-[2,4-difluoro-3-[5-(3-fluoropyridin-4-yl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]propane-1-sulfinamide 3-[(6S)-6-ethyl-2-cyclopropylmorpholine-4-carbonyl]-5,7-dihydropyrrolo[3,2-d]pyrimidin-4-one [4-(2,5-dimethylphenyl)piperazin-1-yl]-(6,7-dihydro-5H-cyclopenta[b]pyridin-3-yl)methanone (E)-3-(4-butoxyphenyl)-N-[(2R,3S,5R)-6-hydroxy-3-phenoxazin-10-yloxan-2-yl]prop-2-enamide 6,7-dimethyl-1'-[(4-propanoylphenyl)methyl]spiro[5,8-dihydropteridine-2,4'-piperidine] (3S)-3-[3,5-dimethyl-4-oxo-6-[4-(trifluoromethyl)phenyl]pyrimidin-2-yl]sulfanylpentanenitrile 4-[(2,6-dichlorobenzoyl)amino]-3-hydroxy-N-methylpyridine-2-carboxamide 4-(2,3-dihydroxypropoxy)-3-iodobenzenesulfonamide 6-methoxy-N-(oxan-4-yl)pyrazine-2-carboxamide N-(4-chlorophenyl)-2-[3,7-dimethyl-5-oxo-1-phenyl-6-[3-(trifluoromethoxy)phenoxy]thieno[2,3-d]pyridazin-4-ylidene]acetamide 1-(2,5-difluorophenyl)piperidine 3-[3,5-bis(trifluoromethyl)phenyl]-1,2-oxazol-4-amine 5-bromo-N-(3,4-dimethoxyphenyl)pyrimidine-2-carboxamide 1-(4,6-diaminopyrimidin-5-yl)ethanone;hexane;2-methoxy-3-pentoxypropane 2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-ium-3-yl)-5-ethyl-6-[methoxy-[1-[[(E)-2-(methylideneamino)prop-1-enyl]-propylcarbamoyl]piperidin-4-yl]amino]-3H-pyrrolo[3,4-f]benzimidazole-7-carboxylic acid 5-methylspiro[chromene-2,3'-pyrrolidine] (2R)-N-[2-[[2-ethyl-5-(1,3-thiazol-4-yl)benzoyl]amino]-4-methoxyphenyl]pyrrolidine-2-carboxamide (5E)-5-[2-(3,4-dichlorophenyl)sulfanylpropylidene]-1-(4-phenoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione N-[(3R,4S)-1-benzyl-4-[[6-(2-oxopyrrolidin-1-yl)pyridine-3-carbonyl]amino]piperidin-3-yl]-5-methyl-6H-1,2,4-oxadiazine-3-carboxamide ethane;2-methylhexane;4-[1,1,2,2-tetrafluoro-5-(3,5,7-trimethyloctoxy)pentan-3-yl]benzoic acid 4-[(2,6-dichlorobenzoyl)amino]-1H-pyrazole-5-carboxylic acid 1-[(Z)-[(3,5-dibromophenyl)hydrazinylidene]methyl]naphthalen-2-ol 2-N,4-N-bis[5-bromo-6-(methylamino)pyrimidin-4-yl]cyclohexa-1,3-diene-1,2,4-triamine 2-(5,7-dimethyl-1H-indol-3-yl)ethanol;2-[3-hydroxy-4-[2-hydroxy-3-(morpholine-4-carbonylamino)propoxy]phenyl]-N-(oxolan-3-yl)acetamide [5-chloro-2-(2-methylanilino)pyridin-3-yl]oxyboronic acid 4-[[1-(2,3-dihydro-1H-indene-2-carbonyl)piperidin-4-yl]methoxy]-5-cyclopropyl-2-fluorobenzoic acid 2,4-dimethyl-6-[3-methylidene-5-(1-methylpyridin-1-ium-2-carbonyl)cyclohexen-1-yl]pyridazin-3-one (1R)-3-[[2-[4-(2,4-dioxo-1H-quinazolin-6-yl)piperazin-1-yl]acetyl]amino]-N-methylidenecyclopentane-1-carboxamide 3-chloro-N-cyclopropylsulfanyl-2,4-difluoroaniline 5-bromo-2-(1,4-dimethyl-3H-pyrrol-2-ylidene)-6-[4-[1-methoxy-2,2-bis(sulfanyl)ethyl]piperazin-1-yl]-3H-pyridine 2-(4-chlorophenyl)-3,5-dimethyl-6-pentan-3-yloxy-1H-pyrazolo[1,5-a]pyrimidin-7-one 2-bromo-N-hexyl-N-(1,2,4-triazol-4-yl)benzamide 4-chloro-N,2,6-trimethylaniline;ethane 5-(4-methoxyphenyl)-N-[3-(1H-pyrrol-2-yl)phenyl]-1,3,4-thiadiazol-2-amine 3-[(3R,4S)-1-benzyl-4-hydroxypyrrolidin-3-yl]-N-cyclopentylpropanamide;hydrochloride ethane;N-[4-(5,7,11,12-tetrazatricyclo[7.4.0.02,6]trideca-1,3,6,8,10,13-hexaen-13-yl)phenyl]acetamide N-[2-amino-3-fluoro-4-[6-(morpholine-4-carbonyl)pyridin-2-yl]phenyl]-5-methoxypyrazine-2-carboxamide 2-[4-(7,8-dichloro-5,6-difluoronaphthalen-2-yl)oxyphenyl]ethanol N-[(4,5-dimethyl-1,3-thiazol-2-yl)methyl]-3-(imidazol-1-ylmethyl)piperidine-1-carboxamide N-(1,4-dioxan-2-ylmethyl)-2-(3-hydroxy-3-methylpiperidine-1-carbonyl)-6-methylpyridine-4-carboxamide 4-methyl-N'-[3-[6-methyl-3-(4-phenylpiperazine-1-carbonyl)indol-1-yl]prop-1-enyl]benzenecarboximidamide 2-[6-chloro-4-(trifluoromethyl)pyridin-3-yl]oxypyridine 1-[6-(trifluoromethyl)pyridin-3-yl]butan-2-one 2-cyclobutyloxy-6-(4-methylsulfinylpiperazin-1-yl)pyridine-3-carboxamide 2-[(4aS,8aR)-3-methyl-1-oxo-6-phenyl-2,4,5,7,8,8a-hexahydropyrrolo[1,2-d][1,4]diazepine-9-carbonyl]benzonitrile;formic acid 2-[4-[(3R)-1,5-dioxohexan-3-yl]sulfonylphenyl]acetic acid 2-(5,6-dimethylnaphthalen-1-yl)oxyethanamine 4-[(1S)-1,2-difluoroethyl]-N-[4-fluoro-3-[[7-oxo-8-propan-2-yl-6-(trideuteriomethoxy)pyrido[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidine-1-carboxamide 2-[4-(hydroxymethyl)-3-phenyl-1,3-thiazolidin-5-ylidene]acetic acid [(1-cyclopentylpiperidin-4-ylidene)methoxy]methanol 5-[(2S)-2-[3,4-bis(trifluoromethyl)phenyl]pyrrolidine-1-carbonyl]furan-2-sulfonamide 1-azido-2-butan-2-yloxy-3-methoxybenzene 4-benzyl-3-methoxycarbonyl-1,2,5-oxadiazole-4-carboxylic acid 3-[2,6-dichloro-4-[(2-phenylimidazo[1,5-a]pyrazin-8-yl)amino]benzoyl]iminopropanoic acid 4-[(2-methoxybenzoyl)amino]quinoline-7-carboxylic acid (3E,5Z)-6-amino-4-(methylamino)hexa-1,3,5-trien-2-ol;N'-[3-formamidopropanoyl(propyl)amino]naphthalene-2-carbohydrazide N-[2-[4-(hydroxymethyl)phenyl]propan-2-yl]pyrazine-2-carboxamide 7-(6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazine-7-carbonyl)-3-methoxy-2H-isoquinolin-1-one N-[(5R)-3,4-dihydro-2H-chromen-5-yl]-5-methylthieno[2,3-d]pyrimidin-1-ium-6-amine N-[1-(2-cyanopyrimidin-4-yl)cyclohexyl]cyclopropanesulfonamide 1-[6-chloro-2-(5,8-dioxoquinolin-6-yl)pyrimidin-4-yl]azetidine-3-carboxylic acid (2E)-N,3-dimethyl-2-(4H-quinolizin-2-ylidenehydrazinylidene)butanamide;ethane 2-(3-methylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine N-[(2S)-1-(aminomethylideneamino)-3-methylbutan-2-yl]benzamide 2-[4-chlorobutyl(hexyl)amino]-4-nitrophenol 1-ethyl-2-methyl-5H-pyrazolo[4,3-c]quinolin-3-one 3-bromoprop-2-enal;methanamine;6,7,11,12,14-pentamethyl-8-thia-9,11-diazatetracyclo[7.7.0.02,7.010,15]hexadeca-1(16),2(7),3,5,10,13-hexaene 5-[(2R,4S)-2-[4-(5-chloropentylamino)phenyl]-4-hydroxypyrrolidin-1-ium-1-carbonyl]pyridine-3-carbonitrile (1-azido-2,3-dihydroisoindol-1-yl)phosphane 3-[(4aR,8aS)-2-ethylsulfonyl-4a-methyl-3,4,5,6,7,8,8a-octahydro-1H-isoquinoline-6-carbonyl]benzamide 2-[(2,4-dimethoxyphenyl)methylimino]-5,6-diethoxy-5-hydroxycyclohex-3-en-1-one 2-(azetidine-1-carbonyl)-N,4-dimethyl-5-nitrobenzenesulfinamide 4-[2-[4-(2,3-difluorocyclopropyl)phenyl]phenyl]piperidine 7-methoxy-3-[1-(2,4,6-trifluorophenyl)ethenyl]chromen-4-one 2-[5-chloro-3-(4-methylphenyl)sulfonylindol-1-yl]acetic acid 3-amino-5-[3-methoxy-2,6-di(propan-2-yl)phenyl]imidazole-4-carbonitrile 4-[5,6-dideuterio-2-(trifluoromethyl)phenoxy]-N'-hydroxybenzenecarboximidamide 3-bromo-4,5-difluorobenzenesulfonic acid (1E,3Z)-2-ethenyl-4-[6-(1H-indazol-5-ylamino)pyridine-3-carbonyl]buta-1,3-diene-1,4-diamine;methanol 3-[4-(trifluoromethoxy)phenyl]azetidine (E)-1-[4-[8-chloro-7-hydroxy-6-(2-oxopropoxy)quinolin-4-yl]piperazin-1-yl]-3-cyclopentylprop-2-en-1-one 4-(1,3-benzothiazol-2-yl)-N-[4-(hydroxymethyl)cyclohexen-1-yl]piperazine-1-carboxamide 1-[4-(2,3-dichloro-4-iodophenyl)-6-methyl-5H-pyrrolo[3,4-c]pyridin-1-yl]propan-2-ol 3-(2,4-difluorophenyl)sulfonylpiperidine 5-(4,6-dimethylcyclohexa-1,3-dien-1-yl)oxy-2H-benzotriazole 2-methyl-N-[5-(6,7,8,9-tetrahydro-1H-pyrrolo[3,2-h]isoquinoline-2-carbonyl)pyridin-3-yl]benzamide N-(3,4-dimethoxyphenyl)-2-[(6S)-5-oxo-2-phenyl-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]acetamide 2-[(3-chlorophenyl)methyl]-4-fluorobenzaldehyde;methanol N-benzyl-6-[2-(2-bromophenyl)ethyl]pyridine-3-carboxamide N-[(E)-1-(4,5-dimethoxycyclohexa-2,4-dien-1-yl)-2-methylbut-1-enyl]-N'-(1-pyridin-4-ylethylideneamino)propane-1,3-diamine 1-[[2,5-bis(trifluoromethyl)phenyl]methyl]-N-methoxy-6-oxo-4-pyridin-3-ylpyrimidine-5-carboxamide N-[2-(2,4-dimethylphenyl)propan-2-yl]-2-pyridin-3-ylacetamide (7-chloro-3,4-dihydro-2H-1,5-benzodioxepin-6-yl)methanimine N-[5-(4,7-dimethoxyquinazolin-6-yl)-2-methoxypyridin-3-yl]benzamide 2,2-dichloro-3-[5-iodo-4-(trifluoromethyl)pyridin-3-yl]cyclopropane-1,1-dicarbonitrile 4-[[3-[(3S)-3-[(2,5-dimethylpyrazole-3-carbonyl)amino]pyrrolidin-1-yl]pyridin-4-yl]amino]-N-propan-2-yl-6-(trifluoromethoxy)quinoline-7-carboxamide 5-chloro-N-(2,6-dioxopiperidin-3-yl)-1H-imidazole-4-carboxamide;toluene N-(4-aminocyclohexyl)-5-fluoro-2-pyrrolidin-1-ylpyrimidine-4-carboxamide 3-(2,4-difluorophenyl)sulfanyl-N'-hydroxy-5,6-dimethylpyridazine-4-carboximidamide (3R)-1-benzylsulfonyl-N,2-dimethylpyrrolidine-3-carboxamide 2-(5,6-dimethylpyrimidine-4-carboximidoyl)-N-(6-methoxypyridazin-3-yl)-1H-indol-6-amine 2-[6-(hydroxymethyl)-7-methoxy-5-(1,3-oxazol-4-yl)thieno[3,2-b]pyridin-2-yl]-1-pyrrolidin-1-ylethanone 3-[2-(cyclopropylmethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-hydroxy-5-oxoimidazolidine-4-carboxamide 2-[3,5-dimethyl-1-(4-oxo-3H-quinazolin-7-yl)pyrazol-4-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide 4-[2-(aminomethyl)-5-chlorophenyl]phenol 2-(3-azidopropyl)-6-methoxyphenol (5S)-2,4-dimethylheptane;N'-[4-(1H-imidazole-5-carbonylamino)naphthalen-1-yl]butanediamide 1-(4,4-difluorocyclohexyl)-2-[6-(1H-pyrazol-5-yl)isoquinolin-3-yl]ethanone N-[5,7-dimethoxy-2-[2-(3-morpholin-4-ylsulfonylanilino)pyrimidin-4-yl]-1H-inden-1-yl]propanamide 4-[2-(4-methylsulfonylphenyl)ethylamino]-N-pyrimidin-4-ylbenzamide [2,6-diamino-5-(4-hydroxyphenyl)pyrimidin-4-yl]oxymethylphosphonic acid 2-[(5,6-difluoro-1H-indol-3-yl)methyl]-4-morpholin-4-ylbenzimidazole-1-carboxamide 4-methylsulfanyl-N-[6-[4-(pyridine-3-carbonyl)piperazine-1-carbonyl]pyridin-2-yl]piperidine-1-carboxamide N-[(1S)-5-(4-fluorophenoxy)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-yl]-3-methylbutanamide 3-(N-(2,4-dichloropyrimidin-5-yl)anilino)butanoic acid N-butyl-6-hydroxy-5-[(2R,3S)-1-pyridin-4-yl-5-pyridin-3-yloxypentan-2-yl]pyrimidine-4-carboxamide N-[(Z)-(4-hydroxyphenyl)methylideneamino]-3-methyl-1,2-thiazole-5-carboxamide 1-amino-3-[4-(4-tert-butylphenoxy)piperidine-1-carbonyl]pyridin-2-one (2S)-2-[3-[4-(1H-benzimidazole-2-carbonylamino)phenyl]sulfonylanilino]propanoic acid 2-amino-4-[2-fluoro-5-(trifluoromethyl)phenyl]-6-methylbenzene-1,3-dicarbonitrile N-[(Z)-[4-cyclopentyl-3-ethoxy-5-iodo-2-methyl-1H-pyrrol-3-yl]methylideneamino]aniline 3-[4-hydroxy-5-(6-methoxypyridin-2-yl)-2,5-dioxoimidazolidin-1-yl]propanoic acid N-(1-acetyl-4,5-dihydroimidazol-2-yl)-7H-pyrrolo[3,2-d]pyrimidine-6-carboxamide (4-chloronaphthalen-1-yl)oxymethanesulfonic acid 7-amino-5-[2-(3-methoxyphenyl)sulfanylphenyl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 3-bromo-4-ethyl-2-(trifluoromethyl)benzoic acid N-(1,5-dimethylpyrazol-4-yl)-2-[2-ethoxy-6-propan-2-yl-3-(2H-tetrazol-5-yliminomethyl)phenyl]acetamide 5-(1,3-dioxolan-2-yl)-N-[5-(ethoxymethyl)pyrimidin-4-yl]thiophene-2-sulfonamide 5-(2,4-dimethoxyphenyl)-1-[(3-fluoropyridin-2-yl)amino]pyrazole-4-carboxylate 3-(azetidin-1-yl)-N',2-diphenyl-5H-pyrrolo[2,3-b]pyrazine-7-carboximidamide 4-[[(1R,2S)-1-cyclopropyl-2-methylsulfonylcyclopropanecarbonyl]amino]pyridine-3-carboxamide 2,4-dichloro-N-[1-(5-cyclohexylpyridine-3-carbonyl)pyrrolidin-3-yl]benzamide (E)-3-amino-2-[[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]oxymethyl]but-2-enedioic acid N-[(3S,4R)-1-tert-butylpiperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 6-methyl-2-[4-(trifluoromethoxy)phenoxy]pyridine-3-carboxylic acid 2-[(2E,5Z)-4-chlorohepta-2,5-dien-3-yl]-N-ethyl-1H-imidazole-5-carboxamide 3-[4-(hydroxymethyl)phenyl]sulfonylcyclobutane-1-carboxamide 2,2-dichloro-3-[4-methoxy-3-(trifluoromethyl)phenyl]cyclopropane-1,1-dicarbonitrile 3-methyl-2-(naphthalen-1-ylmethoxy)-3,4-dihydro-2H-quinoline [1-(2-chlorophenyl)pyrrolidin-3-yl]-[4-methoxy-3-(trifluoromethyl)anilino]methanol (2R,4S)-N-[(Z,3E)-1-amino-3-hydroxyiminoprop-1-enyl]-4-methoxy-1-methylpiperidine-2-carboxamide;dihydrochloride 1-[(E)-2,3-difluorohex-2-enyl]-5-[6-[(3R)-pyrrolidin-3-yl]oxypyridin-3-yl]indazole 1-(2,6-dichloro-3-nitrophenyl)sulfonyl-4-piperidin-1-ylindole 2-amino-5-(1H-pyrrolo[3,2-b]pyridine-6-carbonyl)cyclohexane-1,3-dione N-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]aniline 3-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-1-naphthalen-2-ylimidazolidine-2-thione N-(5-chloropyrimidin-2-yl)-5-fluoro-4-(1H-indol-3-yl)-6-methoxycyclohexa-2,4-dien-1-imine (2Z)-4,5-dimethylhepta-2,6-diene;1-[1-(4-methylphenyl)sulfinylpiperidin-3-yl]propan-2-one 4-amino-N-[(2S)-1-hydroxypropan-2-yl]-3,5-dimethoxybenzamide 2-[6-(2,4-dimethylphenoxy)pyridin-3-yl]-N-[[5-(furan-2-yl)-1H-pyrazol-4-yl]methyl]acetamide 5-[2,6-bis(4-fluorophenyl)phenyl]triazinane;formaldehyde 3-[3,4-difluoro-2-(2-fluoro-4-methylanilino)phenyl]propanoic acid 2-[(6,7-dihydropurin-8-yl)oxy]-N'-hydroxypyridine-4-carboximidamide (4E)-4-[[3,5-bis(trifluoromethyl)phenyl]methylidene]-2-chloro-6,7-dihydro-1H-benzimidazole N-cyclopentyl-6-[(1,3-dimethylindazol-5-yl)amino]pyridine-3-carboxamide 1-(4-hydroxy-2-naphthalen-1-ylphenyl)-2,2-dimethylpropan-1-one 1-[3-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]butanoylamino]-5,6,7,8-tetrahydro-4H-cyclohepta[c]pyrazole-3-carboxamide 2-(4-acetylphenyl)-1H-1,5-benzodiazepine-3-carbonitrile 2-(4,6-dimethyl-1H-benzimidazole-5-carbonyl)-N'-[(1S,3R)-3-phenylcyclopentyl]acetohydrazide 1-(2-methylpyridin-4-yl)-3H-pyrrolo[2,3-b]pyridine N-(6-chloropyridin-3-yl)-N-ethenylsulfonylbutanamide 3-[(E)-2-nitroethenyl]-4,5-dihydrobenzo[e]benzotriazole 4-(2,5-dihydroxyphenyl)sulfanylbenzoic acid 1-phenyl-2H-quinazoline N-[1-(4-ethylphenyl)propyl]-2,6-difluorobenzenesulfonamide 4-chloro-3,5-diiodothiophene 2,3-dimethyl-5-oxo-N-[(6-oxo-1H-pyrimidin-4-yl)methyl]-1H-pyrazole-4-carboxamide 2,4-dihydroxy-5-octylbenzenesulfonamide 2-hydroxy-3-(pyridin-2-ylamino)propanamide 6-[(4-bromophenyl)methoxy]-N'-hydroxypyridine-2-carboximidamide (E)-1-aminoprop-1-en-2-ol;ethane;4-methyl-N-[5-(oxan-4-ylamino)pentanoyl]benzamide N-[3-(hydroxymethyl)oxetan-3-yl]-4-phenylbenzamide 2-(methoxymethyl)-1'-[2-(4-phenylpiperidin-1-yl)acetyl]spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,3'-piperidine]-4-one 6-[(2S)-3-methylbutan-2-yl]quinoline N-[1-(6H-benzo[c]quinolizin-5-ium-11-yl)ethenyl]-4-(trifluoromethoxy)aniline N-(4,6-dimethylpyrimidin-2-yl)-5-ethoxypyrazolo[1,5-a]pyridine-3-carboxamide 2,4-dichloro-6-(2H-triazol-4-yl)phenol 1-(4,4-dimethylhexan-2-ylamino)-3-[(4-fluorophenyl)methoxy]propan-2-ol 1-[6-[5-[(2R,4S)-1-acetyl-2-cyclopropylpiperidin-4-yl]oxypyridine-3-carboximidoyl]pyridin-2-yl]-3-[(1R)-1-phenylethyl]urea 3-(2,4-difluorophenyl)azetidine-1-carboxylic acid 1-[(Z)-3-(4-nitropyrazol-1-yl)prop-1-enyl]sulfonylpiperidine N-[3,5-bis(trifluoromethyl)phenyl]-1H-indol-4-amine 2-(4-fluorophenyl)-5,6,7,8-tetrahydroquinoline 4-(2-chloro-6-fluorophenyl)-7,8-dihydroimidazo[1,2-a]pyrimidine 3-(3,5-difluorophenyl)-N-(1H-indazol-6-yl)propanamide 2-chloro-N-[3-(4,6-difluoro-1H-benzimidazol-5-yl)propyl]acetamide 2-[2-[4-amino-7-(piperidin-4-ylmethoxy)quinazolin-2-yl]phenoxy]propanoate 6-(2,6-difluorophenyl)-5-[4-[3-methyl-1-(pyridine-4-carbonyl)azetidin-3-yl]oxyphenyl]pyrazine-2-carboxamide;ethane N-[4-(cyclohexylamino)-3,4-dioxo-1-[2-oxo-2-(quinolin-4-ylmethylamino)ethyl]azetidin-2-yl]formamide;ethane 2-(4-cyclopropyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6-carbonyl)-1H-imidazole-4,5-dicarbonitrile N-[2,4-difluoro-3-(1H-indole-2-carbonyl)phenyl]-2-fluoropropane-1-sulfonamide N-(2,4-dichloropyrimidin-5-yl)-N-[4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]-1-methoxy-3-methylbutan-2-amine 2-azido-N',3-dimethoxybenzenecarboximidamide 2-[3,5-dichloro-4-(2,2,2-trifluoroethoxy)phenyl]sulfanylacetic acid 5-hydroxy-1,8-dimethoxy-4H-chromeno[3,4-c]pyridine N-[(1S,2R)-2-hydroxycyclobutyl]thieno[3,2-b]pyridine-7-carboxamide 1-methyl-N-[4-(2-oxopropylamino)phenyl]imidazole-2-carboxamide N-[(3S,4R)-1-(cyclopropylmethyl)-4-thiophen-2-ylpyrrolidin-3-yl]-3-phenylpropanamide;hydrochloride 1-[4-(trifluoromethylsulfanylamino)phenyl]sulfonylpiperidine-2-carboxylic acid 3-butylbenzenesulfonic acid 2-(4-butoxyphenyl)propanoate N-[2-methyl-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyridin-3-yl]methanesulfonamide 3-[[6,7-dimethoxy-4-(2H-quinolin-1-yl)phthalazin-1-yl]amino]-5-fluorophenol (E)-2,3-diamino-3-[4-methyl-5-(1-piperidin-1-ylethenoxy)pyridin-2-yl]prop-2-enenitrile 1-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)azepane-4-carbonitrile 2-azido-1,3-dimethylindole 1-(4-propylthiadiazol-5-yl)nonan-3-ol (2R)-2-[(4-chloro-3-nitrophenyl)methyl]-4-hydroxy-N-propan-2-ylpentanediamide 1-[5-cyano-2,3-dimethyl-6-(2-methyl-4-propan-2-ylphenyl)-4H-pyridin-4-id-7-yl]-3-cyclopentylurea;iridium N-cyclohexyl-1,2,3,4,5,6-hexahydroindolo[2,3-b]quinoline-11-carboxamide 1-[4-chloro-3-(2-phenylethoxy)pyridine-2-carbonyl]piperidine-4-carboxylic acid 1-[(2-fluorophenyl)methyl]-N-[2-oxo-1-(2,2,2-trifluoroethyl)piperidin-3-yl]pyrazole-4-carboxamide 2-[[5-chloro-4-methyl-1-(3-morpholin-4-ylpropoxy)indole-7-carbonyl]amino]spiro[3.3]heptane-6-carboxylic acid N-azido-4-(1H-benzimidazol-2-yl)pentanamide 1-[3,5-bis(trifluoromethyl)phenyl]-2-(4-nitropyrazol-1-yl)ethanol 1-azido-2-chloro-4-(cyclopropylmethoxy)benzene 1-[3-(4-fluorophenyl)pyrrolidin-2-yl]sulfonyl-2-propan-2-ylpiperidine 1-N,6,8-trimethylisoquinoline-1,2-diamine (2R,3S)-N,1,5-trimethyl-2-pyridin-3-ylpyrrolidine-3-carboxamide 1-cyclopropyl-N'-[(4S)-2-(2,6-dichlorophenyl)-5-oxopyrrolidine-3-carbonyl]-N'-methylmethanesulfonohydrazide (E)-1-[4-[5,6-difluoro-7-[1-[1-(4-methylphenyl)ethoxy]ethenyl]quinolin-4-yl]piperazin-1-yl]-3-(1H-indol-2-yl)prop-2-en-1-one N-[5-cyano-4-(3,4-difluorophenyl)-6-methylpyridin-2-yl]-4-methoxybutanamide N-(1,3-benzothiazol-2-yl)-4-chloro-N'-hydroxy-5-(trifluoromethylsulfanyl)thiophene-2-carboximidamide 2-methyl-2-[3-(1H-pyrrol-2-yl)phenyl]propanenitrile N-[4,5-bis(ethenyl)furan-2-yl]hydroxylamine N-[2,4-difluoro-3-[5-(6-piperidin-1-ylpyridin-2-yl)pyrazolo[4,3-b]pyridin-2-yl]phenyl]benzamide 2-azidooxy-N,N-dimethyl-4-(trifluoromethyl)aniline 2-[2,6-difluoro-4-(1-propan-2-ylpiperidine-4-carbonyl)phenyl]iminoacetamide 2-N,6-N-bis[2,6-di(propan-2-yl)phenyl]pyridine-2,6-dicarboxamide;1H-pyrazol-5-olate;tin(4+) 2-(cyclopropylmethoxy)-1-[6-(2,5-dimethylphenyl)pyridine-3-carbonyl]pyrrolidine-2-carboxamide (Z)-2-[[6,9,11-trioxo-7-(propylamino)anthracen-2-yl]methylideneamino]-3-trityloxyprop-2-enamide 4-[(2-fluorobenzoyl)amino]-N-methylbutanamide N-butanoyl-3,5-dichloro-4-methylthiophene-2-carboxamide 2-(2,4,6-tribromophenoxy)benzonitrile 3-[2,6-difluoro-N-(3-methylbut-2-enyl)anilino]propane-1,2-diol 3-(4,5-dichloro-1H-indol-3-yl)propanoic acid 3-(2,4-dimethylphenyl)-7-[4-(4-fluoro-2-hydroxyphenoxy)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide 4-azido-2,5,6-trichlorobenzenesulfonic acid N-[(E)-(3,4-dichlorophenyl)methylideneamino]-2-(pyridine-3-carbonylamino)pyridine-4-carboxamide 2-chloro-1-[4-[5-(3,5-difluorophenyl)-5-methylhexan-2-yl]piperazin-1-yl]ethanone 1-[(2R,5S)-5-hydroxypyrrolidine-2-carbonyl]-4-hydroxy-N'-(3-methylphenyl)piperidine-4-carboximidamide 1-(2,5-dimethylpyrazol-3-yl)-N-[(4R,6S)-6-phenylpiperidin-3-yl]cyclopropane-1-carboxamide 4-methylsulfanyl-N'-[5-methyl-2-[2-(trifluoromethoxy)phenyl]-1,3-thiazol-4-yl]benzohydrazide 4-N,4-N-diethyl-2,5-bis(4-fluorophenyl)imidazole-1,4-dicarboxamide 2-(4-chlorophenyl)-5,6,7,8-tetrahydro-3H-pyrido[3,4-d]pyrimidin-4-one 1,3-dihydroxy-6,9-dioxoxanthene-2,7-disulfonic acid;4-[[(Z)-2-[2-(methylamino)phenyl]-3-oxoprop-1-enyl]carbamoyl]benzonitrile 4-[2,3-dihydroxypropyl(1,1,1,2,3,3,3-heptafluoropropan-2-yl)amino]-N-pyridin-2-ylbenzenesulfonamide 5-[[(4S)-2-amino-1,3-thiazolidine-4-carbonyl]amino]-N,2-dimethylpyrazole-3-carboxamide N-[5-[2-(dimethylamino)ethyl-[3-(2,3-dioxopyrrolidin-1-yl)propyl]amino]naphthalen-1-yl]quinoline-8-sulfonamide N-(6,8-difluoro-1H-imidazo[4,5-b]pyridin-2-yl)cyclopropanesulfonamide 3-(4,5-dimethyl-1H-pyrrol-2-yl)-5-[[2-fluoro-6-methoxy-4-[2-(4-methylpiperazin-1-ium-1-ylidene)hydrazinyl]phenyl]carbamoylamino]benzoic acid 2-cyclopropyloxy-N-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-ylmethyl)acetamide 2-(3,4-dichlorophenyl)-N-[1-(6-fluoro-1H-benzimidazol-2-yl)propan-2-yl]acetamide 3-methyl-N-[(1S)-1-phenylethyl]-1,2,4-oxadiazole-5-carboxamide 2-bromo-1,5-bis(phenylsulfanyl)pyrrole N-[4-[4,5-bis(ethenyl)-1H-imidazol-2-yl]phenyl]sulfanylacetamide 1,2-dichlorobenzene;ethane 2-[(E)-1,3-bis(4-hydroxyphenyl)prop-2-enylideneamino]oxybutanamide 6-[(2-methoxypyridin-4-yl)methylamino]-3-methylidene-1,5-dihydroimidazo[2,1-b]quinazolin-2-one 3-(2,2-dimethylpropanoyl)-5-[1-[(3R)-3-fluoropyrrolidin-1-ium-1-ylidene]ethyl]-N-methoxy-4-oxothieno[3,2-c]quinoline-9-carboxamide 2-(3,5-ditert-butylphenyl)quinoline N-[1-(4-chlorophenyl)ethenyl]formamide;N',2,3-trimethylpropanimidamide 4-[[1-[2-(6-fluoro-4H-1,3-benzodioxin-8-yl)ethyl]piperidin-3-yl]methoxy]-5-iodo-1H-pyridazin-6-one 3-(4-butoxy-N-methoxycarbonylanilino)propanoic acid 6-amino-7-methylsulfonyl-3H-quinazolin-4-one [5-[4-(3,5-dimethoxyphenyl)-2,6-bis(ethenyl)quinolin-8-yl]-3H-1,3,4-oxadiazol-2-ylidene]hydrazine [4-(3,5-difluoropyridin-2-yl)piperazin-1-yl]-phenylmethanone 4-chloro-N-[1-(5,6-dimethylpyridine-3-carbonyl)piperidin-3-yl]benzamide N-[1,4-dihydroxy-5-(3-phenylphenyl)hexyl]acetamide 6-hydroxy-5-[(3R)-2-oxa-9,11,15,18-tetrazatetracyclo[8.8.0.03,7.012,17]octadeca-1(10),12(17),13,16-tetraen-14-yl]hexanoic acid [4-chloro-5,7-dihydroxy-6-(4-methylphenyl)naphthalen-1-yl]urea [(Z)-(4-hydroxy-3,5-dimethoxyphenyl)methylideneamino]urea 3-[3-fluoro-2-(trifluoromethyl)phenyl]sulfanyl-1,4-dihydro-1,2,4-triazol-5-one 3-[[2-bromo-5-(trifluoromethoxy)phenyl]methyl]-1,4-dihydropyrazol-5-one 1-[(2,4-dimethylphenyl)methylamino]-3-heptan-3-ylthiourea 2-[(6-cyclopropyl-4-oxopyran-3-carbonyl)amino]acetic acid 2-[2,5-dichloro-N-(3-methylbut-2-enyl)anilino]ethanol (E)-1-[4-(difluoromethoxy)phenyl]-2-[5-ethenyl-1-(1-propan-2-ylpiperidin-4-yl)pyrazol-4-yl]but-2-en-1-one 1-azidooxy-2,3,4,5,6-pentafluoronaphthalene 3-(2,5-diphenylpyrazol-3-yl)-N-[(Z)-1H-indol-2-ylmethylideneamino]propanamide 3,5-dichloro-N-[1-(2,3-dihydroindol-1-yl)ethenoxymethyl]-4-methylaniline 6-[(2,3,4-triethoxyphenyl)methyl]-1H-benzimidazole N-[1-(4-fluorophenyl)ethyl]-3,7-dimethoxyquinolin-8-amine 2-[6-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]benzoic acid 5-(4-azidocyclohexyl)pyridine-2,3-diamine 2-[4-(3,5-dimethylphenyl)piperazin-1-yl]-N-[(6-fluoropyridin-3-yl)methyl]-N-methanimidoylpyrimidine-4-carboximidamide 1-[(2R)-butan-2-yl]-4-methoxy-2-propan-2-yl-6-(trifluoromethyl)benzimidazole 1-[(2S,4R)-4-hydroxy-6-iodo-2-methyl-3,4-dihydro-2H-quinolin-1-yl]ethanone N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-2-[1-(2-oxoethylamino)cyclopentyl]oxysulfonyl-2-[(E)-prop-1-enyl]acetamide N-[4,5-dihydroxy-1-(oxan-2-yl)pyrrolidin-3-yl]benzamide N-(3,5-difluorophenyl)-1-[4-(2-methylpropoxymethyl)triazol-1-yl]propan-2-amine 2-(methylamino)acetaldehyde;3,6,7,8-tetrahydro-2H-furo[4,5-e]indole-1,9-dione N-(2,3-dimethylphenyl)-1-(2-hydroxyethyl)-4-pyrazol-1-ylpiperidine-4-carboxamide N-[3-(3-fluorophenyl)propyl]-2-[5-[4-[4-(methoxymethylamino)piperidine-1-carbonyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl]-2-oxoacetamide 1,2-dimethoxy-N-[(Z)-1H-indol-3-ylmethylideneamino]benzimidazole-5-carboxamide 2-[(4-methoxyphenyl)iminomethyl]quinoline-8,9-diol (5Z)-5-[(2,4-dichlorophenyl)methylidene]-1-(4-ethoxyphenyl)-2-sulfanyl-6H-pyrazolo[4,3-d]pyrimidin-7-one 4-chloro-7-methyl-N,1-dioxoindole-2-carboxamide 2,6-bis(3-phenylpropyl)phenol 1-(cyclopropanecarbonyl)-7-[[3,5-difluoro-2-(4-fluorophenyl)pyridin-4-yl]methoxy]-2H-pyrido[3,2-e][1,2,4]triazine-8-carboxylic acid 6-(1,3-benzodioxol-5-yl)-2-butyl-N-[4-chloro-2-methoxy-5-(3-methyltetrazol-3-ium-1-yl)phenyl]pyrimidine-4-carboxamide 4-[(Z)-1,2-diphenylethenyl]cyclohepta-2,4,6-triene-1,4-diamine (2R)-4-[5-chloro-1-(2-methylpropanoyloxymethyl)indole-2-carbonyl]-2-methylpiperazine-1-carboxylic acid 5-(3,4-dimethoxyphenyl)-2-ethyl-7,8-dihydro-1,6-naphthyridine N-(5,7-dimethoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-4-[(4-methoxyphenyl)methoxy]benzamide;hydrochloride 4-amino-N'-(cyclohexylmethyl)-5,6-dihydrofuro[2,3-d]pyrimidine-7-carboximidamide N-[2-(4-fluorophenyl)ethyl]-3-[(1Z,7Z)-3-methylidenecyclonona-1,5,7,9-tetraen-1-yl]aniline 2-hydroxy-N,3,4-trimethyl-6-[[(E)-(1,3-thiazol-4-ylhydrazinylidene)methyl]amino]benzamide 1-(2,6-dichlorophenyl)-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine 4-azido-2,3-bis(3,5-difluorophenyl)furan 2-[1-(4-methylphenyl)piperidin-3-ylidene]propanedioic acid 3-(7-oxobenzo[d][2,1]benzoxaphosphepin-6-yl)-3H-isoquinoline (Z)-1-chlorobut-2-ene;ethane;N-methylpropan-1-amine;6-[4-[(2E,4Z)-2-(3-methylphenyl)hexa-2,4-dienoxy]piperidin-1-yl]-5-nitropyridine-3-carbonitrile 2-[4-(1,3-benzothiazol-2-yl)cyclohexa-2,4-dien-1-ylidene]propanedinitrile 1-methyl-5-[(3R)-piperidin-3-yl]oxybenzimidazole 2-[4-(3,5-difluorophenyl)piperidin-1-yl]-N,N-dimethylacetamide [6-(4,5-dihydroimidazol-1-ylmethyl)pyridin-3-yl]-(2-pyridin-3-ylazepan-1-yl)methanone 1-ethenyl-3,7-dimethyl-5-phenyldiazenyl-6H-pyrazolo[4,3-d]pyrimidin-7-one 2-azido-1-cyclopentylethenoxybenzene 2-[4-bromo-N-(cyanomethyl)anilino]benzenesulfonic acid 2-methylsulfanyl-3-(5,6,7,8-tetrahydroquinazolin-4-yloxy)phenol 3-[2,5-dimethyl-4-(oxiran-2-ylmethoxy)phenyl]propanoic acid N-[4-(7-cyanoquinoxalin-5-yl)oxycyclohexyl]cyclopropanecarboxamide 2-[4-(difluoromethoxy)phenyl]-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine 4-[2-fluoro-5-(trifluoromethyl)phenyl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 2-ethylsulfanyl-4,6-dimethoxypyridine 7-chloro-8-hydroxy-2-thiophen-3-yl-1,4-dihydro-[1,4]oxazino[5,6-c]quinoline 1-methyl-4-phenylquinolin-2-one 1-(4-azidobutyl)-2,3-dimethoxybenzene N-[(3S,7R,8aS)-3-propan-2-yl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-5-cyclobutyl-1,2-oxazole-3-carboxamide 4-azidooxy-2,6-bis(2-ethoxy-2-oxoethyl)benzoic acid N-[(2S,3R)-1-amino-4-methylpentan-2-yl]-5-[[2-fluoro-4-(trifluoromethoxy)phenyl]methoxy]pyridine-3-carboxamide 3-[(E)-2-iodoethenyl]furan 3-cyclopropyl-N-[1-(2,4-dimethoxyphenyl)ethyl]aniline 2-(5-carbamimidoylindol-1-yl)propanoic acid 4-(5-oxopyrrolidine-2-carbonyl)benzoic acid (2R)-1-[(3,4-dimethoxyphenyl)sulfonylamino]-N-[3-(4-methylpiperazin-1-yl)propyl]pyrrolidine-2-carboxamide;2,2,2-trifluoroacetic acid 2-[4-fluoro-3-(trifluoromethyl)phenyl]-N,1-dimethylimidazole-4-carboxamide (2R)-2-(3,6-dichlorocarbazol-9-yl)-N-[4-(N'-hydroxycarbamimidoyl)phenyl]propanamide (1S,3R)-N,3-dimethyl-2,3-bis(phenylmethoxy)cyclopentan-1-amine N-butyl-N-(2,4-dichloropyrimidin-5-yl)-2H-tetrazol-5-amine 5-chloro-4,6-dimethylthieno[2,3-d]pyrimidine;2-hydroxyacetaldehyde 4-[3-(1H-imidazol-5-yl)propyl]-2,3-dimethoxyphenol [(2S)-1-methylsulfanyloxy-3-(4-nitrophenyl)propan-2-yl]azanium 5-[3-[4-(5-ethylthiophene-2-carbonyl)piperazin-1-yl]propoxy]-6-phenylmethoxyhexanoic acid 5-[3-(2,6-dichlorophenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-N,N-dimethyl-2-oxopentanamide 7-[6-(2,6-difluorophenoxy)-4-[3-(dimethylamino)propoxy]pyridine-3-carbonyl]-N-hydroxy-2,5,6,8-tetrahydro-1H-isoquinoline-3-carboxamide;ethane (2S)-4,5,6,7,8-pentadeuterio-1-[2-fluoro-3-[[5-methyl-2-(propan-2-ylamino)pyrimidin-4-yl]amino]phenyl]-2H-isoquinolin-3-one 4-[6-(dibutylamino)hexyl]-7-(1H-indol-5-yloxymethyl)pyrrolo[2,3-d]pyrimidine-2-carboxamide N-(5-ethyl-2-methoxyphenyl)-1-[4-[(4-hydroxypiperidin-1-yl)methyl]phenyl]triazole-4-carboxamide 2-(5,7-dihydropyrrolo[3,4-b]pyridin-6-yl)-2-oxoacetamide 5-[[4-fluoro-3-methyl-2-(methylamino)butanoyl]amino]-2,4,6-triiodobenzene-1,3-dicarboxylic acid 3-(1H-indol-6-yl)pyrazin-2-amine N-[(3R,4S)-4-methylpiperidin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine;hydrochloride 3-chloro-N-(1,4-dimethylpyrrolidin-3-yl)-5-(trifluoromethyl)pyridine-2-carboxamide 2,4-dinitro-1-(6-nitronaphthalen-2-yl)sulfanylcyclohexa-2,5-dien-1-ol (2-chloro-4,6-dimethylphenyl)-[1'-[(3R)-piperidine-3-carbonyl]spiro[piperidine-4,3'-pyrrolo[2,3-c]pyridine]-2'-yl]methanone 2-azido-6,7-dimethoxynaphthalene 3-(furan-2-yl)-1,4-dioxobenzo[f]chromene-7-carbonitrile 2-[(4,5-dimethylpyrazol-1-yl)methyl]-N-[5-(2H-tetrazol-5-yl)oxolan-3-yl]benzamide 1-[2-chloro-4-(3-cyclohexyl-1,2,4-oxadiazol-5-yl)phenyl]-N-methylethenamine [[3-fluoro-4-(triazol-2-yl)phenyl]methyl-sulfanylamino]sulfanium N-[(1S)-2-(4-methoxyphenyl)-1-[6-oxo-3-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]pyridazin-1-yl]ethyl]-6-methylpyridine-3-carboxamide N-[3-(2,4-dioxocyclopentyl)-1H-indol-5-yl]-4-piperazin-1-ylbenzamide 1-(2-methylpropyl)-3-[2-(3-nitrophenyl)ethylamino]thiourea 2-N,6-N,6-trimethylpyrazolo[1,5-a]pyridine-2,7-diamine 3-(1,5-dimethylpyrazole-4-carbonyl)-2-methylsulfonyl-8-oxa-2-azaspiro[4.5]decane;formic acid 2-(3,4-dichlorophenyl)-N'-[2-hydroxy-3-[(3-methylphenyl)sulfonylamino]propyl]butanediamide (5R)-N-(4-methylphenyl)-2-[(3S,6R)-3,7,11-trihydroxyundecanoyl]-8-oxa-2-azaspiro[4.5]decane-4-carboxamide 1-[(2-ethyl-1,3-thiazol-4-yl)methyl]indole-3-carboxamide [2-(dihydroxymethyl)-6-methoxyphenyl]-(4-methoxy-1H-indol-3-yl)methanone 6-amino-7-[(1-phenylcyclobutyl)methylamino]heptanoic acid N-[(E)-2,5-dimethyl-6-oxohept-3-en-4-yl]benzamide 6-methyl-5,7-dihydrothieno[3,2-f][1]benzothiole N-[4-(1,1-dioxo-1,4-thiazinan-4-yl)phenyl]cyclopropanesulfonamide 2-[(5-chloro-3,4-dimethylpyridin-2-yl)methoxy]pyridine;ethane 1-[4,5-dimethyl-3-(1H-pyrazol-4-yl)thiophen-2-yl]ethanethiol 2-[4-(3,5-dimethylpyridin-1-ium-2-yl)phenyl]ethanamine;bromide 5-benzylsulfanyl-4-chloro-1H-triazolo[4,5-d]pyrimidine (Z)-N,2-dimethyl-3-[(6E)-6-[(4E)-8-oxo-4-[phenyl(pyrrolidin-1-yl)methylidene]cycloocta-4,7-dien-1-ylidene]heptoxy]but-2-enamide 4-[(3R)-3-aminopyrrolidine-1-carbonyl]-6-methyl-2,3-dihydro-1H-pyrrolizin-7-one 1-[4-(2,5-difluorophenoxy)cyclohexyl]propan-1-amine N-azido-2-propan-2-yloxybenzamide 5-bromo-4-tert-butyl-2-[2-(3-methoxyphenyl)ethyl]-1H-pyrimidin-6-one N-[4-(cyclohexa-1,3-dien-5-yn-1-ylamino)phenyl]naphthalene-2-carboxamide (5R)-2,5-dimethyl-6-[(1R,3S)-3-[methyl-[4-[(E)-2-(7-methyl-1H-indazol-5-yl)ethenyl]pyrimidin-2-yl]amino]cyclopentyl]hexanoic acid 3-(furan-2-yl)-1,7-dihydropyrazolo[4,3-d]pyrimidine N'-(2,3-dimethylphenyl)-4-[3-(8-ethoxy-7-fluoroimidazo[1,5-a]pyridin-3-yl)-4,4,4-trifluorobutanoyl]piperazine-1-carboximidamide 5-(methyliminomethyl)-6-(1H-pyrazol-4-yl)pyridine-2,3-diamine (E)-1,3-diamino-N'-[4-fluoro-2-[1-(methylsulfonylmethyl)cyclopropyl]phenyl]but-2-enediamide 4-[2-(6,7-dimethoxyquinazolin-4-yl)ethynyl]benzonitrile;4-(2H-tetrazol-5-ylmethylidene)piperidine 2-[(6S)-6-[[(2R)-2,3-dihydroxypropyl]amino]-7-[(4-fluorophenyl)methyl]-5-methyl-8-[(4-methylsulfanylpiperazin-1-yl)methyl]-6H-naphthalen-2-yl]acetaldehyde 5-[(3S,4R)-1-acetyl-4-methoxypyrrolidin-3-yl]-2-[3-chloro-2-fluoro-6-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-one 2-[(5Z)-3,4-dihydroxy-6,7-dimethoxy-1-methylocta-5,7-dien-4-yl]-3-prop-2-ynylbenzoic acid 5-chloro-3-[3-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]propoxy]pyridine-2-carbonitrile N-[(E)-2-aminoethenyl]-1-(3,4-dimethoxyphenyl)-6-[4-(trifluoromethyl)phenyl]benzo[h]phthalazine-7-carboxamide 1-(4-hydroxyphenyl)-2-[[2-(6-methylheptoxyamino)pyridine-3-carbonyl]amino]-7,8-dihydro-5H-pyrrolo[3,4-f]benzimidazole-6-carboxamide N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)phenyl]-3,4-dihydroxybenzamide;hydrochloride 4-[(2S)-1-[6-(5,7-dihydropyrrolo[3,4-b]pyridin-6-ylmethyl)pyrazine-2-carbonyl]piperidin-2-yl]-2-methoxybenzonitrile 3-(4-bromophenyl)-2,6-dichloropyridine 7-methyl-5,6-dipropoxy-2-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine 6-fluoro-N-methylsulfonyl-1,2,3,4-tetrahydronaphthalene-1-carboxamide 3-azidooxy-5,6-dimethylthieno[2,3-b]pyridine 2-cyclopropyl-4-[(2S)-2-methyl-1,3-dihydroinden-2-yl]-5H-indeno[2,1-b]pyridine 1-(4-chlorophenyl)sulfonyl-5-[2-methyl-3-(oxan-4-ylmethoxy)quinoxalin-6-yl]pyrazole-4-carbonitrile (1S)-5,7-difluoro-2-methylsulfonyl-3,4-dihydro-1H-isoquinoline N-[4,6-diamino-1-(5-cyanopyridin-2-yl)hexylidene]hydroxylamine 1-methyl-2-[3,4,5-tris(trifluoromethyl)phenyl]piperazine 5-(2-methyl-1,3-thiazol-4-yl)-2-propan-2-ylphenol 3-[2-(3,4-dichlorophenyl)ethylamino]-5-methyl-6H-[1,2]oxazolo[4,5-d]pyrimidin-7-one 2-[N-(benzenesulfonyl)-4-fluoroanilino]-5-chlorobenzoic acid N-(4-anilinophenyl)-N-hexadecanoylbenzamide 2-azido-N,5-dibenzylaniline 2-(4-benzylpiperazin-1-yl)-N-[(2S,3S)-2-(4-chlorophenyl)-6-methoxy-3-methyl-5-oxo-2,3-dihydro-1H-imidazo[1,2-a]pyridin-8-yl]acetamide 6,7-bis(9H-fluoren-1-yl)-N-propan-2-ylnaphthalen-2-amine 6-[3-(dimethylamino)propyl]-4,5,7-trideuterionaphthalene-1,2-dione N-[1-[5-bromo-2-(5,6-dimethylpyridine-3-carbonyl)phenyl]ethylideneamino]acetamide 1-N',5'-N'-ditert-butylspiro[cyclohexane-1,3'-indole]-2',5'-diamine (2S)-2,6-diamino-3-methyl-N-[3-(3-phenylpyrrolidine-1-carbonyl)phenyl]hexanamide 7-azido-4,8-dimethylchromen-2-one 4-[8-(2-oxo-1H-pyrrol-3-ylidene)quinoline-5,7-diium-3-carbonyl]piperazine-1-carboxylic acid 4-fluoro-1,3-dihydroxyindene-2-carboxylic acid (4R,5S)-N-[3-(1H-benzimidazol-2-yl)cyclobutylidene]-7,7-difluoro-10-methyl-17-oxa-12-azatetracyclo[8.6.0.02,9.011,15]hexadeca-1(16),2(9),10,14-tetraene-4-carboxamide 3,8-dimethyloctane;ethane;4-(5-formamidopentanoylamino)pyridine-2-carboxylic acid 1-(1-ethylpiperidin-4-yl)-6,7-dihydro-5H-pyrazolo[3,4-c]pyridin-4-one N-[4-(5,6-dimethylpyrimidin-2-yl)oxyphenyl]acetamide 2-[N-(cyanomethyl)anilino]benzenesulfonic acid N-ethyl-3-methyl-2-[(Z)-1-[3-(trifluoromethyl)phenyl]but-1-enyl]aniline 1-[4-(7,8-dihydrothieno[2,3-f]quinolin-9-yl)piperazin-1-ium-1-ylidene]ethanol;methane 4-methyl-2-(7-oxospiro[1,3-dihydroisoquinoline-4,1'-cyclobutane]-2-carbonyl)pyridine-3-carbonitrile N-methyl-4-[1-[2-[3-methyl-5-(trifluoromethyl)pyrazole-1-carbonyl]piperidine-1-carbonyl]cyclohexanecarboximidoyl]benzamide 1-(7-cyclopentyloxynaphthalen-2-yl)sulfonyl-N,N-dimethylpiperidine-4-carboxamide 2-[1-[2-amino-3-(3,4-dichlorophenyl)propanoyl]-4-cyanoazepan-4-yl]acetamide 3-[4-(5-aminopyridin-2-yl)pyridazin-1-ium-1-yl]propanoic acid 4-ethyl-2-[[5-methoxy-4-[3-(trifluoromethoxy)phenyl]pyridine-2-carbonyl]amino]benzoic acid 5-[2-fluoro-4-(7H-purin-6-yl)phenyl]-1,3-oxazole 3,5-bis[(Z)-prop-1-enyl]benzoic acid 1-[(2R)-2-methylpyrrolidin-1-yl]-5-phenyl-3H-2,1-benzoxaborole 3-(5-phenylpentanoyl)chromen-2-one [(3aR,6aS)-1-(4-fluorophenyl)sulfonyl-2,3,3a,5,6,6a-hexahydropyrrolo[3,2-b]pyrrol-4-yl]-(3-methoxyphenyl)methanone N-[1-(2,4-difluorophenyl)cyclopropyl]-2-oxopiperidine-3-carboxamide [(1S)-2,3-dihydro-1H-indene-1-carbonyl]-oxoazanium;3-ethoxypropane 4-amino-2-(3,5-dimethoxyphenyl)-N-[(2R)-2-hydroxy-4-(2-oxoimidazolidin-1-yl)butyl]pyrimidine-5-carboxamide [4-(azetidine-1-carbonyl)phenyl]urea 5-azido-2-chloro-4-(6-methoxypyridin-3-yl)pyrimidine 4-(3-ethoxyphenyl)-1,2,3,6-tetrahydropyrimidine 2-[[5,7-dichloro-1-(4-methoxybutyl)indazol-3-yl]methylidene]cyclohexane-1,3-dione 4-[1,3-dimethyl-5-(piperidine-1-carbonyl)pyrazol-4-yl]-2H-phthalazin-1-one 4-[3-(difluoromethyl)-4-methoxyphenyl]-6,7-dihydro-2H-furo[2,3-d]pyridazine N-[1-(2,6-dimethylphenyl)pyrrolidin-3-yl]-N-(oxetan-3-yloxy)formamide 5-[3,4-bis(phenylmethoxy)phenyl]-1,2-oxazol-3-one 5-[3-(2,4-dihydroxyphenyl)propanoyl]benzene-1,3-dicarboxylic acid 3-(4-bromobutoxy)-1H-indole 4-[(E)-2-(4-hydroxyphenyl)ethenyl]sulfanylbenzoic acid 1-azido-3-ethylsulfonylbenzene 1-(4,5-dichloro-2-methoxybenzoyl)-N-[2-oxo-6-(trifluoromethyl)-3H-imidazo[1,2-a]pyridin-7-yl]pyrrolidine-2-carboxamide (4-azidopiperazin-1-yl)-[3,5-bis(trifluoromethoxy)phenyl]methanone (NE)-N-[1-amino-2-(methyliminomethyl)butylidene]-4-[(3-chlorophenyl)methoxy]piperidine-1-carboxamide;methanimine 2-(1H-benzimidazol-2-yl)-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-4-chloro-5,6-diethynoxyquinazoline-7-carboxamide 5-(4,5-diphenyl-1H-imidazol-2-yl)pentan-1-amine (5S)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide 2-[1,3-dioxo-4-(prop-2-enoylamino)isoindol-2-yl]-N,5-dimethoxypentanamide 2-[4-[6-(butanoylamino)-1H-benzimidazol-2-yl]phenyl]sulfanyl-2-methylpropanoic acid 6-[1-(3,4-dimethoxyphenyl)ethyl]-N-[2-[methyl-[2-(5-oxohexan-2-yl)prop-2-enoylamino]phosphoryl]ethyl]pyridine-3-carboxamide 2-[4-(5-aminopyrazin-2-yl)-3-fluorophenyl]-1,2-dipyridin-2-ylethanone (2Z,5R)-5-[(4-fluorophenyl)methyl]-2-[(Z)-(3-hydroxyphenyl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one 5-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(3-methylbut-2-enyl)amino]-3H-1,3,4-thiadiazole-2-thione 1-[2-[6-(trifluoromethoxy)pyridin-3-yl]pyrrolidin-1-yl]propan-1-one 1-(cyclopropylamino)-3-[[(2S,4R)-4-fluoro-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]methyl]urea 3-[2,4-dichloro-5-(phenylmethoxycarbonylamino)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile (Z)-2,3,4-triphenyl-1H-[1]benzoxepino[5,4-c]pyrazole 2-[2,4-dichloro-6-[(E)-1-pyridin-3-ylethenyliminomethyl]phenyl]sulfanyl-N-methylethanamine 3-[(4aR,9aS)-7-bromo-1-(4-methoxybutyl)-2-methylidene-5-propan-2-yl-3,4,4a,9a-tetrahydropyrido[4,3-b]indol-6-yl]-1H-pyridin-2-one [(2R,3S)-3-amino-4,4,4-trifluoro-1-hydroxybutan-2-yl]oxybenzene 1-cyclopenta-2,4-dien-1-yl-3H-indol-2-one N-azido-2-[3-(1,5-dihydropyrazol-2-yl)phenyl]ethanamine [(4R,5S)-2-benzoyl-3-phenyl-1,3-thiazolidin-4-yl]-(1,6-dihydropyrrolo[3,4-c]pyrazol-5-ylmethylideneamino)methanone 4-[[2-[(2,6-dioxopiperidin-3-yl)methyl]phenoxy]carbonylamino]butanoic acid 3-azido-1,2-dimethylindole N-[[4-(5,6-dimethyl-2H-pyridin-1-id-3-yl)phenyl]methoxy]cyclobutanamine N-(2,6-diethylphenyl)-5-[[4-fluoro-3-(trifluoromethyl)phenyl]sulfonylamino]-1H-indole-2-carboxamide 2-[3-(N-[[2,4-bis(trifluoromethyl)phenyl]methylideneamino]anilino)propoxy]phenol 2-N-(5-aminopyridin-3-yl)-5-chloro-4-N-[4-[5-(ethoxymethyl)furan-2-yl]cyclohexyl]pyrimidine-2,4-diamine 3-amino-4-cyano-5-[3,4-difluoro-2-(trifluoromethoxy)phenyl]-1H-pyrrole-2-carboxamide 5-chloro-4-[6-[(3R,4S)-3-ethyl-4-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-benzimidazol-2-yl]-N-(1,3-thiazol-2-yl)thiophen-2-amine 5-[(Z)-[7-cyclopropylimino-5-[4-hydroxy-2,6-dioxo-1-(pyridin-3-ylmethyl)pyrimidin-5-ylidene]pyrazolo[1,5-a]pyrimidin-3-ylidene]methyl]-1,3-diethylbenzimidazol-2-one ethane;(Z)-2-methylidene-3-[6-methyl-5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl]iminobut-1-en-1-amine 2-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-[(Z)-(4-hydroxy-3-iodo-5-nitrophenyl)methylideneamino]acetamide N-[2-(7,8-dihydronaphthalen-1-yl)ethyl]propanamide 2-[3,5-dichloro-4-(4-hydroxyphenyl)phenyl]-4,6-dioxo-1,3-diazinane-5-carbonitrile (3Z)-4-methylidene-N-[1-[6-oxo-5-(trifluoromethyl)-1H-pyridazin-4-yl]pyrrolidin-3-yl]hepta-1,3-diene-2-sulfonamide 2-[7,9-diethoxy-10-(1H-inden-5-yl)phenanthren-3-yl]acetaldehyde 2-amino-4-(8H-[1,3]dioxolo[4,5-g]chromen-6-yl)-4H-pyran-3,5-dicarbonitrile 2-[2,5-dimethyl-6-(4-methylsulfanylphenyl)-3-propoxyphenoxy]butanedioic acid (5Z)-3-methyl-2-phenylimino-5-[[4-[3-(trifluoromethoxy)phenyl]furan-2-yl]methylidene]-1,3-thiazolidin-4-one (E)-4,8-difluoro-3-methyl-1-phenyloct-5-en-3-ol 5-ethenyl-4-(1-methoxycyclobutanecarbonyl)thiophene-3-carbonitrile 2-[4-hydroxy-5,8-dioxo-6-(2-phenylsulfanylethoxy)-6H-naphtho[1,2-b]chromene-10-carbonyl]benzoic acid 2-azido-3,4-dimethylisoquinolin-1-one [4-[bis(prop-2-enyl)amino]piperidin-1-yl]-(3-chloro-2,5-dihydropyrrol-1-yl)methanone 1-[5-ethenyl-4-(oxan-4-ylamino)pyridin-2-yl]-3,6-dihydro-2H-pyridine-4-carboxylic acid 2-[1-(methoxymethyl)cyclopentyl]pyridine 2-[4-(difluoromethyl)pyrimidin-5-yl]oxy-N-(1,3-thiazol-2-yl)-7-azaspiro[3.5]nonane-7-carboxamide (7R)-2-(4-fluorophenyl)-N,7-bis[4-(trifluoromethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)-6,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide 2-[[(1R)-1-azidooxy-2,3-dihydro-1H-inden-5-yl]oxymethyl]-5-chloropyridine N-(1-benzofuran-2-ylmethyl)-N',3-dimethylcyclohepta-1,4,6-triene-1-carboximidamide [4-(3,3-dichloroprop-2-enoxy)phenyl]-methylidene-(pyridine-4-carbonylamino)azanium 4-[2-(3,5-dimethylpyrazol-1-yl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-[4-(2,5-dioxopyrrolidin-1-yl)phenoxy]-N,N-dimethylbenzamide 4-methyl-N-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)phenyl]benzamide 4-(2,3-difluorophenyl)imino-1-ethyl-5-methylimidazolidine-2-thione N-[5-[3-(4-thiophen-2-yl-1H-pyrrolo[3,2-c]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]cyclopropanecarboxamide 2-azido-N,N-diethylbenzamide N-[4,5-bis(ethenyl)-2-methylidenepyridin-1-yl]-7-oxodecanamide 5-bromo-4-cyclopropyl-2-(1,3-oxazol-2-yl)-1H-pyrimidin-6-one (2Z,4E)-1-[4-[5-fluoro-6-(methylamino)pyrimidin-4-yl]piperazin-1-yl]-3-methylidene-N-propylhexa-2,4-dien-1-imine 1-[[(2S,4R)-3-fluoro-4-hydroxypyrrolidine-2-carbonyl]amino]-N-methylpyrrole-3-carboxamide (6-bromo-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)-(6-fluoro-1H-indol-2-yl)methanone 3-[(6Z)-6-(1H-indol-2-ylmethylidene)cyclohexa-2,4-dien-1-ylidene]oxypropanoic acid N-[4-(2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-5-carbonyl)phenyl]acetamide N-[4-(dimethylsulfamoyl)phenyl]-2-fluoropyridine-3-carboxamide N-[3-(difluoromethyl)-5-methyl-1H-pyrazol-4-yl]-4-[5-[2-[(dimethylamino)methyl]morpholin-4-yl]pentanoyl]piperazine-1-carboxamide 6-[3-(2,6-dimethylpyridine-4-carbonyl)phenyl]cyclohexa-1,5-diene-1-carbonitrile 3-bromo-2-(4,5-dihydrobenzo[e][1]benzazepine-6-carbonyl)-7-ethylcyclohepta-2,4,6-trien-1-one 5-ethenyl-6,7,8-trifluoro-1H-benzo[g]isochromene 4-chloro-2,7-di(propan-2-yl)pyrido[2,3-d]pyrimidine N'-[[4-(2,2-difluorocyclohexyl)phenyl]methoxy]-3-ethanimidoyl-N-ethenyl-N'-methyl-1H-pyrrole-2-carboximidamide 2,4-dichloro-5-iodopyrimidine 2-[[[3-methyl-5-(trifluoromethyl)benzoyl]amino]methyl]pyridine-3-carboxylic acid 1-(4-azidooxyphenyl)-5-methylsulfonyltetrazole 1-[2,6-dichloro-N-(4-propylphenyl)-1H-pyridazin-5-yl]azetidine-3-carbonitrile N-(3-azidopropyl)-4-chlorobenzenesulfonamide 5-(2,2-dimethylpropylamino)-N'-hydroxypyridine-4-carboximidamide 2-[3-(difluoromethoxy)pyridin-4-yl]cyclobutan-1-ol 4-[3,5-bis(trifluoromethyl)anilino]-N-[2-oxo-2-[[4-[3-(trifluoromethoxy)phenyl]pyrimidin-2-yl]amino]ethyl]benzamide 1-azidosulfanyl-3-butan-2-yl-5,6-dimethoxy-2-methylnaphthalene 2-[[1-[(4,5-dimethylthiophene-3-carbonyl)amino]cyclopentanecarbonyl]amino]acetic acid 3-[2,4-bis(2-phenylethenyl)phenyl]-5-fluoropyridine 1-methoxy-2,3-dimethyl-4-(4,4,5,5,6,6,7,7,8,8,9,9,10,10,11,12,12,12-heptadecafluorononoxy)benzene N-(1,2-dihydropyridazin-3-yl)-4-[[6-fluoro-1-methylidene-7-(3-morpholin-4-ylpropoxy)quinazolin-4-ylidene]amino]benzamide 6-chloro-2,4-dihydroxybenzenesulfonic acid 2-[7,8-difluoro-5-(4-methylpiperazine-1-carbonyl)-3,4-dihydro-1H-isoquinolin-2-yl]-4-(4-morpholin-4-ylcyclohexyl)oxybenzaldehyde (1R,2S)-2-amino-N-[8-fluoro-7-methyl-4-oxo-6-(3,3,3-trifluoropropoxy)quinazolin-3-yl]cyclopentane-1-carboxamide (3S,4R)-2-methyl-1-[(2S)-2-propanoyloxy-3-[(2-quinolin-7-ylacetyl)amino]propanoyl]piperidine-4-carboxylic acid (2-aminopyrimidin-5-yl)-[4-[2-(dimethylamino)ethoxy]phenyl]methanone;hydrochloride 2-(2,4-dichloro-3-nitrophenyl)acetaldehyde 3-(1-azidopiperidin-2-yl)oxy-6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazole 2-(4-methylcyclohexyl)oxyiminopropanal;N,5,6-triethylnaphthalen-1-amine 2-[[3-fluoro-4-(trifluoromethyl)phenyl]carbamoylamino]acetamide (4S,5R)-3-cyclopropyl-6,7-dimethoxy-1-azatricyclo[7.3.1.05,13]trideca-9(12),10-diene 2-azido-6-bromo-3,4-dihydro-1H-isoquinoline 4-amino-6-[[3,5-difluoro-2-(hydroxymethyl)phenyl]methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 1-(2,4-dibromophenyl)-2-methylpentane-3-sulfonic acid 2-[4,5-dimethyl-1-(4-phenylsulfanylphenyl)pyrazol-3-yl]propanoic acid N-[5-(2-fluorophenyl)sulfanyl-4,6-dioxo-3-propanoylthieno[2,3-d]pyrimidin-7-yl]acetamide N-(1,3-benzodioxol-5-ylmethyl)-6-oxo-4H-furo[2,3-c]pyrrole-5-carboxamide N-[1-(2-fluorophenyl)ethenyl]-6-methoxypyrazine-2-carboxamide 3-[(2S)-2-amino-4-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butanoyl]piperazine-1-carbonyl]benzonitrile 6-[4-(2-ethylbutyl)phenyl]hexan-3-ol (2S)-4-[3-methylsulfonyl-4-[(3R,5S)-3,4,5-trihydroxypyrrolidin-1-yl]phenyl]butanoic acid 5-chloro-2-[(1,3-dimethylpyrazol-4-yl)sulfonylamino]benzoic acid (4-benzylpiperazin-1-yl)-[6-(2,4-dichlorophenyl)-5H-pyrazolo[3,4-d]pyrimidin-4-ylidene]methanolate 5-tert-butyl-N-[2-(methylamino)ethyl]thiophene-3-carboxamide 3-(2-cyclohexylethoxy)-5-(1-methoxybutan-2-yloxy)benzonitrile 4-[2-methyl-6-(4,5,6,7-tetrahydro-3H-benzimidazol-5-yl)pyridin-4-yl]oxyaniline 6-hydroxy-5-[[2-(4-methylphenyl)sulfonylphenyl]iminomethyl]-1,3-dipropylpyrimidine-2,4-dione 6-[4,5-bis(ethenyl)pyridin-2-yl]-10-propan-2-yl-1,3,8,11-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene (2S)-4,5-dimethyl-6-oxo-1H-1,5-benzodiazepine-2-carboxylic acid;ethane 5-(3,4-dimethoxyphenyl)-2-(furan-2-ylsulfonylamino)pentanoic acid 2,6-difluoro-N-(1H-pyrazol-5-yl)benzamide N-[(3S)-5-chloro-2,4-dimethylhexan-3-yl]-5-phenyl-1H-pyrazole-3-carboxamide 6-bromo-4-N,5-bis[(Z)-[4-(diethylaminomethoxy)phenyl]methylideneamino]pyrimidine-2,4-diamine 2-[3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethanesulfonamide (2S,3aS,7aR)-N-pyridin-2-yl-6-(thiophen-2-ylmethyl)-3,3a,4,5,7,7a-hexahydro-2H-furo[2,3-c]pyridine-2-carboxamide;2,2,2-trifluoroacetic acid 2-[3-(2,6-dimethoxyphenyl)propyl]propanedioic acid 3-(cyclopentylmethyl)-7-(3,5-dichlorophenyl)-2H-1,3-benzoxazin-4-one ethane;4-[6-ethoxy-5-(4-fluorophenyl)pyridin-2-yl]-1-methylpiperazine [1-[2-(4-chlorophenyl)-3-ethylsulfonylimidazo[1,2-a]pyridin-6-yl]piperidin-4-yl]-morpholin-4-ylmethanone 3-[4-(methylsulfamoyl)phenoxy]propanoic acid 4-[5-ethylsulfonyl-6-(3,4,5-trifluorophenyl)pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidine 5-azido-4,6-dibromopyrimidine (1S)-1-[4-chloro-5-[1-(difluoromethyl)pyrazol-3-yl]thiophen-2-yl]-2-(propanoylamino)ethanesulfonic acid 2-[[4-(2,3-dihydropyridin-6-yl)pyrimidin-5-yl]methylideneamino]benzonitrile 2-amino-N-[4-[5-(methylamino)pyridin-2-yl]phenyl]-4-propan-2-ylidenecyclohexane-1-carboxamide 2-(2,6-dimethylphenyl)-7-[1-[3-(pyridin-4-ylamino)propoxy]ethenyl]pyrido[1,2-a]pyrimidin-4-one 1-[4-(4,6-dimethyl-2-oxopyran-3-yl)phenyl]-5H-pyrazolo[4,3-c]pyridin-4-one 1-methyl-5-[2-(4-thiophen-3-ylcyclohexa-1,3-dien-1-yl)ethynyl]pyrrolo[2,3-b]pyridine 4-bromo-2,5-dimethyl-N-(3-morpholin-4-ylpropyl)-N-pyridin-3-ylaniline 1,7-difluoro-3-(2-methylbutan-2-yl)-5-pentan-2-ylbenzimidazol-2-one 3-[(4-azidophenyl)methyl]-5-fluoro-1H-benzimidazol-2-one 1-[(3aR,6R)-2-benzylsulfonyl-5-oxo-3,4,6a,7,8,9-hexahydro-1H-pyrrolo[3,4-h]isoquinolin-6-yl]-3-methylbutan-2-one 5-[3-(2-fluoroethylamino)butanoyl]-1-methylpyridin-2-one 3-[(5Z)-4,9-dimethylidene-7,8-bis(2-phenylethynyl)undeca-5,10-dienoxy]propanoic acid 1-(2-bromoethyl)pyrene N-(2,2-diethoxyethyl)-4-methoxy-6-methyl-N-phenylpyrimidin-5-amine 1-(4-chlorophenyl)-3-[3,5-difluoro-2-[2-methyl-6-oxo-4-(trifluoromethyl)pyrimidin-1-yl]phenyl]urea 3-amino-N'-(3,4-dichlorophenyl)pentanehydrazide 4-(1,3-benzodioxol-5-ylmethyl)-7-chloro-2H-isoquinolin-1-one 4-[2,3-difluoro-6-(propoxymethyl)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 2-[N-(4-nitrobenzoyl)-4-phenoxyanilino]propanoic acid 5-[1-(4-chlorophenyl)-2,4-difluoro-3-methylcyclobutyl]-1,3-benzothiazole;ethane ethane;2-[3-[5-(hydroxymethyl)furan-2-yl]propanoylamino]benzamide 2-(3,4-dichlorophenyl)-N-methyl-2-phenylpropanamide 1-bromo-4-fluoro-3,5-diiodo-2-methylsulfanylbenzene 4-[2-(difluoromethoxy)phenyl]-N,3-dimethylaniline;ethane 2-[3-[(6S)-1,6-dimethyl-6,7-dihydro-4H-pyrano[4,3-c]pyrazole-3-carbonyl]-5-fluoro-4-phenylmethoxyphenyl]acetamide (3E)-3-benzylidene-6-bromo-2,4a-dimethyl-1H-quinoxaline 4-[(3R)-2,6-dioxopiperidin-3-yl]oxybenzonitrile;hydrochloride 4-[2-hydroxyethyl(propyl)amino]-5-iodo-1H-pyrimidin-6-one 5-(5,7-dimethoxy-1H-indole-2-carbonyl)-N-[(2S)-1-fluoropropan-2-yl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 2-[[4-(6-cyano-3-methylindol-1-yl)phenyl]sulfonylamino]ethoxymethanesulfonate N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-methoxyethanimine 4-[1-(6-ethoxypyridine-3-carbonyl)azetidin-2-yl]oxypyridine-2-carboxamide 6-chloro-2-N,4-N-bis[(2E)-penta-2,4-dienyl]pyridine-2,3,4-triamine 4-[2,3-bis(ethenyl)phenyl]dibenzofuran 5-[2,6-bis(trifluoromethyl)phenyl]-1H-pyrazol-3-amine N-[3-(4,5-dihydro-1H-imidazol-2-yl)propyl]-6-methoxy-1,1a,2,7b-tetrahydrocyclopropa[c]quinolin-9-amine 4-chloro-6,9-diethylcarbazole-1-carboximidamide (Z)-N-[2-hydroxy-1-(3-methoxyphenyl)ethyl]pent-2-enamide 2-[3-(4-chlorophenyl)sulfanylimidazo[1,5-a]pyridin-1-yl]-N-[1-(4-methoxyphenyl)ethyl]acetamide 1-cyclopentyl-6,7-dimethoxyisoquinoline 4-[1-(1,2-benzoxazol-5-yl)-3-methyl-6-oxopyridazin-4-yl]-N-[2-(2-hydroxyethoxy)ethyl]piperazine-1-carboxamide;hydrochloride 1-(3-cyclopropylbut-3-enoxy)-4-(1-methylcyclohexa-2,4-dien-1-yl)benzene N-[1-(4,5-dimethyl-6-oxo-1H-pyrimidine-2-carbonyl)piperidin-3-yl]but-2-ynamide N-[(2S,4R)-1-[[(1R)-cyclohexa-2,4-dien-1-yl]methylamino]-3,3,3-trifluoro-2-hydroxy-4-phenylbutan-2-yl]-6-[3-[3-(cyclopropanecarbonylamino)phenyl]phenyl]imidazo[1,5-a]pyridine-8-carboxamide N-[1-[6-(difluoromethoxy)pyridin-3-yl]ethyl]-2,5-bis(3-fluorophenyl)triazole-4-carboxamide 1-(4-bromophenyl)sulfonyl-3-diazourea 6-methoxy-N-[(5Z)-2-oxo-4-sulfanylocta-5,7-dienyl]naphthalene-1-carboxamide 5-benzylsulfanylnaphthalene-2-sulfonamide 1-(2,4-dichlorophenyl)-N-[(E)-[3,5-dibromo-2-hydroxy-4-(trifluoromethoxy)phenyl]methylideneamino]-6-oxopiperidine-3-carboxamide 2-[(4-phenylcyclohexa-1,5-dien-3-yn-1-yl)amino]ethanol 1-[[2-methyl-4-(2,2,3,3-tetrafluoropropoxy)phenyl]methylideneamino]cyclopropane-1-carboxylic acid N-[5-[3-(2,2,6,6-tetramethylpiperidin-4-yl)triazolo[4,5-c]pyridazin-7-yl]-1H-pyrazol-3-yl]benzamide 3-[(2R)-2-amino-1,3-thiazol-4-yl]-N-[[5-[methyl(pyridin-3-ylsulfonyl)amino]-1H-indol-2-yl]methylidene]benzamide N-(6-bromo-1,3-benzothiazol-2-yl)-4-[[3-(dimethylamino)propanoylamino]methyl]benzamide 5-[4,8b-bis(methylimino)-3a,7a-dihydrocyclohepta[d]imidazol-2-yl]quinoline-2-carbonitrile 3-(benzenesulfonyl)-1H-quinolin-2-one 4-[2,6-dimethoxy-4-(trifluoromethyl)phenyl]-3-phenyl-4H-chromene (6-amino-1,3-benzothiazol-2-yl)-[3-(difluoromethoxy)phenyl]azanium;bromide N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethynyl]-2-oxochromene-3-carboxamide 1-(2-ethoxypyridin-3-yl)-N-[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]-6-iodobenzimidazole-5-carboxamide 3-chloro-6-[4,5,6-tris(fluoromethyl)pyridin-2-yl]oxypyridazine 3-methyl-6-[1-(2-propanoyloxyphenyl)sulfonylpyrrolidin-2-yl]pyridine-2-carboxylic acid 3-[(2-aminophenyl)carbamoyl]-1-(4-ethoxyphenyl)pyrrolidine-2-carboxylic acid [2-(4-fluorophenyl)quinolin-3-yl]methanamine (4R)-1-methyl-3,9-diphenyl-5,6,7,8-tetrahydropyrimido[4,5-b]quinoline-2,4-dione 4-[5-(2,3,5-trimethylcyclopenta-1,3-dien-1-yl)thiophen-2-yl]-N-(3,4,5-trifluorophenyl)pyrimidin-2-amine 4-[2,5-dimethyl-3-(trifluoromethyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile N-(2,3,4,5-tetrahydropyrido[2,3-e][1,4]diazepin-7-ylsulfonyl)-2H-chromene-4-carboxamide N-[(2S)-4-azidooxy-1-methoxybutan-2-yl]-1H-benzimidazole-4-carboxamide 2-(6-chlorohexyl)tricyclo[4.3.0.03,8]nona-1(6),7-dien-4-ol N-[3-[(2,6-dimethylphenoxy)methyl]piperidine-1-carbonyl]acetamide (1S,2R)-N-[(Z)-3-anilinoprop-2-enimidoyl]-2-phenylcyclopropane-1-carboxamide N-[3-(4-methyl-1,2,4-triazol-3-yl)phenyl]sulfonylprop-2-enamide N-(4-acetamidobutyl)-2,3,4,5,6-pentachlorobenzamide 7-(furan-3-yl)-N-[4-methoxy-3-(4-morpholin-4-ylpiperidin-1-yl)phenyl]pyrido[2,3-d]pyrimidin-4-amine (2Z)-4,8-difluoro-N'-[3-fluoro-5-methyl-1-(2H-thiopyran-6-yl)pyrazolo[3,4-b]pyridin-6-yl]-2-(3-hydroxypropylidene)-7H-chromene-3-carboximidamide (2S)-3,3-difluoro-2-methyl-1-[4-(trifluoromethoxy)phenyl]pyrrolidine (1S,5R)-N,N'-bis[(4-methoxyphenyl)methyl]-2-oxobicyclo[3.1.0]hexane-6-carboximidamide N-[2,4-difluoro-3-(2-methyl-5,8-dioxoquinazolin-6-yl)phenyl]cyclopropanesulfonamide N-[6-(3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-2-carbonyl)pyridin-2-yl]acetamide 4-[[(3S)-3-aminopyrrolidin-1-yl]methyl]-5,6,7,8-tetrahydrocinnoline-3-carboxamide 4-[2-(6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-1-yl)ethoxy]benzaldehyde 2-[1,4-bis(4-chlorophenyl)-5-cyanoimidazol-2-yl]sulfanylacetic acid 2-hydroxyimino-1-(4-methylphenyl)-2-[(E)-phenylcarbamothioylhydrazinylidene]ethanone N-(3,5-dichloropyridin-4-yl)-1-hydroxy-3H-2,1-benzoxaborol-6-amine 6-methyl-5-(3,4,5-trimethoxyphenyl)spiro[1H-2-benzofuran-3,4'-piperidine] (5R)-6,8-diazaspiro[4.5]decan-5-ol;N-ethyl-2-[4-[4-fluoro-3-(trifluoromethoxy)phenyl]-3-(trifluoromethyl)phenoxy]acetamide 2-(methylamino)-4,6-di(propan-2-yl)phenol 3-(2,4-dichlorophenyl)sulfanyl-2H-thieno[2,3-d]pyrimidine 5-chloro-N-(1,4-diazabicyclo[3.2.2]nonan-9-ylmethylidene)quinoline-8-carboxamide N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-pyrimidin-5-ylpyrrolidine-1-carboxamide 4-amino-1-(2,3-dihydro-1H-inden-5-yl)pyridin-1-ium-3-carboxylic acid N-benzyl-2,4-dichloro-N-(2-methylpropyl)pyrimidin-5-amine 3-methylsulfanyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carboxamide 5-amino-6-[(3S)-3-(hydroxymethyl)piperidine-1-carbonyl]naphthalene-2-sulfonic acid (2S,4R)-4-[2-(5-cyclohexyloxypyridin-3-yl)imidazol-1-yl]pyrrolidine-2-carboxylic acid;dihydrochloride 2-[4-amino-6-[(5-fluoropyridin-3-yl)methoxy]pyrimidin-5-yl]acetamide 1-[2,5-diethyl-4-(5-fluoropyridine-3-carbonyl)piperazin-1-yl]-2,2,2-trifluoro-N-hydroxyethanesulfonamide 5-(5-azidooxy-2-methylphenyl)-3-[1-(cyclopropylmethyl)pyrazol-4-yl]-1H-pyrrolo[2,3-b]pyridine 1-[[5-chloro-2-(trifluoromethyl)phenyl]methyl]indole (Z)-3-amino-2-(ethylaminomethyl)but-1-en-1-ol;4-[[[(E,4S)-8-[(4R,6S)-2,6-dimethylpiperidin-1-yl]-7,8-dihydro-6H-quinolin-5-ylidene]amino]oxy]aniline 6-[4-(4-methylphenyl)piperidin-1-yl]pyrimidine 5-cyclohexa-1,3-dien-1-yl-1-pyridin-2-yl-N-(4-sulfamoylphenyl)pyrazole-4-carboxamide N-[5-cyano-4-(3,3-difluoroazetidin-1-yl)pyridin-2-yl]-7-formamido-6-methoxy-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide 4-[4-(benzoylsulfamoyl)-N-cyclohexylanilino]butanoic acid N-(cyclopentylmethyl)-4,4-difluoro-1H-indazole-6-carboxamide 5-[2-(4-bromophenyl)-4-oxoimidazolidine-1-carbonyl]-N-methylpyridine-3-sulfonamide 2-N-methyl-1-N-[3-(trifluoromethoxy)phenyl]cyclopropane-1,2-dicarboxamide 2-[3,5-dichloro-4-(3-methylbutoxy)phenyl]acetohydrazide 3-[(2E,4Z)-5-bromohepta-2,4-dienyl]-2H-1,3-benzoxazole (5E)-5-[[3,5-diiodo-4-[(2R)-pentan-2-yl]oxyphenyl]methylidene]-2-(4-ethylphenyl)imino-1,3-thiazolidin-4-one N-[(3R)-4-[1,3-benzodioxol-5-ylsulfonyl-[(6-cyanopyridin-2-yl)methyl]amino]-3-hydroxybutyl]-7-methoxynaphthalene-1-carboxamide 1-ethyl-2,4-dimethylnaphthalene;5-ethyl-3-methylheptane;(3E)-penta-1,3-diene 5-[(2S)-4,8-dimethyldecan-6-yl]oxycarbonylnaphthalene-1-carboxylic acid (1-ethyl-4,5-dihydroimidazol-2-yl)-phenylmethanone 2-chloro-5-(1,1-dimethylbenzo[f]quinoxalin-3-ium-6-yl)benzaldehyde N'-[(2S)-1-hydroxybutan-2-yl]-4-[1-[3-(trifluoromethoxy)phenyl]-1,2,4-triazol-3-yl]pyridine-2-carboximidamide 2-[4-(difluoromethyl)phenyl]-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine 3-(2-butoxypyridin-4-yl)pyrazolo[1,5-a]pyrazine 3-[4-(diethylamino)butyl]-6,11b-dihydrothiochromeno[2,1-c]quinazoline-12,13-dione 4-[3-(2-chloroethylamino)propyl]phenol;hydrochloride 2-[(3Z)-4,5-dimethylhepta-1,3,6-trien-3-yl]-6-methylidene-7-[4-(2-methylphenyl)butylsulfanyl]-1H-imidazo[4,5-d]pyridazine ethane;N-(2,4,6-trimethylphenyl)-5,7-dihydropyrrolo[3,4-b]pyridine-6-carboxamide 2-amino-4-[3-chloro-2-fluoro-5-(trifluoromethyl)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile 1,2-dichloropentan-3-one;6-methyl-4-[(3Z)-3-propylidenepiperidine-1-carbonyl]-1H-pyridin-2-one 1-[4,5,8a-trimethyl-7-(2-phenylpropanoyl)-3H-pyrazolo[1,5-a]pyridin-6-yl]-3-[6-chloro-3-fluoro-4-[[[(Z)-hydrazinylidenemethyl]amino]-methylsulfamoyl]naphthalen-2-yl]urea 2-[[5,6-bis(4-methoxyphenyl)pyridazine-3-carbonyl]amino]-3H-benzimidazole-5-carboxylic acid 2-[(3S)-5-[4-chloro-3-(trifluoromethyl)phenyl]-1-(cyclopropanecarbonyl)-4,6-difluoro-2,3-dihydroindol-3-yl]acetic acid 2-ethylhexoxy(propan-2-yloxy)phosphoryloxybenzene 4-cyclopentyloxy-N',5-dimethylbenzenesulfonohydrazide 1-[4-(9,10-dioxoanthracen-2-yl)oxybutanoyl]pyrrolidine-2-carboxylic acid 4-(3,5-dinitrophenyl)-1H-pyrazole 1-(4-methylphenyl)-5,6-dihydro-4H-pyrazolo[3,4-d]pyrimidine [2-(aminomethyl)phenyl]sulfanylaminooxybenzene (1R,2S)-6-chloro-1-fluoro-5-hydroxy-2-methyl-2H-anthracene-9,10-dione N-[(3S,4R)-1-cyclopentylpiperidin-4-yl]-5-methylpyridin-2-amine 1-[(4-methoxyphenyl)methyl]-2-phenylpiperidine ethane;4-methyl-N-[2,3,5,6-tetrafluoro-4-(2-iminocyclohexylidene)phenyl]benzamide 2-[4-(1-aminoethyl)phenyl]-N'-hydroxy-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-5-carboximidamide (3-chlorophenyl)methyl-[2,4-dichloro-5-[(E)-4-morpholin-4-ylbut-2-enoyl]phenyl]azanide N-azido-2,4-dichlorobenzenesulfonamide 2-[5-methyl-4,6-dioxo-1-(4-phenylsulfanylcyclohexa-2,4-dien-1-ylidene)pyridazin-3-yl]acetic acid 1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl)-3-(triazol-1-ylmethyl)piperidine 3-[(3,5-dimethylpyrazole-1-carbonyl)amino]-2,3-dihydropyridine-6-carboxylic acid 2-[3-(5-chloropyridin-1-ium-2-yl)oxypropanoyl]oxybenzoic acid 2,4-dioxo-5-[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]-3H-thieno[2,3-d]pyrimidine-6-carbonitrile 6-(1,3-benzothiazol-2-yl)-5-methylcyclohexa-1,4-diene-1,2-diamine N-[5-[2-(dimethylamino)pyrimidin-4-yl]-6,7-dihydro-1H-indazol-3-yl]benzamide 3-(9,10-dimethoxyanthracen-2-yl)propanoate N-[3,5-difluoro-4-(4-fluorophenoxy)phenyl]-4-morpholin-4-yl-6-oxo-1H-pyridazine-3-carboxamide 4-(benzenesulfonamido)-3-[3,5-dichloro-2-oxo-6-(trifluoromethylsulfanyloxyamino)pyridin-1-yl]benzamide 1-azido-2,3-bis(trifluoromethyl)naphthalene 1-[2-(4-azidophenoxy)ethyl]piperidine 5-[3,4-bis(phenylmethoxy)phenyl]pyrrolidin-2-one;propane N-[2-methyl-4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butanoyl]prop-2-enamide N'-[6-(4-methoxyanilino)pyridin-3-yl]ethane-1,2-diamine N-[(3,5-dimethylphenyl)methyl]cyclopropanamine;ethane 2-(2,2-diethoxyethyl)-4H-1,3-benzothiazine 5-(4,6-dimethoxypyrimidin-2-yl)isoquinoline;8,8,11-trimethyl-7,9,10,12-tetrahydro-6H-pyrrolo[3,2-a]phenanthridin-9-ol (7R)-2,3-dimethyl-5-oxo-N-(2-phenylethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide N-[4-(3-cyclobutylpropoxy)phenyl]-2,4,5-trimethylpyrazole-3-carboxamide 2-amino-4,6-bis(trifluoromethyl)pyridine-3,5-dicarbonitrile 1-azidooxy-3,5-dichlorobenzene 1-(2,6-dichlorophenyl)sulfonyl-N-[(4-ethylsulfanylphenyl)methoxy]-2-sulfanylideneimidazolidine-5-carboxamide 2-[(5-chloropyridin-2-yl)methylidene]propanedinitrile 4-[[5-chloro-1-(oxolan-3-yl)pyrrolo[2,3-b]pyridin-4-yl]methoxymethyl]benzenesulfonamide (1-methylsulfonylpiperidin-4-yl)-[4-(5-phenyl-3,6-dihydro-2H-pyridin-1-yl)piperidin-1-yl]methanone N-[2,5-di(propan-2-yl)phenyl]-3-oxobutanamide 3-(2,6-dichlorophenyl)-7-[4-methyl-1-(oxan-4-ylmethyl)piperidin-4-yl]-8H-imidazo[5,1-c][1,4]thiazin-6-amine 1-(4-azidophenyl)sulfanylpyrrolidine 1-(2,6-dimethylphenyl)-3-[[3-fluoro-5-(trifluoromethoxy)phenyl]sulfonylamino]urea (2R)-2-[(3S)-5-fluoro-1-phenylpentan-3-yl]cyclohexane-1-carboxylic acid (2S,3R)-N-[2-(4-chlorophenyl)propan-2-yl]-2-(2,4-dioxopyrimidin-1-yl)-3-methylpentanamide (Z)-3,7-diethyl-6-hydroxynon-5-en-4-one;iridium;2-phenyl-4-(1-propan-2-ylpyrazol-4-yl)pyridine N-azido-4-(2,5-difluorophenyl)piperazine-1-carboxamide 3-(2,4-dichlorophenyl)-6-[4-(5-ethylpyridin-2-yl)oxypiperidine-1-carbonyl]-7-methyl-1H-quinazoline-2,4-dione 3-[(2,5-dihydroxyphenyl)diazenyl]-4H-1,2,4-triazin-6-one 1-(2,4-dichlorophenyl)-N-[5-(furan-3-ylmethylsulfanyl)pyridin-2-yl]pyrazole-3-carboxamide 2-[(4R)-6-amino-3,4-dihydro-2H-thiochromene-4-carboximidoyl]phenol (2S)-4-(1H-imidazol-5-ylmethylideneamino)-N,3-diphenylbutanamide 1-ethyl-4-[4-(2-hydroxypropan-2-yl)cyclohexa-2,4-dien-1-yl]sulfonyl-3,5-dihydro-2H-1,4-benzodiazepine-8-carboxamide (2R,3aS,9aR)-6-methyl-N-[2-(4-pyridin-4-ylpiperazin-1-yl)ethyl]-2,3,3a,5,7,8,9,9a-octahydrofuro[3,2-b]azepine-2-carboxamide 1-[(E)-3,7-diethyloct-4-enyl]naphthalene N-(4-bromobutan-2-yl)-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide N-(5-cyanopyridin-2-yl)cyclopropanecarboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]acetamide 3-N-(4-bromophenyl)-1H-1,2,4-triazole-3,5-diamine;4-chloro-N-[2-methoxy-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]benzamide N-[4-(diethylamino)phenyl]-2,6-bis(1,3,5-triazin-2-yl)pyridine-4-carboxamide (3S)-5-amino-N-[1-cyclopropyl-4-fluoro-6-[(2R)-1,1,1-trifluoropropan-2-yl]benzimidazol-2-yl]-4-(dimethoxymethyl)-3-fluoropentanamide 6-[2,4-dihydroxy-5-(3-methylphenyl)phenoxy]-N-hydroxyhexanamide 2-(4,5-dimethyltriazol-1-yl)-N-ethyl-2-[6-(3,3,5,5-tetramethylpiperidine-1-carbonyl)pyridin-2-yl]acetamide 4-(3,5-diethylimidazol-4-yl)-2-piperidin-1-yl-[1]benzofuro[2,3-d]pyrimidine;hydrochloride 1-[3,5-bis(trifluoromethyl)phenyl]-N-deuterio-2,2-dimethoxyethanimine 3-[5-methoxy-2-(2,4,6-trifluoroanilino)pyrimidin-4-yl]-N-[1-(sulfanylmethyl)piperidin-3-yl]benzamide 7-[4-[2-(diethylamino)ethoxy]-2,3-bis[4-(dimethylamino)phenyl]azetidine-1-carbonyl]naphthalene-2-sulfonamide 1-(3,5-difluorophenyl)-2,2,2-trifluoroethanone 7-methoxy-2-[4-(trifluoromethyl)phenyl]chromene-4-thione (2-cyclopropylphenyl)methoxycarbonylimino-[1-[4-fluoro-3-(trifluoromethyl)phenyl]azetidine-3-carbothioyl]azanium 2-[1-carboxypropan-2-yl(prop-2-enyl)amino]benzoic acid N-ethyl-3,4,5-trifluoro-2-[(1R)-1-naphthalen-1-ylethoxy]aniline 3-(2,5-dimethylpyrrolidin-1-yl)sulfonylquinoline N-[[1-[(2-hydroxy-5-nitrophenyl)methyl]piperidin-4-ylidene]methyl]acetamide (2E,4Z)-3,5-dihydroxyhexa-2,4-dienoic acid;N'-[6-(pyridine-3-carbonylamino)hexyl]propanediamide N-[(1Z,3E)-2-[2-[(4,5-diphenylthiophen-2-yl)methoxy]ethylamino]penta-1,3-dienyl]propanamide ethane;2-[[6-(4-methylphenyl)pyridine-3-carbonyl]amino]propanoic acid 2-amino-9-[(4R)-1,3-dihydroxypropan-2-yl]-7H-purin-8-one;cyclohepta[d]pyrimidin-4-amine 4-[2-hydroxy-3,5-di(propan-2-yl)cyclopenta-1,4-dien-1-yl]-2,6-bis(sulfanyl)phenol 2-[4-(4,5-dihydro-1H-imidazol-2-yl)-3-fluorophenyl]-7-methoxyquinoline 2-[1-(4-methylphenyl)indol-3-yl]acetamide 2-(cyclobutylmethyl)-4-[1-[(5-fluoropyridin-3-yl)amino]ethylideneamino]-6,7,8,9-tetrahydropyrimido[5,4-b]azepine-5-carbonitrile 4-[(3S)-2,6-dioxopiperidin-3-yl]oxy-N-hydroxybenzamide 6-(3,4-dimethoxybenzoyl)-2-[(3S)-1-propanoylpyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 6-[2,5-dimethyl-1-(1H-pyrazol-4-yl)pyrrole-3-carbonyl]-2-(4-fluorophenyl)-N-hydroxyheptanamide (Z)-3-amino-N'-methoxy-2-methylidene-4-[5-[methyl(3-methylbutyl)amino]pent-1-ynylsulfanyl]but-3-enimidamide;ethane 2-amino-9,10-dihydroxy-1H-anthracene-9,10-dione 2-[[(3S,4R)-3-hydroxypiperidin-4-yl]methyl]isoindole-1,3-dione 7-fluoro-2,4-dihydroxynaphthalene-1,3-disulfonic acid 2-[1,3-dihydroxy-6-[(4-nitrophenyl)methylsulfanyl]isoindol-2-yl]acetic acid 5-fluoro-2-[6-fluoro-7-(4-methylpiperidin-1-yl)-3H-imidazo[4,5-c]pyridin-2-yl]-8-methoxy-[1,2,4]triazolo[1,5-a]pyridine (2S)-2-amino-3-[6-(trifluoromethylsulfanyl)indol-1-yl]propanoic acid 1-(5,8-difluoroquinolin-3-yl)-2-[6-hydroxy-7-(4-methylpiperazin-1-yl)quinolin-4-yl]oxyethanone 3-(2,4-difluorophenyl)sulfanyl-6-methoxy-N-[[2-(trifluoromethylsulfanyl)phenyl]methylideneamino]pyridin-2-amine 3-amino-N',2-dimethyl-5-[methyl(oxan-4-yl)amino]benzenecarboximidamide;ethane [4-[4-[3-(dimethylamino)propoxy]phenyl]piperazin-1-yl]-(5-methoxyspiro[2H-1-benzofuran-3,3'-pyrrolidine]-1'-yl)methanone 1-[3-[4-(cyclohexylmethoxy)phenoxy]phenyl]ethanone 4-[3-(1,1-difluoropropyl)phenyl]piperidine;ethane 2-bromo-5-[3-[[2,6-di(propan-2-yl)phenyl]iminomethyl]pyrrol-1-id-2-yl]phenol 5-(cyclopenten-1-yl)-2,4-dimethoxyaniline 2-amino-4-(4-hydroxypiperidin-1-yl)-5,6,7,8-tetrahydroquinazoline-6-carbonitrile (5E)-2-cyclohexylimino-5-[(7-fluoro-1,3-benzodioxol-4-yl)methylidene]-1,3-thiazolidin-4-one 2-azido-3-methyl-6,7-dihydrocyclohepta[d][1,2]thiazole (6S)-3,4-bis(chloromethyl)-8-oxatetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),10,12,14-tetraene 1-benzylsulfanyl-3,5-bis(chloromethyl)benzene ethane;3-(4-fluorophenyl)-2,5-dimethylpyridine N-cyclohexa-1,3-dien-1-yl-5-(4-nitrophenyl)-3,6-dihydro-1,3,4-thiadiazin-2-imine 5-[1-(2-fluorophenyl)ethyl]pyrimidine 2-[4-[(6-butylbenzo[b][1,4]benzothiazepine-3-carbonyl)amino]piperidin-1-yl]acetic acid 4-[(3-chloropyridin-2-yl)diazenyl]aniline;ethane 2,4-dimethyl-7H-pyrrolo[3,4-b]pyridine;(5Z)-N-ethyl-6,10-dimethyl-2,3-dihydrotriazolo[1,2-a]azocin-5-amine (3-methylsulfonylphenyl)-[4-propan-2-yl-2-[(pyridine-4-carbonylamino)methyl]pyrrolidin-1-yl]azanium 1-(1H-indol-2-yl)-4,4-dimethoxybutane-1,3-dione 2-amino-N'-(3-bromophenyl)-6-[1-methoxyethyl(methyl)carbamoyl]pyridine-4-carboximidamide 4-[[3-(dimethylamino)cyclohexyl]amino]-2-propan-2-ylidene-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidine-1,8-dione 1-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)pyrrolidine-3-carboxylic acid 2-[[2-hydroxy-5-(trifluoromethyl)phenyl]methylideneamino]benzonitrile (E)-3-[5-(ethoxymethyl)naphthalen-2-yl]prop-1-en-1-amine 1-[(Z,4E)-4-ethylidene-3-methylhept-2-en-2-yl]-9H-fluorene 4-[(2R)-3-amino-1-oxo-1-sulfanylpropan-2-yl]benzoic acid 4-[[2,6-dichloro-4-(trifluoromethyl)phenyl]carbamoylamino]-3-ethylsulfonylbenzoic acid 2-methoxycarbonyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carboxylic acid 1-(2,3-dimethoxyphenyl)-N-[3-[(4S)-2'-oxospiro[3H-chromene-4,5'-imidazolidine]-4'-yl]-1,2-benzothiazol-6-yl]cyclopropane-1-carboxamide 4-[5-[1-(3,5-dimethoxyphenyl)ethylidene]-4-oxopiperidin-3-yl]benzoic acid N-[3-[4-(benzylamino)-1,2,5-oxadiazol-3-yl]phenyl]-2-bromo-6-chlorobenzamide N-[6-(1H-imidazol-5-yl)quinolin-4-yl]cyclohexanecarboxamide 2-azido-N,N-dimethylquinazoline-4-carboxamide 3-[4-chloro-2-(trifluoromethyl)phenoxy]-5-fluoro-N-propan-2-ylpyridine-2-carboxamide ethane;6-fluoro-5-(4-fluorophenyl)-1-methyl-3H-indol-2-one 3-[(2,4-dichloropyrimidin-5-yl)-(furan-2-ylmethoxycarbonyl)amino]butanoic acid 6-(4-methoxyphenyl)sulfonyl-3,4,5,7-tetrahydropyrrolo[2,3-c]pyridine 1-(4-aminopiperidine-1-carboximidoyl)sulfonyl-3-[5-methyl-6-[2-oxo-8-[3-(trifluoromethoxy)phenyl]-1,3-dihydropyrido[2,3-b]pyrazin-7-yl]pyridin-3-yl]urea 2-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-N-(5-cyclopropylsulfonylpyridin-2-yl)-6-oxo-1H-pyrimidine-4-carboxamide 2-[2-(3,5-difluorophenyl)-5-methylmorpholine-4-carbonyl]benzonitrile 1-azidooxy-N,3-diphenylmethanesulfonamide 2-[4-(azidomethyl)phenyl]-N-methylethanamine [(2S,4R)-4-methylpiperidin-2-yl]-[2-(triazol-1-yl)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl]methanone 5-chloro-N-methyl-4-[2-(propan-2-ylamino)ethyl]thiophene-2-sulfonamide 5-chloro-N-[(2S)-1-hydroxypropan-2-yl]-4-[2-methoxyethyl(methyl)amino]thiophene-2-carboxamide N-[2-(4-chloroanilino)-1,3-thiazol-5-yl]-N'-(2-hydroxyethoxy)-2-(1H-indol-6-ylsulfanylamino)acetohydrazide 2-(1,3-benzothiazol-2-yl)benzene-1,4-diol 6-chloro-4-methoxycarbonylnaphthalene-2,3-dicarboxylic acid 6-(1,3-benzodioxol-5-yl)imidazo[2,1-b][1,3]thiazol-3-one 6-[4-[3-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]sulfonylphenyl]pyrazin-2-amine 2-bromo-5-chloro-4-methylpyrazolo[1,5-a]pyridine 1-azido-4-(2,4-dichlorophenyl)piperazine N'-[4,6-dichloro-5-(trifluoromethyl)pyrimidin-2-yl]benzohydrazide 1-[4-methyl-2-(3,5,6,7-tetrahydropyrrolo[3,4-d]pyrimidin-4-ylidene)-4a,5,8,9,10,11-hexahydrocycloocta[b]indol-1-yl]prop-2-en-1-one 1-methyl-4,10,10a-trioxo-5H-benzo[b]carbazole-7-carbonitrile 4-(2-ethylsulfanylphenoxy)-1-oxidopyridin-1-ium 4-N-[4-(2,5-dimethylphenyl)butan-2-ylideneamino]benzene-1,4-diamine (6S,9R)-9-(4-fluorophenyl)-2-[(4-methylphenyl)methylsulfanyl]-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 2-[2,3-dibromopropyl(methoxycarbonyl)amino]benzoic acid 1-[(E)-2-(4-hydroxyphenyl)ethenyl]naphthalene-2-sulfonic acid 1-(3,4-difluorophenyl)-2-[6-ethyl-3-methoxy-2-(oxan-4-ylamino)quinoline-5-carbonyl]prop-2-en-1-one 2-[5-(1,3-benzodioxol-4-yl)-6-methylpyrazolo[4,3-b]pyridin-2-yl]propanoic acid 3-(9,9-diethylfluoren-4-yl)-N-phenylaniline;methane 4-[(E)-2,3-dimethylbut-1-enyl]-1-[2-[5-[(2R)-pyrrolidin-2-yl]pentoxy]ethylamino]anthracene-9,10-dione [4-[1-(2,6-dimethylphenyl)imidazol-2-yl]-7H-tetrazolo[5,1-c][1,4]benzoxazin-8-yl]oxymethanamine 4-bromo-N'-hydroxynaphthalene-2-carboximidamide N-(3-chlorophenyl)-4,5-dimethylcyclohexa-2,4-diene-1-carboxamide N-methyl-3-nitro-N-(2-phenoxyethyl)aniline [5-(1H-indol-4-yl)cyclohexen-1-yl]methanol 2-(N-ethyl-3-nitroanilino)benzenesulfonic acid 4-(2-methoxyphenyl)-6-oxo-2,3-dihydro-1H-pyridine-5-carboxylic acid 4-[1-azidosulfanyl-2,3-bis(benzenesulfonyl)-9H-fluoren-4-yl]morpholine 1-azidooxy-4,7-dimethyl-2H-naphthalene (3R)-4-amino-2,5-dihydroxy-N-methylsulfonyl-3-[5-(4-phenylphenyl)thiophen-3-yl]pentanamide 4-chloro-N,2-dimethyl-3-oxobutanamide;(E)-[5-[3-(3,5-difluorophenyl)-6-oxopyridazin-1-yl]pyridin-2-yl]oxy-ethylidene-prop-1-ene 3-[2-[3-(dimethylamino)propoxy]phenyl]-N,4-diphenylbenzamide 5-ethyl-N-[[2-(2,3,4,5-tetramethoxyphenyl)imidazol-1-yl]methyl]-6H-indolo[2,3-b]quinoline-11-carboxamide N-[6-aminosulfanyl-5-(4-fluorophenoxy)pyrimidin-4-yl]hydroxylamine 5-[5-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]-1-[2-(5-ethyl-1H-imidazol-2-yl)propan-2-yl]-6-methylidenepyridine-3-carbonitrile 4-[3-amino-6-(1,5-dimethylpyrazol-4-yl)pyrazin-2-yl]piperazine-1-carboxylic acid (2R,4S)-1-[3,5-bis(trifluoromethyl)benzoyl]-N-[[2-chloro-6-(difluoromethoxy)phenyl]methyl]-4-fluoropyrrolidine-2-carboxamide 4-[1,3-benzothiazol-2-yl(butanoyl)amino]benzenesulfonic acid 4-(2,5-dimethylphenyl)sulfonylmorpholine 2-[3-(2,6-dichlorophenyl)-2-oxopropyl]benzamide (3S)-N-[2-(dimethylamino)ethyl]-1'-[[4-(4-fluorophenyl)phenyl]methyl]-6-methoxyspiro[1,2-dihydroindene-3,4'-piperidine]-2'-carboxamide N-(2,5-dichlorophenyl)-2,4,6-trimethyl-N-phenacylbenzenesulfonamide N-[4-(3,4-difluorophenyl)-5-pyridin-2-ylpyrimidin-2-yl]-2-methoxyacetamide;ethane 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[3-(trifluoromethoxy)phenyl]sulfinylurea N-[3-methoxy-4-(2-piperidin-1-ylethoxy)phenyl]methanimine N-azido-5-nitroindole-1-carboxamide 2-amino-4,5-dimethylbenzenesulfonic acid;N'-(3,4-dihydro-1H-isoquinolin-2-yl)-N-methylidenemethanimidamide N-[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]-3-hydroxyazetidine-1-carboxamide 3,5-dichloro-N-(1H-indol-6-ylmethylideneamino)benzamide 2-[(3S)-4-(2,5-dimethylphenyl)sulfonyl-6,8-difluoro-1,4-dihydroquinoxalin-2-yl]acetic acid 2-[[4-(4,6-diphenylpyrimidin-5-yl)phenyl]methylidene]indene-1,3-dione N-[(2S)-1-hydroxypropan-2-yl]benzamide;4-[[3-(trifluoromethylsulfanyl)phenyl]carbamoylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acid 2,6-dibromo-4-[(E)-[4-cyclopropylimino-2-[[3-(2-methoxyphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]pyrazolo[1,5-a][1,3,5]triazin-8-ylidene]methyl]phenol 1-(5,6-dihydropyrido[2,3-b]pyrazin-7-yl)ethanone 3-(5-carbamoylpyridin-2-yl)-N-[[4-(4-methylphenyl)sulfanyloxolan-2-yl]methyl]piperidine-1-carboxamide 4-[2,6-difluoro-N-(2-methylpropyl)anilino]butan-1-ol 3-[2-(trifluoromethyl)phenyl]propanehydrazide 4-methyl-6,8-diazatetracyclo[7.5.0.02,7.010,14]tetradeca-1(9),2,4,6,10(14),11-hexaene 2-(3,4-dimethyl-1,2-oxazol-5-yl)benzenesulfonamide 2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)cyclopropan-1-one N-[4-(2,3-dimethylphenoxy)phenyl]quinoline-6-carboxamide 5-azido-1-methylpyrazolo[3,4-c]pyridine 3-(4,6-difluoro-1H-benzimidazole-2-carbonyl)-N-[(1S)-1-phenylethyl]imidazolidine-4-carboxamide [(2R)-4-(3,6-dimethylpyrazolo[1,5-a]pyridine-2-carbonyl)morpholin-2-yl]methanolate [3-[5-(cyclobutanecarbonyl)-1,2,4-oxadiazol-3-yl]piperidin-1-yl]-(oxolan-2-yl)methanone 2-(dimethylamino)-N-[5,7,10-trioxo-6-phenyl-3,9-bis(propanoylamino)anthracen-1-yl]acetamide 3-[4-(2,6-difluorocyclohexa-1,5-dien-1-yl)pyrazol-1-yl]-N'-hydroxybenzenecarboximidamide (2S)-N,2-dihydroxy-2-[(5R)-5-methyl-4-oxo-9-(2,2,2-trifluoroethyl)-1,3-diazatricyclo[6.3.0.02,4]undeca-10-en-11-yl]-3-phenylpropanamide 6-[(4,4-difluoropiperidin-1-yl)methyl]-3-methylimidazo[2,1-b][1,3]thiazole N-[4-(4-aminoanilino)phenyl]sulfonylbenzamide 3-(1H-pyrazol-5-yl)-4,5-dihydro-1H-benzo[g]indazole 2-[(5Z)-4-oxo-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetamide 2-methyl-3-[(7R)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid N-[(4S)-1,3-thiazolidin-4-yl]-2-[4-[3-(trifluoromethoxy)phenoxy]piperidin-1-yl]pyrimidine-5-carboxamide 3-(5,6-dimethoxypyridin-3-yl)-2H-pyrazolo[3,4-d]pyrimidine (3R)-1-[4-chloro-2-methyl-6-(4-phenylphenyl)sulfanylpyrimidin-5-yl]pyrrolidin-3-amine 2,3-diiodo-4-(methoxymethyl)thiophene [4-amino-3-(ethoxymethyl)piperidin-1-yl]-[4-chloro-2,6-difluoro-3-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)phenyl]methanone 3-N,5-dimethyl-7-N-(pyridin-2-ylmethyl)triazolo[4,5-d]pyrimidine-3,7-diamine;ethane 2-chloro-3-(4-iodophenyl)pyridine (E)-N,3-dimethyl-4-[1-[2-methyl-6-(trifluoromethoxy)pyridin-4-yl]azetidin-3-yl]but-2-enamide N-[4-(hydroxymethyl)cyclohexyl]-3,4-dihydro-1H-isoquinoline-2-sulfonamide 1-(3-bromophenyl)-6-oxopiperidine-2,4-dicarboxylic acid N'-[2,3,5,6-tetrafluoro-4-(3,3,3-trifluoropropylamino)phenyl]-N-(1H-pyrazolo[4,3-b]pyridin-3-ylmethoxy)oxamide 1-[4-(2-chloroacetyl)phenyl]-3-methylcyclohex-4-ene-1,3-dicarboxylic acid 2-(6-oxobenzo[c]chromen-7-yl)oxyacetic acid (5R)-2-amino-N'-[4-cyano-3-(trifluoromethyl)phenyl]-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carbohydrazide N-azido-1,3,5-trimethylpyrazolo[4,3-d]pyrimidin-7-amine 1-[3-(2-methylphenyl)buta-1,3-dienyl]imidazole N-(4,6-dimethylpyrimidin-2-yl)-5-(1-ethylpiperidin-3-yl)-1H-pyrazole-3-carboxamide 6-[2,5-dimethyl-1-[(3S)-pyrrolidine-3-carbonyl]pyrrol-3-yl]hexanoic acid N-[(1R)-5-chloro-2,3-dihydro-1H-inden-1-yl]benzamide [4-(4,4,5,5-tetramethyloxaborolan-2-yl)phenyl]-[3-(trifluoromethoxy)pyrrolidin-1-yl]methanone 3-[7,9-dimethyl-2-[4-(oxan-2-yloxy)anilino]purin-6-yl]sulfanylpropan-1-ol 2-[4-[5-(3,5-dimethyltriazolo[4,5-b]pyridin-7-yl)-1-methylbenzimidazol-2-yl]butanoylamino]ethanesulfonic acid 4-[4-[(1R,2S)-2-[4-[(E)-3-methoxybut-2-enyl]piperidine-1-carbonyl]cyclopropyl]phenyl]benzoic acid [4-(aminomethyl)phenyl]-[7-(5-fluoro-3,4-dihydropyridin-6-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]methanone 3-[4-[4-(1,6-diazocin-5-yl)phenoxy]piperidin-1-yl]sulfonylbenzoic acid 2-(2,6-difluorophenyl)-N-[(4-hydroxy-3-methoxyphenyl)methylideneamino]propanamide 1-[3-ethyl-2,6-difluoro-4-(oxiran-2-ylmethoxy)phenyl]ethanone 4-[5-methylsulfonyl-6-(2,2,3-trifluoropropoxy)pyridin-3-yl]-6-[6-(oxolan-3-ylmethylamino)pyridazin-3-yl]pyrazolo[1,5-a]pyridine-3-carbonitrile 3-azidooxy-1,6,7,8-tetrahydrocyclopenta[e]indole 2-[3-(hydroxymethyl)piperidine-1-carbonyl]-4,6-dimethoxybenzaldehyde 2-[4-fluoro-3,5-di(propan-2-yl)phenyl]acetic acid N-[2,4-dihydroxy-5-(3-methylcyclohexa-1,5-dien-1-yl)phenyl]-6-hydroxyhexanamide 7-[(4-chlorophenyl)methyl]-3-hydroxy-2H-pyrrolo[3,4-f]isoindol-1-one 4-[(4R,5S)-7-chloro-4,5-dihydroxy-2-methoxy-1-methyl-3,4-dihydro-1H-isoquinolin-8-yl]benzenesulfonamide N-[2-(4-hydroxyphenyl)ethyl]-1,3-dimethyl-5-propan-2-ylpyrazole-4-carboxamide (2-fluoro-3-octan-4-ylphenyl)boronic acid 2-[1-(cyclopropylmethoxy)isoquinolin-3-yl]-N-[(2S)-3,4-dihydro-2H-chromen-2-yl]acetamide 4-tert-butyl-N-[[1-[(2S)-3,3,3-trifluoro-2-hydroxypropanoyl]piperidin-4-yl]methyl]benzamide 5-azidooxy-1,2-dimethylindole 2-[(1E,3Z)-5-aminohexa-1,3,5-trienyl]-5-chloropyrimidine-4,6-diamine 3-[1-(cyclobutylmethyl)piperidin-4-yl]oxy-5,6-dimethylpyridazine 5-[4-(cyclopropylmethoxy)phenyl]-1,3-oxazole;N-ethanimidoyl-2-pyrrolidin-1-ylpyridine-4-carboximidamide N-[(4E)-5-(furan-2-ylmethoxymethylimino)-3,7-dihydrofuro[3,2-e][1]benzofuran-6-ylidene]hydroxylamine 4-methylsulfanyl-3,5-dinitrobenzoic acid [4-amino-2-(3-bromopyridin-2-yl)imino-1,3-thiazol-3-yl]urea 2-methyl-6-[3-(trifluoromethoxy)phenyl]pyridine 2-ethyl-3-(methylamino)benzo[f]benzimidazole-4,9-dione N'-(dimethylamino)-N-[5-fluoro-1-[[4-[4-(trifluoromethoxy)phenoxy]phenyl]methylcarbamoyl]naphthalen-2-yl]ethanimidamide N-[3,5-bis(trifluoromethyl)phenyl]-4-(2-oxopiperidine-1-carbonyl)piperidine-1-carboxamide [3-chloro-5-(trifluoromethyl)phenyl]-(2,5,6-tetrahydro-1H-benzo[h]quinolin-7-ylamino)methanol 5-[(1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl)amino]quinoline-8-carbonitrile 2-(4-bromophenyl)-N-(diaminomethylideneamino)-N,5-diethyl-1H-imidazole-4-carboxamide 3-butan-2-yl-4,5-dimethoxybenzaldehyde N-[2-(dimethylamino)ethyl]-3,4-dihydro-1H-naphthalene-2-carboxamide 5-methyl-2-(oxolan-3-yl)pyrazole-3-carboxamide 1-(2-chlorophenyl)-4-(4,5-dihydro-1,3-oxazol-2-ylmethoxymethyl)piperidine (4S)-1,3-dimethyl-5,6-bis[[4-(2,4,4-trimethylpentan-2-yloxy)phenyl]sulfonyl]-2,4-dihydropyrimidine 7-(3,4-dimethoxyphenyl)pyrido[2,3-b]pyrazine [1-carboxy-3,5-di(propan-2-yl)pyrazol-4-yl]iodanuidyl-naphthalen-1-ylazanium 3-(2,5-dimethoxyanilino)sulfanyl-4-propylbenzoic acid 2-[(1S)-1,6-dimethyl-3,4-dihydro-2H-naphthalen-1-yl]phenol 4-ethyl-5-[(Z)-3-pyridin-2-ylprop-1-enyl]imidazolidine-2,4-dione N-[2,6-di(propan-2-yl)phenyl]-1-oxopropane-2-sulfonamide N-(3,4-dimethylphenyl)-2-[6-hydroxy-2-(2-methoxyethyl)-1-oxoisoquinolin-4-yl]acetamide 2-[(5,5-dimethylhexylamino)methyl]-3H-thieno[3,2-d]pyrimidin-4-one 4-[4,4-bis(3-fluorophenyl)butyl]aniline;ethane 1-methyl-4-[(3-phenylmethoxyphenyl)methyl]piperazine 5-bromo-3,4-diethyl-1H-pyrimidine-2,6-dione 1-azidooxy-2,3,4-tris(ethenyl)benzene ethane;6-methyl-1-[(E)-1,3,3-triphenylprop-2-enoxy]naphthalene 2-[1,6-dimethyl-4-[[4-(trifluoromethoxy)phenyl]carbamoylamino]cyclohexa-2,4-dien-1-yl]acetic acid 1-[4-[(E)-2-nitroethenyl]phenyl]naphthalene (2S)-N-(4,5-dimethyl-1H-pyrazol-3-yl)azepane-2-carboxamide;hydrochloride 2-[(4Z)-4-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-3-oxo-1-phenylpyrazolidin-2-yl]acetic acid 3-[(3aR,7aS)-2,5-dioxo-1,3,3a,4,6,7,7a-octahydrothieno[3,4-c]pyridine-7-carbonyl]-N,N-dimethylbenzamide 3-butyl-4-[5,6-difluoro-2-(hydroxymethyl)pyridin-3-yl]-N'-hydrazinylbenzenecarboximidamide N-[4-amino-2-(difluoromethyl)phenyl]-2-chloro-5-[(3,3-dibromo-1-hydroxypropyl)sulfonylcarbamoylamino]benzamide 3-[4-(cyclobutylmethoxy)phenyl]-N'-hydroxypyridazine-4-carboximidamide 2-[4-(2,5-dihydroxyphenyl)-6-methylpyrimidin-2-yl]sulfanyl-N-[(3-hydroxyphenyl)methylideneamino]acetamide (2S,4R)-N'-diazenyl-5-fluoro-3-hydroxy-4-methoxyimino-7-morpholin-4-yl-N-phenylspiro[1H-quinoline-2,1'-cyclopentane]-6-sulfonamide (2R,3S)-N,3-dimethyl-1-(oxan-4-yl)-5-oxo-2-phenylpyrazolidine-3-carboxamide 1-methyl-5-(3-methylcyclohexyl)oxypyrazole N-[(2S)-1-amino-3-(2,4-difluorophenyl)-3-methylbutan-2-yl]formamide 5-benzylsulfonyl-2,3-dimethoxyphenol [2-chloro-5-fluoro-4-(hydroxymethyl)phenyl]-spiro[1H-3,1-benzoxazine-4,3'-pyrrolidine]-2-one 4-[2-(aminomethyl)phenyl]-1-azido-N,N-dibutylpiperidin-3-amine 1-[(4R)-6,7-dimethoxy-3,4-dihydro-2H-chromen-4-yl]pyrrolidine;hydrochloride 1-chloro-2,3-bis(ethenyl)naphthalene N-[3-[[5-cyano-6-(7,8-dimethyl-1-oxoisoquinolin-2-yl)pyridin-3-yl]amino]prop-1-en-2-yl]-N-ethylformamide 1-(6,7-dimethyl-2-phenylpyrazolo[4,3-c]pyridin-5-yl)ethanone (2S)-4-methyl-5-oxo-3,4-dihydro-1H-1,5-benzodiazepine-2-carboxylic acid 2-[[7,8-dichloro-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]isoindole-1,3-dione 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;8-ethyl-3-methyl-2-phenylisoquinolin-1-one 2-[3,5-dibromo-4-[(E)-3-cyanopent-1-enyl]sulfanyloxyphenyl]acetic acid 2-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-3-[4-(trifluoromethoxy)phenyl]sulfonylpropanoic acid 6,8-dibromo-4-oxochromene-3-carboxylic acid 2-methyl-4-[2,3,5,6-tetradeuterio-4-(trifluoromethoxy)phenyl]-N-[2-(propan-2-ylsulfonylamino)-1,3-thiazol-5-yl]pyrazole-3-carboxamide 1-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonylamino)phenyl]cyclopropane-1-carboxylic acid (3Z)-7-fluoro-1-[4-methyl-2-(trifluoromethoxy)phenyl]-3-[3-(1H-pyrazol-5-ylamino)butan-2-ylidene]-2H-isoindole-5,6-dione 2-[2,5-dichloro-N-(2,3-dihydroxypropyl)anilino]acetamide 2-[5-(4,4-dimethylpiperidin-1-yl)pyridin-3-yl]-6-hydroxyiminocyclohexa-2,4-dien-1-one N-[(2,4-dichloropyrimidin-5-yl)methyl]-7H-purine-6-carboxamide 2-amino-4-[3-(1,3-dioxolan-2-yl)phenyl]-6-methylbenzene-1,3-dicarbonitrile 1-[[5-(5,7-difluoroquinolin-6-yl)thiophen-2-yl]methyl]pyridine-4-carboxylic acid N-[4-chloro-3-(trifluoromethyl)phenyl]-5,7-dihydropyrrolo[2,3-d]pyrimidine-6-carboxamide 1-(6-bromopyridin-2-yl)butan-2-ol 3-methyl-2,7-bis[(4-methylphenyl)methyl]inden-1-one 2-[4,7-dimethyl-3-[(2E)-2-[1-(4-nitrophenyl)ethylidene]hydrazinyl]imidazo[4,5-b]pyridin-5-yl]oxyacetic acid 2-[3-methylbutoxy(phenacyl)amino]acetamide (2S,4R)-1-[5-chloro-3-(4,6-dimethoxypyrimidin-2-yl)imidazo[1,2-a]pyridine-7-carbonyl]-4-fluoropyrrolidine-2-carbonitrile 6-hydroxy-5-[(2E)-5-oxohepta-2,6-dienyl]-1H-pyrimidine-2,4-dione 3-[(2E)-2-[(3,5-dichlorophenyl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one 7-azido-4-ethoxynaphthalene-2,6-diol 2-[1-(4-chlorophenyl)sulfonyl-7-fluoroindol-3-yl]acetamide [2-[(3,4-dimethylphenyl)methoxy]phenyl]boronic acid N-[2-(4-methylpiperazin-1-yl)-5H-pyrrolo[3,2-d]pyrimidin-4-ylidene]hydroxylamine 1-(4-cyanophenyl)-N',N'-dimethyl-1-(3-nitrophenoxy)methanediamine 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonylamino)-3-thiophen-2-ylpropanoic acid N-[4-[3-(dimethylamino)propoxy]phenyl]-7,11,14-trihydroxy-2,10-dioxatricyclo[7.6.0.03,8]pentadeca-1(15),2,4,6,12,14-hexaene-17-carboxamide [2-[4-chloro-3-(5-methylsulfonylpentoxy)phenyl]-1,3-thiazol-4-yl]-(2,6-diethylmorpholin-4-ium-4-ylidene)methanolate [4-[(5S)-6-amino-3,7,9-triazatricyclo[6.4.0.02,4]dodeca-1(8),6,9,11-tetraen-5-yl]phenyl]-(morpholin-4-ylmethyl)-oxoazanium (6R)-2-[3-[1-(4,5,6,7-tetrahydro-1H-indazole-5-carbonyl)azetidin-3-yl]oxyphenyl]-6-(2,2,2-trifluoroethyl)oxan-4-ol 2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5-[1-[3-hydroxy-2-oxo-2-(1-pyridin-4-ylcyclobutyl)ethyl]piperidin-4-ylidene]-7,8-dihydropyrimido[4,5-d]pyrimidin-6-one 5-fluoro-1-methyl-4,6-dihydropyrrolo[3,2-c]pyrazole;5-[(2E)-penta-2,4-dien-2-yl]-N-propan-2-ylpyridin-2-amine 1-(3-cyclohexa-1,5-dien-1-ylpropanoyl)naphthalene-2-carbonitrile 3-[1-[(4R)-2,2-dimethyloxan-4-yl]imidazol-2-yl]pyrazolo[1,5-a]pyridine [4-(2,5-dimethylbenzoyl)piperazin-1-yl]-[5-(methoxymethyl)thiophen-3-yl]methanone N-[(2S,3R)-1-amino-4,4-difluoro-3-hydroxybutan-2-yl]-7-cyclopropylsulfonylimidazo[1,5-a]pyridine-6-carboxamide N-(4,5-dimethylpyrimidin-2-yl)-4-[(3-fluorophenyl)methoxy]benzenesulfonamide 2,6-dimethoxyacridine;ethane 4-(4,5-dimethylfuran-2-carbonyl)-12-phenyl-1,4,8-triazacyclotetradecane-2,9-dione N-[4-amino-6-(methylamino)pyrimidine-5-carboximidoyl]-2-[3-fluoro-1-(3,3,3-trifluoropropyl)piperidin-3-yl]acetamide (3-propan-2-yloxyphenyl)methanamine;dihydrochloride 1-chloro-2-ethyl-3,4-dimethylthioxanthen-9-one 1-[(2R)-4,5-dimethyl-2-phenylcyclopent-3-en-1-ylidene]-3-ethoxyiminopropan-2-one 3-[2-[3,5-dichloro-4-[3-cyano-6-(1H-pyrazol-4-yl)pyrazin-2-yl]oxyphenyl]ethylamino]propanenitrilium 5-[3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxypyridine-3-carbonitrile 2-[6-(3,5-dimethyl-1,2-oxazol-4-yl)pyridin-3-yl]-8-(2,6-dipropylpyrimidin-4-yl)oxyimidazo[1,2-a]pyrazine 6-methyl-8-pyridin-3-ylimidazo[1,2-b]pyridazine 2-N,4-N-bis(2-bromophenyl)-1,3,5-triazine-2,4,6-triamine (3S,4R)-2-(hydroxymethyl)-1-[[(2R)-oxolan-2-yl]methyl]-3-thiophen-2-ylpiperidine-3,4-diol 3-chloro-2,5-bis(methylsulfanyl)pyridine 2-(4,5-dimethylthiophene-2-carbonyl)pyrrolidine-1-carboxylic acid 7-(dimethylamino)-5-methylsulfonylspiro[1,3-dihydroquinazoline-2,4'-piperidine]-4-one [3-(2-aminopyridin-4-yl)-5-ethoxy-1H-indol-7-yl]methanesulfonamide (4aR,10bR)-8a-methyl-9-(trifluoromethoxy)indeno[1,2-c]chromene 5-(4-fluorocyclohexa-1,3-dien-1-yl)oxy-2,3-bis[(E)-2-methylidenepent-3-enoxy]pyridine N-[4-(furan-3-yl)phenyl]-6-methoxyquinazolin-4-amine [4-(2,3-dihydroindol-1-ylsulfonyl)phenyl]boronic acid 5-cyclopropyl-N-cyclopropylsulfanyl-4-(2,2-dimethylpiperidin-1-yl)pyridin-3-amine 2-(3-fluorophenyl)-N-methyl-N-[[6-[4-[2-(trifluoromethyl)benzoyl]piperazine-1-carbonyl]pyridazin-3-yl]methyl]acetamide 2-[3,5-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]thieno[3,2-b]pyridine 5-[(2,4-dichloropyrimidin-5-yl)-(4-hydroxybutyl)amino]naphthalene-2-sulfonic acid (5E)-5-[(2,4-dihydroxyphenyl)methylidene]imidazolidine-2,4-dione N-[(3S)-1-(1H-benzimidazole-2-carbonyl)piperidin-3-yl]-2,5-dimethylfuran-3-carboxamide 2-(2,2-dihydroxy-4-oxo-5-phenylmethoxypentyl)propanedioic acid 2-(5,7-dihydroindolo[2,3-b]carbazol-12-yl)-4-nitrobenzonitrile 2-[1-(9,10-dichloro-4-oxo-6,7-dihydropyrimido[6,1-a]isoquinolin-3-yl)but-1-en-2-yl]benzonitrile N-[2,4-dichloro-3-(1,6-naphthyridin-5-yl)phenyl]-1,7-dimethyl-4-oxopyrrolo[3,2-c]pyridine-3-carboxamide 3-azidooxy-4,6-dipropylbenzene-1,2-disulfonic acid N-[2-fluoro-3-(4,4,5,5-tetramethyloxaborolan-2-yl)phenyl]pyridine-2-carboxamide (2S)-3,4,7-trihydroxy-1-[4-[6-(2-methoxyethyl)quinoline-2-carbonyl]piperazin-1-yl]heptane-2-sulfonamide (5E)-2-cyclopentylimino-5-[[3,4-dihydroxy-5-(2-methoxycarbonylphenoxy)phenyl]methylidene]-1,3-thiazolidin-4-one 5-azidooxy-4-methyl-6-phenylsulfanylpyrimidine 2-[2-amino-4-(4-phenylpiperidin-1-yl)butanoyl]sulfanylacetic acid 3-(3-fluorophenyl)-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-ylmethyl)propanamide N-[(1S)-2-cyanocyclohexyl]-4-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-7-ylsulfonylmethyl)-N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)benzamide 4-[2-(1,3-dioxoisoindol-5-yl)oxyethyl]-N-ethylmorpholine-2-carboxamide 2-amino-N-(3,3-difluorobutan-2-yl)pyrimidine-5-carboxamide 3-[(4-methoxyphenyl)sulfonylamino]-N,N-dimethylbenzamide N-(2,6-dimethylphenyl)sulfanyl-N',N'-diethylpropane-1,3-diamine 2-methoxy-N'-[(1E,3Z)-5-(4-phenylmethoxypiperidin-1-yl)hepta-1,3-dienyl]benzohydrazide N-[5-(2,4-difluorophenyl)sulfonyl-1H-indazol-3-yl]-4-morpholin-4-yl-6-pyrrolidin-1-ylpyrimidine-2-carboxamide 5-[2-[6-(1,3-benzodioxol-5-ylamino)pyrimidin-4-yl]ethynyl]thiophen-2-amine [2-[5-(2,3-dichlorophenyl)-1H-imidazol-4-yl]ethylcarbamothioylamino]urea (3R)-N-[1-[4-[[[5-(hydroxymethyl)furan-2-yl]methylamino]methyl]cyclohexyl]-6-phenylhexa-2,4-dien-3-yl]piperidine-3-carboxamide 3-[(1R)-1-[4-chloro-2-fluoro-5-[5-[(3,3,3-trifluoropropylamino)methyl]pyridin-3-yl]phenyl]ethoxy]cyclobutan-1-ol 2-(4-methylphenyl)sulfonyl-N-[(5S,7R)-7-nitro-6,9-dioxo-5-propan-2-ylidenedecoxy]acetamide N-benzyl-2-[1-(3,4-dimethoxyphenyl)-3-ethyl-5-oxo-4H-pyrazol-4-yl]-2-oxoacetamide 6-[(3S,4R)-1-benzyl-3-methoxypiperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidine 2-azido-5-(4,5-dimethyl-1H-imidazole-2-carbonyl)benzoic acid (2-aminopyridin-4-yl)-[1-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)pyrrolidin-3-yl]methanone;benzene N-[(3S)-8-chloro-1-oxoisoquinolin-3-yl]-6-(2,5-difluorophenyl)pyridine-3-carboxamide N-[3-amino-6-(2,4-difluorophenyl)pyridin-2-yl]methanesulfonamide 3-(4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidine-2-carbonyl)benzamide N-(4,4-dimethylpent-1-en-2-yl)-5-[3-[7-(5-fluorothiophen-2-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-indazol-5-yl]pyridin-3-amine N-[2-(3,4-dimethylphenyl)propan-2-yl]-5-fluoropyridine-3-carboxamide 2-fluoro-5,6-dimethylbenzenecarboximidate 5-methyl-4,10-dihydro-[1,2]thiazolo[3,4-b][3,1]benzoxazin-1-amine 4-[2-(2,5-dioxoimidazolidin-1-yl)ethyl]-N-hydroxypyridine-3-carboxamide 4-[(1R,2S)-1-amino-2-hydroxypropyl]benzonitrile 2-[2-fluoro-3-(methanesulfonamido)phenyl]acetamide [2-fluoro-4-methylsulfonyl-5-(trifluoromethoxy)phenyl]boronic acid N-[3,4-difluoro-5-(2-phenylpropoxy)phenyl]formamide 2,5-dioxopyrrolidine-1-carboxylic acid;2-[5-(3-phenoxyphenyl)-3-thiophen-2-ylpyrazol-1-yl]acetaldehyde 3-amino-N'-[2,4,6-trimethyl-4-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]pyridine-2-carboximidamide 4-[(2,3-dimethyl-1H-indol-7-yl)amino]piperidine-1-carboxylic acid N-[4-(2-hydroxy-3,5-dimethoxyphenyl)-6-methylpyrimidin-2-yl]cyclopropanecarboxamide 2-azidooxy-5-methylsulfonylpyridine N-(2,4-difluorophenyl)formamide;2-methyl-3-(1H-pyrrolo[2,3-b]pyridin-5-ylmethoxy)aniline 2-[6-fluoro-3-hydroxy-4-[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]indazole-1-carbonyl]-6-fluorobenzonitrile 1-(oxan-2-yloxy)isoquinoline N-[4-(trifluoromethoxy)phenyl]-3,4,5-tris(phenylmethoxy)benzamide 4-[4-methyl-3,6-dioxo-2-(phenylsulfanylmethyl)piperazin-1-yl]benzamide N-[2-amino-6-(3,5-dimethyl-1,2-oxazol-4-yl)pyridin-3-yl]-3-(trifluoromethoxy)benzamide 4-[3-(4-chlorophenyl)-1H-1,2,4-triazol-5-yl]-N-propan-2-ylaniline 2-(3-azidooxypropylsulfanyl)-1,3,4-trimethylbenzene 6-[(1R,2S)-2-hydroxycyclopentyl]oxy-5-[3-(trifluoromethyl)phenyl]isoquinoline-8-carbonitrile 3-hydroxy-2,2-bis(4-methylsulfanylphenyl)-1,8-naphthyridine-4-carboxylic acid 3-[2-[(4-ethylphenyl)methoxy]phenyl]-N-(thiophen-3-ylmethyl)propanamide N-(3,4-difluorophenyl)-2-hydroxy-6-oxopiperidine-1-carboxamide 2-bromo-N-hexyl-6-methoxy-4-nitro-N-prop-2-enylaniline 4-[N-(2-carboxyethyl)-3-nitroanilino]-2-hydroxybenzoic acid 2-[2-(3,4-dimethylphenoxy)ethylamino]-1-(6-fluoro-3,4-dihydro-1H-isoquinolin-2-yl)ethanone 2-methyl-3-[[4-(5-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]amino]propanoic acid 1-(6-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-propanoylpiperidine-4-carboxamide 1-cyclopentyl-6-[(1S,2R)-2-pyrimidin-2-ylcyclopropanecarbonyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one [2-amino-3-(1,2-dihydroindol-6-yl)propanoyl]oxidanium 2-methyl-N-[(1S,3R)-3-[[6-(oxan-4-ylamino)pyrimidine-4-carbonyl]amino]cyclohexyl]pyrimidine-5-carboxamide N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]-3-pyridin-2-ylsulfanylpropanamide 4-[2-(cyclopentylmethylamino)ethylamino]isoindole-1,3-dione;ethane 4-(6-fluoroquinoline-2-carbonyl)-5,5-dimethyl-1-pyridin-3-ylpyrrolidin-2-one 1-[4,5,5,8,8,11,14,17-octamethyl-6,7,12-tris(2-methylphenyl)-3,17-dioxa-19-azapentacyclo[12.8.0.02,10.04,9.015,20]docosa-1(21),2(10),4,6,8,13,15(20),18,20-decaen-3-yl]ethanone 5-[2-(diethylamino)-6-fluoropyridin-4-yl]-N',3,4-trimethoxypyridine-2-carboximidamide 2-amino-N-[(4-bromothiophen-2-yl)methylidene]-3-hydroxybutanamide 1-[4,5-diamino-6-(methoxymethyl)pyrimidin-2-yl]-3-[3-methyl-5-(3-methylphenyl)but-2-enyl]urea 2-chloro-N-(6,7-dimethoxyquinolin-4-yl)acetamide [6-(3,5-dimethyltriazol-4-yl)isoquinolin-3-yl]carbamic acid 2-amino-8-[3-[(4-chlorophenyl)methyl]-6,7-dihydro-4H-triazolo[1,5-a]pyrazin-5-yl]-N,N-dipropyl-3H-1-benzazepine-4-carboxamide;formic acid N-[2,4-bis(phenylmethoxy)phenyl]-2-cyclobutylacetamide 1-(4-chlorophenyl)sulfonyl-3,6-dihydro-2H-pyridine 3-(3,5-dichlorophenyl)-N'-hydroxyimidazo[1,2-a]pyridine-7-carboximidamide 6-methoxy-N-(3,4,5-trifluorophenyl)-7-(1H-pyrrolo[2,3-b]pyridin-5-yl)quinazolin-4-amine 3-[3-(4-chlorophenyl)sulfanylpyrazin-2-yl]sulfanyl-N,N-dimethylpropane-1-sulfonamide N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-oxo-6,7-dihydropyrazolo[1,5-a]pyrazine-5-carboxamide 1-(2-aminophenyl)-7,9-dimethoxycarbazole-3-thiol 1-[(3aR,6aS)-2-pyrimidin-2-yl-3a-(5-pyridin-4-yl-1H-1,2,4-triazol-3-yl)-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl]-2-phenylethanone 5-azidooxy-2-butylsulfanyl-6,7-dichloro-4-methoxyquinoline 1-[4-(2,5-dimethylcyclohexyl)oxyphenyl]pyrrolidine 3-[4-(aminomethyl)phenyl]-N-methoxycyclohexan-1-imine 6-chloro-2,9a-dimethyl-8H-[1,3]dioxolo[4,5-g]isoquinolin-10-one N-[5-(2-methylbutanoylamino)pyridin-2-yl]sulfonyl-6-[4-(trifluoromethoxy)phenoxy]naphthalene-1-carboxamide 2-(5-ethyl-1H-pyrazol-3-yl)-6-[[1-[4-[5-(trifluoromethyl)pyridin-2-yl]oxybutanoyl]piperidin-4-ylidene]amino]pyrimidine-4-carbonitrile 2-[[5-(4-chlorophenyl)furan-2-yl]methylideneamino]-N,N,1-triethylpyrrolidine-3-carboxamide 2-[azido(phenylmethoxy)methyl]oxirane N-(2,4-dichloropyrimidin-5-yl)-N-(1-phenylethyl)nonanamide 4-[3-(4-bromophenyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-[1,3-difluoro-6-(5-heptylpyridin-2-yl)naphthalen-2-yl]propan-2-ol 1-methyl-3,5-bis(phenylmethoxy)piperidine 2-[(5Z)-5-[(4,7-dimethylquinazolin-6-yl)hydrazinylidene]-3-methoxy-1-propan-2-ylpyrazol-4-ylidene]propanenitrile 2-[4-[3-methylbut-1-en-2-yl(pyridin-3-yl)amino]pyrazol-1-yl]ethanol 4-[2-(6-ethylsulfonylpyridin-3-yl)sulfanyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]naphthalen-1-ol N-[4-(5-azidopentoxy)phenyl]-4-chlorobenzamide N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1-methyl-2-oxo-5-thiophen-2-ylpyridine-3-carboxamide N-[(4-fluorophenyl)methyl]-2-pyridin-3-yloxyquinolin-8-amine 3-[[3,4-bis(ethenyl)phenyl]sulfonylamino]propanamide;5-fluoro-2-pyridin-2-ylpyrimidine 5-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-octylamino]naphthalene-2-sulfonic acid 4-tert-butyl-1-(2,3-dihydro-1H-tetrazol-5-ylmethyl)piperidine 5-fluoro-2-methyl-N-[1-[2-(3,4,5-trimethoxyphenyl)acetyl]piperidin-4-yl]benzamide 2-fluoro-4,5-dimethoxy-N-(2-oxoazepan-3-yl)benzamide 1-[3-[(2R)-6,15-dibromo-13-chloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl]piperidin-1-yl]-3,3-bis(methylamino)propan-1-one 1-(2,3-dihydro-1H-inden-5-yl)sulfonyl-4-[(4S)-4-fluoropyrrolidin-3-yl]piperazine 3-[1-azido-2-(4-chlorophenyl)ethyl]-5,6,7,8-tetrahydrocinnoline [5-[6-(dimethylamino)pyridin-2-yl]pyridine-3-carbonyl]chloranium 4-methyl-2-[5-(1,3-thiazol-2-yl)-4-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-2-yl]pentanamide N-(3,4-dimethoxyphenyl)-1-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-6-yl)cyclopentane-1-carboxamide N-(1-bromo-6,7-dihydrobenzo[d][1]benzazepin-11-ylidene)hydroxylamine N-[5-[4-(4-propan-2-ylpiperazine-1-carbonyl)phenyl]pyridin-3-yl]carbamate 3-[N-methylsulfonyl-4-(pyridin-2-ylsulfamoyl)anilino]propanoic acid (7R)-5-methyl-N-naphthalen-1-yl-2-pyridin-3-yl-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide [4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-[(5R,7S)-2,5,7-trimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazol-3-yl]methanone N'-amino-4-[2,6-dimethyl-5-(trifluoromethyl)pyrimidin-4-yl]piperazine-1-carboximidamide 3-[2,6-di(propan-2-yl)phenyl]-1-methoxybutan-2-one 5-ethyl-4,6-difluoronaphthalene-2-carboxamide 1-methyl-3-[4-(1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl]urea (3Z,5E)-N-[3-[7-(4-fluorophenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-2H-pyrazolo[3,4-b]pyridin-5-yl]hepta-1,3,5-trien-2-amine 4-[6-(6-chloro-7-fluoroimidazo[1,2-a]pyridin-3-yl)pyrimidin-4-yl]morpholine 2-hydroxy-5-methylbenzenesulfonate 2-(cyclopropylamino)-5,8-dimethylnaphthalene-1,4-dione N-[3-[(Z)-aminomethylideneamino]oxypropyl]-1,2,4-triazol-4-amine 3-[(4-azidophenyl)methyl]pyrimidin-2-one 4-(4-chlorophenyl)-2,5-dimethylpyridine;ethane 6-(dimethylamino)-3-methyl-1,4-benzothiazin-2-one 2-[(3S,4R)-4-[(5-chloropyrimidin-2-yl)amino]-1-methylsulfonylpyrrolidin-3-yl]-N,N-dimethylacetamide 1-[(1R)-3-(4-phenylphenyl)cyclopentyl]propan-2-one 2-[(2E,5S)-4-oxo-2-[(Z)-1H-pyrrol-2-ylmethylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 3-[1-(4-bromophenyl)triazol-4-yl]propanoic acid (2R)-2-(5,7-dihydroxynaphthalene-1-carbonyl)oxy-4-methylpentanoate 4-[(5R)-6-[3-chloro-2,6-difluoro-5-(trifluoromethyl)phenyl]-3-oxo-4,5-bis(prop-1-enyl)-4H-pyridazin-1-yl]benzaldehyde (5E)-1-prop-2-enyl-4,6,9-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-3,5,7,10,12,14,17-heptaene 2-[4-chlorobutyl(ethenoxysulfonyl)amino]benzenesulfonic acid (2-butylphenyl)-(2-cyclohexylimino-5,6,7,8-tetrahydro-1H-quinolin-3-yl)methanone (5Z)-5-[[3,4-difluoro-2-[[1,3]thiazol-2-yl(methyl)amino]phenyl]methylidene]imidazolidine-2,4-dione 1-[(2,4,6-trimethylphenyl)sulfonylamino]propane-2-sulfonic acid 7-chlorospiro[3,4-dihydropyrano[2,3-b]pyridine-6,1'-cyclohexane] N-[4-(6,11-dihydropyrrolo[2,1-c][1,4]benzodiazepine-5-carbonyl)phenyl]-3,5-dimethylbenzamide (6-chlorocyclohexa-1,5-dien-1-yl)-[4-[2-hydroxyethyl(methylsulfonyl)amino]naphthalen-1-yl]azanium 2-[1-(furan-2-ylmethylamino)propan-2-ylideneamino]acetaldehyde 5-(2,4-dichlorophenoxy)-3-[(4R)-6-fluoro-1,2,3,4-tetrahydronaphthalene-2-carbonyl]pyrimidin-4-one 2-(3,4-dihydroxyphenyl)-5-hydroxycyclohexa-1,3-diene-1,4-dicarboxylic acid N-[1,2-diamino-3-(4-fluorophenyl)propan-2-yl]-1-methylcyclohexane-1-carboxamide 6-chloro-3-[(4-chlorophenyl)methyl]-2H-1,3-benzoxazin-4-one 3-(1H-benzimidazol-2-yl)-N,N'-dimethyl-N-prop-2-ynylpropanimidamide 5-amino-1,3-dimethylpyrazole-4-carboxamide;N-[2-cyclohexyl-2-(2H-tetrazol-5-yl)ethyl]formamide 2-(3,5-dichlorophenyl)-N-[1-(3-oxoazepane-4-carbonyl)azetidin-3-yl]acetamide (3E)-6,7-dimethylocta-1,3,5-triene;3-(1,1,1-trifluoropentan-2-yloxy)benzaldehyde 3-(azepin-1-yl)pyridine-2,6-diamine 3-(2,4-dihydroxyphenyl)-N,1,2-trimethylpyrazole-4-carboxamide 3-(7-hydroxy-1H-benzimidazol-2-yl)-5-[(4R,6S)-8,9,10,11-tetrahydroindolo[2,3-a]quinolizin-6-yl]pyridine-4-carboxylic acid 2-[4,5-dichloro-1-ethyl-3-(methoxymethyl)pyrazol-4-yl]-7H-purine 2-amino-N'-[3,4-difluoro-5-(trifluoromethyl)phenyl]benzenecarboximidamide (5S,7R)-N-[(4-methylsulfonylphenyl)methyl]-1,3,4,5,6,7,8,9,10,11-decahydropyrazolo[3,4-b][1,2,5]triazecine-5-carboxamide (2R)-4-[2,6-dichloro-3-[(2,2-dimethylpropanoylamino)methyl]phenoxy]-N-hydroxybutanamide N-[2,4-difluoro-3-(3-methylbutanoylamino)phenyl]-1H-pyrrole-3-sulfonamide N-(4-carbamoylphenyl)-4,6-dichlorohexanamide (2Z)-2-(3,5-dimethyl-1H-pyrrol-2-yl)-N-[1-(3,4-dihydro-2H-quinolin-1-yl)ethenyl]-5-fluoropenta-2,4-dien-1-amine 2-azido-6-[5-(3,4-dihydropyridin-5-yl)pyridin-1-ium-2-yl]pyridine 2-[(2R)-1,1-bis(4-fluorophenyl)-1,3-dihydroxypropan-2-yl]cyclohexan-1-one (2R)-6-[4-chloro-3-(2,6-difluorophenyl)quinolin-7-yl]oxy-1,2-oxazolidine-2-carboxylic acid (E)-N'-[amino-[1-[4-[3-[4-(dimethylamino)butyl]piperazine-1-carbonyl]phenyl]-2,6-naphthyridin-7-yl]amino]hex-2-enediamide (3R)-4'-chlorospiro[1H-indole-3,5'-oxane]-2-one 2-(5-methoxycyclohepta-1,3,6-trien-1-yl)-N-[[4-(1-pyridin-2-ylethylamino)phenyl]methyl]acetamide 6-[1-(4-methoxyphenyl)-3-methylpyrazole-4-carbonyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 5-[(4-ethoxycarbonylphenyl)methyl]-6-propan-2-ylpyridine-3-carboxylate 2-[4,7-dimethyl-3-(5-methylthiophen-2-yl)-8,10b-dihydropyrazolo[1,5-d][1,4]benzoxazepin-6-yl]acetate N-[(2,4-dimethoxyphenyl)methyl]-1-[[5-(1H-indole-3-carbonyl)pyridin-2-yl]amino]-2,2-dimethylcyclopentane-1-carboxamide 2-[1-(5-azidopyridin-2-yl)pyrrolidin-3-yl]ethanamine N-[2-(4,5-dihydro-1H-imidazol-2-yl)ethyl]-3-nitroaniline (5-butoxypyridine-2-carbonyl)oxidanium 2-(3-chlorophenoxy)-N'-hydroxypyridine-4-carboximidamide 1-benzylsulfonyl-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-ylmethyl)pyrrolidine-2-carboxamide 1-[3-(4,6-dimethylpyrimidin-2-yl)sulfanylpropyl]-7H-purine-2,6-dione (3S)-N-(1H-indol-4-ylmethyl)-6-methoxy-2,3-dihydro-1-benzofuran-3-carboxamide 1,3-dimethyl-6-[(6S)-3-methylidene-6-propan-2-ylidenecyclohexen-1-yl]naphthalene 2-[(E)-3,5-bis(hydroxymethyl)hex-1-enyl]-7-methoxychromen-4-one 3-(6,7-dihydrocyclohepta[d]pyrimidin-4-ylamino)butanamide 2-hydroxy-5-[2,3,6-trimethyl-4-(oxolan-2-ylmethoxy)phenyl]sulfanylcyclohepta-2,4,6-trien-1-one 4-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenyl]-6,7-dihydroquinoline 3-[1-[4-(2-cyclopentylpropan-2-yl)phenyl]sulfanylpyrrolidin-2-yl]-5,6-dihydro-1H-benzimidazole 1-(5,6-dimethoxypyridin-3-yl)-N-[6-fluoro-5-(2H-pyrazin-1-ylmethyl)pyridin-2-yl]pyrazolo[4,3-c]pyridine-3-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]-5-(2H-tetrazol-5-yl)pentanamide 5-(4-methoxyphenyl)-N,1-dimethyl-3,6-dihydro-2H-pyridine-3-carboxamide 2-(2,3-dihydrothieno[3,4-b][1]benzofuran-6-yl)acetamide 5-(4-chlorophenyl)-N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]-1H-pyrrole-3-carboxamide (2R)-2-[3,5-bis(trifluoromethyl)phenyl]-3-[3-chloro-6-(1H-pyrrolo[2,3-b]pyridin-4-yl)indazol-1-yl]propanamide 4-bromo-5-ethyl-3,7-dimethoxynaphthalene-2,6-diol 3-(4-ethylphenyl)-1,5-dihydrochromeno[2,3-d]imidazole 3-[5-(1H-indol-2-yl)-4-methoxy-1,2-oxazol-3-yl]phenol 5-bromo-4-[3-methylbutyl(propan-2-yl)amino]-1H-pyrimidin-6-one 2,5-diiodo-3-(methylideneamino)aniline [(3aR,7aS)-1-(4-fluorophenyl)-2,2-dimethyl-3,3a,5,6,7,7a-hexahydropyrrolo[3,2-b]pyridin-4-yl]-(4-chloropyridazin-3-yl)methanone 3-ethyl-4,5-dimethoxy-N-(3-phenylprop-1-en-2-yl)aniline 4-amino-2-methyl-5-[3-(trifluoromethoxy)phenyl]thiophene-3-carbonitrile 6-[(3-chlorobenzoyl)amino]-2-[4-(trifluoromethoxy)anilino]quinoline-4-carboxylic acid;dihydrochloride 3-[3-(3,4,5-trimethoxyphenyl)prop-1-enyl]-2H-furan 1-butoxysulfanyl-4,5-dichloro-3-(4-phenoxyphenyl)sulfinylbenzene 3-(benzylideneamino)-6,7-diethyl-2-methylchromen-4-one N-(1,4-dihydropyrimidin-2-ylmethylidene)-3-ethoxybenzenesulfonamide 4-(2-fluorophenyl)-6,7-dihydropyrazolo[1,5-a]pyridine N-[2,4-difluoro-3-(6H-pyrrolo[1,2-a]pyrimidin-7-ylsulfonyl)phenyl]methanesulfonamide N-(4-cyano-3-fluorophenyl)-N-[2-hydroxy-2-(5-thiophen-2-ylfuran-2-yl)ethyl]-1H-pyrrole-2-carboxamide N-[(4,5-dimethyl-1H-pyrazol-3-yl)methyl]-5-hydroxypyrrolidine-2-carboxamide 2-[3-[4,5-dimethoxy-6-(methylsulfanylamino)pyrimidin-2-yl]phenyl]-1,3-thiazole-5-carbonitrile 1-(4-fluorophenyl)-N-[6-methyl-5-[3-(7-pyridin-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]methanimine (3Z)-7-cyclopropyl-4,8-dimethyl-1,2-bis[4-(trifluoromethyl)phenyl]-6H-benzo[f]benzimidazole (2S)-1-[4-cyano-3-(trifluoromethyl)phenyl]-N,N-dimethylpyrrolidine-2-carboxamide N-(5-bromothiophen-2-yl)sulfonylacetamide 4-azidooxy-5-(2,2,3,3-tetrafluoropropyl)pyrimidine 1-(2,2-dimethylcyclobutyl)-N-[4-[5-[4-fluoro-3-(trifluoromethoxy)phenyl]-7-sulfanylidene-6H-pyrazolo[1,5-a]pyrimidin-3-yl]pyridin-2-yl]methanesulfinamide (6R,7S)-3-[(4-fluorophenyl)carbamoylamino]-8-oxo-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 2-[(3R)-1,6-dimethylpiperidin-3-yl]-5-methoxy-8-(4-methylcyclohexa-1,5-dien-1-yl)sulfanyl-3H-quinazolin-4-one (5-chloropyridin-3-yl)-[2-[1-[4-ethyl-6-(1-methylpyrazol-4-yl)pyridine-2-carbonyl]pyrrolidin-3-yl]oxyphenyl]methanone 2,4-bis(methoxycarbonyl)-3-[4-(trifluoromethyl)phenyl]sulfanylbenzoate 2-fluoro-N,6-dimethyl-4-(1H-pyrrolo[2,3-b]pyridin-5-yl)aniline;propane 1-amino-4-methylsulfanylbenzene;N,2,5-triphenylbenzenesulfinamide 2-bromo-6-phenylpyrazolo[1,5-a]pyrimidine 2-(4-azidopyridin-3-yl)-1,3-thiazole 2,4-ditert-butyl-6-[(3-ethoxyphenyl)iminomethyl]phenol 2-azido-5-methoxy-1,3,4-thiadiazole N-(3,5-dichlorophenyl)-2-[3-(4-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]propanamide 5-[7-fluoro-3-(4-thiophen-2-yl-1H-imidazo[4,5-c]pyridin-2-yl)-2H-indazol-5-yl]pyridin-3-amine 1-[6-(azetidine-3-carbonyl)pyridin-2-yl]-N,N-dimethylpyrrolidine-2-carboxamide 1-[2-chloro-6-(trifluoromethyl)phenyl]ethylideneazanide 5-[[2,4,6-trimethyl-N-(pyridin-3-ylcarbamoyl)anilino]diazenyl]naphthalene-1,7-disulfonic acid 1-benzyl-5-ethenoxypyridin-2-one 4-[(5-acetylcyclohexen-1-yl)methoxy]benzaldehyde N'-[3-ethyl-4-(trifluoromethoxy)phenyl]oxamide 2-(cyclopropylmethoxy)-4,7-dimethylpyrrolo[2,3-d]pyrimidine 4-[[2-(2,3-dihydro-1H-inden-5-yl)ethylamino]methyl]-6-phenylpyridine-2-carbonitrile 4-[(6-chloropyridine-3-carbonyl)amino]benzenesulfonic acid 3-fluoro-4-[6-methylsulfonyl-2,3,3a,4,5,9b-hexahydropyrido[3,4-b]indole-1-carbonyl]benzoic acid 4-bromo-3-cyanobenzoate 1-azido-4-butan-2-yloxy-3,5-dimethoxy-N-propan-2-yloxybenzenesulfonamide 5-chloro-2,6-dimethoxybenzene-1,3-dicarboxylic acid 2-(5-azidopentoxy)quinoline 2-(3,5-dichlorophenyl)-N-[4-[[2-[2-hydroxyethyl(methylsulfonyl)amino]pyridin-4-yl]oxymethyl]-1,3-thiazol-2-yl]acetamide 6-cyclobutyl-3H-thieno[2,3-d]pyrimidine-4-thione N-ethyl-3,4,7-trimethylphenanthrene-1-carboxamide (3,5-dimethylpyrazol-1-yl)-[4-[2-fluoro-6-methoxy-4-(trifluoromethyl)phenyl]piperazin-1-yl]methanone 2-[5-amino-1-[2-(difluoromethyl)phenyl]pyrazole-3-carbonyl]-3,4-dihydro-1H-isoquinoline-7-carboxylic acid 3-[(2,6-dimethoxyphenyl)methyl]-1-[3-(4-methylpiperazin-1-yl)propanoylamino]piperidine-3-carboxamide 1-(3,5-dichlorophenyl)-N-[4-[6-(3,3-dimethylbut-1-en-2-ylamino)pyridin-3-yl]phenyl]cyclopropane-1-carboxamide (E)-3-[3-[4-(4-chlorophenyl)-5-oxo-1H-1,2,4-triazol-3-yl]-4-ethoxyphenyl]prop-2-enoic acid 2-[4-(oxan-4-yloxy)phenyl]prop-2-enamide 2-[(2,5-dichlorophenyl)sulfanylmethylidene]propanedioic acid 2-[(2,6-dimethylphenoxy)methyl]-3H-pyrido[2,3-d]pyrimidin-4-one N-[4-(aminomethyl)cyclohexyl]pyridine-2,5-diamine N-[4-chloro-2-(trifluoromethyl)phenyl]-3,6-dioxocyclohexene-1-carboxamide N-[1,3-benzodioxol-5-yl-(4-methoxyphenyl)methylidene]hydroxylamine 3-(2-chlorophenyl)-N-[5,7-dimethoxy-2-oxo-1-[4-(trifluoromethyl)phenyl]quinolin-6-yl]propanamide N-[3-(azetidin-1-yl)butan-2-ylidene]-4-phenylmethoxypiperidine-1-carboximidamide N-[3,5-bis(trifluoromethyl)phenyl]-1,2-dihydropyridine-4-carboxamide 5-[3-fluoro-2,6-di(propan-2-yl)phenyl]-4-hydroxypiperidine-2,6-dione 4-[4-(4-ethenylphenyl)butoxy]benzoate 4-amino-3,5,6-trichlorophthalic acid 3-[(6S)-2,6-dimethylmorpholine-4-carbonyl]-N'-hydroxy-5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboximidamide N-[2-(5-methoxy-1H-indol-3-yl)ethyl]acetamide 2-(5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)-6-piperidin-4-ylpyrimidin-4-amine;fluoromethane 1,3-bis[2,6-di(propan-2-yl)phenyl]-4-[(Z)-prop-1-enoxy]imidazol-1-ium;dibromomethane 2-N,5-N-bis(3-aminophenyl)pyridine-2,4,5-triamine N-methyl-2-(1-oxo-3,4,5,6,7,8a,9b-hexahydroindeno[2,1-c]pyridine-2-carbonyl)benzamide 1-(cyclopentylmethyl)-4-ethoxybenzene;1-[4-fluoro-2-(trifluoromethyl)phenyl]butan-2-one 5-[(3S,5R)-3,5-dimethylpiperazine-1-carbonyl]-N-[4-fluoro-2-(trifluoromethoxy)phenyl]pyridine-2-carboxamide (1-hydroxycyclobutyl)-[4-methoxy-3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methanone 3,4-dichloro-N-[1-(2-chloroethyl)cyclopropyl]aniline 1,5-dihydro-[1,3]thiazolo[5,4-c]isoquinoline-2,3-dithione 2-[2,6-difluoro-4-(triazol-1-ylmethyl)phenyl]-N,1-diethylbenzimidazole-5-carboxamide 4-tert-butyl-N'-[(Z)-[2,6-dichloro-5-(trifluoromethoxy)phenyl]methylideneamino]benzenecarboximidamide 1-[2,5-difluoro-4-(1H-pyrrolo[3,2-c]pyridine-2-carbonyl)phenyl]ethanone 1-ethenyl-3,5-difluorobenzene;N'-[(2Z)-hepta-2,6-dien-2-yl]-4-methylbenzenecarboximidamide N-(cyclohexylmethyl)-2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxyethanamine;6-(difluoromethoxy)-1H-indole-3-sulfonamide 2-[4-(3,3a,4,5,6,7a-hexahydro-1H-pyrrolo[3,4-c]pyridine-2-carbonyl)piperazin-1-yl]-N-methylpyrimidine-5-carboxamide;2,2,2-trifluoroacetic acid 3-[4-amino-7-methyl-6-oxo-2-(2,2,2-trifluoroethyl)sulfanylpyrido[2,3-d]pyrimidin-8-yl]benzonitrile 2-[(3-methylphenyl)methoxy]cyclohepta-1,3-diene N-[1-[3-[(4-fluorophenyl)methyl]triazolo[4,5-d]pyrimidin-5-yl]piperidin-4-yl]-1H-indole-2-carboxamide 2-[8-(2,6-dimethylphenyl)-1-methoxyisoquinolin-3-yl]benzimidazole-5-carboxamide 3-azido-6-bromonaphthalene-1,2-dione N-methyl-1'-[3-(trifluoromethoxy)benzoyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide N-[6-[5-fluoro-4-(trideuteriomethoxy)pyridin-2-yl]pyridazin-3-yl]-1-(methylamino)cyclopropane-1-carboxamide N-[1-(4-tert-butylphenyl)ethylideneamino]pyrimidin-2-amine 5-chloro-3,4-dihydroisoquinoline;N-[2-(2-chlorophenyl)ethyl]-6-pyrrolidin-1-ylpyrimidin-4-amine 2,5-dichloro-N-(4-methoxyphenyl)sulfanyl-3H-thieno[3,2-d]pyrimidin-4-imine 2-amino-4-(2,6-difluoro-4-methoxyphenyl)-6-ethoxy-4H-pyran-3,5-dicarbonitrile 4-methyl-1-[(2-pyrrolidin-1-ylpyrimidin-5-yl)methyl]piperidine-4-carboxylate 3-[4-(methoxymethyl)cyclohexyl]-1-methyl-6-pyrimidin-2-ylquinazoline-2,4-dione 6-(3-chloropropoxy)-N'-hydroxypyridine-2-carboximidamide 4-[2-chloro-3,5-di(propanoyl)phenyl]pyridine-2-carboxylic acid 2-cyclopropyl-4-(4-phenoxybutoxy)benzaldehyde 2-(N-(4-phenyl-1,3-thiazol-2-yl)anilino)propanoic acid 2-bromo-4-[(3S)-5,7-dimethoxy-1-phenyl-2,3-dihydroindene-1-carbonyl]phenol 3-[[1-cyclopropylsulfonyl-2-(oxan-4-yl)pyrrole-3-carbonyl]amino]pyridine-2-carboxylic acid [6-[(5R)-3,4-dihydroxy-5-methoxycarbonyl-2-methylphenyl]-9H-xanthene-3-carbonyl]azanium 1-[2,6-di(propan-2-yl)phenyl]-3-[5-(2-morpholin-4-ylethoxymethyl)pyridin-2-yl]sulfonylurea 6-[5-(4,5-dihydrothieno[3,2-d][1]benzazepine-2-carbonyl)cyclooctyl]-1,3-benzothiazol-2-amine (4S)-2,2-difluoro-N'-methanimidoyl-3,4-dihydrochromene-4-carboximidamide 6-(5-chloro-2-methoxypyridin-3-yl)-N,1-dipropylpyrrolo[3,2-c]pyridine-4-carboxamide 2-[4-(3,5-difluorophenyl)-6-(trifluoromethyl)pyridin-3-yl]acetamide N-methoxy-4-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]benzamide (3E,4Z)-5-[4-[3-(2-ethoxyethylamino)propyl]phenyl]-6-fluoro-2-methylidenehepta-3,5-dienal;propanoic acid 2-azidooxy-N-(3,4-dichlorophenyl)propanamide N-[5-[1-methyl-4-[(1-methylsulfonylcyclopropyl)amino]pyrido[3,2-d]pyrimidin-6-yl]pyridin-3-yl]methanesulfonamide (2S)-2-[(3,4-dimethoxyphenyl)sulfonylamino]-3-[5-ethenyl-1-ethyl-6-oxo-2-(3,3,3-trifluoropropyl)pyrimidin-4-yl]propanoic acid 4-[[2,6-difluoro-3-(5-fluoro-4-hydroxy-1H-benzimidazole-2-carbonyl)phenyl]methyl]piperazin-2-one N-[1-(3,4-dimethoxybenzoyl)piperidin-2-yl]prop-2-enamide 3-(2,4-dimethylphenyl)-N'-methylsulfonylpropanehydrazide 2-(5-bromopyridine-3-carbonyl)-4,4,7-trifluoro-N,N-dimethylheptanamide 1,3-dichlorobutane;N-[1-(methylamino)propan-2-ylidene]benzamide (2E,4Z)-5-amino-2-[[amino-(3-methoxyphenyl)methylidene]carbamoyl]penta-2,4-dienoic acid N-butyl-2-methoxy-N-(2H-tetrazol-5-yl)acetamide (5R)-2-[(2S,7S)-9-oxononanoyl]sulfanyl-3,4-dihydro-1H-isoquinoline-6-carboxylic acid N-[5-(4-methoxyphenyl)-1,2-dihydro-1,3-benzothiazol-6-yl]acetamide N-[4-(dimethylamino)-6,7,8,9-tetrahydropyrimido[5,4-b]indolizin-10-yl]cyclohexanecarboxamide (5-methylpyrazine-2-carbonyl)-[4-[4-(trifluoromethoxy)phenyl]piperazin-1-yl]azanium 6-[4-(2-methylpropylamino)phenyl]cyclohexa-1,5-diene-3-sulfonic acid 6-[3-[4-(aziridin-2-yl)-5-chlorothiophen-2-yl]phenyl]-1,1,1-trifluorohexan-2-one 4-[5-[(2,6-dichlorobenzoyl)amino]pyridin-3-yl]-N-(4-fluorophenyl)piperazine-1-carboxamide N-[2-(4-ethylphenyl)ethyl]-1,3,5-trimethylpyrazole-4-carboxamide [2-(5,6-dimethylpyridin-3-yl)-1,3-thiazol-4-yl]-(4-methylpiperazin-1-yl)methanone 2-azido-N,N-dimethyl-6-nitroaniline N-[3-(7-methoxy-1,4a-dimethyl-2,3,4,9-tetrahydroindeno[2,1-b]pyridin-5-yl)propyl]acetamide 4-[(1R)-2-aminocyclopentyl]benzenesulfonamide;hydrochloride 4-cyclohexyloxy-6-[(2,3,5-trifluorophenyl)methyl]pyrimidine [[2-(4-ethylsulfonylphenyl)acetyl]amino]thiourea 1-(3-methyl-4,5,6,7-tetrahydrobenzotriazol-5-yl)-3-(3,3,5,5,8,8-hexadeuterio-2,8-diazaspiro[3.5]nonan-2-yl)propan-1-one 1-amino-N-[(E)-(2,4-dimethoxyphenyl)methylideneamino]-2H-pyridine-3-carboxamide 4-hydroxy-6-(3,5,8-trimethyl-7,8-dihydronaphthalene-2-carbonyl)oxybenzoic acid 3-hydroxy-1,4-dihydroisoquinoline-2-sulfonamide 5-(1,3-benzothiazol-2-yl)-6-chloro-N-[4-methoxy-3-methyl-5-(trifluoromethyl)phenyl]pyridine-3-carboxamide 2-cyclopropyl-1'-(pyridine-3-carbonyl)spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,4'-piperidine]-4-one N-[6-cyano-2,5-bis(ethenyl)pyridin-3-yl]-4-methoxybenzenesulfonamide 3-[4-[2,5-bis(4-aminophenoxy)phenyl]sulfonylphenoxy]aniline 1-(7-fluoronaphthalen-2-yl)sulfonyl-4-[2-methoxy-4-[5-(trifluoromethyl)pyridin-3-yl]phenyl]piperazine (4S)-6,8-dibromo-7-chloro-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepine N-[3-amino-5-(4-hydroxyphenyl)pyrazin-2-yl]thiophene-2-carboxamide;ethane 2-[(1S)-1,3-diphenylpropyl]-1,4-bis[2-(trifluoromethoxy)ethyl]piperazine N-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]formamide;4-(methoxymethyl)-N-methylpyridine-2-carboxamide 3,4-dihydro-1H-isoquinolin-2-yl-[5-(4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-5-carbonyl)thiophen-3-yl]methanone 5-(azidomethyl)-4,6-difluorobenzene-1,3-disulfonic acid 4-(3,5-diethoxyphenyl)cyclohexan-1-amine (5E)-2-cyclopentylimino-5-[(7,8-dimethoxy-4H-1,3-benzothiazin-2-yl)methylidene]-1,3-thiazolidin-4-one 2-(7,8-dihydronaphthalene-2-carbonyl)benzoic acid 3-[2-(2,6-dimethylmorpholine-4-carbonyl)anilino]-1-[(2R,5S)-5-fluoropyrrolidin-2-yl]pyrazole-4-carboxamide;hydrochloride 5-chloro-4-(3,6,7-trifluoro-2H-chromen-2-yl)benzene-1,2-diol 2-hydroxy-3,3-dimethylbutane;N-methylidene-4-[4-[(E)-pent-1-enyl]phenoxy]benzamide 1-[3-[[5-(3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl)-1,3,4-oxadiazol-2-yl]amino]phenyl]pyrrolidin-2-one 2-[3,5-dimethyl-1-(4-oxo-6,7-dihydro-3H-pyrrolo[3,2-d]pyrimidin-2-yl)pyrazol-4-yl]-N-[(4-methoxyphenyl)methyl]acetamide 2-amino-3,5-difluorobenzenesulfonic acid;ethane 1-[(2R)-3,3-difluorocyclopentyl]-6-[4-[5-(dimethylamino)pyrazine-2-carbonyl]phenyl]-4-(triazol-1-ylmethyl)pyridin-2-one 2-[1,3-dioxol-4-yl(ethyl)amino]benzoic acid 2-N,6-N-bis(4-butoxyphenyl)-9H-fluorene-1,2,6-triamine 1-(3,4-dihydro-2H-chromen-5-ylmethyl)azetidine;ethane 5-[4,6-bis(2-methylpropyl)-1H-triazin-2-yl]-N'-hydroxypyrazine-2-carboximidamide 2-[(1S)-1-[[6-oxo-4-(trifluoromethyl)-1H-pyrimidin-5-yl]oxy]ethyl]pyridine-3-carbonitrile 1-[(3S,4R)-4-hydroxy-1-[5-(2-methoxypyridin-3-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl]pyrrolidin-2-one 2-[(3S,4R)-3-[3-[(2-fluoro-6-propan-2-ylphenyl)carbamoylamino]phenoxy]-4-hydroxypiperidin-1-yl]acetic acid 3-bromo-6-methyl-N-(3-morpholin-4-ylpropyl)thieno[2,3-b]pyridine-2-carboxamide 2-[(5S,10bS)-7-methoxy-5-thiophen-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-chlorophenol 1-cyclopentyl-5,6-diethylbenzimidazole 3-cyclopentyl-2,5-dihydroxynaphthalene-1,4-disulfonic acid 7-hydroxy-5,6-diphenyl-3H-[1,3]oxazolo[4,3-b]quinoline [4-hydroxy-3-(5-methyl-1H-pyrazole-3-carbonyl)phenyl]urea [1-methyl-6-oxo-5-(pyridin-2-yldiazenyl)pyrimidin-4-ylidene]cyanamide (1R,2S)-3-azido-5-[[4-fluoro-6-(1H-indol-2-ylmethoxy)-7-methoxyquinazolin-8-yl]methylamino]cyclopentane-1,2-diol 1-(3,5-dichlorophenyl)sulfonyl-4-[(2-methyltetrazol-5-yl)methoxy]indole 4-methyl-3-[(Z)-6-oxooct-5-enoxy]-N-[4-[4-(5H-[1,2,4]triazolo[3,4-a]quinazolin-8-ylamino)butoxy]phenyl]benzamide [(2R)-1-(5,6-dichloropyridine-3-carbonyl)piperidin-2-yl]carbamic acid 2-(1,3-benzoxazol-2-yl)-N-[2-[(6S)-5-oxo-4,6-dihydroimidazo[1,2-b][1,2,4]triazol-6-yl]phenyl]cyclopropane-1-carboxamide N-[4-[[2-(benzylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino]cyclohexyl]acetamide 6-[4,5-bis(ethenyl)thiophen-2-yl]-8H-furo[3,2-c]azepine (3-methylpiperidin-1-yl)-[5-phenyl-7-(trifluoromethoxy)pyrazolo[1,5-a]pyrimidin-2-yl]methanone (E)-1-[4-chloro-3-(1,2,5-triazin-2-yloxymethyl)phenyl]-N-ethoxy-1-(1H-imidazol-5-yl)methanimine 1-[3-(2,6-dimethylpyridin-4-yl)phenyl]-4-methoxybutan-1-one 4-N,8-diamino-4-N-benzylnaphthalene-1,4-dicarboxamide N'-[(Z)-2,3,3a,4-tetrahydro-1H-indol-5-ylmethylideneamino]-N-[(3-chlorophenyl)methyl]oxamide 1-[2,6-di(propan-2-yl)phenyl]butane-1,3-diamine 7-(1,3-benzothiazol-2-yl)-4-hydroxy-6-methyl-5-nitroso-3H-pyrrolo[2,3-f]benzimidazol-1-ium-8-carboxylic acid 4-azidosulfanyl-2,3-dimethylaniline 3-(4-azidophenyl)-2-chlorothiophene (4S,7R)-3-methyl-4-(3-propoxyphenyl)-2,4,5,7-tetrahydropyrazolo[3,4-b]pyridin-6-one N-cyclohexyl-3-phenylmethoxybenzamide;4-(2,5-difluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine 2-[1-(2-azidoethyl)pyrazol-3-yl]pyridine [(2R,3S)-3-methyl-2-phenylheptanoyl]azanium N-[5-chloro-2-(5-cyanothiophen-3-yl)phenyl]sulfanyl-N',2-dimethylpropane-1,3-diamine 6-chloro-2,3,4-trideuterio-N'-ethylbenzohydrazide N-(2-cyanobutanoyl)naphthalene-1-carboxamide;toluene 6-(1H-indazol-5-yl)quinoxaline 4-(2,5-dihydroxypyrrol-1-yl)benzaldehyde 5-[2,6-bis(methoxymethyl)phenyl]-2-propan-2-ylidene-1H-naphthalene 2-(2,6-dichlorophenyl)imino-5-(quinolin-8-ylmethylidene)-1,3-thiazolidin-4-one 1-methylsulfonylpyrrolo[3,2-b]pyridine-6-carboxamide 2-(5,6-dichloropyridin-3-yl)sulfonyl-7a-methyl-1-[4-(trifluoromethoxy)phenyl]-5,6,7,7a-tetrahydropyrrolo[1,2-c]imidazole-3a,4,7-trione 1-[3,3-difluoro-2-hydroxy-4-(trifluoromethyl)piperidin-1-yl]-6-methoxy-7-pyrrolidin-1-yl-4H-quinoline-2-carboxylic acid 3,5-dichloro-4-(4-methylsulfonylphenoxy)pyridine 2-amino-4-[1-(3,4-dihydro-2H-chromen-6-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one 3-[4-(3,5-dimethyltriazol-4-yl)pyridin-2-yl]-6-methanimidoyl-7H-pyrrolo[1,2-c]imidazol-8-ium-1-amine [3-[2-(4,5-dimethylpyrazole-1-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]pyrrolidin-1-yl]-phenylmethanone N-methyl-5-[(4-oxo-3H-phthalazine-1-carbonyl)amino]furan-2-carboxamide N-[(2S)-1-amino-5-[[4-chloro-3,5-bis(trifluoromethyl)phenyl]methoxy]pentan-2-yl]-4-ethynylbenzamide;ethane 2-methoxy-5-(3-methylbutanoyl)benzoic acid 1-[(3S)-4-azidopiperidin-3-yl]indole 6-azidooxy-5,7,10-trimethyl-2-methylsulfanyl-1H-naphtho[2,3-h]quinoline 6-(4-tert-butylphenyl)-3-cyclohexylpyrazolo[5,1-c][1,2,4]triazole 4-fluoro-1,3-diphenylazetidine 1-(2,2-dimethylpropyl)-3-[4-(oxolan-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one 2-azidooxy-5-(1H-imidazol-2-yl)pyrimidine [1-(2,3-dihydropyrrolo[2,3-b]pyridine-1-carbonyl)cyclopropyl]methanol N-[(3Z)-hexa-1,3,5-trien-2-yl]-6-imino-N-methyl-3-pyridin-4-yl-1H-pyridazine-5-carboximidamide 1-(2,4-dichlorophenyl)-3-ethyl-N-[3-(hydroxyamino)-3-oxopropyl]-7-methoxy-8-(trifluoromethyl)indolizine-6-carboxamide N-[2-(4-methoxyphenyl)ethyl]-2-oxo-1,3-dihydrobenzimidazole-5-carboxamide 1-[2,3-di(propan-2-yl)phenyl]-3-ethyl-4-methoxypiperazine [4-(difluoromethyl)phenyl]-[3-(4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-5-carbonylamino)pyrrolidin-1-yl]methanone 2,3-bis(4-bromophenyl)-1H-imidazole 1,4-bis(2-methylpropyl)piperidin-4-ol;1-[2-(2H-tetrazol-5-yl)phenyl]propan-2-one 7-(2,4-dichlorophenyl)sulfonyloxyheptylcarbamic acid N-[(2S)-1-(2,5-diaminopyridin-4-yl)oxypropan-2-yl]-1-methoxyisoquinoline-3-carboxamide 5-[[5-(2,4-dichlorophenyl)furan-2-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one 6-methoxy-1-methyl-3,4-dihydro-2H-quinoline;3-[4-(5-propan-2-ylpyrazin-2-yl)phenyl]oxetane 2-ethyl-1-[3-(oxolan-3-ylmethoxy)pyridin-4-yl]sulfonylpyrrolidine-2-carboxamide N-(4-chlorophenyl)-1'-[(3,5-dimethylphenyl)methyl]spiro[7H-furo[3,4-d]pyrimidine-5,3'-azetidine]-2-imine 5-(5-fluoropyridin-3-yl)-4,6-dimethoxypyrimidine 1-amino-5,10-dihydrobenzo[b][1]benzoxepine-3-carboxylic acid;2,6-diaminohexanoic acid N-(3,4,5-trimethylpyrazol-1-yl)-2-(3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)acetamide;dihydrochloride 4-[(7-tert-butylquinoxalin-2-yl)amino]phenol 2-methyl-4-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[6-(1-methyltriazol-4-yl)cinnolin-3-yl]piperidine-4-carboxamide 1-N-(4,6-dimethoxypyrimidin-2-yl)butane-1,3-diamine (E)-4,4-difluoro-N-[2-(1H-indole-3-carbonyl)phenyl]but-2-enamide 2-[4-(3,5-dimethylbenzoyl)phenoxy]acetate 5-[4,5-bis(3-hydroxypropyl)pyridin-2-yl]benzene-1,3-diol;butane 1-[(3,5-dichlorophenyl)methyl]-4-propanoylpiperidine-4-carboxamide 2-[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]-6,7-dihydro-5H-quinolin-8-one 5-[(E)-2-(6,7-dimethoxy-3,4-dihydroisoquinolin-1-yl)ethenyl]-N,4-dimethyl-1H-pyrazol-3-amine 2-(4,6-dimethyl-1H-benzimidazol-2-yl)-3a,4-dihydroindene-1,3-dione 4-[1-[(5Z,7E)-3,9-dihydrocycloocta[c]pyridine-8-carbonyl]piperidin-4-yl]morpholin-3-one (3R,4S)-1-(cyclohexylmethyl)-N-[[4-(2H-tetrazol-5-yl)phenyl]methyl]-4-(trifluoromethoxy)pyrrolidine-3-carboxamide 2,4-diaminopyrrolo[2,3-d]pyrimidine-7-carboxylate (2S)-2,4-dihydroxy-1-methyl-3-[4-[6-[[(3R)-oxolan-3-yl]amino]pyrazin-2-yl]phenyl]-7-(trifluoromethyl)pyrido[2,3-d]pyrimidin-3-ium-2-ol 7-[(6,8-dimethoxy-2H-quinolin-1-yl)sulfonyl]-3,4-dihydrochromen-2-one 3-(N-[3-nitrophenyl)methyl]anilino)phenol 3-[1-(2-ethoxypyridin-4-yl)piperidin-3-yl]-1H-benzimidazole-2-thione N-(3,3-dimethylbut-1-en-2-yl)-5-[7-fluoro-3-[4-(furan-3-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-2H-indazol-5-yl]pyridin-3-amine N-ethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-6-carboxamide 2-methyl-N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)-2-(trifluoromethoxy)phenyl]propanamide;hydrochloride (E)-3-[2,6-bis[4-fluoro-3-(trifluoromethyl)phenyl]pyridin-4-yl]-1-chloroprop-1-en-2-ol 5-(1H-indole-2-carbonyl)-N-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 1-(4-methylphenyl)sulfonyl-N'-(2-morpholin-4-ylethylamino)piperidine-3-carbohydrazide (2S)-2-[(4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(5-methylthiophen-2-yl)butanamide N-(3,5-difluorophenyl)-6-morpholin-4-ylpyrimidine-4-carboxamide 2-(3-chlorophenyl)-N-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]acetamide 5-chloro-6-phenyl-N-[2-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine 1-(4-methylsulfonylphenyl)-2-oxopyridine-3-carboxylate 2-[N-(3-methylbut-2-enyl)anilino]-1-phenylethanone 3-(1,4,5,6-tetrahydropyrimidin-2-yl)-9H-fluorene 3-chloro-1H-indole;3-(cyclohexylamino)-5-[[3,3,5,5-tetramethylpiperazin-4-ium-1-ylidene]amino]benzoic acid [7-(3,4-dimethoxyphenyl)-2,6-bis(methylsulfanylmethyl)pyrazolo[1,5-a]pyrimidin-5-yl]-[4-(3-hydroxypropyl)piperazin-1-yl]methanone 2-[(2R,4S)-1-acetyl-2-benzamido-6-oxopiperidin-4-yl]acetic acid 2-[6-(aminomethyl)pyridin-3-yl]-1H-quinazoline-2,4-diamine;dihydrochloride 4-(5,6-dimethylimidazo[2,1-b][1,3]thiazol-3-yl)-N,N-diethylbutan-1-amine 4-N-methyl-2-N,6-N,10-triphenylphenothiazine-10,9-diamine (Z)-3-[5-methyl-4-[(E)-2-phenylethenyl]-1H-imidazol-2-yl]-N-propan-2-ylidenebut-2-en-2-amine 7-chloro-3-(5,6,7,8-tetrahydroquinolin-2-yl)imidazo[1,5-a]pyridine 3-cyclopentyloxy-4,5,6-trifluorobenzene-1,2-dicarbonitrile N-methylsulfonyl-1H-indazole-3-carboxamide 4-[5-(4,4,5,5-tetramethyloxaborolan-2-yl)pyridin-3-yl]butanal 6-[5-(2,2-difluoroethoxy)pyridine-3-yl]-4-oxo-1-propan-2-yl-1H-pyridazine-3-carboxylic acid 5-[(3S)-2-acetyl-3-(4-hydroxyphenyl)-3,4-dihydropyrazol-5-yl]-1-(3,4-dimethylphenyl)-6-hydroxypyrimidine-2,4-dione 3-(1H-pyrrole-2-carbonyl)imidazole-4,5-dicarbonitrile 2-[1-[(Z)-butan-2-ylideneamino]piperidin-4-yl]-N-pyridin-3-ylacetamide 2,6-diethyl-N'-[2-(2-ethoxypropanoylamino)-5-pyridin-3-ylphenyl]benzenecarboximidamide N-cyclopropyl-1,2-dimethyl-N-[(4-methylsulfinylphenyl)methyl]indole-3-carboxamide N-[4-(2,5-dichlorophenyl)sulfanyl-1,3-thiazol-2-yl]-2-[1-(dimethylamino)ethyl]pyridine-4-carboxamide 1-azidosulfanyl-2,3,4,5-tetrachlorobenzene N-(2-fluoro-6-methylphenyl)-5,7-dihydroxy-4-oxochromene-3-carboxamide 2-(1,3-benzoxazol-6-ylamino)pyridine-4-carboxylic acid 4-[(1S,3R)-2-amino-3-[[methyl-[(E)-2-phenylethenyl]carbamoyl]amino]cyclohexyl]butanoic acid 2-[[5-(3,4-dimethoxyphenyl)thiophen-3-yl]methylamino]-N-hydroxyacetamide 4-(2,6-difluoroanilino)-5-ethanimidoyl-1H-pyrimidin-6-one (2R,5S)-5-[(5-fluoropyrimidin-4-yl)amino]oxolane-3,4-diol 1-[3-chloro-4-(trifluoromethyl)phenyl]-5,6-dihydro-4H-pyrazolo[3,4-e]indazole 2-[3,5-bis(trifluoromethyl)phenyl]-4-methoxy-1,2-dihydropyrimidine 3-benzyl-4-(2,4-dichlorophenyl)-N'-[2-methylsulfanyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazine-1-carboximidamide 5-[3-(6-bromopyrimidin-4-yl)oxyanilino]oxypentanoic acid 5-benzyl-2-[1-(benzenesulfonyl)piperidin-4-ylidene]pyrrolidine 3-[4-(dimethylamino)butoxy]-2,5,6-trifluorobenzenethiol 3-[1-azidooxy-2,4-bis(phenylmethoxy)butan-2-yl]-5-ethoxyphenol 2-[(3R,4S)-6-fluoro-3,4-dimethyl-5-oxo-1,2,3,4-tetrahydro-1,5-benzodiazepine-8-carbonyl]oxypropanedioic acid N'-[6,7-dichloro-1-(cyclopropylmethyl)-4,5-dihydroindazole-3-carbonyl]-2-nitrobenzohydrazide [1-[(2R)-2-[[(2S,4R)-2-(1H-benzimidazol-2-ylmethoxycarbonylamino)-3,4-dihydro-2H-chromen-4-yl]carbamoyl]pyrrolidine-1-carbonyl]cyclopropanecarbonyl]oxidanium (3E)-5,6-dichloro-3-[(E)-2-iodoethenyl]imino-1H-indol-2-one 3-ethyl-1-[2-(4-methoxyphenyl)ethyl]pyrrolidine 2-[4-(6-azidopyrazin-2-yl)piperazin-1-yl]ethanol N'-(4,6-dimethoxypyrimidin-2-yl)-9H-fluoren-1-amine 2-[3-[(7-chloroquinolin-4-yl)amino]propyl]-1,3-oxazole-5-carboxylic acid N-[1-(4-methoxyphenyl)propan-2-yl]-4,4-dimethyl-2,3-dihydroisoquinoline-1-carboxamide (4-hydroxyphenyl)-[2,3,5,6-tetrafluoro-4-methoxy-6-(trifluoromethyl)cyclohexa-1,3-dien-1-yl]methanone (NE)-2-methyl-N-[(3S,4R)-3-phenyloxan-4-ylidene]propane-2-sulfinamide (1R)-2,2-dimethyl-N'-[(4-phenyl-5-propylpyridin-3-yl)methyl]cyclohexane-1-carbohydrazide;1H-indole N-(3,5-dimethylphenyl)-2-ethoxy-4-(6-oxo-4H-triazin-1-yl)benzamide 2-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]propanoic acid 2-N,4-N-bis(3H-azepin-6-ylmethylideneamino)benzene-1,2,4,5-tetramine 4-[(Z)-1,3-bis(benzenesulfonylmethylsulfanyl)prop-2-enylidene]-N,N'-diethylpiperidine-1-carboximidamide 1-azido-2,3-dichloro-4-[(4-chlorophenyl)methyl]benzene 2-[2,4-bis(aminomethyl)phenyl]-3H-quinazolin-4-one 2-[(3,4-dimethoxyphenyl)methyl]-5-N,5-N-bis[(E)-1-hydroxyprop-1-enyl]pyridine-2,5-dicarboxamide 4-[(2S,3S)-1-[5-chloro-6-methyl-7-(trifluoromethyl)-1H-indole-2-carbonyl]-2-ethylpiperidin-3-yl]benzonitrile 5-[3-(1H-indol-2-yl)-1,2,4-oxadiazol-5-yl]-2,6-dimethylpyran-4-one 2-(3-aminophenyl)-6-[1-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]pyridazin-3-one 2-(N-benzyl-4,5-dimethyl-2-phenyldiazenylanilino)acetonitrile 3-[[4-(2,4-dimethoxyphenyl)-5-pyridin-2-ylimidazol-1-yl]methyl]thiophene-2-sulfonic acid 5-bromo-4-[(2,3-difluorophenyl)methylamino]-1H-pyrimidin-6-one (4R)-1-(4,6-dimethylpyrimidin-2-yl)-3-phenylimidazolidine-4-thione N-(4-azidophenyl)-2,3-dihydro-1H-isoindole-5-carboxamide 1-bromo-2,3,4-trifluoro-5-methylbenzene;ethane N-butyl-1,3-benzodioxol-5-amine;1,4-difluorobenzene 3-[2-bromo-N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)anilino]phenol 1-(cyclopropylmethyl)-3-(3,5-difluorophenyl)-4-[2-(4-morpholin-4-ylanilino)pyrimidin-4-yl]imidazolidin-2-one 2-methylsulfanyl-N-[4-(trifluoromethoxy)phenyl]quinoline-3-carboxamide (3-azido-4,6-dihydrothieno[2,3-c]pyrrol-5-yl)-[3-(trifluoromethyl)phenyl]methanone (3-aminopyrazol-1-yl)-[2-methyl-4-nitro-5-(trifluoromethyl)anilino]methanol N-[(3R)-1-[2-(4-fluorophenyl)acetyl]pyrrolidin-3-yl]methanesulfonamide (3R,4S)-3-hydroxy-4-[4-(methoxymethyl)phenyl]piperidine-1-carboxylic acid 4-[3-(2,6-dichlorophenyl)-1H-1,2,4-triazol-5-yl]-2-methoxyphenol 5-[2,4-difluoro-3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidine-2,4,7-trithione 7-ethenyl-5-methylidene-2,3-dihydrothieno[3,4-b][1]benzothiepine 4-[3-cyano-4-[(1S)-1-methyl-6-oxo-2,3-dihydropyridin-5-ylium-3-yl]thiophen-2-yl]benzonitrile N-methyl-1-[5-(2,3,4,5-tetrahydropyridine-6-carbonyl)pyridin-2-yl]piperidine-4-carboxamide 1-(2,3-dihydroindol-1-yl)-3-[4-hydroxy-5-(5-hydroxy-1H-indole-2-carbonyl)-6-methylidenepyrimidin-1-yl]propan-1-one N-(2,5-dichlorophenyl)sulfonyl-4-methoxypiperidine-1-carboxamide 2-[4-[5-chloro-1,3-dioxoisoindol-2-yl]cyclohexyl]acetic acid 1-methyl-7-[3-(piperidine-1-carbonyl)anilino]pyrido[2,3-b]pyrazin-4-one 4-[4-(2,3-dihydro-1H-inden-5-yl)phenyl]-2-methoxycarbonylbenzoate 3-[2,4-dimethyl-6-oxo-5-(trifluoromethoxy)pyrimidin-1-yl]benzoic acid (2S,4R)-1-[(2-phenylquinoline-3-carbonyl)amino]-4-phenoxypyrrolidine-2-carboxylic acid 6-[4-(3,5-dimethylphenyl)piperidine-1-carbonyl]-4H-pyrazino[2,3-b][1,4]oxazin-3-one 2-(4-aminopiperidin-1-yl)-N,5-dimethylbenzimidazole-1-carboxamide (4E)-2-[3-fluoro-5-(trifluoromethyl)phenyl]-4-[(Z)-2-fluoroethylidenehydrazinylidene]cyclohexane-1,3-dione 1-(3,4-dimethylphenyl)-6-hydroxy-5-[(2-oxochromen-7-yl)oxymethyl]pyrimidine-2,4-dione 5-(2,6-dichlorophenyl)-N'-hydroxypyrazine-2-carboximidamide 2-[1-azidooxy-2-methylpropan-2-yl]oxynaphthalene (1S)-4-ethyl-6,7,8,9-tetrahydro-3H-cyclopenta[c]isoquinoline (2S,4R)-6-chloro-N-[5-cyano-2-methoxy-3-(methylamino)phenyl]sulfonyl-4-hydroxy-1-[2-oxo-2-[(3R)-piperidin-3-yl]ethyl]-3,4-dihydro-2H-quinoline-2-carboxamide 4-[[5-(aminomethyl)-1,3,4-oxadiazol-2-yl]methoxy]benzoate 4-[(2,6-dimethoxyphenyl)carbamoyl]piperazine-1-carboxylic acid 3-amino-5-(2,6-dichloro-4-fluorophenyl)-1H-pyrazole-4-carbonitrile 1-[5-methyl-3,4-bis(phenylmethoxy)pyridine-2-carbonyl]piperidine-4-carboxylic acid 2-methyl-N-[(1S)-1-phenylprop-2-enyl]propane-2-sulfonamide 2-[(6R,9aS)-1-hydroxy-3,4,6,7,8,9,9a-hexahydro-2H-quinolizin-2-yl]acetic acid;3-fluoro-N-methylpyridine-4-carboxamide 3-[4-amino-5-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N-cyclohexa-1,5-dien-3-yn-1-ylbenzamide 5-(2-amino-6-methylpyridine-4-carbonyl)-3a-(hydroxymethyl)-1,3,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-one;hydrochloride 2-[N-(benzenesulfonyl)-4-fluoroanilino]acetamide N-azido-2,4-dimethoxybenzamide (3S)-1-[5-cyclopropyl-4-[(1S,2R)-2-methylcyclopentyl]oxypyridin-2-yl]pyrrolidine-3-carboxylic acid 2-[5,6-bis(4-chlorophenyl)-1H-imidazo[1,2-b]pyrazol-3-yl]acetamide 4-[(2,4-dichlorophenyl)-diethoxyphosphorylmethyl]-1-[(3,5-difluorophenyl)sulfanyl]piperidine (3-azido-1,2-oxazol-5-yl)-[4-(3,4-dichlorophenyl)piperazin-1-yl]methanone 2-bromo-N-butyl-4,5-dimethoxybenzenesulfonamide (3S)-3,5-dibenzyl-1-methylpiperazine 1-[4-[5-amino-6-(quinoline-2-carboximidoyl)pyrazin-2-yl]piperazin-1-yl]prop-2-en-1-one 1-phenyl-3,3a,7a-tetrahydrobenzo[e]isoindole 4-cyclobutyloxycarbonylbenzenesulfonic acid 3-benzyl-2-[(2,5-dimethoxyphenyl)methylideneamino]benzoic acid 1-phenyl-2,3,4-tripropoxybenzene 3-[4-(6-chloroquinoline-8-carbonyl)piperazin-1-yl]oxolane-2,5-dione N-[(3R,7S)-2,11-dioxo-5-thia-1-azabicyclo[12.4.0]octadeca-10,13,15,17-trien-3-yl]-2-phenoxyacetamide [4-(azidomethyl)phenyl]sulfonyl-propan-2-ylideneoxidanium 2-(2,3-dihydroindol-1-ylmethyl)-5-(4-hydroxyphenyl)-1H-[1]benzoxepino[4,5-c]pyrrole-3,9-dione [2-hydroxy-3-(1H-indol-3-yl)propoxy]phosphinous acid 4-[3-bromo-2-(methylsulfonylcarbamoylamino)benzoyl]piperidine-1-carboxylic acid 1-[(4R,5S)-2-fluoro-4-hydroxy-5-methyloxolan-3-yl]-5H-pyrazolo[3,4-d]pyrimidin-4-one N'-hydroxy-4-(3-hydroxypropylsulfanylmethyl)pyridine-2-carboximidamide 3-amino-5-(3,4,5-trifluorophenyl)-1H-pyrazole-4-carboxamide 2-[2,6-bis(ethenyl)phenyl]iminopropanedinitrile (2S,4R)-4-(3,5-difluorophenyl)-6-[ethyl(methyl)amino]-1-(1H-indol-2-ylsulfonyl)piperidine-2-carboxylic acid 4-[(Z)-[[2-[[(1R)-1-phenylethyl]amino]pyrimidin-5-yl]hydrazinylidene]methyl]phenol 2-(3,5-diethylpyrazol-1-yl)pyridine 2-[[5-chloro-3-(cyclopropylamino)pyrazine-2-carbonyl]amino]ethylcarbamic acid 6-methyl-2,4-bis(phenylmethoxy)quinoline N-[3-(methoxymethyl)-1H-indol-2-yl]-2,2-dimethylbutanamide 2-[(3R,5S)-1-[3-(dimethylamino)phenyl]sulfonyl-5-methoxypiperidin-3-yl]-N,N-dimethylacetamide 4-[[3-(2-azidoethyl)phenyl]methoxy]benzonitrile 2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)morpholine-4-carboxamide;dihydrochloride N-[5-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-3-yl]-5-fluoropyridine-3-carboxamide 3-[(2S)-1-benzylpyrrolidine-2-carbonyl]-4-hydroxy-5,6,7,8-tetrahydrocinnoline-1-carboxylic acid [2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-[3-(triazol-1-yl)pyrrolidin-1-yl]methanone (3S)-3-[[6-chloro-5-fluoro-2-[4-(hydroxymethyl)piperidine-1-carbonyl]-1H-indol-3-yl]amino]butanoic acid 4-[(2R)-2-methylpyrrolidine-1-carbonyl]benzaldehyde 1-N'-[5-[7-(5-fluorothiophen-2-yl)-3H-imidazo[4,5-c]pyridine-2-carboximidoyl]pyrimidin-4-yl]-1-N-methylethene-1,1-diamine 4-[(1E)-3-bromobuta-1,3-dienyl]-2-chloropyridine 1-N,3-N-dimethyl-1-N-[2-(4-methylphenyl)ethyl]benzene-1,3-disulfonamide N-[4-(2,4-difluorophenoxy)phenyl]-1H-pyrazolo[3,4-b]pyridine-5-carboxamide N-[[4-(3,5-difluorophenyl)thiophen-2-yl]methyl]carbamate 5-[[4-(2-azidoethynyl)phenyl]methyl]-1,3-thiazolidine 1-[(4R)-3,7-dimethyloctoxy]-2-propan-2-ylbenzene 2,3-difluoro-1H-indene;5-[4-(4-ethylsulfonylpiperazin-1-yl)phenyl]-3-methoxy-7-methylidenepyrazolo[1,5-a]pyrimidine 1-[4-amino-5-(7,8,9,10-tetrahydrophenanthridin-6-yl)pyrimidin-2-yl]piperidine-3-carboxamide (E)-3-[4-[3,6-dimethyl-4-[1-oxo-2-(trifluoromethyl)phthalazin-5-yl]oxypyridin-2-yl]naphthalen-1-yl]prop-2-enoic acid [3-chloro-4-[(2,3-difluorophenyl)methoxy]-5-ethylphenyl]phosphane 1-[3,5-difluoro-4-(trifluoromethyl)phenyl]ethanamine;4-(3-piperidin-4-ylpropoxy)pyridine (E)-3-(2,5-dimethoxyphenyl)-1-[4-hydroxy-5-(3-methylbut-2-enoxy)cyclohepta-1,4,6-trien-1-yl]prop-2-en-1-one 5-(bromomethyl)-1,3-bis[2-(4-ethoxyphenyl)acetyl]imidazolidine-2,4-dione 3-(2,6-dichlorophenyl)-7H-[1]benzofuro[2,3-b]pyridine;ethane 1-[5-amino-3-(3-fluorophenyl)-4,6-dioxo-1,2,4a,8b-tetrahydropyrido[4,3-d]pyrimidin-7-yl]prop-2-ynylideneazanide 4-[[2,3-bis(ethenyl)-6-(4-fluorophenyl)pyridin-4-yl]methoxycarbonylamino]pentanoic acid N-(2,5-dimethylphenyl)-4-(2,3-dihydroindol-1-ylsulfonyl)benzamide 2-[4-(3,4-dichlorophenyl)butyl]-1-(3,5-difluorophenyl)sulfanyl-9H-xanthene (3S)-1-[5-(5,7-dimethoxyquinoxalin-2-yl)sulfanylpentyl]pyrrolidin-3-ol 2-[4,6-difluoro-1-methyl-5-(morpholine-4-carbonyl)indol-3-yl]-N-[(Z)-hydrazinylidenemethyl]-2-oxoacetamide 4-[(3R)-3-aminopyrrolidine-1-carbonyl]-7-fluoro-2H-isoquinolin-1-one 5-chloro-1,3,4-triethylpyrazolo[3,4-b]pyridine 1-azido-3-(3,4-dimethoxyphenyl)-9H-fluorene [(1E)-2-chloro-3-cyclopropylbuta-1,3-dienoxy]benzene 2-hydroxy-3,3,6,7-tetramethyl-5-(2,4,6-trihydroxyphenyl)chromene-2-carboxylic acid ethane;(Z)-3-[4-(7-fluoronaphthalen-1-yl)piperidin-1-yl]-2,5-dimethoxyhept-3-enoic acid N-[3-[(dimethylamino)methyl]phenyl]-4,6-dioxo-1H-1,2,5-triazine-2-carboxamide 2-[(1S)-1-hydroxyethyl]-6-methoxy-3H-quinazolin-4-one ethane;ethene;N-(5-methylpentan-2-yl)-4,5,6,7-tetrahydrothieno[3,2-b]pyridine-2-carboxamide 2-ethylsulfanyl-6,7-dimethylquinoline 1-azido-4,7,10,13,15,16-hexazahexacyclo[13.6.0.02,9.03,8.011,15.017,22]docosa-2(9),3(8),4,6,11,13,18,20-octaene 2-(2,3-difluoro-4-hydroxyphenyl)-5H-benzo[b]azepine-7-thione 2-N-(4-cyclopentyloxyphenyl)-4-N-[4-(1,3-oxazol-5-yl)phenyl]-5-(trifluoromethyl)pyrimidine-2,4-diamine 1-[(2S)-2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)pyrrolidin-1-yl]-2-piperidin-1-ylethanone (2E)-4-(2,3,5,6,7,8-hexahydronaphthalen-1-ylmethylidene)-2-[2-methoxy-6-(trifluoromethyl)phenyl]iminocyclopentan-1-one 3-[[(2R,4S)-4-ethoxypyrrolidine-2-carbonyl]amino]-N-propyl-1H-pyrazole-5-carboxamide N-[2-(5,6-dimethylbenzimidazol-1-yl)ethyl]-4-pyridin-3-ylpiperazine-1-carboxamide 1-[[3-(4,5-dihydropyrimidine-2-carbonyl)phenyl]methyl]-N'-[1-[hydroxy(methoxy)methyl]-6-(trifluoromethyl)indazol-4-yl]pyrrolidine-2-carboximidamide N-[1-(2,6-difluorophenyl)pyrrolidin-3-yl]spiro[1H-isoquinoline-4,1'-cyclopropane]-2-carboxamide 5-(3,4-dimethoxyphenyl)-N-[(2R,6S)-1-hydroxy-5-oxo-2H-pyrrol-3-yl]furan-2-carboxamide 3-(1-phenyl-5,6-dihydro-4H-cyclopenta[c]pyrazol-3-yl)propanoic acid N-[(1R,2S)-2-hydroxycyclohexyl]-2-methoxy-3-(1-propan-2-ylpyrazol-4-yl)quinoline-6-carboxamide 2-[3-ethylsulfonyl-4-[3-methyl-6-(trifluoromethyl)imidazo[4,5-b]pyridin-2-yl]pyrazolo[1,5-a]pyridin-2-yl]propan-2-ol 3-[(3S)-1-(benzenesulfonyl)piperidin-3-yl]-6-propanoyl-2,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-[4-(5-azido-1H-1,2,4-triazol-3-yl)phenyl]quinoline 3,5-dichloro-4-[(2E)-2-ethylidene-7-methyl-6-phenylocta-3,8-dienoxy]phenol N-(2,6-difluorophenyl)-7-methyl-4-oxo-3H-thieno[3,2-d]pyrimidine-5-carboxamide 2-[[4-(dimethylamino)phenyl]methylidene]propanedioic acid [4-(3,5-dimethoxyphenyl)-6-[2-hydroxy-2-(oxan-4-yloxy)ethoxy]quinazolin-7-yl]-pyrrolidin-1-ylmethanone (3Z)-3-(aminomethylidene)-1-[4-[6-methoxy-7-(4-morpholin-4-ylphenyl)quinolin-4-yl]piperazin-1-yl]butane-2,4-dione 5-chloro-N-[(Z)-1-[3,5-dichloro-2-[[1-(1H-indazole-4-carbonyl)azetidin-3-yl]methoxy]phenyl]prop-1-enyl]-2-fluorobenzenesulfonamide 2-chloro-1,5-dimethylindole;2,4-diaminopyrimidine-5-carboxamide [1-(2,6-dimethylpyrimidin-4-yl)pyrrolidin-3-yl]urea (3S)-1,1'-dibenzylspiro[indole-3,4'-piperidine] 2-(3-pyridin-4-ylbutanoyl)cyclopentan-1-one 1-[5-[4-amino-6-[methyl(oxan-4-yl)amino]pyrimidine-5-carboximidoyl]-2,3-dihydroindol-1-yl]ethanone (5-fluoropyridin-3-yl)-[2,4,6-trimethyl-3-[(5R)-5-methyl-1-(oxetan-3-yl)pyrrolidin-3-yl]oxyphenyl]methanone 4-methyl-3,5-diphenyl-1H-imidazole [3-amino-6-(2,5-dimethyl-1H-imidazol-4-yl)-1-benzothiophen-2-yl]-phenylmethanone 1-[(E)-2-nitroethenyl]sulfonyl-4-[3-(trifluoromethoxy)phenyl]benzene 2-amino-N-[(Z)-1-aminobut-1-enyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-3-carboxamide;5,6,7,8-tetrahydronaphthalene-2-thiol (3R)-1-[4-(3,5-dimethylphenyl)phenyl]pyrrolidine;methanimine (E)-3-[(1R,2S,6S)-2,4-dimethylcyclopentyl]-1-(7-fluoro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)prop-2-en-1-one N-[[1-[3-(3,4-dimethylphenyl)propanoyl]piperidin-4-yl]methyl]-5-oxo-6H-benzo[b][1,4]benzoxazepine-3-carboxamide 2-[2,4-bis(2-aminoethoxy)anilino]-1-[2-(trifluoromethyl)phenyl]ethanone 4-(2,3,6,7-tetrahydroazepin-1-yl)benzaldehyde N-[2-[[5-cyano-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]-5-ethoxyphenyl]prop-2-enamide N-[2,6-dichloro-4-(4-fluorophenyl)pyridin-3-yl]hydroxylamine [(1E,3Z)-1-ethenylsulfanyl-2-methylhexa-1,3,5-trien-4-yl]benzene 4-(2,3,5-trifluoro-1-benzothiophene-7-carbonyl)-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboxylic acid N-[4-[3-(6-chloropyridin-2-yl)propoxy]phenyl]-5,7-difluoro-1H-indole-2-carboxamide 1-N-cyclopentyl-4-N,6-dimethoxybenzene-1,2,3,4-tetraamine ethane;1-(4-methylphenoxy)anthracene-9,10-dione 2-[6-methyl-4-oxo-1-(1,3-thiazol-5-yl)pyridazin-3-yl]propanenitrile 5-(3,4-difluorophenyl)-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),5-dien-10-one ethane;2-methyl-2,3-dihydrothieno[3,4-c]pyran-4,7-dione 2-[4-(azetidine-1-carbonyl)-3-fluorophenyl]-1,1-dioxo-1,2-benzothiazol-3-one;ethane 3-(azidooxymethyl)-1,4-bis[2-(trifluoromethyl)phenyl]pyrrole 2-methyl-N-(6-oxopyridazin-3-yl)propanamide (1S,4R)-N-methyl-2-[2-[5-methylidene-6-oxo-4-(trifluoromethyl)pyrazin-2-yl]pyridin-3-yl]sulfonyl-4-phenylcyclopentane-1-carboxamide 4-(2,3,5,6-tetramethylphenyl)butanal 5-[4-chloro-N-(2,2-diethoxyethyl)anilino]naphthalene-2-sulfonic acid 2-chloro-4-[6-(trifluoromethyl)pyridin-3-yl]-8H-pyrido[1,2-a]pyrimidine (2R)-3-azidooxy-1-[[3-methyl-4-[(2,6,7,8-tetrahydrothiopyrano[2,3-b]pyridine-5-carbonylamino)methyl]benzoyl]amino]propane-1-sulfonic acid 3-methylsulfanyloxybenzaldehyde;propane 2-(3,4-dimethylphenyl)sulfanyl-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazine 1-[2-(benzylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]-N'-ethyl-N,N-dimethylazetidine-3-carboximidamide 1,2,3-trimethylbenzimidazole-5-sulfonate 7-(3,4-dimethoxyphenyl)-2-(6-methylpyridin-2-yl)-5-methylsulfanylpyrido[4,3-d]pyrimidine 7-(2-fluorophenyl)-6,8-dihydroimidazo[1,5-a]pyrazine 5-[4-(3,4-dichloroanilino)quinazolin-6-yl]oxypentanal 1-cyclobutyl-6-[(5-cyclopropyl-4,7-dimethylpyrazolo[1,5-a]pyridin-2-yl)amino]-4-oxopyridazine-3-carboxylic acid 3-[4,6-bis(2,2,2-trifluoroethoxy)pyrimidin-5-yl]-1H-indole 2-[(3R)-1-(2-cyclopropylacetyl)piperidin-3-yl]-7-methylsulfonyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one N-(5-cyclopropyl-1H-pyrazol-3-yl)-3,4-dimethoxybenzamide 3-chloro-4,5-diethylpyridine (3R,5R)-4-chloro-5-[[2-(3-methoxyphenyl)acetyl]amino]-N-(2-oxooxolan-3-yl)-1-propan-2-ylpyrrolidine-3-carboxamide N-[(Z)-[1-benzyl-3-fluoro-4,5-di(propan-2-yl)pyridin-2-ylidene]amino]methanamine (4aS,9aR)-8-[[2-fluoro-5-(trifluoromethyl)phenyl]methoxy]-1,2,3,4,4a,10-hexahydroacridine ethane;5-[4-(8-fluoro-3,7-dimethylquinolin-6-yl)phenyl]sulfanyl-2-methylsulfanyl-1H-pyrimidine-2,4-diamine N-[4-(6-oxo-3-phenylpyridazin-1-yl)cyclohexyl]propanamide 4-[6-(3,5-dichlorophenyl)pyridin-2-yl]cyclohexan-1-ol 6-azidooxy-3-phenoxycyclohexa-1,5-diene 2-(4,5,6,7-tetrachloro-1,3-dioxoisoindol-2-yl)oxyacetic acid 4-tert-butyl-2,5-di(propan-2-yl)-1H-pyrazol-3-one 3-(dimethylamino)-N-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-ylmethyl)cyclobutane-1-carboxamide (3,5-dimethoxyphenyl)-[7-[[3-[(4-ethylpiperazin-1-yl)methyl]-4-fluorobenzoyl]amino]-2-hydroxycyclohepta-1,6-dien-1-yl]-methylideneazanium N-[(E)-1-methylsulfanylprop-1-enyl]benzamide 1-azido-4-(4-bromophenyl)-3,5-dimethylpyrazole 2-(1H-indol-3-yl)-4,5-dimethoxybenzenethiol 7-[(4S)-4,5-dihydroxypentyl]pyrrolo[2,3-d]pyrimidine-6-carboxamide 3-(3-phenylmethoxynaphthalen-2-yl)-1H-1,2,4-triazole 4-N-azido-5,6-dimethylpyrimidine-2,4-diamine N-(2,4-difluorophenyl)-5,8-difluoro-6H-benzo[b][1]benzazepine-11-carboxamide N-[2-(3,4-dimethylphenyl)ethyl]-1-pyrimidin-5-ylcyclopentane-1-carboxamide 5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-7-yl)pyrimidine 2-(3,5-dimethoxyphenyl)-1H-imidazole;hydrochloride 4-[5-(trifluoromethyl)pyrazole-1-carbonyl]benzoate 5-(4,5-dimethyl-1H-pyrrole-2-carbonyl)-N-[2-hydroxy-3-methoxy-6-(propanoylamino)phenyl]-1-methylpyrrole-3-carboxamide (2E,4Z)-5-[[2-hydroxy-3-[(2-methylphenyl)carbamoylamino]propoxy]carbonylamino]-6-nitrohepta-2,4,7-trienoic acid 3-ethylsulfonyl-6-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyridine-2-carbonitrile 5-azido-7-bromoimidazo[1,2-a]pyridine 4-[2-(1,3-benzodioxol-5-yl)pyrrolidin-1-yl]-6H-pyrrolo[2,1-c][1,2,4]triazin-7-one N-[4,4-bis(methylperoxy)-1-oxobutan-2-yl]-7-chloroquinoline-3-carboxamide 3-[4-(4,5-dihydro-1H-imidazole-2-carbonyl)phenyl]-4H-pyrimidin-6-one 5-[3,5-bis(trifluoromethyl)phenyl]-N-pyridin-4-ylpentanamide 7-(azidomethyl)-5,5,6-triphenylcyclohepta-1,3-diene 2-[3-(4-fluorophenyl)sulfanyl-2H-pyridin-1-yl]acetic acid N-[2-(dimethylamino)ethyl]formamide;3,4-dihydro-1H-isochromene 1-[[5-amino-6-(methylamino)pyridazine-4-carbonyl]amino]-2,3,3a,4,9b-hexahydro-1H-cyclopenta[c]chromene-8-carboxylic acid [1-(2,4-dimethylphenyl)cyclopropanecarbonyl]oxidanium N-[(2R)-3-(4-hydroxy-1H-indol-3-yl)propanoyl]-6-nitrohexanamide 3,5-dibromo-4-chloro-1H-indole ethane;1-[(E)-2-methyl-3-phenylprop-2-enyl]-4-[2-(4-methylphenoxy)ethoxy]piperidine (Z)-3-[2-chloro-4-[1,2,5-thiadiazol-4-yl(propanoyl)amino]phenyl]-4-iminopent-2-enimidamide 4-[(6-chloropyridine-3-carbonyl)amino]-N-methyl-1H-pyrazole-5-carboxamide [2-methyl-1,3-bis(methylideneamino)indol-6-yl]boronic acid ethene;4-[1-(4-ethenylphenyl)ethenyl]aniline N-cyclopropyl-2-[4-[6-(3,5-dimethoxyanilino)pyrimidine-4-carboximidoyl]phenoxy]acetamide N-(3,5-dimethylphenyl)-4-[(2E,4Z)-hepta-2,4,6-trien-2-yl]-7-(1H-indazol-6-ylmethoxy)quinoline-2-carboxamide;ethane ethane;1-[5-(6-methoxyquinolin-4-yl)oxypyridin-2-yl]pentan-3-imine 2,3-diethyl-8,9-bis(4-methoxyphenyl)-1H-purine-2,6-diamine 5-chloro-4-[(2,6-dimethoxycyclohexyl)amino]-1H-pyrimidin-6-one 3-amino-N-[2-(dimethylamino)ethyl]-5,6-dimethoxy-4H-cyclopenta[b]thiophen-2-amine 6-(1,3-dimethylpyrazol-4-yl)sulfonyl-2-oxo-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidine-4-carboxylic acid N-ethyl-4-[5-(methylamino)-3,6-dioxomorpholine-2-carbonyl]-N-[3-(trifluoromethyl)phenyl]benzamide 2-[(6-chloropyridazin-3-yl)-methoxycarbonylamino]propanoic acid (2E,4Z)-2-ethenyl-5-ethylhexa-2,4-dienoic acid;N'-[[3-[6-(methoxycarbonylamino)pyridine-3-carboximidoyl]phenyl]methyl]oxamide 3-[8-(4-phenylmethoxycyclohexyl)oxyisoquinolin-6-yl]benzenesulfonamide 2-(1,3-benzothiazol-6-yl)butanenitrile N-methyl-2,3,5-tri(propan-2-yl)aniline;hydrochloride (2R)-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide 5-(1H-indole-2-carbonyl)-N,3-dimethyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-4-carboxamide 4-[(2Z,5R)-2-[(Z)-1-(furan-2-yl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]butanoic acid 3-[5,6-dihydroxy-4-methyl-2-oxo-1-(4-phenylphenyl)pyridine-3-carbonyl]piperidine-2,6-dione 4-[3,6-diphenylhexyl(ethenyl)amino]butanoic acid 3-(aminomethylidene)-4-cyano-5,6,7-triethoxyisoindole-1-carboxylic acid 2-[(4R)-3-amino-1-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]benzoic acid N-[4-(5-bromopyridin-2-yl)oxybutyl]aniline 1-[5-(3,4-dichlorophenyl)-6-methyloxan-2-ylidene]propane-2-thione 4-[3-(5,7-dimethylquinoxalin-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl-[(1E)-2-(methylideneamino)buta-1,3-dienyl]amino]-5-propan-2-yl-2-quinolin-6-ylbenzamide [2-azido-1-(benzylamino)cyclohexa-2,4-dien-1-yl]-phenylmethanone 2-(4,5-dihydroimidazol-1-yl)-N-methyl-4-(6-pyridin-3-ylimidazo[1,2-a]pyrimidin-7-yl)aniline N-(4,5-dihydropyrimidin-2-yl)-3-fluoro-4-morpholin-4-ylaniline 4-azido-N-cyclohexyl-3,5-dimethoxybenzamide 2-amino-N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]pyridine-3-carboxamide 1-[(3E,5Z)-hepta-1,3,5-trien-3-yl]oxy-4-propan-2-ylbenzene 3-[4-bromo-1-(2,6-dichlorophenyl)pyrazolo[3,4-c]pyridin-7-yl]oxypropan-1-ol 4-[(2,3-dimethoxyphenyl)methylamino]-5-iodo-1H-pyrimidin-6-one 5-[4-(4-azidophenyl)but-1-enyl]-3-cyclopropyl-2,4-dimethoxypyridine 4-[3-(2,5-dimethylhexan-2-yl)phenyl]phenol 3-(dimethylamino)-N,2-bis(sulfanyl)benzamide 1-[6-azidooxy-1-butyl-2,3-dihydroinden-5-yl]ethanone 2-[6-(4,5-dihydro-1H-imidazol-2-yl)isoquinolin-3-yl]isoindole-1,3-dione N-[[4-chloro-3-(5-cyanopyridin-2-yl)phenyl]methoxycarbamoyl]formamide N-[(4-fluorophenyl)methyl]-2-methoxy-7,8,9,10-tetrahydrophenanthridin-6-amine 1-[(3S,4R)-1-tert-butylpiperidin-4-yl]-2-thiophen-2-yl-6H-pyrazolo[4,3-d]pyrimidin-7-one (4S)-2-amino-N-[5-[2,3-dimethyl-7-[1-(oxan-4-yloxy)ethenyl]-1H-indol-6-yl]-1,3-thiazol-2-yl]-4-propan-2-yl-4,5-dihydro-1,3-thiazolo[4,5-d]pyridazine-6-carboxamide 4-(3,5-dimethyl-1H-pyrazol-4-yl)-2,6-difluorobenzonitrile;ethane 1,2-diamino-4-[3-bromo-4-[(3,5-dichlorophenyl)methoxy]-5-methoxyphenyl]-6-oxopyridine-3,5-dicarbonitrile N-butyl-2,3-dichloroaniline 3-(2,5-dioxopyrrolidin-1-yl)benzenesulfonic acid;3-ethoxypropanoic acid 2-[4-(6-aminopyridin-3-yl)piperazine-1-carbonyl]-5,7-dichlorospiro[6H-pyrazolo[1,5-a]pyrazine-8,4'-piperidine]-3-one 1-[(2R,4S)-2-methyloxan-4-yl]-7-[[4-[4-(trifluoromethoxy)phenyl]benzoyl]amino]indole-2-carboxamide 4-[(E)-2-[3,5-bis(trifluoromethyl)phenyl]ethenyl]-2H-benzotriazole 2-(4,5-dihydro-1H-imidazol-2-yl)phenol;2-(3-hydroxyphenyl)-N-[5-(hydroxymethyl)thiophen-2-yl]propanamide 1-(2,5-difluorophenyl)-N-[3-fluoro-4-methyl-7-(2-morpholin-4-ylethoxy)quinolin-8-yl]methanesulfonamide 3-(2,2-dimethylpropanoyl)-4-[1-(thiophen-2-ylmethoxy)ethenyl]-6,7-dihydro-5H-cyclopenta[c]pyridin-1-one (Z)-2,3,4,5-tetrafluoro-N-[1-[(E)-5-phenylpent-2-enyl]piperidin-4-ylidene]benzenesulfonamide [1-(2,3-dihydroindole-1-carbonyl)piperidin-4-yl]-[(5R,7S)-2,5,7-trimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazol-3-yl]methanone 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-4-methyl-N-(4-phenylphenyl)aniline 1-cyclohexa-2,4-dien-1-yloxy-3-(2-methylidenepentyl)benzene 2-(5-methylfuran-2-yl)-4,6-bis(trichloromethoxy)pyrimidine 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-4-[1-(3-methoxypropyl)piperidin-4-yl]-1H-1,2,4-triazol-5-one [(E)-4,5-diamino-1H-indol-3-yl]carbamic acid 4-[(3S)-4-azidomorpholin-3-yl]pyridin-2-amine 7-(4,4a,8b-dihydrodibenzothiophen-3-yl)-4-iodo-1H-indole 3-[(2R)-1-[2,4-difluoro-6-(4-pentylcyclohexen-1-yl)phenyl]propan-2-yl]pyridine 4-amino-N-(8-carbamoylspiro[1,3-dihydroisoquinoline-4,1'-cyclopentane]-7-yl)benzamide N-(7-hydroxynaphthalen-2-yl)naphthalene-1-carboxamide 1-phenyldecane-4,5-diol 2-(N,4-dimethylanilino)-3-[4-hydroxy-3-(propanoylamino)phenyl]chromene-4-thione N-(1,5-dimethylpyrazol-4-yl)sulfonyl-2-(4-methoxypiperidin-1-yl)acetamide 5-[2,6-dichloro-4-(trifluoromethyl)phenyl]-3H-1,3,4-oxadiazol-2-one N-[(4S)-5-[3,5-difluoro-2-(methylamino)phenyl]sulfonyl-7-hydroxy-6,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-ethylbenzamide 4-methyl-3-[(2S)-1-oxo-3-phenyl-2H-1,2-benzodiazepin-6-yl]-5-propanoyloxypentanoic acid [5-(3-azidopropyl)thiophen-2-yl]methanol 1-[4-[[6-(methoxymethyl)pyridine-2-carbonyl]amino]phenyl]cyclopropane-1-carboxylic acid 6-[4-chloro-2-(hydroxymethyl)anilino]sulfanyl-3,5-dimethoxyphenol 2-cyclohexyloxy-4,6-diethoxybenzene-1,3-dicarbonitrile 4-chloro-2-methylsulfonylpyrimidine N-[6,7-dimethoxy-4-(oxolan-3-yl)quinazolin-2-yl]acetamide (4S,5R)-4-azido-5-fluoro-6,7-dimethoxy-1-[2-methyl-6-(4-phenylmethoxypiperidin-1-yl)pyrimidin-4-yl]-4,5-dihydro-3H-2-benzazepine N-[2-(4,4-difluoropiperidine-1-carbonyl)phenyl]-3H-benzimidazole-5-carboxamide 1-(6-methoxypyridin-3-yl)pyrrolidine-2,5-dione (5R)-3-benzylsulfanyl-2-methylidenespiro[7H-pyrrolo[3,4-b]pyridine-5,9'-xanthene] N-[4,5-dimethoxy-2-(phenylmethoxyamino)phenyl]-1H-pyrrole-3-carboxamide 5-(8-aminooctoxy)quinazoline-2,4-diamine 4-bromobenzenesulfonamide;ethane 2-methyl-6-[[5-(trifluoromethoxy)pyridine-3-carbonyl]amino]cyclohexane-1-carboxylic acid 2-[1,3-bis(methylamino)propyl]naphthalene-1,4-dione;ethane;ethanol [4-(methoxycarbonylamino)phenyl]sulfonylcarbamodithioic acid 1-(3,4-difluorophenyl)sulfonyl-N-methylpyrrolidine-2-carboxamide 7-azidooxy-4H-1,3-benzodioxine 6-[(3R,4S)-1-cyclohexyl-4-phenylpyrrolidine-3-carbonyl]-1H-pyrimidine-2,4-dione 3-(4-fluorophenyl)-N',2-dimethylbutanehydrazide ethane;3-(2,4,6-trimethylphenyl)-5H-imidazo[1,2-b]pyridazine (3E)-N'-[4-chloro-2-fluoro-5-[1-(oxan-2-yl)pyrazol-4-yl]phenyl]-2-methylidenepenta-3,5-dienimidamide 6-(4,5,7,8-tetramethyl-1-benzofuran-2-carbonyl)cyclohexa-1,3-diene-1-carboxamide 2-methyl-4-(1H-imidazo[4,5-f]quinolin-7-id-8-yl)-3-propan-2-yl-1H-pyridin-2-ol;platinum 4-(3,5-difluorophenyl)-1H-pyrrole-2,5-dione 2-(4-bromophenyl)-6,6-dimethyl-4H-1,3,5-triazine 2-[4-methyl-3,5-bis(prop-1-en-2-yl)phenyl]-N-(pyridin-2-ylmethoxy)acetamide 6-(3,5-dimethylanilino)pyridine-2,4-dicarbonitrile 5-[2-(methoxymethyl)phenyl]-2H-triazole-4-carbonitrile (1-azidoindazol-3-yl)-(2,5-dimethoxyphenyl)methanone N-(2,3-dimethylphenyl)-5,6,7,8-tetrahydronaphthalene-1-sulfonamide 5-(4-chlorophenyl)-N'-hydroxy-1H-pyrazole-3-carboximidamide N-[1,3-dimethyl-5-(trifluoromethoxy)pyrazol-4-yl]-7-(3-hydroxypentanoylamino)-2-oxochromene-3-carboxamide [4-(2,3-dihydropyrrol-1-yl)-2-phenylsulfanylphenyl]methylphosphane 3-[4-[(E)-2-(2,5-dimethylphenyl)ethenyl]anilino]chromen-2-one N-[5-(4-chlorophenyl)-1,2-oxazol-3-yl]-2-(1H-indol-3-yl)-2-oxoacetamide 3-[4,6-difluoro-5-(trifluoromethyl)pyridin-2-yl]cyclobutan-1-one 1-[(4aR,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-2-(2H-triazol-4-yl)ethanone 3-[(5R)-4,5-bis(ethenyl)-2-oxo-1H-imidazol-3-yl]-N-phenylazetidine-1-carboxamide 2-[(2Z,5S)-4-oxo-2-[(E)-3-phenylpropylidenehydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 5-bromo-1-methyl-3-[(E)-prop-1-enyl]indole 1-[2,6-di(propan-2-yl)phenyl]-3H-imidazole-2-thione N-(2-benzylsulfanyl-3,4,6-trihydroxyphenyl)sulfonylacetamide 2-(N,3-dimethyl-4-sulfoanilino)acetic acid 5-amino-4-[3-bromo-2-hydroxy-6-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 4-[(2,5-dibromothiophen-3-yl)methyl]benzonitrile [1-(azidomethyl)cyclobutyl]oxymethylbenzene (Z)-2,6,6,7-tetrafluoro-3,4-dimethylhept-4-enal;1,8,12-trimethoxy-14-oxatetracyclo[13.2.1.05,18.07,17]octadeca-2,4,6,9(18),10,16-hexaene 7,9-dimethoxy-2,3,4,6-tetrahydropyrimido[1,2-a]indole 1-[2-(2,5-dimethylpyrrol-1-yl)ethyl]-3-phenylsulfanylpyrrolidine 2,2-dimethyl-N-[6-(piperidin-4-ylmethoxy)pyridin-3-yl]pyrrolidine-1-carboxamide 2-[1-(3-fluoro-4-hydroxy-5-methoxyphenyl)ethyl]cyclohexan-1-one N-[2,6-bis(2-methoxyethoxy)phenyl]-5-propan-2-yl-1H-pyrrole-3-carboxamide 4-fluoro-3-[[(5-methylcyclohexa-1,3-dien-1-yl)amino]methyl]benzamide 5-[2,4-bis(aminomethyl)phenyl]sulfanyl-4H-1,3,4-thiadiazin-2-amine 1-(3,4-dichlorophenyl)-N'-[2-(4-ethylanilino)ethyl]methanediamine 5-(4-chloro-3-fluorophenyl)-2,3-dihydro-1H-indene 3-[(1Z)-2,4-dimethylpenta-1,4-dienyl]-6-ethoxybenzene-1,2-diol 2-methyl-N,N'-diphenylcyclopropane-1-carbohydrazide N-[(3R)-5,6-dimethyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]acetamide 3-[(2,6-difluorobenzoyl)amino]-1-ethynylindazole-4-carboxylate 1,2,3-trifluorobenzene;5-(1H-pyrazol-4-yl)-3-pyridin-4-ylcinnoline ethene;(7-ethylnaphthalene-1,4-diium-5-ylidene)azanide 2-(2,3-dihydroxypropoxy)isoindole-1,3-dione 2-[5-methyl-2-(trifluoromethyl)phenyl]acetonitrile;propane (6R)-7-[3,5-dimethyl-1-phenyl-2-sulfanylideneimidazole-4-carbonyl]-6-methyl-3-propanoyl-2H-[1,3]thiazolo[5,4-c]quinolin-4-one 3,5-bis(trifluoromethyl)benzoic acid;1-cyclopropylidene-4H-quinolin-7-ol 2-[(1E)-3,7-difluoroocta-1,6-dienyl]-6-hydroxybenzaldehyde 2-[4-methylsulfonyl-3-(trifluoromethyl)phenyl]-6H-1,3,5-triazine 2,4-dimethyl-3-phenylquinoline;ethane 2-(N-ethylsulfonyl-3-nitroanilino)propanoic acid 2-(benzenesulfinyl)-4,5-dihydro-1H-pyrrolo[3,2-d][1]benzazepin-6-one 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-6,8-difluoroquinoline 2-[(1R,5S)-6-(methylaminomethyl)-3-azabicyclo[3.1.0]hexan-3-yl]-N-(5-propan-2-ylpyridazin-3-yl)acetamide 4-[(6-cyclobutyl-2-methylpyrimidine-4-carbonyl)amino]benzoic acid [4-(5,7-dimethoxynaphthalen-1-yl)phenyl]-diphenylphosphane 3-[(6Z,8E)-10-ethylsulfonyl-6-methylundeca-2,4,7-trienyl]benzoic acid 1-[(2,5-difluorophenyl)methyl]-4-[5-(2-ethoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyridin-2-one [5-amino-7-(1H-indol-2-yl)imidazo[4,5-b]pyridin-3-yl]-[6-fluoro-8-(4-methoxyphenyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]methanone [(4-tert-butyl-2,3,5,6-tetrafluorophenyl)-dideuteriomethoxy]phosphane N-[2-(diethylamino)ethyl]-4-[3-[[1-[6-(trifluoromethyl)pyridin-3-yl]pyrrol-2-yl]amino]quinoxalin-2-yl]benzamide (3R)-N,N-dimethyl-1-[3-[1-(2-morpholin-4-ylethyl)benzimidazole-5-carbonyl]phenyl]piperidine-3-carboxamide 1-(2,3-dihydro-1H-inden-5-yl)-4-methoxypyrazolo[3,4-d]pyrimidine N-[(3,5-difluorophenyl)methyl]-6-propanoyl-6-azaspiro[2.5]octane-8-carboxamide (1R,2S)-3-[[2-(4-carbamimidoylanilino)-5-[4-methyl-3-(trifluoromethoxy)phenyl]pyrimidin-4-yl]amino]cyclopentane-1-carboxylic acid 1-(4-methoxyphenyl)-3,5-dipyridin-2-ylpyrrole-2-carbonitrile 2-(1H-benzo[e]benzimidazol-2-yl)-3,4-dihydropyridine N-(4-aminophenyl)benzenesulfonamide 3-(2-chloroacetyl)-5-methoxybenzoic acid ethane;2-methyl-5,6,7,8,9,10-hexahydrocycloocta[b]pyridine 4-[1,3-dihydroxypropan-2-yl(5,7-dimethoxyquinazolin-4-yl)amino]butylazanide N-[4-(benzylamino)pyridin-3-yl]-2-(1H-pyrrol-3-yl)acetamide 1-azidosulfanyl-2,3-bis(4-chlorophenyl)benzene (5S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-oxo-1,3-oxazolidine-5-carboxamide 3-(2,6-dimethylmorpholine-4-carbonyl)-N-[(E)-1-phenylethylideneamino]benzamide 6-amino-4-(2,5-difluoro-4-methoxyphenyl)-3-methyl-1H-pyridin-2-one N-[5,7-dihydroxy-8-(3-methoxypropylsulfanyl)naphthalene-2-carbonyl]acetamide 2-amino-N-(9,10-dioxoanthracen-1-yl)propanamide 1-[4-[2-(5,6-dimethylpyridin-3-yl)ethynyl]pyridin-2-yl]ethanone 5-(1H-indol-2-yl)imidazo[2,1-b][1,3]thiazole N-(4-azidobutyl)aniline N-(3,5-dichlorophenyl)-2-[1-[(Z)-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)methylideneamino]-5-sulfanyltetrazol-2-yl]acetamide N-(2,2-dimethyl-3H-1-benzofuran-6-yl)benzamide 6-[6,7-dimethoxy-1-(2-nitrophenyl)-3,4-dihydro-1H-isoquinoline-2-carbonyl]-N-ethylpyridine-3-carboxamide 3-[(2,4-dimethoxyphenyl)methyl]-5,6-dihydroxy-1H-pyrimidine-2,4-dione 2-[(2,4-diaminophenyl)diazenyl]phenol 4-[7-(3,5-dimethylphenyl)imidazo[1,2-a]pyridin-3-yl]pyrimidin-2-amine 3-[2-(1-cyclopentylethenylamino)phenyl]-2-propan-2-ylideneimidazolidine-4,5-dione [4-[[2-[[[(1S)-2,3-dihydro-1H-inden-1-yl]amino]methyl]-5-methoxyphenyl]methyl]-3-fluorophenyl]phosphonic acid 2-azido-1-(4-bromophenyl)piperazine 3-[4-(3,5-dimethylphenyl)piperazin-1-yl]cyclobutane-1-carboxylic acid 1-phenylspiro[1H-2-benzofuran-3,4'-piperidine] 3-[3,5-dichloro-4-[(4-chlorophenyl)sulfonylamino]phenyl]propanoic acid 4-amino-2-[(E)-4-[3,5-dimethoxy-N-(methylcarbamoyl)anilino]but-1-enyl]-6-morpholin-4-ylpyrimidine-5-carboxamide N-(3,3-dimethyloxan-4-yl)-2-fluoro-6-[methyl-[(5-methylfuran-2-yl)methyl]amino]benzamide 2-[(5,6-dimethylpyridine-3-carbonyl)amino]propanoic acid 2-[(3R)-1-(6-aminopyridine-3-carbonyl)pyrrolidin-3-yl]oxybenzonitrile 5-[3,6-difluoro-1-(2H-tetrazol-5-yl)indole-4-carbonyl]-N'-hydroxypyridine-2-carbohydrazide 3-(4-azidooxyphenyl)-2H-1,5-benzodioxepine 2-[1-(4,6-dichloropyrimidin-5-yl)ethoxy]-N,N'-dimethyl-6-morpholin-4-ylpyrimidine-4-carbohydrazide N-(2,5-dichlorophenyl)-N'-(6-methoxypyridazin-3-yl)-2-methylpropanehydrazide (2S)-N,1-dimethyl-6-[3-[4-[1-(5,5,8,8-tetramethylnaphthalen-2-yl)cyclopropyl]phenyl]propanoylamino]piperidine-2-carboxamide 6-[[2-[5-chloro-1-(3,4-dichlorophenyl)-3,6-dihydro-2H-pyridin-4-yl]benzoyl]amino]pyridine-2-carboxylic acid 4-[2,6-dichloro-3-(trifluoromethyl)phenyl]aniline 5-(4,6-dimethylpyrazolo[1,5-a]pyrazine-2-carbonyl)pyrrolidin-2-one 4-benzylsulfinyl-1,3,5-triazine 7-(5-chloropyridin-2-yl)oxy-N-cyclopropylsulfonyl-4,4a,5,6,8,9-hexahydropyrido[3,4-d]azepine-3-carboxamide 4-[[(Z)-1-amino-3,3-dimethylbut-1-enoxy]methyl]benzoic acid 3-(dimethylamino)-N-[6-ethyl-1-oxo-5-phenylmethoxy-2,3-dihydroinden-4-yl]propanamide 4-(2,6-dichlorophenyl)-1H-[1]benzothiolo[3,2-d]pyrimidine-2,5-dione N-ethyl-1,3-dimethoxy-2H-quinoxalin-2-amine 2-[4-(carbamoylsulfamoyl)-N-(2,4,6-trimethylphenyl)sulfonylanilino]propanoic acid 2-(4-ethylanilino)benzonitrile 2-[3-(4,5-dimethylpyrazol-1-yl)phenyl]sulfonylpropanoic acid 6-[1-(4-tert-butylphenyl)ethylamino]-1,3-dimethylpyrimidine-2,4-dione 3-(4-azidobutoxy)aniline 3,4-dibutyl-7,8-bis(ethenyl)naphthalene-2,6-disulfonic acid 2-[4-[(3S)-oxolane-3-carbonyl]piperazin-1-yl]sulfonylbenzaldehyde 3-(1-methylpyrazol-4-yl)sulfonylpyridine-2,6-dicarboxamide 1-(5,6-dimethylthieno[2,3-d]pyrimidine-4-carbonyl)-N-pyridin-3-ylpiperidine-4-carboxamide 2-[4-(3,5-difluorophenoxy)butyl]benzenesulfonic acid (5S)-5-butyl-2-[4-chloro-3-fluoro-5-(3,3,4,4,5,5-hexafluorocyclopenten-1-yl)phenyl]imino-5-methylimidazolidin-4-one (5S)-3,4-dibenzyl-5-[2-[4-(4-bromophenyl)piperazin-1-yl]ethyl]-1,3-oxazolidin-2-one 3-azido-2,4,6-trimethoxybenzoic acid (4aR,8aS)-2-[5-fluoro-3-methyl-6-oxo-1-[3-(trifluoromethoxy)phenyl]pyridazine-4-carbonyl]-10-propanoyl-4,4a,5,8a-tetrahydropyrazino[2,1-c][1,4]benzoxazin-1-one (2S)-2-[[4-[1-[4-(1,3-benzodioxol-5-yloxy)butanoyl]piperidin-4-yl]oxycyclohexanecarbonyl]amino]-3-(3-fluorophenyl)propanoic acid [(Z)-4-aminooxy-3,5-dimethylhex-3-enoyl]oxy-[4-[2-fluoro-6-(hydroxymethyl)phenyl]phenyl]borinic acid;ethane 2-(2,3,4,5-tetrahydrobenzo[g]quinolin-7-yl)ethanesulfinic acid 7-[2-(dimethylamino)ethylsulfanyl]-N-phenylquinoline-3-carboxamide 2-(2,4-dibromophenyl)-N-(1H-indol-5-ylmethylideneamino)-1H-benzimidazole-2-carboxamide 1-amino-2-[5-[6-(difluoromethyl)imidazo[1,2-a]pyridine-3-carboximidoyl]pyrimidin-4-yl]oxyethanol N-[(3R)-2,7-dioxoazocan-3-yl]-2-methoxy-5-[4-methoxy-3-(3-pyrrolidin-1-ylpropoxy)phenyl]benzamide 4-[(Z)-2-chlorobut-1-enyl]-5-ethoxycarbonylpyridine-3-carboxylic acid N-[3-(6-cyclobutyloxypyridin-2-yl)phenyl]acetamide 2-(4-methylphenyl)-5,6,7,8-tetrahydrothieno[3,2-b]azepine (2E,5S)-3-ethyl-5-[(4-methoxyphenyl)methyl]-2-[(Z)-(2-propan-2-yloxyphenyl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one 3-[2,3-bis(1H-indol-4-yl)imidazol-3-ium-4-yl]butanenitrile;bromide N-(2,3-dichlorophenyl)-7H-purine-8-carboximidate 2-[(6S)-3-tert-butylsulfanyl-5-methoxycarbonyl-8-oxo-5,6,7,9-tetrahydropyrido[2,1-c][1,4]oxazepin-6-yl]acetic acid 1-methyl-3,5-bis(trifluoromethyl)benzene;5-methylidenecyclohexa-1,3-dien-1-ol N-[2,4-dimethyl-5-(methylaminosulfanyl)phenyl]sulfanyl-1-phenylethanamine 2-methoxy-6-(5-methylthieno[3,4-b]pyridin-7-yl)sulfonylphenol 5-[5-[(3,3-difluoropyrrolidin-1-yl)methyl]pyridin-3-yl]-N-methanimidoyl-7-(2-methylphenyl)isoquinoline-3-carboxamide 5-chloro-4-[(2,2-dimethylpropanoylamino)methyl]-N-phenylthiophene-2-carboxamide 2-methylsulfanylthieno[3,4-d]pyrimidine-6-carboxamide 5-[(E)-6,8-dihydroxyoct-1-enyl]naphthalene-2-sulfonic acid N-[4-(diethylamino)-3,5-bis(trifluoromethyl)phenyl]acetamide 2-methyl-1-phenyl-3H-1,4-benzodiazepine 1-(azidooxymethyl)-2,4,5-trifluorobenzene 3-[(4-methylphenyl)sulfonylamino]piperidine-1-carboxylate 1-(2,4,6-trimethylphenyl)isoquinoline (4-methylpiperidin-1-yl)-[6-methyl-5-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidin-7-yl]methanone 7-methoxy-2-[(4-piperidin-1-ylsulfonylpiperazin-1-yl)methyl]quinazoline [5-fluoro-2-methyl-3-(2,3,4,5-tetrahydroindol-1-yl)phenyl]methanamine 7-(6-chloropyridazin-3-yl)-8-methoxy-1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazole 1-[6-(trifluoromethyl)cyclohexa-2,4-dien-1-yl]naphthalene [4-azidooxy-2,6-di(propan-2-yl)phenyl]urea 4-[(1R,2S)-2-methyl-6-oxocyclohexyl]benzaldehyde [3-(2H-benzotriazol-5-yl)phenyl]methanamine 6-hydroxy-3-[(2E)-4-methoxypenta-2,4-dien-2-yl]chromen-4-one 2-[4-(1H-indol-3-yl)butanoyl]pyrrolidine-2-carbonitrile (3S)-N-[(4,6-dimethylpyridin-2-yl)methyl]-1-(oxan-4-yl)pyrrolidine-3-carboxamide 4-[1-(4-methoxy-3,5-dimethylpyridin-2-yl)-2-phenylethyl]benzoic acid N-(6,7-dimethoxyquinazolin-4-yl)cyclopropanecarboxamide 3-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]benzoic acid 2-amino-N',N'-bis[(4-chlorophenyl)methyl]butanediamide N-[(6-imidazol-1-ylpyridin-3-yl)methyl]decanamide 2-[2,5-dichloro-N-(3-methylbutyl)anilino]decanoic acid 4-chloro-6,7,8-trimethylpyrrolo[3,2-g]quinazolin-9-amine 3-ethyl-1,2,4a,5-tetrahydropyrazino[2,1-c][1,4]benzoxazine 3-[(1S)-1-aminoethyl]-7-methoxy-1H-quinolin-2-one 2-[(2-ethylphenyl)carbamoylamino]-N,3,5,6-tetramethylbenzamide 1-(azidomethyl)-N,N'-bis[2-(trifluoromethoxy)phenyl]cyclopropane-1-carboximidamide 4-[[(1,6-dimethylpyrazolo[3,4-b]pyridine-5-carbonyl)amino]methyl]benzoic acid 3-[(2,6-dioxopiperidin-3-yl)carbamoylamino]-N-methoxy-4-methylthiophene-2-carboxamide 1-[[4-(trifluoromethyl)phenyl]methylamino]azetidine-2-carboxylate 3,5-diphenyl-4-[[(E)-3-thiophen-2-ylprop-2-enoyl]amino]pyrrole-1-carboxamide 2-[4-azido-5-(2-methoxyphenyl)pyrimidin-2-yl]sulfanylethanol 3-methyl-4-[(2R)-6-[4-[2-(5,7,8,11-tetrahydro-[1]benzoxepino[4,3-d]pyrimidin-4-ylamino)ethyl]piperazin-1-yl]hexan-2-yl]sulfanylbutanenitrile 1-[4-(azidomethyl)phenyl]sulfanyl-9H-fluorene 1-(3,5-dimethylphenyl)-3-[4-methoxy-2-(4-oxo-3H-quinazolin-2-yl)butan-2-yl]urea 4-azido-6,8-dichloro-2,3-dihydrochromene 2-[2,6-bis(2,4,4-trimethylpentan-2-yl)phenoxy]-N-[(Z)-1H-indol-3-ylmethylideneamino]acetamide 2-[(1S)-1-(4-ethylcyclohexa-2,4-dien-1-ylidene)propoxy]phenol 7-(diethylaminomethyl)-N,N-bis[(4-nitrophenyl)methyl]-3H-benzimidazole-5-sulfonamide 1-(3-chloro-2,4-dimethylphenyl)-N-[5-(furan-2-yl)-1H-imidazol-2-yl]ethanimine 1-[4-chloro-2-(3-morpholin-4-ylpropoxy)phenyl]-N-methylcyclohexan-1-amine (5E)-2-imino-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidin-4-one N-[(2,3-dimethoxyphenyl)methyl]-4-oxo-3H-quinazoline-7-carboxamide 2-[4-(3-fluorophenoxy)-2-nitrophenyl]-1,3-benzothiazole 2-amino-9-[(4R,5S)-4-hydroxy-5-methoxyoxolan-2-yl]-1H-purin-6-one;sulfuric acid 2-(4-aminophenyl)pyridine-4-carboxamide 5-[2-(4-aminophenoxy)ethyl]-1,3-thiazolidine-2,4-dione 4-chloro-3-[1-(2,6-dimethylphenyl)ethoxy]benzaldehyde 2-chloro-4-phenylsulfanylbenzonitrile;3,4-dihydroxypenta-1,4-dien-3-olate;methanol;uranium(2+) 1-[4-hydroxy-6-(methyliminomethyl)-2,3-dihydroindol-1-yl]ethanone 2-chloro-3-[[(4-ethylphenyl)methylideneamino]methyl]aniline 4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1,3-dicarboxamide N-[3,5-bis(trifluoromethyl)phenyl]-1-cyano-2-[6-[(4Z,8E)-8-[(2,3-dichlorophenyl)carbamoylamino]tetradeca-4,8,10-trienoxy]pyridin-3-yl]cyclopropane-1-carboxamide 2-azidooxy-1,3,5-triethylbenzene 2-(3,4,5-trimethoxyphenyl)heptan-4-ol 4-(3-aminophenyl)piperazine-1,4-dicarboxylic acid 6-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]-7,8-dihydroquinoline-5,8a-dione N-[2-[6-chloro-1,3-dimethyl-4-oxo-7-(trifluoromethoxy)quinazolin-2-yl]sulfanylethylidene]acetamide 2-amino-1,4-dihydroindeno[1,2-c]pyrazole-5-carboxylate 2-amino-9-[4-(2,3-dihydro-1H-inden-5-yl)cyclopenta-1,3-dien-1-yl]-8-propoxypurin-6-amine (3-methoxy-4-propylphenyl)-piperidin-1-ylmethanone N-butanoyl-4-hydroxyimino-4-(trifluoromethoxy)butanamide;3-chloro-2,6-dipropyl-5H-pyrimido[5,4-d]pyridazin-7-one [3-[(6-aminopyridin-1-ium-2-yl)methoxy]azetidin-1-yl]-phenylmethanone (3aR,6aS)-2-[4-chloro-3-(trifluoromethyl)benzoyl]-3a-(hydroxymethyl)-1,3,4,5,6,6a-hexahydrocyclopenta[c]pyrrole-3-carboxylic acid 2-[4-(5,6-dihydronaphthalene-1-carbonyl)phenyl]-1,3-benzoxazole-4-carboxamide 2-[4-(5-azido-3-phenylpyrazin-2-yl)oxybutanoyl]benzonitrile [1-ethoxy-2-(4-nitrophenyl)propan-2-yl]urea 2-[4-(dimethylamino)phenyl]-N-[3-[2-oxo-2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-ylamino)ethoxy]phenyl]acetamide 1-[4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]phenyl]pyrrolidine 2-[3-(azidomethyl)-5-cyclopropylphenyl]-4,6-bis(trichloromethyl)pyrimidine 3-ethoxy-N'-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(2H-tetrazol-5-yl)amino]propanehydrazide [6-(2,4-dichlorophenyl)-4-(furan-2-ylmethoxyimino)pyridin-3-ylidene]-oxoazanium 5-azido-6-[2,3-bis(4-chlorophenyl)pyridin-4-yl]imidazo[1,2-a]pyrazine 6-amino-2-butoxy-9-[(4R)-5,7-dihydroxy-8-methyl-3,4-dihydro-1H-isoquinolin-2-yl]purine-8-carboxamide 5-azido-2,4-bis(2-methoxyphenyl)-1H-pyrazol-3-one 3-(4,5-dihydro-1H-pyrazol-5-yl)quinoline 1-N,3-N-bis(2-ethoxyphenyl)benzene-1,3-dicarboxamide 2-[1,3-bis(ethenyl)cyclopenta-1,4-dien-1-yl]propane-2-sulfonic acid (2S,6R)-10-hydroxy-8-methoxycarbonyl-9-oxo-7-phenylmethoxy-5-thiapentacyclo[10.8.0.02,6.07,11.013,18]icosa-1,3,7(11),8,12,14,16,19-octaene-4-carboxylic acid 2-[[7-chloro-5-(4-hydroxyphenyl)sulfonyl-3-methoxypyrazolo[1,5-a]pyrimidin-2-yl]amino]ethanethiol 1-bromo-3-(4,4-dimethylpent-1-en-2-yl)benzene;ethane 5-(cyclohexyloxymethyl)-1-[4-[2-(2,6-dichlorophenyl)ethylamino]cyclohexyl]indazole-3-carboxylic acid;hydrochloride 4-(azidomethyl)-1-(2,5-dichlorophenyl)sulfanylpiperidine 6-ethyl-N-[1-(4-fluoro-3-methoxyphenyl)piperidin-4-yl]pyridazine-3-carboxamide N-[4-(benzylamino)-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]-1H-pyrrole-3-carboxamide 6-(4,4,5,5-tetramethyl-1H-imidazol-2-yl)-1H-benzimidazole 4-(azidooxymethyl)-2-[2,6-difluoro-3-(trifluoromethoxy)phenyl]pyridine (2S)-6,8-dimethoxy-N-[5-methyl-1-[[6-(trifluoromethyl)pyridin-3-yl]methyl]pyrazol-4-yl]-2-propan-2-yl-3,4-dihydro-1H-isoquinoline-2-carboxamide (2R)-1,3-dimethyl-N-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl)-2,3-dihydroindole-2-carboxamide;hydrochloride [3-(6-methoxycarbonylnaphthalen-2-yl)phenyl]-oxoazanium 4-[2,3-difluoro-4-[(E)-hept-1-enyl]phenoxy]phenol 1-(3,4-dihydronaphthalen-2-yl)-N-[[4-(2,3-dimethoxyphenyl)sulfonylpiperazin-1-yl]methylsulfanyl]-7-ethoxy-6-fluorobenzimidazole-5-carboxamide [4-[4-(2,6-diphenyl-1,2-dihydro-1,3,5-triazin-4-yl)-1-methylpyridin-1-ium-2-yl]-3-methylphenyl]-methylideneborane 7-butanoyl-6-(2,4-difluorophenyl)-3-propylsulfanyl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one (4-benzylpiperazin-1-yl)methanesulfinate 2-[7-methyl-3,5-bis(phenylmethoxy)-4H-oxazin-6-yl]propanoic acid [4-(3,3-dimethylpentan-2-ylidene)-5,6-dihydroxycyclohexa-2,5-dien-1-ylidene]-(dimethylamino)azanium N-ethyl-2-[4-(3-phenylpropanoyl)piperazin-1-yl]pyrimidine-5-carboxamide N-[(3S,4R)-1-tert-butyl-3-[[1-cyclohexylethoxy(3-fluorophenyl)methyl]carbamoyl]piperidin-4-yl]-5-(2,6-difluorophenyl)-1H-pyrazole-3-carboxamide 5-chloro-N-[3-(cyclopropylmethoxy)phenyl]sulfanyl-2,4-difluoroaniline 3-[(4Z)-4-ethenylhepta-2,4,6-trien-2-yl]benzonitrile (2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methoxy]cyclohexanecarboxamide 2-[3,5-dimethyl-N-(2-oxopropyl)anilino]decanoic acid N-[(4S,5R)-3-methyl-6-oxo-2-pyridin-3-yl-1,2,4-triazin-5-yl]pentanamide 2-[3-fluoro-5-(trifluoromethyl)phenyl]sulfanyl-N-[5-(6-hydroxypyridin-2-yl)-1,3,4-thiadiazol-2-yl]acetamide (E)-N-[5-[2,3-bis(ethynyl)phenyl]pentanoylamino]-4,5-dimethoxy-6-oxohex-2-enamide 6-[2,3-dihydroxypropyl(phenacyl)amino]-4-hydroxynaphthalene-2-sulfonic acid (2R,5S)-1-azido-5-phenylpyrrolidine-2-carboxylic acid 5-[2-(4-chloroanilino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]pyridine-3-carboxylic acid 1-[(2,4-dimethylphenyl)methyl]-3-(diphenylcarbamothioylamino)thiourea 4-amino-2-[(3-ethoxy-1H-pyrazol-5-yl)methylsulfanyl]-1H-pyrimidin-6-one N-[1,3-bis(4-bromophenyl)propan-2-ylideneamino]acetamide 2-amino-5,6-dimethyl-4-[3-(trifluoromethyl)phenyl]pyridine-3-carbonitrile 5-ethyl-3-[[(4R)-1-methylpyrrolidine-2-carbonyl]amino]thiophene-2-carboxylic acid 2-(2-methoxyethyl)-3,4-dihydro-1H-isoquinoline-7-carboxylic acid [(Z)-3-amino-4,4,5,7,7-pentamethyloct-6-enylidene]azanium;(5Z)-5-ethylidene-2H-cycloocta[b]pyridine N-azido-3-(2,6-dichlorophenyl)-1,2,4-triazin-5-amine 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]ethanethiol N'-[5-(3,5-dichloropyridin-4-yl)sulfanyl-1-(cyclopropylmethyl)-2-(trifluoromethoxy)benzimidazol-4-yl]ethane-1,2-diamine 2-(5-fluoro-2,3-dihydroindol-1-yl)benzoate N'-[(Z)-1H-indol-3-ylmethylideneamino]-2-[4-methoxy-5-methyl-2-propan-2-ylsulfanyl-3-[2-[(2,2,2-trifluoroacetyl)amino]ethyl]phenoxy]ethanimidamide 3-benzyl-7-[(2,6-dichlorophenyl)methyl]-1-(3,5-difluoro-4-hydroxybutanoyl)-8,9-dihydropyridazino[3,4-e]indole-2,4-dione N-[3-chloro-4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,11-tetraen-3-ylsulfonyl)phenyl]acetamide [2-methyl-4-[4-[4-[(2E,4Z)-5-methylidenehepta-2,4,6-trien-3-yl]cyclohexyl]butanoyl]phenyl]boronic acid 3-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide 2-[4-(1H-pyrrol-2-yl)phenyl]acetonitrile 2,4-dibutyl-6-[2-(1H-imidazol-5-yl)ethyliminomethyl]phenol (6S,9aS)-N-benzyl-8-[(3-chlorophenyl)methyl]-2-ethyl-4,7-dioxo-6-propan-2-yl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide 1-[3-(1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]-2-azabicyclo[3.2.0]heptane 4-[4-(aminomethyl)phenyl]-2-propoxybenzaldehyde 5-[1-(1H-benzimidazol-2-ylmethyl)triazol-4-yl]-3-piperidin-1-yl-1,2,4-oxadiazole;dihydrochloride 4-(6-methoxypyridin-3-yl)-N,N-dimethylaniline N-[4,5-dichloro-2-(hydroxymethyl)phenyl]-3-[2-[1-(cyanomethyl)cyclopropyl]pyridin-4-yl]-1-ethoxyisoquinoline-6-carboxamide 2-[(5-fluoropyridin-3-yl)amino]-N-[6-(4-methoxyphenyl)pyridazin-3-yl]acetamide [5-azidooxy-2-methyl-3-(4-phenoxybutoxy)pentan-2-yl]benzene 5-cyclopropyl-4-[7-(1,2,4-triazol-1-yl)pyrido[3,4-b]pyrazin-5-yl]oxypyridine-2-carboxamide (3E,5Z)-3-benzylidenehepta-1,5-dien-4-amine 4-amino-2-fluoro-1,5-dimethylpyrrolo[2,3-b]pyridine-6-carboxamide 2-methyl-4,6-bis(methylamino)benzo[de]isoquinoline-1,3-dione 3-(1,5-dimethylpyrazole-4-carbonyl)-2-methylidenespiro[1H-indole-3,4'-piperidine] (2S)-3,6-diamino-N-[2-oxo-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methylamino]ethyl]hexanamide;dihydrochloride [2-[(3S)-3-amino-3-hydroxypropyl]sulfonylphenyl]methanol 2-[1-(5,6,7,8-tetrahydro-1H-1,4-diazocin-2-yl)piperidin-3-yl]quinazoline [5-chloro-2-(cyclohexyloxyamino)phenyl]methanethiol 1-ethenyl-3,5-dimethoxybenzene;2-[(4-ethoxyphenyl)iminomethyl]phenol 5-ethyl-1-(2,3,4,5,6-pentafluorophenyl)pyrrole-3-carboxylic acid 3-hydroxy-5,6-dimethyl-N-[(1R)-1-phenylethyl]pyrazine-2-carboxamide 5-[(2,3-dichlorophenyl)methyl]-1H-indazole 7-[2-(5-fluorothiophen-2-yl)sulfanylacetyl]-N,3,4a,5,6,8,9,10,11,12,12a-decahydro-1H-pyrido[3,4-d]azecine-2-carboxamide (Z)-N'-[2-(3,6-dihydro-2H-pyran-4-yl)quinazolin-4-yl]ethene-1,2-diamine 5-(3-chloro-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonyl)-N-methylfuran-3-carboxamide 1-(3,4-dihydro-1H-isoquinolin-2-yl)-5-[[(1R,2S)-2-hydroxycyclohexyl]amino]sulfanylpentan-1-one (5R)-3-azido-7-[3,4-dimethoxy-2-(2-phenylethylcarbamoylamino)phenyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-5-carboxamide 4-(azidomethyl)-1,3,5-triphenylpyrazole 2-methyl-N-(1-pyrimidin-4-ylpiperidin-4-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine;dihydrochloride 3-[(1S,5R)-1-tert-butyl-2-azabicyclo[3.2.0]heptan-2-yl]aniline 4-chloro-N-(2,6-dimethylphenyl)-3-[2-oxo-2-propoxy-2-(pyrazin-2-ylamino)ethoxy]benzenesulfonamide N-(4-amino-1,3,5-triazin-2-yl)-4-fluorobenzamide 2-[4-(2,6-difluorophenyl)butyl]-3H-isoindol-1-one 2-N-(5,8-dimethoxy-4-oxo-3H-quinazolin-6-yl)benzene-1,2-dicarboximidamide 1-(4-bromophenyl)sulfonyl-3,5-difluorobenzene 4-[[[(2R)-butan-2-yl]amino]methyl]-2-chlorophenol N-(4,5-diaminopyridin-2-yl)hexanamide 3-[4-(2,2-difluoropropyl)phenyl]-8-ethyl-1-methoxychromeno[4,3-c]pyrazole 4-methyl-N-phenyl-3-[2-(trifluoromethoxy)pyridin-4-yl]aniline 1-[(3R,4S)-4-(hydroxymethyl)-2,2-dioxo-7-phenyl-1-oxa-4,6-diazaspiro[2.5]octan-3-yl]-3-propan-2-ylurea (2S)-1,5-dimethyl-2,6-diphenylpiperidine;ethane (3S)-N-[4-amino-2-chloro-6-[[2,5-difluoro-4-(1H-pyrazol-4-yl)phenyl]methoxy]pyrimidin-5-yl]oxolane-3-carboxamide N-[2-[3,4-bis(ethenyl)phenyl]propan-2-ylideneamino]-N',N'-dimethylmethanediamine [4-(4-methylcyclohex-3-en-1-yl)phenyl]boronic acid 4-[(3S)-1-[3-(2,6-difluorophenyl)propanoyl]piperidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-6-one N-[(Z)-4-aminobut-2-enyl]-5-chloro-1,3-benzothiazol-2-amine 3-[5-bromo-4-(methoxymethyl)-1,2,4-triazol-3-yl]piperidine;hydrochloride 4-tert-butyl-2-(1,3-dioxolan-2-yl)phenol 2-[3-(4-phenylphenyl)carbazol-9-yl]benzene-1,4-dicarbonitrile N-[(6-amino-2,4-dimethylpyridin-3-yl)methyl]-5-chlorothiophene-3-carboxamide (5-fluoropyridin-3-yl)-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone 2-(3-methoxyphenyl)-N-[4-[2-(4-methylpiperazin-1-ium-1-ylidene)hydrazinyl]phenyl]pyrimidin-4-amine 1-(2,4-diaminophenyl)butan-1-one (5-chloropyrimidin-2-yl)-[3-methoxy-4-(1H-pyrrol-2-yl)phenyl]methanone 3-azido-2,6-difluorobenzenesulfonic acid 2-(3,4-dimethoxyphenyl)-5-[2-(4-methylpiperazin-1-yl)ethoxy]pyrido[3,4-b]pyrazine 1-[6-chloro-3-(morpholine-4-carbonyl)quinolin-7-yl]-2H-pyridine-3-carboxamide 2-bromo-N-[2-methyl-4-[(2-methylphenyl)diazenyl]phenyl]-N-(3-nitrophenyl)benzamide 1-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-3-[2-(1H-indol-3-yl)ethyl]urea N-[2,5-dichloro-3-(2-nitrobutoxy)phenyl]acetamide 5-[4-azido-6-(2,3-difluorophenyl)pyridin-2-yl]-1H-pyridazin-6-one 5-amino-N-[1-(2-methoxyethyl)pyrazol-3-yl]-6H-thieno[3,2-b]pyrrole-4-carboxamide;1-pyrrolidin-1-ylpropan-1-one (2S)-4-[(4-cyanophenyl)methyl]pyrrolidine-1,2-dicarboxylic acid 1-[4-(dimethylamino)phenyl]-3-(5,6-dihydronaphthalen-2-yl)urea N-(2,3-dihydroxypropyl)-2-[4-methoxy-3-[3-[6-methoxy-5-(trifluoromethyl)pyridin-2-yl]prop-1-ynyl]phenyl]acetamide 3-(1-azidopropan-2-yl)-5-propoxyphenol (5S,7R)-N-[1-(2-chlorophenyl)cyclopropyl]-2-(3-methoxypropyl)-5,7-dimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carboxamide 1-[2-(1,3-dihydroisoindole-2-carbonyl)phenyl]ethanone (2R)-3-[2-chloro-4-[4,5-dimethyl-2-oxo-1-[4-(trifluoromethoxy)phenyl]pyrrolidine-3-carbonyl]phenoxy]-N-formyl-2-hydroxypropanamide N-[2,4-dimethyl-5-[4-(trifluoromethoxy)phenyl]pyrazol-3-yl]formamide;N'-ethyl-N-[2-(6-fluoroimidazo[1,2-a]pyridin-2-yl)-8-azabicyclo[3.2.0]heptan-3-yl]ethane-1,2-diamine [3-(cyclopropylmethoxy)phenyl]-methyl-(naphthalen-1-ylmethylidene)azanium 3-(5-chloropyridin-2-yl)-1,5-dimethylpyrazole (2R,3S)-1-[5-chloro-6-(difluoromethoxy)pyridine-3-carbonyl]-N-[(4-methyloxan-4-yl)methyl]-2-phenylpiperidine-3-carboxamide 2-(4,6-dimethoxypyrimidin-5-yl)-3H-pyrido[2,1-f][1,2,4]triazin-4-one 3-[2-[3-chloro-4-[(2,4-difluorophenyl)methoxy]anilino]quinazolin-6-yl]cyclohexane-1-carboxylic acid 5-fluoro-7,8-dimethyl-1H-pyrano[2,3-c]pyridine-2-thione 3-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2-methoxybenzamide 4-N-cyclohexyl-2-(1H-indol-3-yl)pyrimidine-4,5,6-triamine (3E,5Z)-1-butyl-4-N-[2-(diethylamino)ethyl]-7-(naphthalen-1-ylmethoxy)hepta-3,5-diene-3,4-diamine 4-[5-(3-bromophenyl)-6H-1,2,4-oxadiazin-3-yl]benzoic acid 1-[3,4-di(butan-2-yl)phenyl]isoquinoline;ethane (Z)-3-(4,5-dihydro-1H-imidazol-2-ylamino)-1-[8-fluoro-2-(pyridin-3-ylmethyl)-6H-benzo[c]chromen-5-yl]prop-1-en-2-ol 1-[3-(azidomethyl)-5-chlorophenoxy]naphthalene 4-tert-butylbenzenesulfonamide;cyclohexane;ethene 2-[(6R)-6-azido-5,6,7,8-tetrahydronaphthalen-2-yl]ethanol 3-[[(Z)-2,4-difluoro-1H-indole-6-carbonyl]amino]-5-methylsulfonylbenzoic acid 4-methoxy-7,8-dihydrothieno[2,3-f][1]benzothiole N-[2-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-3H-benzimidazol-1-ium-5-ylidene]-2-[4-(trifluoromethyl)phenoxy]acetamide 1-[5-(aminomethyl)cyclopenta-2,4-dien-1-yl]-3-naphthalen-2-ylpropane-1,2-dione 6-chloro-2-[2-fluoro-5-(1,3-thiazol-4-yl)phenyl]quinazoline-7-thiol 6-(methoxymethyl)-5-(2-quinolin-3-ylpropanoylamino)naphthalene-1,7-disulfonic acid 4-[4-(3,4-dihydro-1H-isoquinoline-2-carbonyl)piperidin-1-yl]oxane-4-carbonitrile 2-[3-amino-4-(3,5-dimethylphenyl)butanoyl]oxyacetic acid N-[(1S,2R)-2-azidocyclopentyl]-2-phenylethanesulfonamide N-[(Z)-(2,3-dihydroxyphenyl)methylideneamino]-2-pyridin-1-ium-1-ylacetamide 3-[(1S)-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylimidazolidine-2,4-dione [1-(5,6-dimethylpyrrolo[2,3-b]pyridine-1-carbonyl)piperidin-4-yl]urea 4-[[4-(5-azidopyrimidin-2-yl)piperazin-1-yl]methoxy]benzonitrile 4-chloro-N'-cyclopropylbenzenecarboximidamide (Z)-N'-[2-(3,4-dimethoxyphenyl)ethyl]-4-iminopent-2-enimidamide N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-prop-2-enylhexadecanamide N-[(4-fluorophenyl)methyl]-2-(3-hydroxy-3-methylbutanoyl)-5,7-dihydro-4H-furo[2,3-c]pyridine-6-carboxamide 6-[2-(hydroxymethyl)phenyl]-2H-1,4-benzothiazin-3-one 2-[2,4-dichloro-5-[[3,6-dioxo-2,4-bis(phenylmethoxy)cyclohexa-1,4-dien-1-yl]amino]phenoxy]acetic acid 3-(4-tert-butylphenyl)-5-chloro-2,3-dihydro-1H-pyrazole N-[2-methyl-1-(4-pyrazol-1-ylphenyl)propan-2-yl]-5-methylsulfanyl-4-(trifluoromethyl)pyrimidin-2-amine 2-[[5,6-dichloro-1-(4,4,4-trifluorobutyl)benzimidazol-2-yl]sulfanylmethoxy]-3H-pyrido[2,3-d]pyrimidin-4-one 4-[3-cyclopropyl-5-[(2R)-1,1,1-trifluoropropan-2-yl]-2H-pyrrol-4-yl]pyridine;ethane 2-[(2,6-dichlorophenyl)methyl]-4-oxo-3H-quinazoline-8-carboxylic acid 4-[1-(4-bromophenoxy)ethyl]-5-methylfuran N-(1,2-dihydronaphthalen-1-yl)naphthalene-2-carboxamide 3-[4-(5,7-dimethoxyquinolin-4-yl)piperazin-1-ium-1-ylidene]propanenitrile (2R,3S)-2-[(2-bromophenyl)methyl]-1-ethoxycarbonylpiperidine-3-carboxylic acid 6-bromo-2-(1,3,5-trimethylpyrazol-4-yl)quinoline N-[(2,4-difluorophenyl)methyl]-7-hydroxy-6-(oxan-4-yl)spiro[1,3-dihydroquinoline-2,4'-piperidine]-1'-carboxamide 2-azido-4,5-diethoxytriazole 5-benzylsulfonyl-2,4-dichlorobenzenesulfonic acid 4-(3,6-dihydro-2H-pyran-4-yl)-1-methoxy-9,10-dioxoanthracene-2-carboxamide 1-[2,5-difluoro-4-(trifluoromethyl)phenyl]-N'-hydroxypyrazole-3-carboximidamide 4-[[(3R)-oxolan-3-yl]oxymethyl]-3,5-dihydro-2H-1,4-benzoxazepine N-[3-(2,4-dichlorophenyl)-3-hydroxypropyl]-6-fluoro-3-methylpyridine-2-carboxamide 5-(1-acetylpiperidine-4-carbonyl)-N,N-dimethyl-2,3-dihydrofuro[3,2-b]pyridine-7-carboxamide (1Z)-5,5-dimethyl-2-methylidene-1-[2-(oxan-4-yloxy)ethyl]-3H-imidazo[1,2-a]imidazole 5-(3,4-difluorophenyl)sulfonyl-N'-hydroxy-1H-1,2,4-triazole-3-carboximidamide 3-(1H-pyrrolo[2,3-c]pyridin-2-ylmethylidene)pentan-2-one 4-(1H-indol-6-yl)thiophene-2-carboxylate 4-amino-2-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-2-yl)phenol 4-(2,3-dihydrothieno[3,2-c]pyrazole-5-carbonyl)-2-fluorophenol 2,4-dimethyl-N-[(1S)-1-phenylethyl]imidazo[2,1-b][1,3]benzothiazol-7-amine 3-[[2,6-dimethyl-4-[5-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyridin-3-yl]phenyl]methyl]pyrrolidine-2,5-dione ethane;1-methyl-3-(2,2,5-trimethyloxolan-3-yl)benzimidazole 2-(3,5-difluorophenyl)-3-(4,6-diphenyl-1,3,5-triazin-2-yl)quinoxaline 5-chloro-2-fluoro-4-[6-(oxan-3-yl)-1H-benzimidazol-2-yl]phenol 1-[3-(2,5-difluorophenyl)-3,4-dihydropyrazole-2-carbonyl]-2-methylpyrrolidin-2-one 1-(4-azidobutyl)anthracene 3-[6-[(5,7-dimethylquinolin-2-yl)amino]pyridin-3-yl]benzonitrile 2-[4-[(E)-but-1-enyl]phenyl]-6,7-dimethoxy-3H-quinazolin-4-one 2-ethyl-4-(3,3,5-trimethylpentan-2-yl)aniline 4-(1,3-benzothiazol-2-yl)-5-imino-1-[2-(methoxyamino)phenyl]-2H-pyrrol-3-ol (7R)-3-[(2S)-butan-2-yl]-9-[2-(6,7-difluorobenzimidazol-1-yl)acetyl]-1,9-diazaspiro[4.5]decane-2,8-dione [3-[1-(benzenesulfonyl)-4-chloroindol-2-yl]phenyl]azanium 5-azido-3-(2,6-dimethylpyridin-4-yl)oxypyridine 2-amino-N-[(3S,4R)-1-[1-[(4-fluorophenyl)methyl]indazole-7-carbonyl]-4-hydroxypyrrolidin-3-yl]pyrimidine-5-carboxamide 4-[5-methyl-6-[2-(1,3-thiazol-5-yl)pyridine-4-carbonyl]pyrimidin-4-yl]morpholin-3-one 1-ethyl-5,7-dimethoxyimidazo[4,5-c]quinoline 1-[4-[(5,8-dichloronaphthalen-2-yl)sulfonylamino]naphthalen-1-yl]-3-propan-2-ylurea 3-[2,5-difluoro-4-[[3-fluoro-2-methyl-6-[methyl-(5-methylpyrimidin-2-yl)amino]phenyl]sulfamoyl]phenyl]propanoic acid 4-[3-(dimethylamino)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl]morpholin-3-one 4-(5,6,7,8-tetrahydronaphthalen-1-yloxy)butanoic acid 2-[(4-aminophenyl)-hydroxymethyl]-5,6,7,8-tetrahydronaphthalen-1-ol N'-(2,3-dihydroindol-1-yl)sulfonyl-3-[4-(2,2,2-trifluoroethoxymethyl)phenyl]benzenecarboximidamide 4-[3-amino-6-(2,5-dimethoxyphenyl)pyrazin-2-yl]benzaldehyde;N-methylmethanamine 2-[4-(difluoromethyl)pyrazol-1-yl]-N-[1-(1,3-thiazol-4-yl)ethenyl]cyclohexane-1-carboxamide (Z)-1,1-difluoro-4-imino-4-[2-methoxy-5-(trifluoromethylsulfanyl)phenyl]but-2-en-2-amine 4-[5,6-bis(trichloromethyl)pyridin-2-yl]-1H-indole ethane;4-N-[3-[(1E,3Z)-hexa-1,3-dienyl]cyclopenta-2,4-dien-1-ylidene]cyclohexane-1,4-diamine N-[[(2S,4R)-1-[1-(6H-pyrrolo[3,2-f][1,7]naphthyridin-9-ylmethyl)piperidine-4-carbonyl]-4-(trifluoromethoxymethyl)pyrrolidin-2-yl]methyl]ethanesulfonamide N-(4-hydroxybutyl)-2,6-dimethoxybenzamide 3-benzamido-N-(5,6-difluoro-2-methyl-1H-indol-3-yl)benzamide;ethane (1R)-3,6,9,9-tetramethylfluoren-1-amine 2-(2,2-dimethylbutanoyl)benzaldehyde N-(5-amino-2,3-dihydroindole-1-carboximidoyl)-4-cyanobenzamide;6-ethyl-2-[(4-propanoylmorpholin-3-yl)methoxy]pyridine-3-carboxylic acid 5-[(2E,4Z)-hepta-2,4,6-trien-3-yl]oxy-1H-pyridine-2-thione 4-(methoxymethyl)-N,2,3,5-tetrahydro-1H-pyrido[4,3-b]indole-8-carboxamide 2-methylpropane;7-(3-methylpentanoyl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-one 7-(4-methylpiperazin-1-yl)-3,8-diphenyl-5H-pyrido[2,3-d]pyridazine 7-cyclopentyl-2,6-dimethoxypurine 1-(4,5-dimethyl-2-phenyl-3H-pyrrol-6-yl)ethanone 1-N,3-N,5-trimethyl-4-propanimidoylbenzene-1,3-diamine 2-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)piperidin-2-yl]cyclopentan-1-one 5-[4-(1,3-diazepan-2-yl)phenyl]-8H-pyrido[4,3-d]pyrimidin-7-one 2-(4-tert-butylphenyl)-1-[2,6-dichloro-4-(hydroxymethyl)phenyl]ethanone N-[(E)-1-aminopropylidenecarbamothioyl]benzamide 2,4-dioxospiro[1H-pyrido[3,4-d]pyrimidine-8,3'-cyclobutane]-5-carboxylic acid 4-[3,5-ditert-butyl-2-(cyanomethoxy)phenyl]sulfonylmorpholine 6-benzyl-4-(ethoxymethyl)-N,8-dioxo-2,3,5,6,7,9-hexahydro-[1,3]thiazolo[3,2-a][1,3]diazepine-7-carboxamide 2-[[(3,4-dichlorophenyl)sulfonylamino]methyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide 2-[4-(1,3-benzothiazol-5-ylmethyl)piperazin-1-yl]ethanol 2-(3,5-dimethylbenzene-6-id-1-yl)quinolin-8-ol;6H-cyclopenta[b]pyridin-4-ide;iridium 6-[[(3R,4S)-1-(5-fluoropyrimidin-2-yl)-3-methoxypiperidin-4-yl]amino]pyridazine-3-carbonitrile;hydrochloride 3-amino-1-(2,5-dihydroxyphenyl)naphthalene-2-sulfonic acid N-[2-(1,3-dioxol-4-yl)ethyl]-5-methoxy-6H-indeno[1,2-c]quinoline-9-carboxamide N-[(6-methoxynaphthalen-1-yl)methyl]-5H-pyrrolo[3,2-d]pyrimidine-4-carboxamide 1-(dichloromethyl)benzene;palladium(2+);1,2,3,4,5-pentafluorobenzene-6-ide 2-[(E)-but-1-enyl]-3,4-dimethoxy-N,N-bis[4-(trifluoromethoxy)phenyl]aniline 2-bromo-6,7-dimethoxy-N'-(2-phenylethyl)quinoline-4-carboximidamide 4-(5,6,7,8-tetrahydroquinazolin-2-ylamino)phenol 2-(3-chlorophenyl)-N-[5-methyl-4-(piperazine-1-carbonyl)thiophen-2-yl]acetamide;hydrochloride 3-ethyl-1,2-dimethylindole 3-(2,5-dimethylpyrrol-1-yl)sulfonylphenol 5-(2-methoxyphenyl)sulfonyl-1H-indole 5-bromo-N'-[4-[2,3-dichloro-6-(methylsulfanylamino)phenyl]thieno[3,2-d]pyrimidin-7-yl]furan-2-carboximidamide (4-benzylpiperazin-1-yl)-[3-methoxy-5-(trifluoromethylsulfanyl)phenyl]methanone 3-amino-4-(methylamino)benzenesulfonamide 2-[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]butanamide;4-oxopyrido[3,2-d]pyrimidine-7-carboxylic acid 7-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]-6-fluoro-1H-quinolin-4-one 2-[4-(benzylamino)phenyl]-N,5,7-trimethylimidazo[1,2-a]pyridine-3-carboxamide 2-(4-iodophenyl)-N-methyl-3H-indene-1-carboxamide [5-chloro-3-(2,6-difluorophenyl)-1H-indol-7-yl]methanol 4-[1,3,4,7-tetramethyl-6-(2-nitrophenyl)naphthalen-2-yl]naphthalene-2,3-dione (4S)-3-methyl-1,4-bis[2-(3,4,5-trimethoxyphenyl)ethynyl]pyrrolidine N-[2,5-difluoro-4-(trifluoromethyl)phenyl]-4-methoxybutanamide 2-[1-(dimethylamino)propan-2-yloxy]pyrido[3,4-d]pyrimidine-8-carboxylic acid 5-[3-(1,2-difluorocyclopropyl)-4H-quinazolin-6-yl]-6-methoxypyrazine-2-carboxylic acid 6-methyliodanuidyl-N-phenylnaphthalen-2-amine 3-(4-azidobutyl)-2H-triazolo[4,5-d]pyrimidine 2-ethyl-5,6-dimethoxy-2,3-dihydroinden-1-one 4-N-[(3Z,5E)-hepta-1,3,5-trien-2-yl]-6-phenylpyrimidine-2,4-diamine 2-amino-N,N-di(butan-2-yl)benzamide 3-azido-6,7-dimethoxyisoquinoline (2S)-1-(2,5-difluorophenyl)-2-methylpentan-3-amine [3-azidooxy-1-(benzenesulfonyl)butan-2-yl]benzene N-[(3R,4S)-1-azido-4-[2-(5-chlorothiophen-2-yl)sulfonylacetyl]piperidin-3-yl]benzamide 2-[(4-methylphenoxy)methyl]piperidine-1-carboxylic acid 4-[(2Z,5R)-2-[(E)-1-phenylpropylidenehydrazinylidene]-4-(pyridine-3-carbonyloxymethyl)-1,3-thiazolidin-5-yl]butanoic acid (E)-2-(N,4-dimethylanilino)-3-[1H-imidazol-5-ylmethoxy-[3-(trifluoromethyl)phenyl]boranyl]prop-2-enenitrile (6-methyl-2,5-diphenylpyridin-3-yl)phosphane 4-(2-azidooxyphenoxy)-1,3-benzodioxole (Z)-2-benzamido-3-hydroxyprop-2-enamide;1-[6-(diethylamino)-7H-purin-8-yl]piperidine-4-carboxamide [3-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)phenyl]carbamic acid 5-(1,3-benzodioxol-5-ylmethyl)-2-cyclopropyliminoimidazolidin-4-one 6-fluoro-7-(3-fluorophenyl)quinoline 3-[(5S)-2-azido-1,4-dioxan-5-yl]aniline [4-[(E)-2-(3,5-dimethylcyclohexa-1,3-dien-1-yl)ethenyl]phenyl]-naphthalen-1-ylmethanone 1-(4-chloro-2,5-difluorophenyl)-3-[4-ethyl-6-(1-ethylcyclohexyl)cyclohexa-1,3-dien-1-yl]urea 3-[1-[(2R,6S)-2,6-dimethyloxan-4-yl]imidazol-2-yl]quinoline 6-N,7-bis(2-methoxyphenyl)imidazo[1,2-b]pyridazine-3,6-diamine 5-methyl-2-(1,4-oxathian-2-yl)-1H-pyrimidine-6-thione ethane;3-(2-methylpyrimidin-5-yl)oxypropanamide 3,5-dimethoxy-1-[(4R)-2-methyloxepane-4-carbonyl]pyridin-2-one 3-[4-(benzylamino)-2-nitrophenyl]oxetan-3-ol (2R)-1-[5-[6-(azidomethyl)quinolin-8-yl]pyridin-3-yl]oxy-3-cyclopentylpropan-2-amine 5-(2,3-dimethylphenyl)-6H-naphthalene-1,3-dione N-(3,5-dimethylphenyl)-4-[4-[2-[5-(trifluoromethoxy)indol-1-yl]ethyl]piperazin-1-yl]benzenesulfonamide 3-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[(4-oxo-3H-quinazolin-2-yl)methyl]prop-2-enamide 3-[3-fluoro-4-(1H-pyrazol-5-yl)phenoxy]-2,6-dimethylbenzonitrile 2-(3,4-difluorophenyl)-6-[4-(4-heptylcyclohexyl)cyclohexyl]naphthalene N-ethylsulfanylmethanamine;1-(4-methoxyphenyl)pyrrolidine 6-[2,2,4-trimethyl-5-oxo-3-(phenylmethoxycarbonylamino)pyrrol-1-yl]hexanoic acid 4-(azidomethyl)-6,11-dihydrobenzo[c][1]benzoxepine 2-(benzimidazol-1-id-4-yl)pyridine;N-tert-butyl-1,3-diphenylpropan-2-amine;platinum(2+) 2-[6-tert-butylsulfanyl-7-oxo-3-(1H-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-N-(4-propan-2-ylphenyl)acetamide 3-(6-chloropyrazin-2-yl)oxybenzene-1,2-dicarbonitrile 1-[3-methylbutyl(1,2,4-triazol-4-yl)amino]propan-2-one N-methyl-4-[2-[(4-oxocyclohexanecarbonyl)amino]ethoxy]benzamide 5-tert-butyl-1-[(2,3-dimethoxyphenyl)methyl]imidazole 3-(6,7-dihydro-4H-pyrano[2,3-c]pyrazol-1-yl)-N-methylsulfonylbenzamide 1-[5-[2-(3-fluorophenyl)ethyl]-6H-cyclopenta[b]pyrrol-6-yl]propan-2-one 3-[4,5-bis(ethenyl)furan-2-carbonyl]chromen-4-one 5-[[7-(2,4-difluorophenyl)quinolin-3-yl]methylidene]-1,3-thiazolidine-2,4-dione 2-(3,5-dichlorophenoxy)-N-[(1Z,4E)-3-methyl-4-[(5-phenylpyridin-2-yl)amino]hepta-1,4,6-trienyl]propanamide (6R)-3,5-dimethyl-8-oxo-7-[[2-[6-(trifluoromethyl)pyridin-3-yl]acetyl]amino]-4-thia-1-azabicyclo[4.2.0]octane-2-carboxylic acid 1,3-ditert-butyl-5-(dimethylamino)pyrazole-4-carboxylic acid 4-[4-methyl-1-[(2S)-2-methylbutanoyl]piperidin-4-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one 2-(2,4-difluorophenyl)-6,7-dimethoxy-1H-isoquinoline 3-[(1E,3Z)-2,3-dimethylhexa-1,3,5-trienyl]-4-phenylmethoxyaniline [4-(2,3-dimethylphenyl)sulfanyl-3-fluorophenyl]phosphane N-methoxy-6-(2,3,4,5,7-pentamethylcyclohepta-1,3,5-trien-1-yl)-[1]benzothiolo[3,2-c]chromene-9-carboxamide 2-[(1S)-2,3-dihydro-1H-inden-1-yl]-6-methoxyisoquinolin-1-one 2-(1,5-dimethylpyrazol-4-yl)oxypyridine 4-(4-methylphenyl)sulfanylpentylphosphane 2-[4,6-dimethyl-5-(3-oxo-1H-isoindol-2-yl)pyrimidin-2-yl]oxyacetic acid 2-(2,4-dimethylanilino)-N-[(Z)-1H-indol-3-ylmethylideneamino]benzamide 4-chloro-3-hydroxy-N'-(6-methylheptanoyl)thiophene-2-carbohydrazide (6R,9S)-2-amino-9-(4-chlorophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 4-[3-cyano-6-(2,6-dichlorophenyl)pyridin-2-yl]-N'-methanimidoylpiperazine-1-carboximidamide 5-[2-(4-butylcyclohexyl)ethynyl]-6-(3,5-difluorophenyl)-1,2,3-trifluoronaphthalene 5-azido-1,4-dimethyl-2,3-bis(3-phenylpropyl)benzene 3-aminosulfanyl-4-[1-(2,5-dichloropyrimidin-4-yl)pyrrolidin-3-yl]oxybenzonitrile 3-(azidomethoxy)-1,2-dichloro-4-phenylbenzene 7-bromo-5-phenylspiro[1,3-dihydro-1,4-benzodiazepine-2,4'-piperidine] 2-methyl-5-[2-(3-methylphenyl)propan-2-yl]-1H-indene [3-[[1-[3,5-bis(trifluoromethyl)phenyl]triazol-4-yl]methoxy]phenyl]methanimine 5-hydroxy-4-[2-(1,3,5-trimethylpyrazol-4-yl)phenyl]-7H-pyrrolo[3,4-f]isoindole-6,8-dione 4-amino-6-[(3-chloroquinolin-8-yl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 1-methoxy-4-(5-phenylhexan-2-yl)benzene 2-[3-methylbut-2-enyl(1,2,4-triazol-4-yl)amino]acetic acid N-[2,6-difluoro-4-(1H-pyrrolo[3,2-b]pyridin-5-yl)phenyl]benzenesulfonamide (2R)-2-[3-[[4-ethoxycarbonyl-1-(1H-indole-6-carbonyl)piperidin-4-yl]amino]-5-methylphenyl]butanoic acid 1-(2,3,4-triphenylnaphthalen-1-yl)propan-1-one 6-[(1Z)-1,3-diamino-2-methylbuta-1,3-dienyl]-5-ethoxypyridine-3-carbonitrile 2-bromo-N,N'-diethylbenzenecarboximidamide 1-(3,4-dihydroisoquinolin-5-yl)-2-ethoxybutan-1-one N-[4,5,6-trifluoro-2-(propanoylamino)phenyl]carbamate 2-[1-(2-azidoethyl)piperidin-4-ylidene]-6,11-dihydrobenzo[c][1]benzoxepine 1-[2,3-difluoro-4-(trifluoromethyl)phenyl]-3,5-bis(trifluoromethyl)pyrazole (2S)-1-[2-oxo-2-[(2S)-pyrrolidin-2-yl]acetyl]-N-[[2-oxo-4-propan-2-yl-3,5-bis(trifluoromethyl)pyridin-1-yl]methyl]pyrrolidine-2-carboxamide 5-[(E)-3-amino-4,4-difluoro-2-methylbut-1-enyl]-N-[1-hydroxy-3-[2-[2-[4-hydroxy-4-(4-iodobenzoyl)piperidin-1-yl]ethoxy]phenyl]propan-2-ylidene]furan-2-carboxamide (E)-3-[4-hydroxy-2-methoxy-5-(4,5,6,7-tetrahydro-1H-indol-2-ylsulfonylcarbamoyl)phenyl]prop-2-enoic acid 2,3-dimethylpyridine;ethane;2-(5-hydroxy-1H-indol-3-yl)-6-[[4-(4-methoxyphenyl)piperazin-1-yl]methyl]pyran-4-one 1-[4-(2,5-dimethylpyrrol-1-yl)phenyl]ethanone;ethane;N'-methyl-3-phenylpropane-1,2-diamine 3-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-[3-hydroxy-4-(trifluoromethoxy)phenyl]propanamide 4-(2,3,5,6,7,8,9,10,11-octahydropyrido[1,2-a]azocine-3-carbonyl)-1H-pyridin-2-one;dihydrochloride 5-ethenyl-2-methoxybenzenesulfonic acid 3-[4-chloro-2-fluoro-5-(1,2-thiazol-4-yl)phenyl]-7-[4-ethyl-6-(methanesulfonamido)pyridin-2-yl]-2H-furo[2,3-e]indole-2-carboxylate (5E)-2-(4,6-dimethylpyrimidin-2-yl)imino-5-[(3-ethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 3-[8-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]imidazo[1,5-a]pyridin-6-yl]pyridine-4-carboxylic acid 2-[5,7a-dihydrobenzotriazol-2-yl(2,3-dihydroindole-1-carbonyl)amino]ethanesulfonic acid [(E)-2,3-dihydro-1H-thieno[2,3-g][1,4]benzoxazin-7-yl]methanol 5-hydroxy-4-[3-[[3-methyl-6-(4-methylpiperazin-1-yl)cyclohexa-2,4-dien-1-ylidene]amino]phenyl]-7-propan-2-yloxychromen-2-one (2R)-1-[4-azido-5-chloro-6-(cyclopropylmethoxy)pyrimidin-2-yl]oxy-3-(methanesulfonamido)butan-2-ol 1-(cyclohexen-1-yl)-4-[3-[2-methoxyethyl(methyl)amino]propoxy]naphthalene-2-carboxylic acid 2-[(2,6-dichlorobenzoyl)amino]-3-[8-(3-iodophenyl)quinolin-5-yl]oxypropanoic acid 2-[(6R)-4,5,10,11-tetrahydro-[1]benzoxepino[3,4-d]pyrimidin-6-yl]acetic acid 3-(2-azidophenyl)-1,5-dimethylpyrazole 3-(1,2-dihydroacenaphthylen-5-yl)-1H-pyridazin-6-one 4-[2-[2,6-dichloro-3-(ethoxymethyl)phenyl]ethynyl]benzamide (2S)-N-[1,3-dihydroxy-2-[(4-methylphenyl)sulfonylamino]propan-2-yl]-1,1,1-trifluoro-N'-methylpyrrolidine-2-carbohydrazide 1,3-diethyl-4-(phenyliminomethyl)benzene;N-[(Z)-2-(methylideneamino)ethenyl]-N'-pentylethenamine N-(3,4-difluorophenyl)-6,7-dihydro-1-benzofuran-2-carboxamide 5-cyclopropyl-N'-hydroxy-3-(trifluoromethoxy)pyridine-2-carboximidamide 2-(5,6-dimethylpyridine-3-carbonyl)-4-oxo-N'-[(1R)-3-phenylcyclopenten-1-yl]pyrrolidine-1-carboximidamide 2-tert-butyl-1'-[(4,5-dimethoxypyrimidin-2-yl)methyl]-6-methylspiro[3H-chromene-2,4'-piperidine]-4-one 6-bromo-3-[(2Z)-5,8-dimethylcycloocta-2,7-dien-1-ylidene]-4H-chromene 2-[4-(azidomethyl)phenyl]naphthalene 5-[(Z)-2-aminobut-1-enyl]-N,N-bis[3-(dimethylamino)propyl]naphthalene-1-sulfonamide 1-phenylmethoxy-9H-thioxanthene-2,4,7-triamine 1-(7-benzylsulfanyl-1H-indol-3-yl)ethanethione 4-[3-[(5-fluoro-2,4-dihydroxyphenyl)methylamino]phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile N'-azido-4-(2,6-dibromophenyl)-1,3-thiazol-5-amine 3-methyl-2,4-dinitro-1H-pyridine-2-carboxylic acid 3-[6,8-dioxo-9-[4-(N'-phenylcarbamimidoyl)anilino]-1H-purin-2-yl]benzenecarboximidamide 4-chlorobenzenethiol;2-(1H-indol-5-yloxy)butanoic acid (5Z)-5-[[2-[2,4-bis(methoxycarbonyl)phenoxy]phenyl]methylidene]-2-imino-1,3-thiazolidin-4-one N-(8,9-diethoxy-3,4-dihydro-1H-pyrano[4,3-c]quinolin-10-yl)-2-phenylacetamide 1-(4-acetylphenyl)sulfonylpyrrolidine-2,5-dione 4-amino-3,5,6-trichloropyridine-2-carboxylic acid 5-azido-2-(1H-indol-2-yl)-1,3-benzothiazole 6-(4,5-dihydro-1,3-thiazol-2-ylamino)pyridine-3-carboxylic acid 5-chloro-N,N-dimethyl-2-[[3-(2-oxopiperidin-1-yl)phenyl]sulfanylamino]benzamide 2-[(1R)-3,3-dimethylcyclohexyl]oxy-N-[6-(4-ethylpiperazin-1-yl)pyridin-3-yl]thieno[3,2-d]pyrimidin-4-amine 4-[(2-chloroacetyl)-(3-ethoxy-3-oxopropanoyl)amino]benzenesulfonic acid [2-[(4R)-1-(1,3-benzothiazol-6-ylsulfonyl)piperidin-4-yl]oxypyridin-4-yl]methanamine 2-[3,5-dimethyl-4-(prop-1-enylamino)phenoxy]acetonitrile 3-[2-(4-propan-2-ylphenyl)ethynyl]-5-(trifluoromethoxy)phenol ethane;2-methyl-6-[4-(trifluoromethoxy)phenyl]pyrazolo[1,5-a]pyrimidine N-[(4R)-6,9-diazaspiro[2.5]octan-7-yl]-2-[1-(6,8-difluoroquinoline-3-carbonyl)piperidin-4-yl]acetamide 2-chloro-N,5-dimethoxyaniline;N-(1-formylpyrrolidin-3-yl)-4-morpholin-4-ylbenzamide 2-(4-azidophenyl)sulfanylacetic acid 2-[4-ethylsulfonyl-6-(trifluoromethyl)pyridin-3-yl]propanenitrile 2-[3-[(E)-3-hydroxybut-1-enyl]-4,7-dimethoxynaphthalen-1-yl]prop-2-enenitrile 5-ethynylnaphthalene-1,2,6-tricarboxylic acid 2-[7-fluoro-8-(methoxymethyl)naphthalen-1-yl]-5-(3-methoxyazetidine-1-carbonyl)benzonitrile (3R)-6,8-difluoro-1'-methylspiro[2H-pyrrolo[2,3-b]quinoline-1,4'-cyclohexane]-3-one 5-(1H-imidazo[4,5-b]pyridine-6-carbonylamino)-3-methylthiophene-2-carboxylic acid 2-(2-methylpropanoyloxy)benzenesulfonate 4-[7-amino-6-bromo-2,8-dimethyl-3-[2-(trifluoromethyl)phenyl]indolizine-1-carbonyl]-N'-methanimidoylpiperazine-1-carboximidamide [4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl]-(2,6-dimethylpyridin-3-yl)methanone 2-[2-(4-cyclopropylphenyl)imino-3,6-dihydro-1H-pyridin-5-yl]acetonitrile 4-(4-ethylcyclohexa-1,5-dien-1-yl)-2-propan-2-ylidene-5H-benzo[e]benzotriazole N-[1-cyclopentyl-3-(dimethylamino)propan-2-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide N-[4-[4-(cyclopentylamino)cyclohexyl]phenyl]-2-fluorobenzamide 7-[(6-bromonaphthalen-2-yl)sulfonylamino]-4-methoxyspiro[3H-chromene-2,1'-cyclobutane]-8-carboxylic acid 1-cyclopentyl-4-[(2,3-dichlorophenyl)methoxy]benzotriazole 6-[(2,5-dimethylphenyl)methoxy]-4,8-dihydrobenzo[e]indole-3-carboxylic acid 4-[2-(4-propan-2-yloxyphenyl)ethynyl]phenol 4-methyl-2-[4-(1,3-oxazole-5-carbonyl)morpholin-3-yl]-1H-pyrimidin-6-one (4-chlorophenyl)-[1-(2,3,4,5,6-pentafluorophenoxy)cyclopentyl]methanone 6-bromo-7-[4,5-bis(ethenyl)-1H-pyrrol-3-yl]-2,3-dihydrothieno[3,4-b][1,4]dioxine N-[2-(dimethylamino)ethyl]-3-[(1R,4E)-1-methoxyhepta-1,4-dien-2-yl]-5-propan-2-ylidenebenzenecarboximidate 2-[3-(cyclobutadienyl)phenyl]-4,6-dihydrazinylpyridine-3,5-dicarbonitrile (2-chloropyridin-3-yl)-phenylmethanone N-methylmethanesulfonamide;(4R)-3-[[(1R)-2,2,2-trifluoro-1-(4-fluorophenyl)ethoxy]carbonylamino]azepane-1-carboxamide 3-(5-azidooxy-2-methylphenyl)-1,2,4,5-tetrazine 1-[1-(benzenesulfonyl)pyrrole-2,3-dicarbonyl]piperidine-2-carboxylic acid 5-ethyl-7,9-dimethoxy-1,3,3a-trimethyl-2-(4-methylphenyl)indeno[2,1-b]fluorene 1-[4-(3,5-dimethylphenyl)piperazin-1-yl]propan-2-one;ethane 2-[4-(cyclopropylamino)piperidin-1-yl]-N'-hydroxypyridine-4-carboximidamide [2-azido-1-[[3,5-bis(trifluoromethyl)phenyl]methoxy]propan-2-yl]cycloheptane 7-ethyl-6,8-difluoro-N-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]quinazolin-4-amine 4-[2-(4-azidopiperazin-1-yl)ethyl]benzonitrile 4-cyclohexa-1,5-dien-1-yl-2-[4-(5-fluoropyridin-3-yl)-1H-benzimidazol-2-yl]-1H-imidazo[4,5-c]pyridine N-[5-(2,4-dihydroxyphenyl)-3-(1H-indol-3-ylmethylideneamino)thiophen-2-yl]formamide 1-[[2-fluoro-4-(trifluoromethyl)phenyl]carbamoyl]piperidine-3-carboxylic acid 3-[5-(2,5-dimethylimidazol-1-yl)-4-methoxypyridin-2-yl]-3-azaspiro[5.5]undecane (6Z,7E)-8-[2-(3,4-dimethoxyphenyl)ethylimino]-5,9-bis(ethenyl)-8,10-dihydrobenzo[b]anthracen-11-ol 2-[3-(8,9-dimethoxy-1,4-dihydroanthracen-9-yl)propyl]naphthalene 2,4-dichloro-N-(2-nitrophenyl)-N-[3-(trifluoromethyl)phenyl]pyrimidin-5-amine 1-(2,4-dichlorophenyl)sulfonyl-3-propan-2-ylazetidine 2-[3-(1,3-benzothiazol-6-yl)-4H-imidazol-5-yl]ethanamine;butane;cyclohexane [(3S)-3-(3,5-difluorophenyl)pyrrolidine-1-carbonyl]boronic acid [4-(3,5-dimethylphenyl)piperazin-1-yl]-(1-methylpyrazol-3-yl)methanone 3-(azepan-1-yl)benzaldehyde;butane 4-[(3Z,5E)-6-aminohexa-1,3,5-trien-2-yl]-N-methylaniline 2-(cyclohexylmethoxy)-7-ethyl-4,8-dimethylquinoline [3-(benzylsulfonylamino)-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-5-ylidene]urea;hydrochloride 1-azido-2,4-dipropylbenzene 4-cyclopropyl-5-methoxypyridine-3-carboxylic acid (2S)-N-[4,5-bis[(2-methylpropan-2-yl)oxy]thiophen-2-yl]-2-(3-chlorophenyl)-5,7-dimethyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-4-carboxamide (E)-3-(5,6-dihydroxynaphthalen-2-yl)-N-[4-methoxy-2-(pentanoylamino)phenyl]prop-2-enamide 4-[(7S)-6-amino-5,6,9,10-tetrahydronaphtho[2,3-b][1]benzofuran-8-yl]phenol;cyclohexa-3,5-diene-1,2-diimine 2-[2,3-dimethyl-4-(4-methylsulfanylbenzoyl)oxyphenyl]acetic acid (3aR,4R,7aS)-5-benzyl-N-ethyl-1-methyl-2,3,3a,4,6,7,7a-octahydropyrrolo[3,2-c]pyridine-4-carboxamide;formic acid 5-[(4-bromophenyl)carbamoylamino]-N-tert-butyl-2,3-dihydroxybenzamide;propane N-(1,3-benzothiazol-2-yl)-4-(dipropylamino)benzamide N-[2,5-dichloro-4-(trifluoromethyl)phenyl]-N'-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]carbamimidothioate (2R,6R)-4-(4-fluorophenyl)-N-[[1-[6-(trifluoromethylsulfanylamino)pyridine-3-carbonyl]piperidin-2-yl]methyl]bicyclo[3.1.0]hexane-2-carboxamide 1-[5,6-difluoro-2-(hydroxymethyl)-3H-inden-1-yl]pyrrolidine-2-carboxamide (5E)-2-imino-5-[(4-methoxynaphthalen-1-yl)methylidene]-3-(naphthalen-1-ylmethyl)imidazol-4-one 4-amino-5-chloro-6-(1-methylsulfinylbutan-2-ylsulfanyl)pyrimidine-2-carboxylic acid 4-ethylsulfonyloxybenzenesulfinate 5-(2,4-dihydroxy-6-methylphenyl)-N-[1-(4-pyrrolidin-1-ylpiperidine-1-carbonyl)cyclohexa-2,4-dien-1-yl]-1,3-oxazole-4-carboxamide N-benzyl-2-chloro-4-(5,6-dichloro-3H-indol-1-ium-1-yl)pyrimidine-5-sulfonamide N-(2,6-dioxopiperidin-3-yl)-N-[1-(3-methoxyphenyl)ethyl]formamide 5-[3-(4-cyclohexyloxyphenyl)propanoyl]-2,4-dimethyl-1H-pyrimidin-6-one 2-(1,2,3,6-tetrahydropyridin-4-yl)indole 4-[(3S)-1,5-dioxo-2-[[4-(trifluoromethyl)phenyl]methyl]pyrrolidin-3-yl]butanoic acid 2-[3,5-dichloro-4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1-hydroxy-N'-iminoindole-6-carboximidamide 2-(1,3,4,9a-tetrahydrofluoren-9-yl)naphthalene 4-[(2,6-difluorophenyl)methyl]-5-iodo-2-piperidin-1-yl-1H-pyrimidin-6-one 4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butanoate N-(4-hydroxyphenyl)-2,3-dioxoaziridine-1-carboxamide 2-chloro-1-[3,3-di(propan-2-yl)cyclohexa-1,5-dien-1-yl]oxyethanethiol 4-[2,5-dichloro-3,6-bis(methylsulfanyl)naphthalen-1-yl]oxyphenol 1-azidooxy-2,3,4-tris(ethenyl)benzene N-[4-(chloromethyl)pyridin-2-yl]-N-cyclopropylformamide 2-[[7-chloro-4-oxo-3-phenyl-5-(propanoylamino)quinazolin-6-yl]amino]acetamide 3-[2-(4-bromophenyl)ethyl]oxan-3-ol 3-[3-aminopropyl(2,6-difluorohexyl)amino]-1-cyclohepta-1,4,6-trien-1-yl-3H-inden-5-ol N'-[5-[4-methyl-1-(2-oxooxolan-3-yl)pyrazolo[3,4-b]pyridine-6-carbonyl]-6,7-dihydro-4H-furo[3,4-c]pyridin-7a-yl]methanimidamide 1-(2,3-dimethylphenyl)-5H-pyrazolo[4,3-c]quinolin-4-one 2-methoxycarbonyl-1,3-dihydropyrrolo[2,3-c]pyridine-6-carboxylic acid N'-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-(2-methoxyethoxy)quinoline-6-carboximidamide 3-(dimethylamino)-4,5-dimethoxybenzamide;2-ethylnaphthalene N-[1,3-dihydroxy-4-oxo-2-(phenylsulfanylmethyl)butan-2-yl]carbamate 2-[(2,4-dimethoxyphenyl)methyl]-8-oxa-5-azaspiro[3.5]nonane 3-cyclopropyl-2-[(4-methoxyphenyl)sulfonylamino]-N,N-dimethyl-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-10-carboxamide 4-(6-chloropyridin-3-yl)-N-(2,2-dimethoxyethyl)-2,5-dioxoimidazolidine-1-carboxamide 4-[6-(4,4-difluoropiperidine-1-carbonyl)-2-methylthieno[3,2-b]pyridin-7-yl]oxybenzonitrile 1-(4,6-dimethylpyrimidin-2-yl)-N-[[(2R,3S)-2-phenyloxolan-3-yl]methyl]ethanamine 4-(3,5-dimethyl-2H-pyrrole-4-carbonyl)-3,5-dihydro-2H-1,4-benzoxazepine-8-carboxylic acid;ethane 2-(4-phenylpiperazin-1-yl)ethanol;hydrochloride 2-[2,4-dichloro-N-(1,3-thiazol-5-yl)anilino]acetamide 1-(2,4-difluorophenyl)-3-(2,5-dimethoxyphenyl)-5-[(E)-1-propan-2-ylsulfanylethenyl]pyrazole 3-azido-4,5-bis(phenylmethoxy)benzoic acid 1-[2-(2,3-difluorophenoxy)ethyl]pyrazole 4-[[2-[[cyclopentylmethyl(ethyl)amino]methyl]phenyl]sulfamoyl]benzoic acid 1-(2-azidoethyl)-4-[2-methoxy-5-(2,3,6-trifluorophenyl)pentan-2-yl]piperidine N-[(2S,3R)-1-cyclopropyl-5-oxo-2-pyridin-3-ylpyrrolidin-3-yl]-4-propanoylbenzamide 3-[2,2-dimethylpropanoyl(naphthalen-1-yl)amino]propanoic acid 1-[6-azido-5-(difluoromethyl)pyridin-2-yl]pyrazole 5-(4-chloro-3-fluorophenyl)-2-[2,6-difluoro-4-[(E)-hex-1-enyl]phenyl]pyrimidine 3-benzyl-5-methylbenzene-1,2-disulfonic acid N-(4-fluorophenyl)-1,7-dimethyl-2-oxoquinoline-3-carboxamide 4-[4-(2,3-dichlorophenyl)-5-methoxy-1H-pyrazole-3-carbonyl]benzoic acid 1-bromo-2,3-diiodo-5-methoxybenzene [6-(4-tert-butylcyclohexyl)oxy-1H-indol-2-yl]-phenylmethanone 4-[(7S)-2,3-dimethyl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl]benzamide 2-(3,4-dichlorophenyl)imino-5-[(2-methylsulfanylpyrimidin-4-yl)methylidene]-1,3-thiazolidin-4-one 2-[5-methoxy-6-(trifluoromethyl)-1H-benzimidazol-2-yl]-4,5-dihydro-1H-imidazole 1-(4-hydroxyphenyl)cyclohexa-3,5-diene-1,2-disulfonamide 1-(4-chlorophenyl)-7,11b-dihydrobenzo[c]chromen-6-one 3-(1,4-dimethylbenzotriazol-5-yl)-2,3-dihydroisoindol-1-one 5-chloro-N-[4-[[3-(2,6-dioxopiperidin-1-yl)-2-methylbutanoyl]amino]cyclohexyl]pyridine-2-carboxamide 1-benzyl-4,5-dimethoxypiperidine;ethane 3-[2,6-dichloro-N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-nitroanilino]butanoic acid N-cyclohexyloxy-1,3-oxazole-2-carboxamide 2-(3,5-dimethoxyphenyl)-1H-pyrrolo[2,3-c]pyridine 2-N-(4-fluorophenyl)-6-[1-methyl-5-(trifluoromethoxy)pyrazol-3-yl]pyrimidine-2,4-diamine 2-[(2Z,5S)-2-[(Z)-[4-(3-methylphenyl)sulfanylphenyl]methylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 1-(2,3-dimethylphenyl)sulfonyl-4-[(3S)-3-phenylpiperazine-1-carbonyl]piperidin-4-ol 4-N-methylsulfanyl-1-N-[1-(2H-tetrazol-5-yl)cyclohexyl]benzene-1,4-diamine 6-bromo-3-(2,4,5-trimethoxyphenyl)pyrido[1,2-a]pyrimidin-4-one 5-bromo-3-(2,6-difluorophenyl)-4H-quinazoline 5-tert-butyl-1,2-dimethoxy-3-(2,4,6-trimethylphenyl)benzene N-[2,4-dichloro-3-(7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)phenyl]propane-1-sulfonamide 2-[(5R)-3-hydroxy-5,6-dimethoxyhexyl]pyridine-4-carboxamide 1-(3-chlorophenyl)sulfonyl-2,4-dimethylbenzene [2-methylpropanoyloxy(phenyl)methyl]-triphenylphosphanium (Z)-1,5-diphenylhex-4-en-2-ol 2,3-difluoro-4-[(2R)-9-methoxycarbonyl-8-methylnonan-2-yl]benzoic acid N'-(benzenesulfonyl)benzenecarboximidamide (2S)-N-(1,3-benzothiazol-5-yl)-5-methoxy-2-propanoylcyclohexane-1-carboxamide 2-[4-[4-amino-6,8-difluoro-7-(3-fluoroanilino)pyrimido[5,4-d]pyrimidin-2-yl]phenyl]propan-2-ol;ethane ethane;1-(3-methoxyphenyl)pyrrole ethane;methanamine;(E)-4-[1-[2-[[6-(trifluoromethyl)pyridine-3-carbonyl]amino]phenoxy]butyl-[3-(trifluoromethyl)phenyl]phosphaniumyl]but-2-enoate 4-(3,5-dimethylpyridin-2-yl)-N'-hydroxybenzenecarboximidamide 3-(4,5-dimethoxypyridin-2-yl)-N-[[2-ethoxy-6-(trifluoromethyl)pyridin-3-yl]methyl]-1H-indole-7-carboxamide 2-[4-(benzenesulfinyl)phenyl]acetonitrile N-[(4-chlorophenyl)methyl]-3,3-difluoropiperidine-2-carboxamide;5-methoxy-2H-triazole-4-carboxylic acid 3-(4-morpholin-4-yl-6,7-dihydrothieno[3,2-d]pyrimidin-1-ium-5-carbonyl)cyclohexane-1-carboxylic acid 1-chloro-3,4-dimethyl-2-(2-methylbutan-2-yl)naphthalene (2-chlorophenyl)-[4-(3,6-dihydro-2H-pyran-4-ylmethoxy)phenyl]methanone (6R)-3-[4-[2-[(3,5-dichlorophenyl)methyl]hydrazinyl]piperidine-1-carbonyl]-6-ethyl-6,7-dihydro-5H-triazolo[4,5-c]pyridin-4-one (1S,2R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-5-cyano-2-hydroxycyclohexane-1-carboxamide (5S,8aR)-7-[5-(2-methylpyrazol-3-yl)pyrimidin-4-yl]-1,5,6,8,8a-hexahydro-[1,3]oxazolo[3,4-a]pyrazin-3-one 5-[2,3-bis(ethenyl)phenyl]-1,10-phenanthroline 2,7-dibromo-5H-furo[3,4-d]pyrimidine 4-(2-diazohydrazinyl)-1H-pyrrolo[3,2-c]pyridine-7-carboxylic acid 5-(4-azido-3,5-dichlorophenyl)-N'-hydroxypyrazine-2-carboximidamide N-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-2-(4-cyclohexylpiperazin-1-yl)ethanamine N-[(5Z)-5-[[4-(3,4-difluorophenyl)phenyl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]-4-fluorobenzenesulfonamide N-(4,5-dihydro-1H-imidazol-2-yl)-4-propan-2-yl-3-thiophen-2-ylpiperazine-1-carboxamide 4-[2-[(2-methoxyphenyl)methyl]-1,3,4,6,7,8,9a-hexahydropyrido[1,2-a]pyrazin-7-yl]benzenesulfonamide (4S)-3-[2-chloro-6-methyl-4-(3-pyridin-4-ylpropoxy)benzoyl]-1,3-thiazolidine-4-carboxylic acid 1-methyl-N-(4-pyridin-2-yloxyphenyl)pyrazole-3-carboxamide (4R)-3-[(2S,3aS,7aR)-6-[[4-(trifluoromethyl)phenyl]carbamoyloxy]spiro[3.5]nonan-2-yl]-1,3-thiazolidine-4-carboxylic acid N-[4-[3-ethenyl-5,6-dimethoxy-1-(2-morpholin-4-ylethyl)indol-2-yl]phenyl]pyrrolidine-2-carboxamide 2-[(1S)-2-hydroxy-1-pyridin-3-ylethyl]piperazine-1-carboxylate N-[5-(1H-benzimidazol-2-yl)pyridin-3-yl]cyclopropanecarboxamide 3-(dimethylamino)-2,4-dioxobenzo[g]pteridine-7-carboxylic acid 4-[2-(5,6-dihydro-1H-benzimidazol-3-ium-3-yl)ethylidene]-2-methoxyimino-N-(3-sulfanylpropoxy)cyclohexa-2,5-dien-1-imine 3-bromo-7,9-dimethoxy-2,2-dimethyl-1H-pyrrolo[2,1-a]isoquinoline 6-[2,3-dihydroxypropyl(2-hydroxyethyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 2-(3,5-dichloropyridin-4-yl)-N-propan-2-yl-5-[[6-[1-(trifluoromethyl)cyclopropyl]pyrimidine-4-carbonyl]amino]oxy-1H-indole-7-carboxamide 4-[5-[(1,3-diethoxy-1,3-dioxopropan-2-yl)amino]thiophen-2-yl]-2-methoxybenzoic acid 2-azido-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde 4-[2-(4-fluoro-3,5-dimethylphenyl)-1,3-thiazol-5-yl]-N'-(trideuteriomethoxy)benzohydrazide 3-(4-ethoxy-N-hexylanilino)propane-1,2-diol 3-(4-cyclopropylphenyl)-N-[(2S,3R)-1-methyl-2-(2-methylpyrazol-3-yl)piperidin-3-yl]propanamide 2-[[5-(4-chlorophenyl)furan-2-yl]methylsulfanyl]-1-nitro-4-phenylimidazole 3-(4-chlorophenyl)sulfanyl-2-methoxy-7H-purine 6-[3,5-bis(trifluoromethyl)phenyl]-N-[5-chloro-2-methoxy-4-[(2S)-4-methyl-2-propanoylpiperazine-1-carbonyl]phenyl]-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxamide 2-ethyl-7-(3-methoxybutyl)-4,5,6,8-tetrahydropyrazolo[1,5-a][1,4]diazepine;hydrochloride N'-[4-[(6,7-dimethoxy-1,5-naphthyridin-4-yl)oxy]-3-fluorophenyl]-N,N,N'-trimethylethane-1,2-diamine;ethane 2-[6,7-difluoro-4-(4-methylpiperazin-1-yl)quinazolin-8-yl]phenol (5Z)-2-(4-fluorophenyl)imino-5-[(1,3-thiazol-2-yldisulfanyl)methylidene]-1,3-thiazolidin-4-one 2-(3,5-dimethylphenyl)sulfonyl-N-[(1R)-4-hydroxycycloheptyl]acetamide 4-[(2R,5S)-4-[(3-chlorophenyl)methyl]-2,5-dimethylpiperazine-1-carbonyl]-2-cyclopropyl-1H-pyrimidin-6-one 6-[(4,5-diamino-2-phenyltriazol-1-yl)methyl]naphthalen-2-ol 2,3-difluoro-1-[4-(4-methylcyclohexen-1-yl)phenyl]-4-propylbenzene N-(3,5-dimethylphenyl)-2-[(6S)-6-ethyl-4,8-dioxo-7-propanoyl-1,3,6,9-tetrahydropyrazolo[4,3-h][1,5]benzothiazepin-2-yl]acetamide (2S)-1,4-dimethyl-5-[2-methylsulfanylethyl(2-phenylethyl)carbamoyl]oxy-2-propan-2-ylpyrrolidine-3-carboxylic acid 3-(3-ethylsulfanylanilino)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carboxylic acid N-cyclopropyl-3-[5-[1-(2,4-difluorophenyl)ethyl]-1H-pyrazol-3-yl]benzamide N-[(E)-1H-indol-3-ylmethylideneamino]-2-[methyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]acetamide 2-[4-(4,4,5,5-tetramethyl-1H-imidazol-2-yl)phenyl]pyridine 5-(N,4-dimethylanilino)-6-ethoxycarbonylpyridine-3-carboxylic acid 3-(4-fluorophenyl)-N-methyl-6-[4-(triazol-1-yl)phenyl]-2,5-dihydropyrazolo[3,4-h]quinoline-8-carboxamide 2-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-4-phenylbenzenesulfonamide 5-[4-(2-azidophenyl)piperazin-1-yl]-6-methoxypyridazine-3,4-diamine 2-(3,4-dihydro-1H-naphthalen-2-ylideneamino)benzoic acid 2-methyl-N-(4-methylphenyl)sulfanylquinazolin-4-amine N-[(Z)-(3,5-dichloro-2-hydroxyphenyl)methylideneamino]-4-nitrobenzamide [(1Z,3E)-1,4-bis(4-fluorophenyl)penta-1,3-dienyl]hydrazine 1-(3,4-dimethoxyphenyl)sulfanyl-4-pentoxypiperazine N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-(2H-thiopyran-6-yl)-2-pyrimidin-2-ylethanamine N-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethyl)-N-[3-(trifluoromethoxy)phenyl]pyrrolidine-1-carboxamide N-[(3E)-2,6-dimethylocta-1,3,5,7-tetraen-4-yl]-8-(5H-pyrrolo[2,3-b]pyrazin-7-yl)isoquinolin-3-amine 4-[3-(furan-2-yl)pyrrolidine-1-carbonyl]-N,5-dimethylthiophene-2-sulfonamide 4-[1-(4-bromophenyl)triazol-4-yl]oxane 1-[(E)-4-naphthalen-2-ylbut-3-enyl]azepane 3-[4-(2,6-diphenylpyrimidin-4-yl)dibenzofuran-1-yl]pyridine 1-[[6-[(E)-4,4-dimethylpent-2-enoyl]pyridin-3-yl]methoxy]-N-(5-fluoropyridin-2-yl)isoquinoline-7-carboxamide 2-[N-(2,3-dihydroxypropyl)anilino]-2-methylpropanoic acid 1-azido-3-[2,6-di(propan-2-yl)phenyl]thiourea 5-cyclopropyl-N-[1-(2,4-dimethoxyphenyl)ethylideneamino]-7-oxo-6H-pyrazolo[1,5-a]pyrimidine-3-carboxamide 4-[2,3-dimethylbutoxy(phenyl)methylidene]-1-methylcyclohexane-1-carboxylic acid N-(5-azido-2,3-dihydro-1H-inden-1-yl)-4-methoxybenzenesulfonamide [(3S,4R)-1-benzylpiperidin-3-yl]-phenylmethanol 4-azido-5-methyl-1-[(3,4,5-trifluorophenyl)methyl]pyrazole 2-(4-chloro-3,5-dimethylpyrazol-1-yl)-N'-hydroxypyrimidine-4-carboximidamide N-(2,5-dioxohexan-3-yl)-4-fluorobenzamide N-[3-(2,3-dihydroindole-1-carbonyl)phenyl]benzamide 5-methoxy-6,6a,7,8,9,10-hexahydrobenzo[b][1]benzazepine 7-[(2R)-1-methoxypropan-2-yl]-5-(5H-pyrrolo[3,4-b]pyridin-6-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxylic acid 2-cyclopropyl-6-[(3-methoxythiophen-2-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (E)-3-[6-[2,4-dimethyl-5-[(4-pyridin-2-ylpiperidin-1-yl)methyl]furan-3-carbonyl]indol-1-yl]prop-2-enal 1-azidooxy-3,4-dichloro-2-(6-propan-2-yloxynaphthalen-2-yl)oxy-5-(2H-triazol-4-yloxy)anthracene 2-(4,6-diaminopyrimidin-5-yl)ethanol;N,2-dimethoxybenzamide N-(3,5-dichlorophenyl)-2,4,6-trimethyl-N-octylbenzenesulfonamide N-(3-chlorophenyl)-2-[(2Z,5R)-2-[(Z)-1-(4-hydroxyphenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetamide (1-benzoylpiperidin-4-ylidene)-ethoxymethanolate 4-(N-(6-bromo-1,3-benzothiazol-2-yl)anilino)benzenesulfonamide N-(2,6-dimethylphenyl)-3-(1H-imidazole-5-carbonylamino)-1H-pyrazole-5-carboxamide 1,3-diphenylbicyclo[1.1.0]butane 3-[4-[(2S,5R)-2,6-dimethylpiperazine-1-carbonyl]phenyl]sulfanyl-2-fluorobenzonitrile N-[2-(1-methylpyrazol-4-yl)-3H-benzimidazole-5-carboximidoyl]cyclopropanecarboxamide [(E)-1,2-bis(4-hydroxyphenyl)but-2-enyl]phosphonic acid 1-[5-(4-fluorophenyl)-7-(methylamino)pyrazolo[1,5-a]pyrimidin-3-yl]ethanone 4-chloro-2,3-bis(2-methylphenyl)quinoline [2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]phosphonic acid (4S)-N-(3,4-dichlorophenyl)-1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazole-4-carboxamide 3,4-dichloro-N'-[5-(3-methoxyphenyl)-1H-pyrazol-3-yl]benzenecarboximidamide 2-[3-[5-(oxolan-2-ylmethoxy)pyridin-1-ium-2-yl]-1H-pyrazol-5-yl]phenol N-(4-ethoxy-2,6-dimethylphenyl)sulfonylacetamide 4-chloro-1,3,5-trimethylpyrrolo[2,3-b]pyridine N-[(1S)-5-methylcyclohexa-2,4-dien-1-ylidene]-2-phenylsulfanylbenzamide 2-(2,6-dichlorophenyl)-N-[3-[(3S)-oxolane-3-carbonyl]-1,3-thiazolidin-4-yl]acetamide (5Z)-2-[4-bromo-3,5-bis(trifluoromethyl)phenyl]imino-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-4-one 2-fluoro-4-[1,3]thiazolo[5,4-c]pyridin-5-yl-N-[5-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]benzamide 2-[4-[(3S)-1,5-dimethylpiperidin-3-yl]piperazin-1-yl]quinoline 2-N,5-diphenyl-3,4-bis(1-pyridin-2-ylethenoxy)benzene-1,2-dicarboxamide 2-[(1R,2S)-2-aminocyclohexyl]oxy-4-methylphenol N-[3-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)phenyl]-6-piperidin-1-ylpyridazine-3-carboxamide 2-[3,5-bis(trifluoromethyl)phenyl]cyclopropan-1-amine N-[(1S)-1-[4-[7-amino-8-ethyl-6-(methoxymethyl)imidazo[1,2-b]pyridazine-3-carbonyl]phenyl]ethyl]acetamide 4-methyl-2-propyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 7-[3,5-difluoro-2-(trifluoromethyl)phenyl]heptanoic acid 4-(4-chlorophenyl)-2,3,6,7-tetramethylimidazo[1,5-a]pyridine 2-[4-[2-azidooxy-1-(4-tert-butylphenyl)ethoxy]phenyl]-5-methylthiophene N-[5-(1,2,3,6-tetrahydropyridin-4-yl)pyridin-2-yl]formamide 2-[4-methyl-3,5-bis(trifluoromethyl)phenyl]-1,6-naphthyridine N-(5,6-dimethyl-1,3-benzothiazol-2-yl)-6-[4-(trifluoromethylsulfonyl)phenyl]piperidine-3-carboxamide 4-[2-(1,3-dioxoisoindol-2-yl)ethoxy]pyridine-2-carboxamide N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-ethyl-2-[4-[(1-methoxycyclobutyl)methylamino]phenyl]-7-methylimidazo[1,2-a]imidazole-8-carboxamide [2-(azidooxymethyl)phenoxy]methanesulfonic acid 4-[3,5-dimethyl-1-(6-pyrrolidin-1-ylpyridazin-3-yl)pyrazol-4-yl]pyrimidine 4-(3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclohexane-1-carboxylic acid 1-[(2,5-dichlorophenyl)methyl]-3-hydroxy-3H-indol-2-one N-[[1-(4,7-dichlorobenzoyl)piperidin-3-yl]methyl]-2-fluoro-6-methoxybenzamide 2-cyclohexyl-N-(3,5-difluoropyridin-2-yl)sulfonylacetamide 1-(2,6-dimethylphenyl)pyrazole 3-ethyl-6-[4-(1-methoxypropan-2-yl)piperazin-1-yl]pyridazine 1-(5-methylfuran-2-yl)-3-[3-[4-[[3-methylidene-6-(trifluoromethoxy)-1,2-dihydroinden-2-yl]amino]piperidine-1-carbonyl]phenyl]urea N-[5-fluoro-4-[8-(2-methylpyrimidin-4-yl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]-7,8a-dihydronaphthalene-1-carboxamide 4-[1-(1H-indazole-5-carbonyl)piperidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-6-one 5-(2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)pyrimidine-2-carboxylic acid 2-(4-aminophenyl)-6,7-dimethoxychromen-4-one 2-[1,1-difluoro-5-(4-fluorophenyl)pentyl]-6-hydroxy-3H-isoindol-1-one 7-[4-(1,3-benzodioxol-5-yl)-6-chlorocyclohepta-2,4,6-trien-1-ylidene]-2H-azepine [2-amino-5-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)phenyl]methanol 5-[4,6-bis(2-pyridin-3-ylethynyl)-1H-benzimidazol-2-yl]thiadiazole 4-cyclohexyloxybenzenethiol 1-(4,5-dimethyl-1H-pyrazol-3-yl)-6-fluoro-7-piperazin-1-ylquinolin-4-one;hydrate 1-azido-3,7-dimethyl-4-[5-(2-pyrrolidin-1-ylethoxy)benzimidazol-1-yl]pyrazolo[3,4-d]pyrimidine 5-(3-bromo-4-fluorophenyl)-N-(4-cyclobutylpyridin-2-yl)pentanamide;1,1,1-trimethoxypropane 4-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)naphthalen-2-ol ethane;1-(3-methoxypropyl)-4-(trifluoromethylsulfanyl)benzene 1-azido-N,N-dimethyl-2H-indole-3-carboxamide N-[(E)-3-(4-hydroxyphenyl)propylideneamino]-3,5-dimethoxybenzamide 3-methyl-1-[2,4,6-tri(propan-2-yl)phenyl]sulfonylindole 1-benzyl-4-N-(5,6-dihydroquinolin-8-yl)-1,4-diazepane-3,4-dicarboxamide 3-[1-(methylamino)ethenyl]-4-propoxyaniline (NZ)-N-[[4-[2,6-bis(2-methylbutan-2-yl)phenoxy]phenyl]methylidene]hydroxylamine 1-[2,3-bis(2-butoxyethylsulfanyl)butan-2-yl]-4-methoxybenzene 7-(trifluoromethyl)-4H-pyrrolo[1,2-a][3,5]diazepine N-[2,3,5,6-tetrachloro-4-(chloromethyl)phenyl]acetamide 1-[4-[(2,6-dichlorophenyl)methyl]piperazine-1-carbonyl]-3H-pyridin-2-one 4-methyl-2,6-dipentoxybenzenesulfonic acid 3-[2,6-difluoro-4-(N'-hydroxycarbamimidoyl)phenyl]-1H-pyrazole-5-carboxylic acid 2-[(5S,10bR)-9-chloro-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol N-[(2S,3R)-1-(cyclobutanecarbonylamino)-2-methylhexan-3-yl]-1H-indazole-5-carboxamide N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-ylmethyl)pyrrolidine-2-carboxamide 2-[4-ethylsulfonyl-3,6-dioxo-1-(pyrazine-2-carbonyl)piperazin-2-yl]acetamide (3R)-N,N-diethyl-1-[2-(2-oxo-1H-pyrido[2,3-b][1,4]thiazin-7-yl)-6-phenylimidazo[1,2-a]pyridin-5-yl]pyrrolidine-3-carboxamide 4-(3-bromopyridin-2-yl)oxy-N,N-dimethylpyridine-2-carboxamide 4-azido-1-chloro-2-ethyl-3,6-dimethoxybenzene 4-(3-chlorophenyl)-2,5-dimethylfuran 1-[6-(4-chlorophenyl)pyrazin-2-yl]ethanone 2-[(E)-but-1-enyl]sulfanyl-4,6-dichloropyrimidine (4-nitrophenyl)-(3,4,5-trihydroxyphenyl)methanone 1-benzyl-5-chloro-3-propan-2-ylindole 4-(1H-indazole-5-carbonylamino)piperidine-1-carboxylic acid [6-[2,6-difluoro-4-(2-methylsulfonylethoxy)phenyl]-3-propanoylpyridin-2-yl]boronic acid 3-(4,5-diamino-2H-triazolo[4,5-i][1]benzazepine-9-carbonyl)benzoic acid 2-azido-6-(4-fluorophenyl)sulfanyloxane 3-(4,5-dihydro-1H-imidazol-2-ylamino)benzaldehyde 3-[(6-chloropyridin-3-yl)methylideneamino]oxypropan-1-amine 2-chloro-N,N-dimethyl-5H-indolo[3,4-d]pyrimidin-6-amine;3,3-difluoro-1,4-bis(methoxymethyl)pyrrolidine N-[2-(N'-hydroxycarbamimidoyl)phenyl]-2,3-dimethyloxolane-2-carboxamide N-(2-azidopyridin-3-yl)-4-fluorobenzamide 2,5-bis[(2-methylpropan-2-yl)oxycarbonyl]terephthalic acid N-(2,6-dibromopyridin-4-yl)-N-[4-(quinoxalin-2-ylsulfamoyl)phenyl]hexadecanamide 2-chloro-4-[1-methyl-3-(trifluoromethoxy)pyrazol-4-yl]benzonitrile 2-[(6-chloropyridin-3-yl)-ethenylsulfonylamino]decanoic acid 6-[3-[2,6-di(propan-2-yl)anilino]penta-1,4-diynyl]benzene-1,2,3,5-tetrol 7-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-9-(4,6-diphenyl-1,3,5-triazin-2-yl)pyrido[3,4-b]indole 1-N,1-N'-bis[2-(pyridine-4-carbonyl)phenyl]ethenedihydrazide 1-[4-(2,6-diphenylpyridine-4-carbonyl)phenyl]ethanone 5-(azidomethyl)-4-[1,3]dioxolo[4,5-b]pyridine 4-[(5Z)-5-[[2-methoxy-5-nitro-4-(trifluoromethyl)phenyl]methylidene]-4,4-dimethyl-2-sulfanylideneimidazolidin-1-yl]benzenecarboximidamide 2-[4-(chloromethyl)phenyl]benzo[f]chromen-1-one 2-(6,7-dimethoxyquinazolin-4-yl)oxy-N,N'-diethylpropane-1,3-diamine 1-N,3-N-bis[4-chloro-2-methoxy-5-(morpholine-4-carbonyl)phenyl]propanediimidamide (5S,7R)-N-[1-(4-chlorophenyl)ethyl]-7-(trifluoromethyl)-5-(3,4,5-trimethoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide 2-methyl-N-(7H-pyrrolo[3,4-b]pyridin-1-ium-6-ylidene)propanamide (2R)-3-phenyl-1-[(4S)-4-propan-2-yl-2,5-diazabicyclo[10.4.0]hexadeca-1(12),13,15-trien-14-yl]propan-2-ol 3-N-[1-(5-aminothiophen-2-yl)ethylideneamino]thiophene-2,3-diamine (4-bromo-3,5-dimethoxyphenyl)-[2-[5-(trifluoromethyl)pyrimidin-2-yl]azepan-1-yl]methanone 1-(2-bromophenyl)sulfanylnaphthalene N-[4-(diethylamino)phenyl]-3,5-dihydroxybenzamide 2,6-dichloro-N-[(Z)-1H-pyrrol-2-ylmethylideneamino]pyridine-4-carboxamide 2-[5,6-dimethyl-4-[(Z)-prop-1-enyl]pyridin-3-yl]iminopentanal 2-(3,4-dichlorophenyl)-2-hydroxy-2-phenylacetamide N-[2-amino-5-(4-chlorophenyl)phenyl]formamide 3-fluoro-2,4-diiodobenzoate (6R)-3-ethylsulfanyl-6-[4-(trifluoromethoxy)phenyl]-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-1-one 2-amino-4-[4-(cyclopropylmethoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile N-[(3-cyanophenyl)methyl]-2,5-dihydroxy-6-oxo-1H-pyrimidine-4-carboxamide 2-[2-(4,4-difluoropiperidin-1-yl)ethoxy]-7-(5,6-dihydrofuro[3,2-b]thiophen-3-yl)quinoline 3-hydroxy-2-[4-(7H-purin-8-ylmethoxy)phenyl]-1,5,6,7,8,9-hexahydrocyclohepta[f]benzimidazole (3aR,7aS)-2-benzylsulfonyl-N-pyrimidin-5-yl-1,3,3a,4,6,7-hexahydropyrano[3,4-c]pyrrole-7a-carboxamide;formic acid ethane;[(5R)-3-methyl-2,6,10-triazabicyclo[10.4.0]hexadeca-1(16),12,14-trien-13-yl]-phenylmethanone N-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonyl)phenyl]thiophene-3-sulfonamide 6-(2,3-dihydroimidazo[1,2-c]quinazolin-9-yloxy)heptanoic acid (6-chloropyridin-3-yl)-[4-[1-(4-cyanophenyl)sulfonylpyrrolo[2,3-b]pyridin-5-yl]pyrazol-1-yl]carbamic acid 4-[2,5-difluoro-4-(trifluoromethyl)phenyl]-1H-tetrazol-5-one 1-[(3R)-5,7-dibromo-2,3-dihydro-1H-inden-4-yl]ethanone [6-(dimethylamino)pyridine-3-carbonyl]oxyboronic acid 1-[(3R)-5-azido-2,3-dihydro-1,4-benzodioxin-6-yl]pyrrolidine 5-[3,4-bis(fluoromethoxy)phenyl]-2-phenylmethoxyaniline 3-(3,4-dihydroxyphenyl)-5-[3-(2H-triazol-4-ylmethoxycarbonylamino)propanoyl]furan-2-carboxylic acid 2-[N-(carboxymethyl)-4-fluoroanilino]acetic acid N-[4-amino-3-(3H-benzimidazole-5-carboximidoyl)phenyl]-6-pyridin-2-ylcyclohepta-1,3,5-triene-1-carboxamide 4-(1,3-benzodioxol-5-yl)-2-[4-[(3E)-hexa-1,3,5-trien-3-yl]oxyphenyl]-N'-methylbutanimidamide N-[(3-fluoro-4-methylphenyl)carbamoyl]propanamide 1-[(5S)-2,8-dimethyl-3,4,6,10b-tetrahydro-1H-pyrazino[2,1-a]isoindol-5-yl]propan-1-one N-[(3,4-difluorophenyl)methyl]-4-oxo-1H-quinoline-7-carboxamide 2-(3,4,5-trimethoxyphenyl)quinoline-7-carboxamide (2S)-N,3-dimethylbutanamide;ethane;8-methoxy-5-methyl-7-methylidenebenzo[d][2]benzoxepin-6-one 3-[(4S,5R)-2-amino-6-chloro-5-methyl-4-phenylmethoxyhexanoyl]-N-[2-(dimethylsulfamoyl)ethyl]-N-methyl-1H-indole-7-carboxamide 2-(dimethylamino)-N-[4-[(7Z,9E,11E)-5-ethenylimino-10,12-dihydroindolo[3,2-a]carbazol-12-yl]phenyl]acetamide 6-(cyclohexylamino)pyridine-2,3-dicarboxylic acid 1-(1-azido-4,5-dimethylpyrazol-3-yl)-2-methoxypyridin-1-ium 5-[(E)-2-(2,4-dichlorophenyl)ethenyl]-1H-pyrazole 5-[2-(benzenesulfonyl)ethyl]-N,1H-pyrazole-3-carboxamide 3-[(E)-5-amino-5-iminopent-2-enoyl]benzonitrile;butane 4-(2,6-dichlorophenyl)-N-[1-[(E)-3-[7-[dimethylamino(piperidin-4-yl)amino]quinolin-5-yl]prop-2-enoyl]pyrrolidin-3-yl]butanamide 2-azidooxy-5,6-bis(propylamino)benzo[de]isoquinoline-1,3-dione (3S,4R)-1-[2-(diethylaminomethyl)pyrimidin-5-yl]sulfonyl-3,3,6-trimethylpiperidin-4-ol 5-[(E)-1,2-diphenylethenyl]pyridine-3-carboxamide (3Z)-5,6-dimethoxy-3-[[2-(4-methylphenyl)imino-1,4-dihydroimidazol-3-ylidene]amino]chromen-2-one N-[4-[3,5-dichloro-2-(1-oxo-2H-isoquinolin-7-yl)phenoxy]-6-methoxyquinolin-7-yl]piperidine-4-carboxamide (2S)-2-(2,3,5,6-tetrabromophenyl)oxirane (2S,4R)-N-[[1-(benzenesulfonyl)piperidin-3-yl]methyl]-4-hydroxypyrrolidine-2-carboxamide [1-[(3,5-difluorophenyl)methyl]pyrazole-4-carbonyl]azanium 2-[2,5-dioxo-4-(3-phenylpropyl)pyrrolidin-1-yl]acetic acid 2-[4-(8,9,11-trioxonaphtho[1,2-g]isoquinolin-6-yl)sulfanylphenyl]acetonitrile N-[3,5-dimethyl-4-[[(1R)-1-phenylethyl]carbamoylamino]cyclohexa-2,4-dien-1-ylidene]acetamide 2-[7-(4,6-dichlorobenzotriazol-1-yl)heptanoylamino]acetic acid N-[6-(1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinolin-1-yloxy)pyridin-2-yl]-2-chlorobenzamide 4-(2-methyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carbonyl)oxy-1H-triazole-5-carboxylic acid 5-azido-3-(1,2-benzoxazol-6-yl)furan-2-carboxylic acid 1-[(4R)-3,3-difluoropiperidin-4-yl]indole 2,6-dimethyl-4-(2-pyridin-3-ylethynyl)phenol 3-(2,6-difluorophenyl)-4-[4-fluoro-5-(hydroxymethyl)-1H-pyrazole-3-carbonyl]piperazin-2-one 2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine;4-(2H-thieno[3,2-b]pyrrol-5-yl)benzoic acid N-[2-[4-(4-aminobutyl)piperidine-1-carbonyl]imidazo[1,2-a]pyridin-6-yl]formamide (3E)-1-[4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxy-2,6-diethylphenyl]-3-[3-ethylidene-8-methyl-4-[3-(trifluoromethyl)phenyl]iminocyclohexa-1,5-dien-1-yl]penta-1,3-dien-1-ol N-[5-(2,3-dihydro-1H-indene-2-carbonyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl]cyclopentanecarboxamide;hydrochloride N-[2-hydroxy-4-(trifluoromethyl)phenyl]-3-(3-hydroxypyrrolidine-1-carbonyl)piperidine-1-carboxamide 4-(2,3,5,6-tetrafluorophenoxy)piperidine 2-(3,4-difluorophenyl)-1H-benzimidazole-4-carboxamide 3-[2,6-di(propan-2-yl)phenyl]-5-methylbenzonitrile [(E)-1-(2,4-dihydroxyphenyl)ethylideneamino]urea [(2R)-2-(difluoromethyl)azetidin-1-yl]-[5-(3,4,4a,5,6,7,8,9,10,11,12b-decahydrophenanthren-2-yloxymethyl)furan-2-yl]methanone 4-[4-methyl-2,6-bis(trifluoromethyl)phenyl]pyrimidine;2-(3-oxobutanoylamino)acetic acid 1,2-dimethyl-N-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide 4-[2-(3,5-diphenylphenyl)phenyl]-6-[9-ethylcarbazol-2-yl-1-[(Z)-prop-1-enyl]benzo[e]indol-7-yl]pyrimidine (2R)-3-methyl-4-oxo-4-[[4-(thiophen-2-ylsulfanylamino)phenyl]sulfonylamino]butanoic acid 3-cyclohexa-1,5-dien-1-yl-6-methylidene-4-propylthieno[2,3-b]pyridine (1-ethyl-2,6-dioxopiperidin-3-yl)-[6-[[4-[(2-methoxyphenyl)methylideneamino]benzoyl]amino]hexan-3-yl]carbamic acid N-[2-(4-chlorophenyl)ethyl]-3,3-dimethylbutanamide 3-[4-[[2-[4-(1,1-dioxothietan-3-yl)oxyphenyl]-5-hydroxypyridine-4-carbonyl]amino]benzoyl]-N'-methylbenzohydrazide N-[1,3-di(propan-2-yl)pyrrolidin-4-yl]-7-methoxyquinoxalin-6-amine 1-[4-(cyclopropylmethylamino)-6-fluoroquinolin-3-yl]ethanone [3-[4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethoxy)phenyl]piperidin-1-yl]-thiomorpholin-4-ylmethanone;dihydrochloride N-(4-bromobutan-2-yl)-N-[4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]nonanamide (2E)-6-(3,4-dichlorophenyl)-N'-hydroxy-1-methanimidoyl-2-[3-(piperidine-1-carbonylamino)propylidene]pyridine-3-carboximidamide 6,7-dihydro-5H-pyrazolo[3,4-f][1]benzazepine-9-carboxylic acid 2-(6-hydroxynaphthalen-1-yl)-5-[3-(7-methoxy-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)propylsulfonylamino]benzoic acid 3-(4-bromophenyl)sulfonyl-1H-triazole 1,3-difluoro-2-iodobenzene;ethane 2-methylsulfonyl-4H-furo[3,2-b]pyridine 2-[(1R)-6-[[4-[2-cyclopropylethynyl(difluoromethoxy)methyl]triazol-1-yl]methyl]-3,4-dihydro-1H-isochromen-1-yl]acetic acid 3-azidooxy-2,6-dichloropyridine 2-methoxy-N-methyl-4-[7-(methylamino)-4H-azepin-3-yl]benzamide 2-(5-fluoroquinolin-8-yl)oxypyridine-3-carboxamide 2-benzyl-N-methyl-1-phenylpropan-2-amine 4-[4-(3,5-difluorophenyl)sulfonylbutyl]benzenesulfonamide 3-[3-(2,6-dimethylphenoxy)-1H-pyrazole-5-carbonyl]pyrrolidine-1-carboxylic acid (3R,4S)-3-(2-oxochromen-7-yl)oxycarbonylpiperidine-4-carboxylic acid 6-amino-2-[1-(3,3-dimethylbutanoyl)pyrrolidin-3-yl]-3H-quinazolin-4-one 5-(2-bromo-3,4-dihydroxy-6-methylphenyl)-1-methylpyrazole-3-carboxylic acid 4-[(7R)-8-[2-(1H-imidazol-5-ylmethoxy)ethyl]-11-(methanesulfonamido)-2,3,9,12-tetrazatricyclo[6.3.1.04,12]dodeca-1,4(12),5,7,10-pentaen-7-yl]benzamide 1-[3-(3,5-dimethyl-4H-imidazol-2-yl)phenyl]-N'-ethoxy-1-(2-fluoro-6-methylphenyl)ethane-1,2-diimine ethane;N-methylethanamine;(3E,5Z)-4-methylidene-2-propylhepta-1,3,5-triene;1-[2-(1H-pyrrol-3-yl)acetyl]piperidine-2-carboxamide 2-[3,4-dimethoxy-5-[(5-oxo-7-propanoyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)amino]phenyl]ethyl-trimethylazanium 1-[2,5-di(propan-2-yl)phenyl]-3,6-dihydro-2H-quinoline 3-[2,6-dichloro-4-(1H-pyrazol-5-yl)phenyl]oxolan-2-amine [2-(1H-indol-3-yl)-4,5-dihydrothieno[2,3-g]indazol-7-yl]boronic acid N-[(5E)-3,4-bis(phenylmethoxy)octa-1,5-dien-2-yl]-4-chloro-N-ethylbenzenesulfonamide N-(2-chlorophenyl)-N'-[(2S)-1,1-dicyclopentylpropan-2-yl]-4-methoxy-3,5-bis(trifluoromethyl)benzenecarboximidamide N-[2-(2,4-dioxocyclohexyl)-1,3-dioxoisoindol-5-yl]ethanesulfonamide 2-[2,6-dimethyl-4-(4-phenylphenyl)phenyl]propan-1-amine N-(1,3-dihydroxypropan-2-yl)-5-methoxy-2,8-dimethyl-2,3-dihydronaphthalene-1-carboxamide 2-chloro-4-[6,7-difluoro-1-(3-methylphenyl)sulfonylindole-3-carbonyl]oxybenzoic acid 4-[azido(phenyl)methyl]benzenesulfonamide 3-[4-(trifluoromethyl)phenyl]sulfinylbenzaldehyde 1-bromo-3-methyl-5-nitro-2,4-diphenylbenzene;toluene 5-chloro-3-ethyl-2-[(1R)-4-(propan-2-ylamino)cyclohexa-2,4-dien-1-yl]indole-1-carboxylic acid (4R)-6,10-difluoro-5-methoxycarbonyl-1,2,3,4-tetrahydroanthracene-9-carboxylic acid 2-chloro-4-[3-(1-fluoroethyl)-1H-pyrazol-5-yl]phenol 3-(2,4-dimethoxyphenyl)-N'-ethyl-6-hydroxy-N-[2-(5-propan-2-yl-1,3-oxazol-2-yl)ethyl]pyridazine-4-carboximidamide 1-azidooxy-2-methoxybenzimidazole 5-methyl-2,7,9,12-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5-triene;hydrochloride 1-[4-[bis(2-methylpropyl)amino]phenyl]-3,9-dihydrocyclohepta[c]pyridine-4-thione 3-bromo-5-fluorothieno[3,2-b]pyridine 3-(2,6-difluorophenyl)-4-hydroxy-5-methylbenzoic acid 2-azidooxy-1,3-diphenylbenzene 2-fluorobuta-1,3-diene;N-methylhexan-2-amine;5-(3-methylphenyl)pyrimidine-4,6-diamine 5-[3-(4-methylcyclohexa-1,3-dien-1-yl)phenyl]-2H-tetrazole (3R)-6'-chlorospiro[1,2-dihydroindene-3,4'-piperidine] ethane;5-methyl-4,6-diphenylpyrimidine 2-amino-5-[4,4-difluoro-3-(methoxyiminomethyl)butanoyl]-6-(4-methylsulfonylphenyl)-1H-pyrrolo[2,3-f]indazole-7-carboxylic acid 1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-[6-[5-(furan-3-yl)-2H-pyrazolo[3,4-b]pyridine-3-carbonyl]-2,3-dihydro-1,4-benzodioxin-8-yl]ethanone 3-[(4-bromophenyl)methoxy]-N'-hydroxypyridine-2-carboximidamide 4-(2-bromobutyl)naphthalene-1,7-disulfonic acid N-[5,6-bis(4-chlorophenyl)pyridin-3-yl]ethanesulfonamide 2-(4-azidobutanoylamino)benzenesulfonic acid 4-[N'-(2,6-dichlorobenzoyl)carbamimidoyl]-3,5-dimethoxybenzamide 5-amino-4-[7-[(3-chlorophenyl)methoxy]-2,3-dihydro-1H-inden-4-yl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 3-azido-1,2,4,5-tetrafluoronaphthalene 2-[3-methylbutyl(2H-tetrazol-5-yl)amino]octanoic acid 7,8-difluoro-2H-quinoline-1-sulfonamide 3-(6,7,8,9-tetrahydroimidazo[1,5-a]azepin-5-yl)-N'-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)propanehydrazide 4-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-methoxycarbonylamino]benzenesulfonic acid N-[(1S,2R)-2-[(1R)-5-chloro-8-fluoro-1H-naphthalene-1-carbonyl]cyclohexyl]methanesulfonamide 5-[(4-aminophenyl)diazenyl]-1,3-dimethylimidazole-2-thione (NZ)-N-[1-(4-fluorophenyl)propylidene]hydroxylamine;5-[3-[7-(2,2,6,6-tetramethyloxan-4-yl)oxyhepta-1,3,5-trien-3-yl]-5-(trifluoromethyl)phenoxy]pyridine-3-carbonitrile 2-(2,4,6-trichloro-N-hexylanilino)decanoic acid [(2R,3S)-2-[4-methyl-6-[(5-phenylthiophen-2-yl)methoxy]pyridin-3-yl]oxolan-3-yl]methanol 1-(5-methyloxolan-2-yl)-5-oxo-N-phenylpyrazole-3-carboxamide 3-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]butan-2-one;2-(4,6-dimethoxypyrimidin-2-yl)-2-hydroxyacetamide 4-fluoro-2,5-dimethyl-N-[6-(3,3,3-trifluoropropanoyl)pyridin-2-yl]benzamide N-[[4-(methanesulfonamido)phenyl]methyl]-3,4,5-trimethoxybenzamide 4-benzyl-5,6-dihydro-[1]benzothiepino[3,2-d]pyrimidine 3-[2-ethoxy-4-(trifluoromethyl)phenyl]oxirane-2,2-dicarbonitrile 2-[2-(dimethylamino)ethoxy]-6-methyl-N-quinolin-5-ylbenzamide 1-ethyliodanuidyl-3-fluorobenzene [2-[4-(1H-indazole-3-carbonylamino)phenyl]pyrrolidin-1-yl]borinic acid 1-[4-(3,5-dimethylcyclopentanecarbonyl)phenyl]-3-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]urea N-[2,4,6-tri(propan-2-yl)phenyl]dibenzofuran-3-amine (2S)-2-[(5R)-3,5-dimethyl-4,5,6,7-tetrahydroindazol-1-yl]-3-phenylpropanamide 5-azido-1,3,3a,4,6,6a-hexahydrocyclopenta[c]pyrrole 1-[(E)-3-methoxyprop-2-enyl]sulfonyl-4-propan-2-ylbenzene [(3-hydroxy-2,4-dimethylphenyl)sulfonylamino]urea 4-[4-(2,5-dihydrofuran-3-ylsulfonyl)piperazine-1-carbonyl]benzonitrile 6-[6-(3,4-dichlorophenoxy)pyridin-2-yl]sulfonyl-2-phenyl-1,3,5-triazine 2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-ylmethylideneamino)ethanol 2-[4-[[(3S,4R)-1-benzyl-3-propan-2-ylpiperidin-4-yl]methoxy]phenyl]sulfanylacetic acid N-azido-3,5-difluorobenzenesulfonamide 2-(3,5-dichlorophenyl)-1-[4-(6-fluoro-1H-indole-2-carbonyl)piperazin-1-yl]ethanone 3-chloro-N-[(1R,2S)-2-hydroxycyclohexyl]pyridine-4-carboxamide N-azido-N,2-dimethyl-6-(trifluoromethyl)aniline N-cyclopropyl-2,6-difluoro-4-[(4E)-4-[[5-(hydroxymethyl)oxolan-3-ylidene]hydrazinylidene]hexa-1,5-dienoxy]benzamide 5-(4-methoxyphenyl)-7-methylsulfanyl-1H-thieno[3,2-d]pyrimidine-2,4-dione 4-[[6-cyclopropyl-3-ethoxycarbonyl-5-(3-fluorobenzoyl)pyridine-2-carbonyl]amino]benzoic acid (5R)-2-[3-[(1S)-cyclohexa-2,4-dien-1-yl]propanoylamino]-N-(oxolan-2-ylmethyl)-5-phenyl-3,7-dihydro-1H-1,4-benzodiazepine-6-carboxamide 1-(3,5-dichloropyridin-4-yl)-2-[[1-[[4-(trifluoromethoxy)phenyl]methyl]benzimidazole-2-carbonyl]amino]benzimidazole-5-carboxylic acid 3-amino-N,2-dimethylbenzimidazole-5-carboxamide N-[4-[3-fluoro-5-methoxy-2,6-dimethyl-4-(oxan-4-yl)phenyl]pyridin-2-yl]propanethioamide 2-chloro-N-(4-methylphenyl)-5-nitropyrimidin-4-amine (4Z)-3,5-diamino-N-[5-[2-[4-[hydroxy-[4-(methylaminomethyl)phenoxy]amino]piperidine-1-carbonyl]pyridin-4-yl]oxy-6-oxocyclohexa-1,4-dien-1-yl]pentanamide 4-[(E)-[3-chloro-5-ethoxycarbonyl-6-methyl-2-[(4S)-4-phenylpentanoyl]oxypyridin-1-ium-1-ylidene]methyl]cyclohexane-1-carboxylic acid 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-N'-methanimidoyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboximidamide [2-[2,4-difluoro-3-(2H-tetrazol-5-yl)phenyl]cyclopropyl]methanamine N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-methylpyridine-3-carboxamide 2-(3-methoxy-4,5-diphenylpyrazolo[3,4-b]pyridin-1-yl)-1,3,4-oxadiazole 3-[(4Z,8E)-11-methyldeca-1,4,8-trien-4-yl]benzoic acid [(1R)-2-(4-cyclopentyloxyphenyl)-1-[3-fluoro-5-[3-(4-methylpiperazin-1-yl)propoxy]phenoxy]ethyl]oxidanium N-[[2-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)pyridin-3-yl]methyl]-4-phenylbutanamide 4-(2,3-dimethylbenzimidazol-5-yl)sulfonylphenol (Z)-3-hydroxy-2-[4-methoxy-6-oxo-1-[[5,5,5-trifluoro-1-[4-(3-hydroxypropyl)phenyl]pentan-2-ylideneamino]methyl]pyridin-3-yl]prop-2-enenitrile 3-methyl-5-(2-methylbutanoylamino)benzenesulfonic acid 1-[1,4-dimethyl-2-(4-phenylbut-3-enyl)-5-propan-2-ylidenecyclohexa-1,3-dien-1-yl]oxy-3-ethenyl-5-propan-2-ylbenzene 2-(4-chlorophenyl)sulfanyl-3H-pyrido[3,4-d]pyrimidine [1-[(4-chlorophenyl)methyl]indol-3-yl]-[(2R,6S)-6-hydroxyoxan-2-yl]methanone 2-(4-ethyl-3,5-dimethoxyphenyl)acetic acid 4-methyl-2-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]quinoline 5-chloro-4-[1-(2-cyclopropyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperidin-3-yl]oxy-2-fluorobenzonitrile 2-[3-fluoro-4-(trifluoromethyl)phenoxy]-5-(1,1,1,3,3-pentadeuteriopropan-2-yloxymethyl)pyridine N-[4-(diethylamino)phenyl]-5,6,7,8-tetrahydroindolizine-3-carboxamide;ethane 4-[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6-one [(4-anilinophenoxy)-oxidophosphinothioyl]oxymethylphosphonic acid 2-[4-(8-amino-1,3-dimethylimidazo[1,5-a]pyrazin-6-yl)phenyl]propanoic acid;N-(oxetan-3-ylidene)hydroxylamine 2-(hydroxymethyl)-6-[2-(4,5,6,7-tetrahydro-1H-indazol-5-ylamino)pyrimidin-4-yl]-3,4-dihydro-2H-chromen-8-ol N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[4-hydroxy-5-(indole-1-carbonyl)-2-oxo-1,3-thiazolidin-3-yl]acetamide N-[1-[4-(3,4-dichloroanilino)-7-ethoxyquinazolin-6-yl]piperidin-4-yl]acetamide 1-(4-propanoylpiperazin-1-yl)-2-[(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)methoxy]ethanone 2-hydroxy-5-(N-propylanilino)benzoic acid N-[5-[4-fluoro-3-[7-(3-methylphenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]pentanamide 4-[2,6-dichloro-3-(methanesulfonamido)phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile N-[3-amino-4-(2,5-difluorophenoxy)cyclohexyl]-1,3-benzothiazole-6-sulfonamide 6-(4-benzylpiperazine-1-carbonyl)-5-methoxy-3H-1,3-benzoxazol-2-one 2-[3-chloro-5-(2,6-difluorophenyl)pyridin-4-yl]sulfanyl-4-methyl-1H-pyrimidin-6-one 1-methyl-6-(3,5,6-trifluoropyridin-2-yl)cyclohexa-3,5-diene-1,3-dicarboxylic acid 2-[2,5-dimethyl-4-(3-oxobutoxy)phenyl]acetic acid 2-ethoxy-N-[(4S)-4-hydroxypentan-2-yl]-5-[2-[[1-[4-(trifluoromethoxy)phenyl]pyrazol-3-yl]amino]pyrimidin-4-yl]benzamide 5-chloro-2,3-di(piperidine-1-carbonyl)benzaldehyde 4-(3,6-dichlorocarbazol-9-yl)benzaldehyde;2,4-dihydroxypentanal 2,3-diethoxycyclohepta-1,3-diene;4-(N-methylanilino)aniline N-(2,4,6-trimethylphenyl)dibenzofuran-1-amine 1,2-bis(2,6-dimethylphenyl)hydrazine;(4S)-3-methoxy-4-methylpiperidine N-[5-[[6-(3,4-dihydropyridin-5-yl)-1H-benzimidazol-2-yl]methoxy]-1H-indazol-3-yl]furan-2-carboxamide 2-[3-amino-6-(2,4-difluorophenyl)isoquinolin-5-yl]oxyacetonitrile (2S,3aS)-1-[2-[4-methyl-5-[(2Z)-2-[(6E)-7-methyliminoocta-1,3,6-trien-3-ylidene]hydrazinyl]-2H-pyridin-1-yl]acetyl]-N-propan-2-yl-3,3a,4,9b-tetrahydro-2H-chromeno[4,3-b]pyrrole-2-carboxamide N-(4-chlorobutyl)-1,3-thiazol-2-amine 2,4-diiodo-3-methoxycarbonylbenzoic acid 4-[2-(4-bromophenyl)butanoyl]-1,3,5-trimethylpyrrole-2-carboxylic acid 2-chloro-N-methylaniline;3-(4-formamidoanilino)-5-oxobenzo[b][1,8]naphthyridine-6-carbonitrile 2-[3-(4,5-dihydroimidazol-1-ylmethoxy)phenyl]ethanol 6-(2-azidophenyl)-1,3-dimethylpyrazolo[3,4-d]pyrimidin-4-amine 1-[2-[5-(2,6-difluorophenyl)-3H-1,4-benzothiazepin-2-yl]ethyl]-N,N-dimethylpiperidine-4-sulfonamide [4-(4-methoxyphenyl)piperazin-1-yl]-[4-methyl-3-[2-(quinolin-6-ylamino)acetyl]phenyl]methanone 3-[2,6-dichloro-4-(trifluoromethyl)phenoxy]oxolane 5-(4-azidophenyl)-4,5,6,7-tetrahydro-1H-indazole 4-amino-3-(3,5-dimethoxyanilino)butanamide;N'-methylmethanediamine 5-(2,3-dimethoxyphenyl)pentan-2-one 2-chloro-N-[4,5-difluoro-3-(trifluoromethyl)-1H-pyrazol-5-yl]pyridine-3-carboxamide 5-[5-(3,4-dimethoxyphenyl)furan-2-yl]-1H-pyrazole [3,5-bis(trifluoromethyl)phenyl]-[4-(4-propan-2-ylphenyl)piperazin-1-yl]methanethione 4-amino-6-(methoxycarbonylamino)pyridine-3-carboxylic acid 1-(2,3-dihydro-1H-inden-2-yl)-N-[6-(5-methoxypyridin-3-yl)cinnolin-3-yl]piperidine-4-carboxamide N-methylsulfonyl-N-(3,4,5-trifluorophenyl)butanamide 1-[5-(azidomethyl)-2,4-dichlorophenyl]imidazole 4-[5-(4-tert-butylphenyl)sulfonylpentanoyl]benzonitrile 1-[2,5-bis(trifluoromethyl)phenyl]piperidine (2S)-1-N,2-N,3-N,4-N,4,5,6-hexamethyl-2-(9-oxothioxanthen-2-yl)heptane-1,3,4-tricarboxamide 4-[[3,5-dimethyl-4-(1-methylidenepyridazin-1-ium-4-yl)oxyphenyl]carbamothioylamino]benzoic acid N-[2-(3,4-dimethoxyphenyl)ethyl]-6-(4-fluorophenyl)benzo[b][1,4]benzothiazepine-3-carboxamide (3S,6R)-4-azido-5-bromo-N-[[2,6-dichloro-4-(trifluoromethyl)phenyl]methyl]-1-propanoyl-6-propan-2-yloxycarbonylpiperazine-2-carboxamide 4-(6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl)-N-[1-[3-methoxy-2-(trifluoromethyl)phenyl]ethyl]-6-pyrrolidin-1-ylpyridazin-3-amine (5E)-2-(4-chlorophenyl)imino-5-[(3,7-dimethyl-1,3-benzothiazol-3-ium-2-yl)methylidene]-1,3-thiazolidin-4-one 1,3-diphenyl-5-prop-2-enoxybenzene 4-[(4-fluorophenyl)sulfonylmethyl]-3,5-dioxocycloheptane-1-carboxylate 2-[2-(hydroxymethyl)phenoxy]-4-nitrophenol 2,4-dichloro-N-(4-phenoxyphenyl)aniline N-[3-(4,5-dimethylimidazol-1-yl)propyl]-2,4-dihydroxy-N-methyl-6-oxocyclohexa-2,4-diene-1-sulfonamide N-[(2R)-1-[4-(azidomethyl)phenyl]-5,7-dichloro-3,4-dihydro-2H-quinolin-6-yl]cyclopentanecarboxamide 4-[azido(fluoro)methyl]-5,7-difluoroquinoline 5-chloro-N-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]pyrimidine-4-carboxamide N-[2,5-dimethyl-4-(1-thiophen-3-ylpyrazol-4-yl)phenyl]formamide 2-(2,4-dichlorophenyl)-1-[4-(pyrimidin-5-ylmethoxy)-3H-indol-2-yl]ethanone N-[1,1-dioxo-2-(trifluoromethyl)thiolane-3-carbonyl]quinoline-8-sulfonamide 2-[7-(3,4-difluorophenyl)-2-oxo-1,6-naphthyridin-3-yl]-N-methyl-2-(1-propan-2-ylpiperidin-3-yl)acetamide 2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-ium-3-yl)-4,5-dimethoxy-N-propan-2-ylpyrrolo[3,2-d]pyrimidine-7-carboxamide 2-[6,7-dimethyl-4-oxo-3-(pyridin-4-ylmethyl)quinazolin-2-yl]sulfanyl-N-[2-(1H-indol-3-yl)ethyl]acetamide;methane 2-cyclohexyl-N,N-dimethyl-3H-imidazo[4,5-c]pyridine-7-carboxamide 2-hydroxy-4-methyl-5-[(1R,2S)-2-methyl-2,3-dihydro-1H-inden-1-yl]-N'-propan-2-ylbenzenecarboximidamide N-[6-(6,7-dihydro-4H-pyrano[2,3-c]pyrazol-1-yl)pyridin-2-yl]-3,5-bis(trifluoromethyl)benzamide N-benzyl-5,6-diphenyl-1,2,4-triazin-3-amine N-[(4-fluorophenyl)methyl]spiro[1,4-dihydroquinoline-3,2'-cyclopropane]-2-imine N-(4,5-dichloro-2-methylphenyl)-2-[(1,3-dimethyl-6-propanoyloxybenzimidazol-1-ium-2-yl)amino]acetamide 5-[(3R)-3-methylmorpholin-4-yl]-2-quinolin-8-ylbenzenesulfonamide 2-[(1,3-dimethylpyrazol-4-yl)sulfonylamino]-N-(5-phenylpentan-2-yl)acetamide (3R)-2,7-dimethyl-10-[4-[3-(methylaminosulfanyl)phenyl]piperazin-1-yl]-1H-phenothiazine-3-carbohydrazide;ethane 2-(4-chlorophenyl)imino-5-[(4-hydroxyphenyl)methylidene]imidazolidin-4-one 1-[4-(2,3-dichlorophenyl)-5,6-dimethylpyrimidin-2-yl]piperidine-4-carboxylic acid N-[3-chloro-4-(4,5-dihydroimidazol-1-yl)phenyl]formamide;formic acid 4-bromo-5-(5,6-difluoro-2-hydroxy-3-methylphenyl)pyridine-2-carboxylic acid (1Z)-2-N',3-N'-dibenzyl-1-N-prop-2-ynylspiro[1-benzothiophene-2,9'-xanthene]-1',3',6-triamine;toluene 2-[N-(benzenesulfonyl)-2,4-difluoroanilino]decanoic acid 3-[4-(1,1-difluoroethyl)phenyl]-7-[3-(dimethylamino)prop-1-ynyl]-5H-pyrrolo[2,3-b]pyrazine-2-carboxamide N-[2-[2-[(1R)-6-chloro-2,3-dihydro-1H-inden-1-yl]acetyl]phenyl]-2-methoxyethanesulfonamide 1-cyclopropylsulfonyl-3-[6-(4-methoxypyrimidin-5-yl)isoquinolin-3-yl]urea 5-cyclopropyl-N-methoxy-N,2,4-trimethylbenzamide 4-(3,3-dimethylazetidine-1-carbonyl)-N'-[1-[2-fluoro-5-methoxy-4-[(pyridin-4-ylamino)methyl]phenyl]ethylideneamino]-5H-pyrimidine-4-carboximidamide 1-cyclohexyl-2-[4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)piperazin-1-yl]ethanone 1-(5-tert-butylpyrazole-1-carbonyl)-N-(5,6-dimethylcyclohepta-1,4,6-trien-1-yl)piperidine-4-carboxamide N-cyclobutyloxy-4-(3-hydroxypropanoylamino)-2-methylbenzamide (4S)-4-tert-butyl-1-(4-ethoxyphenyl)-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 6-(2,5-difluorophenyl)-3-ethylsulfanyl-7-propanoyl-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one N-azido-6-(2,2,2-trifluoroethyl)thieno[3,2-d]pyrimidin-4-amine (5-azidooxypentylsulfinyl)benzene 2-(4-butyl-5-methoxycarbonyl-6-oxo-1H-pyrimidin-2-yl)acetic acid [3-(1,1-difluoroethyl)phenyl]urea;(E)-N'-[4-[3-[2-(dimethylamino)ethoxy]anilino]pyrido[3,4-d]pyrimidin-6-yl]prop-2-enehydrazide N-[5-tert-butyl-2-(methylamino)pyridin-3-yl]sulfonyl-6-[2,4-difluoro-5-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)phenyl]pyridine-3-carboxamide 1-[4-(2,3-dihydro-1H-tetrazol-5-yl)phenyl]pyrrole-2,5-dione 6-[[1-methyl-5-(trifluoromethoxy)indol-3-yl]methyl]pyridine-2-carboxylic acid 3-(2,5-difluoroanilino)benzoic acid N-[3-(4,5-dichloroimidazol-1-yl)propyl]aniline 2-[1-(1H-indole-3-carbonyl)piperidin-4-yl]acetonitrile 4-[[4-(4-azidophenoxy)thieno[3,2-d]pyrimidin-6-yl]methyl]morpholine N-[4-(2,6-dimethylphenoxy)phenyl]acetamide 2-[4-(1,4,5,6-tetrahydropyrimidin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-3-one 4-[1-(5-methylpyridine-3-carbonyl)piperidin-4-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one N-[(2S,3R)-1-ethyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]-2,6-dimethoxybenzamide 6,7-bis(4-methoxyphenyl)-9H-fluoren-2-ol 3-methoxy-2,4-dioxo-5-propanoyl-1H-pyrimidine-6-carboxylic acid 3,5-diamino-N'-[amino(methyl)amino]-6-chloropyrazine-2-carboximidamide 3-bromobenzenesulfonate;1,2-dihydrocyclopenta[b]indol-3-ylmethanone [2-(3-fluorophenyl)-1,3-thiazol-5-yl]-[4-[(5-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl]methanone;2,2,2-trifluoroacetic acid 4-(6-azidohexoxy)benzonitrile 5-[2-[(4S)-4,8-dimethylnonanoyl]oxypropoxycarbonyl]pyridine-3-carboxylic acid 1,2-dihydroquinoline;2-[[5-(4-ethoxyphenyl)-4-methyl-6-oxo-1H-pyrimidin-2-yl]sulfanyl]acetic acid 2-(3,5-dichlorophenyl)-5,8-dimethoxynaphthalene-1,4-dione 2-(4,5-dimethyl-1,3-thiazol-2-yl)-6-[[2-hydroxyethoxy(phenyl)phosphoryl]amino]phenol (1S)-N,2,3-trimethyl-1-phenylcyclohexa-2,4-dien-1-amine 2-amino-4-[3-methoxy-4-(trifluoromethyl)phenyl]-6-methylbenzene-1,3-dicarbonitrile 4-[2-(1,3-dioxobenzo[de]isoquinolin-2-yl)ethyl]benzoic acid 1-[4-[2-[4,5-bis(ethenyl)thiophen-3-yl]ethynyl]phenyl]ethanone 4-(4-aminophenyl)sulfanyl-2,3-dimethoxyphenol N-[2-hydroxy-1-(3-methoxyphenyl)ethyl]-5-oxohexanamide 4-methyl-2-(3-pyrimidin-5-ylpropanoylamino)-1,3-thiazole-5-carboxylic acid N-[2-(1H-benzimidazol-5-yl)ethyl]-4,4a,5,6,7,8,8a-octahydro-3H-quinoline-2-carboxamide 4-methyl-N-[5-[3-(1H-pyrrolo[2,3-c]pyridine-2-carbonyl)phenyl]imidazo[1,2-a]pyridin-8-yl]benzenesulfonamide N-[2-methyl-4-(2,2,3,3,3-pentafluoropropoxy)phenyl]furan-2-carboxamide 4-[4-(cyclobutylmethoxy)-2,5-dimethylphenyl]-7-[(1S)-3-oxocyclohexyl]pyrrolo[2,3-d]pyrimidine-6-carbonitrile [4-(2,3,4a,5,6,7,8,9,10,11,11a-decahydrobenzo[b]quinolizin-4-yloxy)piperidin-1-yl]methanol 2-hydroxy-5-phenyldiazenylnaphthalene-1,7-disulfonic acid [2-(1-benzofuran-2-yl)phenyl]boronic acid N-[4-chlorobutyl-(8-hydroxy-6-sulfonaphthalen-2-yl)amino]sulfonylbenzamide 2-N,4-N-bis(2-methoxyphenyl)-1,3,5-triazine-2,4,6-triamine 2-(1,3-benzodioxol-5-ylmethylideneamino)-4,6-bis(3,5-difluorophenyl)pyridine-3-carbonitrile [4-(aminomethyl)-4-fluoropiperidin-1-yl]-[5-[3-chloro-7-(2,6-difluorophenyl)-2,8b-dihydropyrazolo[3,4-d]pyrimidin-4-yl]pyridin-2-yl]methanone 3-cyclobutyl-N-[5-(2,4-dioxoimidazolidin-1-yl)pentyl]-1H-pyrazole-5-carboxamide 2-[(2R,6S)-2,6-dimethylmorpholine;ethane;N-[5-formamido-4-[4-(1H-indol-3-yl)piperidin-1-yl]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]formamide 2-cyclohexyloxy-N'-hydroxypyrimidine-4-carboximidamide 7-cyclohexyl-N-[(2S,3R)-1-oxo-2-phenylazetidin-3-yl]-5,6-dihydropyrrolo[2,3-d]pyrimidine-4-carboxamide 4-(2,3-difluorophenoxy)-6,7-dimethoxyquinoline 6-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]pyrazolo[1,5-a]pyridine-3-carboxylic acid 5-amino-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 3-[[2,5-dimethyl-4-(1-phenylethylidene)cyclohexa-1,5-dien-1-yl]amino]benzamide 2-[2-[4-(2,3-dichlorophenoxy)piperidin-1-yl]ethylsulfanyl]-N-(pyridin-4-ylmethoxy)acetamide;ethane 2-(2-butan-2-ylphenyl)quinoline N-[(2S)-1-[3-[5-[amino(hydroxy)methyl]thiophen-2-yl]phenyl]-5-oxopyrrolidin-2-yl]prop-2-enamide 3-benzyl-2H-azirine 2-[(3R,4S)-1-benzyl-4-ethoxypyrrolidin-3-yl]-N-methyl-N-(3-morpholin-4-ylpropyl)acetamide N-[2-(7,8-dihydronaphthalen-1-yl)ethyl]-1H-imidazole-5-carboxamide (4S)-1-cyclohexyl-3-methoxy-4-(3-nitrophenyl)azetidin-2-one 2-[1-(3,5-dimethoxyphenyl)cyclopropyl]acetonitrile 2-[3-(1,2-oxazol-3-yl)propanoyl]-6H-[1,2,4]triazolo[1,5-c]quinazolin-5-one N-[1-(benzenesulfinyl)piperidin-4-yl]-3,5-dimethoxy-2-methylbenzamide;ethane 1-azido-4-fluoro-2,3-diphenoxybenzene 1,2-diamino-6-oxo-4-(5-piperidin-1-ylpyridin-3-yl)pyridine-3,5-dicarbonitrile 6-methyl-N'-(2-oxo-1H-pyridin-4-yl)pyrimidine-4-carbohydrazide N-[3,5-difluoro-4-(1-methylbenzimidazol-2-yl)phenyl]-2,6-dimethoxypyridine-3-carboxamide 7-chloro-2,3,9-trimethylphenazine 6-(2,3-dihydroindole-1-carbonyl)-3H-thieno[3,2-d]pyrimidin-4-one 3-[4-(bromomethyl)-1,2-dihydroindol-3-ylidene]-7H-indol-6-ol 5-(3-azidophenyl)-2,4-dimethoxypyrimidine 3-(4-azidobutoxy)aniline 3-[1-(5-tert-butyl-2-ethoxyphenyl)propan-2-yl]-N,N-dimethylaniline 6-[(2,5-dimethoxyphenyl)methyl]-2-pyridin-3-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3,4-dibromo-7-oxo-4H-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid 1-[(4S)-5-(3-chlorophenyl)-2,5-dihydrofuran-4-yl]ethenol 1-[2,6-di(propan-2-yl)phenyl]-3-(5-ethylpyridin-2-yl)sulfonylurea 4-[2,3-dihydroxypropyl(ethyl)amino]-N-pyrimidin-2-ylbenzenesulfonamide 2-methyl-4-[1-(2,3,5,6-tetrafluorophenyl)imidazol-4-yl]pyridine 7-(2,4-dimethoxyphenyl)-6-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indole;ethane N-[(3S)-1-[3-(5,7-dimethylquinolin-8-yl)phenyl]pyrrolidin-3-yl]carbamate 3-[4,7-dihydroxy-2-(4-methoxyphenyl)-1,3-benzothiazol-6-yl]propanoic acid 6-chloro-4,5-dihydrothieno[3,2-b]pyrrole 2-[5-(2,3,4a,5,7,8,8a-octahydropyrano[3,2-b]pyridin-4-yl)-4,6-dimethoxypyrimidin-2-yl]phenol 1-methyl-3,5-diphenyl-4H-indeno[1,2-c]pyrazole [(3S,4R)-3-hydroxy-4-phenoxypyrrolidin-1-yl]-[4-methyl-3-(2H-tetrazol-5-yl)phenyl]methanone 3-(1H-indol-2-ylmethylidene)azepane 2-(3,4-dimethoxyphenyl)-1,5-dioxo-6H-thiopyrano[2,3-d]pyrimidine-2,4-diamine 3-(2,4-dichlorophenyl)-6-[2-[4-[4-(2-methylpropyl)piperazin-1-yl]anilino]pyrimidin-5-yl]quinazolin-4-one 2-[(5,6-dichloropyrazin-2-yl)amino]-2,3,4,7,8,9,10-octahydropyrimido[4,5-b]quinoline-1,6-dione [2-[(Z)-but-1-enyl]phenyl]-phenylmethanimine 3-[[[1-(2,6-difluorophenyl)piperidin-4-yl]amino]methoxy]-N'-hydroxypyridine-2-carboximidamide 2-[(Z)-1-chloroethenyl]-1,3,4,9-tetrahydropyrido[3,4-b]indole 4-[2,5-difluoro-4-(3-fluoropropyl)phenyl]-N,N-bis[(E)-1H-indol-6-ylmethylideneamino]aniline 7-[(4-chlorophenyl)methyl]-8-hydroxy-5,6,8,11-tetrahydrobenzo[b][1,4]benzodiazepine-3-carboxylic acid 3-(3,4-dihydroxyphenyl)-7-[(4-methoxyphenyl)sulfonylamino]chromene-2-thione (2S)-N-(4-bromophenyl)-3,3-dimethyl-2-[(6-phenylpyrimidine-4-carbonyl)amino]butanamide 2-(4-aminocyclohexyl)oxycarbonylbenzoate 4-[(6,8-dimethoxyquinazolin-2-yl)amino]-N,3-bis(ethylaminomethyl)benzamide (5-fluoropyrimidin-2-yl)carbamoylcarbamic acid 4-[2-(aminomethyl)phenyl]-3-[3-(trifluoromethoxy)anilino]piperidine-1-carboxylic acid 2-amino-1,3-benzoxazole-4-carboxylic acid;N'-[4-(4-chlorophenyl)butanoyl]-N,N,4-trimethylpiperazine-1-carboximidamide N-[3-[2-(4-chlorophenyl)ethyl]oxetan-3-yl]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide 3-[3-(benzenesulfonamidomethyl)phenyl]benzenecarboximidamide 2-(6-methoxy-1H-indol-3-yl)ethanimine 1-(3,4-dimethylphenyl)sulfonyl-N'-[5-(trifluoromethyl)pyridin-2-yl]piperidine-3-carboximidamide 2-[[4,5-dimethyl-6-(methylamino)pyrimidine-2-carbonyl]amino]-3-thiophen-2-ylpropanoic acid;ethane 6-chloro-4H-imidazo[1,2-a]1,4]benzodiazepine;(Z)-2-(dimethylamino)-3-fluorobut-2-enenitrile 4-amino-2-[(1E,3Z)-1-aminopenta-1,3-dienyl]phenol;but-1-yne 4-[3-(3,5-dimethylphenyl)propoxy]aniline 1-(2,4-dimethoxyphenyl)-N-[3-(5,6-dihydro-[1,3]oxazolo[4,5-b]pyridin-2-ylamino)phenyl]cyclopropane-1-carboxamide 6-[(5R)-2,4-dimethyl-5-morpholin-4-ylsulfonylfuran-3-carbonyl]-1-[(E)-2-phenylethenyl]pyrrolidin-2-one 4-[3-(2,6-dimethylphenyl)propanoyl]-1-ethylpiperazine-2-carbonitrile 3-[7-[4-(1,5-dimethylpyrazol-4-yl)-2,6-dimethoxyanilino]-3-methylimidazo[4,5-b]pyridin-5-yl]cyclobutane-1-carboxylic acid 3,4-dihydroxy-N'-(4-methyl-1H-indol-5-yl)benzenecarboximidamide 4-ethenyl-2-phenyl-1H-indole N-[4-fluoro-3-(trifluoromethyl)phenyl]cyclopropanesulfonamide (4R)-1,3-dimethyl-4-[(E)-2-(4-methylphenyl)ethenyl]-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 2-[6-(1,4-dioxan-2-ylmethoxy)pyridin-3-yl]-5-phenylcyclohexan-1-one 1-azidooxy-5-ethenylnaphthalene 1-[6-(3,5-dichloropyridin-4-yl)pyridin-2-yl]-N-(1-hydroxyethyl)piperidine-4-carboxamide 3-[[2-hydroxy-5-methyl-4-(trifluoromethoxy)phenyl]diazenyl]-5,7-dihydropyrrolo[3,2-c]pyridazine-6-thione N-[2,3-dihydro-1H-inden-5-yl(pyridin-3-yl)methoxy]pyrimidin-4-amine 4-[(2,3-difluorophenyl)methyl-methylideneamino]piperidine (3-chloropyridine-4-carboximidoyl)carbamic acid N-[2-chloro-3-(3,6-dihydro-2H-pyran-5-yl)phenyl]-4-methoxypyrimidine-5-carboxamide [(5-methylpyridine-2-carbonyl)amino]carbamodithioic acid 6-bromo-2-chloro-3,4-difluoroaniline 2-[[3-(1,2-oxazol-3-yl)-1H-1,2,4-triazol-5-yl]methoxy]ethanamine 2-[(3,4-dichlorophenyl)methylsulfanyl]-6-[5-(4-fluorophenyl)furan-2-yl]-7H-purine N-[4-chloro-3-[2-(cyclopropylamino)ethyl]phenyl]-5,6-difluoro-1H-indole-2-carboxamide 2-[(3S,6R)-5-(4-chlorophenyl)-1,1-dioxothiolan-3-yl]-N-[[2,5-bis(trifluoromethyl)phenyl]methyl]-N-cyclohexylacetamide [(2S)-4-tert-butylmorpholin-2-yl]-[7-chloro-6-fluoro-5-hydroxy-1,3-dihydroisoindol-2-yl]methanone 2-chloro-6-(3,5-difluorophenyl)-8H-pteridine 2-amino-5-(2-bromophenyl)-6H-[1,3]thiazolo[4,5-d]pyrimidin-7-one 1,2-diamino-4-[3-(methylamino)phenyl]-6-oxopyridine-3,5-dicarbonitrile 2-(3,4-dimethoxyphenyl)-5-hydroxy-2,7-diazaspiro[3.4]octane-6,8-dione N-[2-(4-methoxyphenyl)ethyl]-1H-pyrazolo[3,4-b]pyridine-5-carboxamide (2R)-N,3-dihydroxy-1,4-bis[(4-methylphenyl)sulfonyl]-5-oxopiperazine-2-carboxamide 2-(5,7-dimethoxyquinolin-3-yl)-8-ethyl-6H-cyclohepta[d]pyrimidine N-[3-(1H-benzimidazol-2-ylmethoxy)-5-(1H-pyrazol-4-yl)phenyl]cyclopropanecarboxamide [(3R,4S)-1-benzoyl-4-methoxypiperidin-3-yl]-[(3S)-3-fluoropyrrolidin-1-yl]methanone (2S)-3-[4,5-bis(ethenyl)triazol-1-yl]-N-(furan-3-ylmethyl)-2-hydroxypropanamide 3-chloro-4-[(4-cyanophenyl)methoxy]benzaldehyde 5-amino-4-(3-bromo-2,6-dichlorophenyl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 2-(1,3-benzodioxol-5-ylmethoxy)-6-N-phenylpyridine-4,6-diamine;ethane 5-chloro-2,3-dimethylthieno[3,4-b]pyridine;methanol 4-[(3,5-difluorophenyl)methyl]-2-(6-methoxypyridin-3-yl)-1H-pyrimidin-6-one N-[(1R,2R)-2-hydroxycyclohexyl]-4-methoxybenzenesulfonamide 7-methyl-6,11-dihydrobenzo[c][1]benzoxepine 4-[1-(2-chlorophenyl)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-2-yl]-3-methoxyphenol N-[3-chloro-4-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]phenyl]-5-[2-fluoro-6-(trifluoromethoxy)phenyl]furan-2-sulfonamide;hydrochloride 4-N,5-bis(3-cyclopropylphenyl)-2-hydroxybenzene-1,4-dicarboxamide 3,6-dichloro-2-methylpyridine;ethane;8-[(1S)-1-hydroxypropan-2-yl]-N-piperidin-4-yloxyquinoline-3-carboxamide 2-[3,4-dichloro-5-methylsulfonyl-6-(pyridine-4-carbonyl)pyridin-2-yl]benzonitrile N-[2-(5,6-dimethylpyrimidin-4-yl)oxyethyl]thiophene-3-carboxamide N-[1-(2,4-dihydroxyphenyl)ethylideneamino]-3-hydroxybenzamide N-[(2S,3R)-6-chloro-1-methyl-5-oxo-2-phenylpiperidin-3-yl]-4-cyclopropyloxybenzamide 2-[3-(4,4-difluoropiperidine-1-carbonyl)phenyl]-1H-indole-6-carboxamide 2-(7,8-difluoro-3,4-dihydroquinolin-6-yl)acetic acid 1-[(4,5-dimethylfuran-2-carbonyl)amino]-3-sulfamoylurea 4-[2,2-bis(methylamino)ethylimino]-1-(3,5-difluorophenyl)-6-(pyridin-4-ylamino)hexan-3-ol;propane [(3R)-5,8-difluoro-2,3-dihydro-1H-inden-4-yl]carbamic acid 1-[[4-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylcarbamoylsulfamoyl)cyclohexyl]methylideneamino]propan-2-one ethane;(3S,4R)-1-[1-methyl-5-(trifluoromethyl)pyrazole-3-carbonyl]-4-phenylpyrrolidine-3-carboxylic acid 2-(4-aminophenyl)sulfanyl-6,7-dihydro-5H-pyrrolo[1,2-c]imidazole-7a-carboxylic acid 3-[2-(5,8-dimethyl-1,7a-dihydroquinoxalin-6-yl)ethynyl]-N-(pyridin-4-ylmethyl)benzamide 5-[(Z)-2-hydroxy-4-phenylpent-1-enyl]benzene-1,3-diol 3-[2-[(Z)-3-aminoprop-1-enyl]pyridin-4-yl]-N,N-dimethylaniline N-(1,2,3,5,6,7-hexahydropyrrolizin-8-yl)pyridine-3-sulfonamide 2-[6-(1,3-dioxol-4-yl)-7-methoxyquinazolin-4-yl]cyclopropan-1-one 7-chloro-4-ethyl-2,3-dimethylidene-1,4-benzoxazine N-(1,3-benzothiazol-5-yl)-2-methoxyacetamide 6-bromo-2,3-dimethylimidazo[1,2-a]pyridine 3-[3-[(6R)-6-[2-(4-ethylphenyl)ethenyl]piperidin-1-yl]propoxymethyl]pyridine 3-methyl-2-oxo-5-[(2,4,6-trichlorophenyl)methoxy]-1H-indole-3,7-dicarboxamide 1-butan-2-yl-3,5-bis(2-methylbutan-2-yl)pyrazole;platinum(2+) 2-(1,3-benzothiazol-2-ylamino)-4-(pyridine-3-carbonyl)benzenesulfonic acid 3-[4-(2,3-dihydro-1H-inden-5-yl)phenyl]-N,N-dimethylpropan-1-amine 5-[(1S,2R)-2-aminocyclohexyl]pyridine-3-carboxylic acid 2-[(2Z)-4,5-dimethylhepta-2,6-dien-3-yl]sulfanyl-N'-hydroxypyridine-4-carboximidamide 4-[(2Z)-2-ethenyl-5,6-dimethoxyhepta-2,5-dienoyl]benzaldehyde 2-[(3Z)-6-fluoro-2-methyl-3-[(4-phenylphenyl)methylidene]inden-1-yl]acetic acid 4-amino-2-(3,5-difluoropyridin-2-yl)-N'-hydroxybenzenecarboximidamide N-[2,3-dihydroxypropyl(pyridin-4-yl)amino]benzenesulfonamide N-[5-(2-aminoquinazolin-6-yl)-3H-1,2-oxazol-2-yl]-2-bromobenzenesulfonamide 2,4-dimethyl-5-[(3R)-1-propanoylpyrrolidin-3-yl]pyridine-3-carbonitrile 2-[1-[(3,4-dichlorophenyl)methyl]-5-hydroxy-6-oxopyrimidin-2-yl]sulfanylpropanoic acid 2,5-dihydroxybenzoate;manganese(2+) [4-(3,5-dipyridin-2-ylphenyl)cyclohexa-1,3-dien-1-yl]oxymethanol ethane;(3-fluoropyridin-4-yl)oxyboronic acid 5-fluoro-4-phenyl-2H-1,3-thiazin-6-amine 2-(3,4-dimethylphenoxy)-N-[(Z)-1-(4-hydroxyphenyl)ethylideneamino]acetamide 2-azido-5,7-difluoroquinoline 3-[(1R)-1-(4-fluorophenyl)ethyl]-7,7-dimethylbenzo[e]indole 5-[4-(diethylamino)-2-methylphenyl]imidazolidine-2,4-dione N-(2,6-dioxopiperidin-3-yl)-4-methoxybenzamide 1-[3,5-bis(trifluoromethyl)phenyl]-N',2-dihydroxypropanediamide N-[2-amino-1-(cyclohexylmethylamino)propan-2-yl]-5-chloropyridine-3-carboxamide;dihydrochloride 2-[4-(6,7-difluoronaphthalen-1-yl)phenyl]-5-ethoxypyridine N-[5-[7-fluoro-3-(1H-imidazo[4,5-b]pyridin-2-yl)-2H-indazol-5-yl]pyridin-3-yl]pentanamide 5-(difluoromethyl)-N-[2-methyl-4-(1H-pyrazole-5-carbonylamino)phenyl]-1,2-oxazole-3-carboxamide 2-[4-[[2,6-dichloro-5-(pyridine-3-carbonyl)pyrimidin-4-yl]amino]piperidin-1-yl]acetamide 3-[(4-cyclopentylphenyl)methoxy]-2,6-difluorobenzamide 1-(3-azidophenyl)-N-propan-2-ylmethanesulfonamide 1-[3,5-bis(4-chlorophenyl)-2H-pyrrol-4-yl]-N,2,2-trimethylpropan-1-amine N-[(Z)-2,4-difluoropent-1-enyl]-5-(trifluoromethoxy)pyridine-3-carboxamide N-[2-(4,7-difluoro-1H-indole-3-carbonyl)-5-ethoxyphenyl]-2-(trifluoromethyl)benzenesulfonamide 1-[2,6-di(propan-2-yl)phenyl]pyrrolidine-2,5-dione 2-[4-chloro-5-methyl-3-(trifluoromethoxy)pyrazol-1-yl]acetic acid 1-[3,5-dimethyl-4-(oxolane-2-carbonyl)piperazin-1-yl]-3-(5-ethylsulfonylthiophen-3-yl)propan-1-one 3-ethyl-1-(4-methoxyphenyl)sulfonyl-4-methylindole 5-bromo-3,4-dimethoxybenzoate (3S,4R)-3-azido-4-phenylpiperidine 7-cyclopentyl-2-[(2R)-1-[4-(diethylaminomethyl)benzoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 5-(6,7-dihydro-4H-triazolo[1,5-a]pyrazine-3-carbonylamino)-2,4-dihydroxybenzoic acid 3-[4-amino-5-(methoxymethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N-cyclobutyl-4-methylbenzenesulfinamide 3-[(E)-2-nitroethenyl]-2H-1,4-benzodioxine N-[(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]furan-2-carboxamide 4-(1,2-benzoxazol-3-yl)benzoic acid;ethane 4-(2,5-dimethylanilino)-3,7-dihydropyrimido[4,5-b]quinoline-8-thione 4-(3,5-difluorophenyl)-N-[2-(hydroxymethyl)cyclobutyl]piperidine-1-carboxamide 1-[2-amino-3-methyl-4-(methylamino)-5,6-dihydrocyclopenta[b]pyrrol-7-yl]ethanone 1-[2-[3-(1,2-dihydrotriazin-5-yl)-4-methoxyphenyl]-6-(3-morpholin-4-ylquinoxalin-6-yl)sulfanylpyrimidin-4-yl]pyrrolidine-2,5-dione N'-hydroxy-4-[2-(methylsulfonylmethyl)pyrrolidine-1-carbonyl]pyridine-2-carboximidamide 4-ethyl-2-[(3-hydroxypiperidin-1-yl)methyl]-5-iodo-1H-pyrimidin-6-one 6-[4-(dimethylamino)cyclohexyl]oxynaphthalene-2-carbonitrile 4-(6,7-dimethoxyquinazolin-2-yl)morpholine;ethane 2-[3-[(4S)-4,5-diamino-4-hydroxypentoxy]propyl]isoindole-1,3-dione N-[(Z)-1H-indol-3-ylmethylideneamino]pyridine-2-carboxamide 5-[3,5-bis(trifluoromethyl)phenyl]hexanenitrile 2-[(3S)-1-(cyclobutanecarbonyl)piperidin-3-yl]-6-(thiophen-2-ylmethyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-hydroxysulfanyl-5,6,7,8-tetrahydronaphthalene-1-sulfinic acid 5-[3-(1,4-dioxin-2-yl)phenyl]-2,4-bis(phenylmethoxy)pentanamide 1-[3-(dimethylamino)phenyl]-3-naphthalen-2-ylsulfinylurea 6-[1-methyl-5-(2-phenylethyl)pyrazole-4-carbonyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-[2-(cyclopentylamino)ethyl]-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxamide 4-[(E)-3-azidoprop-1-enyl]-2,6-dichlorophenol 5-[1-(4-cyclopropylimidazol-1-yl)-3,3,3-trifluoropropyl]-2-pyrimidin-2-ylpyridine 4-[(Z)-3-amino-2-methanimidoylbut-2-enimidoyl]-5-chloro-N'-propan-2-ylpyridine-2-carboximidamide 2-benzylsulfanyl-8-(4,6-dimethoxypyrimidin-5-yl)-1,7-dihydropurin-6-one 3-(2,4-dichlorophenyl)-1H-indol-5-amine 5-methoxycarbonylimino-2,8-dimethylbenzo[g]chromene-6-carboxylic acid 7-fluoro-N'-(pyridine-3-carbonyl)-1H-indole-2-carbohydrazide 7-amino-2,4-dioxo-5-[2,3,4,5-tetrafluoro-6-(trifluoromethyl)phenyl]-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile (Z)-1,4-diphenylbut-3-en-2-one ethane;(2E)-2-[(2E,5Z)-octa-2,4-dienylidene]-1H-quinoline (E)-2-cyano-3-[1,3-dimethyl-4-oxo-2-sulfanylidene-6-[3-(trifluoromethoxy)phenyl]pyrimidin-5-yl]prop-2-enoic acid 3-(2,4-dimethoxyphenyl)-5-ethyl-N,N-dimethyl-1H-pyrazole-4-carboxamide 2-[1'-(cyclopropylmethyl)spiro[4,5-dihydrothieno[2,3-c]pyran-7,4'-piperidine]-6-carbonyl]pyrazole-3-carboxylic acid [6-[(dimethylamino)methyl]pyridin-3-yl]-[3-[[5-fluoro-4-hydroxy-2-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]phenyl]iminomethyl]-2-hydroxyphenyl]azanium N-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxamide 1-(5,6-dimethylpyridin-3-yl)oxyazetidin-2-one 2,4-dimethoxy-N-[6-(3-phenoxypropanoylamino)hexyl]benzamide 5-[2-(2-propylbutanoylamino)ethyl]-1H-indole-2,3-dicarboxylic acid N-[4-(4-chlorophenoxy)phenyl]-2-methyl-6,7-dihydropyrimido[5,4-d]pyrimidin-4-amine N-methyl-4,5-dinitropyrazole-1-carboxamide 4-[2,6-dichloro-N-(methoxyiminomethyl)anilino]phenol 6-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-2H-phthalazin-1-one (4S)-1-azido-4-butoxy-3,6-dihydro-2H-pyridine 1-[2,3-dichloro-4-[(E)-4,4,4-trifluoro-3-methylbut-1-enoxy]phenyl]-N-[(Z)-ethylideneamino]sulfanylmethanamine N-(3,4-dihydro-2H-chromen-7-yl)-1-methylsulfonyl-4-(trifluoromethoxy)pyrrole-2-carboxamide 3-[3-[4-(4-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-1H-indazol-5-yl]-N-methyl-4-propan-2-ylidenecyclohexa-1,5-diene-1-carboxamide (E)-4-[[1-[(2,6-dichlorophenyl)methyl]triazol-4-yl]methoxy]-4-oxobut-2-enoic acid 3-(5,7-dichloro-2,3-dihydro-1H-inden-4-yl)-4,6-dimethoxypyridazine 7-(difluoromethyl)-2-ethoxyimidazo[1,2-a]pyridine 1-(3,4-dimethoxyphenyl)-2H-quinoline 3-[4-(1,3-dioxolan-2-yl)phenyl]propan-1-ol;ethane 4-[[2,6-difluoro-4-(trifluoromethyl)phenyl]methylamino]piperidine-1-carboxylate 4-(4-propanoylphenyl)sulfonylpiperidine-1-carboxylate 3-[(4-chlorophenyl)methyl]-5,6-dihydro-4H-1,2]oxazine 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]-6-ethoxy-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 2,6-dibutyl-4-(3-chloropropyl)phenol (3S,4R)-3-methyl-1-[[2-methyl-6-(trifluoromethoxy)pyridin-3-yl]methyl]piperidin-4-ol 2-[3-(4,5-dihydropyrimidin-2-yl)phenyl]sulfanylphenol 7-[[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridine (5S)-1-[2-(3,4-dimethoxyphenyl)ethyl]-5-(3-hydroxyprop-1-enyl)pyrrolidin-2-one 1-(2,5-dichlorophenyl)-N-[2-methylsulfanyl-4-(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)phenyl]-5-piperidin-1-ylpyrazole-4-carboxamide ethane;4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxybenzonitrile 2-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[3H-indene-2,3'-azetidine]-1'-ylidene]propanenitrile 4-[(3R,5S)-1-(8-fluoroquinolin-5-yl)-5-methylpyrrolidin-3-yl]oxy-2,6-dimethylpyridine-3-carboxamide 2-[2-(1-aminoethyl)phenyl]benzaldehyde [4-chloro-3-(trifluoromethyl)phenyl]-[1-methyl-7-(pyridin-2-ylamino)pyrazolo[3,4-c]pyridin-5-yl]methanone 2-(7H-pyrrolo[3,2-d]pyrimidin-4-yl)phenol N-(4-chlorophenyl)-3-[6,7-dimethoxy-2-(trifluoromethyl)quinolin-4-yl]propanamide 2-(6-methoxypyridin-3-yl)-5,10,17,19-tetrazahexacyclo[12.11.0.03,12.04,9.016,24.018,23]pentacosa-1,3(12),4(9),5,7,10,13,15,18,20,22,24-dodecaene 2-ethoxy-N-[5-methyl-2-(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)pyrazol-3-yl]acetamide 6-chloro-4-(5-nitrofuran-2-yl)-2,3,5,7,8,9-hexahydrocyclohepta[b]thiophen-1-ol 2-hydroxyethyl(phenyl)sulfanium 2-[3,4-bis(phenylmethoxy)-5-propylphenyl]acetic acid;ethane [6-(2-aminoethyl)-4-chloro-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-yl]methanesulfonamide N-[(3S,4R)-1-azido-2-oxopiperidin-3-yl]-5-chloroquinoline-8-sulfonamide [4-[2-(3,5-dichloropyridin-4-yl)cyclohexen-1-yl]piperazin-1-yl]-naphthalen-1-ylmethanone (E)-N,N-diethyl-3-(2-fluorophenyl)prop-1-en-1-amine (2S,4R)-1-[4-cyano-3-(trifluoromethyl)phenyl]-N-cyclopropyl-N-ethyl-4-methoxypyrrolidine-2-carboxamide N-[1-methyl-5-(6-pyridin-2-ylpyridin-3-yl)imidazol-4-yl]pyrimidin-2-amine 2-[(3R,5S)-4-acetyl-1-benzyl-3,6-dimethoxy-3H-indol-2-ylidene]propanedioic acid 1-azidooxy-4-[3,5-bis(trifluoromethyl)phenyl]benzene N-benzyl-4,6-dimethoxypyrimidine-2-carboxamide;hydrochloride 4-N,6-dibenzyl-3-methanimidoylpyridine-2,4-diamine (2-cyclopropylpyrimidin-4-yl)-[2,8-diaza-7-azoniaspiro[3.5]nonan-7-yl]methanone 2-(1H-indol-3-ylmethylideneamino)-4-methylsulfanylphenol 5-[(2-diazohydrazinyl)methylidene]-4-ethoxycyclohexa-1,3-dien-1-ol 3-[2-(4-methoxyphenyl)cyclopentyl]-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepine;dihydrochloride 3-amino-5-[(3,4-dimethoxyphenyl)sulfonylamino]benzoic acid 1-[(2,4-difluorophenyl)methylamino]-3-hexan-3-ylurea (2R,3S)-N-[(4-methoxyphenyl)methyl]-2-thiophen-2-yloxolane-3-carboxamide N-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-3-fluorophenyl]-1-methylcyclopropane-1-carboxamide (2-methoxyphenyl)phosphanyl-oxophosphanium 1-[2-(1,1,3,3-tetramethylisoindol-2-yl)propanoylamino]pyrrole-2-carboxylic acid N-[[(5S)-3-(6-fluoroquinolin-4-yl)oxycyclohexyl]methylidene]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide 3-[2-amino-6-methyl-5-(3-morpholin-4-ylpropoxy)pyrimidin-1-ium-4-yl]-4-chloro-N-cyclohexylbenzamide 5-amino-N-ethyl-6,8-dihydroxynaphthalene-2-sulfonamide (E)-3-[2,6-dimethoxy-4-(3-pyrrolidin-1-ylquinoxalin-5-yl)phenyl]prop-2-enal 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(5-hydroxycyclopenta-1,3-dien-1-yl)piperidin-4-ol 5-chloro-6,7-dihydroxynaphthalene-2-carboxylic acid 2-[N-(3-hydroxypropyl)-4-sulfoanilino]acetamide (2S)-3-naphthalen-1-yloxy-2-(phenylmethoxycarbonylamino)propanoic acid 3-[(4E,5Z)-4-ethylideneocta-1,5,7-trien-2-yl]-2H-indazole 4-[2-[(4,5-dichlorocyclohexa-1,3-dien-1-yl)amino]quinazolin-6-yl]oxybutanoic acid 4-(4-tert-butylphenyl)-3,6-dimethyl-N-[(Z)-prop-1-enyl]pyridin-2-amine 1-[(4,5-dichloropyridin-3-yl)methoxy]cyclopentane-1-carboxylic acid 2-[3-(cyclopropylmethoxy)-4-methoxyphenyl]butanoic acid 2-[(4R,5S)-1-ethyl-3-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]benzoic acid 1,2-difluoro-6-[2-(4-propylphenyl)ethynyl]naphthalene 3-(4,5-dimethylthiophen-2-yl)oxy-N-[4-(3-phenylpropanoylamino)-1H-indazol-6-yl]benzamide 5-[[2-(4-bromophenyl)-2-ethoxyacetyl]amino]pyridine-3-carboxylic acid 2-[4-methyl-3,5-di(propan-2-yl)phenoxy]-6-propyl-1,2,3,4-tetrahydronaphthalene [(E)-4-aminobut-2-enyl]-triphenylphosphanium 3-bromo-4-(1H-indole-2-carbonyl)pentanoic acid (4R)-1-[[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-N'-hydroxy-2-oxoimidazolidine-4-carboximidamide 2-[6-(4-bromo-3,5-dimethylpyrazol-1-yl)pyrimidin-4-yl]oxyethanol 4-methylsulfonyloxy-2,6-dinitrobenzoic acid N-butanoyl-2,4,6-trimethyl-N-(3-morpholin-4-ylpropyl)benzenesulfonamide 7-(4-fluorophenyl)-9,10-dihydrophenanthrene 1-[4-(1,3-benzothiazol-2-yloxy)phenyl]sulfonyl-5-hydroxyindole-2,3-dione 6-azidooxy-2,3-difluoro-1H-benzimidazole N-[5-[3-(4,6-dimethylpyridin-2-yl)oxetan-3-yl]-1-methylpyrazol-3-yl]propanamide N-[(E)-3,7-dimethyloct-5-enyl]aniline;formaldehyde 2-[(Z)-1-phenylpropylideneamino]oxyacetic acid 4-[1-(3,4-dichlorophenyl)ethylamino]-2-methyl-6-(pyridin-4-ylsulfanylamino)pyridazin-3-one 1-(4-cyclohexylpiperazin-1-yl)-2,3,5,6-tetrahydroazepino[4,3-b]indole;dihydrochloride 1-(3,4-dihydro-2H-quinoline-1-carbonyl)-N-[(5-methylfuran-2-yl)methyl]cyclopropane-1-carboxamide 1-[(3,5-dichloropyridin-4-yl)methyl]pyrrole-2,5-dione 6-methoxy-N-[4-[2-(trifluoromethyl)cyclohexa-1,5-dien-3-yn-1-yl]cyclohepta-2,4,6-trien-1-ylidene]pyridine-2-carboxamide 1,4-dibenzyl-2H-pyridine 2-[N-(4-bromobutan-2-yl)-3-hydroxyanilino]octanoic acid 5-ethyl-2-[(3S)-pyrrolidin-3-yl]oxypyridine 5-[(3,4-dimethoxyphenyl)methyl]-6-hydroxynaphthalene-2-carboxylic acid N-[(3S,4S)-1-benzyl-4-methoxypyrrolidin-3-yl]-N'-[2-(2-methoxyphenyl)ethyl]oxamide 2-(cyclopropylmethylamino)-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one 1-[3-(2-ethoxypyridine-4-carbonyl)phenyl]-N,N',N'-trimethylethane-1,2-diamine 5-(3,4-difluorophenyl)sulfonyl-N-[2-methoxy-6-(trifluoromethyl)pyridin-3-yl]furan-2-carboxamide 2-[1-[(3R)-4,6-dimethyl-3-propan-2-yl-9H-pyrido[3,4-b]indol-3-yl]ethylideneamino]guanidine;hydrochloride 4-methyl-2-(1H-pyrrolo[2,3-b]pyridin-6-yloxy)phenol 2-[1-(1,4-dimethylpiperidine-4-carbonyl)piperidin-3-yl]-6-propanoyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-(2,3-dihydropyrrolo[2,3-c]pyridine-1-carbonyl)-6,7,8,9,10,11-hexahydro-5H-pyrido[3,4-b]azonine-10a-carboxylic acid [1-(cyclopropylmethyl)pyrrolidin-3-yl]-[4-(pyridine-2-carbonyl)piperazin-1-yl]methanone (2S)-1-[3,5-difluoro-4-[7-methyl-6-(1-methylpyrazol-4-yl)-2-oxo-3H-imidazo[4,5-c]pyridin-1-yl]phenoxy]-N,N',N',N',N'-tetramethyloxamide 1-[(3S,4R)-6-fluoro-4-hydroxy-3-[(5-methyl-2H-tetrazol-1-ium-1-yl)methyl]-3,4-dihydro-2H-chromen-7-yl]piperidine-2,6-dione 2-[[4-amino-5-(3,5-dichlorophenyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]methoxy]acetic acid (3S)-3-[4-(4-chlorophenyl)butyl]-1-ethylpyrrolidine 4-[8,14-difluoro-3-methyl-5-(4-pyridin-4-ylphenyl)-6,11,13,15-tetrazatetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),2,4,10(15),12-pentaen-14-yl]morpholine 2-(6-aminopurin-9-yl)ethanesulfonate 1-methyl-4-[3-methylidene-5-oxo-7,8-dihydro-6H-cinnolin-2-yl]pyrrole-2-carboxylic acid (5Z)-2-imino-5-[(4-nitrophenyl)methylidene]-1,3-thiazolidin-4-one 5-(2,3-dichlorophenyl)-N-[4-(difluoromethoxy)phenyl]pentanamide 4-[2,6-difluoro-3-(trifluoromethyl)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one (5R)-N-cyclopentyl-2-(methylaminosulfanylamino)-7,8-dihydro-6H-quinoline-3-carboxamide 2,3-bis(hydroxymethyl)-4-naphthalen-1-yloxyanthracene-9,10-dione 1-[4-amino-5-(azidomethyl)-2-(trifluoromethoxy)phenyl]pyrrolidine-3,4-diol N-methyl-3-methylidene-2H-1,4-benzothiazine-6-carboxamide N-methyl-2-[3-(2,4,6-trimethylphenyl)-1H-pyrazol-5-yl]pyridine-4-carboxamide 1-(3,4,5-trimethoxyphenyl)piperidine-2,6-dione N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2,2-diethylcyclopropane-1-carboxamide [(1E,4Z,7Z)-6-amino-8-[5-chloro-2-(oxan-4-ylmethoxy)phenyl]octa-1,4,7-trienyl]phosphonic acid 1-[(4-azidooxyphenyl)methyl]-2,3,5,6,7,8-hexahydro-1H-pyrrolizine 2-[3-amino-6-methyl-1-(4-prop-1-en-2-ylphenyl)sulfonylindol-5-yl]acetic acid 1-N',3-N'-diphenyl-3-N'-(pyridine-2-carbonyl)butanedihydrazide 7-azido-2,5-dimethyl-3H-imidazo[4,5-c]pyridine 4-ethyl-3-[(2S)-1-phenylpropan-2-yl]benzenesulfonic acid 7-fluoro-6-methoxy-3-[1-[4-(trifluoromethyl)phenyl]propan-2-yl]quinazolin-4-one N-[[(2S)-oxolan-2-yl]methyl]spiro[1,4-dihydroquinoxaline-3,4'-piperidine]-2-imine 7-(4-fluoro-2,6-dimethylphenyl)-2-[3-[(1-iodophosphanylazetidin-3-yl)amino]pyridin-4-yl]thieno[3,2-b]pyridine-5-carbonitrile 4-[4-(2,3-dihydro-1H-tetrazol-5-ylmethoxy)phenyl]-N-[(1S)-1-(4-propan-2-ylpyridin-3-yl)ethyl]benzamide 2-[(6,7-dimethoxy-4H-indeno[1,2-d][1,3]thiazol-2-yl)sulfanyl]ethyloxidanium N-(2,5-dihydroxypentyl)-4-[(Z)-1,3-diphenylprop-1-enoxy]benzamide 2-[2-chloro-N-(1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carbonyl)anilino]propanoic acid (2R)-3-[4,5-bis(ethenyl)furan-2-yl]-2-methyl-N-[[4-(methylaminosulfanyl)phenyl]methoxy]propanamide 6-[2-(4-tert-butylphenyl)quinolin-6-yl]oxyhexanamide 1-azido-2,3-di(propan-2-yl)naphthalene 5-(8,9,10,11-tetrahydrophenanthro[9,10-f]indolizine-11-carbonyl)furan-3-carboxamide 6-[(2R,5S)-2-ethyl-1,3,4,5-tetrahydroazepino[4,5-b]indol-5-yl]-N-(oxetan-3-ylmethyl)pyridine-3-sulfonamide 4-[[(3R)-1,2,3,4-tetrahydroisoquinolin-3-yl]methoxy]pyridine-2-carboxamide 3-[5-bromo-2-ethoxy-4-(methylamino)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 4-amino-N,N-dimethyl-3-[6-(trifluoromethyl)pyridine-2-carboximidoyl]benzenecarboximidamide [6-chloro-1,5-bis(4-methoxyphenyl)hexyl]azanide N-[(2S)-4-methoxyimino-1-phenyl-3,6-dihydro-2H-pyridin-5-yl]quinoline-7-carboxamide 3-(4-chlorophenyl)-N-[2,5-difluoro-4-[5-methylsulfonyl-6-(4,4,4-trifluorobutoxy)pyridine-3-carbonyl]phenyl]propanehydrazide N-cyclopropyl-2,4-dihydroxy-3-(1H-indol-3-yl)-5-propanoylbenzamide (4S)-4,5,6,7-tetrachloro-3-methyl-1-propan-2-ylsulfonyl-2H-benzimidazole 5-(2-nitrophenyl)sulfanylcyclohepta-1,4,6-trien-1-ol 2-[4-bromo-3-(trifluoromethyl)phenyl]acetate 2-[(1R,3S)-3-azidocyclopentyl]sulfanylbenzenesulfonamide 4-(2,6-difluorophenyl)-3-methyl-1H-pyridin-2-one 2-[3-aminopropyl(methyl)carbamoyl]-N,N',2,6-tetramethylcyclohexane-1-carboximidamide;ethanol 3-chloro-N',4-dimethylbenzohydrazide;hydrochloride 6-(2,6-difluorophenyl)-N-[5-[1-[ethyl-[1-(methanesulfonamidomethyl)piperidin-4-yl]amino]ethenyl]pyridin-3-yl]imidazo[1,2-a]pyrazine-8-carboxamide 5-(4-tert-butylphenyl)sulfonyloxy-2,3-dihydroxybenzoic acid 5-[2-(4,6-dimethylpyridin-3-yl)-1H-indol-3-yl]pentan-1-amine 4-azido-1,2,3-trimethoxy-9H-fluorene 5-bromo-N-[(3Z)-7-methyl-4-[3-(trifluoromethoxy)phenyl]hepta-1,3,5-trien-2-yl]-N-propan-2-ylidenepyridine-2-carboximidamide 4-[(Z)-2-chloroethenyl]-5-methoxytriazole-1-carboxamide 2-[(Z)-1,3-diaminoprop-1-enyl]-4-(2-hydroxyethoxy)benzonitrile 7,8-dimethoxychromene-2,4-dione 3-(3,5-dimethylphenyl)-1H-indole 4-chloro-6,7-difluoro-2H-chromene;ethane 4-amino-N-(3,6-dimethylimidazo[1,2-a]pyridin-7-ylidene)benzenesulfonamide 2-[4-methyl-3-(trifluoromethyl)phenyl]sulfanylbenzonitrile N-azido-2,3-dibromoaniline 1-[(4aR,6R)-2-hydroxy-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-6-yl]-3-ethoxy-1-phenylpropan-2-one 2-aminoacetaldehyde;1,4-difluorobenzenethiol;N-[(E)-3-(5-ethylpyridin-2-yl)-5,6-dimethylhex-4-en-2-ylidene]-N'-[2-[1-(3-methoxy-1-methylazetidin-3-yl)pyrazol-3-yl]prop-2-enimidoyl]methanimidamide N-[6-(hydroxymethyl)-1,3,4-thiadiazol-2-yl]-2-methoxybenzamide [(2R,5S)-4-azido-5-methoxycarbonyloxolan-2-yl]-triphenylphosphanium 2-chloro-3-methoxy-6-(1,3-oxazol-5-yl)benzenesulfonic acid N-(2,6-dichlorophenyl)-2-[[5-isocyano-4-(methoxyiminomethyl)-1H-pyrimidin-6-ylidene]amino]acetamide 5-chloro-6-[[2,3-dimethyl-4-[3-(1,4,5-oxathiazepan-4-ium-4-yl)propoxy]phenyl]methylsulfanyl]pyridine-2,3-diamine N-[2-[(3R,4S)-3-methyl-5-oxooxan-4-yl]pyridin-4-yl]acetamide 5-(4-fluorophenyl)sulfinylpentanamide 1-[1-(azidomethyl)cyclopropyl]-4-phenylbenzene N-[(2S)-3-[4-[5-(aminomethyl)pyridin-3-yl]phenyl]-1,1,1-trifluoropropan-2-yl]azetidine-3-carboxamide;dihydrochloride ethane;1-[3-(4-methylphenyl)pyrrolidine-1-carbonyl]pyrazole-3-carbonitrile N'-(6-chloropyridin-3-yl)propane-1,3-diamine;ethane 4-benzyl-2-[(1S)-1-[7-bromo-8-fluoro-1-[(4-methoxyphenyl)methyl]-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]ethyl]-5-hydroxy-1H-pyrimidin-6-one 4-[3-(1-azidopyrrolidin-2-yl)-1H-indol-5-yl]-6,8-dimethoxyquinoline 3-(2,4-dihydroxyphenyl)-N-[(1S)-4-methoxycyclohepta-2,4-dien-1-yl]benzamide 3-hydroxy-1,3-bis(2-hydroxyphenyl)propan-1-one 2-(4-acetamidocyclohexyl)-N-[1-(3,5-difluorophenyl)-2-pyrrolidin-1-ylethyl]-6-oxo-1H-pyrimidine-4-carboxamide (1Z,3E)-N'-(pyridine-4-carbonyl)hexa-1,3-diene-1,5-dicarboximidamide 1-azido-3-(3,5-dichlorophenyl)sulfonylbenzene 2-(3,4-dihydroxyphenyl)-6-methoxychromen-4-one 4-[(2,6-dimethylbenzoyl)amino]-1H-pyrazole-5-carboxylic acid 5-amino-3-[2,4-bis(prop-1-en-2-yl)phenyl]pyrazine-2-carbonitrile 4-(2,3-dihydro-1H-pyrazol-5-yl)-N-[2-methoxy-4-nitro-6-(trifluoromethyl)phenyl]-2-methylaniline 2-[2-amino-5-(4,4-difluorocyclohexen-1-yl)pyrimidin-4-yl]phenol 1-[2-(methoxymethyl)phenyl]-3,6-bis(1-phenylpropan-2-yl)piperidine 2-chloro-N-methylsulfonyl-N-propanoylbenzamide 6-chloro-N-[5-(3-methoxypropanoyl)pyridin-2-yl]-1H-indole-2-carboxamide N-[4,5-difluoro-6-(2H-tetrazol-5-yl)pyridin-3-yl]imidazo[1,5-a]quinoline-8-sulfonamide 1-methyl-4-propan-2-ylsulfinylbenzene;1-[[4-(trifluoromethoxy)phenyl]carbamoylamino]cyclohexane-1-carboxylic acid 2-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-6-oxa-2,9-diazaspiro[4.5]decan-8-one 4-[N-(2,2-dimethoxyethyl)-4-hydroxyanilino]benzenesulfonamide 1-[(3R)-4-[2,5-dimethyl-7-[1-(6-propanoylpyridin-2-yl)piperidin-4-yl]pyrrolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]ethanone 3-(2,4-dihydroxyphenyl)-N'-ethenyl-1H-pyrazole-5-carboximidamide 4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carbonylamino)oxane-4-carboxylic acid;hydrochloride N-(2,4-dichloropyrimidin-5-yl)-4H-1,3-benzoxazin-6-amine 1-[(3aR,7aS)-5-benzyl-2,3,3a,4,6,7-hexahydropyrrolo[3,2-c]pyridin-1-yl]-3,3-dimethylbutan-1-one;formic acid 5-[[(2S)-1-[(2R)-6-cyano-2,3-dimethyl-4-oxohexanoyl]piperidin-2-yl]amino]-N,4-dimethylpyridine-2-carboxamide 2-[4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]-N-[(3-fluorophenyl)methyl]anilino]propanoic acid 4-[4-[2-(dimethylamino)ethylcarbamoyl]-1,3-thiazol-2-yl]benzoic acid 4-chloro-7-hydroxy-6-phenyldiazenylnaphthalene-2,3-disulfonic acid 2-[(3R,5S)-1,7-dioxo-6H-2,6-naphthyridin-3-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide 4-N-[1-(3,5-dimethoxyphenyl)ethyl]-6-methylquinazoline-2,4-diamine (NE)-N-[3-(2,5-difluorophenyl)-1-piperidin-4-yl-3H-imidazo[1,2-a]pyridin-2-ylidene]hydroxylamine 5-[2-(cyclopentylmethylamino)pyridine-3-carboximidoyl]-4-N,4-N-dimethylpyrimidine-4,6-diamine 2-(N-pyridin-3-yl-4-sulfamoylanilino)acetic acid 3-(2,6-diethylanilino)-4H-1,2,4-triazin-5-one 2-methylimino-5-phenyl-1H-pyrimidine-4,6-diamine 2-[1-(4-fluorophenyl)pyrrolidin-3-yl]oxypyridine 2-[4-(3-chloro-2-fluorophenyl)-1,3-thiazol-2-yl]-N'-hydroxypropanediamide 2-azido-5,6-dibutoxypyrimidin-4-amine 1-[4-(5-chloro-2,3-dihydroindole-1-carbonyl)piperidin-1-yl]ethanone [(3R,4S)-3-hydroxy-4-methoxypyrrolidin-1-yl]-[4-(1,2,4-triazol-1-yl)phenyl]methanone 2-[6-methoxy-3,5-di(propanoyl)naphthalen-1-yl]acetic acid 5-chloro-N,3-dimethyl-4-[4-(1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)piperidine-1-carbonyl]pyridine-2-carboxamide N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]isoquinoline-5-carboxamide 1-[6-(4-azidophenyl)pyridin-3-yl]-2,3,3a,4,5,9b-hexahydrofuro[3,2-c]quinoline 2-amino-4-[3-(trifluoromethyl)phenyl]pyridine-3-carbonitrile N-cyclobutylsulfanyl-2,6-difluoro-3-phenylaniline;N-[4-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]sulfanylpyridin-2-amine 3-methyl-N-(1H-pyrazolo[4,3-b]pyridin-6-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine-2-carboxamide 1-[2-methyl-4-[[(E)-1H-pyrazol-5-yldiazenyl]methoxy]phenyl]ethanone 3-[(1S)-2,2,3-trimethylcyclopropyl]benzoic acid 6-butylsulfonyl-4-propanoyl-2,3-dihydrochromene-2-carboxamide N-[(2,3-difluorophenyl)methyl]-7H-purine-6-carboxamide 4-[4-amino-5,7-dichloro-2-(trifluoromethyl)benzimidazol-1-ium-1-ylidene]butanoate 2-[[3-(benzylcarbamoyl)phenyl]methylideneamino]benzoic acid 2-chloro-5-fluoro-4-[3-(thiophene-3-carbonylamino)pyrazol-1-yl]benzoic acid N-[(1R,3S)-3-[[[2-(4-chlorophenoxy)acetyl]amino]methylideneamino]cyclohexyl]-3-ethynylbenzamide 2-[4,5-dimethyl-N-(3-morpholin-4-ylpropyl)-2-phenyldiazenylanilino]octanoic acid N-(2,4,6-trichlorophenyl)pyridine-3-carboxamide 2-methyl-N'-propanoylfuro[3,2-b]pyridine-3-carbohydrazide (E)-3-[2-chloro-5-[1-(4-chlorophenyl)ethylamino]sulfanylphenyl]-N-hydroxyprop-2-enamide;ethane 2-[(5S,10bS)-5-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]-4-chlorophenol 1-[(3S,4S)-4-[(4-fluorophenyl)methyl]oxolan-3-yl]piperidine;2,2,2-trifluoroacetic acid N-methyl-3-(3,4,5-trifluorophenyl)prop-2-enamide 6-methoxy-3H-quinazoline-4,7-dione 2-[1,3-benzodioxol-5-yl-[[2-hydroxyethyl(methyl)carbamoyl]amino]methylidene]propanedioic acid 6-amino-2-[(4,5-dimethyl-1H-pyrazol-3-yl)methylsulfanyl]-3H-quinazolin-4-one 3-(5-propanoyloxypentyl)benzoic acid 3-[(2R)-3,3-dimethylbutan-2-yl]benzaldehyde 4-chloro-2-[3-[(2-fluorobenzoyl)amino]pyrazol-1-yl]benzenesulfonamide 1-[4-methyl-6-(trifluoromethoxy)-2H-chromen-2-yl]ethanone 2-[5-[(3,4-dichlorophenyl)methoxy]pyrazin-2-yl]acetamide 4-[3-(methylamino)anilino]-N-propylpyrimidine-5-carboxamide 6-(1,3-benzodioxol-5-yl)-4-chloro-2-methoxy-7H-purine 2-bromo-1H-pyrazolo[1,5-a]pyrimidin-7-one 5-chloro-N-[(2S)-4,4-difluoro-1-[5-[5-isocyano-3-methyl-6-(1-methylpyrazol-4-yl)pyrazolo[1,5-a]pyridin-7-yl]pyridin-2-yl]butan-2-yl]thiophene-2-sulfonamide 1-[1,3-bis(4-chlorophenyl)-3-hydroxypropyl]pyrrolidine-2,5-dione 3,6-dichloro-1-methylindole 3-[4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]phenol ethane;1-[3-[(E)-3,4,4-trifluorobut-2-enoxy]phenyl]ethanone (2S)-1-[3-(4-methoxyphenyl)cyclohexa-2,4-dien-1-yl]sulfonylpyrrolidine-2-carboxylic acid 2-[3-(aminomethyl)phenyl]-3-phenyl-6,7-dihydrobenzimidazole-5-carboxamide 2-(4-chloro-3-fluorophenoxy)-N-[4-[(7R)-13-ethyl-5,7-dimethyl-6,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-3-yl]but-1-en-2-yl]acetamide 1-(5-azido-2-methoxyphenyl)sulfonyl-4-methylpiperazine 3-[4-(4-aminopiperidine-1-carbonyl)-2-fluorophenyl]-1,5,7-trimethylpyrrolo[3,2-c]pyridin-4-one 1-(3,5-dimethylphenoxy)-4-methoxy-2H-naphthalene 2-methylsulfanyl-7,8-dihydro-6H-quinazoline-5-carboxylate 1-[3-hydroxy-4-methyl-5-(trifluoromethoxy)phenyl]butan-1-one 1-N',2-N'-bis(4,6-difluoro-2H-pyrazolo[3,4-c]pyrazol-3-yl)-1-(6-methylpyridin-2-yl)ethene-1,1-diamine 4-(7-azido-2,3-dihydropyrido[3,2-b][1,4]oxazin-4-yl)pyridin-2-amine N-[(Z)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-2-methylquinoline-4-carboxamide (E)-N'-[3-bromo-4-(trifluoromethylsulfanylamino)phenyl]-1-N,2-N-diethylprop-1-ene-1,2-diamine 5-[2-(4-aminocyclohexyl)-1,3-thiazol-5-yl]-3H-1,3,4-oxadiazol-2-one;hydrochloride N-(2,6-diethylphenyl)-5-fluoro-3-[4-[6-methoxy-7-(morpholine-4-carbonyl)quinazolin-4-yl]piperazin-1-yl]-2-methylbenzamide 3,5-dimethoxy-6-(2-naphthalen-2-ylethynyl)acridine 3-(6-methoxynaphthalen-2-yl)-4,5-dimethylidene-1H-pyrazole 1-(3,4-difluorophenyl)-N-[(2-methoxyphenyl)methyl]-5-oxopyrrolidine-3-carboxamide 2-[2,3-dihydroxypropyl(ethenylsulfonyl)amino]benzenesulfonic acid 1-[4-(aminomethyl)phenyl]-3-ethenoxypropan-2-one 4-(4-chlorophenyl)sulfanyl-2,3-dihydroxy-5-[2-[4-(hydroxymethyl)piperidin-1-ium-1-ylidene]ethylsulfamoylamino]-N-methylbenzamide;formate 1-(5-chloroquinolin-8-yl)oxybutan-2-one 2-[6,7-dihydro-4H-pyrano[4,3-c]pyrazol-1-ylmethyl(2-fluoroethyl)amino]-N,N-dimethylacetamide N-[(3R,4S)-1-butanoyl-4-(2,5-difluorophenyl)pyrrolidin-3-yl]-5-cyclopentyl-1,2-oxazole-3-carboxamide (1S,3R)-2,2-difluoro-N-[(6-pyridin-4-ylimidazo[1,2-a]pyrimidin-2-yl)methyl]-3-[5-(trifluoromethoxy)pyridin-2-yl]cyclopropane-1-carboxamide N-(4-methoxyphenyl)-N'-[6-[5-methyl-2-(methylideneamino)phenyl]pyridin-3-yl]ethane-1,2-diamine 4-[2,4,6-trimethyl-N-[(3-nitrophenyl)methyl]anilino]benzoic acid N-[4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]cyclopropanecarboxamide;ethane 4-[3-(4,5-dihydrobenzo[g][1]benzoxepin-10-yl)propoxy]aniline (2R,4S)-1-[3-chloro-5-fluoro-2-[[2-methyl-6-(tetrazol-1-yl)quinoline-4-carbonyl]amino]benzoyl]oxy-2,4-dimethylpyrrolidine-2-carboxylic acid 1-[2-(6-benzylpyridine-3-carbonyl)pyrrolidin-1-yl]-3,3-dimethylbutan-1-one 3-[(4-chlorophenyl)methyl]-7-ethenoxy-6-(difluoromethoxy)-2-oxo-N-piperidin-4-yl-1H-quinoline-4-carboxamide 2-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(Z)-[(Z)-3-phenylprop-1-enyl]iminomethyl]ethanimine 4-(2,6-diethylphenyl)sulfinyl-7,7-dimethylfuro[3,4-c]pyridine 6-(3,5-difluorophenyl)-2-sulfanylidene-1H-pyrimidin-4-one (7-methylspiro[chromene-2,4'-piperidine]-1'-yl)-(oxan-3-yl)methanone N-[2-(4-fluorophenyl)-5-methylpyrazol-3-yl]-6-(6-methoxypyridin-3-yl)quinoline-7-carboxamide N-[(Z)-1-cyanoethylideneamino]-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide [2,3-difluoro-4-(trifluoromethyl)phenyl]methanamine 2-azido-4-benzyliminohexanamide N-[2-(2,6-diethylphenyl)ethylideneamino]aniline 1-[2,4-bis(methoxymethoxy)phenyl]propan-2-one 4-chloro-N'-(7H-purin-2-yl)benzenecarboximidamide;ethane 4-(4-fluorophenyl)butanamide;2,3,5,6,7,8-hexahydronaphthalene-1,5-dicarboxamide 2-azidooxy-6-(1-methylpiperidin-4-yl)pyridine 2-[azido(phenyl)methoxy]pyrimidine 3-(cyclopentanecarboximidoyl)-2-N,2-N-dimethylbenzene-1,2-diamine 1-cyclohexyl-2,4-diphenylbenzene;iridium(3+);4-methylbenzenethiolate 1-[2,4-dichloro-3-(1H-imidazole-5-carbonyl)phenyl]ethanone 3-chloro-4-[[6-(dimethylamino)pyridin-2-yl]amino]sulfanylbenzenethiol 4-[3-cyclohexylpropyl(2-hydroxyethyl)amino]-1H-pyrimidin-6-one N-(cyclohexylmethyl)-1'-[(2,4-difluorophenyl)methyl]spiro[7,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyridine-6,4'-piperidine]-3-carboxamide;2,2,2-trifluoroacetic acid 3-(4,5-diphenyl-1H-imidazol-2-yl)-N-[(Z)-(4-hydroxyphenyl)methylideneamino]benzamide 4-[[2-(8-bromonaphthalen-1-yl)cyclopropen-1-yl]amino]-3,5-difluoro-N'-hydroxybenzenecarboximidamide 6-methylsulfanyl-3,4-dihydro-2H-chromene;[4-(trifluoromethoxy)phenyl]methanamine 1-(3-chlorophenyl)butan-2-one;[4-(1,1-difluoroethyl)phenyl]methanol 2-[4,5-bis(4-methylphenyl)-1H-imidazol-3-ium-2-yl]phenol 1-amino-N-[(2S)-2-[6-(5,7-difluoroquinolin-4-yl)-3,3a,4,5,7,8,8a-octahydro-2H-pyrrolo[2,3-c]azepine-1-carbonyl]cyclohexyl]piperidine-4-carboxamide 5-amino-3-(2-ethylpyridin-4-yl)-2,3-dihydro-1,2-oxazole-4-carbonitrile (4Z)-4-[amino(1,2-benzothiazol-3-yl)methylidene]-5,5-dimethylpyrazolidin-3-one 2-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)oxyacetonitrile N'-[(Z)-2-aminoethenyl]-4-phenylbenzenecarboximidamide 2-[(3S,7R)-5-methyl-8-[[2-methyl-4-[(4-sulfamoylphenyl)methoxy]phenyl]methylcarbamoyl]nonan-3-yl]oxyacetic acid 2-[(4S)-1-methyl-6-oxo-4-(thiophen-3-yloxymethyl)-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-3-yl]thiophene-3-carbonitrile 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]-N-[3-(4-pyridin-4-ylpiperidin-1-yl)propyl]acetamide 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;N-cyclohexyl-7-fluoro-3-methyl-2,3-dihydroinden-1-imine 2,3-dimethyl-1H-pyrrolo[3,4-c]pyridine-6,7-bis(prop-1-ynyl)-5,6,8,9-tetrahydropyrazolo[4,3-h]quinazoline 3,5-dimethylbenzenethiol;formaldehyde;N-[2-oxo-1-phenyl-3-(propan-2-ylamino)propyl]benzamide 2-[(3R)-1-azidopyrrolidin-3-yl]oxy-N,5-dimethylpyrimidin-4-amine 2-ethyl-3,6-difluoro-N'-hydroxyimidazo[1,2-a]pyridine-7-carboximidamide 1-N,2-N-dibenzylhexane-1,2-diamine 4-N-[(1E,3Z)-2,4-dimethylhexa-1,3-dienyl]-6-methylpyrimidine-4,5-diamine 6-(4-fluorophenyl)pyridine-2,4-diamine;3,4,5-trifluorobenzamide N-[1-(2-hydroxyacetyl)piperidin-4-yl]-6-pyrazol-1-ylpyridine-3-carboxamide [2-(4,5-dihydrobenzotriazol-1-yl)phenyl]boronic acid 1-(5-chlorothiophen-2-yl)sulfonylpiperidin-4-one (2S)-6-amino-2-[4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxyphenyl]-9-methanimidoyl-7H-purin-8-one 6-[[4-(2,2-dimethylpropoxy)-3-methoxyphenyl]methyl]-2-thiophen-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-bromospiro[cyclohexane-1,2'-dioxirane];1-(3-ethylphenoxy)-3,5-dimethylbenzene;N-methylhexanamide (2S,4S)-5-[3-[(4-cyclopropylphenyl)methoxy]pyridin-2-yl]pyrrolidine-1,2,4-tricarboxylic acid (Z,3E)-1-amino-2-[(2R)-4-chloro-7-fluoro-5-propan-2-yl-2H-1,3-benzothiazol-2-id-3-yl]but-2-en-1-one;rubidium(1+) 6-(cyclopropanecarbonylamino)-4-[4-(3,5-dimethyl-1H-pyrazol-4-yl)piperidin-1-yl]pyridine-3-carboxamide 1-(2,4-dinitrophenoxy)-N-hydroxymethanesulfonamide N'-[(3-methoxyphenyl)methyl]-4,6-dimethylpyrimidine-2-carboximidamide 4-chloro-3-nitrobenzenesulfonate 3,5-dichloro-6-(2,4,5-trifluorophenyl)pyridine-2-carboxylic acid 1-[(4R)-2,6-dimethylheptan-4-yl]-3-phenyl-5H-pyrazolo[4,3-c]pyridin-4-one 4-[(2,5-dimethylcyclohexa-1,3-dien-1-yl)methyl]-1-[2-(4-methoxyphenyl)ethynyl]-N-propan-2-ylpiperidine-4-carboxamide;N-methylbutan-2-amine 4-[(2S)-8,8a-dimethyl-1-oxo-8H-2,3-benzoxazin-6-yl]-N-(trifluoromethoxy)aniline N-[3,5-difluoro-4-(1H-pyrrolo[2,3-b]pyridine-2-carbonyl)phenyl]propanesulfonamide N-azido-6,11-dihydro-5H-benzo[b][1]benzazepin-3-amine 7-chloro-N-methylnaphthalene-2-sulfinamide 2-(7-methyl-1H-indazol-5-ylamino)phenol N-[4-(5-phenylfuran-2-yl)cyclohexyl]carbamate 2-[2-amino-6-(cyclopropylmethoxy)pyridin-4-yl]-1,3-thiazole-5-carboxamide N-[4-(7-fluoro-2-methylquinolin-6-yl)oxyphenyl]piperidine-1-carboxamide 2-[4-(2-fluoropropanoyl)phenoxy]-1,3,6-trimethylpyridin-4-one (4R)-5',6'-dihydroxy-3,7'-bis[(4-methylphenyl)sulfanyl]spiro[isoindole-1,2'-indene]-1',3'-dione 3-[3-(furan-2-yl)propanoylamino]butanoic acid N-butyl-N-(4,5-dimethyl-2-phenyldiazenylphenyl)nonanamide 1-(5,7-dihydropyrrolo[3,4-b]pyridin-6-ylmethyl)cyclohexane-1,2-diol 5-(1,3-benzothiazol-2-yl)-N-[[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]methyl]pyrimidin-2-amine 1-[2,6-bis(trifluoromethyl)phenyl]-5-hydroxy-4-nitrosopyrazole 5-[2,6-dichloro-4-(trifluoromethyl)phenyl]imidazolidine-2,4-dione 1-[2-[5-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-[(1R,6R)-3-sulfanyl-3,9-diazabicyclo[4.2.0]octan-9-yl]pyrimidin-2-yl]oxyethyl]imidazolidine-2,4-dione 1-[6-(2,3-dihydro-1H-indene-5-carbonylamino)hexyl]-N-methyl-4-phenylpiperidine-4-carboxamide N-ethyl-3,5-dimethoxy-4-methylbenzamide 2-[(1-methyltetrazol-5-yl)methoxy]-N-phenylethanimidate 1-[(3R,5S)-5-[4-[2-methyl-6-(3,3,3-trifluoropropoxy)pyridin-4-yl]phenyl]sulfonyloxolan-3-yl]ethanol 2-[3-(4,5-dichloro-1H-indole-2-carbonyl)phenyl]acetic acid 5-ethylsulfonylthiophene-3-carboximidamide 1-[4-(1-iodocyclopropyl)phenyl]piperazine 4-[2-(4-methylanilino)ethyl]cyclohexan-1-one N-[6-(2,4-dichlorophenyl)pyrimidin-4-yl]carbamate [2-hydroxy-1-(3,4,5-trimethoxyphenyl)cyclohexyl]-(4-methylpiperazin-1-yl)methanone (E)-2,6-dimethyl-N-[4-methyl-3-[6-oxo-1-[2-oxo-2-[5-(trifluoromethyl)pyridin-3-yl]ethyl]pyridazin-3-yl]phenyl]hept-2-enamide 6-[7-(1,2,4,5-tetrazin-3-yl)heptanoyloxy]hexoxymethylphosphinous acid 2-(2,3-dichlorophenyl)-4H-pyridine 2,4-bis[(E)-2-(3-nitrophenyl)ethenyl]-1,3,5-triazine N-[5-[3-[4-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]cyclopentanecarboxamide 3-[3-aminopropyl(ethylamino)amino]-N-hydroxybenzamide [3-(4,5,6,7-tetrahydro-1H-benzimidazol-2-ylmethoxy)phenyl]methanimine 1-[(2R)-3,7-dibromo-1,2,3,4-tetrahydronaphthalen-2-yl]ethanone [5-(2,3-dimethylimidazol-4-yl)sulfonylthiophen-2-yl]methanol 2-bromo-N,N'-diphenyl-5H-thieno[3,4-b]pyridine-6-carboximidamide N-(3-acetylphenyl)-4-cyclopropyl-2,6-difluorobenzamide 2-[3,4-bis(difluoromethyl)phenyl]sulfanyl-1H-pyridine-2,5-diamine N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methoxy-2-(4-pyrrolidin-3-ylbutoxy)-5-[5-(trifluoromethyl)pyridin-2-yl]benzamide 3-amino-4-[2,6-difluoro-3-(phenylsulfanylmethyl)phenyl]benzoic acid (4E)-4-[[3,5-dibromo-4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-5,5-dimethylpyrazolidin-3-one 3-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethoxy)propane-1-sulfonate 2-[6,7-bis(3-methylbutoxy)dibenzothiophen-1-yl]acetic acid 7-(3-bromophenyl)-2,3-dimethyl-1H-benzimidazol-3-ium 5-amino-3-(2,6-difluorophenyl)-1-methylpyrazole-4-carbonitrile 3-methyl-2,6-bis(methylamino)phenol;5-naphthalen-1-ylhexanal 4-bromo-2-[(2-hydroxynaphthalen-1-yl)methylideneamino]benzenesulfonamide 2,4-dibromo-6-fluoro-5-methylpyrimidine 3-[(E)-2,4-dimethylhex-1-enoxy]cyclobutan-1-amine;ethane 5-[[4-(2-phenylethyl)piperazin-1-yl]methyl]-3H-1,3,4-oxadiazol-2-one;dihydrochloride (1R,2S)-N'-(4-chlorophenyl)sulfanyl-3-[4-[4-ethyl-5-methoxy-6-oxo-7-(trifluoromethyl)cyclopenta[c]pyridin-1-yl]-2-hydroxyphenoxy]cyclopentane-1-carbohydrazide 4-(3-fluoro-5-methoxypyridin-2-yl)-1,3,6-trimethylpiperazine 2-[4-(6-fluoroindol-1-yl)piperidin-1-yl]acetic acid 4-[4-(3,5-difluoropyridin-2-yl)piperazin-1-yl]-6-(oxan-4-yl)-1H-pyrazolo[3,4-d]pyrimidine 4-chloro-1,2,3,6-tetramethylbenzo[h]quinolin-10-ol 5-[2,4-dihydroxy-6-(hydroxymethyl)phenyl]-N-[2-methoxy-3-(morpholine-4-carbonyl)propyl]-1H-pyrazole-3-carboxamide (2S,4R)-1-[1-benzyl-5-ethanimidoyl-3-[2-(methoxycarbonylamino)-2-oxoethyl]pyrrole-2-carbonyl]-N-cyclopentyl-4-hydroxypyrrolidine-2-carboxamide N-[2,3,6-trimethyl-4-(4-nitrophenyl)phenoxy]-1H-pyrazolo[3,4-b]pyridine-5-carboxamide 3-[7-(5-methylthiophen-2-yl)-3H-imidazo[4,5-c]pyridin-2-yl]-5-(1,2,3,6-tetrahydropyridin-4-yl)-1H-pyrazolo[3,4-c]pyridine 3-[(1S,3aS)-2-[(E)-2-(6-chloropyridin-2-yl)but-1-enyl]-5-oxo-1,2,3,3a,4,5,7,8,9,10,10a-dodecahydropyrrolo[3,2-b]azocin-1-yl]propanoic acid (Z)-2-(3,4-dimethylphenyl)-N-[(E)-(2,6-dinitrophenyl)methylideneamino]-3-hydroxybut-2-enamide 2-N,4-N,6-trimethyl-2-N-(1-pyridin-3-ylethylideneamino)pyrimidine-2,4-diamine 2-(ethylamino)-1'-[3-fluoro-4-(trifluoromethoxy)benzoyl]spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,3'-piperidine]-4-one 2-(N-ethylsulfonyl-2,6-difluoroanilino)decanoic acid (E)-N-methyl-3-[4-[2-methyl-3-[1-(5,6,7,8-tetrahydroquinolin-8-ylamino)ethenyl]phenyl]thiophen-2-yl]prop-2-enamide 4-cyclohexyl-7-methyl-2H-benzotriazol-5-amine (2S)-1-(benzylsulfonylcarbamoylamino)propane-2-sulfonic acid 1-[7-(2-chlorophenyl)-5-methyl-4,6,7,8-tetrahydropyrazolo[1,5-a]azepin-3-yl]ethenol 4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]-N-[2-(5-ethyl-1H-imidazol-3-ium-3-yl)ethyl]benzamide N-(1,3-benzodioxol-5-yl)-2-[4-(6-fluoroquinolin-4-yl)cyclohexyl]acetamide 5-[(3S)-7-(2,6-difluorophenyl)-4-oxo-3H-pyrrolo[1,2-a]pyrazin-2-yl]thiophene-2-carboxylate 2-[6-(3,4-dimethoxyphenyl)hexyl]-6-propanoyl-5,6,7,8-tetrahydro-3H-quinazolin-4-one (6R)-6-butoxycarbonyl-5,7-dihydroindolo[2,1-a][2]benzazepine-10-carboxylic acid 2-[1-(2,4-dichlorophenyl)ethoxy]-5-nitropyridine 5-(3,4-dimethoxy-1H-naphthalen-2-yl)-N-(4-methoxyphenyl)-6-oxocyclohexa-1,3-diene-1-sulfonamide 4-[1-(3,4-dichlorophenyl)ethenyl]aniline 4-(2,3-dihydroindole-1-carbonyl)-5-[2-[hydroxy(methyl)amino]ethoxy]-N-methoxy-2H-quinoline-1-carboxamide 2-(3-methylbutyl)-4-propan-2-ylpyrimidine (5Z)-2-(3,4-dimethylphenyl)imino-5-[(1-ethylindol-3-yl)methylidene]-1,3-thiazolidin-4-one 2-[(1S)-7,11-difluoro-6,8,9-triazatricyclo[4.3.0.02,4]nona-6,10-dien-6-yl]-N,N-bis[2-(dimethylamino)ethyl]acetamide 2-[2-(benzenesulfonamido)ethyl]benzenesulfonamide 2-[2-(5-aminopentyl)-4-fluorophenyl]acetic acid 5-(2-hydroxyphenyl)-4-[(E)-pyrrole-3-carbonyliminomethyl]-1,2-dihydropyrazol-3-one 4-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazole-2-carbonyl)-1'-methyl-2-phenylspiro[4H-isoquinoline-3,4'-piperidine]-1-one 1-(2,3-dihydropyrrolo[2,3-c]pyridin-1-yl)ethanone 1-azido-2,5-difluoro-4-(1H-indol-3-yl)acridine 1-[4-(2,6-diphenylpyrimidin-4-yl)phenyl]ethanol 4-chloro-6,7-dimethoxy-8-phenylchromene-2-thione 2-[(3-bromopyridin-4-yl)amino]-N-(3-fluorophenyl)acetamide N-[(3S)-7-amino-4-oxospiro[3H-chromene-2,1'-cyclopentane]-6-yl]-5-cyclobutylpyridine-2-carboxamide 1-(dimethylamino)naphthalene-2,3,4,7-tetracarbonitrile N-[(3R)-4-oxooxolan-3-yl]-2-[6-(trifluoromethyl)pyridin-3-yl]sulfanylacetamide 2-(2-methoxyphenyl)sulfanyl-1,3-benzoxazole 2-[3,5-difluoro-4-[2-(6-fluoronaphthalen-2-yl)ethynyl]phenyl]-5-methoxypyrimidine 1-[(3,5-dimethylpyridin-4-yl)methyl]-N-(2-phenylphenyl)sulfanylpyrrolidin-3-amine 4-[(5-bromopyridin-3-yl)methoxy]piperidine 2-(1H-benzimidazole-2-carboximidoyl)-6-(4-fluorophenyl)phenol N-[3,4-difluoro-2-(1H-pyrrolo[2,3-b]pyridine-6-carbonylamino)phenyl]-5-phenylmethoxy-1H-indole-2-carboxamide 5-amino-N-[2,2-dimethyl-3-(trifluoromethoxy)cyclobutyl]-1H-pyrrole-2-carboxamide 2-benzylsulfonylethanimidamide 2-[[3-(4,6-dimethyl-1,3,5-triazin-2-yl)phenyl]iminomethyl]phenol 4-(diethoxyphosphorylmethoxy)-N'-hydroxybenzenecarboximidamide 1,3-difluoro-7-methoxyanthracene 2-benzylsulfanyl-5-[(4,6-dichloro-1,3,5-triazin-2-yl)amino]phenol N-azido-6-[3-(2,4-difluorophenyl)propanoyl]pyridine-3-carboxamide 3-[1,1-bis(2,4,6-trimethylphenyl)ethyl]imidazole-2,4-dione 2-(4-chlorophenoxy)-N'-[3,5-dimethyl-1-[(4-oxo-3H-quinazolin-2-yl)methyl]pyrazol-4-yl]acetohydrazide 1-[[2-chloro-5-(tetrazol-1-yl)phenyl]methyl]pyrazole 2-(3,4,5-trimethoxyphenyl)acetaldehyde 1-[5-cyclopropyl-4-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylsulfonyl)-2-methoxyphenyl]-3-(oxolan-3-yl)urea [4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]-pyrrolidin-1-ylmethanone N-(3,4-dichlorophenyl)-N-methylpiperidine-4-carboxamide;hydrochloride 2,5-dibutylpyridine N-methyl-3,4-dihydro-1H-isoquinoline-2-carboxamide;3-(5-nitro-1H-indol-3-yl)propanoic acid N-(2,5-dimethylphenyl)-2-[(6S)-2-[(E)-2-[4-ethoxy-3-(1-hydroxyhexoxy)phenyl]ethenyl]spiro[2.5]octan-6-yl]acetamide (1S)-1-azido-5-benzyl-N-[2,4-bis(trifluoromethyl)phenyl]sulfonyl-3,6-dihydro-2H-pyridine-3-carboxamide 3-[6-(dimethylamino)-4-(2-fluoro-4-pyrrolidin-1-ylbutoxy)pyridin-2-yl]-1,5-dimethyl-1,6-naphthyridin-4-one 1-[6-(8,10-dioxo-11H-indolizino[2,3-f][1]benzofuran-9-yl)pyridin-2-yl]-1-phenylmethanol (4-benzylphenyl)-[4-(hydroxymethyl)piperidin-1-yl]methanone 4-[2,3-dimethylbutan-2-yl(methyl)amino]-5-iodo-1H-pyrimidin-6-one 3-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylamino)-N-[(E)-2-iodoethylideneamino]sulfanylpyrrolidine-1-carboxamide 1-[4-(3,5-dichlorophenyl)piperazin-1-yl]-2-(4-piperidin-1-yl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)ethanone;hydrochloride 2-[3,5-dichloro-N-(1,3-thiazol-5-yl)anilino]acetic acid 4-(3,5-difluoro-2-methylphenyl)cyclohexa-1,3-diene-1-carbonitrile 3-(3,5-difluorophenyl)-3-[6-(1H-pyrazol-4-yl)-1,2-benzothiazol-7-yl]propanoic acid 2-(ethylamino)-1,3-bis(4-propan-2-ylphenyl)guanidine 6-[(1S,2R)-2-methylcyclopentyl]oxypyridine-3-sulfonamide (5S)-3,8-dimethyl-2-oxo-N-[(1R)-1-phenylethyl]-6-propan-2-yl-7,9-dihydro-4H-pyrimido[6,1-c][1,4]oxazine-5-carboxamide 2-(1,3-thiazol-5-yl)-4H-pyrano[2,3-b]pyridine-3-carbonitrile 2-[(3S)-1-benzylpyrrolidin-3-yl]oxy-5-pyridin-2-ylsulfonylbenzonitrile 5-(2,3-dichlorophenyl)-7-N-[4-fluoro-3-(methylaminomethyl)cyclohexa-1,3-dien-1-yl]pyrazolo[1,5-a]pyrimidine-3,7-diamine 2-azido-1H-fluorene-4-carboxylic acid 2-[(3R,4S)-4-(1,5-dimethylpyrazole-4-carbonyl)pyrrolidin-3-yl]oxypyridine-4-carbonitrile 3-ethyl-1-methyl-5-[(E)-2-phenylethenyl]imidazolidine-2,4-dione 4-[azido(3,5-dimethylphenyl)methyl]-N,N-dibutylaniline (2S)-1,1,3-trimethylbenzo[e]indole 3-[(2E)-2-(1-benzylsulfanylethylidene)hydrazinyl]-6-methoxy-4H-1,2,4-triazin-5-one 2-(4-fluoro-3-methylphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole 3-amino-1-azido-2-propan-2-ylnaphthalene-2,5-dicarboxylic acid 3-(4,6-dimethylpyrimidin-2-yl)sulfanylbenzoic acid 3-(2,5-diaminophenyl)benzene-1,2-disulfonic acid 1,3-dimethyl-6-(4-methylsulfanylphenyl)-5H-pyrazolo[3,4-d]pyrimidin-4-one 5-[2-(ethoxymethyl)pyrimidin-4-yl]pyrimidine (3S)-N'-[(4,6-dimethylpyrimidin-2-yl)carbamoyl]pyrrolidine-3-carbohydrazide 3-[(2R)-5-[(4-chloro-1H-pyrrolo[2,3-c]pyridin-7-yl)sulfonyl]oxan-2-yl]prop-1-en-1-amine 5-azido-2,3,4,7-tetrahydropyrrolo[2,1-b][1,3]thiazine-6,9-dione [4-(2,3-difluorophenyl)piperazin-1-yl]-[5-methyl-7-(triazol-2-yl)pyrazolo[1,5-a]pyrimidin-6-yl]methanone;1-propoxyhexane 4-chloro-N-[5,6-difluoro-1'-(2-pyridin-3-ylethyl)spiro[1,2-dihydropyrrolo[2,3-b]pyridine-3,3'-cyclobutane]-1-yl]benzamide;formic acid (4S)-3-[(2,4-dichlorophenyl)methyl]-4-methoxypyrrolidine 2-(4-cyclohexyloxyphenyl)-6,11-dihydrobenzo[d][1]benzazepine 2-[(3S)-2,5-dioxopyrrolidin-3-yl]-N-[1-[4-[2-[(E)-hydrazinylidenemethyl]phenyl]phenyl]sulfonylpiperidin-4-yl]acetamide;dihydrochloride N-[2-(2,5-dimethylphenyl)ethyl]-3-(1H-pyrazol-4-yl)morpholine-4-carboxamide N-[5-[(3S,4R)-3-fluoro-1-propanoylpiperidin-4-yl]-2H-indazol-3-yl]-3,4-dimethoxybenzamide 4-ethyl-2-hydroxy-N,N'-dimethylnaphthalene-1-carboximidamide N'-amino-6-[3-(4-hydroxyphenyl)-1H-indazol-5-yl]pyridine-2-carboximidamide 2-[3-(diethylamino)phenyl]iminoacetaldehyde [2-amino-1-(4-methoxycarbonylphenyl)sulfonylindol-6-yl]oxyboronic acid N-[2-(3,4-dimethoxyphenyl)ethyl]-5-oxo-1-[4-(trifluoromethoxy)phenyl]pyrrolidine-3-carboxamide 2-(azidomethyl)-1-ethyl-4,5-dinitrobenzene 4-[2-(azidomethoxy)-5-chlorophenyl]-1,3-thiazol-2-amine N-(4,6-dimethylcyclohexa-2,4-dien-1-ylidene)pyridine-3-carboxamide 3-(4,6-dimethoxypyrimidin-2-yl)-N-[4-hydroxy-1-[(6-morpholin-4-ylpyridin-3-yl)amino]-1,3-thiazol-5-yl]benzenesulfonamide 2,5-diamino-3-[6-(9H-fluoren-1-yl)pyrimidin-4-yl]oxybenzoic acid 4-[3-(2,3-dihydroxypropoxy)anilino]-1H-pyrimidin-6-one 1-[(2S)-3-cyclopentyloxy-2-hydroxypropyl]pyridin-4-one [2-(dimethylamino)pyridin-4-yl]-(3-phenyl-3,6-dihydro-2H-1,4-oxazin-5-yl)methanone 2-[(1R,2S)-2-methylcyclopropyl]-4-(trifluoromethoxy)benzamide 2-methyl-6-[(3R)-1-[1-[[5-methyl-4-phenyl-2-(4-propan-2-yloxyphenoxy)pyridin-3-yl]methyl]piperidine-4-carbonyl]pyrrolidin-3-yl]pyridazin-3-one 3-[(6-aminopyridine-2-carbonyl)amino]cyclobutane-1-carboxylic acid [(2S)-1-oxo-1-phenylpropan-2-yl]carbamic acid 2,3-dihydroxybutanedioic acid;1-[(Z)-2-(4-methoxyphenyl)ethenyl]-2H-naphthalen-1-ol 2-[(5S)-3-methyl-4,8-dioxo-1,2,6,7-tetrahydro-as-indacen-1-yl]acetic acid 5-[(2,4-difluorobenzoyl)amino]-3-methoxythiophene-2-carboxamide 2-[4-(2,2-diphenylethenyl)phenoxy]acetic acid 2-[3-(cyclopentylcarbamoyl)anilino]-4,7-dioxo-N-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 2-amino-4,6-di(butan-2-yl)phenol 2-ethyl-1-methoxy-4-[2-(4-propan-2-ylphenyl)ethynyl]benzene 3-(furan-2-yl)-1,5-dimethoxynaphthalene 2-N,6-N-bis(3-chlorophenyl)pyridine-2,6-diamine 3-(difluoromethyl)-2,5-bis[(4-methoxyphenyl)methylidene]imidazolidin-1-ium 3-chloroprop-1-ene;[4-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]piperidin-1-yl]-[6-methyl-4-[[4-(trifluoromethyl)benzoyl]amino]cyclohexa-1,3-dien-1-yl]azanide 3-[2-(4,4-dimethylcyclohexyl)ethynyl]benzamide 6-[4,5-dimethyl-2-(7H-purin-6-ylamino)phenyl]-8-methoxy-1-propan-2-ylimidazo[4,5-c]quinolin-4-amine 2-[3-(2-fluorophenyl)propoxy]acetate 2-[(4-methoxyphenyl)diazenyl]phenol N-(2,6-dimethoxypyrimidin-4-yl)-1-methyl-5-oxopyrrolidine-3-carboxamide 1-(5-aminopentyl)-N',N'-dimethylindole-3-carbohydrazide N-[(2S,3R)-1-(cyclopropylamino)-4-methyl-1-oxopentan-2-yl]-3,5-bis(trifluoromethyl)benzamide 7-methyliodanuidyloxy-2,3-dihydroinden-1-one N-[2-[4-[2-(2,5-dimethylphenyl)ethynyl]phenyl]ethyl]-4-pyridin-3-ylbenzamide (2S)-1,3-difluoro-2-methylbutan-1-ol;2-(1-ethoxyethyl)-4-(4-ethenylphenyl)-6,6-bis(fluoromethyl)morpholine N-cyclopentyl-5-[4-(2-phenoxyethoxy)phenyl]-1,3,4-oxadiazol-2-amine 2-benzyl-1,3,4-triazine;hydrochloride 3-chloro-4,5-difluoro-N-[1-(hydroxymethyl)cyclobutyl]benzamide 1-[4-fluoro-2,6-di(propan-2-yl)phenyl]-3-(4-methoxy-6-oxo-5H-phenanthridin-8-yl)urea 2-methoxy-4-[[(1R)-1-(5,6,7,8-tetrahydronaphthalen-1-ylamino)butyl]sulfamoyl]benzoic acid 2-(2,3-dihydropyridin-6-yl)-4-ethoxy-1-[3-fluoro-5-(trifluoromethyl)phenyl]sulfonylazetidine-2-carboxylic acid 4-(3,5-dimethylcyclohepta-1,4,6-trien-1-yl)-2,6-dioxo-N-[2-(4-phenylpiperazin-1-yl)ethyl]piperidine-3-carboxamide N-(1,5-dimethylpyrazol-4-yl)-3H-benzimidazole-5-carboxamide 4-[(6R)-7-acetyloxycarbonyl-1-oxo-2,8,9,10-tetrahydrobenzo[h][1,2,4]triazin-5-yl]butanoic acid N-(2-butylpyrimidin-5-yl)sulfanylacetamide 4-(2,5-dimethyl-4-phenylphenyl)pyridine N-azido-1,3-bis(2H-tetrazol-5-ylmethoxy)butan-1-amine 3-[1-(2,4-dimethoxyphenyl)triazol-4-yl]pyridine (2Z,4Z)-2-[3-[4-(3-aminopropoxy)phenyl]-5-sulfanylidene-1H-1,2,4-triazol-4-yl]hepta-2,4,6-trienoic acid 3-benzyl-4H-triazolo[5,1-c][1,4]benzothiazine 3-(6-bromopyridin-2-yl)oxycyclobutane-1-carboxylic acid 4-[1-[2,3-di(cyclobutyl)imidazo[1,2-b]pyridazin-6-yl]pyrrolidin-2-yl]pyridine-3-carbonitrile 5-[2,3-bis(ethenyl)-1,6-dihydroxy-8H-cyclopenta[b]naphthalen-7-yl]benzene-1,2,4-triol ethane;(Z)-2-[(4-fluorophenyl)methylidene]pentanal 5-[(2E,4Z)-5-aminohepta-2,4,6-trien-3-yl]oxypyridine-2-carboxylic acid 6-bromo-2-methoxy-3,4-dihydroquinoline 4-(2-azido-1,3-diphenylpropan-2-yl)aniline 5-[(E)-2,3-dihydrofuran-4-ylidenemethyl]benzimidazole [3-(4-fluorophenyl)sulfonylcyclobutyl]carbamodithioic acid (E)-N-hydroxy-3-[4-[[2-hydroxyethyl(methyl)amino]sulfanylmethoxy]phenyl]prop-2-enamide (3Z)-4-hydroxypenta-1,3-dien-2-one;iridium;2-phenyl-5H-[1]benzofuro[2,3-b]pyridin-7-ide (2Z)-2-(3-cyclopentyloxypyridin-2-yl)-N-ethyl-N-methyl-2-[6-methylidene-5-oxo-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-ylidene]acetamide 3,5-dihydrobenzo[e]indazole;hydrochloride [3-[4-(1H-indole-2-carbonyl)piperazin-1-yl]azetidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone 2-[(1R)-1-cyclohexylethoxy]-6-nitroaniline (2R,4S)-N-[(Z)-(5-chloro-3-ethyl-1H-indol-2-yl)methylideneamino]-2-phenylpiperidine-1-carboxamide 3-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]-N-pyridin-3-ylpropanamide 4-[4,6-bis(2-methylpropoxy)pyrimidin-5-yl]sulfonyl-N-(1H-pyrazol-4-yl)benzamide [5-[3,5-bis(trifluoromethyl)phenyl]sulfanyl-2,4-dihydroxythiophen-3-ylidene]oxidanium 1-(4,6-dimethoxypyridin-2-yl)pyrrolidine-3-carboxylic acid 3-hydroxy-6,7-dimethoxy-4-[(5-phenylcyclohexa-1,5-dien-1-yl)methyl]chromen-2-one 2-(5-methyl-1,3-thiazol-4-yl)-N-[(6-oxo-1H-pyrimidin-4-yl)methyl]acetamide 3-[(2,5-dichlorophenyl)sulfonylamino]-N-hydroxy-4-[methyl-[1-(2-oxopyrrolidin-1-yl)piperidin-3-yl]carbamoyl]-6-(trifluoromethoxy)naphthalene-2-carboxamide 1-[5-[4-methoxy-2-(trifluoromethyl)benzoyl]-3a-methyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-1-yl]ethanone 3-methyl-4-(2,5,8,11,14-pentazatetracyclo[7.6.0.02,6.010,13]pentadeca-1,3,5,9,12,15-hexaen-14-yl)phenol 2-(4-chloro-3-fluorophenoxy)-N-[3-[(2R,6S)-6-hydroxypiperidine-2-carbonyl]-1-bicyclo[1.1.1]pentanyl]acetamide N-[4-(3,6-dihydro-2H-pyran-4-ylmethoxy)phenyl]sulfanylpyrimidin-2-amine 1-[(E)-2-[3,5-difluoro-4-(2-fluoro-4-methylphenyl)phenyl]ethenyl]-4-ethoxy-2-fluorobenzene 2-[3-(cyclopropylsulfanylamino)phenyl]pyrimidine-5-carboxylic acid 1,3-diamino-2-phenylpropane-2-sulfonic acid N-[4-amino-1-(6-carbamoylpyridin-2-yl)-3,4-dioxobutan-2-yl]-3-pyridazin-4-ylimidazole-4-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]-3-[4-[2-hydroxyethoxy(dimethoxy)methyl]thiophen-2-yl]propane-1,3-dione 1-[1-azido-2-(4-methylphenoxy)ethoxy]-3,5-dichlorobenzene (2R)-1-[2,4-bis(aminomethyl)phenyl]sulfonylpyrrolidine-2-carboxylic acid 4-amino-2-[(1S)-1-[4-(2,3-dimethylindazol-6-yl)phenyl]ethoxy]pyrimidine-5-carboxylic acid 2-(cyclopropanecarbonylamino)-N-[5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridin-2-yl]-7,8-dihydro-5H-pyrido[3,4-b]pyrazine-6-carboxamide 1-(6,8-dimethyl-3,4-dihydro-2H-quinolin-1-yl)propan-1-one N-ethyl-4-[7-methoxy-2,3-dihydro-1H-imidazo[1,2-a]benzimidazole-8-carboximidoyl]piperazine-1-carboxamide 6-(cyclopentanecarbonyl)-2,3-dimethoxybenzoic acid N-[3-(dimethylamino)propyl]-5-[4-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]-1H-indazole-3-carboxamide (E)-1-[4-(2,5-difluorophenyl)piperazin-1-yl]but-1-en-1-amine 2-(4-oxoquinazolin-3-yl)-N-[6-(piperidin-1-ylmethoxy)-5,6,7,8-tetrahydronaphthalen-1-yl]acetamide (3R)-1'-[4-chloro-3-fluoro-2-(trifluoromethyl)phenyl]spiro[1H-indole-3,3'-piperidine]-2-one 4-[3,5-bis(trifluoromethyl)phenyl]-N'-(1H-indole-2-carbonyl)cyclohexane-1-carbohydrazide 7-[[6-[2,4-dimethyl-5-(oxetan-3-yloxy)phenyl]pyrimidin-4-yl]amino]-1-ethylindole-4-carbonitrile N-[4-(azepane-1-carbonyl)phenyl]quinoline-2-carboxamide N-(2,3-dihydrothieno[3,4-b][1,4]oxazin-5-yl)-3-methoxybenzamide 1-(4-bromophenyl)-2-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]ethanone N-[2-(4-bromophenyl)ethyl]-1,1-dioxo-3,4a,5,6,7,8,8a-octahydro-2H-thiepino[2,3-c]pyrrole-4-carboxamide N-benzyl-4-oxo-1H-quinoline-3-carboxamide (2R)-4-[2-cyclopropyl-6-[1-(2,3,5,6-tetrafluorophenyl)ethenylamino]pyridin-4-yl]piperazine-2-carboxylic acid 2-[4-[[4-(3,5-dichloropyridine-2-carbonyl)morpholin-2-yl]methoxy]phenyl]-6H-pyrrolo[3,4-d]pyrimidin-5-one N-[(4S,5R)-1,3-benzodioxol-5-yl]-6-chloro-2-methylsulfanyl-7-[1-(6-propanoylpyridin-2-yl)piperidin-4-yl]oxyquinazolin-4-amine 4-(3,5-ditert-butylphenyl)benzenethiol 2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethanol 5-tert-butyl-N-[[6-(4,4-difluoropiperidine-1-carbonyl)pyridin-2-yl]methyl]-3-(2-hydroxyethoxy)pyrazole-1-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N,4-dimethylpiperazine-1-sulfonamide 2,5-dichloro-N-(3-methylsulfanylphenyl)benzenesulfonamide (4-methylphenyl)methoxy-[[6-[(E,3Z)-5-pyridin-2-ylidenepent-1-enyl]pyrimidin-4-yl]amino]methanol [4-[(3E,5Z)-1-fluorohepta-3,5-dien-3-yl]piperidin-1-yl]-naphthalen-2-ylmethanone (Z)-N',2-dimethyl-3-[5-(1-propan-2-ylpyrazole-4-carbonyl)cyclooctyl]but-2-enimidamide 6-(aminomethyl)-N-[2-[1-[4-(trifluoromethoxy)phenyl]ethylcarbamoyl]pyridin-3-yl]pyridine-3-carboxamide 1-[(2S)-4-[4-(4-methylphenyl)sulfonylpiperazine-1-carbonyl]oxan-2-yl]pyrimidine-2,4-dione 5-[(3E)-4,6-dimethylnona-1,3,7-trien-2-yl]-1,2,4-oxadiazole N-[(6-fluoro-5H-pyrrolo[2,1-c][1,4]benzodiazepine-11-carbonyl)amino]formamide;methoxyethane 3-(benzimidazol-1-yl)-4,6-difluoro-1H-indole 1-(2,4-dimethylcyclohexa-1,3-dien-5-yn-1-yl)-6-fluoro-9H-carbazole 2-(N-hexadecanoylanilino)acetic acid (3,4-dichlorophenyl)-[1-[2-methoxy-5-[methyl(1H-pyrazolo[4,3-d]pyrimidin-7-yl)amino]benzoyl]piperidin-3-yl]carbamic acid 6-chloro-3-[(4-ethoxyphenyl)diazenyl]-1H-indole-2-carboxylic acid 2-hydroxy-1,2-diphenylnonan-5-one N-[[2,3-difluoro-4-(4-methylsulfonylphenyl)phenyl]methoxy]-1H-pyrrolo[2,3-c]pyridine-5-carboxamide 3-azido-1,2,4,5-tetrabromobenzene 3-chloro-5,6-dimethyl-N-[1-(2-oxo-2-pyrrolidin-1-ylethyl)pyrazol-4-yl]thieno[2,3-b]pyridine-2-carboxamide (4Z)-2-methyl-4-[[4-[4-(4-methylphenyl)sulfanylbutoxy]phenyl]methylidene]-1,3-oxazol-5-one 1,1,2,3-tetramethyl-7-nitroindene 3-methyl-6-[2-[(4S)-1,4,5,7-tetrahydropyrano[3,4-c]pyrazole-4-carbonyl]thieno[3,2-b]pyridin-7-yl]oxyimidazo[1,2-a]pyridine-2-carbonitrile 5-benzyl-3,7-dimethyl-6,8-dihydro-[1]benzothiolo[2,3-d]pyrimidin-4-one;N-[(3,4-dichlorophenyl)methylideneamino]formamide 6-[(E)-2,3-diaminobut-1-enyl]-4H-imidazo[5,1-c][1,4]benzothiazin-8-ol 4-[2-[4-(1H-indole-3-carbonyl)piperazin-1-yl]ethoxy]benzaldehyde 3-[4-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(2-methoxyethyl)amino]phenyl]butane-1,1-diol [7-hydroxy-5-[4-(1,3,5-trimethylpyrazole-4-carbonyl)piperazin-1-yl]-1H-indol-2-yl]-[4-[(Z)-prop-1-enoxy]phenyl]methanone 5-(2,6-dimethylphenoxy)-1H-imidazo[4,5-b]pyridine 5-(4-fluorophenyl)-2-phenyl-1,3-dihydropyrazole 1-[2-chloro-3-(trifluoromethyl)phenyl]-3-[1-[4-[5-[4-(dihydroxymethyl)phenyl]-3-(ethoxymethyl)-1,2,4-oxadiazol-2-ium-2-yl]anilino]cyclohexyl]urea (2R)-N-[6-(difluoromethyl)pyridin-3-yl]-1,4-dithiane-2-carboxamide 5-(azidomethyl)-2-methylsulfonylpyridine 4-cyclohexa-1,3-dien-5-yn-1-yl-1-methoxy-2-(trifluoromethyl)benzene;ethane 2-[1-(cyclohexylmethoxy)-3,6-dihydro-2H-pyridin-4-yl]pyrimidine N-[6-(1,3-dimethylpyrazol-4-yl)cinnolin-3-yl]formamide 1,2-dichloro-5-(2-ethylhexoxy)-3-(trifluoromethyl)benzene 6-bromo-3,5-dichloropyridine-2,4-diamine 2-[4,5-dichloro-2-(methylideneamino)anilino]-N-[(Z)-(1H-pyrrol-2-ylhydrazinylidene)methyl]acetamide 2-(1H-indazol-4-yl)-1,3,6,7-tetrahydroimidazo[4,5-c]pyridine 5-[2-fluoro-6-[2-(1,3-thiazol-4-yl)ethoxy]phenyl]pyrimidin-2-amine 1-(2,4,6-trichlorophenoxy)-3-[2-(4-phenylpiperazine-1-carbonyl)anilino]propan-2-one N-[2-[[5-chloro-6-(3,4,5-trimethoxyanilino)pyrimidin-4-yl]amino]phenyl]-2-(difluoromethyl)-2-sulfanylideneacetamide;ethane 2-(1,5-diphenylpyrazol-3-yl)-4,6-bis[(Z)-prop-1-enoxy]pyrimidine 4-(5-methylthiophen-2-yl)-2,6-dimorpholin-4-ylpyrimidine-5-carbonitrile 1-[1-cyclopropyl-4-fluoro-2,5-bis(trifluoromethyl)indol-3-yl]ethanone 5-methoxy-4,6-dimethyl-7-[(4-methylpiperazin-1-yl)methyl]-2,3-dihydroinden-1-one N-(4-hydroxycyclohexyl)-4-[2-[(5-methoxypyridine-3-carbonyl)amino]phenoxy]piperidine-1-carboxamide 4-(cyclopentylamino)-6,7-difluoroquinoline-3-carboxamide 5-(difluoromethyl)-2-[4-(3,3-difluoroazetidin-1-yl)piperidine-1-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyridin-4-one (3S)-N-benzyl-1-[4-chloro-2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]piperidine-3-carboxamide N-(2,4-difluorophenyl)-3-[1-(1,5-dimethylpyrazol-4-yl)ethoxy]pyrido[2,3-b]pyrazin-6-amine 2-[(3R)-5-(4-chlorophenyl)-1-cyclopropyl-2-oxopyrrolidin-3-yl]acetic acid 1-[[2-chloro-4-(trifluoromethyl)phenyl]carbamoylamino]-3-[3,5-dimethoxy-4-(phenoxymethyl)phenyl]thiourea N-[4,5-dichloro-2-[(3S)-4,4,4-trifluoro-3-methylbutanoyl]phenyl]-1-benzothiophene-6-carboxamide 3-benzyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carboxamide 5-[(2R)-2-methylmorpholine-4-carbonyl]pyrazine-2-carboxamide 3-(ethoxymethyl)-1,5-diphenyl-2H-pyridine 2-[(2-ethoxyphenyl)methylidene]morpholine N-(4-methylpyridin-2-yl)-6-phenylimidazo[1,2-b]pyridazine-7-carboxamide 2-[(3-hydroxyphenyl)diazenyl]-5-octoxyphenol 1-[(2S,4R)-4-hydroxy-2-phenyl-1-oxa-9-azaspiro[5.5]undecan-9-yl]-4-pyrrolidin-1-ylbutan-1-one 4-methoxy-5-(2-phenylethyl)piperidine 3-(5,5-dimethyl-4H-imidazol-1-yl)-N-[2-oxo-2-[3-(trifluoromethoxy)anilino]ethyl]propanamide 3-amino-N-[4-(2-hydroxyethyl)-2-methoxyphenyl]propanamide N-[(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-2,3-dihydroimidazo[1,2-c]quinazoline-8-carboxamide 1-[5-(4-fluorophenyl)furan-2-yl]sulfinyl-6-methoxyindole (2S)-4-amino-2-[[5-methyl-6-[2-(trifluoromethyl)phenyl]pyridine-3-carbonyl]amino]butanoic acid 4-azido-N,2-dimethylbenzenesulfonamide 2-[2-(5-chlorobenzotriazol-2-yl)phenyl]benzene-1,3-diol 2-[(4-acetylpiperazine-1-carbonyl)amino]-N-[1-cyclohexyl-3,3-dimethylbutan-2-yl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide N-[2-(6,7-dimethoxy-3-oxoquinoxalin-4-yl)propanoylamino]-1-phenylcyclopropane-1-carboxamide N-methyl-4-[2-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-3-yl)ethynyl]benzamide N-[4-methoxy-2,6-di(propan-2-yl)phenyl]acetamide 2-[(3R,4S)-3-amino-1-methylpiperidin-4-yl]-N-(2,5-dimethylphenyl)ethanimidate N-(4,5-dimethyl-2-phenyldiazenylphenyl)-2H-tetrazol-5-amine 1-[6-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-2H-chromen-3-yl]pyrrolidine 2-[(7-aminonaphthalen-1-yl)methoxy]acetic acid 6-[4-chlorobutyl(2,2-dimethoxyethyl)amino]-2-sulfanylidene-1H-pyrimidin-4-one 2-(azetidin-1-yl)-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one N-(5-methylthiophen-2-yl)sulfonylacetamide 4-[(3R)-2,2-dimethylmorpholin-3-yl]-3-nitrobenzoic acid 3-(3,4-dimethoxyphenyl)butane-2,1,4-trione;ethane 2-[(4S,8aS)-8a-(hydroxymethyl)-3,4,6,7,8-pentahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-N-(5,6-dichloropyridin-3-yl)acetamide 2-(4-chlorophenoxy)-N'-hydroxypyridine-3-carboximidamide 4-[1-(4-ethoxy-3-methylphenyl)-2,3-dihydrotetrazol-5-yl]pyridine (1S)-N-methyl-2,3-dihydro-1H-indene-1-carboxamide;5-[[4-(piperidine-4-carbonylamino)phenyl]carbamoyl]pyrrolidine-1-carboxylic acid N-methyl-2-[1'-(thiophene-3-carbonyl)spiro[4,7-dihydrotriazolo[5,1-c][1,4]oxazine-6,3'-pyrrolidine]-3-yl]acetamide;2,2,2-trifluoroacetic acid 3-[4-chloro-5-(2,2,2-trifluoroethoxy)pyridin-2-yl]-1-methyl-6-(trifluoromethyl)imidazo[4,5-c]pyridin-2-one 1-ethyl-N-[[3-methoxy-4-(2H-tetrazol-5-yl)phenyl]methyl]piperidine-2-carboxamide 4-N,4-N-diethylquinazoline-2,4-diamine 2-[(4-methylpyridin-3-yl)oxymethyl]-N-pyrrolidin-1-ylsulfonylcyclohexane-1-carboxamide (E)-N'-[5-chloro-2-(3,4-difluorophenyl)sulfinylpyridin-3-yl]-N-ethylbut-1-ene-1,4-diamine 2-[(4-fluorophenyl)methoxy]-N-[4-(3-hydroxypropylsulfamoyl)-1H-indol-7-yl]pyridine-3-carboxamide 3-amino-5-(4,5-dimethylcyclohexa-1,3-dien-1-yl)pentan-2-one;ethane 1-chloro-4-[3-(2,3-dichlorophenyl)propoxy]-2-methylbenzene 5-N-[2-(dimethylamino)ethyl]-3-N,4-dimethylpyrimidine-2,5-diamine 4-[3-(2,5-difluorophenyl)propyl]-1-methoxycyclohexa-1,3-diene 2-(5-bromothiophen-2-yl)-3,4-difluoroaniline (4S)-2,4-diamino-7-benzyl-5-[2-chloro-6-(difluoromethoxy)phenyl]-4H-pyrano[3,2-c]quinoline-3-carbonitrile N-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carboxamide 2-[4-[(E)-3-(3,5-dimethoxyphenyl)prop-1-enyl]-1-oxoisoquinolin-2-yl]acetonitrile 3-[(3,6-dioxocyclohepta-1,4,6-trien-1-yl)methoxy]-N-[(2S)-1-methoxypropan-2-yl]benzamide [1-(2,3-dihydro-1H-inden-5-yl)-2,3-dimethylbutylidene]hydrazine 2-chloro-5-[1,3-dioxoisoindol-2-yl]pyridine-4-carbonitrile (E)-3-[4-methoxy-6-(trifluoromethyl)pyridin-2-yl]prop-1-ene-1,1,3-triol 1-(2,4-dichlorophenoxy)-3-[2-ethyl-5-(4-methylphenyl)pyrazol-3-yl]urea 7-[6-(4-azidophenyl)pyridin-2-yl]furo[3,2-c]pyridine 1,3-dichloro-5,6-bis(fluoromethyl)naphthalene (Z)-1-[3,4-difluoro-2-(triazol-2-yl)phenyl]-N-[(4-phenoxyphenyl)methoxy]ethanimine 2-methyl-N-[5-(5-phenyl-1H-imidazol-4-yl)cyclohexa-1,3-dien-1-yl]propanamide 5-[2-(4-cyclopropylphenyl)ethynyl]pyridine-3-carbonitrile 5-(2,4-dichlorophenyl)sulfanyl-1-methylideneindole-3-carboxylic acid 1-[5-[5-(2-fluoro-3-methylphenyl)-4,5-dihydro-1H-imidazol-2-yl]-6-methoxypyridin-2-yl]piperidine-4-carboxylic acid;dihydrochloride (E)-1-[4-[(Z,2E)-4-amino-2-ethylidenehex-3-enoyl]piperazin-1-yl]-3-[4-(difluoromethoxy)phenyl]prop-2-en-1-one (1-aminocyclohexyl)-(3,4-diphenylpiperazin-1-yl)methanone (4E)-2,3-dimethylhepta-1,4-diene;ethane;1-[6-methoxy-5-methyl-4-[(4-methylphenyl)methoxy]pyridin-2-yl]ethenamine 5-(4,6-dimethylpyridin-2-yl)oxycarbonyl-1-[(2S)-1-phenylbutan-2-yl]-3,6-dihydro-2H-pyridine-4-carboxylate 1-[4-(3-cyclopropylpyrazol-1-yl)piperidin-1-yl]ethanone 4-azido-N',2,3-trichlorobenzohydrazide 2-[3-(3,5-difluoropyridin-4-yl)-1H-indol-6-yl]cyclohexan-1-ol 1-[(4-chlorophenyl)methyl]pyrrolidine;2,3-diaminoquinoxaline-6-carbonitrile N-[(E)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]-2-[4-(4-fluorobenzoyl)phenoxy]acetamide 3-[[2-(4-chloroanilino)-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxybenzamide (3S)-2-N-[2,6-dimethyl-4-(1H-pyrazol-5-ylmethoxy)phenyl]pyrrolidine-1,2-dicarboxamide 1-(4,4-dimethylcyclohexa-1,5-dien-1-yl)naphthalene 2-[(1R)-1-ethylsulfinylethyl]-5,6,7,8-tetrahydro-3H-pyrido[4,3-d]pyrimidin-4-one 2-[(1S)-1-naphthalen-1-ylethoxy]propanoic acid 4-(7-methoxy-2,3,5,6,8,9-hexahydrobenzo[d][1]benzazepine-10-carbonyl)pyrrolidin-2-one 4-fluoro-6-[(E)-pent-3-enyl]naphthalene-2,7-diol 4-methyl-3-[2,2,2-trifluoro-1-[8-(4-pentanoyl-2H-pyridin-1-yl)naphthalen-2-yl]ethoxy]benzonitrile N-[(2S)-1-[(5-methoxypyridine-3-carbonyl)amino]propan-2-yl]-7-propyl-4,10,11-trioxa-1,8-diazatricyclo[7.4.0.03,7]trideca-9,12-diene-12-carboxamide 4-chloro-N'-hydroxy-1,3-benzoxazole-2-carboximidamide 2-(dimethylamino)-6,7-dimethyl-4-[(1R)-5-methylcyclohexa-2,4-dien-1-yl]pyrrolo[3,4-d]pyrimidin-5-one 4-[5,5-bis(4-chlorophenyl)hexanoylamino]benzoic acid (2S)-5,6-dimethyl-N-propan-2-yloxy-3,4-dihydro-1H-naphthalene-2-carboxamide 5-chloro-1,3-diethylbenzene;(E)-N-[(2R)-4-ethoxy-1-[6-oxo-6-(phenylmethoxyamino)hexanoyl]pyrrolidin-2-yl]but-2-enamide 5-[1-(2,6-dichlorophenyl)piperidin-4-yl]-2-methoxy-3H-pyrido[2,3-d]pyrimidin-4-one 3-N-(4,5-dimethylfuran-2-yl)benzene-1,3-disulfonamide 2-[3,4-dichloro-5-(1H-pyrrole-2-carbonyl)phenyl]propanamide N-(2,6-dibromopyridin-4-yl)-2-methoxy-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)acetamide 3-[3-[2-(3,5-dimethoxyanilino)ethyl]pyridin-4-yl]sulfanylaniline 5-amino-2-(3,4-dimethylphenoxy)benzonitrile 4-[6-fluoro-2-[3-(hydroxymethyl)phenyl]-1,3-benzothiazol-5-yl]phenol 2-[(2,3-difluorobenzoyl)amino]-5-sulfooxycarbonylterephthalic acid 1-amino-3,3-difluoro-2H-acridin-4-one N-[(1Z,3E)-4-fluorohexa-1,3-dienyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide N-cyclopropyl-2-[3-(difluoromethoxy)phenoxy]acetamide (2S,4R)-1-[3-(2-butylphenyl)propanoyl]-N-cyclohexyl-4-hydroxypyrrolidine-2-carboxamide 5-chloro-6-methyl-2,3,4,9-tetrahydro-1H-carbazole N-[(2S)-3-methyl-1-oxobutan-2-yl]formamide;methylidene-[1-oxo-7-[6-(2-phenylmethoxyethylamino)hexylsulfonylmethyl]-2H-isoquinolin-5-yl]azanium N-[2,6-di(propan-2-yl)phenyl]-1-phenylmethoxymethanimine 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]-5-(methoxymethyl)pyridine 2-(1H-imidazol-5-yl)-3-[4-(2-pyrrolidin-1-ylethoxymethyl)phenoxy]cyclobutan-1-one 1-(3,4-difluorophenyl)-N-(2H-pyrazolo[3,4-b]pyridin-6-yl)methanesulfonamide (3S)-2,6-dimethyl-4-propan-2-yl-3,5-dihydro-1H-2,7-naphthyridin-4-imine 4-[1-(2,3-dihydronaphthalen-1-yl)cyclopropanecarbonyl]oxybutanoic acid 3-[(2Z)-2-[1-(4-aminophenyl)propylidene]hydrazinyl]-4H-1,2,4-triazin-5-one 2-[2,4-difluoro-N-(3-methylbut-2-enyl)anilino]acetonitrile 2-(3,5-dihydroxyphenyl)-7-methylheptanoic acid 2-[3-(4-benzoylpiperazine-1-carbonyl)piperidin-1-yl]-N,N-dimethylpyrimidine-5-carboxamide 5-[2-[4-(3,6-dihydro-2H-pyran-4-yl)phenyl]cyclobuten-1-yl]-1-ethoxycarbonylpiperidine-3-carboxylic acid 6-[[4-(trifluoromethyl)phenyl]methylamino]spiro[2H-1-benzofuran-3,4'-piperidine]-5-ol 2-hydroxy-4-(3-methylsulfonylbenzoyl)cyclopentane-1-carboxylic acid 4-(methoxymethyl)-2-[(1R,3S)-3-(4-pyrazol-1-ylpiperidin-1-yl)cyclopentyl]-1H-pyrimidin-6-one 2-[2-(3,4-dimethoxyphenyl)ethyl]-6-methoxy-5H-pyrrolo[2,3-b]pyrazine 2-[6-(4-tert-butylcyclohexen-1-yl)pyridine-3-carbonyl]-8-oxa-2,5,11-triazabicyclo[10.4.0]hexadeca-1(16),12,14-triene-13-carboxylic acid 6-[4-[3-[6-ethoxy-2,2,7-trimethyl-9-(oxan-2-yl)purin-8-yl]propyl]piperidine-1-carbonyl]pyridine-3-carbonitrile 3-[4-chlorobutyl(methoxycarbonyl)amino]benzenesulfonic acid 2-amino-6-[(4-oxo-3H-quinazolin-2-yl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonitrile 4-[2,3-dihydroxypropyl(2,2-dimethoxyethyl)amino]benzenesulfonamide ethane;N-[2-(methylamino)ethyl]-3-phenylpropanamide 5-ethylsulfonyloxy-6-methylpyrazine-2-carboxylic acid (E)-3-[2-ethoxy-4-[[1,1,3]trimethyl-5-oxo-4-(3-phenylpropanoylamino)-6H-pyridazin-6-yl]anilino]prop-2-enoic acid N'-[4-chloro-2-(trifluoromethyl)phenyl]sulfanylacetohydrazide 4-N-azido-1,3-bis(2-methylpropoxy)benzene-1,4-disulfonamide 4-(1H-benzimidazol-2-yl)-N-[6-(2,5-dimethylpyrrolidin-1-ium-1-carbonyl)-1,3-benzothiazol-2-yl]butanamide (2S,3R)-1-ethyl-N-[1-[4-fluoro-6-oxo-5-(trifluoromethyl)-1H-pyridazin-3-yl]piperidin-4-yl]pyrrolidine-3-carboxamide [3-amino-2-[4-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]prop-2-enylidene]azanium N-[4-(2-nitrophenyl)butanoyl]bicyclo[1.1.1]pentane-1-carboxamide 2-(1,3-benzodioxol-5-yl)-N-hydroxy-3H-benzimidazole-4-carboxamide 2-(4,5-dimethylpyrimidin-2-yl)benzene-1,3-diamine;hydrochloride (E)-3-[(2R,4S,5R)-2-(2,3-dihydro-1H-indene-1-carbonyloxymethyl)-3,4-dihydroxy-6-(hydroxymethyl)oxan-5-yl]prop-2-enoic acid 7-ethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine 1-[(4R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazin-4-yl)azepan-4-yl]pyrrolidin-3-ol 2-[N-[(4-nitrophenyl)methyl]-3-sulfoanilino]propanoic acid 4-[2-(methoxymethyl)-4-(1,3-oxazol-5-yl)phenyl]morpholine (2R)-2,4-diamino-N-[1-[(3R,5S)-3,5-dimethylpyrrolidine-1-carbonyl]piperidin-4-yl]-4-phenylbutanamide 3-(2,6-diethylphenyl)imino-7-[(2Z,4E)-1,5-dihydroxyocta-2,4-dien-3-yl]sulfanylheptane-2,4-diol (E)-3-[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]-2-sulfanylprop-2-enoic acid (E)-N,3-dimethyl-4-[2-methylidene-3-[3-oxo-6-(quinolin-4-ylamino)pyridazin-1-yl]pyrrolidin-1-yl]but-2-enamide 2-[2-chloro-6-fluoro-3-(propanoylamino)phenyl]acetic acid 3-[6-(2,4-difluorophenyl)pyridin-3-yl]-5-methylideneheptanoic acid 1-benzyl-4-[(3E)-hexa-1,3,5-trien-2-yl]piperazine 2-chloro-4,6-dimethoxy-N-phenylbenzamide 1-(3,5-dichlorophenyl)sulfonyl-4-[5-methyl-6-(1H-pyrazol-5-yl)pyridin-2-yl]piperazine ethene;4-[(1E,3Z)-1,2-dichlorohexa-1,3,5-trienyl]benzonitrile 2-(1H-benzo[g]indol-3-yl)decanoic acid N-[1-(2,5-dimethoxyphenyl)propan-2-yl]-1H-benzimidazole-4-carboxamide 1-[3,4-bis(2-phenylethynyl)phenyl]piperidine (E)-3-[5,7-bis(ethenyl)quinolin-8-yl]prop-2-enenitrile;methanol 2,4-dichloro-N-[5-chloro-3-(2-methoxyphenyl)pentyl]aniline 4-(cyclohexylamino)-2-[1-methyl-5-[3-(piperidine-1-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]pyrazol-4-yl]pyrimidine-5-carbonitrile (2R)-1,3-bis[3-[4-(dimethylamino)butyl]phenyl]propane-2-thiol;hydrochloride (2R,3S)-3-phenyl-2-[3-[4-(pyridin-2-ylamino)piperidine-1-carbonyl]phenoxy]butanamide 3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-7-methylsulfanylchromene 2,4-ditert-butylthieno[3,2-b]pyridine 3-(2-chlorophenyl)-2-(2,6-dimethoxyphenyl)-4H-chromene (2R)-3-[1-methoxy-6-(3,4,5-trimethoxyphenyl)naphthalen-2-yl]propane-1,2-diol 2-[2,6-dimethyl-4-(3-nitroso-1H-indene-2-carbonyl)phenoxy]acetic acid 1-(5-chloro-2-hydroxyphenyl)-3-imino-6,7-dimethoxy-4H-quinoxalin-2-one 5-amino-4-(3-bromo-2,6-difluorophenyl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 4-(2,6-dimethylphenyl)-2-phenyl-1,3-dioxolane 3-cyclopropylsulfonylpyridine-2,4-diamine N-[(2S)-3,4-dihydro-2H-chromen-7-yl]-6-methoxy-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide 5-bromo-3-[2,6-dichloro-4-(trifluoromethyl)phenyl]-1-methyl-1,3-dihydrofuro[3,4-c]pyrrole 1-[4-(azidomethyl)phenyl]ethanesulfonate N-[[2,3-difluoro-4-(trifluoromethyl)phenyl]methyl]pyridine-3-carboxamide 4-(2,5-dimethoxyphenyl)-N,N-bis[2-(trifluoromethyl)phenyl]aniline 1-(8,9,10,11-tetrahydrobenzo[d][3]benzazepin-6-yl)butan-2-amine (2-chloropyrimidin-4-yl)-(2,4-dimethoxyphenyl)methanone ethane;5-methylnaphthalene-2,3-dithiol N-benzyl-1-(4-but-2-enoxyphenyl)methanimine 2-(3,4-dimethoxyphenyl)-4-methyl-5H-1,2,4-triazole [4-(4-hydroxybutan-2-yl)piperidin-1-yl]-[7-methyl-5-(2,3,5-trifluorophenyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone 5-chloro-4-N-(3-fluorophenyl)pyrimidine-2,4-diamine (2S)-4,6-diamino-1-[[4-[[2-methylpropanoyl-[[5-(trifluoromethoxy)thiophen-2-yl]methyl]amino]methyl]phenyl]methylamino]hexane-3,5-diol 2-[3-hydroxy-4-(4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-5-carbonyl)phenyl]acetonitrile 2-[3,5-dichloro-4-(1H-indole-2-carbonyl)phenyl]-6-(hydroxymethyl)oxan-4-ol;ethane 3-[3-ethoxy-5-(2H-tetrazol-5-yl)phenyl]-4,6,7-trimethylchromene 7-(2,4-dimethylphenyl)naphthalene;ethane N-[2,4-dimethyl-5-(pyridine-4-carbonyl)phenyl]pyridine-3-carboxamide 4-azido-2,6-dimethoxybenzoic acid N-[(Z)-(3,5-dibromo-2-hydroxyphenyl)methylideneamino]-1-benzofuran-2-carboxamide 4-chloro-7-methyl-6-(trifluoromethoxy)quinoline (Z)-1-N-methyl-1-N,2-N'-diphenylpent-1-ene-1,2,4,5-tetramine 1-(2,3-dimethylphenyl)sulfanylpiperidine 1-(4,6-dimethoxypyrimidin-2-yl)azetidine-3-carboxylic acid 3-[(3S,4R)-3-fluoro-1-(4-propanoylphenyl)sulfonylpiperidin-4-yl]-5-methoxy-2-methyl-6H-pyrazolo[4,3-d]pyrimidin-7-one ethane;2-methyl-1-(5,7,10,11-tetrazatricyclo[7.4.0.02,6]trideca-1(13),3,6,8,11-pentaen-13-yl)propan-1-one (2-chloropyrimidin-5-yl)-[(1S,3R)-3-[5-fluoro-6-(2-methoxypyridin-4-yl)indazol-1-yl]cyclopentyl]methanone 2-[2,3,5,6-tetrafluoro-4-(hydroxymethyl)phenyl]-3H-isoindol-1-one 4-[(2,5-dimethylphenyl)methylidene]piperidine;hydrochloride 5-(2,6-dimethylphenyl)quinoline 6-methoxy-N,5-dimethyl-N-[(1-methylimidazol-2-yl)methyl]pyridine-3-carboxamide 7-chloro-6-(3,4-dichlorophenyl)imidazo[1,2-b]pyridazine 4-[(2Z)-2-(3-oxo-6,7,8,9-tetrahydrooxy-4H-quinolizin-1-yl)penta-2,4-dienoyl]piperazine-1-carboxylic acid (1S)-N,2-diethyl-6-methoxy-2-[(E)-4-oxohex-2-en-3-yl]-1,3-dihydroindene-1-carboxamide (4S)-2-[5-[6-amino-1-[3,3-difluoro-2-(3-hydroxyphenyl)butanoyl]pyrazolo[4,3-c]pyridin-3-yl]pyridin-3-yl]oxepane-4-carboxylic acid 2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonylamino]-5-fluorobenzoic acid (2E)-N,3-bis[4-[difluoro(phosphanyl)methoxy]phenyl]-2-hydroxyiminopropanamide 3-(4-tert-butylphenoxy)sulfonylbenzenethiol [2-(2-fluorophenyl)morpholin-4-yl]-(3,5,6-trimethylpyridin-2-yl)methanone N-[3,4-bis(ethenyl)cyclohexa-1,5-dien-1-yl]-9H-fluoren-9-amine 1-[5,8-dimethyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]ethanone;2,2,2-trifluoroacetic acid 3-aminosulfanyl-6,7-difluoroquinoline-8-carboxylic acid 2-cyclohexa-1,3-dien-1-yl-2-(2,4-dihydroxyphenyl)ethanol 1-[3,4-dimethyl-5-(1H-pyrazol-4-yl)phenyl]-3-methoxypropan-2-one 3-[(2-chloro-5-methoxyphenyl)methyl]-5-(dimethoxyphosphorylmethylidene)-1-[(2R,3S)-2-hydroxyhexan-3-yl]-2H-pyrido[2,1-f][1,2,4]triazine-4,6-dione 4-[(3R,5S)-7-chloro-5-phenyl-1,2,3,4-tetrahydropyrido[4,3-b]indol-3-yl]phenol ethane;6-(4-methylphenyl)naphthalene-2,3-diamine 1-ethyl-5,6,7-trimethoxyisoquinoline;hydrate 1-chloro-2-(3-chloropropoxy)benzene;ethane 1-(cyclopropylmethyl)-3-[(3,5-dichloropyridine-4-carbonyl)amino]thiourea (2S,4R)-1-[3,4-difluoro-2-[[methyl(propan-2-yl)amino]methyl]phenyl]sulfonyl-4-fluoropyrrolidine-2-carboxylic acid 2-(4,5-dichlorothiophen-2-yl)-N-[[4-(hydroxymethyl)phenyl]methyl]acetamide 4-[5-[(E)-2-chloroprop-1-enyl]thiophen-2-yl]pyridine 1-[5,7-dichloro-6-(methylamino)pyrazolo[4,3-b]pyridin-2-yl]ethanone 2-(N,4-diaminoanilino)ethanol 2-[2-(3-cyclopropylpyridin-4-yl)ethynyl]-1H-quinoline 2-methyl-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]-N-phenacylpropanamide 3-N-(2,4-dimethoxyphenyl)-6-(1H-indazol-5-ylamino)-2,7-naphthyridine-3,8-dicarboxamide 3-[2-(4,4-difluoropiperidin-1-yl)ethoxy]pyridine 2,3-bis(4-butylsulfanylphenyl)propanedioic acid N-benzyl-1,4-diazacyclododecan-1-amine 2-[(3S,4R)-4-[(4-chlorophenyl)carbamoyloxymethyl]-1-(oxan-4-yl)pyrrolidin-3-yl]benzoic acid 4-[(1E,3E)-4-hydroxy-3-methoxybuta-1,3-dienyl]benzaldehyde 4-azidooxy-2-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline (E)-N-[2-(cyclopropylsulfonylamino)-4,6-difluorophenyl]-3-[[2,5-dimethoxy-4-[6-[(2R)-oxepan-2-yl]oxypyridin-3-yl]phenyl]methylideneamino]-N'-methanimidoylbut-2-enimidamide 2-[4-(4-methoxypyridin-3-yl)phenyl]propanoic acid 4-(4-azidocyclohexyl)oxybenzene-1,3-diamine 1-bromo-4,5-di(propan-2-yl)imidazole N-[5-(4-chlorophenyl)-2-oxo-1H-pyridin-3-yl]-3,3a,4,7a-tetrahydroisoindole-1-carboxamide 1-[(5R,7S)-3-chloro-4,5,6,10-tetramethoxy-9-oxa-2-thia-14-azatricyclo[13.4.0.05,10]nonadeca-1(19),15,17-trien-12-yl]ethanone N-(1,2-diphenylethenyl)-2-[3-(3-methoxyphenyl)-5-(trifluoromethyl)pyridin-2-yl]sulfanylpropanamide 2-[3-(2,5-dioxopyrrolidin-1-yl)-2-hydroxypropyl]isoindole-1,3-dione 2-amino-5-(3,4-dichlorophenyl)sulfanylphenol 1-(4-ethenylphenyl)-3,5,6-trifluorobenzimidazol-2-one N-[5,6-bis(methylsulfanyl)pyridin-2-yl]-3-[2-ethyl-4-(trifluoromethyl)phenyl]propanamide 4-[6-(2,4-difluorophenyl)pyrimidine-4-carboximidoyl]-5-methylsulfanylthiophene-3-carboxamide N-[4-(2,6-dipyridin-3-ylphenyl)-1-hydroxybutan-2-ylidene]hydroxylamine;ethane N-[(E)-1-aminobut-2-enylidene]-6-chloro-3,4-dihydroquinoline-8-carboxamide;hydrochloride (2R)-N-methyl-3-[[4-[1-[4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethyl]piperazin-1-yl]sulfonylamino]-2-(oxan-4-ylamino)propanamide 2-[(1R,5S)-3-acetyloxy-6-oxobicyclo[3.1.0]hexanyl]-5-methyl-4H-benzotriazole-6-carboxylic acid 3-[1-hydroxy-2-(naphthalen-1-ylamino)ethyl]phenol 2-[1,3-benzothiazol-2-yl(2,4-dichloropyrimidin-5-yl)amino]ethanol 5-[8-chloro-1,7-dihydroxy-3-(2-methoxyphenyl)benzo[f]chromen-2-yl]-6-methoxynaphthalene-2-carboxylic acid N-ethenylsulfonyl-2-methoxy-N-(4-nitrophenyl)acetamide 3-[4-methyl-2,5-bis(trifluoromethyl)anilino]propanenitrile (1S,3S)-N-[2-[4-chloro-5-hydroxy-6-(trifluoromethyl)pyrimidin-2-yl]oxyphenyl]sulfanyl-3,4-dimethylcyclopentane-1-carboxamide 2-[(1,4-dimethylimidazol-2-yl)sulfonylamino]-3-[5-(2-ethoxyphenyl)furan-2-yl]propanoic acid 3-[(7S)-4-(2,6-dimethylphenyl)sulfonyl-7-propan-2-yl-1,4-diazepane-1-carbonyl]benzoic acid 3-[2,6-difluoro-N-(methoxyiminomethyl)anilino]phenol 2-[(6S)-6-ethylmorpholine-4-carbonyl]-N-(1H-pyrazol-5-ylmethyl)imidazo[1,2-a]pyridine-7-carboxamide 4-fluorobenzenesulfonate;2-methylpropanedioic acid 4-bromo-6-(cyclopropanecarbonylamino)-N-[4-methyl-1-[(2R)-4,4,4-trifluorobutan-2-yl]piperidin-3-yl]pyridine-3-carboxamide 5-[2,3-dichloro-4-(trifluoromethyl)phenoxy]-N'-hydroxypyridine-2-carboximidamide ethane;2-(3,4,5-trimethoxyphenyl)propanoic acid 1-[7-(2,5-dimethylphenoxy)sulfanyl-6-fluoro-4H-azepin-3-yl]cyclopropane-1-carboxamide 1-[7,8-bis(4-chlorophenyl)-2-oxo-9H-purin-3-yl]propan-2-one 1-[2,6-dichloro-4-(2-methylpropyl)phenyl]ethanimine 1-[2,6-di(propan-2-yl)phenyl]-3-[5-(5-methylpyridin-2-yl)hexa-1,5-dien-4-yloxy]urea N-(diaminomethylidene)-7,8-bis(ethenyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide 2-bromo-4,5-dimethylpyridine;ethane 2-amino-6-[[3,5-dichloro-4-(3-methoxypropoxy)phenyl]methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-[6,8-dichloro-2-(methylamino)purin-9-yl]cyclopentan-1-ol 2-amino-1-(4-chlorophenyl)-6-fluoro-8-methoxyquinazolin-4-one (6-chloro-2,3-dihydro-1H-indol-5-yl)-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methanone 2-[4,5-bis(phenylmethoxy)cyclohexa-1,3-dien-1-yl]oxyacetate 3-(2,4-dichlorophenyl)propanehydrazide;hydrochloride 4-azido-2,5-dimethyl-N-[3-(4-nitrophenoxy)phenyl]pyrazole-3-carboxamide 3-[4-(benzenesulfonamido)phenyl]-5,6-dimethoxy-1H-indole-2-carboxamide 2-[[(E)-3-methylbut-1-enoxy]methoxy]-4,6-bis(trichloromethyl)aniline (2-chloro-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-3-yl)-[4-(1H-pyrazol-4-yl)piperidin-1-yl]methanone N-[2,2,2-trifluoro-1-(4-phenylmethoxypiperidin-1-yl)ethyl]methanesulfonamide 4-[N-ethylsulfonyl-2,6-difluoro-3-(trifluoromethoxy)anilino]butanoic acid [3-bromo-1-(4-methoxynaphthalene-2-carbonyl)indol-4-yl]-pyridin-4-ylmethanone N-[1-(3,5-dimethoxyphenyl)-2-hydroxyiminoethylidene]propanamide N-ethyl-4-[2-[(6-methoxypyridine-3-carbonyl)amino]imidazo[1,2-a]pyridin-5-yl]-N-[3-(trifluoromethyl)phenyl]piperazine-1-carboxamide N-[(4,6-dimethylpyridin-3-yl)methyl]-8-[2-ethoxy-5-(1H-pyrazol-4-yl)phenyl]-7-fluoro-[1,2,4]triazolo[1,5-c]quinazolin-5-amine 2-(1-bromo-2H-pyridin-4-yl)-6-propanoyloxybenzoic acid 1-methyl-N-(6-pyridin-2-ylisoquinolin-3-yl)piperidine-4-carboxamide N-[3,5-difluoro-4-(methylamino)phenyl]-2-hydroxy-3-(1H-pyrazole-5-carbonylamino)-2-(trifluoromethyl)propanamide 2-[(2Z)-2-[1,5-bis(4-methoxyphenyl)-3-methyl-6-oxopyrimidin-2-ylidene]hydrazinyl]-N'-hydroxyethanimidamide 2-[(5Z)-4-oxo-5-(quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid 2-[5-carbamoyl-2-methyl-9-(3,4,5-trifluorophenyl)carbazol-4-yl]oxyacetic acid 2-[3,5-ditert-butyl-4-hydroxy-N'-(6-oxobenzo[c]chromen-8-yl)anilino]ethanol;ethane 2-[(6-methyl-5H-indolo[3,2-c]quinolin-12a-ium-11-ylidene)amino]propan-1-ol 3-[(1S)-1,2-diphenylethyl]-8-methylbenzo[f]quinazolin-1-amine N-(2,6-dimethoxypyrimidin-4-yl)-4-[ethenylsulfonyl-(3-ethoxy-3-oxopropanoyl)amino]benzenesulfonamide 2-methylsulfanyl-4,8-dipyridin-2-ylpyrazolo[1,5-a][1,3,5]triazine [4-(2,3-dihydrofuran-5-yl)naphthalen-1-yl]boronic acid 3-(6,7-dihydronaphthalen-1-yloxy)-N-[2-[4-(2-hydroxyethylamino)phenyl]ethyl]propanamide 6-tert-butyl-1'-[(1-methylpyrazol-4-yl)methyl]spiro[3,4-dihydrochromene-2,4'-piperidine] 2-(ethylaminomethyl)-7H-purin-6-amine;hydrochloride (2-aminophenyl)sulfanylsulfanium 3-[3-chloro-4-(1,2,4-triazol-1-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 2,4-dinitro-1H-pyrrolo[2,3-b]pyridine 2-(3-methoxyphenoxy)-N'-(2,4,6-trichlorophenyl)acetohydrazide 3-(2,3-dihydro-1H-pyrrolo[3,4-c]pyridin-7-ylmethyl)benzaldehyde 1-(4,6-dimethylpyrimidin-5-yl)-3-[[2-fluoro-4-(trifluoromethoxy)phenyl]methylamino]propan-2-ol (1R,3S)-3-[[4-(2-methyl-6-pyrimidin-5-ylindazol-4-yl)pyridin-2-yl]amino]cyclohexane-1-carboxylic acid 3-ethyl-2-[(2Z)-2-hydroxyimino-2-[5-methoxycarbonyl-1-methyl-4-oxo-6-(trifluoromethyl)pyridin-2-yl]ethyl]butanoic acid 3-(aminomethylidene)-4,5,7-trihydroxychromene-2-thione;ethane 2-[3-(5-bromopyridine-2-carbonyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-2-yl]acetic acid 4-[6-chloro-2-(2,4,6-trifluorophenyl)pyrimidin-4-yl]-N-ethylbenzenesulfonamide 1-(4-ethoxyphenyl)-3,5,6,7-tetrahydrocyclopenta[d]pyrimidine-2,4-dione N-(4-methoxyphenyl)-2-(1,6,8-trimethyl-3-oxoimidazo[5,1-c][1,4]thiazin-1-yl)acetamide 4-methylsulfonyloxybenzenesulfonic acid (4-methylsulfonylphenyl)-[(3R,5S)-3-pyridin-2-yloxy-1-oxa-9-azaspiro[4.5]decan-9-yl]methanone 1-[4-(2,3-dihydro-1H-isoindole-5-carbonyl)morpholin-2-yl]-N-methylmethanesulfonamide 2-[4-fluoro-6-(hydroxymethyl)pyridin-3-yl]acetamide 7-methyl-N-[1-(oxan-4-yl)ethylidene]pyrazolo[5,1-b][1,3]benzothiazole-2-carboxamide N-(2,4,5-trihydroxyphenyl)benzamide 3-(2,3-dihydro-1H-indene-5-carbonylamino)-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylic acid 4-[5-cyano-6-(4,4,4-trifluorobutyl)naphthalen-2-yl]sulfonyl-3-methylpiperazine-1-carboxylic acid 3-(2-propan-2-ylphenyl)imidazolidine-1-carboxamide 1-[(6E)-6-ethylidene-2-methylpiperidin-3-yl]pyrazolo[4,3-c]pyridine 1-(6-azidohexyl)triazolo[4,5-b]pyridine 2,3-dimethylspiro[5,7-dihydropyrazolo[4,3-b]pyridine-6,1'-cyclopropane]-4-one 1-[(2,5-dimethylphenyl)methylamino]-3-propan-2-ylurea ethane;N-(4,6,7,8-tetrahydrothieno[3,2-c]oxepin-5-ylmethyl)propanamide 2-cyclopropyl-1,3,4,5-tetrahydropyrido[4,3-b]indole N-(4-methylphenyl)sulfanyl-6-oxoheptanamide 5-azidooxy-4-methylsulfanylbenzene-1,3-dicarbonitrile 3-(4-chlorophenyl)-2,2,5-trimethylheptanamide [(3R,4S)-1-tert-butyl-4-[3-chloro-5-fluoro-2-[[6-fluoro-2-methoxy-8-(trifluoromethyl)quinazolin-4-yl]amino]phenyl]piperidin-3-yl]carbamic acid 3-azidooxy-5,6-dimethylpyridine-2-carboxylic acid 5-(4-bromophenoxy)-1-[3,5-dichloro-2-hydroxy-6-(trifluoromethyl)phenyl]pentan-1-one 1-[6-amino-5-(1,3,4-thiadiazol-2-yl)pyridin-2-yl]-6-(2-methoxyethoxy)pyrazolo[3,4-b]pyridine-4-carboxamide 3-(4,7,10-triazaspiro[5.6]dodecan-11-yl)benzoic acid 4-[2-(2,3-dihydro-1H-inden-5-yl)ethynyl]pyridine 2-[1-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-4-cyclohexyl-2-ethyl-6-oxopyrimidine-5-carbonyl]-3-hydroxybenzoic acid 2-amino-4,6-ditert-butyl-8,9-dimethoxypyrimido[5,4-c]azepine-5,7-dione 2-ethyl-7,7-dimethyl-5H-[1,3]thiazolo[4,5-c]pyridine;N-ethynyl-6-phenylpyridazin-3-amine 6-(4,5-dihydro-1H-imidazol-2-yl)-N-piperidin-3-ylquinoline-4-carboxamide N-methyl-4,6,8,10-tetrahydro-3H-imidazo[1,2-a]azocine-7-carboxamide;hydrochloride N-[2-chloro-4-[1-(2,3-dihydro-1H-pyrrole-5-carbonyl)piperidin-4-yl]phenyl]acetamide 1-[4-[5-(cyclopropylmethoxy)pyrazine-2-carbonyl]piperazin-1-yl]ethanone 2-(2,3,5,6-tetrafluorophenoxy)benzenesulfonic acid N-[4-[4-(cyclohexylcarbamoylsulfamoyl)phenyl]-3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl]benzamide (NZ)-N-[1-[3-fluoro-2-(trifluoromethyl)phenyl]ethylidene]hydroxylamine 2-(4-hydroxy-3,5-dimethoxyphenyl)-N-[2-[2-hydroxy-5-[1-(4-pentylanilino)ethenyl]phenyl]ethyl]acetamide 6,7-dimethoxy-4-(3-nitrophenyl)sulfonylquinoline ethane;N-[3-(1H-indol-4-yl)phenyl]-2-methylpyrazole-3-carboxamide 2-amino-1,5-dimethyl-3H-pyrrolo[2,3-d]pyrimidine-4-thione N-[5-[3-(7-pyridin-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-2H-pyrazolo[3,4-b]pyridin-5-yl]pyridin-3-yl]cyclopentanecarboxamide 2-amino-6-methyl-1,4-bis[(2-nitrophenyl)methylidene]naphthalene-2-carboxylic acid 1-(4,7-dimethoxynaphthalen-2-yl)ethanone 2-(azidomethyl)-3,4,5-trifluoro-6-phenylaniline 5-(methoxymethyl)-1-[2-[(E,3Z)-4-methylidenehepta-1,3,6-trienyl]phenyl]tetrazole N-[1-(4-aminophenyl)propyl]-2,2-dichloro-3-(3,5-dichlorophenyl)cyclopropane-1-carboxamide 1-[(3,5-dimethylphenyl)methylamino]-3-naphthalen-2-ylthiourea 2-[4-[(7S)-4,8-dimethyl-6,7-dihydro-5H-pyrido[3,4-d]pyrimidine-2-carbonyl]phenoxy]-N-phenylacetamide (3Z)-5-methoxyhexa-1,3,5-triene;2-[1-(4-phenoxyanilino)propan-2-yl]guanidine 1-(2,2-difluoroethyl)-3-[4-(4-oxo-2,3-dihydro-[1]benzofuro[2,3-d]pyrimidin-8-yl)pyrazol-1-yl]azetidine-3-carbonitrile 5-(3,5-dimethyltriazol-4-yl)pyridine-2-carboxamide 2-[N-(1,3-thiazol-5-yl)anilino]octanoic acid 1-[3-(3,4-difluorophenoxy)-2-hydroxypropyl]-2-phenylpiperidine-2-carboxylic acid 1-[(2S)-4,6-diaminohexan-2-yl]oxycarbonylbenzotriazole-5-carboxylic acid;hydrochloride 4-[5-[6-(2,5-dimethoxyphenyl)pyridazin-3-yl]oxypentyl]morpholine 3-(4,6-dimethoxypyrimidin-2-yl)cyclohexa-1,5-diene-1-carboxamide (3R)-1-azidooxy-2,6-ditert-butyl-3-propan-2-ylbenzene 4-[3-(2,3-dihydro-1H-indole-6-carbonyl)phenyl]-1H-pyrimidin-6-one 5-[[4,6-bis(ethenyl)-1H-pyrimidin-2-ylidene]amino]pyridin-2-amine 1-(4,5-dichloro-2-hydroxyphenyl)-3-[2-methoxy-4-(trifluoromethyl)phenoxy]propan-2-one (4Z)-2,5-bis[(6-nitronaphthalen-1-yl)methyl]-4-[(3-nitrophenyl)methylidene]-1H-imidazol-5-one 5-(1,3-benzoxazol-2-yl)-4-N-(4-fluorophenyl)pyrimidine-4,6-diamine;methanol (5R)-3,9-diazaspiro[4.5]decan-8-ol;1-[2-fluoro-4-(trifluoromethyl)phenyl]-2,2,2-trifluoroethanone 3-cyclohexyl-5-[4-(trifluoromethoxy)phenyl]pyridine 3-N,5-N-bis(2-hydroxyethyl)benzene-1,3,5-tricarboxamide (5R)-2-[3-fluoro-4-(trifluoromethyl)phenyl]-8,8-dimethyl-N-[(1R,6S)-2,2,6-trimethylcyclohexyl]-5,7,9,10-tetrahydro-3H-pyrimido[4,5-b]quinoline-4-carboxamide N-[4-(difluoromethyl)phenyl]-4,5-dihydro-1H-imidazole-2-carboxamide (1-azidooxy-2,3,4,5,6-pentachlorophenoxy)benzene 1-azidooxy-2-tert-butylperoxy-4,6-dimethylbenzene 7-tert-butyl-5-(4-nitrophenyl)pyrrolo[2,3-b]pyrazine (5R)-2-cyclopentylimino-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 4-[3,5-bis(trifluoromethyl)phenyl]oxan-2-ol 6,6-dimethyl-2-(4-nitrophenyl)cyclohexa-1,3-diene-1-carboxylic acid 2-(6-methoxy-1H-benzimidazol-2-yl)aniline 1-(4,6-dimethylpyridin-3-yl)sulfonyl-N-[2-(methylamino)ethyl]piperidine-4-carboxamide;hydrochloride 6-chloro-4-[5-(difluoromethyl)pyridin-2-yl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 6-N-(2,3-dimethylphenyl)-4-N-(1-propanoylpiperidin-4-yl)pyrimidine-4,6-dicarboxamide (2R)-N-[[3,5-dimethoxy-4-[6-[5-methyl-1-(pyridin-3-ylmethyl)pyrazol-4-yl]pyrrolo[2,1-f][1,2,4]triazin-4-yl]oxyphenyl]carbamothioyl]-2,3-dihydroxypropanamide (2R,3aS,7aR)-6-[(4-methylphenyl)methyl]-N-pyrazin-2-yl-3,3a,4,5,7,7a-hexahydro-2H-furo[2,3-c]pyridine-2-carboxamide;2,2,2-trifluoroacetic acid 6-(4-phenylphenyl)cyclohexa-2,4-dien-1-imine 2-[4-(benzylamino)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-c]azepin-2-yl]phenol 1-[2-ethyl-4-(5-fluoropyridin-3-yl)phenyl]-N-methoxy-3H-pyrazole-2-carboxamide [3,4-difluoro-2-(2H-tetrazol-5-yl)phenyl]hydrazine N-[(2,4-dimethoxyphenyl)methyl]spiro[1,3-dihydroisoquinoline-4,1'-cyclopropane]-2-imine 4-[(1S)-3-methylcyclopentanecarbonyl]-6,7,8,9-tetrahydrothieno[2,3-c]isoquinolin-5-one N-[3-(difluoromethoxy)phenyl]-2-[4-oxo-5-[(4-propan-2-ylpiperidin-1-yl)methyl]quinazolin-3-yl]acetamide 2-[6-(benzylamino)pyridin-3-yl]-1,7-dihydropurin-6-one 3-(5-ethylsulfanylpyridin-2-yl)sulfanylbenzonitrile N-[4-[2-[(1-methylpyrrolidin-3-ylidene)amino]phenyl]phenyl]-2,6-di(propan-2-yl)aniline 2,6-dichloro-N-[(4S)-6-fluoro-7-(2-hydroxy-4,4-dimethylpentoxy)-4-phenyl-1,3-benzothiazol-2-yl]benzamide 2,2-difluoropropane;3,4-dimethoxy-N'-[(1E)-1-[2-[(1E,3Z)-5-(methylaminomethyl)penta-1,3-dienyl]anilino]buta-1,3-dien-2-yl]benzenecarboximidamide 1-[4-[2-(3,5-dichlorophenyl)ethyl]piperazin-1-yl]ethanone 2-cyclopropyl-6-[(3-ethoxyphenyl)methyl]-5-fluoropyrimidine 1-(2,3-dihydro-1H-inden-1-yl)-N-propan-2-ylpyrazole-4-sulfonamide N-ethyl-4,5-dimethoxy-2-phenylmethoxybenzenesulfinamide N-azido-2-methyl-4,5-dinitrobenzamide 2-fluoro-N-[4-[[6-(2,3,5-trimethylpyrrol-1-yl)pyridine-3-carbonyl]amino]phenyl]acetamide (5S)-3-amino-7,10-dioxo-1,4,7,12-tetrazatricyclo[6.4.0.02,6]dodeca-8,9,11-triene-9-carboxylic acid N-[(3-cyclohexyloxy-5-hydroxyphenyl)methylideneamino]-1,2-benzothiazole-3-carboxamide N-(cyclopropylmethoxy)-4-fluoro-2,3-dihydro-1H-indene-5-carboxamide N'-hydroxy-5,6-dimethyl-3-(2-methylpiperidin-1-yl)pyridazine-4-carboximidamide N-[5-[4-fluoro-3-(7-thiophen-2-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclopentanecarboxamide (2S)-1-[1-(2,4-dimethoxyphenyl)ethyl]pyrrolidine-2-carboxamide 3,5-dimethylbenzenethiol;6-(4-hydroxyphenyl)-N,N,2,4,8-pentamethylnonanamide N-(2-bromopyridin-4-yl)sulfonyl-3,5-dimethoxybenzamide N-[3-(benzenesulfonyl)-2,4-dichlorophenyl]-7-methylsulfonylisoquinoline-1-carboxamide 1-[3-chloro-4-(1,2,3,6-tetrahydropyridine-2-carbonyl)phenyl]propan-1-one 3-[6-methyl-5-(2-morpholin-4-ylethoxy)indazol-1-yl]propan-1-ol 4-azido-2-(3,4-difluorophenyl)aniline 3-(1,1-dioxothiazinan-2-yl)-7-methoxy-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine 5-[(2S)-1-azido-4,4-dimethylpentan-2-yl]-2H-tetrazole 1-[2-(6,7-dimethoxyquinazolin-4-yl)sulfanylethyl]cyclopentane-1-carboxylic acid 2-[(2E,4Z)-5-ethenylsulfanyl-3-methylidenepenta-1,4-dien-2-yl]oxypyridine 1-methoxy-4-[3,4,5-tris(trifluoromethyl)phenoxy]benzene N-[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]-6-[(Z)-1,5-diiminopent-2-en-2-yl]quinazolin-4-amine N-[4,4-difluoro-2-(hydroxymethyl)butan-2-yl]-3-ethoxybenzamide (1-methoxyisoquinolin-6-yl)-[3-(trifluoromethyl)piperidin-1-yl]methanone N-azido-5,6-bis(phenylmethoxy)pyridine-3-carboxamide 2-(4-chlorophenyl)-3,7-dimethylquinoline N-[(4-phenylmethoxy-6,7-dihydro-5H-[1]benzoxepino[5,4-d]pyrimidin-2-yl)amino]pyridine-3-carboxamide N-(2,6-dimethylphenyl)-4-[(3S)-1-methylpiperidin-3-yl]oxypyridine-2-carboxamide 2-(difluoromethyl)-5-[3-methoxy-4-(trideuteriomethoxy)phenyl]sulfonylpyridine 1-(2-phenylphenoxy)-4,5,6,7-tetrahydro-2H-benzotriazole N-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]-6,8-difluoro-1H-indole-2-carboxamide;N-methylethanamine N-[(1S)-1-(4-aminosulfanylphenyl)ethyl]-3-(4-methoxycyclohexa-2,4-dien-1-ylidene)propanamide (2R)-N-[[5-chloro-4-[[3-fluoro-1-methyl-6-[3-[(3S,5R)-1-methylpiperidin-3-yl]propanoyl]indol-7-yl]amino]pyrimidin-2-yl]methyl]oxane-2-carboxamide 1-(2,4-difluorophenyl)-N-[1-(5-fluoropyridin-3-yl)ethoxy]methanimine 3-(8-azido-7-methoxyquinolin-4-yl)benzonitrile 1-[(2R)-1,1,1-trifluoropropan-2-yl]oxyisoquinoline 3-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-N-[(4-ethylsulfanylphenyl)methyl]-N-propan-2-ylbenzamide 4-[4-amino-7-methyl-6-[4-(pyrrolidin-1-ylmethyl)phenyl]pyrrolo[2,3-d]pyrimidin-5-yl]-N-(2-hydroxyethyl)benzamide 4-[3-(2,5-dioxopyrrolidin-1-yl)-5-fluoroquinolin-8-yl]benzoate 2-(3,4-dichlorophenoxy)-N-[5-(furan-2-ylmethoxymethyl)cyclohexa-1,5-dien-1-yl]propanamide (6E)-1,3-dimethyl-8,9-diphenylnona-2,6,8-trien-4-one 2-[7,8-dideuterio-3,6-bis(trifluoromethyl)-9H-pyrazolo[4,3-h]quinolin-5-yl]phenol (2S,6R)-4-[(3S)-4-amino-3-fluorobutyl]-N-methoxy-7-oxo-1-phenyl-2,5-dihydro-1H-pyrrolo[3,2-b]azepine-3-carboxamide 3-chloro-6,7-dimethyl-2H-pyrazolo[4,3-g]quinoline 2-(4-aminopiperidine-1-carbonyl)-5,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-4-one 2-(N-(4-bromophenyl)anilino)acetic acid 2-[(6S,9R)-6-(3,4-dimethoxyphenyl)-8-oxo-5,6,7,9-tetrahydro-4H-[1,2]oxazolo[5,4-b]quinolin-9-yl]benzoic acid 4-[(Z)-2-(furan-3-yl)ethenyl]phenol 2-(N-hexadecyl-4-sulfoanilino)acetic acid 4-methyl-2,5-dinitro-N'-phenylbenzenecarboximidamide 5-chloro-4-[6-chloro-7-fluoro-2,3-dimethyl-1-(2-methylpropanoyl)pyrrolo[3,2-b]pyridin-5-yl]oxy-2-fluoro-N-methylsulfanylbenzamide N-[5,6-dimethyl-3-(trifluoromethyl)pyridin-2-yl]-1H-pyrrole-3-carboxamide;ethane 1-[(2,4-dimethoxyphenyl)methylamino]-3-[(2,5-dimethylphenoxy)methyl]urea 1-[4-(6-ethyl-5,8-dioxopyrimido[4,5-d]pyridazin-2-yl)morpholin-3-yl]-3H-imidazo[4,5-b]pyridin-2-one 4-(5,6,7,8-tetrahydroisoquinolin-3-yloxy)benzenecarboximidamide N-[4-(1,3,4-oxadiazole-2-carbonylamino)butyl]-5-pyrrolidin-1-ylsulfonylthiophene-2-carboxamide N-(5-bromonaphthalen-1-yl)sulfanylcyclohexanecarboxamide 5-[3-(hydroxymethyl)-3,4-dihydropyridin-6-yl]-N,2-dimethylaniline 4-[7,10-dimethyl-9-(3-methylbutoxy)-5,6-dihydrobenzo[h]quinazolin-2-yl]phenol N-(3,5-dichlorophenyl)-2-[4-(2-hydroxypropyl)-2-oxopiperazin-1-yl]acetamide [(2R,3S)-1-cyclopropyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]methanesulfonic acid 4-(3,3-dimethylbutanoylamino)naphthalene-1-sulfonic acid 2-[(2R)-4-ethylpiperidin-2-yl]-6-methoxy-1H-benzimidazole 4-(1,3-benzodioxol-5-yl)-7-[5-chloro-2-[2-methylpropyl(propanoyl)amino]phenyl]thieno[3,2-c]pyridine-2-carboxylic acid 1-(2,2-dimethylpropanoyl)-3-[5-methoxy-8-methylidene-6-[4-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]benzo[f]quinoxalin-7-ium-1-yl]urea (2R,3S)-2-azido-5-[2-(4-fluorophenyl)piperazin-1-yl]-1-(2-propan-2-yloxyanilino)pentane-3-thiol N-(1-methylimidazol-4-yl)-2,3-dihydrothieno[3,4-b][1,4]dioxine-5-carboxamide 2-(3,5-dichloro-N-ethylanilino)decanoic acid 3-(2,5-diphenyl-1H-pyrrol-3-yl)aniline 7-[4-(trifluoromethyl)phenyl]heptanoic acid N-[(Z)-3,5-dihydroxypent-2-enyl]-2-[5-(4-methylsulfanylphenyl)furan-2-yl]acetamide 2-[1-[[(E)-3-aminobut-2-enoyl]amino]ethylamino]-6-bromopyridine-4-carboxamide (E)-3-[4-[2-chloro-4-[(Z,1Z)-1-ethylideneamino]anilino]thieno[3,2-d]pyrimidin-6-yl]-N-methoxyprop-2-enamide [7-amino-5-(2,6-dimethylpyridine-4-carboximidoyl)pyrazolo[1,5-a]pyrimidin-3-yl]-(azetidin-1-ium-1-ylidene)azanium 2-N-(1,3-dimethylindazol-5-yl)-7H-purine-2,8-diamine 4-tert-butyl-N-[1,3-difluoro-2-[4-(trifluoromethoxy)phenyl]propan-2-yl]benzamide 5-(6-methylpyridine-2-carbonyl)-N'-propanoyl-3,4,6,7,8,9-hexahydropyrido[1,2-a]pyrazine-2-carbohydrazide 2-[(3,4-dimethoxyphenyl)methyl]-7-fluoro-3-propanoyl-1-benzofuran-5-carbonitrile 2-[(2,6-dibromopyridin-4-yl)-pyridin-3-ylamino]acetonitrile (2S,3R)-5-[3-chloro-4-(trifluoromethylsulfanyl)phenyl]-1,3-diethyl-2-phenylpyrrolidine 1-(2-methylsulfanyl-4,6-dinitrophenyl)-4-sulfamoylpiperazine 2-(1,5-dihydroxybenzimidazol-2-yl)oxyacetic acid N-(4-azidophenyl)-2-oxopropanamide N'-[2,3-dichloro-4-(3-fluorophenyl)sulfanylthieno[3,2-b]pyridin-7-yl]-N-ethylbutane-1,4-diamine;N-methoxyhydroxylamine 3-[4,5-bis(ethenyl)-2-propan-2-ylidenepyridin-1-yl]-1,6-dimethoxyisoquinoline 2-methylsulfonyl-7H-pyrrolo[2,3-d]pyrimidine 2-(2-hydroxyethoxy)-4,6-dimethylphenol (5S)-5-[(2,3-dimethylquinolin-6-yl)oxymethyl]pyrrolidin-3-ol (E)-1-[4-hydroxy-2,3-dimethoxy-5-[(2R)-2-methylpentoxy]phenyl]-3-(4-hydroxy-3-nitrophenyl)prop-2-en-1-one 2-ethyl-N-(3-phenylbutyl)pyrrolidine-1-carboxamide N-(1-azido-2,4-dioxospiro[3H-chromene-5,4'-piperidine]-6-yl)-2-(4-methoxyphenoxy)acetamide 2-(4,4-dimethyl-1H-quinolin-3-yl)acetate 4-[(2-hydroxy-5-nitrophenyl)iminomethyl]-2,6-diiodophenol 2-[5-(5,6,7,8-tetrahydroquinolin-4-yl)-1H-pyrazol-3-yl]benzamide (E)-1-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-2-yl)-N-ethoxy-1-phenylmethanimine 1-[2-(5,6-dimethoxybenzimidazol-1-yl)ethyl]-3-nitrosoindol-2-ol 6-[3-(2,5-dimethylphenyl)azetidine-1-carbonyl]-4H-chromen-2-one 5-[2-(cyclohexylamino)-1,3-thiazol-4-yl]-7-fluoro-8-(methylamino)naphthalene-2-sulfonic acid 3-chloro-4-[(3E)-hexa-1,3,5-trien-3-yl]oxyphenol N-[(2E,4Z)-3-cyclohepta-1,4,6-trien-1-ylhepta-2,4,6-trienyl]sulfanyl-4-methoxyaniline 1-(4,5-diphenyl-1H-pyrrol-2-yl)ethanone 2-[1-cyclohexyl-3-hydroxy-5-(6-methoxyquinolin-4-yl)pentan-3-yl]benzoic acid 3-bromo-2,5-diphenylthieno[3,4-b]pyridine 3-(5,6-dihydronaphthalen-1-yl)propanenitrile;ethane N-(1-azidopropan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide 2-[3-(5-aminopyridin-3-yl)phenyl]acetic acid 3-[(4S)-2,2-dimethyloxan-4-yl]-6-fluoroimidazo[1,5-a]pyridine 6-methyl-5,10,17-trioxapentacyclo[11.8.0.03,11.04,9.014,19]henicosa-1(13),2,4(9),7,11,15,18,20-octaene 3-[4,6-bis(1H-indol-2-yl)-1,5-dihydropyrimidin-2-yl]-2-(4-chlorophenyl)-1H-indole N-[(E)-1-amino-3-hydroxy-5,5-dimethylhex-2-enylidene]-6-[4-(cyclopropanecarbonyl)piperazin-1-yl]pyridine-3-carboxamide;butane 4-bromo-6,8,9,10-tetrahydro-[1]benzoxepino[3,2-d]pyrimidine 2-amino-1-[4-(1H-imidazol-5-ylmethyl)piperazin-1-yl]propan-1-one;trihydrochloride [3-amino-4-(1,1,1-trifluoropropan-2-yloxy)phenyl]methylidenehydrazine 3-(4-methylphenyl)-1,3,3a,9b-tetrahydrodibenzofuran (Z)-2,3-bis[(4-hydroxy-3,5-dimethoxyphenyl)methyl]but-2-enedioic acid (E)-N'-hydroxy-3-[4-[2-(3-methylbutylamino)-1,3-thiazol-5-yl]phenyl]prop-2-enimidamide 4-(N-cyclohexyl-3-nitroanilino)butan-1-ol (E)-N-[2-(3,4-dichlorophenyl)-3-pyrrolidin-1-ylpropyl]heptanamide 1-[2,3-bis(ethenyl)phenoxy]-3,4,5,6-tetrachlorocyclohepta-1,3,5-triene 7-(6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazine-7-carbonyl)-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one 2-(4,5-dichloroimidazol-1-yl)-N-[3-(N'-methanimidoylcarbamimidoyl)phenyl]acetamide 6-[[6-(4-bromophenyl)pyridazin-3-yl]amino]-2-(oxolan-2-ylmethylamino)benzonitrile N-(2-cyanoethyl)-2-[1'-(thiophene-3-carbonyl)spiro[4,7-dihydrotriazolo[5,1-c][1,4]oxazine-6,4'-piperidine]-3-yl]acetamide (5Z)-2-[3,4-bis(ethenyl)phenyl]imino-5-[[3-iodo-1-methyl-4-[(4-nitrophenyl)diazenyl]pyrrol-2-yl]methylidene]-1,3-thiazolidin-4-one [4-[(3R)-3-(1H-benzimidazol-2-ylmethoxycarbonylamino)pyrrolidin-1-yl]phenyl]carbamic acid 2-(3-carbamimidoylphenyl)-1,3-dioxoisoindole-5-carboxylic acid 2-[(3,4-dichlorophenyl)methylsulfanyl]-6-(5H-imidazo[5,1-a]isoindol-5-ylamino)pyrimidine-4-carboxylic acid ethane;4-[2-(3-hydroxy-5,7-dimethylindol-1-yl)ethyl]benzaldehyde 5-chloro-6-ethoxycarbonylimidazo[1,2-a]pyridine-7-carboxylic acid 1-[3-[7-(3,5-dimethyl-2H-indazole-6-carbonyl)-9-hydroxy-7,8-dihydro-6H-pyrido[4,3-a]pyrrolizin-5-yl]phenyl]pyrrolidine-2-carboxylic acid N-(3,4-difluorophenyl)-N-[2-(cyclopentylamino)-2-oxo-1-pyridin-3-ylethyl]-5-(methanesulfonamido)-3a,6a-dihydro-1H-pyrrolo[3,2-b]pyrrole-2-carboxamide 7-[[(1R,3S)-3-aminocyclopentyl]methoxy]-2-hydroxy-4H-isoquinoline-1,3-dione;hydrochloride (Z)-N-[3-(2,6-dimethoxyphenyl)imino-1-ethyl-4-hydroxyquinoxalin-2-ylidene]-1,2-diphenylethenamine N-[3-[(1Z)-buta-1,3-dienyl]-2-methylphenyl]-6-(4-chlorophenyl)sulfanylhex-5-ynamide;ethane 4-(6,7-dihydro-1H-indole-3-carbonyl)-N-methylpiperazine-2-carboxamide;N-[3-fluoro-5-(2,2,2-trifluoroethoxy)phenyl]formamide (2E,3Z)-N-[2-(5-cyanopyridin-2-yl)ethoxy]-4-methylidene-1-pyrrolidin-1-ylhepta-2,5-dien-2-amine ethane;2-[3-methoxy-4-(2-phenylethynyl)phenyl]propanoic acid 2-amino-1',3-dimethylspiro[fluorene-9,3'-indole]-2'-one (2S)-6-amino-1',1',1',4,5-pentamethyl-3,3a,9b-tetrahydro-2H-pyrrolo[3,2-b]indole-2-carboxylic acid 4-[6-azidooxy-2,3-bis(propan-2-ylamino)phenyl]-2-fluorobenzonitrile (1R)-3-[[2-[5-(furan-2-ylmethylamino)-1,3,4-thiadiazol-2-yl]acetyl]amino]cyclopentane-1-carboxylic acid 1-[(3-chlorophenyl)methyl]-7-nitroindole 3-[3-oxo-7-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonylamino)-1H-isoindol-2-yl]piperidine-1-carboxamide 1-[5-(3,4-dichlorophenyl)pentyl]pyrrolidine;ethane;(4E)-4-ethylidenenona-2,5-diene (E,3S)-2-ethenyl-N'-[3-methoxy-4-(1,3-thiazol-5-yl)phenyl]-3-[1-(methylideneamino)ethenylamino]hex-4-enehydrazide 5-[(3,6-dimethylpyridine-2-carbonyl)amino]-2,4-difluorobenzoic acid 2-[3,5-dichloro-4-[(6-oxo-1-propylpyridazine-3-carbonyl)amino]phenyl]acetic acid (3-chloropyrazin-2-yl)-[4-hydroxy-4-[methoxy(diphenyl)methyl]piperidin-1-yl]methanone (1R)-N-[5,6-bis(ethenyl)pyridin-2-yl]-2-cyclohexa-1,3-dien-1-yl-N-(4-iodophenyl)sulfonylacetamide 1-N',3-N',2-triethyl-1-N',3-N'-dimethylbutanedihydrazide;2-[(5R)-3,7,13-trimethoxy-4-oxo-9-oxa-6-thiatetracyclo[10.2.1.05,14.08,12]pentadeca-1,3,5,7,10,12,14-heptaen-5-yl]acetonitrile 4-[4,6-di(propan-2-yl)pyrimidin-5-yl]oxypyrrolidine-2-carboxylic acid;ethane 5-tert-butyl-4-chloro-2,6-bis(2-methylpropyl)pyrimidine N-(7,7-dimethylcyclohepta[b]pyridin-4-ylidene)hydroxylamine N-(1,2,3,5,6,7-hexahydropyrrolizin-8-ylideneamino)aniline 3-methyl-6-(4-pyridin-2-yloxyphenyl)pyrazine-2-carboxamide 3-[1-(2,6-dimethylpyridine-4-carbonyl)piperidin-2-yl]propanoic acid 2-[4-(2,3-dichlorophenyl)sulfanylpiperazin-1-yl]pyridine-3-carboxamide (1S)-4-[2-azido-6-chloro-3-fluorophenyl]-1-propan-2-yloxybutane-1,3-diol 4-cyclohexyl-2-(methylamino)-5,6,7,8-tetrahydropteridine-6-carboxamide;N-propan-2-yl-1,3-thiazol-2-amine 4-[(6-bromopyridin-2-yl)methoxy]-N-hydroxybenzenecarboximidate 2-azidosulfanyl-5-ethoxypyrimidine (3-aminothiophen-2-yl)-[1,4-diphenylbutyl(methoxycarbonyl)amino]carbamic acid 3-azidooxy-7-[2-(5-fluoropyridin-3-yl)ethynyl]-8a-methyl-6,8-dihydropyrrolo[1,2-a]pyrazine 2-[(5,6-dichlorobenzimidazol-1-yl)methyl]-3H-quinazolin-4-one 1-(2,5-dichlorophenyl)-2-[4-(4-pyridin-4-ylpiperazine-1-carbonyl)phenyl]ethanone;hydrochloride 2-[4-bromo-N-(1,3-thiazol-5-yl)anilino]guanidine 1-(2-methylpyrazol-3-yl)-3-[1-(4-morpholin-4-ylbenzoyl)azetidin-3-yl]urea 4-[2,3-dihydroxypropyl(1,2,4-triazol-4-yl)amino]-N-thiophen-2-ylbenzenesulfonamide 5-N-[(2R)-1-[4-chloro-3-(trifluoromethyl)phenyl]propan-2-yl]-3-N-cyclopentyl-3-N,6-dimethoxypyrazine-2,3,5-tricarboxamide 2-[1-(3-acetylphenyl)piperidin-4-ylidene]propanenitrile N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6-[(E)-2-(furan-2-yl)ethenyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-amine 2-[4-(cyclohexylamino)piperidine-1-carbonyl]-6,7-dihydro-5H-cyclopenta[b]pyridine-4-carboxamide 1-[3-(2,6-dichloro-4-methylphenyl)sulfanylpropyl]piperazine 4-[(3-chlorophenyl)methyl]-2,2-dioxo-1H-1,3,5-triazin-6-one N-[2-[2-[[(E)-1-aminopent-2-enylidene]amino]propyl]phenyl]-5-fluoropyridine-3-carboxamide 1-[3-methylbut-2-enyl(pyridin-2-yl)amino]propan-2-one 3-(5-methylfuran-2-yl)-4,7,8,9-tetrahydropyrazolo[1,5-a]quinazolin-5-one 4-[4-(3-amino-1H-indazole-6-carbonyl)piperazin-1-yl]benzonitrile (5R,7S)-N-(2-chlorophenyl)-5-(4-methylphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide N-[3-(aminomethyl)phenyl]-6-hydroxy-2,4-dioxo-1H-pyrimidine-5-carboxamide 2-[5-(3,4-dimethylphenyl)heptanoylamino]benzoic acid 4-[6-[2-(5-fluoro-1H-indol-3-yl)ethylamino]pyridine-2-carbonyl]piperidine-1-carboxylate 4-[3-hydroxy-5-(2H-tetrazol-5-yl)phenoxy]butanoic acid 2-(5-ethyl-1,3-thiazol-2-yl)-N-[4-fluoro-5-(6-morpholin-4-ylpyridin-3-yl)-2H-indazol-3-yl]acetamide (4aS,7R)-6-methoxy-3a-methyl-N-[(1S)-1-phenylethyl]-4,5,7,8-tetrahydrothieno[2,3-d]azepine-7-carboxamide 4-[(2-chlorophenyl)methylsulfanyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine N-[(2R,3S)-3-methyl-1-methylidenethiiran-2-yl]-4-[5-(trifluoromethyl)pyrimidin-2-yl]-1,4-diazepane-1-carboxamide N-butyl-6-chloroimidazo[4,5-c]pyridin-3-amine [(3R,4R)-1-ethyl-2-oxo-4-phenylpyrrolidin-3-yl]carbamic acid 1-methyl-2-nitro-6H-phenanthridine 6-benzylsulfanyl-3-propyl-2,5-dihydropyrazolo[3,4-d]pyrimidin-4-one 6-azido-2,3-difluorobenzenesulfonic acid 1-methyl-N-[(4-nitrophenyl)methyl]-N-octylpiperidin-3-amine 7-tert-butyl-1,2,3,4,5-pentamethylpyrrolo[1,2-a]quinoxaline (5Z)-2-cyclopentylimino-5-[(2,3-difluorophenyl)methylidene]-1,3-thiazolidin-4-one N-[3-(6-aminopyridin-1-ium-3-yl)phenyl]sulfonylacetamide 5-(chloromethyl)-1,4-diethoxypyrazole 2-[3,4-bis(propylperoxy)phenyl]ethanamine 2-(2,4-dimethylphenyl)imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one 2-[(3S,4R)-1-tert-butyl-3-(cyclopropylmethoxymethyl)piperidin-4-yl]benzonitrile 2-(9H-fluoren-1-yl)-4-phenylbenzenethiol 5-(6-chloro-1H-indazol-3-yl)-2,4-difluorophenol 2-amino-6-(4-hexyl-2-hydroxyphenyl)phenol 5-[3-(trifluoromethyl)phenyl]pentan-1-amine (4S)-4-benzyl-N-[1-cyano-2-[(6-nitroquinoline-8-carbonyl)amino]ethyl]-N-methylpiperidine-3-carboxamide 2-[(1E,3Z)-1-amino-4-piperidin-1-ylhexa-1,3-dienyl]-N-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide 2-chloro-4-ethyl-6-phenylpyridine 1-(4,6-diethyl-2-methoxycyclohexa-1,5-dien-1-yl)-3-hydroxybutan-1-one 3-[[2-(2,6-dioxopiperidin-4-yl)-1H-triazol-1-ium-5-carbonyl]amino]benzamide 6-[5-(2,3-difluorophenyl)-1H-imidazol-2-yl]-4-[2-fluoro-4-(trifluoromethoxy)phenoxy]thieno[3,2-d]pyrimidine 4-(1,3-benzothiazol-2-yl)-N-[4-cyano-2-[4-[3-(dimethylamino)propanoyl]piperazin-1-yl]phenyl]-6-fluoro-2H-chromene-7-carboxamide N-methyl-2,3-dioxospiro[4H-quinoxaline-1,4'-piperidine]-7-carboxamide N-methyl-2,2-bis(3-nitrophenyl)ethanamine 4-[[6-(1,3-benzodioxol-5-yl)pyridin-2-yl]methylamino]-3-fluorobenzenesulfonamide 1-(3,4-dimethoxyphenyl)sulfonyl-3-[2-(1H-pyrrol-2-yl)ethyl]urea 1-[(2,3-dimethylpyridin-4-yl)amino]-N'-hydroxypyrazole-5-carboximidamide 2-[6-fluoro-5-(4-methylpyridin-3-yl)-1H-indazol-3-yl]-7-piperidin-1-yl-1H-imidazo[4,5-b]pyridine 3-(N-[3-chloro-4-(1H-pyrazol-4-yl)phenyl]anilino)propane-1,2-diol 5-amino-4-[2,6-dibromo-4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 4-N-ethenyl-1-N,4-N-bis(3-methylphenyl)benzene-1,4-diamine (E)-3,5-diaminopenta-2,4-dienal;N-[2-oxo-2-(5-phenylmethoxy-1H-indol-3-yl)ethyl]methanesulfonamide 6-hydroxy-N,5-dimethylcyclohexa-1,3-diene-1-carboxamide;(E)-3-[3-fluoro-4-(1H-indol-7-yloxy)phenyl]prop-2-enoic acid 1,3-dimethyl-7-[3-(trifluoromethyl)thiophen-2-yl]imidazo[4,5-b]pyridin-3-ium (5Z)-3-cyclobutyl-6-methylidene-4,8-dihydro-2H-benzo[f]quinolin-7-one (5-benzylsulfonylthiophen-2-yl)urea N-[2-(2,4-dimethylphenyl)ethenyl]-1-[2-hydroxy-3-[[(E)-[(Z)-hydrazinylidenehydrazinylidene]methyl]sulfanylamino]propoxy]naphthalene-2-carboxamide 7-[(2R)-5-ethenyloxolane-2-carbonyl]-2,3,5,6,8,9-hexahydropyrido[2,3-d]azepin-4-one 1-cyclopropyl-4-(dimethylamino)-3-ethylpyrazolo[3,4-b]pyridine-5-carboxamide N-[(6-amino-2,4-dimethylpyridin-3-yl)methyl]formamide;2-fluoro-5-hydroxy-1,2,3,4-tetrahydroisoquinoline 6-(2-azidoethyl)-N,N-bis[(4-methoxyphenyl)methyl]pyridine-3-carboxamide 4-bromo-6,8-difluoroquinoline-3,7-diamine 2-[4,5-bis(4-methoxyphenyl)thiophene-3-carbonyl]benzoic acid 3-[4-[2,6-dimethyl-4-(oxan-2-yloxy)anilino]-7-methoxyquinazolin-6-yl]but-1-en-2-ol 2-(azidooxymethyl)-1,4-dichlorobenzene 2-azido-5,8-dibromoquinoxaline (Z,2R)-1,4-bis(2-aminophenyl)but-3-en-2-amine 5-(1,2-diphenylhydrazinyl)furan-3-carboxylic acid 1-[4-[2-(5,6,7,8-tetrahydroquinolin-2-yloxy)ethyl]piperazin-1-yl]-2,3-dihydro-1H-indene-5-carbonitrile 2-(3,4-dichlorophenyl)-1-[7-methyl-5-(1H-pyrazol-4-yl)-2,3-dihydroindol-1-yl]ethanone [4-(1,1-dideuterioethyl)-6-[5-fluoro-2-(methoxymethyl)pyrimidin-4-yl]-3,8-dihydro-2H-pyrrolo[3,2-c]azepin-1-yl]-(1-propanoylpiperidin-4-yl)methanone 2-N,7-N-diphenylanthracene-1,2-disulfonamide 2-(2,3,4a,5,6,7,8,8a-octahydrobenzo[d][1]benzoxepin-11-yl)-3H-benzimidazole-5-carboximidamide N-[2,5-bis(trifluoromethyl)phenyl]sulfanyl-N-methylhydroxylamine;ethane 1-[2-(4-aminopiperidin-1-yl)-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-4-yl]-N-methylpyrrolidine-3-carboxamide;dihydrochloride (2S)-1,1,1-trifluoro-4-[2-fluoro-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]butan-2-amine N-[2,4-bis(phenylmethoxy)-5-propan-2-ylphenyl]-1,3-thiazole-2-sulfonamide 2-chloro-1-[4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl]ethanone 5-(4,6-dimethoxypyrimidin-2-yl)oxynaphthalene-1,7-disulfonic acid 1-methyl-N-(2,3,4-trihydroxyphenyl)cyclopentane-1-carboxamide 2-[(Z)-(7H-pyrrolo[2,3-d]pyrimidin-4-ylhydrazinylidene)methyl]phenol 5-[[4,6-bis(methylamino)-1,3,5-triazin-2-yl]amino]-2-ethoxyphenol 3-methylsulfanyl-6,6a,7,8,9,10-hexahydro-5H-benzo[b]carbazole-11-carboxylic acid 4-[(3R)-5-(4,4-difluorocyclohexyl)sulfanyl-3-methylpentyl]pyridine 2-[(2E,4Z)-5-(1H-indol-3-yl)penta-2,4-dienoxy]benzonitrile N-[5-[3-(4-piperidin-1-yl-1H-indol-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclohexanecarboxamide (E)-2,3,3-trimethyl-1-[4-methyl-3-(2-methylpropyl)phenyl]sulfanylbut-1-en-1-amine N-[3-methoxy-4,5-bis(phenylmethoxy)-6-(trifluoromethyl)pyridin-2-yl]-3-oxobutanamide N-[4-(2,3-difluorophenyl)sulfanylcyclohexyl]propane-1-sulfonamide N-[(3S,4R)-1-methylpiperidin-4-yl]-5-(2H-pyrrol-4-yloxy)pyridine-3-carboxamide;hydrochloride 4-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazole-3-carbonyl)-N-methylpiperazine-1-sulfonamide 1-[3,5-difluoro-4-(hydroxymethyl)phenyl]-N-(2-phenylethoxy)-2H-pyrrole-5-carboxamide 4-[(3S)-2-amino-5,6-dimethoxycarbonyl-7H-pyrrolo[1,2-b][1,2,4]triazol-3-yl]benzoic acid [4-(3,3-dimethylbut-1-ynyl)-2,6-difluorophenyl]-(pyridin-2-ylmethylideneamino)methanol N-methyl-2,6-dipyridin-4-yloxybenzamide 5-(4,6-dihydropyrrolo[3,2-c]pyrazole-1-carbonyl)benzenesulfonamide 1-[3-azidooxy-2,6-difluoro-5-(trifluoromethyl)phenyl]ethanone 4-(3,5-diaminophenyl)-3,6-bis(propyliminomethyl)benzene-1,2-diol N-butanoyl-2-hydroxy-4-(trifluoromethoxy)benzamide N-[5-bromo-2-(methylamino)phenyl]formamide ethane;1-(3,4,5-trifluorophenyl)piperidine N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-1,3-thiazol-2-amine (2E)-N-[(2R,4Z)-2,5-dihydroxypenta-2,4-dienyl]-2-[1-[4-ethoxy-3-(methylideneamino)phenyl]ethenylhydrazinylidene]butanamide N-(4-phenylbutyl)-6-[2-(phenylsulfamoylamino)ethoxy]hexanamide 2-(3,5-diethoxyphenyl)-N'-methylacetohydrazide 5-(1,3-benzothiazol-2-yl)-N-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]naphthalene-1-carboxamide [(3R)-4-azidopiperazin-1-yl]-(5,6-dichlorobenzimidazol-1-yl)methanone (6R)-2-amino-3,5,7-trimethyl-6-[(2,4,5-trifluorophenyl)methoxy]-1H-pyrido[3,4-e]indole-8-carbonitrile 5-(3,4-dichlorophenyl)-N-methylfuran-2-carboxamide 6-[(4-fluorophenyl)methyl]-1-[2,2,2-trifluoro-1-[2-methoxyethyl(methylsulfonyl)amino]ethyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one 3-hydroxy-2-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)heptanoic acid 5-amino-2-(2-chloropyridine-4-carbonyl)-3,3a,4,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrole-6-carboxylate (2R,3S)-4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfanyl-N-(1H-indazol-6-ylmethyl)-3-methoxy-1-[4-(4-methylphenyl)sulfonylpiperazine-1-carbonyl]pyrrolidine-2-carboxamide 2-[(4S,7R)-4-amino-3-fluoro-8-methyl-1-oxo-5,6-dihydropyrano[2,3-f]benzimidazol-2-ylidene]-N-pyridin-2-yl-3H-benzimidazole-5-carboxamide (2-amino-5,8-dihydroimidazo[1,2-a]pyrimidin-3-yl)-[(3R)-7-ethynyl-6-fluoro-3-propan-2-yl-2,3-dihydro-1,4-benzoxazin-4-yl]methanone 1-(2,5-dimethoxyphenyl)sulfinyl-4-[3-[(2E)-hexa-2,4-dienyl]phenyl]piperazine 2-(4,5-dihydro-1H-indole-7-carbonylamino)thieno[3,2-b]pyran-6-carboxylic acid 1-[4-(aminomethyl)cyclohexyl]oxy-3-(2H-tetrazol-5-yl)propan-2-one;hydrochloride 1-[7-(2,5-dichloropyridin-4-yl)oxy-1H-indol-3-yl]butan-1-one N-(4-aminocyclohexyl)-3-methoxy-5-pyrrolidin-1-ylsulfonylpyridine-2-carboxamide;hydrochloride 4-[6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carbonyl(methyl)amino]benzoic acid (2E,4Z)-3-chloro-6,7-dimethylhepta-2,4-dien-1-amine;ethane;N'-[2-(5-fluoropyridin-2-yl)ethynyl]ethanimidamide 5-(2-morpholin-4-ylethoxy)-N-[1-(oxan-4-ylmethyl)pyrazol-3-yl]pyridine-2-carboxamide [4-[3-(3,5-difluorophenyl)propanoyl]piperazin-1-yl]-pyridin-2-ylmethanone 5-azidooxy-N-pyridin-2-ylpyrimidin-4-amine 3-[2-(3,5-difluorophenyl)ethyl]-1H-quinoxalin-2-one [3,5-bis(trifluoromethyl)phenyl]methanimine;ethane (1S,3R)-2-[[2-[4-(2-aminoethoxy)anilino]-5-fluoropyrimidin-4-yl]methyl]-2-azabicyclo[4.1.0]heptane-3-carboxylic acid 1-(4-ethenylphenyl)-N,N-dimethylpropan-2-amine;hexane 2-(4,6-dioxospiro[1H-pyrrolo[3,4-c]pyrrole-3,4'-piperidine]-1'-carbonyl)-N-hydroxyacetamide 4-(1,1,1-trimethoxydecan-2-yl)phenol 6-azidooxy-1-bromo-2,3-dihydro-[1]benzofuro[3,2-c]pyridine 4-(4-chlorophenoxy)-1-[(3R,5S)-3,5-dimethylpiperidin-1-yl]butan-1-one N-(diaminomethylidene)-3-[1,5-bis(4-fluorophenyl)-4-hydroxypyrazole-3-carbonyl]-1H-indole-7-carboxamide 5-(2,5-dichlorophenyl)-4-N-[4-[(4-methylpiperazin-1-yl)methyl]benzenecarboximidoyl]pyrimidine-4,6-diamine 4-chloro-6-[(4R)-1,4-dimethylpyrrolidin-3-yl]oxypyrimidine;2,2-dimethylpropane 5-N-(3,4-dihydroxyphenyl)-2-[(3S)-1-methylpyrrolidin-3-yl]oxypyrimidine-4,5,6-tricarboxamide 2-(3,5-difluorophenyl)-N-[1,4-dimethyl-7-[4-(trifluoromethoxy)phenoxy]naphthalen-2-yl]acetamide 1-(3-fluorophenyl)sulfonyl-2,5-dimethylbenzene (2S)-N-[5-(3,4-dichlorophenyl)sulfonyl-1H-indazol-3-yl]-4,4-difluoropyrrolidine-2-carboxamide 1-(2,4-dichlorophenyl)-6-hydroxy-5-[[[3-methyl-4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]amino]methyl]pyrimidine-2,4-dione 6-[4-amino-3-[(Z)-1-methyliminobut-2-en-2-yl]imidazo[4,5-c]pyridin-6-yl]-3H-thieno[3,2-d]pyrimidin-4-one 4-[(3R)-1-butanoylpiperidin-3-yl]-2-methyl-1H-pyrimidin-6-one (4S)-N-[(2,3-dichlorophenyl)methyl]-1'-ethylspiro[5,7-dihydropyrazolo[3,4-b]pyridine-4,3'-indole]-2'-carboxamide N-butylformamide;N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)formamide 1-[4-methyl-6-(4-pyrimidin-2-ylpiperazin-1-yl)pyrimidin-2-yl]-3-(2-methylpyrazol-3-yl)sulfanylazetidin-3-ol 4-[3,5-bis(2-carboxyethyl)phenyl]-1H-pyrrole-3-carboxylic acid 5-(5-bromopyridin-3-yl)pyrazolo[1,5-a]pyrimidine 2-[N-(benzenesulfonyl)-4-chloroanilino]acetic acid 1-[2-(4,5-diphenyl-1H-imidazol-2-yl)pyrrolidine-1-carbonyl]imidazolidin-2-one 4-ethoxy-5-methyl-N-[2-(1,3,7-trimethylindol-2-yl)ethyl]oxan-2-amine 5-bromo-4,7-difluoro-2-propan-2-ylquinoline 2-amino-7,8-dihydro-6H-pyrrolo[1,2-a]pyrimidine-3,4-dione;1-methyl-3-(2-phenylethynyl)benzene ethane;2-methylbut-1-ene;N,3,4-trimethyl-5-(2-oxopropoxy)benzamide 2-azido-1,3-dichloro-4,5-bis(methylsulfanyl)benzene N-(2,4-dinitrophenyl)-N-methylsulfonylhexadecanamide 3-(2,4,6-trimethylphenyl)propylphosphonic acid 4-[(2-butoxy-2-oxoethyl)-[(4-nitrophenyl)methyl]amino]benzoic acid 3-(4-methoxyphenyl)-1,3-diazepane-2,7-dione [1-(4-methylsulfonylphenyl)cyclopropyl]-[(3R,5S)-3-methyl-5-pyridin-2-ylpiperidin-1-yl]methanone N-(2,6-dimethylphenyl)-5-methoxypyrazine-2-carboxamide 4-N-(2,4-dinitrophenyl)-3-fluoro-6-pyridin-4-ylpyridine-2,4-diamine (3aR,7aS)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-5-(oxane-4-carbonyl)-3,3a,6,7,7a-hexahydro-1H-pyrrolo[3,4-c]pyridin-4-one;2,2,2-trifluoroacetic acid N-(2,4-dichloropyrimidin-5-yl)-1,3-thiazol-2-amine 4-(4-tert-butylphenyl)-3-[[4-chloro-2-(trifluoromethyl)anilino]methyl]pyrrolidine-1-carboxylic acid 4-(1-butylpiperidine-3-carbonyl)-6-hydroxy-3,5-dihydropyrrolo[3,4-c]pyrrol-1-one 2-chloro-6,7-dimethoxy-4a,10a-dihydroanthracene 3-(2,4-dichlorophenyl)-1-(4-fluoro-2,6-dimethylanilino)pyrrolidine-2,5-dione 2-[(3,4-dichlorophenyl)methylamino]-N'-hydroxypyrimidine-5-carboximidamide N-[3-hydroxy-4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonylamino)butyl]-1H-indazole-3-carboxamide N-cyclohexyl-1-[5,6-dimethoxy-1-(2-methylsulfanylethyl)benzimidazol-2-yl]piperidine-4-carboxamide [(3S,4R)-1-(2-hydroxyethyl)-4-pyridin-4-ylpyrrolidin-3-yl]urea 2-[(4-aminophenyl)methyl]-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one (2R)-6-chloro-N-[3-fluoro-5-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydroquinoline-2-carboxamide N-[(2S)-5,7-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl]-6-(5-methoxypyridin-3-yl)-3H-benzimidazole-5-carboxamide N-[1-(3,5-dichlorophenyl)-2-methylpropyl]-6-oxo-2-piperidin-4-yl-1H-pyrimidine-4-carboxamide 2-(1,3,5-trimethylpyrazol-4-yl)pyridine-3-carboxamide 5-(2-azidoethyl)-3-(4,4-difluoropiperidin-1-yl)pyridine 6-[2-(5-methyl-1,3-dioxan-2-yl)ethoxy]-4H-pyrido[3,2-b][1,4]thiazin-3-one 4-[2-(3,3a,5,6a-tetrahydro-2H-cyclopenta[b]pyrrole-1-carbonyl)thieno[3,2-d]pyrimidin-4-yl]oxypiperidine-1-carboxylic acid 2-[6-[5-(azetidin-1-ylmethyl)pyridin-3-yl]isoquinolin-3-yl]acetamide 4-[[1-(cyclohexylmethyl)azetidine-2-carbonyl]amino]benzoic acid 2-[(E)-5-ethenylhept-1-en-3-ylideneamino]oxy-4-nitroaniline;methanimine 7-ethoxy-4,9-difluorofluoren-2-amine (3aR,7aS)-5-[2-(4-chlorophenyl)ethyl]-N-(thiophen-2-ylmethyl)-2,3,4,6,7,7a-hexahydrofuro[3,2-c]pyridine-3a-carboxamide;2,2,2-trifluoroacetic acid 3-methyl-4-[(E)-2-phenylethenyl]cyclohexa-1,5-diene-1,2-disulfonic acid 2,6-bis[3-(trifluoromethyl)phenyl]pyridine 5-[(E)-3-amino-1-hydrazinylbut-2-en-2-yl]pyridine-2,4-diamine;hydrochloride 2-[5-(4-chlorophenyl)-4,6-dimethylpyrimidin-2-yl]sulfanyl-N'-hydroxyethanimidamide (3R)-6-chloro-5-[(2,4-dimethoxyphenyl)methylsulfanyl]-1'-propanoylspiro[1H-indole-3,4'-5,7-dihydropyrazolo[3,4-b]pyridine]-2-one N-(5,8-dimethylquinolin-6-yl)pyridine-3-carboxamide N-[(4-methoxyphenyl)methyl]spiro[1,4-dihydroquinoline-3,2'-piperidine]-2-imine 1-phenyl-2-(trifluoromethyl)piperidine [2-(1H-indazole-6-carbonyl)-2,7-diazaspiro[3.4]octan-7-yl]-(oxetan-3-yl)methanone N-[(Z)-butan-2-ylideneamino]-4-ethylaniline;7-methoxy-1,3-dimethylimidazo[4,5-c]quinolin-2-one 4-[(3R)-4-[(2S)-2-aminopropanoyl]morpholin-3-yl]benzoic acid N-[(E)-4,4-difluoro-3-methylpent-1-enyl]-3-methylsulfanylbenzamide 2,4-diamino-6-(2,3-dihydro-1-benzofuran-5-yl)pyridine-3,5-dicarbonitrile 2,4-dimethyl-5-[3-(trifluoromethoxy)phenyl]-1H-pyrimidin-6-one 4-(1,2-dimethylindol-3-yl)piperazine-1-carboxylic acid 3-[2-(4-methoxyphenyl)phenoxy]cyclobutan-1-amine N-(4-acetylphenyl)-2,4-dichloro-5-[(Z)-1-hydroxypent-3-enyl]benzenesulfonamide (2Z)-2-(4,4,6,7-tetramethyl-3H-1,2-dioxepin-5-ylidene)acenaphthylen-1-one (3,5-diethylphenyl)methanesulfonic acid 2-[(E)-1-chlorobut-1-enyl]-3,5-bis(ethenyl)pyrazine (2S,3R)-2-[(4-ethyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N'-hydroxy-3-(oxolan-2-ylmethoxy)butanehydrazide N-methyl-4-[(6-methylthieno[2,3-d]pyrimidin-4-yl)amino]butanamide;hydrochloride 2-[4-(1H-indole-3-carbonyl)piperazin-1-yl]acetaldehyde 3-[2,4-dihydroxy-6-(4-nitrophenoxy)phenyl]propanamide 1-[2,6-di(propan-2-yl)phenyl]-3-[3-methoxybutyl(methyl)amino]sulfanylurea [2-(9H-fluoren-1-yl)pyrazol-3-yl]phosphane 1-[3-(4,6-diphenyl-2H-1,3,5-triazin-3-id-2-yl)carbazol-9-yl]-3-(5-methylpyridin-2-yl)imidazo[1,5-a]pyrazine;platinum(2+) [4-(1,4-diazepan-1-yl)-3-hydroxy-5-iodophenyl]carbamic acid 3-azido-1,4-dimethylpyrrole;N'-ethyl-N-[(2Z)-5-methylideneocta-3,7-dien-2-yl]ethane-1,2-diamine 1-[2,4,6-tris(trifluoromethyl)phenyl]ethanone (3S,6R)-1-benzoyl-3-[2-[(2Z)-1-(4-fluorophenyl)-2-(1-hydroxyethylidene)hydrazinyl]ethyl]-6-methylpiperazine-2,5-dione N-(1,3-benzothiazol-2-yl)-4-oxo-2,3-dihydrochromene-7-sulfonamide 2-[5,6-bis(4-chlorophenyl)pyrazin-2-yl]sulfanyl-N'-diazenylethanimidamide 1-cyclohexyl-4-methoxy-6,7-dihydronaphthalene 1-[(2S)-5-(4-chlorophenyl)pyrrolidin-2-yl]-3-[5-(furan-2-yl)-1,2-oxazol-3-yl]propan-1-one 2-[1-(2,6-difluorophenyl)propoxy]-N'-(4,5-dihydropyrazolo[1,5-a]pyrimidin-7-yl)-3H-pyrrolo[2,3-c]pyridine-6-carboximidamide N-[5,6-bis(phenylmethoxy)pyridin-3-yl]-1-methyl-3-pyridin-3-ylpyrazole-4-carboxamide 3-(1,2,4-triazin-5-yl)-2H-benzo[e]benzimidazole N-[2-(4-azidooxybutylsulfanyl)ethyl]-5,6,7,8-tetrahydroquinolin-8-amine 4-azido-2-tert-butyl-3-iodopyridine [4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]-(3-propan-2-ylidenecyclobuten-1-yl)methanone [1-[3-(6-methoxypyridin-3-yl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidine-2-carbonyl]carbamic acid 5-[[7-[3-(2-methylpyridin-4-yl)propoxy]thieno[3,2-c]quinolin-4-yl]amino]pentanamide 4-[(3R)-1,3-bis(dimethylamino)-2-methylidenepentan-3-yl]-N-hydroxybenzamide 1-(6-tert-butyl-2,3-dihydro-1,4-benzothiazin-4-yl)ethanone (1S)-3,4-bis[4-(trifluoromethylsulfonyl)phenyl]cyclohexan-1-amine 6-chloro-4-(3,5-dibromophenyl)-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 2-[3-amino-5,6-bis(4-chlorophenyl)pyrazin-2-yl]oxyacetic acid 3-methyl-4-(2,2,2-trifluoroethoxy)-N-[(E)-1-pyrimidin-5-ylpropylideneamino]benzamide 3-[(E)-1-[1-methyl-6-oxo-4-(trifluoromethyl)pyrimidin-5-yl]pent-2-en-2-yl]benzonitrile (E)-N-[[7-[2-cyclopentyl-1-(2,5-difluorophenyl)ethoxy]-6-methylsulfanyl-4H-thiopyrano[3,2-d]pyrimidin-3-yl]methyl]-N',N'-dimethylbut-2-ene-1,4-diamine N-(azidooxymethyl)-2,6-dichloroaniline 3-benzyl-2,6-dihydropyrazolo[4,3-d]pyrimidin-7-one 6-chloro-4-[4-(hydroxymethyl)phenyl]sulfanyl-2H-isoquinolin-1-one 4-[(2E)-3,7-dimethylocta-2,6-dienoxy]benzaldehyde 3-[5-tert-butyl-2-(2,4-dioxopyrimidin-1-yl)phenyl]-N,N-dimethylpropanamide 6-chloro-3-(cyclopropylmethylamino)pyridine-2-carboxamide 6-[(E)-2-pyridin-4-ylethenyl]thieno[3,2-d]pyrimidine 3-[3-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydrocinnoline N-[(1S,2R)-2-hydroxycyclobutyl]-6-methoxypyridine-3-carboxamide 6-chloro-N-[2-(dimethylamino)ethyl]-4,5-didehydroquinoxaline-2-carboxamide N-[(Z)-3,7-dimethyloct-2-enoxy]benzamide (2S)-1-[2-[(5R)-5-[[5-chloro-6-(trifluoromethyl)pyridine-3-carbonyl]amino]cycloocten-1-yl]acetyl]piperidine-2-carboxylic acid 6-chloro-4,4-difluoro-1,3-dihydroisoquinoline-2-carboxylic acid 4-[8-(2,6-dimethylcyclohexa-1,3-dien-1-yl)oxy-5-methylspiro[3H-chromene-2,4'-piperidine]-4-yl]benzoic acid 1-methyl-2-(4-methylsulfonylcyclohexa-1,3-dien-1-yl)benzene N-(2,3-dihydro-1H-inden-5-ylmethyl)-4-methoxy-6-oxo-1H-pyridine-3-carboxamide 2-(1,3-benzothiazol-2-yl)benzoate 6-(cyclohexylmethoxy)-1-cyclopentyl-4H-3,1-benzoxazin-2-one N-methyl-3-(4-methylpiperazin-1-yl)aniline [2-bromo-4-(2,5-dimethylphenyl)phenyl]-(3,4-difluorophenyl)methanone 2-amino-4-[2,5-dimethyl-3-(trifluoromethoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile 4-[3-(2,6-dichloroanilino)-2-hydroxypropoxy]benzenesulfonic acid [4-methyl-3-(2,3,5-trifluorophenyl)piperazin-1-yl]-[6-(3,3,3-trifluoropropoxy)pyridin-3-yl]methanone 3-[2-[(1R)-3-chlorocyclopentyl]oxyethoxy]-N,N-dimethylbenzamide 4-(cyclobutylmethyl)-3-methylsulfanyl-6-(trifluoromethoxy)benzene-1,2-dicarbonitrile 2-(4-aminophenyl)benzoate 1-(3-fluorophenyl)sulfonyl-7-methoxypyrrolo[2,3-c]pyridine N-[2,3-bis(ethenyl)-4-(methylideneamino)phenyl]-5-methoxy-1-benzofuran-2-carboxamide N-(4,5-dimethylpyridin-2-yl)-1H-imidazole-3-[5-(hydroxymethyl)oxolan-2-yl]methanesulfonamide 4-[(3S)-1-[2,6-difluoro-4-[(3R,5S)-3,4,5-trimethylpiperazine-1-carbonyl]phenyl]pyrrolidin-3-yl]oxybenzonitrile N-benzyl-3,5-bis(dimethylamino)-2-hydroxybenzamide (4R)-4-[4-(3,5-difluorophenyl)imidazol-1-yl]oxolan-2-one 1-[4-[(2R)-5-chlorospiro[3H-1-benzofuran-2,3'-pyrrolidine]-1'-yl]phenyl]-4-methoxypyrimidin-2-one [3-(1-hydroxynaphthalen-2-yl)oxyphenyl]boronic acid [(2S)-2-benzamido-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]carbamic acid 2,3-bis(dichloromethyl)pyridine N-benzyl-N'-[3-(1,1-difluorobutoxy)phenyl]methanimidamide 7-benzyl-2,7-diazaspiro[4.5]decan-1-one 2-(4-butyl-3,5-dimethoxyphenyl)pentanal 2-(4-methylphenyl)-N-[1-(2,3,4,5-tetrahydrobenzo[c]quinolizin-6-ylsulfanylmethylamino)propan-2-ylidene]propanamide N-ethyl-2,4,5-trifluoro-3-hydroxybenzohydrazide 2-[(2,3-dimethoxyphenyl)methyl]-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-phenylpyrazol-3-yl]-2-methoxyacetamide N-[4-(2,3-dihydro-1H-inden-5-ylamino)pyrimidin-5-yl]-1-[(Z)-prop-1-enyl]-6-pyridin-4-ylbenzimidazole-2-carboxamide (2S)-1-N,3-N-dibenzyl-1-N-[1-[2-(5-formamido-1H-imidazol-4-yl)ethylamino]-7-methylnaphthalen-2-yl]-4-oxopyrrolidine-1,3-dicarboximidamide 1-methyliodanuidyl-3-[(2E)-penta-2,4-dien-2-yl]benzene 3-[1,6-di(propan-2-yl)naphthalen-2-yl]oxybenzonitrile N-(2,6-dimethylphenyl)-5-[(Z)-3-fluoropent-1-enyl]thiophene-2-carboxamide N-benzyl-1-[(3,4-dichlorophenyl)methyl]-2-oxoimidazolidine-3-carboxamide 5-(6-acetamidopyridazin-3-yl)oxy-2-fluorobenzoic acid;5-bromopyrimidine 5-chloro-4-fluoro-2,3-dimethylacridine 2-[4-[[2,3-difluoro-6-(4-pentylphenyl)phenoxy]methyl]-3,5-difluorophenyl]-5-ethoxypyrimidine 1-[4-(2,3-difluorophenyl)piperazine-1-carbonyl]piperidine-4-carboxylic acid [1-(2,6-dichlorophenyl)piperidin-3-yl]-(7-methoxy-4,5-dihydroimidazo[1,2-a]quinolin-3-ylidene)methanamine 5-[[(2S)-1-methyl-3,6-dihydro-2H-pyridin-4-yl]methoxy]-1,2,3,4-tetrahydroisoquinoline N-(3,4-dichlorophenyl)sulfonylcyclopropanecarboxamide 2-[5-chloro-7-fluoro-6-(1,3-oxazol-4-yl)-1H-indol-3-yl]ethanol 1-(2,2-difluoroethyl)azepane;4-[[2-hydroxypropoxy(methylsulfanylamino)phosphoryl]methyl]benzonitrile 1-(3,5-dimethyl-6-oxo-4H-thieno[2,3-c]pyrrole-4-carbonyl)piperidine-2-carboxamide 1,3-dibromo-5-[4-[[2-(3,4-dichlorophenoxy)-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]sulfinylbenzene 2-amino-5-methyl-3H-quinazoline-4,8-dione;N-[(2S)-1-(methylideneamino)propan-2-yl]-6-oxohexanamide (5R)-3,3-dimethyl-4-[6-methylidene-1-(4-phenylphenyl)cyclohexa-2,4-dien-1-yl]morpholine [1-(5,6-dimethyl-2,4-dioxopyrimidin-1-yl)-2-hydroxypropan-2-yl]carbamic acid 3-(2,4-dioxopyrimidin-1-yl)-N-[(1S)-1-(1H-imidazol-5-yl)ethyl]propanamide N-(cyclohexylmethyl)-2-[(3S,4R,5R,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxybenzamide (2R,3S)-N',3-dihydroxy-2-[[4-(pyrrolidine-1-carbonyl)phenyl]methyl]butanediamide 6-hydroxy-1-[2-(4-methylpiperazin-1-yl)-5,6-dihydrobenzo[h]quinazolin-8-yl]-5H-pyrazolo[3,4-d]pyrimidin-4-one (5R)-N-(3,4-dichlorophenyl)-2-(2-methylpiperidin-1-yl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 1-[4-(3,5-dimethylanilino)quinolin-2-yl]cyclopentan-1-ol N-[(E)-(2,4-dihydroxyphenyl)methylideneamino]-3-methoxy-1H-pyrazole-5-carboxamide 3-[(4-chlorobenzoyl)amino]-N-methyl-4-oxo-5-phenylpentanamide [2-chloro-5-(trifluoromethyl)phenyl]-propan-2-yloxyphosphane 2-hydroxy-4,5-bis(trifluoromethyl)benzenesulfonamide 3-(2-hydroxy-4,5-diphenyl-1H-indol-3-yl)propanamide 4-[5-fluoro-2-(trifluoromethyl)phenyl]sulfonyl-1-methylpiperazine-2-carboxylic acid 4-(2,3-dihydro-1H-inden-5-ylamino)quinoline-2-carboxamide 6-cyclopropyl-N-methoxy-1H-indole-2-carboxamide 3-(2,4-dimethoxyphenyl)-2-hydroxypropanoic acid (2S,5R)-1-azido-4,7-dibromo-3,5-bis(phenylmethoxy)heptan-3-ol 2-[3,4-dichloro-5-(trifluoromethyl)phenyl]-6-iodo-3H-quinazolin-4-one 2-amino-4-[(5Z)-6-hydroxyhexa-1,3,5-trienyl]benzenecarboximidamide [(Z)-2-[4-[3,5-dichloro-6-methyl-4-(pyridin-3-ylmethoxy)pyridin-2-yl]pyrazol-1-yl]ethenyliminomethyl]carbamic acid 1-azidooxynaphthalene-2-carboxylic acid 1-[2,5-difluoro-4-(trifluoromethyl)phenyl]-3-[6-ethoxy-2-[4-(methylaminomethyl)piperidine-1-carbonyl]pyridin-3-yl]urea 4-methylpentacyclo[10.7.1.02,5.08,20.013,18]icosa-1(19),2(6),3,7,9,11,13,15,17(20),18-decaene;propane 2,3-dibutyl-6-[(4-fluorophenyl)methyl]cyclohexan-1-one 4-[2-(3-methyl-1,3-benzothiazol-3-ium-2-yl)ethenyl]benzene-1,3-diamine;iodide N-[5,6-dichloro-4-(trifluoromethyl)cyclohexa-1,3-dien-1-yl]benzamide N-azido-6-ethoxy-5,7-difluoroquinoline-8-carboxamide 2-fluoro-6-[(1-methylcyclopropyl)amino]-4-(2,2,2-trifluoroethoxy)benzoic acid N-[5-[3-(4-pyridin-2-yl-1H-benzimidazol-2-yl)-1H-indazol-5-yl]pyridin-3-yl]propanamide N-[4,5-dichloro-2-(trifluoromethyl)phenyl]-2-[[3-[4-oxo-6-(1H-pyrazol-5-yl)quinazolin-3-yl]cyclopentyl]amino]acetamide 5-methyl-7-(1H-pyrazolo[3,4-d]pyrimidine-4-carbonyl)-2-pyridin-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-one 1-[4-(3,3-dimethylpentanoyl)phenyl]-2,2-difluoropropan-1-one 1-[5,6-dimethyl-2-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]-N,N-bis(pyridin-4-ylmethyl)piperidin-4-amine 2,4-diamino-N-[(3R)-1-[(3S,5R)-3-chloro-5-hydroxypiperidine-1-carbonyl]piperidin-3-yl]pyrimidine-5-carboxamide [(3R)-4,7-dichloro-2,5-dioxo-3-phenyl-1,3-dihydroimidazo[1,2-a]quinolin-9-yl]boronic acid [4-(6-chloro-1H-benzimidazol-2-yl)piperidin-1-yl]-[5-methyl-2-[3-(trifluoromethoxy)phenyl]-1,3-oxazol-4-yl]methanone [3-(4,5,6,7-tetrahydrothieno[2,3-c]pyridine-2-carbonyl)phenyl]carbamic acid (2S)-N-[(3R,4S)-4-methoxypiperidin-3-yl]-2-[2-oxo-2-(4,4,6,7-tetramethyl-1H-isoquinolin-2-yl)ethyl]pyrrolidine-1-carboxamide;hydrochloride 2-hydroxy-3,5-dimethoxybenzamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]sulfanylethanethiol N-[(2S,5R)-2-tert-butyl-5-[[4-(1,3-dimethylpyrazol-4-yl)benzoyl]amino]piperidin-1-yl]carbamate N-[4-chloro-3-[2-(propylamino)imidazo[1,2-b]pyridazin-6-yl]phenyl]-2-fluorobenzamide N-[3-[2-(1H-indazol-5-ylamino)thieno[3,2-d]pyrimidin-7-yl]phenyl]formamide 5-N-benzyl-2,3-dimethylbenzene-1,4-diamine 4-(4-bromophenyl)sulfanylthiophene 2-[1-methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indazol-3-yl]oxyethanol 2-azido-5-[4-(trifluoromethyl)phenoxy]pyridine (3R)-4,4-dimethyl-3-[1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]pentanoic acid N-[1-[[(1R,2S)-2-aminocyclohexyl]methylsulfonyl]piperidin-4-yl]-N'-ethyl-2-fluorobenzenecarboximidamide (E)-N'-[1-(3,5-difluorophenyl)ethyl]-4-[2-fluoro-6-hydroxy-4-(2-methoxypyridin-4-yl)phenyl]but-3-enimidamide [(2S)-1-[5-fluoro-6-methoxy-8-(3,3,3-trifluoropropylamino)imidazo[1,2-a]pyridine-2-carbonyl]pyrrolidin-2-yl]methylcarbamic acid (2S,4R)-1-[6-chloro-8-fluoro-7-(2-fluoro-6-hydroxyphenyl)-1-oxo-2H-isoquinolin-3-yl]piperidine-2,4-dicarboxamide 2-azido-6,7-dichlorochromene 1-[(3R)-2,5,7-trimethyl-6-propan-2-yloxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]piperidine-2-carboxylic acid 3-chloro-2-(4-ethoxyphenyl)sulfonylpropanenitrile (Z)-3-ethoxy-4,8-dimethylnon-5-enal;N'-[(E)-2-(dimethylamino)ethenyl]-N-propan-2-ylmethanediamine;3-[5-(4-fluorophenyl)cyclohepta-1,6-dien-1-yl]thiophene;propane (2E,5Z)-3-cyclohexylhepta-2,5-dienal;5-[1-hydroxy-2-oxo-2-[3-(4-phenylpiperazine-1-carbonyl)anilino]ethyl]-N,4-dimethyl-1,3-thiazole-2-carboxamide 3-[4-chloro-6-[[7-fluoro-5-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indazol-3-yl]oxymethyl]pyrimidin-2-yl]propan-1-amine 2-(5-bromopyridin-3-yl)ethanethioamide 1-[2-(4-azidooxyphenyl)ethyl]piperidine 1-(4-ethyl-3-methoxyphenyl)sulfanyl-N',2-dihydroxy-3H-pyrazole-5-carboximidamide 3,5-diphenyl-2H-1,4-benzothiazin-6-ol 1-amino-3-(4-butylphenyl)urea 3-(2,6-dimethylphenyl)bicyclo[4.1.0]heptane (3S)-3-[5-bromo-2-oxo-1-(pyridin-4-ylmethyl)pyridine-3-carbonyl]oxy-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxylic acid 2-[3,5-bis(trifluoromethyl)phenyl]-N,4-diphenylaniline 4-tert-butyl-N-[5,6-dimethoxy-2-(1H-pyrazol-4-yl)thieno[3,2-b]pyridin-7-yl]benzenesulfonamide [4-[2-(trifluoromethyl)phenyl]phenyl]phosphane [4-[(2-methylimidazo[5,1-b][1,3]thiazol-3-yl)methyl]piperidin-1-yl]-(6-methylpyridin-3-yl)methanone (2S,4R)-1-[(2S)-3-methyl-2-[[(2S)-2-[(3S)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]oxybutanoyl]amino]butanoyl]-N-[(2S)-1-phenylpropan-2-yl]-4-[(3-phenylmethoxycyclobutanecarbonyl)amino]pyrrolidine-2-carboxamide N-[2,5-dimethoxy-4-(3,4,5-trifluorophenyl)phenyl]propanamide 3-azido-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]benzamide 2-(4-aminophenyl)propanamide;2,3-dihydro-1H-indene (5R)-4,8-dioxo-2-[3-(trifluoromethoxy)anilino]-N,5-dipropyl-7,9-dihydro-6H-imidazo[1,5-b]isoquinoline-5-carboxamide N-[2,4-difluoro-3-[5-(oxan-3-ylmethoxy)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl]but-3-enamide (2E,6Z)-N-benzyl-5-methylidenenona-2,7-dien-1-imine (4R)-2-cyclohexylimino-5',7'-dimethoxy-1-phenylspiro[5H-indole-3,9'-xanthene]-4-amine 2-[5-carbamoyl-9-[(4-ethylphenyl)methyl]-2-thiophen-3-ylcarbazol-4-yl]peroxyacetic acid 3-[4-methylsulfonyl-2-(trifluoromethyl)phenyl]azetidine N-(5,6-dimethylpyrimidin-4-yl)-2,3,4,9-tetrahydropyrano[2,3-h]isoquinoline-8-carboxamide 2-[4-[(7S)-5-oxo-6,7,8,9-tetrahydropyrimido[5,4-c]quinolin-2-yl]piperazin-1-yl]benzonitrile N-benzyl-4-[(2E,5Z)-hepta-2,5-dien-2-yl]oxy-3-methylaniline;(4Z)-2-ethylidenehexane;(E)-pent-2-ene 2-[3-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-4-propan-2-yl-1H-pyrazol-5-yl]-1-[6-(2-oxa-6-azaspiro[3.3]heptan-6-ylsulfonyl)-2,3-dihydroindol-1-yl]ethane-1,2-dione 1-[3-ethylsulfanyl-5-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]-N'-[(E)-4-[6-methoxy-7-(trifluoromethyl)quinazolin-4-yl]but-1-enyl]ethane-1,2-diamine (4aR,7aS)-2-[5-(azidomethyl)pyridin-3-yl]-1,3,4,4a,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazine 3-N-[(2S)-4-aminobutan-2-yl]-6-chloropyrazine-2,3-diamine;ethane [7-(dimethylamino)naphthalen-1-yl]sulfonylazanide 4-(cyclohexylmethoxy)-5,6,7,8-tetrahydroquinoline 3-(1,2-benzothiazol-5-yl)-4H-1,2,4-oxadiazol-5-one N-[2-[4-amino-3-(methyliminomethyl)phenyl]pyridin-4-yl]-5-cyano-6-(difluoromethoxy)pyridine-2-carboxamide 4-[2-(3,5-dimethylphenyl)ethynyl]-1H-tetrazol-5-one N-[5-bromo-3-methyl-2-(propanoylamino)phenyl]-1,2,4-triazine-3-carboxamide 2-[(E)-2-(7,8-dihydronaphthalene-1-carbonyloxy)-3-methylpent-3-en-2-yl]oxyacetic acid [5-chloro-2-(triazol-2-yl)phenyl]-[(1R,3S,4S)-3-hydroxy-4-[[methyl(methylsulfanyl)amino]methyl]cyclopentyl]methanone 1-[2,6-difluoro-3-[[(1R)-2-phenylmethoxycyclopentyl]amino]phenyl]ethanone [4-[2-[(1,3-dihydroxypropan-2-ylamino)methoxy]phenyl]oxan-4-yl]urea 4-[4-[[(2,6-dioxopiperidin-3-yl)-methylamino]methyl]cyclohexyl]-N-methylbenzamide 2-[1,4,6-tris(trifluoromethyl)carbazol-9-yl]benzaldehyde 4-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)cyclopropanecarbonyl]oxybenzoic acid (4S,7aR)-3-methyl-1'-[[1-[4-(trifluoromethoxy)phenyl]imidazol-2-yl]methyl]spiro[5,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c]imidazole-4,4'-piperidine]-2'-one (3-chlorophenyl)-[4-(2,6-difluoro-4-methoxybenzoyl)piperazin-1-yl]methanone;ethane 3-[4-(dimethylamino)pyrimidin-2-yl]phenol 3-chloro-5-[(4Z)-4-[hydroxy-(3-methylphenyl)methylidene]imidazol-1-ium-1-yl]benzonitrile N'-(aminomethyl)-5,6-dichloro-3-[methyl-[1-[2-[4-(trifluoromethyl)phenyl]benzoyl]piperidin-4-yl]amino]pyrazine-2-carboximidamide (2S)-N,1-bis[(4-methylphenyl)methyl]pyrrolidine-2-carboxamide 2-[4-[(3S,5R)-3-amino-5-methylpiperidin-1-yl]pyridin-3-yl]-1H-indole-7-carboxamide [(E)-1-[[3-hydroxy-2-[4-[hydroxy(phenylsulfanyl)methylidene]piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinolin-6-yl]amino]-5-oxopent-2-en-2-yl]urea 2-[3,5-difluoro-4-(1H-indole-2-carbonyl)phenoxy]acetonitrile 3-hydroxy-4-[(1S)-2-phenylmethoxycarbonylcyclopropyl]butanoic acid 2-chloro-N-(1-cyclopropylethenyl)-5,6-dimethylpyrimidin-4-amine 4-benzyl-3-[(2,2-dimethylcyclopentylidene)methyl]benzoate (3Z)-2-cyclohexa-1,5-dien-1-yl-N-methoxy-6-[4-[4-(trifluoromethoxy)phenoxy]piperidin-1-yl]hexa-3,5-diene-1-sulfonamide 2-[6-(4-butylcyclohexyl)-1,3-difluoronaphthalen-2-yl]-5-heptoxypyrimidine N-butyl-4-(1H-indazol-3-yl)aniline N-(2,3-dihydro-1H-inden-5-ylmethoxy)-6,7-dihydro-4H-pyrano[4,3-d][1,2]oxazole-3-carboxamide 3-(5-ethylsulfonylpyridin-2-yl)-1,7-naphthyridine 4-fluoro-2-(1H-pyrazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine 1-[2,3-di(propan-2-yl)phenyl]-5-phenylcyclohexa-3,5-diene-1,2-diamine (3-aminocyclopentyl)-[3-[(4-propan-2-ylphenyl)methoxy]azetidin-1-yl]methanone (5R,6S)-4-[2-ethyl-3-[3-fluoro-5-[6-fluoro-7-(methylamino)pyrido[2,3-d]pyrimidin-4-yl]phenyl]propanoyl]-1,3-diazabicyclo[3.2.0]heptane-2,5-dione 3-(3,5-dimethylphenyl)-1,2-oxazol-4-amine N-[4-[[2,6-bis(trifluoromethyl)phenyl]carbamoylamino]cyclohexa-1,5-dien-1-yl]-4-ethynoxybenzamide 2-amino-4,5-dioxodibenzothiophene-1,3-disulfonic acid 5-[3-chloro-4-(trifluoromethoxy)phenyl]-2,3,6,7-tetrahydrofuro[3,2-c]pyridine 1-[5-[(Z)-2-aminoethenyl]cyclohepta-1,3,6-trien-1-yl]-N'-[5-chloro-4-[2-fluoro-3-(2-methoxyethylsulfanyl)phenyl]pyridin-2-yl]ethane-1,2-diamine N-(4,5-dichloropyrimidin-2-yl)-6-(1,3-thiazol-5-ylsulfamoyl)cyclohexa-1,3-diene-1-carboxamide 7-(2,6-dichlorophenyl)-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]-6H-pyrido[2,3-d]pyridazin-5-imine [4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]-methylidyneazanium 4-(1,3-benzoxazol-2-ylamino)-1-[(2S,5R)-2,5-dimethylpyrrolidine-1-carbonyl]piperidin-4-ol 2-[5-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]-N'-(3,4,5-trimethoxybenzoyl)piperidine-1-carboximidamide 2-chloro-N-[4-[3-(1,3-dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrazin-5-yl]cyclohexyl]pyridine-4-carboxamide 3-benzyl-2-[(2,5-dimethoxyphenyl)methyl]-N-propanoylbenzamide 5-methyl-3,4,6,7-tetrahydro-2H-quinoline;(9R)-4,8,13-trimethyltetracyclo[10.7.0.02,11.04,8]pentadeca-1(12),2,5,14-tetraene (2S)-1-[3-cyano-4-[5-[[ethyl(1,3-thiazol-2-ylmethyl)amino]methyl]thiophen-2-yl]-6-phenylpyridin-2-yl]oxypyrrolidine-2-carboxylic acid 5-(6-aminopurin-9-yl)-2-methoxypentane-1,3-diol (2-tert-butylindolizin-6-yl)urea (2S,3aS)-2-ethenyl-N'-(1H-indole-5-carbonyl)-4-methoxy-5-[5-(trifluoromethyl)pyridin-2-yl]-3a,7a-dihydro-1-benzofuran-2-carbohydrazide 2-[5,6-bis(ethenyl)pyridin-3-yl]oxypropanoic acid 3-amino-2-[2,5-dimethyl-4-(1,1,2,2,3,3,4,4,4-nonafluorobutyl)phenyl]propanoic acid 4-[1-[5-(difluoromethyl)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]piperidin-3-yl]oxybenzonitrile 1-(5-bromo-3-methylpyridin-2-yl)oxy-2,4-dimethoxybenzene N-[1-(2,3-dihydro-1H-inden-5-yl)ethylidene]hydroxylamine 1-cyclopropyl-7,8-dimethoxy-N'-(1-phenylethenyl)pyrazolo[4,3-c]cinnoline-5-carboximidamide 2-[6-(1-methylpiperidine-4-carbonyl)spiro[3,4-dihydronaphthalene-2,4'-piperidine]-1'-yl]acetonitrile 1-(2,4-dichlorophenyl)-5-(1,3-thiazol-2-ylamino)indole-2-carboxylic acid 4-[5-methyl-2-(3,4,5-trifluorophenyl)imidazo[1,2-a]pyridin-3-yl]phenol 5-methyl-3H-1,4-benzodiazepine-7,8-diol 4-[3-(trifluoromethoxy)phenyl]-1H-pyrazolo[4,3-c]pyridine N-(2,6-difluorophenyl)-N-methylsulfonylbutanamide 5-cyclohexyl-1,3-difluoro-2-(4-methylphenyl)benzene 2-(8-oxononyl)-2,3-dihydrofuro[2,3-f]quinoline-4,9-dione N-(1,3-benzothiazol-2-ylsulfanyl)aniline 3-[(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carbonylamino)methyl]thiophene-2-carboxylic acid (3S,4R)-2-(hydroxymethyl)-6-oxo-4-[(2S)-4-phenylbutan-2-yl]oxyoxane-3,5-dicarbonitrile 5-[4-(2,3-dihydroindole-1-carbonyl)anilino]-1,4,6-trimethyl-3-propanoylpyrimidin-2-one 3-N,6-N-bis(1H-imidazol-2-ylmethylideneamino)-9,10-dihydroanthracene-2,3,6-triamine 4-[N'-[1-(3-cyanophenyl)ethyl]carbamimidoyl]benzoic acid 2-[1-(4-fluorophenyl)-5,6-dimethylbenzimidazol-2-yl]propan-2-ol 2-[2-(1,4-dimethylcyclohexa-2,4-dien-1-yl)ethynyl]naphthalene N-(2-bromophenyl)-2,4-dichloro-6-ethylaniline 1-[[(5Z,7E)-5-methylundeca-5,7,9-trien-4-yl]sulfonylmethylamino]pyrazole-3-carboxylic acid 4-(1,3-benzothiazol-2-yl)-5-imino-1-propan-2-yl-2H-pyrrol-3-ol 4-chloro-7-cyclohexyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine 4-(9,9a-dihydrocarbazole-3-yl)pyridine-2,3-diamine 2-[3,5-difluoro-4-(methanesulfonamido)phenyl]butanamide 1-methyl-5-[2-(4-phenylcyclohexyl)ethynyl]triazole [2-(4-chlorophenyl)-5,6-dihydro-4H-1,3-thiazin-4-yl]-[5-ethoxy-1-methyl-4-(4-methylphenyl)pyrazol-3-yl]methanone 4-[3,5-difluoro-2-(trifluoromethyl)phenyl]-1-methylpyridin-2-one (6-ethylpyridin-2-yl)-[3-hydroxy-5-[4-[(E)-2-phenylethenoxy]phenyl]-1,2-dihydroimidazol-4-yl]methanone (2S)-N'-hydroxy-2-methyl-4,4-diphenylbutanehydrazide 2-[[4-(aminomethyl)phenyl]methyl-[(2,6-dichlorophenyl)methoxycarbonyl]amino]acetic acid 2-[4-chloro-3-(2,5-dioxopyrrol-1-yl)phenyl]-N-[(E)-[4-methoxy-6-(morpholin-4-ylmethyl)cyclohexa-2,4-dien-1-ylidene]amino]acetamide 2-chloro-4,5-difluorobenzenethiol 2-[(3R,5S)-4-benzylsulfonyl-1-(2-methoxyethyl)-5-propan-2-ylpyrrolidin-3-yl]acetic acid 3-[(1S)-2-methylsulfonylcyclopent-2-en-1-yl]benzoic acid 7-[(2R,5R)-5-[3-(cyclopropylmethoxy)phenyl]-2-ethyloxolan-2-yl]heptanoic acid (3-chloro-2,6-difluorophenyl)methylcarbamoyloxidanium 1-chloro-3-[(2,4-dibromophenyl)methyl]benzene 3-azido-6-[4-(2,4-difluorophenyl)piperazin-1-yl]pyridazine (4aR,6S)-1-[2-oxo-3-[4-(trifluoromethyl)phenyl]propanoyl]-4a-(5-phenylpentoxycarbonylamino)-6-thiophen-2-yl-2,3,4,5,6,7,8-hexahydro-1H-isoquinoline-8a-carboxylic acid 1-[[1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]methyl]-5-oxopyrrolidine-3-carboxylic acid N-[2-(1,3-benzodioxol-5-yl)ethyl]-2-(oxan-4-yl)acetamide N-[5-(6-fluoroquinolin-4-yl)oxypyridin-2-yl]-1,3-dihydroisoindole-2-carboxamide 2-(4-fluoroanilino)-N-[(E)-2-nitroethenyl]acetamide (2Z,5R)-2-[(Z)-(3-methoxy-4-phenylmethoxyphenyl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one (2E,4Z)-5-[6-(1H-pyrrolo[3,2-c]pyridin-2-ylmethoxy)quinolin-4-yl]penta-2,4-dien-2-amine 4-methoxy-5,6-dimethyl-2-propan-2-ylquinoline 2-[5-methyl-6-[2-(5,6,7,8-tetrahydronaphthalen-1-yl)ethyl]naphthalen-2-yl]-4,5-dihydro-1H-imidazole 5-cyclohexyl-2,4-dihydroxy-N'-[[1-(methoxymethyl)cyclopropyl]amino]benzenecarboximidamide 2-(azidooxymethyl)pyridine-3,5-dicarbonitrile N-[[4-(1H-imidazol-5-yl)phenyl]methyl]cyclohexanamine 1-butyl-3-[5,6-dimethoxy-2-(4-phenylpiperidin-1-yl)-3H-quinazolin-4-ylidene]urea N-ethyl-2-[methyl(2-methylpropyl)amino]quinoline-3-carboxamide 4-chloro-N,5-dimethyl-2-(2,3,4-trifluorophenyl)aniline 3-[(E)-2-[4,5-dimethoxy-1,3-bis(phenylsulfanyl)cyclohexa-2,4-dien-1-yl]ethenyl]-N-ethyl-6-fluorochromen-4-imine N-[2,6-bis(4-fluorophenyl)pyridin-4-yl]quinolin-3-amine (4S)-6,7-dichloro-8-[(2R,3S)-5-fluoro-2,3-bis(phenylmethoxymethyl)oxolan-2-yl]-1-[(4-methoxyphenyl)methyl]-4H-chromeno[4,3-c]pyrazole 3-(4-fluorophenoxy)-N,N-dimethylpropan-1-amine;2-[4-(8-fluoroquinolin-6-yl)oxypiperidin-1-yl]ethanol 2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-N'-methanimidoyl-6-pyrrolidin-1-ylpyrimidine-4-carboximidamide 1-cyclohexylsulfanyl-2,3-difluorobenzene N-(1,2,3,4-tetrahydroquinolin-4-yl)-1H-pyrazolo[3,4-b]pyridine-5-sulfonamide 2-[(Z)-(4-butoxycarbonylphenyl)methylideneamino]oxyacetic acid 6-[4-(2,3-dichlorophenyl)sulfonylmorpholin-3-yl]-1H-pyridin-2-one 5-[(E)-2-(2-chlorophenyl)ethenyl]-2-N,4-N-bis(3-fluoropropylsulfonyl)pyridine-2,4-diamine N-ethyl-5,6,7,8-tetrahydro-4H-cyclohepta[d][1,3]thiazol-2-amine 4-[[(2S)-1-amino-3-phenylpropan-2-yl]carbamoyl]-1-methylpyrrole-2-carboxylic acid N-(2,6-dimethylphenyl)-4-[3-[2-(dimethylamino)ethoxy]phenyl]-3-[2-(furan-2-carbonylamino)propanoylamino]benzamide 5-(4-bromophenyl)-7,12-difluoro-1,8,9,11-tetrazatricyclo[8.4.0.02,7]tetradeca-2(7),3,10,12-tetraene 5-chloro-2-[[6-(trifluoromethyl)pyridine-3-carbonyl]amino]benzoic acid 1-[7-chloro-3-ethyl-2-(methoxymethyl)pyrazolo[1,5-a]pyridin-6-yl]-1-phenylpropan-2-one;2,4,8,11-tetraoxatricyclo[7.3.0.03,7]dodeca-1(9),3(7),10-triene 3-[6-[4-(azidomethyl)-4,5-dihydroimidazol-1-yl]pyridin-2-yl]oxy-N,N-diethylaniline 1-(3,4-dihydropyridin-2-yl)-N-[4-methoxy-2-[3-(trifluoromethyl)phenoxy]phenyl]piperidine-4-carboxamide 4-[N-(4-bromobutan-2-yl)-3,5-dichloroanilino]-N-(2-phenylpyrazol-3-yl)benzenesulfonamide 5-[4-(1,2-dihydroxyethyl)phenyl]-1H-indazole-3-carboxylic acid 4-[2-[3,5-bis(trifluoromethyl)anilino]-1H-benzimidazole-4-carbonyl]piperazine-1-carboxylate 2-(5,6-diethylpyrimidin-4-yl)-3,3a,4,5,7,8,8a-octahydro-1H-pyrrolo[3,4-d]azepine [1-benzylsulfonyl-5,7-di(propan-2-yl)indol-4-yl]methylhydrazine (2S)-4-[3-fluoro-5-[2-methyl-1-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)propan-2-yl]oxyphenyl]butan-2-amine 1,3-bis(ethylsulfanylmethyl)-7-[5-nitro-2-(trifluoromethoxy)phenyl]-4H-quinazolin-4-ol N-azido-4-(5-chloropyrimidin-2-yl)oxypiperidine-1-carboxamide 4-[3-[(2R)-1,5-dimethoxypentan-2-yl]phenyl]-8-methoxypyrido[3,2-d]pyrimidine 5-amino-2-bromo-6-(cyclopenten-1-ylmethyl)pyridine-3-carbonitrile 6-(2-chlorophenyl)-2,3-dihydrothieno[3,4-c]pyridine 1-(1,3-benzodioxol-5-yl)-4-[2-butoxy-4-(2-cyclopropylethynyl)phenyl]sulfanyl-N-methyl-6,7-dihydro-5H-indazole-3-carboxamide 2-[(5-cyanopyridin-3-yl)methylamino]-N'-(3-sulfamoylphenyl)ethanimidamide 2-(3-bromo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)ethanol;hydrochloride 1-[2-(1,3-benzodioxol-5-ylmethoxy)phenyl]sulfonyl-4-(1-hydroxyethyl)piperidine-4-carboxamide 1-amino-N'-methyl-5-[6-(methylsulfanylamino)pyridin-3-yl]benzimidazole-2-carboximidamide 2-[4-[2-(2,6-difluorophenyl)imidazol-1-yl]pyrazol-1-yl]ethanol 5-[(3S,4R)-1-(cyclopropanecarbonyl)-4-methoxypyrrolidin-3-yl]-1-methylpyrazole-4-carboxamide 4-[[2,4-bis(trifluoromethyl)phenyl]methoxyiminomethyl]pyridine-3-carboxylic acid 3-ethyl-N-(2H-pyrimidin-1-yl)benzenesulfonamide 2-(6-chloropyrazin-2-yl)acetamide 3-[2,3-bis(4-chlorophenyl)imidazo[1,2-a]pyridin-7-yl]phenol 2-(1H-pyrazol-4-ylmethylidene)indene 2-[(3S)-1-[7-methoxy-6-(methylamino)imidazo[1,5-a]pyridine-3-carbonyl]piperidin-3-yl]benzonitrile N-[5-cyano-1-(3,4-difluorophenyl)pyrrolidin-3-yl]-5-(dimethylsulfamoyl)pyridine-2-carboxamide N-[(3S,7S,8aS)-2-[(4-fluorophenyl)methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]imidazo[1,5-a]pyrimidine-5-carboxamide [(7S)-2,7-dimethyl-3-(3,4,5-trifluorophenyl)-5,7-dihydro-4H-pyrazolo[3,4-c]pyridin-6-yl]-[1-(3-ethoxypropylamino)pyrazol-4-yl]methanone 3-chloro-5,6-dimethyl-2-[(4-methylphenyl)sulfonylamino]benzenesulfonic acid N-[2-(dimethylamino)ethyl]-3,5-bis(trifluoromethyl)aniline N-[2-amino-6-(2,5-dihydropyrrol-1-yl)pyrimidin-4-yl]-3-[4-(furan-2-carbonylamino)phenyl]propanamide N-[[4-methoxy-3-(2-methylpropanoyl)phenyl]methylidene]hydroxylamine N-(2,3-dihydroxypropyl)-4-nitro-N-[2-[1,2,4]triazolo[4,3-a]pyrazin-5-yl-[1,2,4]triazolo[4,3-a]pyrazin-5-yl]benzamide 2-[[6-chloro-5-methyl-2-[4-[5-(trifluoromethyl)pyridin-3-yl]butanoylamino]benzimidazol-1-yl]methoxy]ethylazanide [3-(cyclopropylmethylamino)thieno[2,3-c]pyridin-6-yl]-(2-morpholin-4-ylethoxy)methanol 7-[(2R)-1,4-bis(benzenesulfonyl)piperazin-2-yl]heptanal 2,7-dimethyl-6-(2,4,6-trimethoxyphenyl)-3H-quinazolin-4-one 3-[2-(4-methoxyphenyl)ethylamino]-2,5-diazatetracyclo[8.6.0.02,7.011,15]hexadeca-1,3,6,9,11(15)-pentaen-13-one 1-(5,6-dimethoxycyclohexa-2,4-dien-1-yl)sulfonyl-3-phenylpropan-1-one N-[(2S)-1,3-dihydroxypropan-2-yl]-4,5-dimethoxythiophene-3-carboxamide 2-[3-azidooxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-4-ethynylpyridine 4-chloro-N-[(E)-2-[4-(4-hydroxyphenoxy)phenyl]but-1-enyl]benzamide N-(2,6-dimethylphenyl)-3-[4-methoxy-3-[(4R)-oxolan-4-yl]sulfonylanilino]pyrrolidine-1-carboxamide 2-[3,5-bis(trifluoromethyl)phenyl]-N-(3-hydroxycyclopenten-1-yl)-N-propanoylacetamide 4-[6-[2-[3,5-bis(trifluoromethyl)phenyl]ethoxy]pyridin-3-yl]-1-(2-hydroxy-3-phenoxypropyl)piperidine-4-carboxylic acid (2S)-3,4-dihydro-2H-chromene;3-[[3-methoxy-4-[(5-phenyl-1,2-oxazol-3-yl)methoxy]phenyl]methylamino]-N,N-dimethylpropanamide 2-(1,3-benzodioxol-4-yl)-5-[3-chloro-4-(difluoromethoxy)phenyl]-6H-pyrrolo[3,4-d]pyrimidin-7-one 2-[(5Z)-2-amino-4,6,7-trimethylideneocta-1,5-dienyl]benzaldehyde 5-chloro-N-(4,4-difluorocyclohexyl)pyridine-3-carboxamide (2-ethylanilino)oxyformic acid 6-[3,5-dimethyl-4-(trifluoromethoxy)phenyl]-N-[3-fluoro-4-(1H-pyrazol-4-yl)phenyl]pyrimidin-4-amine;ethane 3-[2,6-di(propan-2-yl)phenyl]-4H-pyrido[3,2-d]pyrimidine N-(4,5-dihydroimidazol-1-yl)-N,N'-dimethoxy-2-nitrobenzenecarboximidamide (4Z,5E)-3-ethyl-6-methylidene-1-phenyl-4-propylidenepyridine 6-[4-(difluoromethyl)phenyl]-3,5,8-triazabicyclo[4.2.0]octane (1R)-2-[5-(2,6-difluorophenyl)pyrazin-2-yl]cyclobutan-1-ol [4-(6,7,8,9-tetrahydrodibenzofuran-2-yl)phenyl]methanol [4-(2-hydroxyphenyl)-1,3-thiazol-5-yl]carbamic acid N-benzyl-2-(hydroxymethylamino)-3-(2,4,6-trimethylphenyl)propanamide 5-(5-nitropentyl)benzene-1,2,3-triol 2-amino-N-(4-chlorophenyl)sulfonyl-N'-[2,5-dimethyl-6-(oxiran-2-yl)phenyl]pentanimidamide 5-[(1R)-1-(2,6-dichlorophenyl)ethyl]-3H-1,3,4-oxadiazol-2-one;N-[1-[4-[2-[(Z)-3-hydroxy-2-methylidenehex-3-enyl]pyrimidin-5-yl]cyclohexa-2,4-dien-1-yl]ethyl]acetamide 1-(2-chlorophenyl)sulfonyl-5-ethoxy-3-[4-(2-fluoro-4-methylphenyl)cyclohexen-1-yl]indole 4-bromo-2-(3-methylpyrazol-1-yl)benzoic acid 6-azido-8-ethyl-N-[2-(5-fluoropyridin-2-yl)ethyl]quinazolin-4-amine 1-[(1R,2S)-2-azidocyclopropyl]oxy-3-chlorobenzene (2R,5S)-1-[3-cyano-6-(2,2-difluoropropoxymethyl)pyridin-2-yl]-5-methylpyrrolidine-2-carboxylic acid 4-[5-amino-6-(5-chloro-2,3-dimethoxyphenyl)pyrazin-2-yl]cyclohexan-1-ol 6-[(E)-2-amino-1-hydrazinylbut-2-enyl]-3,4-dihydro-1H-quinolin-2-one 1-benzyl-2,5-dimethoxypyrrole N-[5-(azetidin-1-ylmethyl)pyridin-2-yl]imidazo[1,2-a]pyrazine-8-carboxamide 3-methylsulfanyl-N'-phenyl-6,8,10,11-tetrazatricyclo[7.4.0.02,5]trideca-1(9),2,4,6,12-pentaene-10-carbohydrazide 4-(2,3-dichlorophenyl)-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 4-(3,5-dimethylanilino)piperidine-2-carboxylic acid 2-bromo-N-[(5Z)-4,4-dimethyl-3-oxohexa-1,5-dienyl]benzamide 1-[(3R,4S)-3-(dimethylsulfamoylamino)-4-hydroxypyrrolidine-1-carbonyl]pyrazole 6-amino-2,4-dioxo-4-[3-(pyrazol-1-ylmethyl)phenyl]-1,3-diazinane-5-carbonitrile 7,9-dimethyl-3-phenylnaphtho[2,1-e]indazole 1-benzyl-2,3-dimethoxyphenanthrene 4-(N-acetylanilino)naphthalene-2,3-dicarboxylic acid N-[[4-amino-2-(trifluoromethyl)phenyl]methoxy]sulfanylacetamide [4-(1-phenylpropyl)piperazin-1-yl]methanesulfonic acid N-[3-chloro-4-(trifluoromethylsulfanyl)phenyl]-3,4-dihydroxybenzamide 5-(1,3-benzothiazol-2-ylsulfanylmethyl)imidazolidine-2,4-dione 6-methyl-2-(thiophen-3-yloxymethyl)pyrimidine-4-carboxylic acid 4-(2,6-diphenylpyrimidin-4-yl)-3-methoxyphenol 5-(2,6-dimethoxyphenyl)imidazolidine-2,4-dione N-[4-(benzenesulfonyl)phenyl]-2,6-dichloro-N-(2-methyl-5-nitrophenyl)aniline 3-[3-hydroxy-2-(6-methylpyridin-3-yl)quinoline-4-carbonyl]cycloheptan-1-one 1-methyl-4-[(2E,4Z)-6-phenylhexa-2,4-dien-3-yl]piperazine 5-bromo-1-(2,6-diethoxyphenyl)pentan-1-one 3-(2,5-difluorophenyl)-N-[4-[[(5-methylcyclohexa-1,5-dien-3-yn-1-yl)amino]sulfanylcarbamoyl]phenyl]benzamide;ethane [2-carboxy-1-[4-(4,5-dihydro-1H-imidazol-3-ium-3-yl)phenyl]ethylidene]azanide [(3S)-4-[2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoyl]morpholin-3-yl]azanium [4-(3-fluoro-5-pyridin-2-ylpyridine-4-carboximidoyl)oxyphenyl]azanide (4R)-5-(1,3-benzodioxol-5-ylmethyl)-2-benzylsulfanyl-8-(2,6-dichlorophenyl)-4-hydroxy-3-nitroso-7H-pyrrolo[3,4-b]azocin-6-one 1-[(E)-but-2-enoxy]-6-fluoronaphthalene 4-(3,7-dimethylocta-2,6-dienoxy)benzoic acid 6-amino-5,7-dideuterio-2-methyl-4H-thieno[3,2-b]pyridin-5-ol 4-tert-butyl-2-(3,5-dimethoxyphenyl)pyridine N-[2-(4,6-dimethylpyrimidin-2-yl)oxyethyl]ethanesulfonamide N-[(2R)-1-cyanobutan-2-yl]-1-[2-[[4-[(dimethylamino)methyl]cyclohexanecarbonyl]amino]phenyl]pyrazole-3-carboxamide 1,2-difluoro-7,9-dimethyl-3,4-dihydro-2H-pyrido[3,4-b]indol-5-one 1-[4-(azetidine-3-carbonyl)piperazin-1-yl]-2,3-dimethoxybenzimidazole-5-carbonitrile N-[2-(4-azidophenyl)ethyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide 2-[[5,7-dichloro-2-(4-methylbenzoyl)-3,4-dihydro-1H-isoquinoline-6-carbonyl]amino]propanoic acid (7-benzylpyrrolo[2,3-d]pyrimidin-4-yl)hydrazine N-cyclopropyl-3,5-dimethyl-4-[6-(4-morpholin-4-ylbut-1-ynyl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]-1H-pyrrole-2-carboxamide 3-[2-(3,4-dichlorophenyl)-4-(2-methylpropoxymethyl)piperidine-1-carbonyl]benzonitrile N'-(benzenesulfonyl)benzohydrazide 4-chloro-N'-[5-(3,3-dimethylpiperidine-1-carbonyl)-2H-pyrazolo[3,4-b]pyridin-3-yl]-3-fluorobenzenecarboximidamide 4-methyl-7-(1,2,3,6-tetrahydropyridin-5-yl)quinoline 7-(difluoromethoxy)-6-[2-fluoro-4-[4-(4-methylphenyl)cyclohexylidene]phenyl]naphthalene-2-carbonitrile N-(4-azido-3-methoxyphenyl)-5-[2-chloroethyl(propyl)amino]pentanamide (3R,4S)-N-[3-bromo-5-(trifluoromethyl)phenyl]-1-ethyl-4-(1H-pyrazol-4-ylamino)piperidine-3-carboxamide N-[(Z)-3-aminoprop-2-enimidoyl]-5-[4-(2,3-difluoro-4-methoxyphenyl)phenyl]-1-methylpyrazole-3-carboxamide (2R)-4-benzylimino-2-[3,5-difluoro-4-(1H-indole-2-carbonylamino)phenyl]piperidine-1-carboxylic acid 3-[(6S)-4-chloro-8-(trifluoromethyl)-1,2-dihydrochromeno[3,4-c]pyridine-5-carbonyl]benzoic acid 3-(4-oxo-1,5-dihydropyrazolo[3,4-d]pyrimidin-6-yl)-N-piperidin-2-ylpropanamide;hydrochloride 1-[(2S,4R)-5-(4-chlorophenyl)-4-methyloxolan-2-yl]-N-cyclohexylmethanimine [(3R)-1-[(3S)-1,1-dioxothiolan-3-yl]piperidin-3-yl]-[4-[5-fluoro-2-(4-hydroxyphenoxy)pyridin-3-yl]piperazin-1-yl]methanone (2R)-3,4-dihydroxy-1-[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]butan-2-one 5-chloro-4-N-[[1,3-dimethyl-2-(6-methylidenepyrimidin-2-yl)indol-6-yl]methyl]pyrimidine-2,4-diamine 6-(3,4-dimethoxyphenyl)-5-methylcyclohexa-2,4-diene-1-carboxylic acid 2-(dimethylamino)-N-[4,6-bis(trichloromethyl)pyrimidin-5-ium-1-ylidene]benzamide N-(4-chlorophenyl)-6,7-dihydroxy-1,3,8-trimethylnaphthalene-2-carboxamide N-butyl-3-[2-(4,6-difluorocyclohepta-1,3,5-trien-1-yl)pyrazole-3-carbonyl]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide (4Z)-2-methyl-4-[(3-propoxyphenyl)methylidene]-1H-imidazol-5-one N-[(2R)-1-hydroxypentan-2-yl]-6-methoxypyridine-3-carboxamide 2-(4,5-dihydro-1H-imidazol-2-yl)-1-pyridin-2-ylpyrrole 4-[2-[(4-acetamidophenyl)methyl]tetrazol-5-yl]-N-benzylbenzamide 2-(1,3-benzodioxol-5-ylmethoxy)-7-[2-[4-(3-pyrrolidin-1-ylpropylsulfanyl)piperazin-1-yl]ethoxy]quinazoline;hydrochloride 1-[5-[7-fluoro-3-[4-(4-methylpiperazin-1-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-1H-indazol-5-yl]pyridin-3-yl]-N,N-dimethylmethanamine (3-methylpyridin-2-yl)-[3-methyl-1-[4-[2-(trifluoromethoxy)phenyl]piperazine-1-carbonyl]piperidin-3-yl]methanone 1-[(2S)-4-[3-methyl-4-[5-methylidene-7,8-dihydro-6H-naphthalen-2-yl]phenyl]morpholin-2-yl]ethanone 2-[N-(furan-2-ylmethyl)-3-nitroanilino]decanoic acid 2-[4-[(3E)-hexa-1,3,5-trien-3-yl]anilino]-7H-[1,3]thiazolo[4,5-d]pyrimidine-6-thione 3-N,5-N-diphenylaniline (2S)-N-[3-[[5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide (2R)-1-amino-3-[4-(4-fluorophenyl)-5-methyltriazol-1-yl]propan-2-ol 2-[6,7-di(propan-2-yl)thieno[3,2-c]pyridin-4-yl]-N-ethylethanethioamide 2-[4,5-dichloro-3-(trifluoromethyl)pyrazol-1-yl]-2-hydroxyacetic acid 1-(3,4-dimethoxyphenyl)-N'-[3-[methyl-(2-oxochromene-5-carbonyl)amino]propyl]cyclobutane-1-carbohydrazide 2-(5,6-dihydro-4H-cyclopenta[d][1,3]thiazol-2-yl)-N-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]acetamide 2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[1-[5-fluoro-2-(triazol-2-yl)phenyl]ethyl]pyrido[3,4-d]pyrimidine-7-carboxamide 2-hydroxy-1,3-dimethyl-5-[[2-(4-propan-2-yloxyphenyl)imino-4-(trifluoromethyl)-1H-imidazol-5-ylidene]amino]benzimidazole-6-carboxylic acid 3-[4-bromo-N-(cyanomethyl)anilino]propane-1,2-diol 2-[(4,5-dimethylfuran-3-carbonyl)amino]benzenesulfonic acid 2-N-butyl-1,3-benzothiazole-2,6-diamine 3-[(4S,5R)-3,3-difluoro-1-phenylmethoxycarbonylpiperidin-4-yl]oxypyridine-2-carboxylic acid N-(3,5-dichlorophenyl)-2-[2-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]acetamide 1-(4-acetylphenyl)sulfanylpiperidine-2,3-dione;3-methoxypropanamide 1,3-diamino-1-[2-(cyclopropylmethoxy)naphthalen-1-yl]urea N-[4-(4,5-dihydro-1H-imidazol-2-ylsulfanyl)phenyl]-3-oxopiperazine-1-carboxamide;ethane 2-fluoro-4-(2-fluorobenzoyl)benzaldehyde;N'-methoxy-2,2,3-trimethylbutanimidamide 3-azidooxy-6,7-dimethylnaphthalene 3-azido-1,5-dichloro-2,4-bis(ethenyl)benzene N-[2,4-difluoro-3-(5H-pyrido[2,3-d]pyridazine-8-carbonyl)phenyl]propane-1-sulfonamide [2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-4-yl]hydrazine 3-(2,6-dimethylpyridin-4-yl)-2-phenyl-5H-pyrido[1,2-a]benzimidazol-10-ium 7-[(2,5-dimethylpyrazol-3-yl)methoxy]-N,8a-dihydroquinoline-6-carboxamide N-[3,5-bis(trifluoromethyl)phenyl]sulfanyl-2,4-dimethylaniline 1-methyl-2-[(1S,2R)-2-thiophen-3-ylcyclopropyl]hydrazine 2-[5-(azidomethoxy)pyridin-3-yl]-8-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-6,7-dihydro-5H-indolizine-3-carboxamide [4-(2,6-difluoropyridin-3-yl)piperidin-1-yl]-[2-(5-methyl-2H-benzotriazol-4-yl)phenyl]methanone 5-chloro-2,4-difluoro-N-(2-methylphenyl)benzenesulfonamide 1-(3,5-dibromo-4-hydroxyphenyl)-2,3,5,6,7,8-hexahydro-[1]benzofuro[2,3-b]pyridine-4,9-dione 1-[2-(2,6-dioxopiperidin-3-yl)-7-hydroxy-1-oxo-4H-naphthalen-4-id-8-yl]-3-ethylurea;methanol;yttrium N-[2-[4,5-dimethyl-1-(4-methylphenyl)pyrazole-3-carbonyl]-2-azaspiro[4.4]nonan-9-yl]-4-fluorobenzamide 5-[4,6-bis(3-nitrophenyl)-1,3,5-triazin-2-yl]pyrimidine [1-(4,6-dichloropyrimidine-5-carbonyl)piperidin-4-yl]urea 6-[cyclohexa-2,4-dien-1-yl(2,6-dimethoxyphenyl)methyl]-N,N-diethylpyridine-3-carboxamide N-[4-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)phenyl]-2-fluoroethanesulfonamide 2-[1-(4,6-dimethylpyrimidin-5-yl)sulfonylpyrrolidin-3-yl]-7-propanoyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 1-[(6-methylpyridin-2-yl)amino]-3,4-dihydro-2H-1,5-naphthyridine-7-carboxylic acid 4-(7,8-dihydroisoquinolin-1-yl)phenol (5E)-2-imino-5-[(4-methoxyphenyl)methylidene]imidazolidin-4-one 5-[2-chloro-5-(trifluoromethyl)pyrimidin-4-yl]oxy-3,7a-dihydro-1H-isoindole N-(5,7,8,9-tetrahydrobenzo[b][1,4]diazepin-6-yl)propanamide 1-[3-(trifluoromethoxy)phenyl]-5,6-dihydrocyclopenta[c]pyrazole 4-[5-amino-6-(1H-pyrazol-4-yl)pyrazin-2-yl]-N,N-dimethylbenzenesulfonamide;4-[3-(3-tert-butyl-1,2-oxazol-5-yl)quinoxalin-2-yl]phenol N-(1,2-oxazol-5-yl)-3,5-bis(trifluoromethyl)benzamide N'-(3-bromo-5-methoxyphenyl)propanediamide 2-[3-(2-methylphenyl)piperazin-1-yl]-5H-pyrazolo[3,4-d]pyrimidin-6-one N-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)ethanimine;methoxymethane ethene;1-N,2-N'-di(propan-2-yl)naphthalene-2,7-disulfonamide;propane 3-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)sulfanylpiperidine-1-carboxylic acid 5-(4-chlorophenyl)-N'-hydroxypyridine-3-carboximidamide 5-cyclopropyl-4-[(4S)-6-methoxy-3,4-dihydro-2H-chromen-4-yl]pyridine-3-carbonitrile (Z)-2,3-diamino-N'-[1-[4-(trifluoromethylsulfanyl)phenyl]ethyl]prop-2-enimidamide (5-chloro-1-methyl-2,3-dihydroindol-6-yl)-cyclopropylidenemethanol 3,6-dibromo-9H-fluorene 4-N-[1-(azetidin-3-yl)ethenyl]-6-N-ethyl-2-methoxy-5,6-dimethylpyrimidine-4,6-diamine 1-[4-(6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]-2-ethoxy-2-[3-(trifluoromethyl)phenyl]ethanone 2-(benzenecarboximidoyl)-6-chloroaniline 3-(4-benzylpiperazin-1-yl)-6-methoxycarbonyl-7,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxylic acid 5-[(2R,4S)-1-acetyl-2-methylpiperidine-4-carbonyl]-N-cyclopropylfuran-3-carboxamide 1-(3-azidophenyl)-2-(ethylamino)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-one 1-[4-chloro-3-(trifluoromethyl)phenyl]-3,5,6,7-tetrahydropyrazolo[4,3-c]pyridine (E)-3-[4,5-dimethoxy-2-[2,6,12,13-tetraoxo-8-[(E)-2-phenylethenyl]dodecanoyl]phenyl]prop-2-enoic acid 2-[5-methyl-1-(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)pyrazole-4-carbonyl]oxyacetic acid 2,3-diphenyl-5-[(4-phenyl-1,3-thiazol-2-yl)methylidene]-1H-pyrazole-4-carboxamide N-[(3R,4S)-1-[6-(2-chloroethoxy)quinoline-8-carbonyl]-4-phenylpiperidin-3-yl]cyclopropanecarboxamide N-[(1R)-2,3,4,9-tetrahydro-1H-fluoren-1-yl]-5,7-dioxa-13-azatricyclo[6.5.0.02,6]trideca-1,6-diene-12-carboxamide 4-methyl-5,6,7-tripentyl-1H-benzimidazole 1-(2,4-dimethylcyclopenta-2,4-dien-1-yl)sulfanyl-3-(4-ethoxyphenoxy)benzene N-benzyl-4-[2-(3,4-dichlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]-N-ethanimidoylthiophene-2-carboximidamide 1-(5-tert-butyl-2-methoxyphenyl)pyrrolidine;ethane (2R,5R)-2-methyl-4-[3-(1H-pyrazol-4-yl)quinoline-6-carbonyl]oxy-5-[[4-(trifluoromethoxy)phenyl]methylcarbamoyl]morpholine-3-carboxylic acid 3-bromo-7-(5,6-dimethylpyridin-2-yl)-1H-indole 4-methylsulfonyl-N-(2,2,6,6-tetramethylpiperidin-1-yl)pyridin-2-amine N-[2,4-difluoro-3-(8-pyridin-3-ylimidazo[1,5-a]pyrazin-3-yl)phenyl]benzenesulfonamide 4-(3,5-diethyl-4-methoxyphenyl)pyridine;1,4-dimethylbenzene 1-methyl-5-[2-(oxolan-3-yl)ethyl]tetrazole 1-cyclobutylsulfinyl-4-(trifluoromethoxy)benzene;N-[2-oxo-5,6,7,8-tetrahydro-3H-quinazolin-4-yl]pyrrolidine-3-carboxamide 3-[2,4-dimethyl-5-(6-nitro-1H-indol-3-yl)pyrazol-3-yl]propanal 1-[2-hydroxy-4-(hydroxymethyl)phenyl]pyrrole-3-carboxamide 4-[1-(2,4-dihydroxyphenyl)-3-(trifluoromethyl)hexan-2-yl]benzenesulfonic acid N-[(Z)-1-[5-(difluoromethylsulfanyl)pyridin-2-yl]oxyprop-1-enyl]ethanimine (2E,4Z)-2-ethenyl-5-[4-methoxy-3-(methylideneamino)phenyl]hepta-2,4,6-trienamide N-[5-(3,4-dimethylcyclopenten-1-yl)pyrazin-2-yl]-6-(trifluoromethoxy)pyridine-3-carboxamide 5-(5-methoxycarbonylpyridine-3-carboximidoyl)pyrimidine-4,6-diamine 2-[(3-ethoxyphenyl)sulfonylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid 1-[2,5-difluoro-4-(trifluoromethyl)phenyl]-3-propan-2-ylidenepyrazolidine 3-[4-(6-pyridin-2-ylpyrrolo[1,2-a]quinoxalin-9-yl)phenyl]propanoic acid 1-(1,3-benzodioxol-5-yl)-N'-[2-fluoro-4-methyl-5-(trifluoromethyl)phenyl]cyclopropane-1-carboximidamide 4-[2-(3,3,3-trifluoropropanoyl)benzimidazol-1-yl]piperidine-1-carboxylic acid N-ethyl-2,3,4,5-tetrafluoro-6-(triazin-4-ylamino)benzenesulfonamide N-ethyl-2,3,4,5-tetrafluoro-6-(1H-imidazol-5-yl)aniline 6-(2,4-difluoro-3-methylphenyl)pyridine-3-carboxylate 4-[(2Z)-6,7,8-trimethoxy-3,4-dihydronaphthalen-2-yl]butanoic acid N-cyclohexyl-2-(3-cyclopropyloxyphenyl)imidazo[1,2-b]pyridazine-6-carboxamide N-[1-(3-hydroxy-4-propan-2-ylphenyl)ethylideneamino]benzenesulfonamide 2-[[1-(4-fluorophenyl)sulfonylpiperidin-3-yl]methoxy]pyrimidine 2-(1,3-benzothiazol-2-ylsulfanylmethyl)-4-methoxy-5-nitrophenol N-(2,4-difluorophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxamide N-[(E)-3-(6,8-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)prop-2-enyl]-5-phenylpentanamide 2-benzylsulfanyl-3,4-difluorophenol 2-chloro-N-[4-[(5,7-dimethyl-1H-benzimidazol-2-yl)oxy]phenyl]-3-methoxyaniline 2,6-diamino-3,4,5-tricyanobenzoic acid (2E)-2-[3-(bromomethyl)-5,6,7,8-tetrahydronaphthalen-1-ylidene]propanoic acid 2-[2-(1H-indol-4-yl)ethynyl]benzenesulfonamide 2-hydroxysulfanyl-4-[(4-oxo-3H-quinazolin-2-yl)methoxy]benzaldehyde 2-[(3,4-dichlorophenyl)methyl]-1-oxo-5,6,7,8-tetrahydroisoquinoline-4-carboxamide 2-[1-(5-azido-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carbonyl)piperidin-4-yl]-N-ethylacetamide 4-[3-[5-(1,2-dihydropyrazin-6-yl)pyridin-3-yl]oxypropyl]morpholine 5-[3-amino-2-chloro-4-(ethyliminomethyl)phenyl]-N-(3-cyanophenyl)-1,3,4-thiadiazole-2-carboxamide 2-(4-fluorophenyl)-3,5-dimethylpyridine 2-[(1S,3R)-2,3-diphenylcyclopropyl]acetic acid 1-[(3Z)-3,4-dimethoxyhepta-1,3-dien-2-yl]-4-fluorobenzene 5-(3,5-dimethylphenyl)-4H-imidazole 3-(1,2,4-triazol-1-yl)-5,6-dihydro-[1]benzoxepino[5,4-b]pyridine-9-carboxylic acid 3-[[6-[(3S)-3-aminopiperidine-1-carbonyl]pyridin-2-yl]methyl]-4,5-dihydro-1H-1,3-benzodiazepin-2-one;hydrochloride 2,4-difluoro-3-[5-(morpholin-4-ylmethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]phenol 3-[(5Z)-5-[(4-hydroxyphenyl)methylidene]cyclohexa-1,3-dien-1-yl]-N-phenylpropanamide 6-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]hexanamide 3-[1-[(6-chloropyridin-3-yl)methyl]piperidin-4-yl]oxy-5,6-diethoxypyridazine 5-butyl-2,7-dimethyl-1H-indazole 3-(1-azidoethyl)-5-chlorobenzenethiol N-[(Z)-[2,3-bis(ethenyl)cyclopropylidene]methoxy]-1-pyridin-4-ylethanimine 3-(1H-indol-4-yloxy)benzonitrile 4-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)piperazine-1-carboxylate 2-(4-chlorophenyl)sulfanyl-N'-hydroxy-6-(trifluoromethyl)pyrimidine-4-carboximidamide 2-(5-azido-1H-pyrazol-3-yl)-4-fluoroaniline 2-[5-amino-1-(4,5-difluoro-2-methoxyphenyl)pyrazole-3-carbonyl]-3,4-dichlorobenzonitrile 2-[1-azidooxy-6,7-dimethyl-3-(4-methylphenyl)naphthalen-2-yl]acetic acid 3-[[(1R)-1,2-dihydroxyethyl]amino]-2-phenylmethoxybenzonitrile [(E)-2,3-bis(2H-indazole-4-carbonylamino)prop-1-enyl]chloranium 1-[(Z)-[amino-[4-(dimethylamino)phenyl]methylidene]amino]-3-(cyclohexylmethyl)thiourea 2-(2,5-dioxopyrrolidin-1-yl)-N-[3-hydroxy-3-methyl-4-(4-phenylphenyl)butan-2-yl]acetamide;propane 1-[2-(4,5-difluoro-3,6-dihydro-2H-pyridine-1-carbonyl)cyclohexen-1-yl]-2-phenoxyethanone 3-[(2S,4R)-1-cyclopentyl-4-methoxypyrrolidin-2-yl]-5-propan-2-yl-1H-indole 1-azidooxy-2,3-dibromo-4-(1H-indol-2-yl)benzene (4S)-3,7,8-trimethoxy-5-(4-nitrophenyl)-1,2,6,10-tetrahydroazocino[1,2-a]indole [4-azido-3-(2,6-difluorophenyl)cyclohexyl]methanamine N-[2-(3,4-difluorophenyl)ethyl]-6-nitropyridine-3-carboxamide (5Z)-5-[[1-(4-methylphenyl)pyrrol-3-yl]methylidene]imidazolidine-2,4-dione 2-[5-chloro-6-(3,4-dimethoxyphenyl)pyridin-1-ium-3-yl]acetic acid 4-[2-chloro-5-(trifluoromethyl)phenyl]-N,N,3-trimethylpentanamide 5-(4,7-dihydropyrazolo[1,5-a]pyrazin-6-ylmethyl)-2H-isoquinolin-1-one;hydrochloride 4-[(2-methylpropan-2-yl)oxy]-3-phenylsulfanylphthalate 3-amino-5-(6-bromopyridin-2-yl)phenol 3-(N-methylsulfonylanilino)-N'-piperidin-4-ylidenepyridine-2-carboximidamide [(E)-2-[5-(2-chlorophenyl)furan-3-yl]ethenyl]phosphane 3-(N-(2,4-dichloropyrimidin-5-yl)anilino)propane-1,2-diol (2R)-N,4-dimethyl-1-[4-methyl-3-[(Z)-2-(methylideneamino)ethenoxy]phenyl]pentan-2-amine (5Z)-2-(4-ethylphenyl)imino-5-[(7-nitro-1,3-benzodioxol-5-yl)methylidene]-1,3-thiazolidin-4-one 5-[(3R)-1-benzylpiperidin-3-yl]sulfanyl-2H-triazole-4-carboxylic acid 2-(cyclopropylmethylamino)quinoline-4-carboxylate 4-(6,7-dimethylthieno[2,3-d]pyrimidin-4-yl)-1,5,9-trioxa-4-azaspiro[5.5]undecane;hydrochloride 2-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]-5-propoxypyridine (Z)-3-[5-chloro-2-[(4-methylcyclohexyl)amino]pyridin-4-yl]-N',5-dihydroxyhept-6-enimidamide 2-[2-(3,4-difluorophenyl)ethyl]-N-[2-(2-hydroxyethoxymethyl)-4-methylthiophen-3-yl]pyrimidine-5-carboxamide 1-(2,6-difluorophenyl)-7-[3-methylbutanoyl(methylsulfonyl)amino]-4H-chromeno[4,3-c]pyrazole-3-carboxylic acid 3-(1,2,3,4,5,6-hexahydroacenaphthylen-3-yl)-1H-imidazole-3-ium 2-bromo-N-cyclohexyl-N-pyridin-3-ylbenzamide 3-(2,5-dichlorophenyl)sulfanyl-N'-[[4-(methylideneamino)naphthalen-1-yl]diazenyl]benzenecarboximidamide;ethane 1-[(2S)-butan-2-yl]oxy-3,5-dimethylbenzene;ethane;(E)-4-hydroxyhept-3-enal (4S)-N',1-diamino-5-bromo-2-oxo-3,4-dihydroquinoline-6-carboximidamide 5-bromo-4-[(1R)-1-azidoethyl]-2-chlorophenol 3-(6-methoxypyridin-2-yl)-5-(4-phenoxyphenyl)-1,2,4-oxadiazole 4-chloro-N,6-dimethyl-5-pyridin-2-ylcyclohexa-1,3-diene-1-carboxamide [4-[4-(1,3-benzoxazol-5-yl)-2H-pyrimidine-1-carbonyl]phenyl]oxidanium 1-(2,3,4a,5-tetrahydro-1H-[1,4]oxazino[2,3-a]indol-8-yl)propan-1-one;ethane 2-[N-(carboxymethyl)-3-methylanilino]octanoic acid N-[(Z)-2-aminoethenyl]-1-cyclopropylidene-3-[4-(4-hydroxypiperidine-1-carbonyl)phenyl]iminopropan-1-imine 3-(azidomethyl)-1,1,4-triethoxy-2H-naphthalene N-[(3R,4S)-3-fluoropiperidin-4-yl]-7H-purine-6-carboxamide;hydrochloride 3-[6-(2,4,5-trimethylphenoxy)pyridin-3-yl]propanoic acid 4-[(2R)-3-hydroxy-4,5-bis(phenylmethoxy)oxolan-2-yl]-1H-pyrimidin-6-one N-(2,3-dihydro-1H-inden-5-yl)-3-phenyl-7-pyridin-4-yltriazolo[4,5-d]pyrimidin-5-amine 6-[[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]amino]pyridazine-3-carbonitrile 7-(4-acetylpiperazine-1-carbonyl)-3H-thieno[3,2-d]pyrimidin-4-one 4-(7-azido-3-ethylpyrazolo[1,5-a]pyrimidin-6-yl)morpholine 2-(2,5-dimethoxyphenyl)-7-[(3S,4R)-1-(4-fluorobenzoyl)-3-phenylpiperidine-4-carbonyl]-3H-thieno[3,2-d]pyrimidin-4-one 2-[4-(8-fluoro-5-methyl-3,4-dihydro-2H-chromen-6-yl)-1-hydroxy-3,4-dihydro-2H-quinolin-7-yl]acetamide 1-(4-acetyl-2,3-dihydroquinoxaline-1-carbonyl)-N'-hydroxy-3-methoxy-5,6-dihydropyrrolo[2,1-a]isoquinoline-8-carboximidamide 1-[2-(difluoromethoxy)phenyl]-7,8-dihydroimidazo[4,5-g]quinoline 1-[2,5-dimethoxy-4-(trifluoromethyl)phenyl]-3-[4-(6-oxo-1H-pyridin-2-yl)phenoxy]urea N-[2-[(3-aminopyridin-4-yl)methoxy]-6-piperidin-1-ylpyridin-3-yl]-N-ethyl-5-fluorothieno[2,3-d]pyrimidin-4-amine 1-[2,6-di(propan-2-yl)phenyl]-3-[5,5-bis(3-methoxyphenyl)hexa-2,4-dienylidene]urea 5-[3-(4-cyclohexylanilino)phenyl]-2,2-difluoro-1H-pyridine-4-carboxylic acid 3-[5,5-dimethyl-4-(1H-pyrrole-2-carbonyl)-6,7-dihydro-1-benzofuran-2-yl]propanoic acid N-[6-chloro-1,3-benzodioxol-5-yl]-4-(5-ethoxy-1-methyl-2-methylidenepyridin-4-yl)-1H-pyrrole-2-carboxamide (2-azido-1H-indol-5-yl)methanol N-methylsulfonyl-2,3,5-trinitrobenzenesulfonamide 6-[(2Z)-3,7-dimethylocta-2,6-dienoxy]-3-propanoyloxynaphthalene-1-carboxylic acid (2R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[2,6-di(propan-2-yl)phenoxy]hexanamide N-[4-[(6R,11bS)-3-methoxy-5-pyridin-2-yl-10b-(trifluoromethoxy)-1,2,3,5,6-pentahydropyrrolo[2,1-a]isoquinolin-9-yl]phenyl]acetamide 2-[3-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-4-propan-2-yl-1H-pyrazol-5-yl]acetamide (2S)-1,1-bis(4-hydroxyphenyl)propan-2-one;ethane 1-[2,3-di(propan-2-yloxy)phenyl]imidazolidine 7-[4-(dimethylamino)phenyl]-2-morpholin-4-yl-5,6-dihydrocyclopenta[d]pyrimidin-4-amine N'-[2,3-dimethyl-5-(4-nitrophenyl)pyrazol-1-yl]propanehydrazide N-(2,6-dibromopyridin-4-yl)-N-octylacetamide 4-[4-(5,7-dihydroxy-6-methoxyquinazolin-4-yl)piperazine-1-carbonyl]benzoic acid (2E)-N-[[4-(4-tert-butylphenyl)sulfanylphenyl]methyl]-3,7-dimethylnona-2,6,10-trienamide [(3R,5S)-2-methoxy-7,7-dimethyldecan-3-yl]benzene N-[2-(3,4-dichloroanilino)phenyl]acetamide 2-[1-azidooxy-3-(1H-inden-1-yl)naphthalen-2-yl]pyridine (3R)-3-amino-1-benzyl-3,4-dihydro-2H-quinoline-6-carbonitrile 2-[4-(N,5-dimethylanilino)pyrazol-1-yl]-3H-pyrido[2,3-d]pyrimidin-4-one 2-(5,6-dihydronaphthalen-1-yl)-7-methoxyquinoline 4-[4,7-dimethyl-5-(1-propan-2-ylsulfonylcyclopropyl)pyrrolo[3,2-d]pyrimidine-6-carbonyl]piperazine-1-carboxylic acid N-(5-bromo-6-methylpyridin-2-yl)-2-chloroacetamide 1-[3,5-dimethyl-4-(2-morpholin-4-ylethoxy)phenyl]pyrrole-2,5-dione [(3S)-1-[6-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]pyridin-3-yl]sulfonylpyrrolidin-3-yl]carbamic acid 3-methylsulfonyl-2H-indazole (5S)-2-[4-chloro-3-[2,6-dichloro-4-(trifluoromethoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]-5-(hydroxymethyl)oxolan-3-one (6S,9R)-2-amino-9-(3,4-dimethoxyphenyl)-6-(2,5-dimethoxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 5-bromo-2,3-dihydro-1H-indene;N,2-dimethylaniline 2-(4,6-difluorobenzotriazol-1-yl)-4-methyl-N-[2-oxo-3-propan-2-yl-5-(3,3,3-trifluoropropoxymethyl)-4H-1,3-thiazol-2-yl]benzenesulfonamide (2R,4S)-N-[(3-chlorophenyl)methyl]-1-formyl-4-hydroxypyrrolidine-2-carboxamide 2-[3,5-difluoro-4-(trifluoromethyl)phenyl]-6-ethoxy-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene (3S)-1-[6-(dimethylamino)-5-[2-methyl-4-[3-(oxetan-3-yloxy)azetidine-1-carbonyl]phenyl]pyridin-3-yl]piperidine-3-carboxamide (E)-2,3-diamino-N'-[4-(azepan-1-ylmethyl)phenyl]but-2-enimidamide 1,4-dibenzyl-5-chloro-3-methylidenepyrazole 3-chloro-1-methylquinoline;2-ethoxy-5-fluoropyridine 4-bromo-N-[(2R)-butan-2-yl]-5,6-diethoxypyridine-3-sulfonamide 1-(4-chlorophenyl)-5,6-dimethyl-N-[2-(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)ethyl]pyrazolo[3,4-b]pyridine-7-carboxamide 2-(2-azidoethyl)-5,6-dimethoxy-3,4-dihydrochromene 1-(4,4-dimethylpentanoyl)indole-3-carboxamide N-[2-chloro-4-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]acetamide 5-[2-ethoxy-4-(1H-pyrrol-3-yl)phenyl]-1,3-dimethylpyrazole 3-[(E)-1-(2,4-dihydroxyphenyl)propylideneamino]benzoic acid;hydrate 1-[2,4-dimethyl-3-(5-propan-2-ylfuran-2-carbonyl)phenyl]ethanone 1-[(6-chloropyridine-3-carbonyl)amino]butyl-dimethylazanium (6R)-8-oxo-3-[(4-pyridin-2-ylphenyl)sulfonylamino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 4-[1,3-dioxolan-2-ylmethyl(ethyl)amino]-N'-hydroxypyridine-2-carboximidamide 3-[(4,6-dimethylpyrimidin-2-yl)amino]benzamide [3-(1-methyl-7,8-dihydronaphthalen-2-yl)phenyl]boronic acid (NE)-N-[6-imino-2-[1-(pyridin-2-ylmethylideneamino)ethenoxy]cyclohexa-2,4-dien-1-ylidene]hydroxylamine 5-(4-phenyloxan-2-yl)-1,3,4-oxadiazol-2-amine N'-(4-bromobenzoyl)-2,3-dihydroxy-5-oxocyclohexanecarbohydrazide 1-bromo-2-ethoxy-4-[(E)-(5-fluoro-2-methylidenecyclohexyl)methylideneamino]sulfanylbenzene 7-[(2-chlorophenyl)methyl]-4,7-dihydrotetrazolo[1,5-a]pyrimidine 3-chloro-4-[(4-methylphenyl)sulfonylamino]benzoic acid 3-(2,4,6-trichlorophenyl)pyrazolo[1,5-a]pyrimidine 2-(3,5-difluoropyridin-2-yl)benzamide N-(1-amino-3,7-dimethyloctylidene)-5-[4-[2-[2-fluoroethyl(propyl)amino]ethoxy]phenyl]-6-methoxynaphthalene-2-sulfonamide 2,5-dibromo-3-(3,4-dibromophenyl)pyridine 6-[3-(5,6-dimethoxynaphthalen-2-yl)sulfonylpropoxy]-N'-hydroxyhexanimidamide 2-chloro-3-(4,5-dihydro-1H-imidazol-2-yl)benzenethiol (4R)-3,5-dimethyl-4-[5-[1-[2-(trifluoromethoxy)ethyl]pyrazol-3-yl]thiophen-2-yl]-1,3-oxazolidine 4-[3-[2-(2,2,2-trifluoroethoxy)pyridin-4-yl]imidazo[1,2-a]pyrazin-6-yl]piperazine-1-carboxylic acid 1-[1,3,7-trimethyl-5-(2-oxo-3H-1,3-benzothiazol-6-yl)pyrazolo[4,3-d]pyrimidine-8-carbonyl]piperidine-4-carboxylic acid 2-[(3aR,6aS)-5-hydroxy-1,3,3a,4,6,6a-hexahydrocyclopenta[c]pyrrole-2-carbonyl]benzonitrile;ethane (5-bromo-1,3,4-thiadiazol-2-yl)methanediol 2-[4-(1,3-benzodioxol-5-ylsulfonyl)piperazin-1-yl]-N'-hydroxypyrimidine-4-carboximidamide [2-(1,3-benzothiazol-5-yl)-5-methoxyphenyl]boronic acid N-[2,4-difluoro-3-(3-imidazo[1,2-a]pyrazin-6-ylpropoxy)phenyl]formamide 2-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-4-oxo-3H-quinazoline-6-carboxamide 1-(6,7-dimethoxyquinolin-4-yl)-N'-pyridin-2-ylpiperidine-4-carbohydrazide 6-amino-2-(4-cyclohexylanilino)-3H-quinazolin-4-one N-[5-[6-fluoro-3-[4-(2-methylphenyl)-1H-imidazo[4,5-c]pyridin-2-yl]-1H-indazol-5-yl]pyridin-3-yl]benzamide N-(1,2,3,5,6,7-hexahydropyrrolizin-8-ylmethyl)-6H-cyclohepta[d][1,3]thiazol-2-amine N-[4-(methylamino)phenyl]benzamide;hydrochloride 1-[2,5-dichloro-3-(propylsulfanylamino)phenyl]ethanethiol N-benzyl-3,3-diphenylpropanamide N-[4,5-difluoro-2-(1-methoxypropyl)phenyl]propanethioamide (2R)-N-[[3-methoxy-4-[4-(trifluoromethyl)phenoxy]phenyl]methyl]pyrrolidine-2-carboxamide 1-(3,5-dimethylphenyl)-N-[2-(3-oxo-4H-quinoxalin-2-yl)-3H-benzimidazol-5-yl]cyclopropane-1-carboxamide 2-(4,6-dimethylpyrimidin-5-yl)-5-iodo-4-propan-2-yl-1H-pyrimidin-6-one 2-[(5R,10bR)-9-chloro-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 4-[(3,5-dichloro-2-ethylimidazo[1,2-a]pyridin-7-yl)amino]-N-(2-fluorophenyl)-5-methoxypyrrolo[1,2-b]pyridazine-6-carboxamide 2-methyl-N-[[5-(3-phenylphenyl)pyridin-2-yl]methylideneamino]aniline 1-phenyl-2,3-diazaspiro[4.5]decan-4-one 5-[(3-bromophenyl)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine N-[3-(ethoxymethyl)phenyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide 2-[3-fluoro-6-methyl-4-(trifluoromethoxy)cyclohexa-1,3-dien-1-yl]-5-methylthiophene ethane;2-ethoxy-3,4,5,6-tetramethylbenzoate (E,1Z)-1-[(2S)-3-cyclopentyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-2,3'-pyrrolidine]-1'-ylidene]hex-2-en-2-ol 2-ethylpentanal;methoxymethane;N-[(E)-1,3,4-trimethylidenecyclohexa-1,5-dien-1-yl]-9H-fluorene-2-carboxamide 2-(6-methylcyclohexa-1,3-dien-5-yn-1-yl)dibenzofuran N-methoxy-1-[6-(4-morpholin-4-ylpiperidine-1-carbonyl)pyridin-3-yl]cyclopropane-1-carboxamide N-[4-(methylsulfamoyl)phenyl]-1-[1-(1,3-thiazol-2-ylamino)cyclopropanecarbonyl]pyrrolidine-2-carboxamide 2-(2,4-difluorophenyl)-5-[4-(2-iodoacetyl)oxyphenyl]pyrrole-1-carboxylate 3-bromo-4-hydroxy-N-[[1-(trifluoromethyl)cyclopropyl]methoxy]benzamide N-(2,6-dimethylphenyl)-4-[[(1S,5R)-7-ethyl-3-azabicyclo[3.1.0]hexan-3-yl]sulfonyl]benzamide N-(2,5-dichlorophenyl)-1-[4-(3,4-difluorophenyl)-6-methylpyridin-2-yl]ethanimine 3-[4-amino-1-[(2R,5S)-4-propan-2-yloxy-6-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]heptan-2-yl]pyrazolo[3,4-d]pyrimidin-3-yl]-N'-hydroxybenzenecarboximidamide 2-(2,6-dioxopiperidin-3-yl)-4-[methyl-[1-(2H-triazol-4-yl)propan-2-yl]amino]isoindole-1,3-dione 5-cyclobutyloxy-3,4,6-trimethylpyridine-2-carboxamide 6-(3-fluoropyridin-4-yl)oxy-N-phenylisoquinolin-1-amine (5Z)-N,N-dimethyl-4,9b-dihydro-1H-azeto[2,3-a]indole-6-carboxamide;ethane N-[(2,3-difluorophenyl)methyl]-3-hydroxybutanamide N-[(1E)-2-cyanobuta-1,3-dienyl]sulfonyl-4-nitrobenzamide 3-[(2S)-2-azidooxypropyl]-4,5,6,7-tetrahydro-1H-indazole 5-[[1-[(4-fluoro-2,6-dimethylphenyl)methyl]piperidin-3-yl]methoxy]pyridazine [5-amino-1-[4-fluoro-2-(trifluoromethyl)phenyl]pyrazol-3-yl]-pyridin-3-ylazanium 2-[3,4-bis(ethenyl)anilino]acetic acid N-[5,6-dimethyl-1-(2-morpholin-4-ylethoxy)benzimidazol-2-yl]butanamide (1S)-2,2,2-trifluoro-N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]cyclopentane-1-carboxamide N-(3,5-dimethylphenyl)-2-hydroxyiminopropanamide 3-[(3,5-dimethylbenzoyl)amino]pyrrolidine-1-carboxylate 1-[4-[6-chloro-5-(2,3-dimethoxyphenyl)-8-fluoro-4H-quinazolin-3-yl]piperidin-1-yl]prop-2-en-1-one 6-[3-(4-tert-butylphenoxy)propoxy]chromen-2-one 1-[4-fluoro-2-methoxy-6-(4,5,7-trifluorocyclohepta-1,3,5-trien-1-yl)phenyl]ethanol 2-(2-methylbutanoyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carbonitrile N-(2,5-difluorophenyl)sulfanyl-6-methoxyquinoline-3-carboxamide 4-benzyl-5-[(3-ethoxyphenyl)methoxy]-3H-1,3-oxazol-2-one 2-amino-N'-(4-anilinophenyl)-6-hydroxy-5-oxo-7,8-dihydroquinoline-3-carboximidamide 6-azidooxynaphthalene-1,2,3-tricarbonitrile 2-(3,4-dichlorophenyl)-6-[5-fluoro-6-(4-methylpiperazin-1-yl)pyridine-3-carbonyl]cyclohepta-2,4-diene-1,1-dicarboxylic acid N-azido-4-(furan-2-yl)pyrimidin-2-amine 4-[4-methoxy-3,5-bis(2-methylbutanoyl)phenyl]piperidine-1-carboxylic acid 3-azido-1,5-bis[(2-chlorophenyl)methyl]-9H-pyrido[2,3-b]indole (2S)-2-[[(1R,3aR,7aS)-5-cyclohexa-2,4-dien-1-yl-1-[[4-(trifluoromethoxy)phenyl]methyl]-3,3a,4,6,7,7a-hexahydro-1H-pyrrolo[3,4-c]pyridine-2-carbonyl]amino]propanoic acid 2-ethylhexanoic acid;[2-(3-methoxyphenyl)-5,6,7,8-tetrahydroquinazolin-4-yl]-pyrrolidin-1-ylmethanone 1-[3,4-dihydroxy-5-(trifluoromethyl)phenyl]pent-2-yn-1-one 2-[3,4-bis(phenylmethoxy)phenyl]-N-pyridin-3-ylacetamide 5-bromo-2-methylpyridine;ethane 2,4-dioxo-5-propan-2-yloxycarbonyl-1H-pyrimidine-6-carboxylic acid 1-[5-[(4S)-2,8-diazabicyclo[6.2.0]decan-8-yl]pyrazin-2-yl]oxy-3,3,5-trimethylhexan-2-one 3-methyl-2-[[5-[(E)-1,3,3-trideuterio-2-phenylprop-1-enyl]thiophene-2-carbonyl]amino]butanoic acid N-[(1S)-4,6-difluoro-2,3-dihydro-1H-inden-1-yl]-6-methoxypyrazolo[1,5-a]pyridine-2-carboxamide 2-(4-fluorophenyl)-N,1-dimethyl-5-[3-oxo-7-(3-thiomorpholin-4-ylpropoxy)-2-thiophen-2-yl-1H-isoindol-1-yl]-6H-pyrrolo[3,2-b]azepine-3-carboxamide (4-ethoxyphenyl)-oxo-[(2S,3R)-1H-1-pyrrole-3-carbonyl]azanium 2-[2-(dimethylamino)propyl]-6-(4-ethoxyphenyl)-3H-thieno[3,2-d]pyrimidin-4-one 1-[4-[(Z)-3-amino-4,5,5,6,7,8,9-heptamethylnon-2-enoxy]phenyl]ethanone 7-chloro-1-(2,3-dihydro-1H-indol-5-ylmethyl)-3-nitrosoindol-2-ol [5-(4,6-diphenyl-1,3,5-triazin-2-yl)cyclohexa-2,4-dien-1-ylidene]-[2-[2-[methyl-(4-methylphenyl)hydrazinylidene]ethoxy]ethylimino]azanium 6-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]-3H-1,3-benzothiazol-2-one 2,4-dioxo-6-[3-(trifluoromethyl)phenyl]-1,3-diazinane-5-carbonitrile (3S,5R)-1-[8-[(E)-4-(4-methylpiperazin-1-yl)but-2-en-2-yl]quinolin-7-yl]-3,5-dipropylpyrrolidin-2-one 1-(3,5-dimethylphenyl)-4-[4-(6-fluoroquinolin-2-yl)phenyl]pentan-3-one N-[1-(2,4-dihydroxyphenyl)ethylideneamino]isoquinoline-3-carboxamide N-(1,4-dioxan-2-ylmethyl)pyrimidine-5-carboxamide 2-(5-chlorothiophen-3-yl)-7,8-difluoroquinoxaline 1-methyl-3-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonylamino)phenyl]urea 4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]-N'-hydroxypyridine-2-carboximidamide 3-(1,2,4-triazol-1-yl)-2-[4-(trifluoromethoxy)phenyl]-6H-pyrido[1,2-a]pyrimidine 1-[(E)-[5,6-dichloro-3-(ethoxymethyl)indol-2-ylidene]amino]-N-methylmethanamine;uranium(2+) 1-[3-(2,3-dihydro-1H-inden-5-yl)propyl]pyrrolidine;4-methoxybenzamide 2-ethylsulfanyl-4-(methylamino)pyrimidine-5-carboxylic acid 2-[5-[(4R)-1,3-dimethyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]furan-2-yl]acetic acid 3-[(4,5-dichlorocyclohexa-2,4-dien-1-yl)methoxy]-N-[1-[5-(ethoxycarbamoyl)-6-oxo-1H-pyridazin-4-yl]piperidin-4-yl]azetidine-1-carboxamide 2-chloro-N-[(Z)-(4-hydroxyphenyl)methylideneamino]benzamide 4-methyl-2,3-dimethylidene-5-(5-propan-2-ylpyridin-2-yl)pentanenitrile [2-chloro-4-(trifluoromethoxy)phenyl]-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]methanone [(2S,4R)-1-benzylsulfonyl-4-hydroxy-5-(hydroxymethyl)pyrrolidin-2-yl]-phenylmethanone 2-[(3S)-6,7-dimethoxy-4-oxo-3-[[4-[phenyl-[4-[(E)-2-phenylethenyl]benzoyl]amino]phenyl]sulfonylcarbamoylamino]heptanoic acid (3S)-7-amino-6-fluoro-5-hydroxy-2,3-dihydrobenzo[g][1]benzofuran-9-carboxylic acid N-(2,3-dihydroxypropyl)-4-[5-(trifluoromethoxy)pyridin-2-yl]piperazine-1-carboxamide 2-[3-(trifluoromethyl)phenoxy]-N,4-di(propan-2-yl)aniline N-methyl-2-[4-[3-(trifluoromethoxy)phenyl]cyclohexa-1,5-dien-1-yl]ethanamine 4-(1,2-dimethylimidazol-4-yl)sulfonyl-N-propan-2-ylmorpholine-3-carboxamide (6-azido-1-benzothiophen-3-yl)-[5-(1H-pyrazol-4-yloxymethyl)furan-2-yl]methanone 4-[(6,7-dimethoxyquinolin-4-yl)amino]piperidine-1-carboxylic acid 3-(3-methylnaphthalen-2-yl)benzene-1,2-diol 1-phenyl-3-[[4-(piperidine-1-carbonyl)cyclohexa-2,4-dien-1-yl]methoxy]quinolin-4-one 3-methyl-4-[(6-methylpyridin-2-yl)amino]butanenitrile (2R)-N-[4,5-bis(ethenyl)-1H-imidazol-2-yl]-3,3-dimethylbutanamide N-[(Z)-1H-indol-3-ylmethylideneamino]quinoline-6-carboxamide 5-[4-(5-fluorothiophene-2-carbonyl)piperazin-1-yl]sulfonylisoquinoline-1-carbonitrile 4-(6,6-dimethyl-1,4,5,7-tetrahydroindazole-3-carbonyl)-1,3-thiazole-2-sulfonamide 6-methoxy-2-[(3R)-piperidin-3-yl]-1,3-benzoxazole 3-(6-bromopyridin-2-yl)benzene-1,2-diol 5-chloro-2-[3-[(E)-2-nitroethenyl]sulfonylpropyl]pyridine 2,4-diaminopteridine-7-carboxylate 3-amino-1-[4-(2-butan-2-ylphenoxy)phenyl]propane-1,3-dione 2,3-dimethyl-1H-indole;ethane;1-methylsulfinyl-4-[(E)-2-phenylethenyl]benzene N-butyl-3-[4,7-dimethoxy-2-oxo-1-(4-phenylcyclohexa-2,4-dien-1-ylidene)azepan-3-yl]propanamide 5-[2-hydroxy-3-(2,4,6-trimethylphenoxy)propyl]-1,3-oxazolidine-2,4-dione 4-(2-aminoethyl)-1,3-dimethyl-7H-pyrazolo[3,4-b]pyridine-5-thione N-[(4-fluorophenyl)methyl]-1-methoxy-5-methylcyclohexa-2,4-diene-1-carboxamide 2-(1-cyclohexyloxyethoxy)-5-methanimidoylaniline 2-[1-(4,5-dihydropyrimidin-6-yl)-3,5-diphenylpyrazol-4-yl]pyridine (2S)-1-(3,5-difluorobenzoyl)pyrrolidine-2-carboxylic acid;ethane 1-(3,5-dimethoxyphenyl)pyrrolidine;N'-[6-oxo-2-(2-propanoylhydrazinyl)-4,5-dihydropyrimidin-1-yl]-2-pyrazol-1-ylethanimidamide N-[2-(1-ethylpiperidin-3-yl)indazol-5-yl]-6-[[2-(4-fluorophenyl)acetyl]amino]pyridine-3-carboxamide 3-(2,5-dimethoxyphenyl)-7-[3-[4-[(dimethylamino)methyl]piperidin-1-yl]propylamino]-5-methylthieno[3,2-c]quinolin-4-one 2-[5-amino-3-cyano-4-(4-morpholin-4-ylphenyl)-6,7-dihydropyrazolo[1,5-a]pyridin-7-yl]acetamide 3-ethylpentane;2,7,9-trimethylfluoren-1-amine N-[4-(chloromethyl)phenyl]sulfanyl-3,5-difluoroaniline N-[3-(2,4-difluorophenyl)propyl]-5-[5-(triazol-1-ylmethyl)furan-2-yl]-1H-pyrazole-4-carboxamide N-[[1-[4-(difluoromethoxy)-3,5-diethylphenyl]sulfonylpiperidin-4-yl]methyl]ethenesulfonamide 1-[(3R,4S)-3-fluoropiperidine-4-carbonyl]-5,7-dimethyl-2H-pyrido[3,4-b]pyrazin-3-one 2-[6,7-dichloro-3-methyl-4-(4-propan-2-ylphenyl)sulfonylnaphthalen-1-yl]oxyacetic acid 2-amino-9H-thioxanthene-1,6-diol 6-ethyl-2,5-dimethoxy-4-phenyl-3H-1,2-thiazole 2-[5-ethyl-4-(4-hydroxy-3-methoxyphenyl)-2,6-dioxo-1,3,5-triazin-1-ium-3-yl]acetic acid N-[4-hydroxy-3-(5,6,7,8-tetrahydronaphthalen-2-yloxy)phenyl]-4-[2-[methyl(propanoyl)amino]ethylsulfamoyl]benzamide 3-(2,3-dihydro-1H-inden-5-yloxy)-N'-hydroxypyridine-4-carboximidamide 5-[(2R)-4-[6-chloro-3-cyclohexyl-1-(oxetan-3-ylmethyl)indol-2-yl]-2-methylbutanoyl]pyridine-3-carboxylic acid 2-[2,4-dihydroxy-6-[(1S)-3-hydroxycyclohexyl]phenyl]acetic acid 2-methyl-4,6-dimorpholin-4-ylpyridin-3-amine N-cyclohexyl-5,6-dimethylthieno[2,3-d]pyrimidine-4-carboxamide 5-butyl-2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]pyrimidine [2-amino-4-(2,6-difluorophenyl)-5-methylpyrrol-1-ium-3-ylidene]carbamic acid 2,3-dimethyl-2-phenyl-3H-pyridine N-[3-fluoro-5-[2-[5-[5-(pyrrolidin-1-ylmethyl)pyridin-3-yl]-1H-pyrazolo[4,3-b]pyridin-3-yl]-7-thiophen-2-yl-1H-imidazo[4,5-c]pyridin-4-yl]phenyl]-N',N'-dimethylethane-1,2-diamine 2-[2-(2,3-dihydropyridine-4-carbonyl)pyrrolidin-1-yl]-5-fluoropyridine-3-carboxamide N-azido-2-(5-methylpyridin-3-yl)oxyethanamine 1-[3,5-bis(trifluoromethyl)phenyl]-N'-methanimidoylbutane-1,4-diamine 3,5-dichlorobenzenethiol;2-[4-(pyrrolidin-1-ylmethyl)phenyl]pyridine 3-(5,7-dibromonaphthalen-1-yl)-2-methoxycarbonylprop-2-enoate 2-[(7-amino-6,8-dibromopurin-9-yl)methyl]propanedioic acid 2-chloro-N-(4-ethylphenyl)-1,3-benzothiazole-6-carboxamide (5E)-2-cyclohexylimino-5-[(4-hydroxyphenyl)methylidene]-1,3-thiazolidin-4-one 3-(5-methylcyclohepta-1,4,6-trien-1-yl)-7,8-dihydroimidazo[1,2-a]pyrimidine N-(3,5-dimethoxyphenyl)-4-[3-(pyridin-4-ylmethoxy)anilino]quinazoline-8-carboxamide 4-amino-1H-pyrimidin-6-one;7-[3,5-difluoro-2-(tetrazol-2-yl)anilino]-N'-[2-ethylpentanoyl(methyl)amino]thieno[3,2-b]pyridine-5-carbohydrazide 5-[2-(3,4-dichlorophenyl)-1,3-thiazol-4-yl]-3H-thieno[3,2-b]pyran-7-one 6-[(2R)-4-ethylmorpholin-2-yl]pyrimidine-4,5-diamine 3-[2,6-dimethyl-4-(1H-pyrrole-3-carbonyl)piperazin-1-yl]propanenitrile 3-[5-(3,4,5-trifluorophenyl)sulfanylpentoxy]propanenitrile 4-[2,5-dimethyl-3-(propylamino)phenyl]pentanal 2-chloro-N-[4-fluoro-3-[3-(piperidine-1-carbonyl)quinolin-6-yl]phenyl]benzenesulfonamide N-[(3R,7S,8aS)-3-cyclopropyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-3,5-dimethoxybenzamide 2-[4,5-bis(ethenyl)-1,3-thiazol-2-yl]acetaldehyde;(E)-2-methanimidoylpent-3-enenitrile 2-[(4-chlorophenyl)methylsulfanyl]-N-[6,7-dichloro-3-[2-(3,5-dihydroxypyrrolidin-1-yl)ethyl]-2H-indazol-5-yl]-2-pyridin-3-ylacetamide 6-(4,4,5,5-tetramethyloxaborolan-2-yl)-N,3-dihydro-1H-inden-2-imine 4-(3-chloropyridin-2-yl)oxycyclohexan-1-ol 1-(4,6-difluoropyridine-3-carbonyl)-N,5-dimethylpyrrolidine-2-carboxamide N-[(3S,4R)-1-cyclopentyl-4-(dimethylsulfamoylamino)pyrrolidin-3-yl]-2-fluorobenzamide 5-azido-2-(trifluoromethyl)benzenesulfonamide N-azido-2,4-dimethylbenzenesulfonamide N'-(benzenecarboximidoyl)propanediamide 1-[(3R,4S)-4-methylpyrrolidin-3-yl]oxybenzotriazole-5-carboxylic acid;hydrochloride N-(4-tert-butylphenyl)-2,3-dihydrofuran-5-carboxamide 5-[(3R,4S)-3-benzyl-4-methoxypyrrolidine-1-carbonyl]-6-hydroxy-1H-quinolin-2-one (3R)-1,4'-dimethylspiro[2H-indole-3,5'-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine]-5-one;3,4-diethylbenzaldehyde 1-(4-methoxyphenyl)-3-[(Z)-3,5,6-trihydroxyhexan-2-ylideneamino]urea 1-[2,5-dichloro-N-(4-hydroxybutyl)anilino]propan-2-one 5-[3-chloro-4-(4-oxopentanoylamino)phenyl]-1,2-oxazole-3-carboxylic acid (3S,5R)-4-[2-methoxyethyl-[4-(5,6,7,8-tetrahydroquinolin-8-ylamino)butyl]amino]-3,5-dimethylcyclohexan-1-one 3-(1,1-difluoroethyl)-N-[2,6-di(propan-2-yl)phenyl]aniline [2,6-dimethyl-4-(2-pyridin-3-ylethynyl)phenyl]boronic acid 7-fluoro-N'-hydroxy-3-[(1R,5S)-3-oxabicyclo[3.2.0]heptan-6-yl]quinoxaline-6-carboximidamide 2-amino-N-[1-(3-azidopropylamino)-3-hydroxy-1-oxopentan-2-yl]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamide [3-(6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl)cyclopentyl]-pyrrolidin-1-ylmethanone 2-(4,6-dichloropyrimidin-5-yl)ethanamine (2S,5R)-5-benzyl-N-[3-cyano-6-(4-methoxyphenyl)pyridin-2-yl]pyrrolidine-2-carboxamide 5-[2,3,4-tris(ethenyl)pyrrol-1-yl]pyridine-2-carbonitrile (5R,7S)-3-bromo-N-[4-chloro-2-(2H-tetrazol-5-yl)phenyl]-5-(trifluoromethyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide N-[2-(diethylamino)propyl]-1'-methylspiro[4,5-dihydrothieno[2,3-c]pyran-7,4'-piperidine]-2-carboxamide;2,2,2-trifluoroacetic acid 2-[1-(azetidin-3-yl)-5-ethoxyindole-7-carbonyl]cyclohexane-1,4-dione N'-(2,4,6-trichlorophenyl)butanediamide 5-[4-chlorobutyl(hexadecanoyl)amino]naphthalene-2-sulfonic acid 4-[(1,2-dimethylcyclohexylamino)carbamoyl]benzoic acid N-[5,6,7-trichloro-2-hydroxy-1-(3-methylbutoxy)naphthalen-1-yl]acetamide (5S)-2,9-dimethyl-1-oxo-N-[2-(pyridine-3-carbonylamino)ethyl]-6-oxa-2,10-diazaspiro[4.6]undecane-10-carboxamide N-(1,3-benzothiazol-5-yl)-1-cyclohexa-2,4-dien-1-ylcyclopropane-1-carboxamide 1,6-bis(3,5-dimethylpyrazol-1-yl)-4-methoxyacridine 1-azidooxy-2,4,5-trichloro-3-(2,6-dimethylphenoxy)benzene 2-[4-fluoro-2-(trifluoromethyl)phenyl]imino-5,6-dimethoxyindene-1,3-dione 3-[2-(2,3-difluorophenyl)pyrrolidine-1-carboximidoyl]-5-methylbenzamide 1-(3-bromophenyl)sulfonyl-5,8-dihydroxyquinolin-4-one (4Z)-2-methylhepta-1,3,5-triene;6-[3-oxobutyl(prop-2-enoxycarbonyl)amino]naphthalene-2-carboxylic acid 6-amino-1,3-dimethyl-4-(3-nitrophenyl)quinolin-2-one 5-[1-[5-fluoro-2,3-dimethoxy-6-(3-phenylcyclobutyl)indol-1-yl]ethyl]thiophene-2-carboxylate 2-methyl-6-propan-2-ylidene-N-(1,1,3-trimethylbenzo[e]indol-2-ylidene)cyclohexa-2,4-dien-1-imine 1-[3,4-di(propan-2-yl)phenyl]-4-ethylpiperazine;ethane 2-[4-[4-[[6-fluoro-2,3-dihydro-1H-inden-5-yl(hydroxy)methylidene]amino]phenoxy]phenoxy]-N,N-dimethylacetamide 2-[(3R,4S)-3-fluoropiperidin-4-yl]sulfanylpyridine (2S,4R)-1-[2-[[(2S)-2-aminobutanoyl]amino]benzoyl]-N-methyl-4-phenylpyrrolidine-2-carboxamide;hydrochloride 2-(3,4-dimethoxyphenyl)benzaldehyde 4-[3,5-dimethyl-1-(oxan-2-yl)pyrazol-4-yl]sulfonylbenzonitrile 1-[(4aS)-6,6-difluoro-1-methyl-2,3,4a,5,7,8,9,10,11,12b-decahydrobenzo[g]isoquinolin-1-ium-4-yl]ethenamine N-(1-azidobutan-2-yl)-6-(4,5-dihydro-1H-imidazol-2-ylmethoxy)naphthalene-2-carboxamide 5-[4-(2,3-difluorophenyl)piperazine-1-carbonyl]pyridine-2-carbonitrile 5-[2-(2,6-dichlorophenyl)ethyl]-4H-imidazole 3-(2,5-diaminophenoxy)-N-phenylaniline 2-(4,5-diamino-1H-pyrazol-3-yl)benzenesulfonate N-(1H-indazol-6-yl)pyrazine-2-carboxamide 2-[3-(difluoromethoxy)phenyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-5-carboxamide 3-[2-(4-methoxyphenyl)ethyl]-5-(1H-pyrazol-4-yl)pyridine 6-methyl-2,5-diphenyl-3,4-dihydropyridine 2-amino-6-[3,5-difluoro-4-(1-hydroxyethyl)phenyl]-9-(4-fluoropyridin-3-yl)-5,7,8,10-tetrahydropyrido[4,3-b]azocine-3-carbonitrile 5-[1-(2,3,4,6-tetrachlorophenyl)butylideneamino]pyridine-2-carbonitrile 3-azido-5,8-dichloronaphthalene 2-methylpropane;N'-[(2E,5Z)-4,6,9,15-tetramethoxy-11-oxohexadeca-2,5-dienyl]benzenecarboximidamide 3-methylsulfinylspiro[1,2-dihydroindole-4,5'-piperidine];2-(1,2-oxazol-3-yl)propan-2-amine 1-azido-4-(2,4-dibromophenoxy)benzene 4-[6-(2-aminopropylamino)pyrimidin-4-yl]benzonitrile 2-[4-(dimethylamino)-N-ethylsulfonylanilino]acetamide 2-azido-4-(3,5-dichlorophenyl)furan 5-fluoro-N,2-dimethyl-6H-pyrido[3,4-e][1,4]oxazepin-7-amine (5Z)-2-(3,4-dimethylphenyl)imino-5-[[7-fluoro-1-hydroxy-8-[(3-hydroxyphenyl)sulfanylamino]isoquinolin-6-yl]methylidene]-1,3-thiazolidin-4-one 6-methylsulfonyl-N-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyridine-3-carboxamide 2-azido-4-methoxy-3,6-diphenylpyridine 4-[2,5-bis(trifluoromethyl)phenyl]-N-ethoxyaniline N-(4-fluorophenyl)-1-(3-methylquinoxalin-2-yl)pyrazole-3-carboxamide 6,7-dichloro-1'-(4-methylnaphthalene-2-carbonyl)spiro[3H-chromene-2,4'-piperidine]-4-one 3-[6-(cyclopropylmethylamino)pyrimidin-4-yl]imidazo[1,2-a]pyridine-7-carbonitrile 2-(2,6-dioxopiperidin-3-yl)-4-[2-hydroxyethyl(methyl)amino]isoindole-1,3-dione N-[4-(4-chlorophenoxy)phenyl]-2,3-dihydroindole-1-carboxamide (4R)-4-cyclohexyl-N-[1-oxo-3-phenyl-1-[2-[[5-(trifluoromethyl)pyridin-3-yl]amino]ethylamino]propan-2-yl]pentanamide;formic acid (1S)-2-[4-(difluoromethylsulfonyl)phenyl]cyclopropane-1-carbonitrile 5-methyl-N-[(E)-3,4,5-trihydroxy-6-oxohex-1-enyl]pyridine-2-carboxamide 2-[4-(hydroxymethyl)phenyl]-N,5-dimethoxybenzamide N-[4-(dimethylamino)phenyl]-2-[2,6-dimethyl-1-[5-[[2-(oxetan-3-yloxy)acetyl]amino]pyrimidin-2-yl]piperidin-4-ylidene]propanamide 2,2-dimethylbutane;ethanimine;N-[4-(3-methoxypyridin-2-yl)oxycyclohexa-1,5-dien-1-yl]sulfanyl-5-(trifluoromethyl)pyrimidin-2-amine 1-methylsulfonyl-2,3,4,6-tetrahydroazepino[4,5-b]indole N-[2-(diethylamino)ethyl]-3-[5,6-dimethoxy-1'-(thiophen-2-ylmethyl)spiro[1H-indole-3,4'-piperidine]-2-yl]benzenesulfonamide;2,2,2-trifluoroacetic acid 5-[4-(3-methoxyphenyl)piperazine-1-carbonyl]thiophene-2-carboxylic acid N-[4-methyl-2,6-di(propan-2-yl)phenyl]-1-[3-[2-[(2S)-oxolane-2-carbonyl]-3H-pyrrole-5-carboximidoyl]-5-(trifluoromethoxy)phenyl]methanesulfonamide N-[(Z)-1-(4-hydroxyphenyl)ethylideneamino]benzenesulfonamide 6,7-dihydroxy-5-nitrosochromene-2-thione 2-[3,4-dimethyl-1-(2,2,2-trifluoroethyl)cyclohexa-2,4-dien-1-yl]oxynaphthalene 1-(5,6-dimethoxypyridin-3-yl)-7H-imidazo[4,5-c]quinoline 2-(4-azidooxyphenyl)-1,3-benzothiazole N-ethyl-2-[4-[6-(1H-pyrazol-5-ylamino)naphthalen-2-yl]oxyphenyl]acetamide 2-(5-ethyl-3,4-dimethoxycyclohexa-1,3-dien-1-yl)pyridine 2-amino-6,7,8-trimethylquinoline-3-carboxylic acid 2-(methylamino)-4-[6-[5-[3-oxo-2-[1,2,4]triazolo[4,3-a]pyridin-6-yl-2,7-naphthyridin-8-yl]thiophen-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1-carboxylic acid 4-[3-(dimethylamino)pyrrolidine-1-carbonyl]-2,6-difluorobenzonitrile N-[3-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide 5-fluoro-3,3-dimethyl-6-(4-methylphenyl)-1H-indol-2-one (3S,5R)-1-[[4-(2,5-dimethylthiophen-3-yl)phenyl]methyl]-3,5-bis(4-fluorophenyl)piperazine 4-N,6-diethyl-2-[(4-phenylphenyl)methylsulfanyl]pyrimidine-4,5-diamine 5-(3,4-difluorophenyl)-2-oxoimidazolidine-1-carboxamide 3-[2,4-dichloro-6-(trifluoromethyl)anilino]-1-phenylpyrrolidine-2,5-dione 1-[2-(4-methylphenyl)ethenoxy]-N,N-bis(sulfanyl)ethenamine 2-(dimethylamino)-N-[1,3-thiazol-4-yl]pyridine-3-carboxamide N-[4-(3,5-dimethoxyphenyl)pyridin-2-yl]benzenesulfonamide 3-(1H-indol-4-yl)-2-methylpropanamide (3S,4R)-1-[2-cyclopropyl-6-(1H-indol-5-ylmethoxy)pyrimidin-4-yl]-4-fluoropyrrolidine-3-carboxamide 4-chloro-6,8-difluoro-7-[2-methyl-1-(oxan-2-yloxy)propan-2-yl]quinoline (1-acetamidocyclopropyl)methane;3-aminobenzaldehyde;2,4,6-trimethoxy-N-methylaniline 1-[3-fluoro-4-(trifluoromethyl)phenyl]cycloheptane-1,3-diol 2-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-N-pyrimidin-2-ylacetamide N-cyclohexyl-4-ethenyl-3-methylbenzenesulfonamide 1-[2,5-di(propan-2-yl)pyrazol-3-yl]-N-(2-ethylsulfanyl-6-methoxypyridin-4-yl)isoquinoline-7-carboxamide;ethane 3-[[4-azidooxy-2-(9H-fluoren-1-yl)phenyl]methyl]pyridine 4-(2-methylphenyl)-3-[(2,5,6-trifluorocyclohexa-1,3-dien-1-yl)methyl]pyridine 1-(2,6-diethylphenyl)-3,5,7,8-tetrahydro-2H-imidazo[4,5-f]quinoline 5-[4-(2,5-dioxopyrrolidin-1-yl)phenyl]pentanoic acid N-[(1S)-2-cyanocyclohexyl]-4-(7H-pyrrolo[3,2-d]pyrimidin-4-ylamino)benzenesulfonamide 2-[4-(3,5-dimethylbenzoyl)phenyl]sulfanylacetic acid N'-hydroxy-3-[(5-propyl-1,2-oxazol-3-yl)oxy]pyrazine-2-carboximidamide (2S)-2-(phenylmethoxycarbonylamino)pentanoic acid 6-bromo-N-[4-(tert-butylcarbamoyl)phenyl]-1H-indole-2-carboxamide 2-[(3R)-5-(4-chlorophenyl)-6-oxo-1-pentan-2-ylpiperidin-3-yl]-N-[(1S,2R)-1-hydroxy-1,3-dimethoxypropan-2-yl]acetamide 4-[3-[(6R)-3-amino-2,5,5a,7-tetrahydrooxepino[2,3-b]pyridine-6-carbonyl]phenyl]piperazin-2-one 5-chloro-3,4-difluoro-N-[[(2R)-oxolan-2-yl]methyl]benzamide 2-methylbutane;3-[4-(3,4,5-trifluorophenyl)phenyl]propanoic acid N-(1,5-dimethylpyrazol-4-yl)sulfonyl-2-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetamide 1-[2,6-dichloro-4-(trifluoromethyl)phenoxy]propan-1-amine [2-azidooxy-3,4-dichloro-6-(trifluoromethyl)phenyl]urea [(1S)-4-fluorocyclohexa-2,4-dien-1-yl]methanol;N-(5-piperazin-1-ylpyridin-3-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-cyano-2-methoxy-6-(pyrazol-1-ylmethyl)phenyl]-2-ethoxyacetamide 6-cyclohexyloxy-3,4-dihydroindeno[1,2-d]pyrimidine N-cyclohexyl-2-[3-[(1S)-5,7-dichloro-2,3-dihydro-1H-inden-1-yl]propanoylamino]-4-phenylbenzamide 3,5-dichloro-N-[[2-[(1R)-3-[methyl(propan-2-yl)amino]cyclopentyl]oxypyridin-4-yl]methylideneamino]aniline [4-chloro-1-(oxan-2-yl)indazol-6-yl]-morpholin-4-ylmethanone (3E)-4-amino-3-[[5-chloro-2-(tetrazol-1-yl)phenyl]methylidene]azete-2-thione 5-(4-fluorophenyl)-2,3,4,6,7,8-hexahydroquinoline 4-[5-(2-chloro-6-methylphenoxy)pentyl]morpholine 3-(4-fluorophenyl)-1,6-bis(4-methoxypyrimidin-2-yl)pyrazolo[3,4-d]pyrimidine 5-chloro-2-N-[4-(3-piperidin-1-ylpropoxy)phenyl]-7H-purine-2,8-diamine;2-methylpropane (3R,4R)-1-[2-(diethylaminomethoxy)phenyl]sulfonylpiperidine-4-carboxylic acid N-[4-[2-(dimethylamino)ethyl-methylamino]phenyl]-3-[6-[1,1-dioxo-2-[4-[2-(trifluoromethoxy)anilino]cyclohexyl]-1,4-thiazinan-4-yl]pyridazin-3-yl]benzamide 5-(1,6-difluoroindole-3-carbonyl)cycloocta-2,4-diene-6-carboxylic acid 2-[1,6-bis(4-aminophenyl)cyclohexa-2,4-dien-1-yl]aniline 2-(N-(8-hydroxyquinoxalin-5-yl)anilino)propanoic acid 2-cyclopropylsulfanyl-7-(3,5-dimethoxyphenyl)thieno[3,2-d]pyrimidine 5-methyl-2,3,4,9-tetrahydropyrano[2,3-b]indole 3-[2-hydroxyethyl(1,3-thiazol-5-yl)amino]propane-1,2-diol 2-(2,4,5,6-tetrafluorophenoxy)-1H-benzimidazole 3-hydroxy-4,5-dimethoxyanthracene-1,2-disulfonic acid 5-(5-aminopyridine-2-carbonyl)-N-methyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-3-carboxamide 5-chloro-2,3-dimethyl-4-[(4S)-1-(4-nitrophenyl)sulfonylazepan-4-yl]oxypyridine (3aR,6aS)-N-[(4-aminoquinazolin-2-yl)methyl]-5-oxospiro[1,3,4,6a-tetrahydropyrrolo[2,3-c]pyrrole-2,4'-piperidine]-1'-carboxamide;formic acid (2R)-5,5,7-trimethyl-2-phenylnonanoic acid N-(1,3-benzothiazol-5-yl)-2-[4-cyclopropylsulfonyl-1-(2,6-difluorophenyl)-6-oxopyridin-3-yl]acetamide 3-(4,6-dimethylpyrimidine-5-carbonyl)oxy-2,2-difluoropropanoic acid 2-(5-pyridin-3-yl-1,4-dihydropyrido[3,4-d]pyrimidin-2-ylidene)propanedinitrile N-(1,2-dihydropyridin-4-ylmethyl)-N-ethyl-3-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraene-5-carboxamide 5-fluoro-2-[(4R)-3-methylpiperidin-4-yl]oxypyrimidine 6-[(1E,3Z)-4-iminopenta-1,3-dienyl]-N-methylquinolin-2-amine 3-[2-[[7-chloro-4-(furan-2-yl)quinazolin-2-yl]amino]ethoxy]benzamide 1-bromo-3,4-dichloro-2H-pyrrolo[2,3-b]pyridine [1-cyclopropyl-2,6-dimethyl-4-(oxan-3-yl)pyrrolo[3,2-c]pyridin-5-yl]carbamic acid N-[(2-chlorophenyl)methyl]spiro[1,4-dihydroquinoxaline-3,3'-piperidine]-2-imine 1-methyl-4-[2-(3,4,5-trifluorophenyl)ethynyl]benzene N-[(5S,7R)-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]benzamide 4-[2-[5-(3,3-difluoropyrrolidin-1-yl)-6-methoxypyridine-3-carbonyl]-3-(2-ethylphenyl)-3,4-dihydropyrazol-5-yl]-3-fluorobenzonitrile 3-(2-methylpropyl)-7-(morpholin-4-ylmethyl)-8,9-dihydroimidazo[1,5-f]purin-6-one (Z)-2-[amino-(3,4-dimethoxyphenyl)phosphanyl]-N'-[(E)-but-1-enyl]prop-1-ene-1,3-diamine;ethane 3-[2-(hydroxymethyl)but-1-enyl]xanthen-9-one 1-[(2R,3S)-3-phenylbutan-2-yl]pyrrolidine 7-[1-(4,6-diphenyl-1,3,5-triazin-2-yl)carbazol-9-yl]indolo[1,2-a]quinoline 4-N-(2,6-dimethylphenyl)-5H-indeno[1,2-d]pyrimidine-2,4-diamine (2S)-N-[5-chloro-6-(1,3-dimethylpyrazol-4-yl)pyridin-2-yl]-5-[5-fluoro-6-(methanesulfonamido)pyridin-3-yl]-3,3-dimethylpentanamide 4-[6-[(Z)-2-aminoethenyl]pyridin-3-yl]oxycyclohexan-1-one N-[(1S,3R)-3-[4-amino-7-methyl-5-[4-(6-phenoxypyridine-2-carbonyl)phenyl]pyrrolo[2,3-d]pyrimidin-6-yl]cyclopentyl]-2,2-difluoropropanamide 2-bromo-N-[(2R,3S)-2-[(4-ethoxyphenyl)methyl]-5-oxooxolan-3-yl]benzamide N-[3-(2-benzylcyclopropyl)prop-1-en-2-yl]aniline (2-oxo-4-phenylhexyl)azanium 4-amino-1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)pyrimidin-2-one (7R)-3-[2-hydroxy-5-methyl-4-oxo-6-(trifluoromethoxy)pyridin-1-yl]-8,9-dihydrobenzo[f]chromene-7-carboxylic acid 5-[(4R)-6-amino-2,2,7-trimethylnonan-4-yl]oxy-4-N-cyclopentylquinazoline-2,4-diamine N-[2,2-difluoro-2-(4-methylphenyl)ethoxy]sulfanylpiperidine-1-carboxamide 1-[5-(2,3-dimethylphenyl)-4H-pyrrolo[3,2-d]pyrimidin-2-yl]cyclobutan-1-ol 4-(3,5-difluorophenyl)-8-methylsulfonyloxyquinoline-2-carboxylic acid 2-ethyl-6,7-dimethoxy-3-(4-phenylpiperazine-1-carbonyl)chromen-4-one 3,5-dibromo-2H-benzo[h]isoquinolin-1-one 3-[2,5-difluoro-4-(1,2,3,6-tetrahydropyrazin-4-ium-4-yl)phenyl]-4-methoxybenzenesulfonamide;chloride 1-(3-ethylsulfonylphenyl)-3,5-dimethylpyrazole;yttrium 5-(2,4-dihydroxy-6-methylphenyl)-N-[3-(4-methylpiperazine-1-carbonyl)phenyl]pyrazole-1-carbothioamide 1-[4-(3,5-dichlorophenyl)sulfonyl-3-(hydroxymethyl)piperazin-1-yl]ethanone 5-[4,6-bis(3,3-dimethylbutanoyl)furo[2,3-b]pyridin-2-yl]imidazolidine-2,4-dione 5-(1H-indol-3-yl)-4,5-dihydro-1,2-oxazole-3-carboxylic acid (E,3R)-6-cyclohexyl-N-[2-hydroxy-5-methoxy-4-(1H-pyrazole-5-carbonyl)phenyl]hept-5-ene-3-sulfonamide 6-[(2R)-3-amino-2-methylpyrrolidine-1-carbonyl]-3,4-dihydro-1H-quinolin-2-one 4-(3,4,5,6,7,8a,9,10-octahydropyren-1-yloxy)piperidine N-[4-(aminomethyl)phenyl]-2,7-dichloroquinolin-4-amine 4-[N-(2,3-dihydroxypropyl)-2-nitroanilino]benzoic acid 1-[5-(2,4-dimethoxyphenyl)hexanoyl]azepan-3-one;hydrochloride 1-(2,4-dibromophenoxy)-3,3a,5,6,7,7a-hexahydrocyclopenta[b]pyridine 4-[[5-[[2-(cyclohexylmethoxy)ethylamino]methyl]pyridin-2-yl]methoxy]-1H-indole-2,3-dione 1-(5-chlorothiophen-2-yl)sulfinylpyrrolidine;hydrochloride 4-methoxy-N-(1-naphthalen-2-yl-5-oxopyrrolidin-3-yl)pyridine-3-carboxamide (NZ)-N-[1-[3,5-bis(trifluoromethyl)phenyl]ethylidene]-2-methylpropanediamide (E)-1-[4-[5-chloro-2-fluoro-4-(propylamino)benzoyl]piperazin-1-yl]-3-[6,7-dihydro-5H-cyclopenta[b]pyridin-8-ylmethoxy-[(Z)-prop-1-enyl]amino]but-2-ene-1,4-dione N'-(1-cyclopentylethenyl)-N-[4-methoxy-3-(5-phenyl-2H-pyrazolo[3,4-b]pyridine-7-carbonyl)phenyl]acetohydrazide (5S)-2-(3,4-dimethoxyphenyl)imino-1,3-thiazolidin-4-one N-ethyl-2-[3,4,6-trioxo-2-sulfanylidene-1-(2-thiophen-2-ylethyl)thieno[2,3-d]pyrimidin-5-yl]acetamide 3-[2-[4-(difluoromethyl)phenyl]-4-phenyl-1,3-thiazol-5-yl]-2,2-bis(sulfanyloxy)propanenitrile (5R)-7,8-dimethyl-1,4,9,11-tetrazatetracyclo[10.3.0.02,6.07,11]pentadeca-2(6),3,10,12,14-pentaene (Z)-2,3-bis[2,6-diethyl-4-(methoxyamino)phenyl]prop-1-en-1-amine 1-[4-methoxy-2-(3,4,5-trifluorophenyl)phenyl]ethanone 3-fluoro-N,4-dimethyl-2-(oxan-4-yl)benzamide [2-(4-aminoanilino)phenyl]iminoazanide (Z)-N'-[5-cyclopropyl-2-fluoro-4-[3-methyl-6-(triazol-1-ylmethyl)morpholin-2-yl]phenyl]but-2-enediamide 1-(4,6-dimethylpyrimidin-2-yl)oxy-3-dodecylthiourea [[[(2S)-1-carboxypropan-2-yl]amino]-(4-phenylanilino)methylidene]azanide 2-[4-fluoro-3-(trifluoromethyl)phenyl]-5-hydroxybenzonitrile 2-[(3R,4S)-4-hydroxy-1-[5-methyl-6-(2,2,2-trifluoroethoxy)pyridazin-3-yl]pyrrolidin-3-yl]acetic acid 7-(5,6-dimethylbenzimidazol-1-yl)-N-[(3R,4S)-4-ethoxyoxolan-3-yl]quinazolin-2-amine 3-cyclohexylpropanoyl(phenyl)carbamic acid N-[3-[[4,6-bis(2,4-dimethoxyphenyl)-1,3,5-triazin-2-yl]sulfanyl]propyl]benzenesulfonohydrazide (5R)-5-[2-(4-fluorophenyl)ethyl]-3,7,9-trimethoxy-6,12-dihydropyridazino[1,6-c][1,4]benzodiazepine (5E)-3-ethyl-2,6-dioxo-5-[(Z)-prop-1-enyl]-4-pyridin-4-ylcyclohepta-3,5-diene-1,4-dicarbonitrile 2-[1-(4-bromophenyl)ethyl]-4-hydroxypiperidine-1-carboxylic acid [4-[(3S)-3-aminopyrrolidin-1-yl]-2,5,6-trifluorophenyl]carbamic acid 2-(4-methylphenyl)-5,6-dihydropyrazolo[3,4-d]pyrimidin-4-one (2R)-2-[3,5-dichloro-N-(1H-pyrazol-4-ylmethyl)anilino]butanoic acid 1-azido-2,3,4,6-tetramethyl-5-(trifluoromethoxy)benzene N-[2-amino-1-(5-chloropyridin-3-yl)ethylidene]-4-[[(1R,2S)-2-methoxycyclohexyl]amino]benzamide;dihydrochloride 3-(1,3,4,6-tetrahydrobenzo[c][1]benzoxepin-5-yl)propanoic acid 2-[4-(3,5-difluoro-4-hydroxyphenyl)triazol-1-yl]ethoxymethanedithioic acid 5-(2,3-difluoro-4-propoxyphenyl)-1,3,8-trimethylpyrido[3,4-d]pyrimidine-2,4,7-trithione N-[2,4-dichloro-5-(methylamino)phenyl]acetamide 6-(6,6-dimethyl-1,4,5,7-tetrahydroindazol-3-yl)-N-[2-fluoro-6-methoxy-4-(4-propanoylpiperazin-1-yl)phenyl]pyridine-2-carboxamide 2-amino-5-(4-azidophenyl)benzenecarboximidamide 2-[5-fluoro-2-methoxy-4-[3-(trifluoromethyl)anilino]phenyl]acetonitrile 5-amino-2-(cyclohexen-1-yl)-6,7-dihydro-4H-[1,3]thiazolo[4,5-c]pyridine-6-carboxylic acid 2-(3,5-dimethylpiperazin-1-yl)-N-[4-(2H-tetrazol-5-yl)phenyl]pyridine-3-carboxamide 2-[(3,5-dimethylpyridin-4-yl)-propan-2-ylamino]-1-pyrrolidin-1-ylethanone 4-[2-(1-azidooxypropyl)-3-phenylmethoxy-5-pyridin-3-ylsulfonylphenyl]morpholine 6-[[5-aminosulfanyl-2-(3,4-difluorophenyl)pentanoyl]amino]hexanoic acid [2-(2-chlorophenyl)pyrazol-3-yl]methanamine;dihydrochloride [3-(cyclohexylmethoxy)phenyl]-diphenylphosphane 2-[3,5-difluoro-4-(triazol-1-yl)phenyl]acetic acid N-[5-(3-chlorophenyl)-6-methylpyridin-2-yl]pyrrolidine-1-carbothioamide [1-(5-fluoropyrimidin-2-yl)pyrazol-4-yl]-[4-(3,3,3-trifluoroprop-1-enylsulfonyl)piperazin-1-yl]methanone 4-azidooxy-3-ethylsulfanylbenzenesulfonic acid 2-hydroxy-5-methyl-3,4-bis(trifluoromethoxy)benzoic acid 1-cyclohexa-2,4-dien-1-yl-3-[[3-methoxy-5-(2H-tetrazol-5-yl)phenyl]methyl]urea (3S)-N',1-dimethyl-5-oxopyrrolidine-3-carbohydrazide;[2-fluoro-6-[4-(trifluoromethyl)phenyl]benzoyl]carbamic acid 7-(2,4-dimethylphenyl)-2-[3-fluoro-4-(trifluoromethoxy)anilino]cyclohepta-2,4,6-trien-1-one 5-methyl-3-(4-propoxyphenyl)imidazolidine-2,4-dione (5R,7S)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5,7-bis(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide [4-(3-aminopropyl)-1,2,5-oxadiazol-3-yl]oxymethanethione 3-[(2E)-2,4-dimethylpenta-2,4-dienoxy]propylbenzene;propane (2S)-N-(1,3-benzothiazol-5-ylmethylideneamino)-2-methoxypropanamide 3-bromo-N-[4-fluoro-2-(trifluoromethyl)phenyl]-2-oxopropanamide 1-azido-3,5-bis(difluoromethyl)pyrazole 2-N-(1-benzylindazol-5-yl)-4-N,6-N-dimethylpyrimidine-2,4,6-triamine 2-[4-[3-(1,1-dihydroxyethyl)-5-methylpyrazol-1-yl]phenyl]benzoate 5-(trifluoromethyl)-2-[3-(2,2,6,6-tetramethylpiperidin-4-yl)triazolo[4,5-c]pyridazin-6-yl]phenol 3-[6-(5,7-dichloro-2-oxo-1H-quinolin-8-yl)-2,7-naphthyridin-3-yl]propanoic acid 6-(4-cyanobutylamino)pyridazine-3-carbonitrile 2-[4-(methanesulfonamido)-3,5-dimethylphenyl]sulfonyl-N-oxoacetamide (1S,2R)-N-[8-amino-6-(4-methylpyridin-3-yl)isoquinolin-3-yl]-2-phenylcyclopropane-1-carboxamide 2-(2-chlorophenyl)sulfanylbenzoic acid 1-[4-amino-2-(methoxymethyl)butanoyl]pyrazole-3-carbonitrile 5-[(E)-but-1-enyl]-4-hydroxy-2-methylidenethiophen-3-one 1-(3,4-dimethoxyphenyl)hexan-2-one 1-[6-ethenyl-5-(methylideneamino)naphthalen-2-yl]butan-1-one 5-fluoro-N-methyl-N-[3-(1,2,4-triazol-1-yl)butan-2-yl]pyrimidine-2-carboxamide 4-azidooxysulfanyl-2-(trifluoromethyl)pyridine 4-[3-[2,6-di(propan-2-yl)phenyl]imidazol-1-ium-1-yl]butanenitrile 2-(9H-fluoren-1-yl)terephthalic acid 2-[[4-[2-(diethylamino)ethoxy]phenyl]methyl]pyridine-3-sulfonamide N-[2,4-difluoro-3-(propylamino)phenyl]-5-(1H-indol-3-yl)-1-methylpyrazole-3-carboxamide 4-[(2R)-6-azaspiro[2.5]octan-2-yl]-3,5-dimethoxyaniline 5-[(1Z)-buta-1,3-dienyl]-2-methylidenenaphthalene;ethane 5-(2-methylpyridin-4-yl)-3H-1,3-benzothiazol-2-one N-azido-2-(4,6-dichloropyrimidin-2-yl)oxyacetamide 6-[4-methoxycarbonyl-N-(1,3-thiazol-5-yl)anilino]-4-hydroxynaphthalene-2-sulfonic acid 5-amino-7-(pyridin-2-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile N-[1-(3-phenylpropyl)piperidin-4-yl]-5,6-dihydroquinoline-8-carboxamide 6-[(3-chlorophenyl)methyl]-2-pyrrolidin-1-yl-7,8-dihydropyrimido[4,5-d]pyrimidine-5,7-dione N-methyl-2-[(4Z)-2,5-dioxo-4-[(2E,4Z)-2-phenylhexa-2,4-dienylidene]pyrrolidin-1-yl]acetamide 3-[[1-(4-fluorophenyl)ethylcarbamoylamino]methoxy]benzoic acid N-(4,6-dimethylpyrimidin-2-yl)-4-[3-nitro-N-(2-phenylethyl)anilino]benzenesulfonamide 4-[3-[(2R)-1,1-bis[5-chloro-2-(tetrazol-2-yl)phenyl]propan-2-yl]oxy-5-cyclopropylidene-1H-pyrazol-2-ium-2-yl]pyrimidine ethane;4-[3-methylbut-1-ynyl(pentan-2-yl)amino]benzoic acid N-(1,2-dihydropyridin-3-ylmethyl)-4-phenylbutanamide 3-N-[(2S,3R)-1-oxo-3-phenyl-5-[4-[(propan-2-ylamino)methyl]anilino]pent-4-en-2-yl]isoquinoline-1,3-dicarboxamide (2S)-4-[2-oxo-1-phenylmethoxy-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-4-yl)propyl]pyrrolidine-2-carboxylic acid 2-[(Z)-(phenylhydrazinylidene)methyl]-4,5-bis(2H-triazol-4-yl)benzene-1,3-diol (2S,4R)-1-[6-amino-5-(cyclohexa-1,3-dien-1-ylmethoxymethyl)pyrimidine-4-carbonyl]-N-ethyl-4-hydroxypyrrolidine-2-carboxamide [(2R)-1-amino-4-methyl-1,3-dioxopentan-2-yl]carbamic acid;methanethiol;3-[2-methyl-5-[5-(trifluoromethyl)pyridin-2-yl]furan-3-yl]propanal 5-[(4S)-3,3-dimethylpiperidine-1-carbonyl]-N-propan-2-ylfuran-3-sulfonamide N-cyclopropyl-7,8-dimethoxy-1H-2,3-benzothiazin-4-imine (E)-3-[4-(9-methylacridin-10-ium-4-yl)phenyl]-1,7,8,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8,10,12-hexaene 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidine-2,4-dione;bromozinc (5-tert-butylthiophen-2-yl)sulfonylurea 2-methylsulfonyl-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)pyridine-3-carboxamide 5-methyl-6-[4-(2-pyridin-4-ylimidazol-1-yl)phenyl]imidazo[2,1-b][1,3,4]thiadiazole 2-[3,5-bis(trifluoromethyl)phenyl]quinoline (5-amino-2,3-difluorophenyl)-(4,6-dihydrazinylpyrimidin-5-yl)methanone 4-(azidomethyl)-2,6-dibutoxyphenol 4-(2,6-dimethylheptan-3-yl)-1-ethoxy-2-[(Z)-prop-1-enyl]benzene 2-(3,4-dihydro-1H-isoquinolin-2-yl)-7-[(5-ethoxycyclohexa-2,4-dien-1-ylidene)methyl]-N-methylpyrrolo[2,3-d]pyrimidine-6-carboxamide 2-(5,6,7,8-tetrahydronaphthalen-2-yl)propanamide 6-[(2R)-4-hydroxybutan-2-yl]-3H-quinazolin-4-one 1-[2-ethyl-4-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydronaphthalene 4-[(8-bromoquinoxalin-5-yl)-propylamino]butan-1-ol (4-methoxyphenyl)sulfanylmethanesulfonate 1-[1-(2,3-dihydro-1-benzofuran-4-yl)cyclopropanecarbonyl]-N-ethylpiperidine-3-sulfonamide N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1,3-benzothiazol-5-amine 2-(3,4-dichlorophenyl)-6-[(2-fluoro-4-hydroxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-(4-pyridin-2-yl-1H-imidazo[4,5-c]pyridin-2-yl)-5-pyridin-3-yl-1H-pyrazolo[3,4-c]pyridine 5-(1,3-benzodioxol-5-ylmethoxy)-4-bromocyclohexa-2,4-dien-1-imine N-[(1R)-5-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]ethanesulfonamide 3-methyl-1-[4-(2,4,6-trimethylphenyl)butanoyl]piperidine-3-carboxylic acid 3-(3-methylphenoxy)-1-piperazin-1-ylpropan-1-one (3R)-7-[2,6-difluoro-4-(2H-tetrazol-5-yl)phenoxy]-N-hydroxy-8-methoxy-2,3-dihydropyrido[3,2-b][1,4]oxazepine-3-carboxamide 1-(2,3-dihydropyridin-6-yl)-N-methyl-1-[4-[(4Z)-4-[(4-nitrophenyl)hydrazinylidene]but-2-en-2-yl]-2H-pyridin-1-yl]methanimine N'-[4-[(2-methylphenyl)sulfonylamino]pyridin-3-yl]ethanimidamide 2-cyclopropyl-N-[5-(6-oxo-1H-pyrimidin-4-yl)-4,7-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]acetamide N-(3,5-dimethylphenyl)-2-[1-[[5-(2-fluoropropanoylamino)pyridine-3-carbonyl]-formamidomethyl]cyclopentyl]acetamide [4-[7-[2-hydroxy-3-(methylcarbamoylamino)phenyl]quinolin-5-yl]piperidin-1-yl]oxidanium 5-[(2,6-dibromopyridin-4-yl)methylsulfanyl]-3-[4-(dimethylamino)phenyl]-2-prop-1-en-2-ylimidazole-4-carboxylic acid N-[5-chloro-2-(2,6-difluorophenyl)pyrazol-3-yl]-2-fluoro-1H-indole-4-sulfonamide 3-[3,5-dimethyl-4-[(4-nitrophenyl)diazenyl]pyrazol-1-yl]propanenitrile 1-ethyl-N-methyl-4-(3-morpholin-4-ylphenyl)pyrazolo[3,4-d]pyrimidin-6-amine 2-(6-chloropyridin-3-yl)-2-methoxyimino-N-(4-piperazin-1-ylphenyl)acetamide;ethane 4-[6-chloro-8-fluoro-7-(2,3,5,6-tetradeuteriopyridin-4-yl)oxynaphthalen-1-yl]-3-methyl-N-(piperidin-4-ylideneamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide 2-[4-amino-3-(6-amino-5,7-dihydropyrrolo[3,4-d]pyrimidine-2-carboximidoyl)phenyl]sulfanyl-1-morpholin-4-ylethanone 2-[1-(7H-purin-6-yl)pyrrolidin-3-ylidene]acetamide 4-[(3-chlorophenyl)methoxy]-3,5-dinitrobenzamide 6-benzylsulfanylnaphthalene-1,4-diamine 3-(1H-pyrrol-2-yl)-5-[4-[1-(trifluoromethylsulfonyl)piperidin-4-yl]oxyphenyl]-1,2,4-oxadiazole 5-bromo-4-N-[2,6-dichloro-4-(trifluoromethyl)phenyl]pyrimidine-2,4-diamine 2-[(4R)-3,7,9-trimethyl-8-oxo-1-azaspiro[5.5]undecan-4-yl]benzenecarboximidamide 4-(dipropylsulfamoyl)-N-methylbenzenecarboximidate ethane;4-hydroxybutanoic acid;3-[(E)-hex-2-en-3-yl]-1H-indole (5-cyanopyridin-2-yl)-[3-[4-(2,6-difluorophenyl)-1H-pyridazin-2-yl]-4-methoxyphenyl]carbamic acid 3-[1-azido-2-(4-chlorophenyl)ethyl]pyridine 4-ethyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyridin-2-amine 5-[6-chloro-5-(4-methylphenyl)pyridine-2-carboximidoyl]pyrimidin-4-amine ethane;methanamine;1-methylcyclohexa-3,5-diene;9-[(E)-2-phenylethenyl]carbazole 1-methylsulfanyl-2-(phenyldisulfanyl)benzene N-[4,5-bis(ethenyl)-1H-imidazol-2-yl]-4-(trifluoromethoxy)benzamide 5-bromo-2,4-dichloro-3H-isoindol-1-one 5-(1H-benzimidazol-2-yl)-6-phenyl-7,8-dihydrophthalazine N-[2,4-difluoro-3-[5-(4-methylphenyl)pyridine-3-carbonyl]cyclohexa-1,5-dien-1-yl]-4-hydroxybenzenesulfonamide 3-[4,7-diamino-6-chloro-3-(5-ethylpyridin-2-yl)-1-methylpyrazolo[4,3-b]pyridin-5-yl]propanoic acid 6-chloro-3-(1H-indol-2-yl)quinoline 2-[7-[methoxy(pentyl)sulfamoyl]naphthalen-1-yl]-5,6-dihydrocyclopenta[b]thiophene-3,4-dione 1-[3,5-bis(dimethylamino)phenyl]-2-[(2E)-2-ethenylpenta-2,4-dienoxy]ethanone 2-[(3Z,5E)-8-fluoroocta-1,3,5-trien-4-yl]-5-(3-propan-2-yloxyphenyl)quinazoline 1-(6,7-dihydrobenzo[g]indole-3-carbonyl)piperidine-4-carboxylic acid 2-aminooxycarbonyl-3-phenylpropanedioic acid 2-(3,4-difluorophenyl)-5-[6-[2-(dimethylamino)ethoxy]imidazo[1,2-b]pyridazin-3-yl]-1H-imidazole-4-carboxylic acid;2,2,2-trifluoroacetic acid N-[3-methyl-1-[[4-[4-[(5R)-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]butyl]phenyl]methoxycarbonylamino]butan-2-yl]carbamate 1-[3-[(Z)-1-aminobut-2-enyl]-2,5-dihydropyrrol-1-yl]-2-methoxy-2-phenylethanone 6-[4-(2-hydroxyethoxy)phenyl]-N-pyrazin-2-ylpyridazine-3-carboxamide [3-(5-chloropyridin-2-yl)oxypiperidin-1-yl]-(2,3-dihydro-1H-inden-5-yl)methanone 4-(3-propyl-1,2,4-triazol-1-yl)pentanoic acid 5-[6-(butylamino)pyrimidin-4-yl]-1H-pyrazole-4-carbonitrile 4-[3-(2,3-difluorophenyl)propyl]aniline (Z)-3-[3,4-dihydroxy-5-(trifluoromethyl)phenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile (2S)-N-[(1R,3R)-3-benzamidocyclohexyl]pyrrolidine-2-carboxamide 3-[[2-(aminomethyl)phenoxy]methyl]benzonitrile N-[2,3,4-trifluoro-5-(trifluoromethyl)phenyl]formamide N-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)cyclohexyl]naphthalene-2-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]piperidine 2-(3,4,5,6-tetraethoxypyridin-2-yl)acetic acid 1-chloro-4-[(3E)-5,7-dimethylocta-1,3,6-trien-2-yl]benzene;ethane 4-[2-(3,5-difluorophenyl)pyrrolidin-1-yl]-N-(furan-2-ylmethyl)-7H-pyrrolo[3,2-d]pyrimidine-6-carboxamide 4-bromo-2,6-difluorobenzoic acid;3-methylbutanal 2-[2-methylpropyl(1,3-thiazol-2-yl)amino]octanoic acid 4-(6,7,8,9-tetrahydropyrido[1,2-a]benzimidazol-3-yl)piperazine-1,2-dicarboxylate 7-[1-(5-fluoropyrimidin-2-yl)piperidine-4-carbonyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 2-(5,6-dihydropyrido[3,2-d]pyrimidin-4-ylsulfanylmethyl)cyclohepta-1,3-dien-5-yne-1-carboxylic acid 4-[(3-fluorophenyl)methyl]-7,8-dihydroquinoline 4-[4-(dibutylamino)phenyl]-N,3-dimethylaniline 3-amino-6-(4-fluorophenyl)-5H-pyrrolo[2,1-f][1,2,4]triazin-4-one N-butyl-4,6-dimethoxynaphthalene-2-carboxamide 1-methyl-4,5,6,7-tetrahydroindole;1-(2-methoxyphenyl)-3-[3-(pyrrolidin-1-ylmethyl)phenyl]urea (2Z)-2-[5-methylidene-2-(4-propylcyclohexen-1-yl)-1,3-dioxan-4-ylidene]-3-oxobutanenitrile 1-ethyl-6-fluoro-7-(5-methyl-2-pyrimidin-4-yl-1,3-thiazol-4-yl)-3H-imidazo[4,5-b]pyridin-2-one 2-[3-[1,5-bis(4-hydroxyphenyl)pyrazol-3-yl]imidazo[1,5-a]pyridin-1-ium-1-ylidene]-N-phenylacetamide;chloride 1-[3,5-difluoro-4-(5,6,7,8-tetrahydroquinazolin-2-ylsulfanyl)phenyl]ethanone 6-bromo-2,2,3,4,5,7-hexafluoro-1H-indene N-[4-(aziridine-1-carbonyl)phenyl]-2-methoxypyridine-3-carboxamide (4R)-1-[(2S,3S,6S)-2-phenylmethoxy-6-propan-2-yloxan-3-yl]-4-[[2-[4-(trifluoromethyl)anilino]benzoyl]amino]piperidine-3-carboxylic acid 7-hydroxy-N-(3,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,11-tetraen-4-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide 1-(3,4-difluorophenyl)-6-[(2S,5R)-5-hydroxyoxepane-2-carbonyl]-3H-imidazo[4,5-b]pyridin-2-one 1-[2-(4,6-diphenylpyridin-2-yl)oxyethyl]piperidine-3-carboxylic acid 1-[4-(aminomethyl)phenyl]-2-hydroxyethanone;ethane N'-methyl-2-[4-(3,6,11-triazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,10-tetraen-5-yl)cyclohexyl]ethanimidamide 2,6-dichloro-N',4-bis(3-methylbutylsulfanyl)pyridine-3-carboximidamide 4-[[4-(dimethylamino)cyclohexyl]amino]-5,8-dihydropyrido[2,3-d]pyrimidin-7-one N-[2,4-dihydroxy-3-(5-methoxycyclohepta-1,3,6-trien-1-yl)butyl]-2,7-diethynylnaphthalene-1-carboxamide 1-(3,5-dichlorophenyl)-N-[[2-ethyl-4-(trifluoromethyl)phenyl]-(6-oxopiperidin-3-yl)methoxy]methanesulfonamide (4-aminophenyl)-[1-[(E)-3,5-dimethylhex-2-enoyl]piperidin-3-yl]methanone N-[2-(1,3-benzothiazol-2-yl)ethyl]-4-oxopiperidine-1-carboxamide N-[2-(difluoromethoxy)-6-(1,1,1-trifluoropropan-2-yl)pyridin-4-yl]formamide 1-benzylpyrrolidine-2,5-dicarboxylate 3-benzyl-2-hydroxy-4-[(5R)-5H-imidazo[5,1-a]isoindole-8-carbonyl]butanamide 6-methylsulfanyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one 2-[4-(methylamino)phenyl]-N-[3-(1,4,7,10,13-pentazacyclotetradec-1-ylsulfonyl)phenyl]acetamide 3,5-bis(4-nitrophenyl)pyridine 2-[(5S,10bR)-7-methoxy-5-pyridin-3-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 5-[4-amino-3-(methyliminomethyl)phenyl]-2H-pyrazolo[3,4-b]pyridine-3-carboxylic acid 4-(6,11-dihydropyrido[2,3-c][1]benzazepine-5-carbonyl)benzamide N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-3,4-dihydro-2H-chromene-8-sulfonamide N'-[3-chloro-4-(2,6-dimethylphenyl)-5-formamidothiophen-2-yl]ethanimidamide ethane;4-[(3E)-6-fluorohepta-1,3,5-trien-3-yl]oxyphenol (NZ)-N-[1-[4-[2-[2-methoxyethyl(methyl)amino]pyridin-3-yl]phenyl]ethylidene]hydroxylamine 4-[5-(4-aminopiperidine-1-carbonyl)-7-oxo-6H-pyrazolo[3,4-c]pyridin-3-yl]benzonitrile 2-(4,7-difluoroindol-1-yl)acetic acid 4-[(Z)-2-(aminomethyl)-3-fluoroprop-2-enoxy]-N,N-diethylbenzamide N'-[4-[(Z)-2,3-diamino-1-cyanoprop-1-enyl]cyclohexa-2,4-dien-1-ylidene]benzenecarboximidamide 5-chloro-3,7-dimethyl-6H-pyrimido[4,5-b]quinoline N-[4-(3,5-difluorophenyl)-2-methylpentan-2-yl]-6-(1H-pyrrolo[2,3-c]pyridin-7-ium-3-yl)pyrimidin-4-amine 2-[[(1R)-1-azidopropyl]amino]-5,6-dimethoxypyrimidine-4-carbonitrile 2-[4-(3,6-dihydro-2H-pyran-4-yl)phenyl]-N-methoxy-1-oxoisoquinoline-4-carboxamide N-(2,3-dihydro-1H-inden-2-yl)-2-methoxy-6-methylpyrimidine-4-carboxamide 7-(cyclopropanecarbonyl)-2-[(3R,4S)-3-fluoropiperidin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 4-[7-cyclobutylimino-3-[(1R)-1-[3-methoxy-5-(trifluoromethyl)phenyl]ethyl]pyrazolo[1,5-a]pyrimidin-5-ylidene]butanoate 5-methoxy-4-(pyridin-3-ylmethylamino)-1H-pyrimidin-6-one 2-[1-[(5-chloro-3-ethylsulfanylpyridine-2-carbonyl)amino]cyclopropyl]acetic acid 2-(2,3-dimethoxyphenyl)-1-(2-hydroxyphenyl)ethanone 6-amino-4-(4-bromonaphthalen-1-yl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 5-[4-[(1E,3Z)-cycloocta-1,3,7-trien-1-yl]oxyphenyl]-2H-tetrazole N-cyclohexyl-6-(1,2,4-triazol-1-ylmethoxy)pyridine-3-carboxamide N-[2-[4-(difluoromethyl)cyclohexyl]pyridin-3-yl]-1H-pyrrole-3-sulfonamide N-[(3R)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]naphthalene-2-carboxamide 1-(4,4-dimethylpentan-2-ylamino)anthracene-9,10-dione 3-[2,6-difluoro-N-(1H-indol-5-yl)anilino]butanoic acid 1-(3,6-dihydro-2H-pyran-5-yl)-N'-[4-fluoro-7-(3-morpholin-4-ylpropoxy)quinazolin-2-yl]ethane-1,2-diimine 2-chloro-5,6-diethylpyrimidine-4-carboxylic acid;hydrochloride 2-(4-methylphenoxy)benzene-1,3,5-tricarboxylic acid 1-[4-[2-[(Z)-2-aminoprop-1-enyl]phenyl]but-3-ynyl]piperidine-3,6-diol 4-(1H-indazol-5-yl)-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 3-[2,6-dibromo-4-(10-chlorodecoxy)phenyl]prop-2-enoate 6-[(4-chlorophenyl)methylamino]-7,8-dihydronaphthalene-1,2-disulfonic acid (NZ)-N-[1-amino-3-[2,3-difluoro-4-(trifluoromethylsulfanyloxy)phenyl]propylidene]hydroxylamine (2-cyclopropyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-8-yl)methanamine 6,7-dimethoxy-2-[(2R)-2-(4-phenylphenyl)morpholin-4-yl]quinoline-4-carboxylic acid (3S)-6'-fluorospiro[1H-indole-3,5'-4H-chromeno[2,3-c]pyrazole]-2-one N-[4-[3-(aminomethyl)piperidine-1-carbonyl]-2-methoxyphenyl]quinoline-8-sulfonamide 2-[5-(aminomethyl)thiophen-2-yl]-7,8-dihydro-6H-quinazolin-4-amine 1-[(2E)-3,7-dimethylocta-2,6-dienoxy]-4-propan-2-ylbenzene 1-[2,6-bis(trifluoromethyl)phenyl]-5-chloropyrazole 5-(2,4-dihydroxy-5-propanoylphenyl)imino-1-methyl-3-propyl-1,3-diazinane-2,4,6-trione 2-chloro-5-N-(6,7-dihydro-1H-indazol-5-yl)pyridine-3,5-diamine N-[(2S)-2-[4-[(cyclohexylamino)methyl]phenyl]propyl]-N,3-dimethyl-1H-indole-7-carboxamide 2-methylsulfanyl-1,3-benzothiazole;2,6,7,8-tetrahydrobenzo[g][1]benzoxepine 2-(1,3-dioxolan-2-yl)-1-methoxy-4-[2-methylidene-3-[[(E)-4-phenylbut-3-en-2-ylidene]amino]propoxy]anthracene-9,10-dione 3-amino-1-[(E)-3-(4,6-dimethoxypyrimidin-2-yl)sulfanylprop-2-enoyl]azepan-2-one 5-[[3-chloro-4-(trifluoromethyl)phenyl]methoxycarbonylamino]pyridine-2-carboxylic acid N-[6-(hydroxymethyl)-3,4-dihydro-2H-chromen-8-yl]methanesulfonamide (2S)-1,2-diamino-4-methylsulfanylanthracene-9,10-dione N-[(4-fluorophenyl)methyl]-1-(2-hydroxyethylsulfonyl)azetidine-3-carboxamide 1-(2,3-dihydro-1H-inden-5-yl)-N-[1-(4,5-dimethoxy-2-methylphenyl)ethenyl]-N'-propan-2-ylmethanediamine 2-[4-(6-methylpyridine-3-carbonyl)piperazin-1-yl]pyridine-3-carboxamide 5-(3,5-difluorophenyl)sulfonyl-N-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide 1-[(4-bromopyridin-2-yl)methylamino]propan-2-one 2-[3,5-dichloro-N-(cyanomethyl)anilino]acetamide 2-[3-(4-azidophenyl)pyridin-2-yl]oxyacetonitrile 3,9-dimethylfluorene-9-carboxylic acid N-[1-(4-cyclohexylphenyl)-2-imidazol-1-id-3-ylpropan-2-ylidene]hydroxylamine;manganese(2+) 1-cyclopropyl-3-[(2E,4Z)-hepta-2,4,6-trien-2-yl]benzene 6-[2,4-dihydroxy-3-(5-methylcyclohepta-1,4,6-trien-1-yl)-6-pentylphenyl]hexanedioic acid 4-(2,3-dihydro-1H-pyrrolo[2,3-b]pyridin-5-yl)-N-iodo-1-methylsulfanylbutan-1-amine 3-(8,9-dihydrodibenzofuran-4-yl)carbazole;(1Z,6E)-9-methylidene-2H-cycloocta[c]pyridine N-(1,3-benzodioxol-5-ylmethyl)-2-tert-butyl-6-(trifluoromethyl)imidazo[1,2-a]pyridine-8-carboxamide N-[3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl]piperidine-3-carboxamide (4E)-2,5-bis[2-(4-fluorophenyl)ethynyl]hexa-1,4-dien-3-one (7S)-2-amino-5-methyl-4,8-dioxo-7H-pteridine-6-carbonitrile 5-bromo-1,3-dimethyl-N-[2-(4-propanoylphenyl)ethyl]pyrazole-4-carboxamide 3-[1-[4-[2-(2,6-dichloro-3-hydroxy-5-methoxyphenyl)ethyl]piperidine-1-carbonyl]cyclopropyl]-1,1,1-trifluorobutan-2-one 2-(4-carbamimidoylphenyl)-2-[2-[3-fluoro-4-(trifluoromethylsulfonylamino)benzoyl]hydrazinyl]acetic acid;2,2,2-trifluoroacetamide 4-[6-chloro-5-(3,3-difluoropyrrolidine-1-carbonyl)-1H-indole-2-carbonyl]piperazin-2-one 2-(2,5-diaminoanilino)benzoic acid N-[4,6-di(piperidin-1-yl)-1,3,5-triazin-2-yl]carbamate 3-[1,3-bis(4-methylphenyl)sulfanylpropoxy]-2,5-diethylpyridine 7-benzyl-9,11-dihydroxy-5H-naphtho[2,3-b]azepine-6,12-dione 6-(6,7-dihydro-1H-indazole-5-carbonyl)-N,4,5,7,8-pentazatetracyclo[9.7.0.02,4.012,17]octadeca-1(11),2,12,14,16-pentaene-3-carboxamide (3R)-2-methoxy-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)amino]piperidine-1-carboxylate 3-[2,5-difluoro-4-(oxolan-3-ylsulfanyl)phenoxy]azetidine 6-(3-methylphenyl)-4H-pyrido[3,2-d]pyrimidine [(2S,5R)-4-ethyl-5-methoxyoxolan-3-yl]-[4-(1H-pyrazol-4-yl)piperidin-1-yl]methanone 2-[4-(5,6-dihydronaphthalen-1-yl)-1H-pyrazol-5-yl]-N-propan-2-ylacetamide N-[(E)-1H-indol-3-ylmethylideneamino]-2,4-dihydroxy-5-nitrobenzamide 2-azidooxy-4,6-dimethoxyquinazoline 4-[(E)-2-(7-amino-5,6,8,9-tetrahydropyrido[2,3-d]azepin-3-yl)ethenyl]phenol N-(2,3-dihydro-1H-inden-5-yl)-4-hydroxy-4-methoxy-6-oxopyran-3-carboxamide 2-[5-(4-chlorophenyl)-2-methyl-1,3-thiazol-4-yl]-N-[(2R,3S)-2-(1H-pyrazol-4-yl)oxolan-3-yl]acetamide 4-bromo-N,N-bis(prop-2-enyl)aniline (2S)-N-[[3,5-bis[(3,4-dichlorophenyl)methylidene]piperidin-1-yl]methyl]-1-(4-propan-2-ylbenzoyl)piperidine-2-carboxamide 5-[6-[3,5-dimethyl-4-(2-oxopyridin-1-yl)phenyl]-8-ethoxyimidazo[1,2-b]pyridazine-3-carbonyl]-N-methylcyclohexene-1-carboxamide 2-(6,7-dimethoxyisoquinolin-1-yl)acetamide 1-[(2S)-4,6-difluoro-3,5-dihydro-2H-1,4-benzoxazepin-2-yl]butane-1,2-dione (3S)-3-[4-[(2-methoxyquinolin-5-yl)amino]thieno[3,2-d]pyrimidin-6-yl]-1-oxa-7-azaspiro[3.5]nonane-8-carboxylic acid 3-[(Z)-2-(methylideneamino)ethenyl]-N-[3-[[(1S,3R)-3-methylcyclohexanecarbonyl]amino]-4-methyliminopentan-2-yl]benzamide 3-methyl-2-[4-(4-propanoylphenyl)-1,3-thiazol-5-yl]butanoic acid N'-[6-fluoro-4-(trifluoromethyl)pyridin-2-yl]benzohydrazide 4-[(3,5-dimethoxyphenyl)methyl]-3-methylbenzamide (3R,4S)-1-[[5-cyclobutyl-2-fluoro-4-[(E)-2-(4-hydroxyphenyl)ethenyl]phenyl]methyl]-3-[(3Z,5Z)-hepta-1,3,5-trien-2-yl]piperidine-4-carboxylic acid 5-[5-(difluoromethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(6-ethoxypyridin-3-yl)propan-2-yl]pyrimidin-2-amine [6-amino-1-(3,5-dihydroxyphenyl)-1-oxohexan-2-yl]carbamic acid 2-(3,5-difluorophenyl)-1-[(4S)-2-oxa-8-azaspiro[4.5]decan-8-yl]ethanone;ethane 2-(3,4-dihydrocarbazol-9-yl)-N,N-diphenylaniline N-[(Z)-1,2-diaminoethenyl]-3-methoxy-4-[6-oxo-5-(propylsulfanylamino)-1H-pyridazin-4-yl]benzamide [1-cyclopropylsulfonyl-3-(trifluoromethoxy)pyrrolidin-2-yl]-pyrimidin-5-ylmethanone [2-(1,3-benzoxazol-2-yl)pyrrolidine-1-carbonyl]phosphonic acid 1-ethyl-4-(2-pyridin-3-ylethylamino)spiro[2H-indole-3,8'-7H-furo[3,2-g]chromene]-5'-one 2-[5,6-diphenyl-2-(phenylmethoxymethyl)pyrimidin-4-yl]oxypropanoic acid 1-[5-methoxy-2-(3-methylbutoxy)phenyl]-2H-tetrazol-5-one N-methyl-5-(3-propan-2-yloxyphenyl)-6,7-dihydrotetrazolo[1,5-a]pyrimidine-7-carboxamide 2-(6,7-dimethoxyquinazolin-4-yl)-3H-isoindol-1-one 1-cyclopropyl-2,6,8-trifluoro-7-(3-methoxyazetidine-1-carbonyl)quinolin-4-one 4-[5-[3,4-bis(phenylmethoxy)phenyl]-1H-pyrazol-4-yl]benzenesulfonamide 2-[3,5-di(propan-2-yloxy)phenyl]-6,7-dihydro-1H-benzimidazole 3-azido-2,4-dichlorobenzenesulfonic acid [2-aminoethyl(propan-2-yl)amino]-[[4-fluoro-1,3-bis(2-methoxyphenyl)pyrazolo[3,4-d]pyrimidin-6-yl]amino]methanol 3-[[(4-acetamidobenzoyl)amino]methylidene]piperazine-1-carboxylic acid (2-azidooxy-1,2,2-trichloroethyl)benzene (3R)-2,5-diamino-3-benzylsulfanyl-4,6-bis[3-(trifluoromethyl)phenyl]hexanedioic acid 1-[(2R)-1-cyclopropylsulfonylpiperidine-2-carbonyl]-N-[6-fluoro-5-[(E,4Z)-3-methoxyiminohept-4-enyl]pyridin-3-yl]pyrrolidine-2-carboxamide 3-chloro-N-[(Z)-1H-indol-6-ylmethylideneamino]benzamide 3-hydroxy-4,8-dimethyl-10H-phenothiazine 1-(2-azidoethyl)-3,4,5-trifluoro-2-phenylbenzene 2-(1H-indol-3-yl)-N-[5-methoxy-4-(methylideneamino)-6,7,8,9-tetrahydrodibenzofuran-2-yl]acetamide 5-chloro-3-[(Z)-2,2-difluorohex-4-en-3-yl]sulfanylpyridine-2-carbonitrile [(2S)-3,3-diethoxy-1-phenylpropan-2-yl]benzene N-(3,5-dichlorophenyl)-3-oxobutanamide 1-(4,5-dimethylcyclohexen-1-yl)naphthalene 6-azidooxy-2,3-dihydrochromen-4-one (2R)-4-[(1S)-3-methoxycyclopentyl]sulfanyl-2-methyl-1-(4-methylphenyl)sulfonylpiperazine 5-(3-pyridin-4-ylpropoxymethyl)-1H-pyrazole 4-[6-(3-tert-butylpiperazin-1-yl)pyridin-2-yl]oxy-N,N-dimethylpyridin-2-amine 1,3-diphenyl-2H-benzimidazole N-[(Z)-(3,4-dihydroxyphenyl)methylideneamino]-4-oxothieno[2,3-c]quinoline-2-carboxamide 2-chloro-4-ethyl-5,6-difluoropyrimidine;3-[(E)-4-[1-(4-fluorophenyl)ethenoxy]-3,3-dimethylbut-1-enyl]pyridine 4-chloro-N'-hydroxy-5,6-dimethylpyridazine-3-carboximidamide 2-methyl-4-(3,3,5-trimethylcyclohexa-1,5-dien-1-yl)phenol N-[2,6-di(propan-2-yl)phenyl]butanethioamide 1-[2-(benzenecarboximidoylamino)ethyl]piperidine-3-carboxylic acid;hydrochloride N-(1,3-benzodioxol-5-yl)-2-[(4E,6Z)-octa-2,4,6-trien-4-yl]sulfonylacetamide 2-(5-bromothiophen-2-yl)-1H-indole N'-[(E)-3-[2,5-bis(trifluoromethyl)phenyl]prop-1-enyl]-4-cyclobutylidenepiperidine-1-carboximidamide 5-chloro-4,6-diethyl-N-methoxypyrimidin-2-amine 7,12-dichloro-2,8-bis(2H-tetrazol-5-yl)-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene 3-[(Z)-4-[4-[1,3-dioxo-2-[6-(trifluoromethoxy)-1,3-benzothiazol-2-yl]isoindol-5-yl]piperazin-1-yl]but-1-enyl]benzenecarboximidamide 3-methoxybenzenesulfonate;6-[[(1R,2S)-2-phenylcyclopropyl]amino]pyrimidine-4-carboxamide 2-[1-[(4-hydroxyphenyl)methyl]indol-5-yl]acetamide 4-[2-(ethylamino)ethoxy]-N'-methylbenzenecarboximidamide 4-[(3-fluorophenyl)methyl]-2,6-dimethylmorpholine;ethane 3-[N-(2,3-dihydroxypropyl)-2,6-dimethylanilino]butanoic acid N-[3-ethylsulfonyl-5-(trifluoromethoxy)phenyl]cyclopropanecarboxamide 2,3-difluoro-4-[5-[2-(2-methoxyphenyl)ethyl]-1H-pyrazol-3-yl]pyridine N-[2,4-dichloro-5-(1,3-oxazol-2-yl)phenyl]benzamide 1-(2,6-dimethylphenyl)-7-[4-(1,4,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-9,11-dien-11-ylsulfanyl)anilino]-3,5-dihydro-2H-imidazo[1,2-c]quinazolin-8-ol 3-(N-(2,4,6-trichlorophenyl)anilino)propane-1,2-diol N-[(3R)-piperidin-3-yl]-4,6-dihydro-1H-pyrrolo[2,3-c]pyrazole-5-carboxamide;hydrochloride 2-[(3S,5R)-4-hydroxypiperidin-3-yl]-N-methyl-N-(1H-pyrrolo[3,2-c]pyridin-6-ylmethyl)acetamide 2,5-dinitrobenzoate;ethanesulfonic acid 1-chloro-4-methylbenzene;ethane;formaldehyde;3-[(1Z)-2-hydroxybuta-1,3-dienoxy]propanal;methoxymethane N-[1-aminosulfanyl-3-(2-oxopyrrolidin-1-yl)propan-2-yl]benzamide 2-[(1S)-1-azidoethyl]-4,5-bis(phenylmethoxy)benzonitrile N-[6-(N'-diazenylcarbamimidoyl)pyridin-2-yl]-4-phenylbenzamide 1-[2-(azidomethyl)hexanoyl]-4-(4-cyanophenyl)piperazine-2,6-dione N-[[3-bromo-7-[2-(1,8-naphthyridin-2-yl)ethoxy]quinolin-4-yl]methylidene]hydroxylamine 2-(5-methyl-1,3-oxazol-4-yl)benzamide 3-(3,5-dimethoxyphenyl)spiro[4H-1,3-thiazole-2,5'-oxolane] (Z)-1-cyclohepta-2,4-dien-1-yl-N-phenylmethoxyethanimine;ethane N-butyl-2,4,6-trimethoxy-N-(3-methylbut-2-enyl)aniline 4-[2,6-dinitro-N-(1,3-thiazol-5-yl)anilino]butan-1-ol 2-[azido(phenyl)methyl]-4,5-dichloropyridine 4-methyl-2-[(2E)-penta-2,4-dien-2-yl]-3H-1,8-naphthyridine 2-N,4-N-bis[2,6-di(propan-2-yl)phenyl]cyclohexa-1,3-diene-1,2,4,5-tetramine 6-chloro-4-methoxy-3-[1-(3,5,7-trihydroxy-2H-chromen-2-yl)but-1-enyl]benzene-1,2-diol N-(4-chlorophenyl)sulfanyl-1-[4,6-difluoro-1-(4-methoxybutyl)benzimidazol-2-yl]methanamine 4-[2-(methoxycarbonylamino)phenyl]-1H-pyrazole-5-carboxylic acid 3-[(4R)-3-[(2S)-2-hydroxypropanoyl]-2-oxo-5,6-dihydro-1H-pyrimidin-4-yl]-N'-methylbenzohydrazide 2-[4-chlorobutyl(1,3-thiazol-5-yl)amino]benzenesulfonic acid 4-[4-(cyclohexen-1-yl)phenyl]-2,6-difluorobenzonitrile 1-(azidomethyl)-4-chloro-2,3-diethoxybenzene 7-methoxycarbonyl-5,6-dihydronaphthalene-1-carboxylic acid N-(2,6-diethylphenyl)-3-[4-(3-propan-2-ylpyrazol-1-yl)phenoxy]benzamide N-(4-methylphenyl)-2-[4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carbonyl)piperazin-1-yl]acetamide 3-(1,1-difluoroethyl)-5-[[4-ethanimidoyl-2-methylidene-5-(oxetan-3-ylamino)pyridin-1-ium-1-yl]amino]-N-(3-fluoro-4-morpholin-4-ylphenyl)benzamide 4-[4-(2,3-dimethylpiperidine-1-carbonyl)phenyl]-N,N-diethylpiperazine-1-sulfonamide;2,2,2-trifluoroacetic acid N-azido-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide 1-(2,6-dichlorophenyl)-3-hydroxyurea 2-[4-(1,1-difluoroethyl)phenyl]-5-methyl-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one 5-phenyl-4H-1,3,2-benzodioxazine 4-[2,4-bis(4-methylphenyl)phenoxy]-N'-[5-(trifluoromethoxy)cycloocta-1,3-dien-1-yl]benzenecarboximidamide 1-[(3S)-1-methylpyrrolidin-3-yl]-4H-[1,2,4]triazolo[3,4-d][1,5]benzodiazepine N-benzyl-5-cyclopentyl-3,8,10-triazatricyclo[7.4.0.02,6]trideca-1(9),2(6),4,11-tetraene-12-carboxamide;2,2,2-trifluoroacetic acid 3-[(4-fluorophenyl)methyl]-5-(oxan-2-yloxymethyl)furan 3-hydroxy-2-[(5S)-1-methyl-5,6-diphenylcyclohepta-2,4,6-trien-1-yl]cyclohexan-1-one 3-[(E)-[1,4]dioxino[2,3-f]benzimidazol-2-yliminomethyl]-5-ethoxy-1H-indol-2-ol 2-[[7-(3,5-dimethylpyrazol-1-yl)-1,6-naphthyridin-5-yl]oxy]-N-[(4S)-6-fluoro-2,4-dihydrochromen-4-id-4-yl]-2-methylpropanamide;uranium(2+) 2-(3-chloroanilino)-5-methoxy-1-(6-morpholin-4-ylnaphthalen-2-yl)-6,7-dihydropyrrolo[3,2-c]pyridine-3,8-dione 4-tert-butyl-2-(5,6-dihydrocyclohepta[d]pyrimidin-2-yl)phenol (Z)-4,4-diamino-N'-(5-chloropyridin-2-yl)but-2-enimidamide 3-[4-chloro-2,6-di(propan-2-yl)phenyl]-1-sulfanyl-3H-pyrazole 2-[3-(1H-pyrazol-4-yl)phenoxy]pyrazine 6-(2,4-dimethylphenyl)imino-5-hydroxy-3-methylidene-1,3-benzoxazol-7-amine [2-[(3,5-dimethylphenyl)sulfonylamino]quinolin-6-yl]carbamic acid 2-[4-(benzenesulfonyl)piperazin-1-yl]-N-[(Z)-(5-bromo-3,4-dihydroxynaphthalen-1-yl)methylideneamino]acetamide 1-N'-[4-[2-(5-ethoxycarbonylpyridin-3-yl)ethynyl]phenyl]cyclopropane-1,1-dicarboxamide 4-[(E)-[5-(3,5-dichlorophenyl)sulfanylpyridin-2-yl]iminomethyl]-N-[1-(diethoxyphosphorylmethyl)piperidin-4-ylidene]benzamide 2-N-ethyl-5-(4,8,10-triazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),11-trien-11-yloxy)benzene-1,2-diamine N-(1H-indazol-5-yl)-2,7-diazaspiro[4.4]nonane-7-carboxamide 2-bromo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine;hydrochloride N-[4-(2-cyanoethyl)phenyl]-3,5-dimethyl-1H-pyrazole-4-carboxamide 2-[7-(8-fluoro-1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carbonyl)-4H-azepin-2-yl]acetamide N-(4-bromophenyl)-3-[1-[1-[5-cyano-2,6-dimethyl-4-[1-[2-[2-(oxiran-2-yl)ethoxy]ethoxy]ethylideneamino]phenyl]ethenyl]cyclopropyl]thiophene-2-carboxamide N-[2-(1H-imidazol-5-yl)ethyl]-2-(6,7,8,9-tetrahydro-5H-pyrido[3,4-d]azepin-4-ylamino)benzamide N-[3-(1,4-dihydropyridin-2-yl)phenyl]pyridine-3-carboxamide 1-[4-(2-ethylbutoxy)phenyl]sulfonylpiperidine 5-chloro-3-[(4-methoxyphenyl)sulfanylmethyl]-1H-indole 2-hydroxy-N-[4-(trifluoromethyl)phenyl]benzohydrazide 2-[1-[(2,5-dimethylpyrazole-3-carbonyl)amino]ethyl]-1,3-thiazole-4-carboxylic acid 7-(3,5-dibromo-4-hydroxyphenyl)-6-[4-(3,4-dichlorophenoxy)phenyl]-2-methylsulfanyl-N-phenyl-4,5-dihydroazepine-1-carboxamide 4-hydroxy-3-[(4-methoxyphenyl)sulfonylamino]-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]benzamide 1-azidosulfanyl-3,4,5-trimethoxybenzene 2-[5-[4-(1,3-benzodioxol-5-ylmethylamino)piperidine-1-carbonyl]pyridin-2-yl]acetic acid N-[4-fluoro-3-(5-pyridin-2-yl-1,2-dihydrotriazol-3-yl)phenyl]-3-oxo-1H-pyrazole-5-carboxamide 1-[(2S)-2-(dimethylamino)-3,4-dihydro-2H-quinoline-1-carbonyl]-N'-hydroxyimidazole-2-carboximidamide 5-chloro-2-fluoro-4-[1-methyl-3-(oxan-4-yl)pyrazol-4-yl]oxybenzonitrile 5-(1,2,3,4,6,7-hexahydropyrrolo[2,3-c]pyridine-5-carbonyl)pyridine-2-carbonitrile 4-[1-(2,5-dimethoxyphenyl)sulfinylpiperidin-3-yl]-2-methyl-1H-pyrimidin-6-one 3-[2-(2,4-dimethoxyphenyl)ethyl]-2H-tetrazolo[1,5-a]quinazoline 2-[1-(2,6-dichlorophenyl)ethyl]-4-methoxybenzamide 4-[5-bromo-2,3,6,7-tetrafluoro-1-(1H-pyrrole-2-carbonyl)indol-4-yl]oxybutanoic acid 5-[4-[1-amino-2,3,3a,8b-tetrahydrocyclobuta[b]quinolin-4-yl(cyano)methylidene]piperidine-1-carbonyl]pyridine-2-carbonitrile 1-azidooxy-2,3,4,5,6-pentamethyl-9H-fluorene 4-[6,7-dimethoxy-4-[3-(propan-2-ylamino)pyrrolidin-1-yl]quinazolin-2-yl]-N-pyridin-2-ylbenzamide 2-[4-fluoro-N-(3-methylbut-2-enyl)anilino]-1-phenylethanone N-[(Z)-[4-chloro-2-hydroxy-3-(trifluoromethylsulfanyl)phenyl]methylideneamino]pyridine-4-carboxamide 3-[4-amino-2,6-dibromo-5-(trifluoromethyl)phenyl]sulfanylpropanoic acid 4-[(3S,5R)-7-chloro-5-methyl-2-oxo-1,3-dihydro-1,4-benzodiazepine-3-carbonyl]-N,N-bis(3-chlorophenyl)piperazine-1-carboxamide 4-(6-bromo-4-methoxy-1,3-benzodioxol-5-yl)-2-sulfanylidene-3,6-dihydropyrimido[4,5-d]pyrimidin-5-one 3,5-dichloro-N-[5-(2-hydroxy-6,7-dimethoxyquinoxaline-5-carbonyl)pyridin-2-yl]benzenesulfinamide (4S,5R)-5-amino-2,3-diphenylcyclohexan-1-one 3-[(1,2-dimethoxypropan-2-ylamino)methyl]-N'-hydroxypyridine-2-carboximidamide 2-(3,5-difluoropyridin-2-yl)-N-methoxybutanamide 2-[5-[3-(1,1-difluoroethyl)-4-methoxyphenyl]-6,7-dihydro-1H-pyrrolo[2,3-b]pyridin-3-yl]acetamide 1-[1-(4,5-difluoro-2-propoxyphenyl)ethenyl]azetidine 2-methoxy-N-methyl-6-[3-(propanoylamino)pyrrolidin-1-yl]pyridine-3-carboxamide N-[(1R,2S)-2-(3,4-dihydronaphthalen-2-yl)cyclopropyl]-2-oxo-1H-pyridine-3-carboxamide (E)-N'-butyl-1,3-diphenylprop-2-ene-1,3-diimine (Z)-3-cyclohexyl-N',2-dimethoxy-N-(methylideneamino)prop-2-enimidamide;ethane;4-[(4-hydroxyphenyl)methyl]phenol 4-[5,6,7-trimethyl-2-(4-nitrophenyl)imidazo[1,2-a]pyridin-3-yl]phenol [(1R)-5-[4-hydroxy-3,5-bis(methoxycarbonyl)phenyl]-2,7-dihydro-1H-pyrazolo[1,5-a]pyrimidin-8-yl]-phenylcarbamic acid 3-cyclohexylsulfanyloxy-5,6,7,8-tetrahydronaphthalene-1,2-dione 4-(5-iodohexoxy)benzaldehyde 4-[(3aR,7aS)-2-benzyl-5-[[5-chloro-1-(methoxymethyl)benzimidazol-2-yl]methyl]-1,3,3a,4,6,7-hexahydropyrrolo[3,4-c]pyridine-5-carbonyl]cyclohexane-1-carboxylic acid N'-(3,5-dimethylphenyl)-2-(4-methoxy-6-methylpyrimidin-2-yl)sulfanylethane-1,2-diamine (1S)-6,11-dimethoxy-2-propanoyl-1-[[4-[(3R)-oxolan-3-yl]phenyl]methyl]-1,2,3,4-tetrahydrotetracene-5,12-dione 1-[[4-[(6,7-dimethoxyquinolin-4-yl)methyl]phenyl]methyl]pyrimidine-2,4-dione 3-[(4S,5R)-2-amino-6-oxo-1-(2-phenylethyl)-4,5-dihydropyrimidin-4-yl]benzamide 5-(4-aminophenyl)sulfanyl-2,3-dihydroisoindol-1-one 1-[4-[2-amino-5-chloro-6-(pyridine-2-carbonyl)pyrimidin-4-yl]piperazin-1-yl]ethanone N-[4-[3-(2,6-dioxopiperidin-1-yl)propyl]phenyl]formamide;ethane 1-[5-chloro-6-(difluoromethoxy)pyridin-3-yl]butan-1-one 4-methylsulfanyl-2,3,5-trinitrophenol 2-amino-6-ethoxy-4-(2-hydroxynaphthalen-1-yl)-4H-pyran-3,5-dicarbonitrile 5-chloro-4-[(1S)-2,3-dihydro-1H-inden-1-yl]-6-methoxypyrimidin-2-amine;ethane (2E,4Z)-4-methylhepta-2,4-dien-3-amine;N'-[3-[2-(6-phenylpyridin-3-yl)ethynyl]imidazo[1,2-b]pyridazin-7-yl]methanediamine 4-[2-(cyclohexanecarbonylamino)phenyl]-N-methylbenzamide 5-[2-(6-fluoro-1H-indol-3-yl)ethylsulfamoyl]pyridine-3-carboxylic acid 3-butyl-2-hydroxybenzimidazole-1,5-dicarboxylic acid 5-[(2S,4R)-1-ethyl-6-oxo-2-phenylpiperidine-4-carbonyl]pyridine-3-carboxylic acid 5-bromo-3-[1-(cyclopropylmethyl)piperidin-4-yl]oxypyridazine [2-methoxy-5-(trifluoromethyl)anilino]-oxoazanium ethane;2-methylimino-N-[1-(5-nitropyridin-2-yl)piperidin-4-yl]butanamide 5-[1-(4-chlorophenyl)ethylamino]-N'-hydroxypyridine-2-carboximidamide 1-(3-pyridin-2-ylpyridin-4-yl)oxy-N-[2,3,5-tris(trifluoromethylsulfanyloxy)phenyl]ethanimine (1S)-N',2-diphenylethanesulfonohydrazide 3-[2-methylpropanoyl(1,2,4-triazol-4-yl)amino]butanoic acid 2-[N-(3-nitrophenyl)-4-(quinoxalin-2-ylsulfamoyl)anilino]acetamide (4-fluoro-5,6-dihydronaphthalene-2-carbonyl)chloranium (3S)-4-[(1R,6R)-2-(propoxymethyl)-1,3-diazabicyclo[4.1.0]heptan-3-yl]-3-quinoxalin-7-ylbutanenitrile N-[3,5-dichloro-4-(8-fluoro-2,3,6,7-tetrahydroquinolin-1-yl)phenyl]-3,3,3-trifluoropropane-1-sulfonamide [(1E)-1-[4-[4-(5-aminopyridin-2-yl)piperazine-1-carbonyl]phenyl]buta-1,3-dienoxy]methanol;ethane 3-[3-(azidomethyl)phenyl]-1,2,4-oxadiazole 1-(2,6-dichlorophenyl)-4-[4-ethyl-3-(trifluoromethyl)pyrazol-1-yl]piperidine 6-[2,3-bis(methylsulfanyl)phenyl]pyridine-2,4-diamine;dichloroiron 2-(4-fluorophenyl)-1-[[2-[2-(4-methylpiperazine-1-carbonyl)pyrrol-1-yl]acetyl]amino]cyclopropane-1-carboxylic acid 4-(2,6-dihydroxyphenyl)-3-methoxybenzaldehyde 1-benzyl-5,6-bis(ethenyl)imidazole-2-carboxamide 6-[3,4-dimethyl-2-oxo-5-(trifluoromethyl)imidazol-1-yl]hexanoic acid (Z)-N'-[7-amino-2,4-dioxo-1-(pyridin-3-ylmethyl)pyrido[3,4-d]pyrimidin-3-yl]ethene-1,2-diamine N-(2,3-dihydrofuro[3,4-b][1]benzofuran-5-ylmethyl)-N',N'-diethylpropane-1,3-diamine 2-[3-(3,5-difluorophenyl)propyl]-6-iodopyridine N-(3,4-dihydro-2H-chromen-7-ylmethyl)-5-thiophen-3-yl-1,3,4-thiadiazol-2-amine N-[2-[4-(1,3-dihydroisoindol-2-yl)-7H-pyrrolo[2,3-d]pyrimidine-6-carbonyl]cyclohexyl]-2-fluorobenzenesulfonamide 2-[6-ethylsulfinyl-5-(7-methoxy-1,3-benzodioxol-5-yl)pyridin-3-yl]-7-(trifluoromethyl)imidazo[1,2-a]pyridine N-[(1R,2S)-4,6-dimethyl-2-(3-oxo-1H-isoindol-2-yl)cyclohex-3-en-1-yl]-5,7,8-triazaspiro[3.5]nonane-2-carboxamide 2,3-dimethyl-N-[5-methyl-6-(2-methylbenzimidazol-1-yl)pyrimidin-4-yl]butanamide 3-[4-(aminomethyl)phenoxy]-N-[5-(cyclohexen-1-yloxy)pentyl]benzamide 1-(1,3-dimethylpyrazole-4-carbonyl)-3-(hydroxymethyl)-N-phenylazetidine-3-carboxamide N-[3-(4-aminobutyl)phenyl]-1,5-naphthyridine-2-carboxamide 5-[2-(1,3-benzodioxol-4-yl)imidazol-1-yl]-1H-indole 2-[4-[5-methoxy-6-(3,3,5,8,8-pentamethyl-1-oxo-7H-2-benzofuran-5-yl)pyridin-2-yl]sulfonylphenyl]-N-methylbenzamide N-(2-azidophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide 1-azidosulfanyloxynaphthalene N-(4-bromobutan-2-yl)-3-methoxy-N-(6-nitro-1,3-benzothiazol-2-yl)aniline 6-[4-(3,5-ditert-butylphenyl)-5-ethynylthiophen-2-yl]-9-methoxy-8a,10,11,12a-tetrahydroindolo[3,2-c]carbazole 1-[(1R,3R)-3-methylcyclohexyl]-2-[4-[6-methylidene-5-[(Z)-prop-1-enyl]pyridazin-1-yl]phenyl]ethanone 2-(methylamino)-1,3,4,5-tetrahydro-[1]benzothiepino[6,5-c]pyridine-11,12-dione 3-chloro-4-[2-[(4,6-dichlorocyclohexa-1,5-dien-1-yl)carbamoyl]benzimidazol-1-yl]benzoic acid 5-[1,2,3,6-tetramethyl-5-(4-methylphenyl)cyclohexa-2,4-dien-1-yl]benzene-1,3-diol 6-(3,5-dimethylbenzene-6-id-1-yl)-4-(trideuteriomethyl)furo[2,3-b]pyridine;(Z)-6-hydroxy-3,7,8,9-tetrahydropyrimido[2,1-b][1,3]benzoxazine;iridium 2-(2,5-dimethylphenyl)-1,3-benzoxazole;ethane 3-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridine-2-carbonyl]benzaldehyde [4-(3-bromophenyl)piperidin-1-yl]-(6,7-dimethoxyquinazolin-4-yl)methanone 2-cyclopropyl-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridine;3,4-dimethoxybut-1-ene 4-[3-[1-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperidin-3-yl]-2-oxopropoxy]benzonitrile 2-[4-(cyclohexylcarbamoyloxy)phenyl]sulfonylacetic acid 4-[3-(7-ethylazepine-1-carbonyl)phenyl]piperidine-1-carboxylic acid N-[1,3-bis(4-fluorophenyl)cyclobutyl]-2-methoxyacetamide 3-(4-chlorophenyl)-2,3-dimethylhexanal 1,2-dichloroethane;(2Z)-3,4-dimethylpenta-2,4-dienal;ethane;N-[2-methoxy-5-(3-methylhexan-3-yl)phenyl]methanethioamide;3-methylpyridine 2-[4-[(2,6-difluorobenzoyl)amino]phenyl]acetic acid 2-(6,7-dihydro-1H-indole-3-carbonyl)-N-ethylsulfonylbenzamide N-azido-2,6-difluoro-4-methylsulfonylaniline (4R)-3,7,8-trihydroxynaphthalene-2,5-dicarboxylic acid 5-amino-N-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyrazine-2-carboxamide 1-[(3,4-dimethoxyphenyl)methyl]-5-ethynyl-N-methyl-N-propan-2-ylindazole-6-sulfonamide 2-[3-(4-azidooxyphenoxy)propyl]-5-butyl-1,3-dimethylbenzene 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethanone 1-(2-ethylcyclohexyl)indole-3,4-dione 5-[4-methoxy-2-(4-methylphenyl)sulfonylsulfanylpyrimidin-5-yl]-1-morpholin-4-ylpentane-1,3-dione N-[4-(2,3-dihydropyrazine-5-carbonyl)phenyl]-6-(trifluoromethyl)pyridazine-3-carboxamide [3-amino-4-(2,4-dichlorophenyl)pyrrolidin-1-yl]-(3-pyrimidin-2-yloxyphenyl)methanone 3-methyl-N'-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)pyridine-4-carbohydrazide [(E)-5-amino-1-cyclobutylsulfanyl-3-(oxan-4-yloxy)pent-2-enylidene]-(5-chloropyridin-3-yl)azanium 2,3-dichloroprop-1-ene;6-[(Z)-(4-nitrophenyl)methylideneamino]iminocyclohexa-1,3-dien-1-ol (6R)-7-acetyloxy-3-[(3,4-dichlorophenyl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate 7-amino-3-[1-(4,6-dimethyl-2-oxochromen-7-yl)ethoxycarbonyl]thieno[3,2-b]pyridine-2-carboxylic acid N-[5-(2,4-dioxopyrimidin-1-yl)-2,3-dihydrothiophen-2-yl]-2-methylpropanamide 1-azidooxy-4-(cyclopropylmethyl)benzene (E)-2,4-dimethylpent-2-enoic acid;7-ethoxy-3-[3-methyl-4-[[1-(pyrrolidin-3-ylideneamino)piperidin-3-yl]methoxy]phenyl]quinazolin-4-one 4-[4-(3-methylphenyl)pyridin-1-ium-2-yl]benzene-1,3-diol;sulfate 2-fluoro-4-[1-hydroxy-5-(oxolan-3-yl)-3,6-dihydro-2H-pyridin-4-yl]phenol 6-[2-[3,5-dichloro-4-(3-ethylsulfanylpropoxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,4,4a,9a-tetrahydropyrido[3,4-c]azepine 6-methoxycarbonyl-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylic acid 4-[(3-aminoazetidin-1-yl)methyl]-5-methoxy-2,6-dimethylpyridine-3-carbonitrile 2-[(1R)-3,5-bis(phenylmethoxy)cyclohexyl]ethanol 1-(2,3-dimethylphenyl)sulfinyl-5-ethylsulfonyl-4-[[6-(trifluoromethyl)pyridin-3-yl]amino]pyrazole-3-carboxylic acid N-[2-(4-bromophenyl)ethyl]-1,3-dichloro-9H-pyrido[3,4-b]indole-6-carboxamide 4-[2,5-dimethyl-3-oxo-7-(trifluoromethoxy)pyrazolo[4,3-c]quinolin-8-yl]sulfanylbutanehydrazide 3-(3,4-difluorophenyl)-2H-furo[2,3-d]pyrimidine 2-[(4Z,5E)-5-ethylidenesulfanylhepta-1,3,6-trien-3-yl]quinazolin-4-amine 1-(4-methoxy-3,5-dimethylphenyl)-2-nitroguanidine [3-fluoro-4-[(5E)-2,7,7-trimethyl-6H-2,3-naphthyridine-3,9'-diaza-1-carbonyl]phenyl]boronic acid 1-(2,4-dimethoxyphenyl)-5-imino-3-[2-(5-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]imidazolidine-2,4-dione N-(3,5-dibromophenyl)-2-[6-(oxolan-2-ylmethoxymethyl)pyridin-2-yl]acetamide 2-chloro-N,N'-dimethyl-N-[(E)-5-phenylpent-3-en-1-ynyl]ethanimidamide 2-[7-[3-(dimethylamino)azetidin-1-yl]-5,6-difluoro-1H-indole-2-carbonyl]pyridine-4-carboxylic acid 1-[4-methyl-3-(2-methylbutan-2-yl)phenyl]propan-1-one 4-(1,3-dioxoisoindole-2-carbonyl)-N-[(E)-1H-imidazol-5-ylmethylideneamino]benzenesulfonamide 2-[(2S)-1-(cyclohexanecarbonyl)pyrrolidin-2-yl]-6-[(4-methoxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 6-[4-(3,5-diethylpyrazole-1-carbonyl)piperazin-1-yl]pyridine-2-carboxamide 3-(2-chlorocyclohexa-1,5-dien-1-yl)oxyphenol N-[2-(4-hydroxyphenoxy)ethyl]-2,3-dihydro-1H-indene-5-carboxamide (3S,4R)-1-[4-cyano-5-(cyclobutylmethoxy)pyrimidin-2-yl]-4-(4-ethenylphenyl)piperidine-3-carboxylic acid N-[3-(1H-benzimidazol-2-yl)propyl]-4-oxo-7,8-dihydro-6H-pyrano[2,3-e][1,3]benzothiazine-2-carboxamide 4-methyl-3-[2,7,8-trifluoro-5-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]phenol N-[5-[3-(4-piperidin-1-yl-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-yl]cyclohexanecarboxamide 2-[4-(chloromethyl)phenyl]-1-phenoxyethanol 2-bromo-6,9,15-triazatetracyclo[8.6.0.03,8.011,15]hexadeca-1(10),3,5,7,11,13-hexaen-16-one 6-[(4R)-4-methyl-2-oxo-1,3-oxazolidin-3-yl]-5H-cyclopenta[f]benzimidazole-7-sulfonamide 1-[2,6-difluoro-4-(propan-2-ylamino)phenyl]piperidine-4-carboxylic acid N-[(2,5-dimethoxyphenyl)sulfonylmethyl]-1-piperidin-4-yltriazole-4-carboxamide;hydrochloride 1-methoxy-3-[2-(2-propylphenyl)phenoxy]benzene 2-[(5S)-3-(1,2,4-oxadiazol-3-yl)-7-oxo-6H-triazolo[4,5-d]pyrimidin-5-yl]acetic acid (2S)-2,5-diamino-N-[(Z)-(5-bromo-2-hydroxyphenyl)methylideneamino]pentanamide 2-[1,4-dimethyl-3-[(2Z)-penta-2,4-dienyl]-6H-xanthen-9-yl]-5-methoxybenzoic acid N-[4-[1-(butanoylamino)ethyl]phenyl]-2,3,6,7-tetrahydroazepine-4-carboxamide 3-fluoro-4-[(5Z)-2-hydroxyimino-5-[[5-nitro-1-(4-sulfophenyl)pyrazol-4-yl]methylidene]-1,3-thiazolidin-3-ium-3-yl]butane-1-sulfonic acid 4-[4-(trifluoromethyl)anilino]-N'-(2,4,6-trichlorophenyl)benzohydrazide [5-(1H-pyrrol-2-yl)pyrazol-3-yl]methanethiol N-[3-(3,4-dichlorophenyl)propyl]-1-(4-ethoxyphenyl)methanesulfonamide N-[2,4-difluoro-3-[5-(1H-pyrazolo[3,4-c]pyridin-7-yl)thiophen-2-yl]phenyl]-3,5-dimethoxybenzamide N-[1,3-dimethyl-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-3-yl]-1-[2-[ethyl(propyl)amino]ethyl]piperidine-4-carboxamide 4-azidosulfanyl-2-(3-methoxypropyl)-1H-indole 5-[(3R)-3-methylpiperazin-1-yl]quinoline (2S)-N-azido-N'-[4-methoxy-3-(3-methylbut-1-ynyl)phenyl]pentanediamide 5-(2,4-dimethylphenoxy)-N'-hydroxypyrazine-2-carboximidamide N-(1,5-dimethylbenzimidazol-2-yl)-4-[(3S)-3-hydroxypyrrolidine-1-carbonyl]benzenesulfonamide 4-N-[2,4-dimethyl-5-(3-phenylbutanoylamino)phenyl]-6-N-[(1Z,3Z)-penta-1,3-dienyl]-1H-imidazole-4,6-dicarboxamide 2-[4-hydroxybutyl(2H-tetrazol-5-yl)amino]octanoic acid 1-(2,4-dimethoxyphenyl)-3-fluoropyrrolidine 3-amino-1,4-dioxonaphthalene-2-sulfonic acid (3-fluorophenyl)-(8,9,10,11-tetrahydroimidazo[2,1-a]benzimidazol-1-yl)methanone 5-(4-fluorocyclohexa-1,3-dien-1-yl)-2-methyl-7-[methylsulfonyl(propanoyl)amino]pyrazolo[1,5-a]pyrimidine-6-carboxamide N-[(E)-[2-methoxy-6-[(Z)-2,3,4,5,6-pentafluorohex-3-enyl]phenyl]methylideneamino]-1,3-benzothiazol-2-amine N-[3-(diethylamino)propyl]-6,7-bis(methoxymethyl)quinoxaline-2-carboxamide 1-(3,5-difluorophenyl)-2-[3-(1-methylcyclopenta-2,4-dien-1-yl)propyl]-3-oxo-N-[(4-pyridin-2-ylphenyl)methyl]pyridazine-4-carboxamide N-(1,3-benzodioxol-5-ylmethyl)-2-(3,4-dimethoxyphenyl)morpholine-4-carboxamide 2-[4-(5,7-dimethyl-1,3-benzothiazol-2-yl)-5-imino-2H-thiophen-3-yl]propan-1-ol 4-(6-azidohexyl)benzenesulfonic acid [1-hydroxysulfanyloxysulfanyl-2,2,6-trimethyl-4-(5-nitrofuran-2-yl)heptan-4-yl]carbamic acid 3-[1-(2,4-dimethylpentanoyl)piperidin-4-yl]-5-fluoro-1H-benzimidazol-2-one 3-methyl-6-oxo-7H-[1,2]thiazolo[5,4-b]pyridine-4-carboxylic acid 7-(4-methoxyphenyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole;hydrochloride 2-hydroxy-1,5-dimethylpyrrole;platinum(2+);quinolino[7,8-h]quinoline (4-amino-2-chloro-3-fluorophenyl)-[5-hydroxy-7-methyl-6,8-dioxo-5-(pyrrolidine-1-carbonyl)-5H-naphthalen-2-yl]azanium 5-bromo-2,6-difluoro-N'-hydroxypyridine-3-carboximidamide 6-[5-(cyclopentylmethyl)-3,4,6,7,8,9-hexahydropyrazino[1,2-a]indol-10-yl]-N,3-dimethyl-2H-pyrrolo[3,2-c]pyridine-1-carboxamide 6-[5-[(2E,4Z)-hepta-2,4-dien-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-1,3,3a,4,9b-hexahydrobenzo[f]indol-2-one 2-(4-butylphenyl)-N'-propan-2-ylacetohydrazide;hydrochloride (E)-4-[2-(aminomethyl)phenyl]but-3-enoic acid N-[3-(5,6-dihydrobenzo[b][1]benzazepine-11-carbonyl)phenyl]prop-2-enamide 4-[2-(4-propan-2-ylphenyl)butyl]benzoic acid 4-[2-[3,5-dimethyl-1-(1H-pyrrole-2-carbonyl)pyrazol-4-yl]-1,1,1,3,3,3-hexafluoropropan-2-yl]-N,N-dimethylbenzamide 2-(2-methyl-1,3-dioxol-4-yl)-5-propan-2-ylbenzotriazole 6-(4-methylphenyl)sulfonylnaphthalene-2,3-dione 3-[(4-ethylphenyl)methylamino]piperidine-2,6-dione (E)-2-cyano-3-cyclohexyloxy-3-[4-hydroxy-2-methoxycarbonyloxy-5-[2-(2-oxoethylamino)phenyl]phenyl]prop-2-enoic acid 4-amino-1-(3,4-dimethylphenyl)-N-[[6-(trifluoromethoxy)pyridin-2-yl]methyl]pyrazolo[3,4-d]pyrimidine-3-carboxamide N-[2-methyl-4-(trifluoromethyl)phenyl]-3,7-dihydropyrrolo[2,3-d]pyrimidine-4-carboxamide 5-[1-(2,3-dihydro-1H-inden-5-ylsulfonyl)piperidin-4-yl]-3H-1,3a,4,6a-tetrahydropyrrolo[3,4-c]pyrrole;hydrochloride 2-chloro-4,7,8-trimethyldibenzofuran 5-chloro-3,4-dihydro-1H-naphthalene-2,7-disulfonate 4-[(3S,4R)-4-methoxy-1-[3-methyl-5-(trifluoromethyl)benzoyl]pyrrolidine-3-carbonyl]-2H-phthalazin-1-one 2-[(3Z)-5,6-difluoro-2-methylidenehepta-3,5-dienyl]-1-ethenyl-4-(methoxymethoxy)benzene 1-cyclopropylsulfonyl-4-[(2,4-difluorophenyl)methoxy]-3-hydroxypyridin-2-one 3-[3,4-bis(ethenyl)-2H-chromen-8-yl]propanoic acid 4-[6,7,8-trifluoro-3-methoxy-2-[1-(6-methylpyridin-2-yl)propyl]quinolin-5-yl]morpholine 2-(6-chloro-1,3-benzodioxol-5-yl)-N-[4-(3-fluorophenyl)-3-hydroxybutan-2-yl]acetamide 6-[(1S)-2-cyclobutyl-7-methoxy-3H-inden-1-yl]-4-oxoheptanoic acid 1-[[6-[3-(4-cyclopentyloxyphenyl)propanoylamino]pyridine-2-carbonyl]amino]cyclohexane-1-carboxylic acid 4-chloro-N-[2-(diethylamino)pyrimidin-5-yl]benzamide N-methoxy-2-(4-propan-2-ylphenyl)-1,3-thiazole-5-carboxamide (E)-3-[4-[(2,5-dioxopyrrol-1-yl)methoxy]phenyl]-N-(4-methoxy-2-nitrophenyl)prop-2-enamide 1-[6,7-bis(ethenyl)-4-methoxyquinolin-3-yl]ethanone 3-[(4E)-6,7-difluorohepta-1,4,6-trien-2-yl]-5-pyridin-4-yl-1H-pyrrolo[3,2-b]pyridine;ethane 5-(4-aminophenyl)imino-3H-thieno[2,3-d]pyrimidin-4-one 1-[(2,4-dichlorophenyl)methylamino]piperidine-3-carboxamide 5-[(4-methoxyphenyl)methyl]-2-methylidene-1H-pyridine 1-(diaminomethylideneamino)-3-[2,6-dichloro-4-(trifluoromethyl)phenyl]thiourea 5-[5-chloro-2-(tetrazol-1-yl)phenyl]imino-8,8a-dihydro-4aH-naphthalene-2-sulfonic acid 2-[5-(2,5-difluorophenyl)pyrazolo[3,4-b]pyridin-1-yl]acetamide 1-(3,4-dimethoxyphenyl)sulfonyl-3-methylurea 4-azido-2-(3,5-difluorophenyl)pyridine N-methyl-2-[3-(3-oxobutanoylamino)phenyl]acetamide 4-(4-chlorobenzoyl)-N,3-dimethylpiperazine-1-carbothioamide 3-(3-aminophenyl)sulfanyl-5,6-dimethoxy-2-methylaniline 4-[[(1R)-3-bromocyclohexyl]amino]quinoline-6,7-diol 4-[2,6-dimethylmorpholin-4-yl(pentanoyl)amino]benzamide 6-methoxy-2-methylsulfonyl-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)pyrimidine-4-carboxamide N-[(2,4-dichloropyrimidin-5-yl)methyl]-1H-imidazo[4,5-c]pyridine-7-carboxamide 5-cyclopentyl-2,4-dioxo-6-[3-(trifluoromethoxy)phenyl]-1H-pyrimidine-6-carbonitrile 5-bromo-2,3-dihydropyrido[4,3-b][1,4]oxazine 4-(4-methylphenyl)sulfonylmorpholine 6-[1-(2,4-difluorophenyl)ethoxy]-3-iodoimidazo[1,2-b]pyridazine 3-[5-bromo-2-(methoxycarbonylamino)phenyl]sulfanylpropyl-cyclobutylcarbamic acid 2-[3-(4-chlorophenyl)-6-ethyl-5-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-7-yl]acetamide 4-[1-methyl-5-(2H-tetrazol-5-yl)pyrrole-3-carbonyl]-N-[2-oxo-2-(2,2,2-trifluoroethylamino)ethyl]piperazine-1-carboxamide 5-(2,3-difluorophenyl)-1H-pyrazole;ethane 2-[5-(4,4-dimethylcyclohexen-1-yl)pyrazolo[3,4-b]pyrazin-2-yl]-3H-isoindole 4-[2,6-bis(3-methylphenyl)phenyl]-1H-1,2,4-triazole 1,5-dimethyl-3-(trifluoromethyl)pyrazole;3,4-dimethylbenzenethiol;4-methylpiperidine [3-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]phosphane 4-(4-ethenylphenyl)-6,8-dinitrodibenzothiophen-2-amine 6-(2-cyclopropylacetyl)-2-[1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-(4-ethenylcyclohexyl)-1,2-difluoro-7-[6-(fluoromethoxy)naphthalen-2-yl]phenanthrene (5E)-2-phenylimino-5-[(4-propan-2-yloxyphenyl)methylidene]-1,3-thiazolidin-4-one 1-[3-(4-chlorophenyl)-4,5-dimethylthiophen-2-yl]ethanone 7-(1,3-benzodioxol-5-ylmethylidene)-2-[4-cyano-3-(trifluoromethyl)phenyl]-N,N'-bis(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecane-8-carboximidamide 4-chloro-6-(2,3-dihydrofuran-5-yl)pyrrolo[1,2-b]pyridazine 2-[4-(3,5-dimethylpiperidin-1-yl)phenyl]-5-methoxy-3-phenylpyrazine;ethane 1-[1-(4-butoxyphenyl)ethenyl]naphthalene 2-[3,5-bis(trifluoromethyl)phenyl]quinoline [4-(cyclopropylamino)-6,7-dihydropyrrolo[3,2-d]pyrimidin-5-ylidene]methanolate 4-[2,3-dihydroxypropyl(1,1,1,2,3,3,3-heptafluoropropan-2-yl)amino]benzenesulfonic acid N-[5-(cyclopropylcarbamoyl)-2,4-difluorophenyl]carbamate N-[(2-chlorophenyl)methyl]-4,5-dihydropyrazolo[1,5-a]pyridine-3-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-chloro-4,6-dinitroaniline 4-(furan-3-ylmethylamino)-1-(1-propan-2-ylpyrazol-4-yl)pyrrolidin-2-one;2,2,2-trifluoroacetic acid N-[2-(6-azidopyridin-3-yl)-4,5-dimethoxyphenyl]acetamide (4-azidopiperidin-1-yl)-[3-[4-[2-(dimethylamino)ethoxy]phenyl]-5-methylthiophen-2-yl]methanone 6-methoxy-4,9-dimethylacridine 6-azido-2-(4-nitrophenyl)pyridine 2-[2-(7H-purin-6-ylsulfanylmethyl)phenyl]benzonitrile (Z)-2,3-bis[3,5-dichloro-4-(naphthalene-1-carbonyloxy)phenyl]prop-2-enoic acid 3-[(2R,5S)-4-hydroxy-5-[(E)-3-oxo-3-phenylprop-1-enyl]oxolan-2-yl]propanenitrile N-[(1R,2S)-3-hydroxy-2-pyrazol-1-ylcyclobutyl]pyrazine-2-carboxamide N-[(3,5-dibromo-2,4-dihydroxyphenyl)methylideneamino]pyridine-4-carboxamide (E)-3-[3,4,5-trifluoro-2-hydroxy-6-[methyl-(2,3,4,5-tetradeuteriophenyl)sulfonylamino]phenyl]prop-2-enoic acid [4-[(2,6-dichlorobenzoyl)amino]naphthalen-1-yl]azanium 3-[2-[[4-[(4Z)-1-amino-5,5-difluoro-4-[[5-methoxycarbonyl-6-(trifluoromethyl)pyridin-2-yl]carbamoylimino]pentan-2-ylidene]piperidine-1-carbonyl]-cyclopropylamino]ethoxy]cyclobutane-1-carboxylic acid 2,4-dibutyl-6-methoxyphenol 4-(2,6-difluorophenyl)imino-1-[[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]methyl]pyrrolidine-3-carboxamide 1-ethyl-7-[2-(pyridin-4-ylmethoxy)phenyl]-5,6-dihydropyrrolo[3,4-b]pyridine 4-N-[1-[(2R,5S)-3,6-dihydro-2H-pyran-2-yl]ethyl]pyrimidine-4,6-dicarboxamide (3R)-3-[4-[[5-(2,6-difluorophenyl)-1,3,4-oxadiazol-2-yl]amino]phenoxy]pyrrolidine-1-carboxylic acid 4-[(3S)-1-[3-(cyclopropylmethoxymethyl)benzoyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one 2-(3,5-dimethoxyphenyl)cyclohexa-1,4-dien-3-yn-1-ol 2-[[4-(3,5-dimethylpyrazol-1-yl)phenoxy]methyl]propanedioic acid 5-[2-chloro-4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-1-ethyl-3-methylpyrazole-4-carboxamide 4-[2-azido-3-(trifluoromethyl)phenyl]morpholine 4-benzyl-N-[5-[(6-fluorocyclohexa-2,4-dien-1-ylidene)methoxy]pyrimidin-2-yl]piperazine-1-carboxamide 1,6-dibromonaphthalene;dichlorozirconium(2+) N-methyl-1-[2,3,4-tris(trifluoromethoxy)phenyl]methanamine 4-chloro-7-methyl-1,3-benzothiazole;3-[[2,4-dihydroxy-5-(pyridine-4-carbonyl)phenyl]sulfonylamino]-N-ethylpropanamide 6-[2,4-bis(phenylmethoxy)pyridin-3-yl]-N-[1-[5-methanimidoyl-6-oxo-4-(propylideneamino)pyrimidin-1-yl]propan-2-yl]imidazo[1,2-a]pyrazine-8-carboxamide 1-(5-chloro-6-ethylpyrimidin-4-yl)-2,3-dihydroindole 5-[4-(3,5-dimethylthiophen-2-yl)phenyl]imidazolidine-2,4-dione N-[1-(7-propan-2-ylquinolin-4-yl)piperidin-3-yl]ethanesulfonamide 5-[2-(difluoromethyl)phenyl]-4-imino-1-propanoylpyrrolidin-2-one 4-amino-3,5-dichloro-N'-hydroxybenzenecarboximidamide 2-[4-[(Z)-[2-(4-bromophenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]phenoxy]acetonitrile 4-chloro-2-[6-(dimethylamino)pyridin-3-yl]benzamide (Z)-3-[4-chloro-2-hydroxy-5-(morpholine-4-carbonyl)phenyl]-2-cyanoprop-2-enamide 2-methyl-4-(4-methylpiperazin-1-yl)pyrido[3,4-d]pyrimidine 2-azido-5-(1,2,3-trimethylcyclopropyl)pyridine 6-[2-fluoro-4-(trifluoromethyl)phenyl]-N,N-dimethylhexan-1-amine 1-ethoxycarbonyl-3,4,6,7,8,9-hexahydro-2H-carbazole-3-carboxylic acid N-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-2-ethoxybenzamide 2,2-dimethylbutane;4-[5-(3-ethenoxypropoxy)pyridin-2-yl]-N-[2-(methylideneamino)phenyl]piperazine-1-carboxamide 2-(2,3-dihydro-1H-inden-5-ylmethoxy)-4,4,6,7-tetrafluoro-1,3-dioxoisoindole-5-carboxylic acid 2-methylsulfanyl-1H-imidazo[4,5-b]pyridine-7-carboxylic acid [3-(1,2-benzothiazol-6-yl)-1H-indazol-5-yl]boronic acid N-(4,4-difluorocyclohexyl)-4-methoxypyrazolo[1,5-a]pyridine-2-carboxamide 2-[7-(4,6-dimethylpyridin-3-yl)imidazo[1,2-a]pyridin-3-yl]-N-ethoxyacetamide N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)ethyl]-3,3,4,4,4-pentafluorobutanamide 1-[5-(2,4,6-trimethylphenyl)thiophene-2-carbonyl]cyclopropane-1-carboxylic acid N-[5-(3,4-dimethylcyclohexa-1,3-dien-1-yl)pyridin-2-yl]-3-hydroxy-4-nitrobenzamide 2-[N-[(4-chlorophenyl)methyl]-3-cyanoanilino]pyridine-3-carboxylic acid N-[2-(hydroxymethyl)phenyl]-3H-benzimidazole-5-carboxamide (2R)-1-[(1R,3S)-1-fluoropentoxy]-3-methyl-2H-naphthalene 2-[1-(5,6-difluoro-3H-indole-2-carbonyl)azetidin-3-yl]oxy-N,N-dimethylacetamide 3-[4-(6,7-dimethoxyquinazolin-2-yl)phenyl]-5-(trifluoromethyl)imidazolidine-2,4-dione 6-[[4-(azidomethyl)pyrazol-1-yl]methoxy]naphthalene-2-thiol N-(2,5-dichlorophenyl)-2-[4-hydroxy-5-oxo-3-(thiophen-2-ylmethylideneamino)-1H-pyrazol-2-yl]acetamide 5-cyclopentyl-1-cyclohexylpyrazole-3-carboxylic acid 5-[1-(2-carboxyethyl)pyrazol-4-yl]furan-2-carboxylic acid N-(2,3-dihydro-1H-inden-2-yl)-4-methoxyaniline 2-[[4-[(3,5-dimethoxyphenyl)methyl]piperazine-1-carbonyl]amino]acetic acid 2-[(6R)-2,4-dimethyl-5,8-dioxo-6-phenyloctanoyl]benzaldehyde;methoxymethane 2-(4-bromo-3,5-dimethylphenyl)pentanoic acid (2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-1,4-dioxane-2-carboxamide N-methyl-3,4,5-tripropoxybenzamide 4-[5-ethylsulfonyl-6-(1,3-thiazol-2-yl)pyridin-3-yl]-N-[2-methoxy-4-[(1S)-1-(oxolan-3-ylamino)butyl]phenyl]-1,3,5-triazin-2-amine 1-(2,6-dimethylphenyl)-3-[4-[4-[N'-(1-morpholin-4-ylethenoxymethyl)carbamimidoyl]phenyl]phenyl]urea 2-[3-(5-tert-butylcyclohexa-1,3-dien-1-yl)phenyl]-4,4,5,5-tetramethyloxaborolane [1-(4-aminophenoxy)-3,7-dihydrodibenzothiophen-2-ylidene]cyanamide 1-[2,6-bis(methylsulfanyl)pyrimidin-4-yl]propane-2-thiol 2-(2,5-dimethylphenyl)-3-[(E)-2-[6-[1-(1H-indol-4-ylamino)ethenyl]quinolin-8-yl]ethenyl]-5,5-dimethylimidazol-4-one 5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-7-yl)pentane-2,4-dione 3-(methoxymethyl)-1-(4-phenylphenyl)sulfonyl-2,5-dihydroindole 3-cyclopentyloxy-N'-hydroxypyridine-4-carboximidamide 2-methyl-5,7-dihydrobenzo[d][1]benzazepine 6-ethoxy-3,4-dimethyl-2H-pyrazolo[3,4-b]pyridine 1-(4-methylphenyl)-5-[4-(trifluoromethoxy)phenyl]pentane-1,3-dione 6-chloro-2-[3,5-dichloro-4-(3-ethoxycarbonylpiperidine-1-carbonyl)phenyl]-3,7-dioxo-4H-pyrido[4,3-d]pyrimidine-8-carboxylic acid N-(2,6-dichlorophenyl)-1-[(4-methylsulfanylphenoxy)methyl]cyclobutane-1-carboxamide;4-(3,5-difluorophenyl)pyridine 5-[(3S,4R)-1-methyl-4-(2-oxocyclopentanecarbonyl)piperidine-3-carbonyl]-N-pyridin-2-yl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide 4-[(3-propan-2-yl-1,2,4-thiadiazol-5-yl)iminomethyl]benzene-1,2-diol 5-[4-(3,3-dimethylbutoxy)-2,6-difluorophenyl]imidazolidine-2,4-dione 2-(2,6-dioxopiperidin-3-yl)-5-[4-(oxan-4-ylmethoxy)butoxy]isoindole-1,3-dione 2-(5,6,7,8-tetrahydro-4H-[1,3]thiazolo[5,4-b]indol-2-yl)benzoic acid 5-[4-methyl-6-[(Z)-pent-2-en-3-yl]pyrimidin-2-yl]cyclohexa-1,3-diene-1-carbonitrile 2-[(Z)-but-1-enyl]-5-[(5Z,7E)-8,10-difluoro-9-iminohepta-1,3,5,7-tetraenyl]benzonitrile 1-(3,4-dichlorophenyl)-2H-pyridine 2-(5-chloropyridin-2-yl)-1-[4-(2,6-dimethoxyphenyl)piperidin-1-yl]ethanone 1-[4-[[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]iminomethoxymethyl]naphthalen-1-yl]-3-ethylurea N-(3,5-dichlorophenyl)-N-ethylsulfonylbenzamide 6-[2-[(1S)-cyclohex-3-ene-1-carbonyl]-5-methoxyphenyl]-5-methylpyridine-2-carboxylic acid N-[[2-amino-4-(4-chlorophenyl)-6-(4,5-dihydro-1H-imidazol-2-yl)-4-methylcyclohexa-1,3-dien-1-yl]methyl]acetamide 2-[4-[3-[1-(trifluoromethyl)cyclopropanecarbonyl]phenyl]sulfonylpiperazin-1-yl]acetic acid N-(3-chlorophenyl)-4,5-dimethyl-1H-imidazole-2-carboxamide ethane;N-methyl-2,3-bis[(Z)-prop-1-enyl]naphthalene-1-carboxamide 1-[(2R)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-2H-chromen-2-yl]-N',N'-bis[[4-(trifluoromethoxy)phenyl]methyl]cyclopropane-1-carbohydrazide 3-[2-(1H-benzimidazol-2-yl)ethyl]-2-propan-2-ylidene-1,3-oxazolidine N-(azidomethyl)-2,6-dibromoaniline N-[4-(azidomethyl)phenyl]cyclohexanamine 2-[2,5-difluoro-N-(1-phenylethyl)anilino]acetamide (5Z)-2-(5-chloro-3-methylpyridin-2-yl)imino-5-[[1,3-dioxo-4-phenyl-6-(4-propoxyanilino)pyridazin-2-yl]methylidene]-1,3-thiazolidin-4-one 5-(cycloheptylamino)sulfanyl-2,4-dimethoxybenzoic acid 2-cyclopropyl-7-ethoxy-N,4,5,6-tetrahydrobenzo[f]benzimidazole-3-carboxamide 4-azido-2,3-dichlorobenzonitrile 3-[(4,5-dimethylfuran-2-yl)methyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione 2-amino-6,7-dihydrobenzo[d][1]benzazepine-5-carboxylic acid (Z,3S)-4-[(1R)-2-cyanocyclohexyl]-N,N'-diethyl-N-methoxy-3-methylbut-2-enimidamide;(E)-2-methylhept-2-ene 1-(5,6-diphenylpyridin-2-yl)ethanone 3-methyl-5-[(3R)-piperidin-3-yl]oxybenzenesulfonamide 2,3-bis(4-fluorophenyl)-5H-imidazo[1,2-b]pyridazin-6-one 5-(2,6-difluorophenyl)-N-[[3-fluoro-5-(3-methylpyrazine-2-carbonyl)phenyl]methyl]-1H-pyrrole-3-carboxamide 5-cyclohexyl-7-(2,4-difluorophenyl)furo[3,2-b]pyridine (3R)-N-[(3S,4Z)-3-(2,5-dioxopyrrol-1-yl)hexa-1,4-dien-2-yl]-2-oxo-1,3-oxazolidine-3-carboxamide N-(2,6-dichloro-4-nitrophenyl)-N-(3-methylbutyl)ethenesulfonamide ethane;3-[4-(2-ethylbutoxy)phenyl]propan-1-amine N-[3-(2,4-dioxopyrimidin-1-yl)phenyl]-2-(4-methoxyphenyl)acetamide 4-[2,3-dihydroxypropyl(4-hydroxybutyl)amino]benzenesulfonamide 1-(6,7-dihydro-4H-thieno[3,2-c]pyran-4-yl)-N-ethylbutan-2-amine N-[(2R,3S)-1-methyl-2-pyridin-4-ylpyrrolidin-3-yl]ethanesulfonamide N-butan-2-yl-5-hydroxy-1,3,4,9-tetrahydropyrido[2,3-b]indole-2-carboxamide 3-[2-bromoethyl-(6-chloropyridazin-3-yl)amino]propane-1,2-diol N-methoxy-6-[4-(2,2,2-trifluoroethyl)phenyl]pyridine-3-carboxamide 1-[2-[4-(3,5-dimethylphenoxy)butoxy]ethyl]pyrrolidine;methane 2-[4,5-bis(4-ethenylphenyl)-1H-imidazol-3-ium-3-yl]ethanol 5-(4,6-difluoropyridin-2-yl)-4-imino-1-methylimidazolidin-2-one 7-(5,6-dimethoxypyridine-3-carbonyl)-2-[4-(trifluoromethyl)phenyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 2-chloro-4-[(2,6-dimethyl-4-propoxyphenyl)iminomethyl]phenol [2-fluoro-4-[3-(methoxyiminomethyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]methanamine N-[(2,3-dimethylphenyl)-phenylmethyl]-1-[6-methoxy-5-(4-methylimidazol-1-yl)pyridin-2-yl]methanimine (7S)-2-[(3-chlorophenyl)methylsulfanyl]-N-(4-ethoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide 3-amino-5-chloro-1H-pyrrolo[2,3-b]pyridine-4-carboxylic acid;2,2,2-trifluoroacetic acid 2-(difluoromethyl)-N-[1-(5,6-dihydropyrido[4,3-d]pyrimidine-7-carbonyl)azetidin-3-yl]pyridine-4-carboxamide 4-[4-chloro-3-(trifluoromethyl)phenoxy]-N-diazopiperidine-1-sulfonamide N-[4-cyano-2-(5-oxo-1H-pyrazol-2-yl)phenyl]-3,7-dimethylspiro[6,8-dihydroimidazo[2,1-c][1,2,4]triazine-9,4'-piperidine]-1'-carboxamide 3-[4-(cyclohexen-1-yl)phenyl]propanamide;methane 5-hydroxy-4,6-dioxo-8-phenyloctanamide 4-(azidooxymethyl)-5-chloropyrimidine N-[(3R,5S)-1-(cyclobutanecarbonyl)-5-(5-methyl-1H-1,2,4-triazol-3-yl)pyrrolidin-3-yl]benzamide 6-bromo-1,2-dimethylbenzimidazole;ethane N-[2-(2,6-dichlorophenyl)ethyl]quinoline-3-carboxamide;hydrochloride 5-methyl-N-[(3S)-1,2,3,4-tetrahydroisoquinolin-3-yl]furan-2-sulfonamide 1-[2,4-dichloro-3-(trifluoromethyl)phenyl]sulfonyl-3,5-dihydro-2H-benzimidazole (2R,5S)-5-[3-(4-chlorophenyl)propoxy]-6-ethenyl-6-methoxyhexan-2-ol 5-(3,5-dimethylphenyl)-8-thia-2,12,14-triazatetracyclo[7.6.0.02,7.010,13]pentadeca-1(9),4,6,10(13),11-pentaene N-[(4-chloro-2,6-dimethoxyphenyl)methyl]cyclopentanamine 3-[5-tert-butyl-4-(oxiran-2-ylmethoxy)thiophen-2-yl]furan (3R)-4,4,6-trifluoro-3-[[5-[4-[2-methyl-4-[methyl(oxolan-3-yl)amino]benzoyl]piperazin-1-yl]pyridin-2-yl]amino]-7-(trifluoromethyl)-2,3-dihydrochromene-2-carboxylic acid 3-[5-(3,4-dimethoxyphenyl)-2-sulfanylideneimidazolidin-1-yl]butanenitrile 2-benzyl-N',3-dihydroxyimidazole-4-carboximidamide 4-[2-(azetidin-1-yl)ethylamino]-5H-pyrido[3,2-d]pyrimidine-8-carboxylic acid (2E,5Z)-N'-[3,4-bis(trifluoromethyl)phenyl]-2,6-dichloro-5-ethylideneocta-1,7-diene-3,6-diamine 2-(1-benzofuran-5-yl)-N-[4-[(3-formylphenyl)carbamoyl]cyclohexylidene]acetamide 2-[1-(4-methylphenyl)cyclopentanecarbonyl]cyclohexan-1-one 3-[2,5-difluoro-4-(morpholine-4-carbonyl)phenyl]-1H-indole-6-carbonitrile 3-(3,4-dimethoxyphenyl)-2,6-difluorobenzaldehyde 2-[1-(4-methoxyphenoxy)pentyl]oxirane 3-(2,5-dimethylphenyl)sulfanylbutanoic acid 1-[(2,3-dimethylphenyl)methylamino]-3-nonan-5-ylthiourea N-(2,3-dihydrofuran-5-ylmethyl)-2-[6-[[3-fluoro-5-(trifluoromethoxy)phenyl]methylamino]pyridin-3-yl]-4H-thieno[3,2-b]pyrrole-5-carboxamide 7-bromo-2,3-bis(4-chlorophenyl)quinoxaline 2-[4-(3-hydroxyphenyl)phenoxy]-3,5-dipropylphenol 2-[(4-methylpiperazin-1-yl)methyl]-1,3-benzothiazole 2-[3,5-dimethyl-1-(2,4,6-trimethylphenyl)sulfonylcyclohexa-2,4-dien-1-yl]oxy-4-fluorooxane 6-N-(1-cyclopentylpyrazol-4-yl)-7-methoxy-2,3-dihydro-1H-indene-5,6-diamine N-[2,6-dichloro-4-nitro-3-(trifluoromethyl)phenyl]acetamide 3-methoxy-4-methylsulfanylbenzaldehyde;1,2,4-triazol-5-amine [(E)-2-cyanoprop-1-enyl]-[4-(dimethylaminosulfanyl)phenyl]azanium N-butyl-2-[3-[4-(difluoromethoxy)benzoyl]indolizine-1-carbonyl]spiro[6,7-dihydro-5H-pyrazolo[1,5-a]pyridine-4,3'-azetidine]-1'-carboxamide [2-fluoro-4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonylamino)benzoyl]oxidanium N'-[2-fluoro-4-[4-[(6-methylpyridin-3-yl)methoxy]piperidine-1-carbonyl]phenyl]ethanimidamide 3-(5-azidoindazol-2-yl)-1H-pyridazin-6-one (3R)-4-methyl-N-[2-oxo-1-(1,3-thiazol-2-yl)piperidin-4-yl]-3-phenylmorpholine-3-carboxamide 2-bromo-3,5-dimethylimidazo[1,2-a]pyridine 1-[(2,3,4a,5-tetrahydro-1H-pyrazino[2,1-b]quinazolin-9-ylamino)methyl]cyclohexan-1-ol (5S,7R)-N-[[4-(2,2-dimethyloxan-4-yl)phenyl]methyl]-1,5,7-trimethyl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carboxamide (7S)-2,4-dimethyl-5-oxo-8-[3-[3-[1-(2,2,2-trifluoroacetyl)piperidin-4-yl]propoxy]phenyl]-7-thiophen-2-yl-6,7-dihydropyrazolo[1,5-a][1,3]diazepine-9-carboxylic acid N-[(3,4-dichlorophenyl)methyl]-2-[4-(3-fluorophenoxy)piperidin-1-yl]-N-[2-(methoxyamino)prop-2-enyl]acetamide;ethane 2-amino-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6,9-disulfonic acid N-azido-1,5-bis(2-methylbutan-2-yl)naphthalene-2-sulfonamide 2-[(4-bromophenyl)sulfonylamino]-3-[3-fluoro-5-(trifluoromethyl)pyridin-2-yl]propanamide (4S)-1,3-bis(3-bromophenyl)-4-naphthalen-2-ylimidazolidine N-[(1Z,3E)-2-cyanopenta-1,3-dienyl]-4,6-bis(dimethylamino)naphthalene-1-carboxamide (Z)-N',2-dimethylbut-1-ene-1,4-diamine;(4S)-3-methoxy-5,9-bis(phenylmethoxy)nonan-2-one 3-[4-(difluoromethoxy)phenyl]sulfonylpyrrolidine-1,2-dicarboxylic acid 4-hydroxy-2,5-dimethoxybenzamide N-[3-[4-(aminomethyl)cyclohexanecarbonyl]phenyl]-5,7-difluoro-2-oxo-1H-quinoline-3-carboxamide;hydrochloride 6-[2-fluoro-4-[(E)-pent-3-enyl]phenyl]-1,2,8-trifluoronaphthalene 2-(4-bromophenyl)sulfonyl-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline 4-[3-(1H-indol-3-yl)propanoylamino]piperidine-2-carboxylic acid 4-[2-(4,5-dihydroimidazol-1-yl)ethoxy]benzonitrile 1-cyclohexyl-N,N'-dipyridin-2-ylethane-1,2-diamine;hydrate 6-hydroxy-5-[(E)-3-oxo-2-propan-2-yloxyprop-1-enyl]-3,4-dihydro-1H-pyridin-8-one 1-[2-(2,4-difluorophenyl)ethyl]-5-(3,6-dihydro-2H-pyran-4-yl)pyrrolo[2,3-b]pyridine 4-[[4,6-bis(4-methoxyphenyl)-1H-1,3,5-triazin-2-ylidene]amino]phenol 2-amino-3,5,6-trichlorobenzonitrile N-(5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-2-ylsulfonyl)cyclobutanecarboxamide 2-(4-bromophenyl)-1,6-naphthyridine 1-(3,4-dimethylphenyl)-5-imino-4-(6-methoxy-1H-benzimidazol-2-yl)-2H-pyrrol-3-ol 5-methylcyclohepta-1,3,6-triene;N-[[4-(4,5,8,10-tetrahydrothieno[2,3-c][1]benzazepine-7-carbonyl)phenyl]methyl]formamide 3-[6-methyl-2-(trifluoromethyl)pyridine-4-carbonyl]-1,3-oxazolidin-2-one (4-amino-2,6-dichlorobenzoyl)-[3-(naphthalene-1-carbonyloxymethyl)oxetan-3-yl]azanium 1-(5,6-dihydrophenanthrene-1-carbonyl)-N-[[4-ethyl-3-[5-methyl-2-(propan-2-ylamino)phenyl]phenyl]methoxy-pyridin-4-ylmethyl]piperidine-4-carboxamide (2S)-3,3-dimethyl-1-[4-(4-methylphenyl)-6-nitropyridin-2-yl]oxybutan-2-ol N'-[3-(4-methylpiperazin-1-yl)propyl]-2-[3-methylidene-5-phenyl-2-(1H-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidin-7-yl]sulfanylethanimidamide 2-[(1S,4R)-1-methyl-6-nitro-3,4-dihydro-2H-naphthalen-1-yl]acetic acid 6-[5-(2,4-difluorophenyl)pentanoyl]cyclohexa-1,3-diene-1-carbonitrile 6-methyl-3,5-diphenylimidazo[1,2-a]pyridine N-[5-[1-(2,3-dihydro-1H-indene-4-carbonyl)piperidin-4-yl]-2-oxopentyl]cyclohexanecarboxamide (5Z)-2-(4-bromophenyl)imino-5-[(7-chloro-1,3,2-benzodioxaborol-2-yl)methylidene]-1,3-thiazolidin-4-one 1-[(2R,6S)-2-tert-butyl-6-phenylmorpholin-4-yl]ethanone 2-[4-methoxy-5,6-dimethyl-7-(oxiran-2-ylmethoxy)naphthalen-1-yl]oxy-3H-pyrido[3,4-d]pyrimidin-4-one [4-(3,5-dichlorophenyl)sulfanylphenyl]methanethiol;ethane ethane;3-(5-fluoro-1H-indol-2-yl)-1,7-dimethoxyquinolin-4-one 5-(1,2-dihydropyridin-4-yl)-7-phenylindolo[3,2-c]carbazole;ethane 5-[(2,5-difluorophenyl)sulfanylamino]-1-methylindazole-3-carbonitrile 1-butyl-4-(2,6-ditert-butylphenyl)-3,5,6,7-tetrahydro-2H-s-indacene 7-(cyclohexylmethoxy)-3-cyclopropyl-2H-chromene N-(4-methylpyridin-3-yl)sulfonyl-2,5-dioxopyrrolidine-1-carboxamide 5-[(5-fluoroindol-2-ylidene)methyl]-3-piperidin-1-yl-4H-1,2,4-triazin-6-one 4-chloro-3-(2,4-dihydroxyphenyl)-1H-pyridazin-6-one 2-[[2-(4-methoxyphenyl)phenyl]methylamino]acetic acid 5-phenyl-2,4-dihydrotriazolo[1,5-a]pyrimidine;hydrochloride (3R,4S)-4-[5-(2-tert-butylphenyl)-1H-pyrazol-3-yl]-1-ethylpiperidine 2,5-dibromo-4-(3-chlorobutyl)-N,3-dihydroxybenzamide 7-chloro-2,3,4,9-tetrahydro-1H-carbazole 2-(6,8,12,15,16-pentazapentacyclo[10.7.0.03,10.04,8.013,17]nonadeca-1(12),2,4(8),5,9,13(17),14-heptaen-6-yloxy)ethanamine 1-[2,6-difluoro-4-(methylsulfanylamino)phenyl]piperidine-3-carboxylic acid 1-[4-(4,5-dimethylpyrimidin-2-yl)piperazin-1-yl]ethanone 4-(4-azidopiperazin-1-yl)-3,5,6-trichloropyridazine 1-[4-(6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl]prop-2-en-1-one N-[1-(5-fluoropyridin-2-yl)ethyl]-3,4-dimethoxy-6-methyl-2-nitrobenzamide 2-[(Z)-propan-2-ylideneamino]oxy-3H-1,2-benzothiazole-6,7-diamine N-(4-chlorophenyl)-2-[(3-oxocyclohexyl)sulfamoyl]benzamide 5-[2-(4-chlorophenyl)ethoxy]-1-(methylamino)pentan-3-ol (2S)-4,5-dihydroxy-1-[2-methyl-6-phenyl-4-(3,4,5-trifluorophenyl)benzoyl]pyrrolidine-2-carboxylic acid 2-[(4Z,5Z)-4-ethylidenehepta-1,5-dien-3-yl]-N-(1H-indazol-6-yl)imidazo[1,2-a]pyrazin-8-amine;propane 4-[2,3-bis(2,6-dimethylphenyl)benzimidazol-5-yl]-2-fluorobenzonitrile 6-[4-(2,3,5,6-tetradeuteriopyridine-4-carbonyl)piperazin-1-yl]pyridazine-3-carboxamide 3-[4-(benzylamino)-5H-pyrazolo[1,5-a]pyrimidin-6-yl]phenol 4-[[(2R)-1,1-dimethoxypropan-2-yl]amino]-1H-pyrimidin-6-one (2S)-3-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]-2-hydroxy-8-phenyloctanal 4-[4-(2-carboxyethyl)phenyl]-N,N-dimethylbenzenecarboximidamide 3-[(5E)-2-amino-4-methylidene-5-prop-2-enylideneimidazol-1-yl]benzaldehyde;butane;N,4,4-triethylcyclohexanamine N-[1-(2,3-dihydro-1H-pyrrole-5-carbonyl)piperidin-4-yl]-7-methoxyquinazolin-4-amine N-[4-amino-3,4-dioxo-1-(1H-pyrrol-2-yl)butan-2-yl]-5-pyridin-4-yl-1,2-oxazole-3-carboxamide N-[4-(5,7-dimethylpyrrolo[2,3-d]pyrimidin-6-yl)phenyl]cyclobutanecarboxamide 4-[(3,5-dimethylphenyl)methoxy]aniline 1-methyl-4,6-diphenyl-3H-2,1,3-benzoxadiazol-3-ium 3-methyl-5,6-dihydrothieno[2,3-b]thiophen-4-one 5-[2-ethoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine-3-carbonyl]-N-(trideuteriomethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide 1-(4-methylsulfonylphenyl)ethenamine 2-[2-(3-methoxy-3-oxopropyl)-7-(trifluoromethyl)quinolin-8-yl]acetic acid 1-(4-nitrophenyl)-5-[2-[3-(trifluoromethyl)phenyl]ethynyl]triazole 2-cyclobutylsulfanyl-4,7-dioxo-N-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 1-[5-(2-bromopyridine-4-carbonyl)-3,4-dihydro-2H-quinolin-1-yl]ethanone 5-bromo-4,6-dimethyl-2-(4-methylphenyl)pyrimidine N-(6-hydroxy-1,3-benzothiazol-2-yl)-4-nitrobenzamide N-[(1S)-3-(dimethylamino)cyclopentyl]-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine-2-carboxamide 2-[2-hydroxyethyl(1,3-thiazol-5-yl)amino]decanoic acid (1S,3R)-N,3-dimethyl-6-phenylmethoxy-N-propan-2-yl-4-thiophen-2-ylsulfonyl-2,3-dihydro-1H-indene-1-carboxamide 2-[5-(trifluoromethyl)pyridin-3-yl]indole N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2-formyl-1-azabicyclo[3.2.0]heptane-2-carboxamide [4-(1,1-dioxothian-4-yl)-5-methoxy-2-[3-(6-methylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]urea 2-[(1R)-1-(4-fluorophenyl)ethyl]-6-N,6-N-dimethylquinazoline-4,6-diamine 3,4-dicyclohexyl-2-[[(E)-3-[6-[cyclopentylcarbamoyl(methyl)amino]benzimidazol-1-yl]prop-1-enyl]amino]pentanoic acid 4-(azepan-1-yl)-5-chloro-N'-hydroxypyridine-2-carboximidamide 2-(5,8-dimethylpyrido[4,3-d]pyrimidin-2-yl)-3-propan-2-yl-1H-indole 4-fluoro-2-[3-(hydroxymethyl)phenyl]sulfonylphenol 4-bromo-1,2-difluorobenzene;3-cyclohexyl-N-[(2R)-1,1,1-trifluoropropan-2-yl]sulfanylbenzamide 3-methyl-4-[4-(thiophene-2-carbonylamino)piperidin-1-yl]benzoic acid;2,2,2-trifluoroacetic acid 5-amino-4,6-dimethyl-2-(5-nitrofuran-2-yl)pyridine-3-carbonitrile 4-amino-5-[2-(1H-imidazol-5-yl)ethoxy]benzene-1,3-dicarboxylic acid 1-[2,3-bis(ethenyl)-4-phenylcyclopenta-2,4-dien-1-ylidene]fluorene (E)-N-[[4-(2-chloroanilino)sulfanylphenyl]methoxy]-1,3-bis(4-fluorophenyl)propan-2-imine 4-[1,1,2,3,3,3-hexadeuterio-2-(trifluoromethyl)propoxy]carbonylbenzoic acid 3-(2-amino-1,3-benzothiazol-5-yl)-4H-1,2,4-oxadiazol-5-one 1-N'-[4-[7-methoxy-6-(3-pyrrolidin-1-ylpropoxy)quinolin-4-yl]oxyphenyl]-1-N-(4-fluorophenyl)cyclobutane-1,1-dicarboxamide 2-[N-(3-hydroxypropyl)-4,5-dimethyl-2-phenyldiazenylanilino]decanoic acid 4-[(2S)-2-methylpiperazine-1-carbonyl]-N-[6-(trifluoromethyl)pyridin-3-yl]piperidine-1-carboxamide (E)-3-[5-methoxy-7-methyl-2,4-dioxo-8-(oxan-4-ylmethylamino)pyrido[2,3-d]pyrimidin-1-ium-1-ylidene]prop-2-enoic acid 2-[(4R,5S)-1-[(3-chlorophenyl)methyl]-5-cyano-6-hydroxy-4-(hydroxymethyl)-7-oxoheptan-2-yl]guanidine (4S)-N-[5-chloro-3-fluoro-2-methoxy-6-(methylamino)phenyl]-1'-ethanimidoylspiro[2H-indene-3,4'-piperidine]-1-carboxamide 2-methoxy-4-[1,2,3,6-tetradeuterio-4-(2-phenylpropan-2-yl)piperazin-2-yl]phenol 2-[4-[4-(4-hydroxyphenoxy)phenyl]phenoxy]phenol 3,6-difluoro-2-[(E)-hept-3-enyl]-1-benzothiophene 2-azidosulfanyl-1,3-difluoro-4-(4-methoxyphenyl)benzene N-[(4S,5R)-1-(cyclohexylmethyl)-5-(3,4-difluorophenyl)piperidin-2-ylidene]-2-oxopropanamide 1-[5-(3,4,5-trimethoxyphenyl)pyrimidin-2-yl]ethanethiol (E)-1-(5-chloro-2,4-dimethoxyphenyl)prop-1-en-1-amine 3-ethyl-2,5-dimethyl-N-[1-(1H-pyrazol-4-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-6-carboxamide (E)-3-[(2-chlorophenyl)diazenyl]-4-hydroxypent-3-en-2-one 5-[(2,4-difluorophenyl)methyl]-3-[2-(1H-imidazol-2-yl)ethylsulfanyl]-5-methyl-1-pyridin-2-yl-6H-pyrazolo[4,3-d]pyrimidin-7-one 1-[4-(2,6-dichlorophenoxy)-3-nitrophenyl]ethanone 4-(aminomethyl)-2-[3-(hydroxymethyl)phenyl]-1H-pyrimidin-6-one 3-[2-(4,5,6,7-tetrahydrobenzimidazol-1-yl)phenyl]-1,2-dihydrotriazolo[1,5-a]pyridine N-[3-(benzenesulfonamido)phenyl]-2,4-dihydroxy-6-oxopyran-3-carboxamide 2-[azido(difluoro)methyl]sulfonylpyridine 4-[(4R)-3-fluoro-1-[(4-methoxyphenyl)methyl]piperidin-4-yl]benzoic acid 5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)-N-[5-piperazin-1-yl-6-(trideuteriomethoxy)pyridin-2-yl]pyrimidin-2-amine 1-(cyclopropylmethylamino)-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-3,4-dione 5-[1-(4-fluorophenyl)indazol-5-yl]pyrimidine-2,4-diamine (E)-3-[4-[7-ethylsulfanyl-2-[4-(methylamino)phenyl]pyrido[2,3-d]pyrimidin-8-yl]phenyl]prop-2-enamide 5-(2,4-dichlorophenyl)sulfanyl-3H-1,3,4-oxadiazol-2-one N-[(E)-3-[4,5-dimethyl-2-[[5-(trifluoromethyl)pyridine-2-carbonyl]amino]phenyl]but-1-enyl]cyclopropanecarboxamide 4-(2-chlorobenzoyl)-N,3-dimethylpiperazine-1-carboxamide 1-[2,3-difluoro-4-(trifluoromethyl)phenyl]-6,7-bis(trichloromethoxy)phthalazine 3-[(2Z)-4-oxo-5,6-dihydrocycloocta[b]furan-7-yl]propanamide 1-azido-4-(2,6-dichlorophenyl)-5H-pyrazole 2-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylamino)-N-[[1-(oxolan-3-ylmethyl)triazol-4-yl]methyl]acetamide 3-[(2E)-2-[(4-hydroxyphenyl)methylidene]hydrazinyl]-1H-quinoxalin-2-one 4-(5-iodopyridin-3-yl)-2-methylmorpholine 3-[1,1-bis(4-bromophenyl)ethyl]-2H-1,3-oxazole 2-amino-4-[1-(pyridin-3-ylmethyl)imidazol-2-yl]phenol N-(2,3-dihydro-1H-indol-7-yl)-4-fluoro-5-pyridin-4-ylthiophene-2-carboxamide 5-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl)-3H-1,3,4-oxadiazol-2-one (4-ethoxyphenyl)methyl-[2-(naphthalene-1-carbonyl)prop-2-enoyl]azanium N-[(4,5-dimethyl-2-phenylpyrazol-3-yl)methoxy]cyclobutanamine 1-amino-3-(diethylamino)anthracene-9,10-dione [2-(6-aminopyridazin-3-yl)pyrrolidin-1-yl]-[5-(3-methoxyphenyl)-4-methyl-1,3-thiazol-2-yl]methanone;ethane 1-[4-[2-azidooxy-7-(3-ethylsulfonylpropyl)quinazolin-6-yl]phenyl]cyclobutan-1-ol [7-chloro-6-(2,3-difluorophenyl)-2,4-dimethylpyrazolo[1,5-a]pyridin-5-yl]-[4-hydroxy-4-[(6-methoxypyridin-3-yl)methyl]piperidin-1-yl]methanone 4-[2-(6,7-dimethoxyquinazolin-4-yl)ethynyl]benzaldehyde 5-[(3,4-diethoxyphenyl)iminomethyl]-4-hydroxy-3H-1,3-thiazol-2-one 3-hydroxy-5-[3-(2,3,4,5,6-pentafluorophenyl)propyl]benzamide 1-[1-(4-chlorocyclohexyl)ethenyl]-6-[2-methoxy-3-methyl-5-(1,1,2,2,2-pentafluoroethyl)phenyl]pyrazolo[3,4-d]pyrimidine N-[2,3-dimethyl-4-(3-oxomorpholin-4-yl)phenyl]-5-ethoxyimidazo[1,2-c]quinazoline-2-carboxamide 2-(4-azidophenyl)-6-methoxyquinazoline 2-(furan-3-ylmethylamino)-4,5-dihydro-1H-indole-7-carboxamide;hydrochloride 2-[[(5Z)-5-benzylidenepyrrol-3-yl]methoxy]ethanol 2-[1-[(4R)-5,8-dichloro-1-methyl-3,4-dihydro-2H-quinoline-6-carbonyl]piperidin-4-yl]acetonitrile N-(3,4-dichlorophenyl)-1-methylpyrazole-4-carboxamide N-[4-(3-cyclopentyloxy-2-fluorophenyl)pyridin-2-yl]propanamide 1-[[(2S,4S)-4-fluoropyrrolidin-2-yl]methoxy]-3-[1-(1H-pyrrolo[3,2-c]pyridin-2-ylmethyl)piperidin-4-yl]indole (3S)-3,7-dimethyl-2H-1,4-benzoxazine;N,4-dimethylaniline (3S,4R)-N'-azido-1-(4-chlorophenyl)-6-fluoro-2-oxopiperidine-3-carbohydrazide 1-[2,2,2-trifluoro-1-(5-methoxynaphthalen-2-yl)ethyl]pyrazolidin-3-one 1-benzyl-2-ethoxy-4-methylsulfanyl-3,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-6-amine 2-[3,4-difluoro-N-(3-methylbut-2-enyl)anilino]acetonitrile 1-methoxy-3-[2-(4-phenoxyphenyl)ethenyl]benzene 3-(2-diazohydrazinyl)naphthalene-1,4-disulfonic acid 1-(3,4-dimethylphenyl)hexane-2,5-dione 5-(2,4-dihydroxyphenyl)naphthalene-1-carboxylic acid N-[5-(4-ethoxyphenyl)pentyl]pyridine-2-carboxamide 6-[5-(4-hydroxy-3-methoxyphenyl)-1H-pyrazole-4-carbonyl]cyclohexa-2,4-diene-1-carboxylic acid 4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)morpholin-4-yl]-3-methoxybenzoic acid 4-(3,3-dimethylbutan-2-ylamino)-5-iodo-1H-pyrimidin-6-one 4-[5,7-bis(2-methylphenyl)imidazo[1,2-a]pyridin-8-yl]-N,N-dimethylaniline 2,5-dimethyl-N-[1-(pyridine-3-carbonyl)piperidin-4-yl]furan-3-carboxamide (3Z,5E)-2-methylidenehepta-3,5-dienoic acid;3-[(4-phenylbenzoyl)amino]propanamide 3-(4-ethylpiperazin-1-yl)-N'-hydroxypyridazine-4-carboximidamide 2-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)piperidine-1-carbonyl]benzamide N-[5-(1H-indole-2-carbonyl)-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrol-2-yl]acetamide 5-[(4-azidobutylamino)methyl]-2,3-dihydro-1H-indene-4,6-diol 2-(4-methoxycyclohexa-1,3-dien-5-yn-1-yl)-6,7-dihydroimidazo[5,1-b][1,3]thiazin-8-ol 2-tert-butyliminospiro[4H-1,3-thiazine-6,3'-pyrrolidine]-5-carboxylic acid 2-[4-(azidomethyl)phenyl]-6-[(5-chlorofuran-2-carbonyl)amino]hexanoic acid 4-[3,5-difluoro-2-(triazol-1-yl)phenyl]sulfonyl-N-(5-methylpyridin-2-yl)piperazine-1-carboxamide (3R)-2-(2,2-dimethylpropanoylamino)-N-[1-[4-[(E)-3-[2-(ethylideneamino)-6,6-difluorocyclohexa-2,4-dien-1-yl]prop-1-ynyl]phenyl]cyclopropyl]pentanediamide 1-[4-amino-5,7-dichloro-2-(hydroxymethyl)quinazolin-6-yl]ethanone N-[(1R)-2-amino-4,4-difluorocyclohexyl]-6-chloro-8-methoxy-7-(3-morpholin-4-ylpropoxy)-2H-chromene-3-carboxamide 1-(4,5-ditert-butyl-2-phenylpyrazol-3-yl)-N-diazo-9H-fluoren-4-amine N-[(4-phenylphenyl)methyl]decanamide 1-[(2S)-4-azido-1-methoxybutan-2-yl]imidazole N-cyclohexyl-2,4-dinitro-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)aniline (1E)-3-N-[4,5-bis(ethenyl)thiophen-2-yl]sulfanylbuta-1,3-diene-1,3-diamine;ethenamine 2-[N-butyl-4-(dimethylamino)anilino]decanoic acid N-[(2S)-1-[(3S,5R)-4-azido-3,5-dimethylpiperazin-1-yl]-3-cyclohexa-1,3-dien-1-yl-1-oxopropan-2-yl]-4-fluorobenzamide 5-(3,4-dimethylphenyl)sulfanylpyridine-2,3-diamine 6-[1-(2,3-difluorophenyl)ethoxy]pyridine-3-carboxamide 4-methyl-1-(5-phenyloxolane-2-carbonyl)piperidine-3-carboxylic acid 1-[(2,4-dichlorophenyl)methyl]piperidine (2R)-3-methoxy-1,2-diphenylpropane-1,2-dione N-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)ethyl]pyrrolidine-2-carboxamide;hydrochloride N-[(2S)-3,3-dimethylbutan-2-yl]-1H-indazole-5-carboxamide 2-chloro-5,7-dihydroindolo[2,3-c]carbazole 2-(3,5-dimethylpiperidin-1-yl)pyridine;4-[(4E,6Z)-hepta-1,4,6-trien-4-yl]quinoline 2-amino-3-azidooxy-5,6-dimethylbenzoic acid 1-[4-(5,6-difluoro-3-methyl-2H-benzimidazol-1-yl)piperidin-1-yl]propan-1-one 4-[[1-(5-fluoro-2-methoxyphenyl)piperidin-3-yl]methoxy]pyridine (Z)-3-[4-(ethylamino)phenyl]prop-2-enehydrazide 1-cyclohexyl-5,7-dimethoxy-3-phenyl-2H-quinazolin-4-one 3-[2,6-dichloro-4-(trifluoromethoxy)phenyl]-5-(1H-indol-2-yl)-1H-1,2,4-triazol-4-ium 3-[2-(4-chlorophenyl)ethenyl]cyclohex-3-ene-1,2-dione 6-(2,4-difluorophenoxy)-N-[3-(dimethylamino)propyl]-5-(1H-pyrazole-4-carboximidoyl)pyridin-3-amine 1-(2,4-difluorophenyl)-N,2-bis[(3-ethoxypyridin-2-yl)methyl]benzimidazole-5-carboxamide 2-[2-(oxiran-2-ylmethoxy)phenoxy]octanoic acid 1-(3,4-dimethoxyphenyl)-2-[4-hydroxy-4-[1-[3-[5-(trifluoromethyl)pyrimidin-2-yl]oxybenzoyl]piperidin-4-yl]butyl]guanidine 4-[3-(benzenesulfonyl)pyrrol-1-yl]benzonitrile 2-ethyl-1-[2,3,4-tris(trifluoromethoxy)phenyl]-5-[2-(trifluoromethoxy)phenyl]imidazole N-[3-cyclopropyl-4-(4,5-dihydroimidazol-1-yl)phenyl]-2,2,2-trifluoroethanesulfonamide (3R)-2,6-diamino-4-[(1S)-2-azidocyclopentyl]oxy-7-methoxy-5-phenylsulfanylheptanoic acid 1-(benzenesulfonyl)-4-(5-methylthiophen-2-yl)pyrrolo[3,2-c]pyridine 4-(3-cyclohexa-1,5-dien-1-ylphenyl)-6-[4-(9H-fluoren-1-yl)piperazine-1-carbonyl]-1H-pyrimidin-2-one 2-[(4-methoxyphenyl)sulfanylmethyl]-3H-quinazolin-4-one 3-[1-[2-(6,7-dihydroquinolin-5-ylamino)ethyl]piperidin-4-yl]-1H-benzimidazol-2-one;dihydrochloride 7-azido-N,N-diethylnaphthalene-1-sulfonamide 5-(6,7-dimethoxyquinolin-4-yl)oxy-N-[4-fluoro-3-(trifluoromethoxy)phenyl]naphthalene-1-carboxamide 4-azido-6,7,8-trimethoxyquinazoline 2-[5-(6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-ylsulfonyl)-2-methoxyphenyl]-4H-1,3,4-oxadiazin-5-one 5-[5-(4-fluorophenyl)sulfonyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-2-carbonyl]pyridine-3-carbonitrile (4R)-6,8-dichloro-1-methyl-N-[2-[4-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyrazol-1-yl]ethyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-4-carboxamide 2-(hydroxymethyl)-3-[4-[1H-indole-7-carbonyl(propyl)amino]butanoyloxy]pyrrolidine-1-carboxylic acid 2-amino-N'-(4,6-dichloropyrimidin-5-yl)-N-hydrazinylidene-3H-benzimidazole-4-carboximidamide 4-[(2-azidooxyphenyl)methyl]aniline 2-(aminomethyl)-4-[(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethoxymethyl))amino]-1H-pyrimidin-6-one;dihydrochloride 2-[1,4-diphenyl-2-(1H-pyrrole-2-carbonyl)pyrrolo[3,2-c]pyridin-6-yl]acetonitrile 2-[(4-chlorophenyl)methyl]-5-ethoxypyrazole-3,4-diamine 5-[1,2,4]triazolo[3,4-a]phthalazine;hydrate 2-[(4-aminopyrimidin-5-yl)methylamino]acetic acid;ethane 3-ethyl-N'-[5-fluoro-6-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyridin-3-yl]pentanehydrazide 2-[N-(4-bromobutan-2-yl)-2,5-dichloroanilino]phenol 3-methyl-4-oxoquinazoline-6-carboxylate 2-[4-[4-(1H-indole-3-carbonylamino)phenyl]butanoylamino]acetic acid N-ethyl-4,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidine-2-carboxamide;1H-imidazole 4-(3-azidopropyl)-2,5-difluorobenzaldehyde 6-[(3S)-2,4-dioxopyrrolidin-3-yl]-2-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-10H-anthracen-9-one N-methyl-2-[4-(2H-tetrazol-5-yl)piperidin-1-yl]pyridine-3-carboxamide N'-[amino(methyl)amino]-5-hydroxy-1H-indole-2-carboximidamide 6,8-dimethoxy-2-(3-pyridin-4-ylphenyl)quinazolin-4-amine N'-hydroxy-5,6-dimethyl-3-[(3R)-1-propanoylpyrrolidin-3-yl]oxypyridazine-4-carboximidamide 5-azido-7-bromoquinazoline 6-[2-(1,3-benzodioxol-5-yl)ethynyl]-4a-methyl-10H-phenoxazine 1-[(3-bromophenyl)methyl]-4-ethenylpiperazine [3-(5-chloro-2-fluorophenyl)pyrrolidin-1-yl]-[3-methoxy-5-(trifluoromethoxy)phenyl]methanone;methanol 2-[[5-(4,6-diphenylpyrimidin-2-yl)pyridin-3-yl]methylidene]indene-1,3-dione 2-(benzylamino)-N',1-dimethyl-3-oxopyrrolo[2,3-c]pyridine-5-carboximidamide;ethane 2,2-bis(2-methoxyphenyl)propanoate (2-bromo-4,6-dimethylphenyl)methanol ethane;methoxyethane;7-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine N-butyl-3,6-bis(4-chlorophenyl)-2-methoxy-7H-pyrazolo[1,5-a]pyrimidine-8-carboxamide 2-[5-bromo-1-(3,4-dichlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-6-yl]oxyacetonitrile 2-(3-cyclopenta-1,4-dien-1-ylpropanoylamino)thiophene-3-carboxylic acid 1-methyl-3-[5,7,8-trihydroxy-2-(4-hydroxyphenyl)chromen-4-ylidene]urea 3-N,4-N-bis(2-methylpropyl)-1H-indole-2,4-dicarboxamide (3R,5R)-N'-[4-cyano-2-(trifluoromethyl)phenyl]-5-(trifluoromethyl)pyrazolidine-3-carbohydrazide N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N'-[(E)-[4-[1-[4-(trifluoromethoxy)phenyl]-1,2,4-triazol-3-yl]phenyl]methylideneamino]propane-1,3-diamine 2-[4-[(E)-3-[5-methyl-3-(2,3,6-trifluorophenyl)-1H-pyrazol-4-yl]prop-2-enoyl]piperazin-1-yl]pyrimidine-5-carbonitrile [3-amino-2-[1-(2,5-difluorophenyl)pyrrolidin-3-yl]prop-2-enylidene]azanium 2-[[5-(3,4-dimethylphenyl)sulfanyl-6-hydroxy-1H-pyrazolo[4,3-d]pyrimidin-7-ium-7-yl]sulfanyl]-N-(2,6-dimethylphenyl)propanamide N-[(3Z,5E)-3,5-dimethylocta-1,3,5-trien-2-yl]benzamide 4-(6-bromoimidazo[2,1-b][1,3]thiazol-5-yl)phenol 1-[3-(2,4-dichlorophenyl)propanoyl]-2-iminoimidazolidine-4-carboxylic acid 3-(2,2,5,5-tetramethylcyclopenten-1-yl)quinoxaline 4-[1-(4-butylcyclohexen-1-yl)ethyl]phenol (2R)-3-cyclopropyl-2-[6-(3,5-dimethoxyphenyl)pyridine-3-carbonyl]-N-[1-(4-fluorophenyl)cyclopropyl]-2H-indole-1-carboxamide 5-azido-3-(1H-pyrazol-4-yl)quinazolin-4-one 1-(2,3-dimethylcyclohexen-1-yl)-2-hydroxy-N,N-dimethyl-5-phenyldiazenylindole-3-carboxamide 6-[(4R)-6-cyclopropyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,8,11-trien-11-yl]-N-methyl-1H-benzimidazole-4-carboxamide 4-[(3R,5S)-4-acetyl-3,5-dimethylpiperazine-1-carbonyl]benzaldehyde N-[(Z)-1-aminoethylidenecarbamothioyl]-3,4-dichlorobenzamide 1-[(3,4-dichlorophenyl)methyl]-2,6,7,9-tetrahydro-5H-pyrazolo[4,3-b]azepin-8-one N-[1-(2,3-dimethylbutanoyl)piperidin-4-yl]-N'-methoxybenzenecarboximidamide 2-[3-(2,3,4,5-tetrahydro-1H-cyclopenta[b]indole-7-carbonylamino)pyrazol-1-yl]acetic acid 5-(3,4-dihydro-1H-isoquinolin-2-yl)pentan-2-one;ethane N-[2-chloro-6-(difluoromethyl)pyridin-4-yl]-1H-pyrrolo[3,2-c]pyridine-7-carboxamide 2-chloro-N-[(3R,4S)-1-ethylsulfonyl-4-methoxypyrrolidin-3-yl]pyridine-3-carboxamide 4-[(2Z,3Z)-6-chlorohexa-1,3,5-trienyl]sulfonylbenzenesulfonamide N-[(1,5-dimethylpyrazol-4-yl)methyl]-8-fluorospiro[2,3-dihydrochromene-4,1'-cyclopentane]-7-carboxamide 2-[[4-(hydroxymethyl)phenyl]methoxycarbonylamino]-3-thiophen-2-ylpropanoic acid 2-[4-[(1,2-dichlorocyclohexa-2,4-dien-1-yl)sulfamoyl]anilino]-3,6-dimethylpyrimidin-4-one 2-[(E)-3-chloroprop-1-enyl]-4-fluoro-N,N-dimethylaniline 6-tert-butyl-2-(4,5-dihydrothieno[3,2-d][1]benzazepine-6-carbonyl)pyridine-3-carboxylic acid 1-ethylpiperidine;4-(5-methoxypyridin-3-yl)-7H-pyrrolo[2,3-d]pyrimidine 3-azidooxy-5,7-dichloroquinoline 5-[2-cyclopropyloxy-3,4-bis(phenylmethoxy)phenyl]-1,2,4-oxadiazole 2-(3-bromophenyl)-N-[4-[difluoro(phosphanyl)methoxy]phenyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-8-carboxamide 2-[4-(3-chloro-5-fluorophenyl)phenyl]-N-methoxyacetamide [3-(4-chlorophenyl)-2H-chromen-4-yl]carbamic acid N-benzyl-1,2,4-trifluorobutan-1-amine 2-[5-[(dimethylamino)methyl]furan-3-yl]-N-[1,4-dimethyl-5-([1,3]thiazolo[5,4-b]pyridin-6-ylamino)cyclohexa-2,4-dien-1-yl]acetamide 6-methoxy-N,3-dimethyl-5-(4-phenylpiperazine-1-carbonyl)-2H-1,3-benzothiazole-2-carboxamide [5-bromo-1-(5-ethylsulfonylpyridin-2-yl)pyrazol-4-yl]methanol 2-[(4-methoxybenzoyl)amino]cyclohexane-1,3-dicarboxylic acid N-[(5-cyclopentylpyridin-2-yl)methyl]-6-[4-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonylphenyl]-7-fluoroquinolin-2-amine (2R)-N-(4-chlorophenyl)-3,7-dioxooctanediamide 4-methyl-1-(3,4,5-trifluorophenyl)pyrazolidine 3-[(5R)-6,7-dihydroxy-2-oxospiro[1H-indole-3,4'-piperidine]-1'-yl]-2-ethoxybenzoic acid 4-(4-methoxyphenyl)sulfonyl-3-propan-2-ylaniline 1-[3-(2,5-difluorophenyl)sulfonylpyrrolidin-1-yl]propan-1-one 3-azido-2,6-dimethoxynaphthalene 1-phenyl-6,8a-dihydropyrene 5-[(2R)-2,3-dihydroxypropoxy]-4-(4-piperidin-1-ylphenyl)benzene-1,3-dicarboxylic acid 1-[3-(2,5-dimethylfuran-3-yl)propanoyl]-2,3,4a,5,6,7,8,8a-octahydropyrido[3,4-b][1,4]oxazine-9-carboxamide (Z)-3-amino-2-[1,4-dimethyl-6-oxo-5-(trifluoromethyl)pyrimidin-2-yl]oxyprop-2-enamide 3-[(1,2,3,5,6,7-hexahydro-s-indacen-4-ylamino)methylidene]-N-[6-(methylcarbamoyl)-2-phenyl-1H-indol-3-yl]pyrrolidine-2-carboxamide 1-[4-[(dimethylamino)methyl]piperidine-1-carbonyl]-2,3-dihydroindole-5-sulfonamide 2-[2,4-dioxo-1-(3-phenylpropyl)-7,8,9,10-tetrahydropyrimido[1,2-a][1,5]diazepin-6-ium-3-yl]-N-(4-fluorophenyl)acetamide 2-[(1R)-4-chloro-5,8-dimethyl-3,6,9,10-tetraoxoanthracen-1-yl]oxyethanimidate N-(4,4-difluorocyclohexyl)-2-[4-(2-methoxybenzoyl)piperazin-1-yl]acetamide N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-6-bromo-3H-benzo[e]benzimidazole-2-carboxamide 4-[2,3-dihydroxypropyl(phenacyl)amino]benzenesulfonic acid N-azido-2,5-bis(9H-fluoren-1-yl)furan-3-amine 5-chloro-N,N,2-trimethyl-4-[[4-[1-(methylamino)propan-2-yloxy]phenyl]-[3-(trifluoromethyl)phenyl]methyl]aniline 2-(2-hydroxyethyl)isoindole-1,3-dione;2-methoxy-N-[4-[6-[(4-methylcyclohexyl)amino]pyridin-2-yl]phenyl]acetamide 1-(4,5-dimethylpyridine-2-carbonyl)-N-ethylpyrrolidine-3-sulfonamide (Z)-N'-[2-[4-[1-[5-(3,5-difluorophenyl)pyrazin-2-yl]oxyethyl]piperidin-1-yl]pyridin-4-yl]-3,3,3-trifluoroprop-1-ene-1,3-diamine 5-[2,3-dihydroxypropyl(phenacyl)amino]naphthalene-2-sulfonic acid 4-amino-5-(1,3-dimethyl-6-phenylpyrazolo[3,4-d]pyrimidine-4-carbonyl)-2-[(3S)-pyrrolidine-3-carboximidoyl]-1H-pyrazol-3-one 4-(2,5-difluorophenyl)sulfinylbenzaldehyde 6-(6,7,8a,9,10,11,12b-octahydro-5H-cyclohepta[b]indol-5-yl)-2-azido-4-N-(furan-3-ylmethyl)quinazoline-4,6-diamine N-(3,5-dichlorophenyl)-6-methyl-4-oxo-2-[(1R)-1-phenylethyl]sulfanyl-5H-pyrazolo[1,5-a]pyrazine-7-carboxamide 2-methoxy-N-(4-phenylbutyl)propan-1-amine 2-methoxy-3-[[(3S)-pyrrolidin-3-yl]amino]benzamide N-[(3R,4S)-1-(2-cyclopropylpyrimidin-5-yl)sulfonyl-4-methoxypyrrolidin-3-yl]cyclobutanecarboxamide;hydrochloride 2-(4-hydroxy-N-octylanilino)acetic acid 1-[2-(4-benzylpiperazin-1-yl)ethoxy]propan-2-one 5-[(2,3-dimethoxyphenyl)methyl]-3H-pyrido[4,3-d]pyrimidin-4-one 7-ethyl-2,3-dimethyl-1,9a-dihydrocarbazole (E)-1-[4-amino-3-(trifluoromethyl)phenyl]-N'-(4-benzoyl-2,6-dichlorophenyl)ethene-1,2-dicarbohydrazide 6-bromo-3,4-dihydro-2H-1,8-naphthyridine;ethane 3,5-bis(methoxycarbonyl)-2-(trifluoromethyl)benzoic acid [4-(3,4-dimethylphenyl)piperazin-1-yl]-[7-(ethoxymethyl)quinolin-5-yl]methanone (2-cyclopropylfuran-3-yl)-[(4S,5R)-1-methyl-2,7-diazaspiro[4.4]nonan-7-yl]methanone;formic acid 2,3-difluoro-1-[4-(4-pentylphenyl)cyclohexa-2,4-dien-1-yl]-6-[2-[4-(trifluoromethoxy)phenyl]ethynyl]naphthalene 2-[(5R)-5-[3-fluoro-4-[6-[(1E,3Z,5Z)-hepta-1,3,5-trienyl]pyridin-2-yl]phenyl]-2-oxo-4-[3-(trifluoromethoxy)phenyl]pyrrolidin-1-yl]acetic acid 3-[(1R,2S)-5-hydroxy-4-methyl-2-(2-phenylmethoxyethyl)-3H-furan-2-yl]pyrrolidine-2,5-dione 5-(4-bromophenyl)-2-methylpyridine;ethane 2,3-dihydroxy-N'-[3-(1H-indol-6-yl)phenyl]cyclohexane-1-carbohydrazide 3-(2,6-dimethyl-4-nitrophenoxy)oxetane 5-tert-butyl-2,3-dimethoxybenzoic acid 1-methoxy-2,3,4,5-tetranitro-6-phenylbenzene N-(3-fluorophenyl)-4-hydroxy-2,3-dihydro-1H-indene-5-carboxamide N-[1-(3,4-dimethylphenyl)ethenoxy]propan-2-amine N-[4-(3,3-dichloropropanoyl)phenyl]-2-ethoxy-N'-methyl-6-phosphanylpyridine-4-carboximidamide N'-hydroxy-3-methyl-5,6,7,8-tetrahydro-4H-cyclohepta[c]pyrazole-2-carboximidamide 5-(4-azidooxypyridin-2-yl)pyrimidine 6-[5-(benzylamino)-1,3,4-thiadiazol-2-yl]-N-(4-methoxybutanoyl)-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide 7-[(1S)-2-amino-3,3-dimethylbutoxy]-6-chloro-4-[3-(5-methylpyrazol-1-yl)propanoyl]-2,3-dihydro-1H-naphthalene-2-carboxylic acid 1-(4-chlorophenyl)-5-[2-(2,6-difluorophenyl)ethynyl]pyrazole 1-chloro-2-(3,4-dimethoxyphenyl)-3-[(2-ethylimidazol-1-yl)methyl]naphthalene N'-[2,3-bis(4-fluorophenyl)-1,2-dihydroquinoxalin-6-yl]ethane-1,2-diamine 3-amino-4-cyano-5-[4-fluoro-2-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrrole-2-carboxamide 4-(3-methylcyclohexyl)-N-[5-[1-[3-(trifluoromethyl)phenyl]ethoxy]pyridin-2-yl]piperidine-1-carboxamide 1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazin-2-one 5-(3,4-dihydroquinoxalin-2-ylmethylamino)-N'-hydroxypyrazine-2-carboximidamide 3-[(2Z,4E)-5-ethenyl-8-(methylideneamino)octa-2,4,6-trien-4-yl]phenol N-[2-(3,5-dimethoxyphenyl)ethyl]-N-methylpropanamide N-(4-methoxy-3,5-dimethylphenyl)-2H-pyrazolo[3,4-d]pyrimidin-7-amine 4-azido-2,6-dimethylbenzenesulfonamide 2-(3-fluoropyrrolidin-1-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine;hydrochloride N-[(5-ethylsulfonylpyridin-2-yl)methyl]pyridine-3-carboxamide [3-[4-(2,6-dimethylphenyl)triazol-1-yl]benzene-2-id-1-yl]oxy-dideuteriogermane;iridium 2-methyl-1,4,5-triphenylpyrrolo[3,2-c]carbazole 7-bromo-1-(3,4-dichlorophenyl)-6-fluoro-3-nitrosoindol-2-ol 4-amino-N-[[2,3-difluoro-5-(trifluoromethyl)phenyl]methylideneamino]benzamide (2R,3S)-1-azido-2,6-bis(phenylmethoxy)hexan-3-ol N-(1,3-benzothiazol-5-yl)-4-oxo-7-piperazin-2-yl-3H-thieno[3,2-d]pyrimidine-6-carboxamide 2-(1-cyclopropylindol-6-yl)oxypropanoic acid 3-[4-(2,5-dimethylphenyl)sulfonylpiperazine-1-carbonyl]-1H-pyrazin-2-one (3R,4S)-1-acetyl-3-[(2-chlorophenyl)methyl]-N-[2-(2,5-dioxopyrrolidin-1-yl)ethyl]piperidine-4-carboxamide N-(3-acetamidophenyl)-4,7-dioxo-2-propylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 3-[(2E,4Z)-hepta-2,4-dien-6-yn-3-yl]-5-phenylaniline 3-(methanesulfonamido)-4-phenylbenzenesulfinamide;1-methylpyrrolidine N-azido-2,3-diethoxybenzamide 2-(6-bromopyridin-3-yl)-N,4-dihydroxy-5-propan-2-ylbenzenesulfonamide 3-(dimethylamino)-N',2-bis[2-(dimethylamino)ethyl]benzenecarboximidamide 6-(7H-purin-2-yl)spiro[1,3-dihydroquinazoline-4,5'-piperidine]-2-one 3-[6-(azidomethyl)-4-ethoxypyridin-2-yl]-1H-pyrrolo[3,2-b]pyridine 2-(6-chloropyrimidin-4-yl)sulfanyl-N-methylbenzamide 4-azido-3,7-dimethyl-1-propan-2-ylbenzimidazol-2-one 2-cyclobutyloxy-N-[(E)-1H-indol-3-ylmethylideneamino]-6-morpholin-4-ylpyrimidine-4-carboxamide 2-methyl-5-[(2Z)-3,3,7-trimethylocta-2,6-dienoxy]benzenethiol N-[(Z)-2-aminoethenyl]formamide;1,4-diazepane;8-ethoxy-6-methoxy-4H-1,4-benzoxazin-3-one 2-[[3-methyl-4,7,10-tris(2-sulfanylidene-1H-pyrimidin-6-yl)anthracen-9-yl]oxy]ethanesulfonic acid 1-amino-7-chloro-2,3,4,5-tetrahydropyrano[2,3-c]pyridine-8-carboxylate 6-[(3,4-dimethoxyphenyl)methyl]-2-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-[4-(trifluoromethyl)pyridin-2-yl]pyridine-3-carboxamide 4-amino-2,6-dichloro-3-fluorobenzoic acid 4-[3-aminopropyl(methyl)amino]-2-methyl-1H-pyrimidin-6-one 1-[(2S)-4,8-dimethylnonan-2-yl]oxy-3-ethoxybenzene (2E)-N,4-dimethylhexa-2,4-dien-2-amine;8-fluoro-2-[4-(furan-3-yl)phenyl]quinoline 1-methyl-5-[4-(trifluoromethoxy)phenoxy]cyclohexa-3,5-diene-1,2-dicarboxylic acid [3-chloro-5-(4-cyanophenyl)phenyl]methylphosphonic acid 1-(3,5-dichlorophenyl)-4-hydroxypiperidine-4-carboxamide 2,6-dichloro-N-[(2,4-difluorophenyl)methyl]aniline;ethane (3R,4S)-1-[4-cyano-3-(trifluoromethyl)phenyl]-N,N-diethyl-2-methyl-4-(quinolin-8-ylsulfanylamino)piperidine-3-carboxamide 4-N,6-dimethyl-2-[4-(6-pyrrolidin-1-ylpyridazine-3-carbonyl)piperidin-1-yl]pyrimidine-4,5-diamine;formic acid 6-chloro-4-(2,3-dimethylanilino)quinoline-3-carbonitrile N-ethyl-2-[(5-oxo-6H-pyrido[3,4-b]pyrazin-7-yl)amino]-2-phenylacetamide N-(1,3-dimethylpyrazol-4-yl)sulfonylformamide 4-[[6-amino-5-(4-oxoquinoline-1-carboximidoyl)pyrimidin-4-yl]amino]butanenitrile 4-amino-2,6-dimethylbenzenesulfonic acid;[3-[5-[(2,6-dichlorophenyl)methoxy]pyridin-1-ium-2-yl]pyridin-2-yl]methanamine N-[3-(dimethylamino)propyl]-4-[[6-[2-[6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]pyridin-3-yl]pyrazol-3-yl]pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamide [(3R)-3-aminopyrrolidin-1-yl]-[5-azido-2-fluoro-4-methoxy-3-(6-methoxypyridin-2-yl)phenyl]methanone 6-chloro-8,9-dimethyl-5-pentan-2-ylidene-3H-benzo[e]benzimidazole 4-[2-(7,8-dihydro-5H-pyrido[3,4-d]pyrimidin-6-yl)ethoxy]benzonitrile 3-[2-(1,1-difluoroethyl)phenyl]-5-methyl-6H-pyrazolo[4,3-d]pyrimidin-7-one (5R)-7-chloro-1',3-diphenylspiro[1,4-dihydroquinoxaline-2,4'-piperidine] 5-(chloromethyl)-1-[2,6-dichloro-4-[[(3S)-pyrrolidin-3-yl]amino]phenyl]pyrazole-3-carboxamide;hydrochloride N-[1-amino-5-cyclopropyl-4-methoxy-3-(oxetan-2-ylimino)pentan-2-ylidene]-3-chloropyridine-4-carboxamide 5-[4-[(3R)-piperidin-3-yl]phenyl]pyridin-2-amine 3-[7-(dimethylamino)quinazolin-4-yl]oxypiperidine-1-carboxylic acid 2-azidooxycarbonylbenzoic acid [2-methyl-4-(pyridin-3-ylmethylamino)phenyl]-oxoazanium 5-[4-(azetidine-1-carbonyl)piperazine-1-carbonyl]-2-benzylpyridazin-3-one 6-(1,5-dihydropyrrolo[3,4-b]pyrrol-2-ylmethylidene)benzo[c]chromene 1-[3-[4-(1,2,3,6-tetrahydropyridin-5-yl)phenoxy]pyrrolidin-1-yl]propan-1-one 5-(3,4-dihydro-2H-quinoline-1-carbonyl)imidazolidine-2,4-dione N-[2-fluoro-4-(6-methyl-2,3-dihydropyridin-3-yl)phenyl]-8-oxo-7-phenylsulfanyl-5H-imidazo[1,2-a]pyrimidine-3-carboxamide 2-chloro-1-(2,3-dichlorocyclohexa-2,4-dien-1-yl)oxy-6-methoxynaphthalene 2-[(5R,10bR)-9-bromo-5-pyridin-4-yl-5,10b-dihydropyrazolo[1,5-c][1,3]benzoxazin-2-yl]-6-methoxyphenol 4-[3,5-dimethyl-1-(2H-tetrazol-5-yl)pyrazol-4-yl]-6-hydroxybenzo[c]chromen-9-one 3-(2,6-difluorophenyl)-4-phenylchromen-2-one 3-amino-6-[(Z)-1,3-bis(4-methoxyphenyl)prop-2-enylidene]cyclohexa-1,4-diene-1-carbonitrile ethane;2-methylpropan-1-amine;4,5,8-trimethoxynaphthalene-2,3-dione 5-(difluoromethyl)-N-(4-hydroxycyclohexyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 6-azido-1-(2,5-difluorophenyl)indole 3-[(3S)-3-hydroxypyrrolidin-1-yl]-N'-[1-(1H-imidazol-2-yl)-2-phenylethylidene]cyclobutene-1-carboximidamide (3S)-N'-[5,6-difluoro-2-(oxetan-3-ylmethoxy)-1H-indol-3-yl]pyrrolidine-3-carboximidamide 2-(3,4-dichlorophenyl)-N-[2-(diethylamino)ethoxy]-7-propan-2-ylpyrido[1,2-a]pyrimidin-4-imine 4-[3,5-bis(trifluoromethyl)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 4-[2,5-dimethyl-7-(trifluoromethoxy)benzimidazol-1-yl]sulfonylpiperidine-4-carboxylic acid (2S,3R)-4-[(1-methylpyrazol-4-yl)methoxy]-N-(oxolan-3-yl)-6-oxospiro[3.5]nonane-3-carboxamide 5-(4-nitrophenyl)iminopentanoic acid 1-(4,4,6,7,8-pentamethylnonan-5-yloxy)-4-(trifluoromethyl)benzene 2-[4-[3-(hydroxymethyl)phenyl]butoxymethylideneamino]propanoic acid 4-[2-(dimethylamino)ethoxy]-N-(3,6,8,9-tetrahydro-2H-[1,4]oxazino[2,3-f]purin-7-ylmethyl)aniline 2-[3-bromo-4-(4-phenylpiperazine-1-carbonyl)anilino]benzonitrile 4-[3,5-difluoro-4-(trifluoromethyl)phenyl]-2,6-dioxo-1,3-diazinane-5-carbonitrile N-(2-ethylphenyl)-4-methoxyiminobutanamide 2-[5-chloro-2-(2,4-difluorophenyl)sulfonylpyridin-3-yl]-6-methoxy-1H-benzimidazole 2-[(1R,6S)-3,8-dioxo-8-phenyloctanoyl]peroxycarbonylphenolate 5-cyclopropyl-4-[(3,5-ditert-butylphenyl)methoxy]-2-fluoroaniline 1-[(2R)-4,8-dioxo-6-[[3,3,5-trimethyl-1-oxo-7-(trifluoromethylsulfanyl)isoquinolin-2-yl]methyl]octan-2-yl]-3-(diphenylcarbamoylamino)thiourea 2,4-ditert-butyl-6-[(E)-1-[4-hydroxy-3-(trifluoromethoxy)phenyl]-2-nitroethenyl]phenol 6-[3-(4,5-diphenylimidazol-1-yl)phenyl]-2-(9H-fluoren-9-id-1-ylmethoxycarbonylamino)hexanoic acid;yttrium 4-[[(1R)-1-phenylethyl]amino]piperidine-1-carboxylic acid 5-(2,3-dihydroxyphenyl)-4-naphthalen-1-yl-N-propyl-1,2,4-triazole-3-carboxamide 2-amino-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxylic acid (Z)-1,2-dipyridin-2-ylhex-1-en-3-imine [2-methyl-5-[2-[(3E,5Z)-4-propan-2-yloxyhepta-1,3,5-trien-2-yl]oxyethylcarbamoyl]phenyl]boronic acid 3-(5,5-dimethyl-1H-1,2,4-triazol-3-yl)-4-(7-methoxy-2H-indazol-3-yl)pyrazole-1-sulfonamide N-[2-(1H-benzimidazol-4-yl)ethyl]-2,3,6-trifluoropyridine-4-carboxamide 1-[2,5-dimethoxy-4-(3-methylbutanoylamino)phenyl]-N,N-bis[(4-methoxyphenyl)methyl]triazole-4-carboxamide 4-(3-methylphenyl)sulfonyl-1-[3-(1,2-oxazol-5-yl)propanoyl]piperidine-4-carbonitrile 1-[7-(2,3-dichlorophenyl)spiro[5H-pyrido[4,3-d]pyrimidine-8,4'-piperidine]-6-yl]ethanone 2-(4,6-diphenylpyrimidin-2-yl)-1,8a-dihydroquinoline [1-(3,4-dimethoxyphenyl)cyclopropyl]-[4-[5-(3-hydroxyphenyl)-1,2,4-oxadiazol-3-yl]piperidin-1-yl]methanone 1-butyl-3,6-dimethoxy-7,8-dihydroquinolin-2-one 2-[4-(dimethylamino)-N-propylanilino]octanoic acid 3-[2,4-bis(propylsulfanyl)phenyl]pentanenitrile 3-[6-(diethylamino)pyridin-2-yl]-1H-pyrazine-2,5-dione (3-chloro-4-methoxyphenyl)-[4-hydroxy-1,4-di(propan-2-yl)piperidin-1-ium-1-yl]methanone N-(4,5-dihydro-1H-imidazol-2-yl)-5-fluoro-6-[(4-methoxyphenyl)methyl]pyridine-3-carboxamide 2-[5,7-difluoro-6-(3,4,5-trifluorophenyl)naphthalen-2-yl]-5-prop-1-en-2-ylpyridine 2-[4-(cyclohexa-1,3-dien-1-ylmethoxy)-2-ethylphenyl]acetonitrile 3-[[1,1-bis(4-chlorophenyl)butylamino]methyl]phenol 4-azido-2,3-difluoro-5-(4-methoxyphenyl)phenol [4-amino-2-(methylamino)phenyl]-phenylmethanone 7-[(4-methoxyphenyl)methyl]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-2,4-dione 2-[[5-(3,4-dimethylphenyl)-1H-imidazol-2-yl]sulfanyl]-N-(1,2,3,4-tetrahydroisoquinolin-7-yl)pentanamide N-(2,3-dihydro-1H-inden-5-yl)-3,4-difluorobenzamide 7-[(2,6-dichlorophenyl)methyl]-8-[(2,4-difluorophenyl)methoxy]-1,3,5-triazocan-2-one 6-chloro-4-[2-[(3,5-dimethylpyrazol-1-yl)methoxy]phenyl]-2-sulfanylidene-1H-pyrimidine-5-carbonitrile 2-methyl-N-(3-nitrophenyl)-N-[4-[(2-phenylpyrazol-3-yl)sulfamoyl]phenyl]propanamide (3S)-1-[[4-fluoro-6-methyl-2-(triazol-2-yl)pyridin-3-yl]carbamoyl]piperidine-3-carboxylic acid 3-[6-(2-hydroxyethylamino)-4,5-dimethylpyridin-2-yl]phenol (2S)-4-methylsulfanyl-1-phenylmethoxycarbonylpiperidine-2-carboxylic acid 4-(3,4-dichlorophenyl)-2-methylsulfanyl-1H-pyrimidin-6-one (3R)-3-[(4S)-3,3-difluoropiperidine-4-carbonyl]-5-[3-(2-methylquinolin-6-yl)phenyl]pentanoic acid 4-N,6-dibutylpyrimidine-2,4-diamine;hydrochloride 3-(6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazine-7-carbonyl)chromen-2-one 2-N,2-N-dimethyl-6-phenyl-1H-pyrimidine-2,4-diamine [4-[3-(dimethylamino)propyl-ethenylamino]phenyl]-[5-[7-(methoxyamino)quinazolin-2-yl]furan-3-yl]methanone 4-(2,1,3-benzoxadiazol-5-ylmethyl)-8-chlorospiro[2H-isoquinoline-1,1'-cyclopentane]-7-amine 4-azidooxy-6,7,8-trimethoxyquinoline N-[4-amino-1-(cyclohexen-1-yl)-3,4-dioxobutan-2-yl]-5-pyridin-4-ylfuran-2-carboxamide 3-[(1R)-2,5-dimethylcyclopenten-1-yl]-N-(pyridin-4-ylmethyl)propanamide (Z)-4,5-dimethyl-2-[1-[1-(2-phenylethylamino)pentan-3-ylidene]piperidin-4-yl]oxyhex-2-enal (3-azidoazetidin-1-yl)-phenylmethanone 6-(3,4-dimethylpentyl)-N'-hydroxypyridine-2-carboximidamide 2-(4-chlorophenyl)-1H-indene;1,4-dimethyl-2-(3-methylbutoxy)benzene 2-[2-hydroxyethyl(propyl)amino]benzenesulfonic acid 4-methyl-N-[1-(2H-pyran-3-yl)ethyl]piperidine-1-carboxamide 4-amino-6-[[3-(hydroxymethyl)-2,5-dimethoxyphenyl]methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-chloro-N-[(Z)-3-cyano-2-(4-methylcyclohexyl)prop-1-enyl]pyridine-4-carboxamide 1-[2,6-di(propan-2-yl)phenyl]-3-[4-methoxy-5-[3-methyl-6-[(E)-[(E)-1H-pyrazol-5-ylmethylidenehydrazinylidene]methyl]pyrazolo[1,5-a]pyrimidin-7-yl]thiophen-2-yl]urea N-butylformamide;N-(3,5-dichlorophenyl)sulfonylacetamide N-[2-(ethylamino)phenyl]-4,5-dihydrothieno[3,2-d][1]benzazepine-7-sulfonamide 3-[7-(4-fluorophenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-piperidin-4-yl-1H-pyrazolo[4,3-b]pyridine 2-(cyclopropylmethylamino)-4-[6-ethoxy-5-(1-hydroxyethylamino)pyridazin-3-yl]-N,N-dimethylpyrimidine-5-carboxamide 2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine;propane 4-[3-(4-hydroxyphenyl)-5-phenyl-1,2,4-triazol-1-yl]benzoic acid 5-[3,4-dihydroxy-5-(2-methoxyphenyl)sulfonylfuran-2-yl]thiophene-2-carboxylic acid 2-[(Z)-1-amino-3-iminoprop-1-enyl]sulfanyl-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine-3-carboxamide 4-[4-[2-(5,6-dimethylcyclohexa-1,3-dien-1-yl)propan-2-yl]phenoxy]phenol 2-amino-N-[(3S,5S)-1-(8-methoxyquinoxaline-6-carbonyl)-5-methylpyrrolidin-3-yl]pyridine-4-carboxamide 1-[3-(cyclohexylmethyl)-2,5-dimethylimidazol-4-yl]ethenamine N-[1-(3,5-dimethylphenyl)cyclopentyl]formamide N-[(1S)-5-chloro-2,3-dihydro-1H-inden-1-yl]-6-oxo-2-pyrimidin-2-yl-1H-pyrimidine-4-carboxamide 4-[2,6-difluoro-3-(methylamino)phenyl]oxan-4-ol N-(4-nitrophenyl)-N-[2-oxo-2-(propan-2-ylamino)ethoxy]octanamide N-[[1-[1-(cyclopropylmethyl)-3,5-dimethylpyrazole-4-carbonyl]piperidin-2-yl]methyl]ethenesulfonamide N-[4-[2-(methoxymethyl)cyclohexyl]butyl]quinazoline-5-carboxamide (1Z)-N-[(2-iodophenyl)methyl]-N,4-dimethylpenta-1,3-dien-1-amine 4-[5-(1,3-benzoxazol-2-yl)-4-(cyclohexen-1-yl)-6-methoxypyrimidin-2-yl]-N-[4-cyano-3-(trifluoromethyl)phenyl]piperazine-1-carboxamide N-[(1S,2R)-2-methoxycyclohexyl]-7H-purine-6-carboxamide 2-[(4R)-1-cyclopentyl-3,4-dimethyl-7-oxo-6H-pyrazolo[3,4-b]pyridine-5-carbonyl]oxyethanesulfonate N-[1,3,4-trimethyl-2-(4-nitrophenyl)quinolin-6-yl]acetamide (5R)-2,6-diethyl-7-methyl-1'-[[4-(trifluoromethyl)phenyl]methyl]spiro[5H-pyrazolo[1,5-a]pyrimidine-4,3'-indole]-2',6-dione (2S,3R)-N-[(1S)-5-chloro-7-fluoro-2,3-dihydro-1H-inden-1-yl]-1-methylsulfonylpiperidine-2-carboxamide [3-(methylamino)thiophene-2-carbonyl]oxidanium 1-[1-[2-[(4S)-4-acetyloxy-3,3-difluoropiperidin-1-yl]pyridin-4-yl]ethylcarbamoyl]cyclohexane-1-carboxylic acid N-[6-methyl-5-(1,3-thiazol-2-yl)pyridin-2-yl]-7H-purin-2-amine 4-(cyclobutylmethylamino)-2-[3,5-difluoro-N-methanimidoyl-6-(3-pyrrolidin-1-ylazetidin-1-yl)pyridin-2-yl]pyrimidine-5-carbonitrile [4-(trifluoromethyl)phenyl]boronic acid 4-[(3-fluorophenyl)methyl]-1H-pyrazole-5-carboxamide;piperidine 4-[(2R)-3,5-dihydroxypentan-2-yl]oxycarbonylbenzoic acid 5-[(1R)-2-cyclohexyloxy-6-(4,5-dihydro-1H-imidazol-2-yl)-7-methoxy-1-(3-methoxypropylsulfonyl)-3-oxoisoindol-5-yl]-N-methylidenepyridine-3-carboxamide (4S)-1-(4-methylphenyl)sulfonyl-4-[(3R)-piperidine-3-carbonyl]pyrrolidin-2-one;hydrochloride 3-[3-cyclopropyl-4-(furan-2-ylmethoxy)phenyl]oxirane-2,2-dicarbonitrile 4-azidooxy-2,7-dichloro-1H-indole 1-[(4-methoxyphenyl)methyl]-N-prop-2-ynylazepane-3-carboxamide (2S)-2-methoxy-2,4-dimethyl-7-pentoxy-3,4-dihydronaphthalene-1,1-diol 4-[3-(azidomethyl)phenyl]benzenecarboximidamide 7-fluoro-2-[2-[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]-1H-inden-1-yl]-2,3-dihydro-1H-indole N-[(3S,4R)-1-benzylpiperidin-3-yl]-2-(2-chloro-6-fluorophenyl)acetamide;hydrochloride 2-[(4,4-difluorocyclohexyl)methylamino]benzoic acid 2-[(4-ethenylphenyl)methoxy]oxane 6-[1,5-bis(4-fluorophenyl)pyrazol-3-yl]-N-[4-(4-methoxyphenyl)-2-oxo-1H-pyridin-3-yl]hexanamide [1-(5,6-diaminopyrimidin-4-yl)pyrrolidin-3-yl]-morpholin-4-ylmethanone 6-[2,3-difluoro-4-(trifluoromethoxy)phenoxy]-1-fluoronaphthalene [(Z)-3-chlorobut-1-enyl]benzene;N-[2-fluoro-5-(trifluoromethoxy)phenyl]formamide ethane;methanol;[(3R)-4-phenylpiperidin-3-yl]oxymethanethione 3-[5-(cyclohexylmethyl)tetrazol-1-yl]-N-phenylpropanamide 1-[2,4-dimethyl-3-[[4-methylidene-3-(5-methylfuran-2-yl)thieno[2,3-d]pyrimidin-6-yl]amino]phenyl]ethanone 5-(4-azidophenoxy)naphthalene-1,3-dione (5R)-N-(1,3-benzodioxol-4-ylmethyl)-7-chloro-2-(2-fluorophenyl)-6-[1-(4-hydroxybut-2-ynylamino)ethenyl]-5H-imidazo[1,2-a]imidazole-3-carboxamide 3-azido-5,6,7-trimethylthieno[2,3-f]indazole N-[(2S,3R)-1-[3,5-bis(trifluoromethyl)anilino]-3-hydroxy-4-methoxy-4-phenylbutan-2-yl]carbamate N-[(3,5-dimethoxyphenyl)carbamoyl]-2-oxopyrrolidine-1-carboxamide 3-chloro-N'-hydroxy-2,5-dimethylbenzenecarboximidamide 6-fluoro-3-hydroxy-N,3H-anthracene-2-carboxamide N-[4-(2-amino-3-methanimidoylpyridin-1-ium-4-yl)oxyphenyl]-6,7,8,9-tetrahydropyrido[1,2-a]indole-10-carboxamide 2-[3-[(4-chlorophenyl)methyl]-5,6-difluoroindazol-1-yl]acetic acid 2-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)quinazoline 1-(6-aminopurin-9-yl)propan-2-ol;dihydrate N-benzyl-1-hydroxynaphthalene-2-sulfinamide 3-(4-aminooxybutylamino)-7-chloro-1H-quinoxalin-2-one 5-[(2R,3S)-1-(benzenesulfinyl)pyrrolidin-3-yl]oxyisoquinoline N-azido-5-[2,4-bis(phenylmethoxy)phenyl]-1H-pyrazol-3-amine N-(2-chloro-6-hydroxyphenyl)-3,5-dimethyltriazole-4-carboxamide 3-cyclohexyloxy-N'-hydroxypyridine-4-carboximidamide 3-(5,6-diphenylpyrazin-2-yl)-N-[(Z)-[4-(dipropylamino)-2-hydroxyphenyl]methylideneamino]benzamide (E)-3,4,7-trimethylnona-2,5-dienamide;1,4,10-tris[2-(trifluoromethoxy)phenyl]benzo[f]quinoxaline 2-azidosulfanyl-3-(4,5-dimethoxycyclohexa-1,3-dien-1-yl)benzenethiol 6-(3-chlorophenyl)-1H-carbazole 3-[[2-[3-(4-fluorophenyl)-1,2-oxazol-5-yl]cyclopenten-1-yl]methoxycarbonylamino]piperidine-1-carboxylate [3-[[6-methyl-2-(2-propan-2-ylidenehydrazinyl)thieno[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]carbamic acid 2-[5-(dimethylamino)-2-fluoro-3-nitrophenyl]sulfonyl-N,3-dimethylaniline 4-[[5-methyl-2-(6-oxo-1H-pyridin-3-yl)-4,5-dihydro-1H-imidazol-4-yl]methyl]benzonitrile 4-bromo-1-butoxy-2,3-dihydro-1H-indene N-(3-nitrophenyl)-N-propylbutanamide 3-chloro-4-[2-hydroxy-3-(propan-2-ylamino)pyrrolidin-1-yl]sulfonylbenzonitrile (3R,4S)-1-azido-N-[2-[6-(cyclopropylmethoxy)pyridin-3-yl]ethyl]-3,4-dihydroxypiperidine-4-carboxamide N-[4-(6,7-dihydrothieno[3,2-d]pyrimidin-4-ylamino)phenyl]-5-(hydroxymethyl)thiophene-2-sulfonamide (4-chloro-3-methylphenyl)sulfonylmethanamine [3,5-dimethyl-1-(4-phenylbutanoyl)indol-2-yl]carbamic acid N-[(E)-1-[5-[2,3-difluoro-4-(3,3,3-trifluoropropoxymethyl)phenyl]-6-methylidene-2H-thiopyran-4-yl]ethylideneamino]ethanamine N-[5-methyl-6-(6-oxo-1H-pyridin-3-yl)-2,3,4,7-tetrahydro-1H-inden-4-yl]-5-phenylpentanamide N-[3-(dimethylamino)propyl]-5-[4-ethoxy-6-(4-fluorophenyl)-2,4-dioxo-1H-pyrimidin-5-yl]pentanamide N-(2,3-dihydro-1H-inden-5-yl)-6,7-bis[4-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]quinoline-3-sulfonamide N-[4-[2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxypropan-2-yl]phenyl]formamide;ethane N-[(4-tert-butylcyclohexylidene)methyl]-2-methoxy-1,3-thiazole-5-carboxamide N-(2,4-dimethoxyphenyl)-3-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]propanamide 3-[(2,3-dichlorophenyl)methyl]-1-methylpiperidine;hydrochloride 4-ethenyl-2,6-dimethoxybenzaldehyde 7-ethyl-1,4-dimethoxyisoquinoline 2-[4-[(3S)-4-methyl-5-oxomorpholin-3-yl]anilino]-6,7-dihydropyrrolo[1,2-a][1,8]naphthyridine-9-carboxamide (3S,4R)-N-[5-cyclopropyl-2-(6-oxo-1H-pyridin-3-yl)pyrazol-3-yl]-4-(4-ethoxyphenyl)pyrrolidine-3-carboxamide 1-(3-bromophenyl)sulfonylpyrrole 3-[4,6-bis(2-methylbutanoyloxy)naphthalene-2-carbonyl]oxy-1-[3-(4-carbamimidoylphenoxy)propyl]azetidine-3-carboxylic acid 6-[3-methylbutanoyl([1,2,4]triazolo[4,3-a]pyrazin-5-yl)amino]-4-hydroxynaphthalene-2-sulfonic acid N'-[4-chloro-2-methyl-6-(1,3-oxazol-5-yl)phenyl]ethanimidamide (4S)-2-(1,3-benzoxazol-2-ylsulfanylmethyl)-8-methoxy-7-methyl-3,4-dihydrochromen-4-ol 2-[(3Z)-5-[(4,5-dimethoxynaphthalen-1-yl)methylidene]cyclopenten-1-yl]acetic acid 4-[(5R)-5-azidopentyl]benzenesulfonic acid 2-[(4S,5R)-4-(6-cyano-1H-benzimidazol-2-yl)-3,7-dioxo-4,8-dihydropyrazolo[3,4-e][1,4]thiazepin-N-phenyl]acetamide 2-[4-(6,6-dimethyl-1,4,5,7-tetrahydroindazol-3-yl)-6-fluoropyridin-2-yl]oxy-N-[2-(1H-indol-5-yl)ethyl]propanamide (3R)-N-[6-methyl-1-phenyl-4,5-dihydropyrazolo[3,4-c]pyrazol-3-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 4-(3,5-dimethylphenyl)sulfanylpentane-2,5-dione 1-[2-(2,6-dimethylphenyl)propan-2-yl]triazole 1-(4-methylcyclohexa-2,4-dien-1-ylidene)naphthalene;[1-(4-methylphenyl)sulfanylazetidin-3-ylidene]methane 3-chloro-1-ethyl-6,8-difluoroquinolin-4-one N-(2,5-dichlorophenyl)-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide 2-methoxy-4,5,6a,11a-tetrahydroisoquinolino[1,2-d][1]benzazepine 5-[(4-bromophenyl)methyl]-2-methoxypyridine 2-[[3,5-dichloro-4-(4-methylsulfonylphenoxy)phenyl]methylidene]propanedinitrile 2-methyl-5-[5-[(E)-1,3-thiazolidin-4-ylidenemethyl]-2H-tetrazol-2-ium-1-yl]benzoic acid (3R)-5-bromo-3,4-dihydro-1H-isochromene ethane;2-(3-fluorophenyl)-N-[1-[6-methoxy-5-(4-oxobutylsulfonylamino)pyridin-3-yl]pyrrolidin-3-yl]acetamide 2-[(E)-1,2-bis(benzenesulfonyl)but-1-enyl]-3,5-dimethoxyphenol 2-amino-N,6-dimethyl-5-oxopentanamide;(E)-3-(4-chlorophenyl)sulfanyl-3-formamidoprop-1-en-1-olate (E)-3-[4-[2-methoxyethyl(methyl)amino]phenyl]-N,N-dimethylprop-1-ene-1,2-disulfonamide 1-azido-4-[(2R)-3,3-dimethylbutan-2-yl]oxybenzene N-(5,6-dihydrophenanthren-3-ylmethyl)propanamide 3-[[3,5-dioxo-2-(thiophene-2-carbonyl)pyrazolidine-1,4-diyl]amino]benzoic acid 2-[1-(3,4-dimethylphenyl)ethenyl]thiophene N-[(1R)-1-phenylethyl]-5,6-dihydropyrazolo[4,3-d]triazole-7-carboxamide 4-(aminomethyl)-3-[6-(diethylamino)pyridin-2-yl]benzenesulfonamide 2-[[8-(3,5-dimethyl-1H-pyrazole-4-carbonyl)-6,7-dihydro-5H-imidazo[1,5-a]pyrimidin-5-yl]oxy]ethyl-triphenylphosphanium;bromide 1-[2-[3-[(4R)-6,8-difluoro-1-hydroxy-5H--cyclohepta[d]imidazole-4-carbonyl]-2-methylphenyl]ethyl]pyrrolidin-2-one 4-methyl-7,9-dihydro-6H-pyrido[3,2-b]azepine 2-[(1R)-4,6-dichloro-5-phenylmethoxy-2,3-bis(trideuteriomethyl)cyclohexa-2,4-dien-1-yl]acetic acid 1-(2,4-difluorophenyl)-N',3-bis[N'-methyl-N-(1H-pyrazol-5-yl)carbamimidoyl]urea 4-(3-methylsulfanylpropoxy)benzenesulfonamide (2R)-4-methyl-N-[(1S,2R)-1-(oxan-2-yloxy)-2,3-dihydro-1H-inden-2-yl]morpholine-2-carboxamide 4-[(8R)-3-butyl-7,10-dimethoxy-1,2,9,11-tetrahydrobenzo[b]fluoren-6-ylidene]cyclohexa-1,5-dien-1-ol (1R)-1-[5,6-difluoro-2-methyl-3-[[4-(oxan-4-yl)piperidine-1-carbonyl]amino]quinolin-7-yl]-N-methyl-3-pyridin-3-yloxycyclohexa-2,4-diene-1-carboxamide 4-ethenyl-2-(3-hydroxycyclobutyl)sulfanylpyrimidine-5-carboxylic acid 2-N,4-N-dimethyl-1H-indazole-3,5-diamine 5-bromo-3,4-dideuterio-2-iodopyridine N-(4,6-dimethyl-1,2-benzoxazol-3-yl)-4-hydroxy-4-[4-(2H-pyrazin-1-ium-1-ylidene)cyclohexa-2,5-dien-1-ylidene]piperidine-1-carboxamide N-[2,6-dimethyl-4-(1,3-thiazol-5-yl)phenyl]prop-2-enamide;ethane 1-ethyl-2-[(4-hydroxycyclohexyl)methyl]-3H-imidazo[4,5-c]quinoline-6-carbonitrile 6-(5,6-dimethylimidazo[2,1-b][1,3]thiazol-3-yl)sulfanyl-3H-quinazolin-4-one (2R)-2-[4-[di(propan-2-yloxy)phosphorylmethoxy]phenyl]-2,3-dihydro-1-benzofuran N-[2-(azetidin-1-yl)phenyl]-N-cyclopropylformamide 3-fluoro-N-[(1R)-6-methylsulfonyl-2,3-dihydro-1H-inden-1-yl]benzamide 3-benzylsulfanyl-2,4,5,6-tetrafluorobenzenethiol 2-[5-[4,6-bis(ethenyl)naphthalen-1-yl]thiophen-3-yl]-2-oxoacetic acid 2-ethoxy-6,8-dimethoxy-3,4-dihydro-1H-isoquinoline (Z)-2-[amino(methyl)amino]-1-[4-fluoro-3-(trifluoromethyl)phenyl]but-2-en-1-amine 1-N,2-N,3-trimethyl-4-phenylpentane-1,2-diimine 1-bromo-7-[(3Z,5E)-5-chlorohepta-1,3,5-trien-2-yl]oxy-4-hydroxyisoquinoline-3-carboxylic acid;ethane 1-[1-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)piperidine-3-carbonyl]-N'-methanimidoylpyrrole-2-carboximidamide N-[(2S)-1-[2-amino-4-(4-bromophenyl)pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]cyclopropanecarboxamide;hydrochloride [7-(2,6-dimethylpyridin-4-yl)-1-[2-methoxy-5-(trifluoromethyl)phenyl]sulfonyl-3,4,4a,5,6,8,8a-octahydro-2H-1,7-naphthyridin-4-yl]methanol;ethane 2-(7-chloronaphthalen-1-yl)-N-[4-cyano-5-methoxy-6-[3-(1,4-oxazepane-4-carbonyl)phenyl]pyridin-2-yl]acetamide [4-(2,6-difluorophenyl)piperazin-1-yl]-(5H-pyrrolo[3,2-d]pyrimidin-2-ylamino)methanol 2-[6-(1,1-dioxo-1,4-thiazinane-4-carbonyl)isoquinolin-3-yl]-N-hydroxyacetamide 1-[2,6-diethyl-4-(N'-methoxycarbamimidoyl)phenyl]-3-(2-fluoro-6-iodopyridin-3-yl)urea 4-(aminomethyl)-6,8-dichloro-7-methoxyquinoline-5-carbonitrile;hydrochloride 2-[5-[6-(3,4-difluorophenyl)pyridin-2-yl]oxypentanoylamino]-N-methylidenebenzamide 6-(3-azidophenoxy)pyridine-3-carboxamide 7,7-dimethyl-1-phenyl-5,6-dihydropyrrolo[2,3-f]benzimidazol-2-one 5-[3,4-dihydroxy-6-(methoxyamino)oxan-2-yl]-1H-pyrimidine-2,4-dione 1,2-diamino-4-[2-(4-cyanophenyl)sulfanyloxyphenyl]-6-oxopyridine-3,5-dicarbonitrile 2-(2,5-dimethylanilino)-N'-hydroxypyrimidine-4-carboximidamide N-[3-(4-chlorophenyl)-1,2-oxazol-5-yl]-1-ethyl-6-methoxy-7-nitroindole-3-carboxamide 1-azido-2,3-difluoro-4-(trifluoromethyl)benzene 3-(cyclopropylmethoxy)-N,4-diphenylpyridin-2-amine N-azido-5-(3,4-difluorophenyl)-1-(2,6-dimethylphenyl)pyrazole-3-carboxamide 1-[2-(3,5-ditert-butyl-4-hydroxyphenyl)propanoyloxy]-3,3-dimethylbutane-1-sulfonic acid 4-[5-(4-azidopiperidin-1-yl)pentyl]phenol 3-[(1S)-1-aminoethyl]-5-methoxycarbonyl-4-oxothieno[2,3-d]pyrimidine-6-carboxylic acid 1-[4-(1-methylpiperidine-3-carbonyl)piperazin-1-yl]-2-pyridin-2-ylethanone 4-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-N-[4-methoxy-7-(piperidin-4-ylamino)quinazolin-6-yl]piperazine-1-carboxamide [(E)-(3,5-dibromo-2,4-dihydroxyphenyl)methylideneamino]thiourea 2-[4-(cyclopropanecarbonylamino)phenoxy]-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine-4-carboxamide 6-[6-chloro-1,4-dimethyl-5-(2-oxo-1H-pyridin-3-yl)sulfanyl-2-phenylindol-3-yl]hexanenitrile N-[3-(1,2-oxazol-5-yl)phenyl]-4,5-dihydro-1H-imidazole-2-carboxamide 2-[2-(dimethylamino)ethyl]pyrazolo[1,5-a]pyrimidin-3-amine 2-azido-5,7-dihydropyrrolo[3,4-b]pyrazine-6,8-dione 2-[3-(2,4-difluorophenyl)imidazo[1,5-a]pyridin-8-yl]oxy-N-methylethanamine 2-[5-azido-3-(oxolan-2-ylmethoxy)-1,4-diphenylpyrazol-4-yl]pyridine 2-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-3H-benzimidazole-5-carboxamide 2-methyl-5-[6-(trifluoromethoxy)pyridin-3-yl]pyrazole-3-carboxylic acid 4-[(3R)-2,3-dimethylbutoxy]phenol 3-amino-N-[2-(4-chlorophenyl)ethyl]-5-[4-fluoro-3-(morpholine-4-carbonyl)anilino]pyrazine-2-carboxamide 2-chloro-3-[5-(1,4-dioxan-2-yl)pentoxy]pyridine (3S,4R)-1-[(4-chlorophenyl)methyl]-N'-cyano-2-oxo-4-propan-2-ylpyrrolidine-3-carboximidamide 4-azidooxy-2,3-difluoro-5-methylpyridine N-[(E)-1H-indol-3-ylmethylideneamino]-7-morpholin-4-yl-2-phenylpyrazolo[1,5-a]pyrimidine-6-carboxamide N-[2-[4-(dimethylamino)phenyl]ethyl]-5,6-dihydroxy-4-oxo-1H-pyridine-3-carboxamide 1-(azidomethyl)-3-nitronaphthalene 1,3-dimethyl-2,4-bis(4-methylphenyl)-6,7-dihydro-5H-cyclohepta[d]imidazole 2-(4,5-dimethyl-2-propan-2-yloxyphenyl)-6,7,8,9-tetrahydro-[1,3]thiazolo[5,4-b]quinoline-5,12-dione N-[2-methoxy-3-(propan-2-ylsulfonylamino)phenyl]formamide 3-(4-chlorophenyl)-1-[(2S,5R)-2,5-dimethylpiperazin-1-yl]propan-1-one;2-fluoro-5-phenoxybenzenesulfonamide 4-amino-2,5-difluorobenzenesulfonic acid;ethane N-(2,4-dimethylphenyl)-1,3-thiazole-5-carboxamide;ethane (5-bromoindol-1-yl)sulfonylurea 2-[(4-hydroxy-1,3-dihydroisoindole-2-carbonyl)amino]acetic acid 2-[3-(1,3-benzodioxol-4-yl)-6-chloroquinoline-7-carbonyl]oxyacetic acid 1-chloro-4,7-difluoronaphthalene 2-bromo-N-ethyl-6-(5-nitro-1,3-benzoxazol-2-yl)aniline 3-[(2-chlorophenyl)methyl]-6-cyclopropylpyrimidine-4,5-dione 2-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)benzamide 5-ethenyl-3-[(Z)-1-methoxybut-2-enyl]sulfanylpyridine 4-[[(1S)-1-(5,7-dichloroquinolin-8-yl)ethyl]amino]-3-methylidene-N-propan-2-ylpyridine-2-carboxamide 4-N-(6-iodopyrazin-2-yl)-5-methoxy-2-N-[3-methyl-1-(trideuteriomethyl)pyrazol-4-yl]pyrimidine-2,4-diamine [1-(3,4-dihydroxycyclohexa-2,5-dien-1-yl)indol-5-yl]urea 4-[8-amino-1-(3,6-dichloro-2H-pyridin-1-yl)imidazo[1,5-a]pyrazin-3-yl]cyclohexan-1-ol [1-methyl-3-(2-methylidenebutoxy)naphthalen-2-yl]methanol 1-[[4-(5-oxo-3,4-dihydropyrazole-2-carbonyl)phenyl]methyl]indazole-7-carboxamide (2E,5S)-2-[(Z)-1-(4-chlorophenyl)ethylidenehydrazinylidene]-5-[(3,4-dichlorophenyl)methyl]-1,3-thiazolidin-4-one 1-(2-cyclobutylethenyl)-4-[1-[4-fluoro-3-(trifluoromethyl)phenyl]sulfanylpropan-2-yl]piperazine;dihydrochloride 3-[2-amino-1-(4-chlorophenyl)ethyl]-N-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]sulfanylbenzamide 2-[[(3aR,6aS)-1,2,3,4,5,6,6a-octahydrocyclopenta[c]pyrrol-3a-yl]methoxy]-5-chloroquinoline 4-fluoro-3-(1,2,2,3,3,5,5,6,6,7,8,9,10,11,12,12-hexadecadeuterioundecoxy)aniline 2-[(4-bromophenyl)methylsulfanylamino]ethanol ethane;6-methyl-2-oxo-N-[4-(trifluoromethoxy)phenyl]-1,3-dihydroimidazole-5-carboxamide 3-[2,6-bis(methylperoxy)phenyl]-1-phenylpyrazolo[3,4-d]pyrimidine 1-azido-3,6-dihydroxynaphthalene-2-sulfonic acid 3-(1-methylpiperidin-4-yl)-N-[6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[1,5-d][1,4]diazepin-2-yl)pyridin-2-yl]imidazo[1,2-a]pyrazine-6-carboxamide 2-[3,5-dibromo-4-(9H-fluoren-1-yl)phenyl]butanoic acid (2S)-N,3-bis[4-[butanoyl(propyl)amino]phenyl]-2-methoxypropanamide 1-[(2S,3R)-2-hydroxy-4-oxoazetidin-3-yl]-N,5-dimethoxyindole-2-carboxamide (E)-N-hydroxy-3-[3-(4,5,6,7-tetrahydro-1H-indazole-3-carbonylamino)phenyl]prop-2-enamide 2-[4,6-bis(trichloromethyl)pyrimidin-2-yl]oxybenzamide 2-(N-butanoyl-3,4-diethoxyanilino)decanoic acid N-(4,5-dimethylpyridin-2-yl)-3,3-difluorocyclobutane-1-carboxamide 2-amino-8,9-dihydroxy-6a,7,10,11b-tetrahydrobenzo[c]chromen-1-one 3-[[2,4-dichloro-6-(cyclopropanecarbonylamino)benzoyl]amino]-N-methylazetidine-1-carboxamide 2-methyl-4-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)propanoyl]piperazine-1-carboxylic acid 2-[1-[4-(3,5-dichloropyridine-4-carbonyl)piperidin-1-yl]ethyl]-3H-quinazolin-4-one 3,5-diamino-N-[(E)-2-bromopenta-1,4-dienyl]benzamide 1,4-difluoro-2-methylbenzene;6-(5-formylfuran-3-yl)-N-hydroxyhexanamide;methane 2-(4,5-dimethyl-1H-imidazol-3-ium-3-yl)-N-[2-[5-(6-fluoroquinolin-8-yl)-2,5-diazabicyclo[10.4.0]hexadeca-1(16),12,14-trien-2-yl]phenyl]acetamide 3-ethenyl-2-[(4-methoxyphenyl)methylidene]-6-methylindene N-[3-(4-bromophenoxy)phenyl]-2,5-dimethylpyrazole-3-carboxamide N-[2-(4,5-dihydro-1H-imidazol-2-ylamino)ethyl]-3-methoxybenzamide 1-methoxy-3,5-dimethylanthracene 2-bromo-1,3,5-trichloroanthracene 4-[4,6-bis(2,4,6-trimethylphenyl)-1,3,5-triazin-2-yl]benzene-1,3-diol 1-azidooxy-5,6-dibutyl-2H-benzimidazole 2-(5-chloropyridin-2-yl)oxy-N'-hydroxypyrimidine-4-carboximidamide 4-[(1S)-1-hydroxy-2,3-dihydrotetrazol-5-yl]-N-methylbenzamide N-cyclohexyl-4,5,6,7-tetrahydro-1H-benzimidazole-2-carboxamide 5-(2,6-difluorophenyl)-3-[(4-ethylcyclohexa-1,5-dien-1-yl)methylamino]-2-hydroxy-7-methylidenethieno[3,2-b]pyran-6-one 4-[2-(3,5-diaminophenyl)ethyl]-N,1-dimethoxybenzimidazol-2-amine 3-[2-(4-nitrophenyl)ethyl]cyclobutane-1,1,2,2-tetracarbonitrile 2-[6,7-difluoro-3-(4-methylphenyl)naphthalen-2-yl]-5-(2,3-dihydro-1H-inden-5-yl)pentanal 3-[(1Z)-buta-1,3-dienyl]-2-ethenyl-N'-methylidenecyclopenta-1,4-diene-1-carboximidamide;ethane 1,3-dichloro-2-(3-iodocyclohexa-2,4-dien-1-yl)oxybenzene 2-[(Z)-3,7-dimethyloct-1-enyl]phenol;ethane 2-[(4R)-2-oxo-1,3-oxazolidin-4-yl]quinoline-8-carboxamide 2-[4-(3-azidopropyl)phenyl]naphthalene 1-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-N-[4-fluoro-2-[[methyl-(5-propanoyl-4,5-dihydropyrimidin-2-yl)amino]methyl]phenyl]-3-N-methylpyrazole-3,5-dicarboxamide (3S)-N'-cyclohexyl-1-oxo-2,9a-dihydropyrrolo[1,2-a]indole-3-carboximidamide (2-carboxyphenyl)-[4-hydroxyimino-5,6,7,8-tetrahydrocyclohepta[b]thiophen-3-yl]azanium 1-[4,6-dihydroxy-5-(2-methylpropyl)-3-(3-nitrophenyl)sulfonyloxan-2-yl]-1,2,4-triazole-3-carbonitrile 2-(4,5-dihydro-1H-imidazol-2-yl)-1-[4-(trifluoromethoxy)phenyl]-5-[4-(2,2,3,3,3-pentafluoropropyl)phenyl]indole 2-[1,3-bis(4-phenylmethoxyphenyl)propylideneamino]oxyacetic acid 5-[3,4-bis(trifluoromethyl)phenyl]-N-cyclohexyl-2-hydroxypentanamide 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)quinoline;hydrochloride 6-azidooxy-4,4,7-trimethylchromene-2,3-dione 4-[5-(4-chlorophenyl)-2,3-dimethylpyrrol-1-yl]benzoic acid N-(2,5-dimethoxyphenyl)-4-[2-(3,4-dimethylphenyl)ethynyl]benzamide 2-[2,3-difluoro-4-(trifluoromethoxy)phenyl]-6-[4-[2-(5-propyloxolan-2-yl)ethynyl]phenyl]-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene [2-(2-ethyl-5-fluoropyrazole-3-carbonyl)cyclohexen-1-yl]azanide 5-[3,4,6,7-tetramethyl-9-(oxolan-2-yl)carbazol-1-yl]pyrido[3,2-b]indole 2-[(1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]-4,5-dimethylthiophene-3-carbonitrile N'-[4,5-dimethyl-2-(1H-pyrrol-3-yl)pyrazol-3-yl]ethanimidamide (4aR,8aS)-6-[3-[4-cyano-2-[5-methyl-1-(3-methyloxetan-3-yl)pyrazol-4-yl]phenoxy]azetidine-1-carbonyl]-4,4a,5,7,8,8a-hexahydropyrido[4,3-b][1,4]oxazine-3-carbonitrile 4-[2,3-bis(ethenyl)-5-methoxyphenyl]-5,6-dimethoxy-2H-1,7-naphthyridine 1-butyl-4-[2-(3,4-dimethoxyphenyl)ethenyl]cyclohepta-1,3,5-triene N-[2-oxo-1-(6-oxo-7H-purin-3-yl)ethyl]-N-propan-2-ylthiophene-2-carboxamide 1-azidooxy-2,5-dichloro-3-[(4-propan-2-ylphenyl)methoxy]benzene N-[5-(1H-indole-2-carbonyl)piperidin-3-yl]benzamide 5-chloro-2-[3,4-dihydro-1H-isoquinoline-2-carbonyl(methyl)amino]benzoic acid 2-[[7-(3-cyanophenyl)-6-[4-[(dimethylamino)methoxy]phenyl]-1,5-naphthyridin-4-yl]oxy]acetonitrile;ethane 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-oxo-2-[[6-(trifluoromethyl)pyridin-2-yl]amino]ethyl]acetamide (7R)-N,N-diphenyl-7-[4-(trifluoromethoxy)phenyl]-5-(3,4,5-trichlorophenyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide 3-[(2,4-diaminopteridin-6-yl)methyl]-1,5-bis(sulfanylidene)-2H-pyrido[2,1-f][1,2,4]triazin-4-one 3-hydroxy-2,4,6-triiodo-5-propan-2-yloxybenzaldehyde 2-methoxyimino-2-[2,3,6-trichloro-4-(4-hydroxyphenyl)phenoxy]acetaldehyde 2-[4-[5-(1,3-benzodioxol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]piperazin-1-yl]acetic acid [2-(methylamino)pyridin-4-yl]-piperidin-1-ylmethanone 2-methyl-6-(4-propan-2-yloxyphenoxy)-5-[3-pyridin-2-yl-1,2,4-oxadiazol-5-yl]pyrimidin-4-amine 2-[1-(5,6-dichloro-1H-benzimidazol-2-yl)ethyl]-3H-isoindol-1-one 4-[1,2,2,3,3,4,4,5,5,6,6,7,8,9,10,10,11,12-heptadecafluoro-4-(pyridin-2-ylamino)octoxy]phenol (3E,5Z)-7-fluoro-6-methyl-2-methylidene-1H-3-[(6-propanoyloxypyridin-2-yl)methyl]nona-3,5-dienoic acid 4-methyl-6-[6-(1,2-oxazol-3-yl)pyridine-3-carbonyl]piperidin-2-one (4-benzoylphenyl)sulfonyl-[3-hydroxypropyl(pyridine-2-carbonylsulfanylmethyl)carbamoyl]azanium 2-[(4-methoxycarbonylpiperazin-1-yl)amino]-N,5-dimethylbenzamide 2-(5,7,10,16-tetrazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-1(13),3,5,8,11,14(18),15,17,20-nonaen-6-yl)-4,6-dipyridin-3-ylpyrimidine 5-methoxy-4-methyl-7,8-dihydroisoquinoline 2-methyl-N,4-bis(propan-2-yloxy)benzamide 2-methyl-4-[[methylidene(1,3-thiazol-2-yl)amino]methyl]benzoic acid 1-azidooxy-2,3-dichlorobenzene 2-[(3E,5Z)-2-fluorohepta-1,3,5-trien-4-yl]-N-methoxy-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 3-(2-chlorophenyl)sulfanyl-N'-hydroxypyridine-4-carboximidamide (NE)-N-[(2-methylquinolin-4-yl)methylidene]hydroxylamine 5-[(1,3-dioxoisoindol-2-yl)methyl]-N'-hydroxypyridine-2-carboximidamide 5-[3-(cyclobutanecarboximidoyl)-1,2,4-oxadiazol-5-yl]-2-methoxy-N-methylaniline [7-butylsulfanyl-2-(4-chlorophenyl)pyrazolo[1,5-a]pyrimidin-6-yl]methanamine 2-[6-(3,4-difluorophenyl)pyridazin-3-yl]phenol 2,4-dichloro-N-cyclopropyl-5-[3-(1,1,1-trifluoropropan-2-ylideneamino)oxypyrrolidine-1-carbonyl]benzamide 1-cyclopropyl-3,4-bis(sulfanyl)anthracene-9,10-dione 1-(2,6-difluorophenyl)-4-[[5-(oxan-3-ylmethoxy)pyridin-2-yl]amino]pyridazin-6-one N-(1,3-dimethyl-5-oxopyrazolidin-4-ylidene)-2-iodobenzamide 2-ethyl-1',3'-dimethylspiro[4H-indazole-5,7'-6H-furo[2,3-f][1]benzofuran] 2-[5-(3,4-dimethoxyphenyl)-3-sulfanyl-1,2,4-triazol-1-yl]-N-[2-(oxolan-2-yl)ethyl]acetamide N-[(1R,2S)-2-(3-chlorophenyl)cyclopropyl]-5-methylimidazo[1,2-a]pyridine-6-carboxamide 4-N,2-diethylbenzene-1,3,4-triamine;ethane N-methylsulfonylbenzenesulfonamide N-azido-4,6-dimethyl-1H-benzimidazol-2-amine 4-[azido(phenyl)methyl]-2,6-ditert-butylphenol 5-(2,3-dihydro-1H-indol-7-yl)-4,4,5,6,6-pentafluorohexanoic acid 3-(4,5-dihydroxy-2-methylphenyl)-1-[4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]cyclohexyl]imidazo[1,5-a]pyrazin-8-amine N-[(5-chloro-2,3-dihydrothiophen-4-yl)methyl]-1-[2-(cyclobutylamino)pyridin-4-yl]methanamine 3-[5-amino-7-(pyridine-4-carboximidoyl)pyrazolo[1,5-a]pyrimidin-2-yl]sulfanylpropanoic acid 6,7-dimethyl-5,5a-dihydro-4H-benzo[de]quinoline-3-carboxylic acid N-[1-[3-[5-ethylsulfonyl-2-(1,1,2,2,3,3,4,4,4-nonafluorobutoxy)phenyl]propyl]piperidin-4-yl]-N-phenylbenzamide 1-methylsulfinyl-2,3-dihydrodibenzofuran (2S)-2-[4-bromo-2,5-difluoro-3-methyl-6-(methoxymethoxy)phenyl]-1,1,1-trifluoropropan-2-ol 3-(7,8-difluoro-4-oxoquinazolin-3-yl)azetidine-1-carboxylic acid 4-[6-(3,5-dimethylpiperidin-1-yl)pyridine-2-carbonyl]piperazine-1-carboxamide 5-chloro-2,4-dimethylbenzohydrazide 4-ethenyl-N-(2,3,5,6-tetrahydroindol-1-ylsulfonyl)benzamide N-(4-bromobutan-2-yl)-5,6,7,8-tetrahydroquinoxalin-2-amine 1-(4-hexylphenyl)-2,3-dipropoxybenzene N-[1-(4-methylpiperidine-1-carbonyl)cyclopropyl]benzamide 1,3-dimethyl-6-(4-propoxyanilino)pyrazin-2-one 2-fluoro-N-[(2-thiophen-3-yl-1,6-naphthyridin-7-ium-4-yl)carbamoyl]benzamide 4-[2-[4,6-bis(4-propoxyphenyl)pyrimidin-2-yl]-4-methylideneazepan-1-yl]butan-2-one 3-[4-chloro-2-(5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-yl)phenoxy]-N-[(1R)-1-(2,4-difluorophenyl)ethyl]propanamide 2-[1-(2,3-dihydroindole-1-carbonyl)cyclopentyl]-4,5-dimethyl-1H-pyrimidin-6-one [4-(3,4,5-trimethoxyphenyl)-1H-pyrrol-2-yl]methanamine;hydrochloride 6-[4-chlorobutyl(prop-2-enyl)amino]-5-nitronaphthalene-1-sulfonic acid N-[3,5-bis(trifluoromethyl)phenyl]-7-chlorothieno[2,3-c]pyridine-4-carboxamide 5-bromo-1',3'-dimethylspiro[1H-indole-2,4'-piperidine] N-[[3-(4-methoxyphenyl)pyrazin-2-yl]methyl]-1,2,4-triazine-6-carboxamide N-[(2R)-2-[(3-cyanophenyl)sulfonylamino]butyl]-4-[3,3-dimethyl-6-(trifluoromethyl)-2H-indole-1-carbonyl]benzamide 6-(difluoromethoxy)-2,4-difluoroacridine (3R,4S)-3-hydroxy-1-methyl-4-[4-[4-(1,2,2-triphenylethenoxy)phenoxy]butanoylamino]pyrrolidine-3-carboxylic acid 1-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-N-[3-ethoxy-5-(trifluoromethyl)-1H-pyrazol-4-yl]piperidine-4-carboxamide 2-(3,4-difluorophenyl)-1-methyl-N-[6-(2-pyridin-3-ylethynyl)pyridin-3-yl]indole-5-carboxamide 5-ethyl-2,4,6-triiodoaniline 4-[(3S,5R)-3-hydroxy-5-methylpiperidine-1-carbonyl]-6-propan-2-yloxypyridine-2-carbonitrile 4-bromo-2,3-dihydrodibenzofuran 3-[4-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfanylphenyl]-4H-1,2,4-oxadiazol-5-one 2-methyl-N-[5-[6-(4-methylphenoxy)pyridin-3-yl]-1H-pyrazol-4-yl]propanamide 4-[[3-chloro-6-(cyclopropylmethoxy)pyridin-2-yl]amino]-N-(2,6-dioxopiperidin-3-yl)benzenesulfonamide N-[(1R)-4-fluorocyclohex-2-en-1-yl]-6-oxo-2-phenyl-5,7-dihydrofuro[3,4-d]pyrimidine-3-carboxamide [4-[5-(1,2-benzothiazol-3-yl)hexa-1,5-dien-2-yl]piperazin-1-yl]-methylborinic acid 2-chloro-4-[(3,5-dichloropyridin-2-yl)amino]-N-pyrimidin-1-ium-4-ylbenzenesulfonamide N-(3,4-difluorophenyl)-7-hydroxy-2-oxoazepane-1-carboxamide 5-[(3,4-dimethoxyphenyl)diazenyl]-2-hydroxy-1,4-dimethyl-6-oxopyridine-3-carbonitrile 1-[4-(3,5-dichloropyridin-2-yl)oxy-7H-pyrazolo[1,5-a]azepin-6-yl]pyrrolidine-3-carboxamide 2-(3,5-dimethyl-1,2-oxazol-4-yl)-N'-[2-(5-methoxypyridin-3-yl)ethynyl]-1H-imidazo[4,5-b]pyridine-7-carboximidamide 3-amino-4-cyano-5-(3,4-dimethoxyphenyl)-1H-pyrrole-2-carboxamide N-[3-(benzylamino)pyrazin-2-yl]-2,6-dimethoxybenzamide 4-[3-[1-(1,2-benzothiazol-6-ylsulfonyl)azetidin-3-yl]oxyphenyl]butanoic acid (E)-3,4-dihydro-2H-naphthalene;7-methyl-5-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidine-2-carboxamide [4-[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]phenyl]methanamine 2-[7-amino-4-(furan-3-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]propanoic acid 2-(4-azidophenyl)-3,5-dimethoxypyridine 3-(2,4-difluorophenyl)sulfonyl-7-(piperidine-1-carbonyloxy)indolizine-6-carboxylic acid 5-(azidomethyl)-2-methoxy-1-benzothiophene 1-chloro-3-[4-[2,6-difluoro-4-(3,3,3-trifluoropropyl)phenyl]cyclohexen-1-yl]-5-(difluoromethoxy)benzene 1-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethyl)-3-N,5-diethylpyrazole-3,4-diamine (2S,3R,4R)-1-[2-(N'-cyclopentylcarbamimidoyl)propanoyl]-4-hydroxy-3-methoxy-5-phenylpyrrolidine-2-carboxylic acid;hydrochloride (4-benzoylphenyl)methylidene-ethoxycarbonylazanium (2R,3S)-N'-benzyl-1-cyclohexylbutane-2,3-diamine 4-[5-[3-(1,3-dimethylpyrazol-4-yl)phenyl]-6-ethylpyridin-2-yl]morpholine 2-hydroxypropanedioic acid;3-phenylchromen-2-one 4-[1,5-bis(3,5-dimethylphenyl)pentoxy]-N-methylaniline [4-[1-(5-chloropyridin-2-yl)cyclopropanecarbonyl]piperazine-1-carboximidoyl]carbamic acid 3-[2-(2-methoxyanilino)pyrimidin-4-yl]pyridine-2-carbonitrile 3-[3-(dimethylamino)propyl]-6,6a-dihydropyrrolo[2,1-c][1,4]benzothiazine-11-carboxylic acid N-methoxy-2-[3-[(Z)-2-(4-methylphenyl)prop-1-enyl]quinoxalin-5-yl]sulfanylethanamine;3-methyl-4,5-bis(phenylmethoxy)pyridine [1-(4-bromophenyl)ethylsulfanylmethyl]phosphane 1-(3,5-dimethylphenyl)-2-(3-methylbutoxy)ethanone (3S,4R)-3-azido-4-phenyl-1-[[3-(trifluoromethyl)phenyl]methylsulfonyl]azetidin-2-one [3-chloro-4-(2,5-difluorophenyl)pyrrol-1-yl]-pyrrolidin-1-ylmethanone 7-(4-methylpiperazin-1-ium-1-ylidene)-6,8-dihydrofuro[3,2-e]indole 2-cyclohexyl-2-[5-(4-fluorophenyl)thiophen-3-yl]acetic acid 5-benzyl-7,8-difluoro-1H-[1,2,4]triazolo[3,4-c][1,4]benzodiazepine 2-[2-(difluoromethoxy)phenyl]-4,5-dihydrobenzo[g][1,3]benzoxazole [3-(2,6-dimethylpyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]urea 2-[4-(cyclohexylcarbamoyl)pyridin-1-ium-1-yl]acetonitrile;4,6-dimethylpyrimidine 6-azido-N-[2,6-difluoro-4-(pyrrolidin-1-ylmethyl)phenyl]quinazolin-8-amine N-[(1E)-2,6-dimethylhepta-1,4,6-trienyl]-3,7-dihydro-2H-purine-9-carboxamide 1-[5,6-bis(ethenyl)pyridin-3-yl]-2-ethoxyethanone ethane;1-[4-(3-methylbutyl)phenyl]piperazine 5-[4-(2-aminoethyl)phenyl]-1H-indazole-3-carbonitrile 1-[4-(2,3-dichlorophenyl)piperazine-1-carbonyl]pyrazole-3-carboxylic acid 5-[2,6-bis(2-hydroxyphenyl)-4-phenyl-1H-1,3,5-triazin-4-yl]benzene-1,2,4-triol 5-[4-(2,6-difluorophenyl)phenyl]imidazolidine-2,4-dione (3R)-3-(4-fluorophenyl)-1',2'-dimethylspiro[1H-indole-3,4'-6,7-dihydropyrrolo[3,2-c]pyridine]-5'-one 6-azido-3-cyclohexylpyrazolo[1,5-a]pyrimidine N-(5,6-dimethoxypyridin-3-yl)-2-methyl-1-oxoisoquinoline-4-carboxamide 1-[3-methyl-4-(2H-triazol-4-yl)phenyl]benzotriazole 3-benzyl-6-(pyridine-4-carbonyl)-1,5,7,8-tetrahydropyrido[3,4-d]pyrimidine-2,4-dione 3-fluoro-4,5-dimethoxybenzenethiol;7-methylsulfanyl-2-(phenylmethoxycarbonylamino)heptanoic acid 6-fluoro-3H-quinazoline-4,7-dione 6-but-1-en-2-yl-2,4-dimethylcyclohexa-1,3-diene;ethane;N-[4-(4-methylphenyl)phenyl]propanamide 5-[2,5-dimethyl-3-(3-nitrophenyl)pyrrol-1-yl]pyridine-2-carboxylic acid 2-[[5,6-dimethyl-3-(1H-pyrazol-4-yl)-3a,7a-dihydrofuro[3,2-b]pyridin-5-ium-1-carbonyl]amino]ethanesulfonic acid 4-methyl-2-(2-phenylpropanoyl)chromene-5-carboxamide 2-(4,6-dimethylpyrazolo[1,5-a]pyrazine-2-carbonyl)benzoic acid 5-bromo-6-chloro-1,3-benzothiazole;methane 2-methyl-1,3-di(propan-2-yl)pyrazolo[3,4-d]pyrimidine 5-chloro-N-(2,4-dimethylphenyl)quinoline-8-carboxamide 3-[7-(2,5-dimethylphenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-methoxy-N-propan-2-yl-5a,6,8,9,10,10a-hexahydrobenzo[f]quinoline-8-carboxamide (4R)-4-(4-bromophenyl)-1,3-dimethyl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one (2E,4E)-3-[1-[4-fluoro-3-(trifluoromethyl)phenyl]ethoxy]-5-pyrimidin-5-ylhexa-2,4-dienoic acid 2-[4-(azidomethyl)piperazin-1-yl]benzimidazole (E)-3-[4-[1,2-bis(ethenyl)imidazo[4,5-c]quinolin-7-yl]phenyl]prop-2-enal 4-benzylcyclohexan-1-amine N-(4-fluorophenyl)-N'-[(6Z,7E,9S)-11,16-dihydroxy-3-methyl-8-oxo-1-azabicyclo[9.4.0]pentadeca-10,12,14-trien-9-yl]octanediamide 4-(2-aminoethyl)-N-[(1S,3R)-3-[(3-chloroquinolin-6-yl)methyl]cyclopentyl]-1,2-oxazole-5-carboxamide;dihydrochloride 2-[N-(cyanomethyl)-3,4-dihydroxyanilino]acetonitrile 1-[5-[3,4-bis(phenylmethoxy)-5-(phenylsulfanylmethyl)furan-2-yl]-1,2-oxazol-3-yl]propan-1-one (5Z)-2-(2,4-dimethylphenyl)imino-5-[[3-fluoro-4-[2-oxo-2-(propylamino)ethoxy]phenyl]methylidene]-1,3-thiazolidin-4-one 6-(5,5-dimethyl-2,3,4,7-tetrahydro-1H-azepino[2,1-b]quinazolin-9-ylidene)-4H-1,4-benzothiazin-3-one 1-butanoyl-N,2-dimethyl-3,4,6,7,8,9-hexahydropyrido[3,4-b]indolizine-3-carboxamide 2-[(3,5-dichloropyridin-4-yl)sulfanylamino]-N'-hydroxybenzenecarboximidamide N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]-1,3,5-trimethyl-4-(methylamino)pyrazole-4-carboxamide 3-[6-(dimethylamino)hexylsulfanyl]phenol 2-amino-N',7-dimethoxy-9H-pyrimido[4,5-b]indole-3-carboximidamide 3-(azidomethyl)-N-(3,3-difluorocyclobutyl)benzamide 1-[4-(2,2-dimethoxyethyl)phenyl]sulfonyl-6,7-bis(ethynyl)indole 3-[1-[(E)-but-2-enoyl]piperidin-4-ylidene]indole-2,5-dione N-[(6S)-6-(ethylamino)-5,6,7,8-tetrahydrobenzo[f][1]benzothiol-2-yl]-3-(trifluoromethoxy)benzamide 3-[[6-(5-chlorothiophene-2-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]amino]propanoic acid 5-methyl-2-methylidene-7-[[(3S)-pyrrolidin-3-yl]amino]-N-[4-(trifluoromethoxy)phenyl]heptanamide 4-(2,3-dihydroindole-1-carbonyl)benzonitrile 5-[(3,4-difluorophenyl)methoxy]-N'-hydroxypyridine-2-carboximidamide 2-[(Z)-(1,3-diethoxy-6-hydroxyhexan-2-ylidene)amino]-4-nitrobenzonitrile 1-[6-azidooxy-2,3-dichloro-5-(trifluoromethyl)phenyl]-4-chlorobenzene 2-(3-chlorophenyl)-4-[1-(4-fluorocyclohexa-2,4-dien-1-yl)ethyl]pyrimidine 2-(7,8-difluoronaphthalene-1-carbonyl)propanedioic acid 2-(3,4-dimethoxyphenyl)-1-(3-fluoropyrrolidin-1-yl)ethanone 2-[2-(4,5-dihydrobenzotriazol-1-yl)phenoxy]acetonitrile N-[[(1R,3aS,6aR)-5-[5-fluoro-2-(trifluoromethyl)benzoyl]-1,2,3,3a,4,5,6,6a-octahydropentalen-1-yl]methyl]cyclopentanecarboxamide 1-[7-[2,5-dimethyl-4-(oxan-4-yl)phenyl]-3H-azepin-6-yl]-N-[(4-fluoro-3-methoxyphenyl)methyl]ethenamine;formaldehyde (2R)-6-[[(3aR,8aS)-7-[4-(3-chlorophenyl)piperazine-1-carbonyl]-9-methyl-1,3,3a,4,5,6,8,8a-octahydropyrrolo[1,2-a]azepin-2-yl]oxy]-7-fluoro-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxylic acid (2S,3R)-4-methyl-N-[2-(6-oxo-1H-pyrimidin-4-yl)ethyl]-3-phenylmorpholine-2-carboxamide [5-methyl-4-(2,2,3,3-tetrafluoropropoxy)pyridin-2-yl]hydrazine N-(3,5-dichlorophenyl)sulfanyl-4,6-bis(2-methoxyphenyl)pyridin-3-amine;ethane 2-[(6S)-3,5-dioxo-1,4-benzoxazin-7-yl]-N-(5-fluoro-6-methoxypyridin-3-yl)acetamide N'-cyclopropylsulfanyl-4,6-difluorobenzenecarboximidamide 1-[(3S,4S)-4-methyl-2-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-1-yl]propan-2-one 3-hydroxy-N'-(4-nitrophenyl)-2-(1,2,4-triazol-1-ylmethoxy)butanimidamide 1-[[(2S)-2-[[(2R,3R)-2,6-dimethyloxan-3-yl]carbamoyl]morpholin-4-yl]methoxy]-7-ethoxyisoquinoline-6-carboxamide 3-(2-chlorophenyl)imino-4H-1,4-benzoxazin-6-amine 1-[3-[2-(ethylamino)pyrido[3,4-d]pyrimidin-6-yl]phenyl]-N',N'-dimethylbutane-1,4-diamine N-(4-bromobutan-2-yl)-6-chloropyridine-3-carboxamide 3-[4-(difluoromethoxy)phenyl]-5-[1-[2,5-dimethyl-4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperazine-1-carbonyl]cyclopropyl]-1H-imidazo[4,5-b]pyrazin-2-one 2-[[4-(6,7-dimethoxyquinolin-3-yl)phenyl]carbamoylamino]acetic acid 4-(1,3-benzothiazol-2-yl)-N-[4-(2-morpholin-4-ylethoxymethyl)-1,3-thiazol-2-yl]benzamide [6-(4,4-difluoropiperidine-1-carbonyl)pyridin-3-yl]carbamic acid 2-azidooxy-1,3-dimethyl-5-propan-2-ylbenzene 2-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-(3-methylbutylsulfonyl)indole-6-carboxylic acid 2-(cyclopentanecarbonylamino)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-5-carboxylate 1-[(E)-3,3-dimethylbut-1-enyl]-2,4,5-trifluoro-6-propan-2-yloxynaphthalene;ethane [4-[5-(2,3-dihydro-1H-indene-5-carbonyl)-1,6-dimethylpyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]-morpholin-4-ylmethanone 6-(2,4-difluorophenyl)-N-[3-[(2S)-1-hydroxypropan-2-yl]oxyphenyl]imidazo[1,2-a]pyridine-8-carboxamide N-[1-cyclopentyl-2-[(2-methoxyphenyl)methylamino]-2-oxoethyl]piperidine-4-carboxamide;dihydrochloride 2-[3-(3,5-dimethoxyanilino)quinoxalin-2-yl]sulfanyl-1-(4-fluorophenyl)ethanone;4-[6-(3-fluorophenyl)pyrimidin-4-yl]piperidine 1-[(3S)-5-cyclopropyl-2,6-dioxopiperidin-3-yl]-3-[(4-pyrazol-1-ylphenyl)methyl]urea [4-[6-azido-2,5-dichloro-3-(trifluoromethyl)phenyl]piperidin-1-yl]-cyclopropylmethanone N-[2-(1-methylpyrazol-4-yl)ethyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide [2,3-bis(methoxycarbonyl)phenyl]boronic acid [2-amino-3-[4-(1,3-dimethylpyrazolo[3,4-b]pyridine-5-carbonyl)-2,6-dimethylphenyl]prop-2-enylidene]azanium 2-[5-cyano-1-(2,6-dichloro-3,5-dimethoxyphenyl)imidazol-4-yl]propanamide 4-[2-[(3,5-dichlorophenyl)methyl]tetrazol-5-yl]benzaldehyde 4-[(2E,5Z)-6-methoxyhepta-2,5-dienyl]-2-[2-[[methyl(propan-2-yl)amino]methyl]quinolin-6-yl]-1H-pyrimidin-6-one 2-[(6-methylpyridin-3-yl)methylamino]-1,3-benzothiazol-4-ol N-[2-(dimethylamino)ethyl]-1-(4-oxo-3H-quinazoline-2-carbonyl)piperidine-2-carboxamide 5-bromo-4-(3,4-dihydro-2H-chromen-6-yl)-1-[(4,6-dimethoxypyrimidin-2-yl)methyl]pyridin-2-one N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(2H-tetrazol-5-yl)morpholine-4-carboxamide 1-azido-3,5-difluoro-2-nitrobenzene 7-[(4-bromophenyl)methyl]cyclohepta[d]pyrimidin-2-amine 3-[(4-ethenylphenyl)methylamino]propanenitrile;1-fluoro-4-methoxybenzene 4-[(5,6-dichloronaphthalen-2-yl)amino]-N-(2,3-dihydroxypropoxymethyl)butanamide (3-ethoxycarbonylpyridin-2-yl)-methylidene-propan-2-ylazanium 2-[(1,4-dioxonaphthalen-2-yl)methoxy]acetate 2-[(3R)-3-aminopiperidin-1-yl]-6,8-dibromo-N-(cyclopentylmethyl)pyrazolo[5,1-c][1,2,4]triazin-3-amine 4-(2,3-difluorophenyl)benzenethiol 4-[(3R)-3,4-dimethylpiperazin-1-yl]-N-[4-methyl-2-[6-(trifluoromethoxy)pyridin-3-yl]phenyl]-5-(trifluoromethyl)pyrimidin-2-amine 5-[(6-bromo-3,4-dihydro-2H-1,8-naphthyridin-1-yl)sulfonyl]isoquinoline 2-[1'-[2-methylpropanoyl(thiophene-3-carbonyl)amino]spiro[2H-indole-3,3'-pyrrolidine]-6-yl]acetic acid 4-[(3S)-3-cyclopentyl-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione;N-(4-ethylphenyl)sulfanylformamide (3-cyclohexa-1,5-dien-3-yn-1-ylphenyl)boronic acid (4R)-4-[3-ethoxy-4-[[3-fluoro-5-methyl-4-(oxan-2-yloxy)phenyl]methoxy]phenyl]-1,3-dimethyl-6,7,8,9-tetrahydro-4H-pyrazolo[3,4-b]quinolin-5-one 2-[2,6-dichloro-N-(4-hydroxybutyl)-3-methylanilino]propanoic acid 3-[(2E,4Z)-6-[ethenyl-[(2R)-1-hydroxybutan-2-yl]amino]hepta-2,4,6-trien-3-yl]oxy-N'-hydrazinylidenebenzenecarboximidamide;pentane (5Z)-2-imino-5-[[1-[4-methyl-3-[3-(trifluoromethoxy)phenyl]phenyl]pyrazol-4-yl]methylidene]imidazolidin-4-one 1-[2-cyclobutyl-6-(3,5-dichloropyridin-4-yl)pyrimidin-4-yl]oxycyclopentane-1-carboxylic acid 2-(4,5-dihydroimidazol-1-yl)-6H-benzo[c]chromene 2-[N'-(cyclopropylmethyl)carbamimidoyl]-1,3-thiazole-4-carboxylic acid 1-[(3S)-5,6-difluoro-3,4-dihydro-2H-chromen-3-yl]-N-methylidene-1-[4-(trifluoromethoxy)phenyl]methanimine (2-amino-1H-imidazol-5-yl)-[4-hydroxy-4-[(1,3,5-trimethylpyrazol-4-yl)methyl]piperidin-1-yl]methanone 2-cyclopropyl-1'-[[5-(trifluoromethoxy)pyridin-3-yl]methyl]spiro[6,7-dihydropyrrolo[2,1-c][1,2,4]triazine-8,3'-pyrrolidine]-3,4-dione;2,2,2-trifluoroacetic acid 7-(1-methoxypropan-2-ylamino)-5,6-dimethyl-3H-quinazolin-4-one 6-methylsulfanyl-1-phenyl-3,4-dihydro-1H-[1]benzothiolo[2,3-c]pyridine 2-(cyclopropylmethoxy)-N-[1-ethenylsulfanyl-4-(trifluoromethoxy)pentan-3-yl]pyridine-3-carboxamide 3-(benzenesulfonylmethyl)-N-diazobenzenesulfonamide (5S)-2-[(3R,4S)-3-fluoropiperidin-4-yl]sulfanyl-1-(4-methoxyphenyl)sulfonyl-3-methyl-6-(trifluoromethyl)-5H-pyrrolo[3,2-b]pyridine 3-[(2-chlorobenzoyl)amino]-4,5,6,7-tetrahydro-1H-indazole-5-carboxamide 5-[6-(2,4-difluorophenoxy)pyridin-3-yl]-N'-hydroxypyrazolo[1,5-a]pyrimidine-3-carboximidamide 6-[2-chloro-4-(3,3-dimethylbutanoylamino)anilino]-N-(2-hydroxyethoxy)-5-propan-2-ylpyridine-3-carboxamide 1-(2-aminoethyl)-N-phenylmethoxypyrazole-3-carboxamide 1-(benzenesulfonyl)-4-methylsulfanylpiperazin-2-one 2-[2-(3,4-dichlorophenyl)ethylamino]-4-[3-[3-(trifluoromethyl)phenyl]propyl]cyclohepta-1,3,6-triene-1-carboxylic acid 2-[N-(benzenesulfonyl)-4,5-dimethyl-2-phenyldiazenylanilino]acetic acid [4-(4-cyanoanilino)phenyl]methyl-bis[2-(diethylamino)ethyl]sulfanium N-[(4S)-1-acetyl-3,6-dihydro-2H-pyridin-4-yl]-7-fluoro-N'-phenylindole-1-carboximidamide 1-(6-benzylsulfanyl-3,4-dihydro-2H-pyran-5-yl)ethanone 5-[(3,4-dihydroxyphenyl)methyl]imidazolidine-2,4-dione 1-[4-hydroxy-2,5-di(propan-2-yl)phenyl]propane-1-sulfonate 4-methoxy-N-[(E)-1H-indol-3-ylmethylideneamino]benzenesulfonamide 3,6-dicyclohexyl-1H-quinolin-2-one 2-[1-(5-chloropyridin-2-yl)-4,6-dioxo-8H-pyrazolo[3,4-e][1,4]thiazepin-7-ylidene]propanedinitrile 1-(azidomethyl)-2,4-dichloro-5-fluorobenzene N-(2,6-dimethoxypyrimidin-4-yl)-4-[ethylsulfonyl(phenacyl)amino]benzenesulfonamide 4-[(2S)-3,4-dimethylpentan-2-yl]pyridine 3-[2-methyl-4-[(2E)-penta-2,4-dien-2-yl]imidazol-1-yl]propanenitrile 1-[(E)-2-chlorohex-3-enyl]-2,5-difluoro-4-methoxybenzene (4-azidopyrimidin-5-yl)-[3-bromo-2,6-difluoro-5-[methyl(oxan-2-ylmethyl)amino]phenyl]methanone [4-(3,5-dichloropyridin-2-yl)piperazin-1-yl]-(6-methoxypyrimidin-4-yl)methanone 5-[1-azido-2,2-dimethylpropyl(cyclohexa-2,4-dien-1-ylidene)amino]benzene-1,3-diamine 4-[8-amino-3-(1H-pyrazol-5-yl)imidazo[1,5-a]pyrazin-1-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]cyclohexane-1-carboxamide (2Z,3Z)-2-ethylidene-5-methyl-6-prop-1-en-2-yl-4-pyridin-2-ylhexa-3,5-dienenitrile 5-amino-N'-[2-[3,4-bis(phenylmethoxy)phenyl]ethyl]pyridine-3-carboximidamide;hydrochloride 4-azidooxy-5,6-dimethyl-2-(methylideneamino)benzenesulfonamide 4-(5-chloro-2-fluorophenyl)-N',N'-dimethylpiperidine-1-carbohydrazide N-(7-cyano-2,3-dihydro-1H-inden-4-yl)methanesulfonamide 1-(3,5-dichloropyridine-4-carbonyl)-2-[(2S)-oxolan-2-yl]pyrazolidin-3-one N-[(Z)-1H-indol-3-ylmethylideneamino]-4-propan-2-ylbenzenesulfonamide 1-[(4R,5S)-2,2-dimethyl-5-phenylcyclopropyl]pyrrolidine 2-(1-ethylcyclopentyl)-4-methoxybenzaldehyde 3-[2-(4-fluorophenyl)sulfonylethylamino]thiophene-2-carboxylic acid N-[6-[1-(benzylsulfonylamino)cyclobutyl]pyridazin-3-yl]-2,4-dimethylpyrazole-3-carboxamide (3R)-N,2-dimethyl-4-oxo-1,3,8,11-tetrazatricyclo[8.6.0.03,7]hexadeca-9,12-diene-5-carboxamide (3E,5Z)-N-[2-methyl-4-[2-[4-[(3-methylazetidin-1-yl)methyl]phenyl]thieno[3,2-b]pyridin-7-yl]oxyphenyl]hepta-1,3,5-triene-3-sulfonamide 2-(3-methylthiophen-2-yl)-7,8-dihydrochromene-4-thione N-(5-ethylsulfonylpyridin-2-yl)-1-methyl-3,4-dihydro-2H-isoquinoline-7-carboxamide N-[4-(2,2,2-trifluoroacetyl)phenyl]-3,5-dihydropyrazole-2-carboxamide N'-[(2Z,4Z)-3-cyanohexa-2,4-dienyl]-N-[4-(1H-indole-6-carbonylamino)phenyl]oxamide 2-[(E)-2-[4,5-bis(4-chlorophenyl)furan-3-yl]ethenyl]-1-cyclohexa-1,5-dien-1-ylbenzimidazole 4-chloro-N-[2-methyl-5-(morpholin-4-ylmethyl)pyrazole-3-carboximidoyl]benzamide 5-[3,4-difluoro-2-(2-fluoro-4-methylanilino)benzoyl]-N-ethylimino-1-methoxy-4-methylidenepyridine-3-carboxamide 1-benzyl-3-[5-(trifluoromethyl)pyridin-2-yl]thiourea [3-methoxy-4-(1,2,4-triazol-4-yl)phenyl]methanamine;dihydrochloride (5S,7R)-3-chloro-N-cyclohexyl-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide N-[(1R)-3-azidocyclopentyl]-5,6-dichloro-2-oxochromene-3-carboxamide 3-(2-tert-butylpyridin-4-yl)-4-methoxypyridine 4-azido-7,8,9,10-tetrahydrotetracene (Z)-2,3-bis[3-methylbutyl(pentyl)amino]-N'-(1-pyridin-4-ylethylidene)prop-2-enediamide 2-(3,4-dihydro-2H-quinolin-1-yl)-1,3,10-triazatetracyclo[6.5.0.02,6.07,12]pentadeca-5,7,9-triene [3-(dimethylamino)piperidin-1-yl]-[2-fluoro-5-nitro-6-[4-(trifluoromethylsulfanyl)pyrazol-1-yl]pyridin-3-yl]methanone N-[5-(4-fluorophenyl)-1,2-oxazol-3-yl]-3-methylidenepentanamide 4-chloro-2-ethyl-7-nitroquinoline (2R,3S)-N-[(1R)-1-(3-chloro-4-fluorophenyl)ethyl]-4,4,4-trifluoro-2,3-dihydroxybutanamide 2-(3-bromoquinolin-8-yl)oxyacetic acid 2-[4-(3,5-dimethyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]acetic acid N-(1,3-dioxol-4-yl)-2-methoxy-5-propan-2-ylidenebenzenesulfonamide 2-N-[2-(1H-imidazol-5-yl)ethyl]-4-N-phenylbenzene-1,2,3,4,5-pentamine 6-chloro-N,N-diphenylnaphthalene-1-sulfinamide 3-benzyl-2,4-dichloro-1-fluorocyclohexa-2,4-diene-1-carboxylic acid 3-[(1S,4R)-2-methyl-4-phenylcyclopentanecarbonyl]oxypyrrolidine-1-carboxylic acid N-(5-bromopyridin-3-yl)sulfonylcyclohexanecarboxamide 4-(2,3-difluorophenyl)-5,7-dihydro-4H-thieno[2,3-c]pyran 5-bromo-3,8a-diphenyl-1H-benzo[g]indole 2-[6-(4-ethylpiperazin-1-yl)pyridin-3-yl]pyridine-4-carbonitrile 4-amino-6-[(3,4-dichlorophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-[1-(4-chlorophenoxy)ethyl]-4-methylsulfonyl-6-(trifluoromethyl)-3,4-dihydropyridine 5-bromo-4-cyclopropyl-2-methyl-1H-pyrimidin-6-one 5-[2,3-dimethyl-4-(3-oxomorpholin-4-yl)phenyl]-N-ethoxyfuran-3-carboxamide 3-[2,4-dimethyl-6-(1H-pyrrol-3-yl)phenyl]-N,N-diethylpropan-1-amine 3-[(3,5-diethylphenyl)methoxy]phenol [(2S,3R)-4-azido-1-(methylamino)-3-phenylbutan-2-yl]carbamic acid 2-methyl-2-[5-(phenylsulfanylamino)pentylamino]propanenitrile 3-(3,5-dimethylpyrazol-1-yl)benzoic acid 6-ethylimino-2,3,5-triphenyl-5H-[1,3]thiazolo[2,3-b]pyrazine-7,8-dione 2-(3-tert-butyl-4-methoxyphenyl)oxane 6-bromo-5-chloro-1H-indazole 2-[4-(2,6-diphenylpyrimidin-4-yl)pyridin-1-ium-1-yl]acetic acid;hydroxide 2-[5,6-dichloro-3-oxo-7-(pyridin-2-ylmethoxy)-1H-isoindol-2-yl]acetic acid 4-(3,5-dimethoxyphenyl)-2-ethyl-1H-pyrimidin-6-one 2-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]pyridine-3-thiol [4-(aminomethyl)phenyl]-[2-butan-2-ylidene-3,7-di(propan-2-yl)octan-3-yl]azanium;bromide 4-[3-(6,7-dimethoxyquinolin-4-yl)propyl]-N-(2,5-dimethoxyphenyl)piperazine-1-carboxamide N-[(Z)-(4-hydroxyphenyl)methylideneamino]-5,7-dinitro-1H-indole-2-carboxamide 4-N-[4,5-diethoxy-2-(methylideneamino)phenyl]quinazoline-4,6-diamine 4-N-[(3E)-3,5-diaminohepta-1,3-dien-2-yl]benzene-1,4-disulfonamide (2R)-N'-hydroxy-2-[2-(methylamino)propanoylamino]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboximidamide 6-[(5S,7R)-3-methyl-4,8-dioxo-2-propyl-1,3,7-triazaspiro[4.4]nonan-7-yl]pyridine-3-carboxamide 3-[2,3-bis(ethenyl)-1H-indol-5-yl]pentanamide;(Z)-but-2-enedioic acid 5-methyl-6-(trifluoromethoxy)chromene-2,4-dione 5-(2,3-dihydronaphthalen-1-ylmethoxy)-N'-hydroxypyridine-2-carboximidamide 1-(2,5-dimethylphenyl)-3-[6-hydroxy-4-oxo-6-[(5-sulfamoylthiophen-2-yl)methylidene]cyclohexa-2,4-dien-1-ylidene]urea 2-(3-propan-2-yloxyphenyl)benzo[g][1,3]benzothiazole 1,3-diamino-1-[2-[(4-benzylpiperidin-1-yl)methyl]naphthalen-1-yl]urea 2-methoxy-4,8-dimethyldibenzofuran N-(2-aminoethyl)-4-methoxy-7,8-dihydronaphthalene-1-carboxamide 3-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylamino)propanamide N-[1-(4,4-difluorocyclohexyl)pyrrolidin-3-yl]-6-methoxypyridine-2-carboxamide 5-(4-chlorophenyl)sulfanylpentylazanium;(2R,3S,4S,6S)-2,4,6-trimethoxy-1,2,3,4-tetrahydronaphthalene-1-carboxylate N-[2-(3-chlorophenyl)ethyl]pyrido[4,3-d]pyrimidine-7-carboxamide 1-(2-methylheptan-4-yloxy)-6,7,8,9-tetrahydrobenzo[e]isoindole N-(3-amino-5,6,7,8-tetrahydronaphthalen-2-yl)-5-chloro-4-methoxy-2-[1-oxo-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]butan-2-yl]benzamide 2-(9H-fluoren-1-yl)hexanedioic acid 5-[4-(2,6-difluorophenyl)piperidine-1-carbonyl]thiophene-3-carbonitrile (3S)-1-cyclopropylsulfonyl-N-[2-hydroxy-5-(trifluoromethoxy)phenyl]piperidine-3-carboxamide 6-[4-(3,4,6,7,8,9-hexahydro-1H-pyrido[3,4-b]indole-2-carbonyl)phenyl]benzenesulfonamide 1-(3,4-dimethoxyphenyl)sulfonyl-2,3-dimethylazepane;hydrochloride N-(2-bromoethyl)-N-(4-chlorophenyl)butanamide 1-(azidooxymethyl)-3,5-dichlorobenzene 6-(4-methylphenyl)sulfinyl-3-nitropyridine-2,4-diamine (5E)-1,4a-dimethyl-5-[6-(6-morpholin-4-ylpyridine-2-carbonyl)pyrimidin-4-yl]-7-propanoyl-4,10b-dihydropyrazolo[3,4-b]quinolizin-9-one 2-[3,5-ditert-butyl-4-(2,4-dimethoxyphenyl)phenyl]ethanethiol 2-amino-5,6-difluoronaphthalene-1-sulfonic acid N-(4-ethylphenyl)-2,5-dimethoxybenzenesulfonamide 6-[2-(4,5-diethoxy-3-methoxycyclohexa-1,3-dien-1-yl)ethenyl]quinoxaline N-cycloheptylthieno[2,3-b]pyrazine-7-carboxamide 4-(2,3,6-triiodophenoxy)carbonylbenzoic acid N-[6-(3,5-dimethylpyrazol-1-yl)-2-[4-[[(2R)-2-(hydroxymethyl)morpholin-4-yl]methyl]phenyl]pyrimidin-4-yl]acetamide 6-[[6,7-dimethyl-4-oxo-3-(2-propan-2-yloxyphenyl)quinazolin-2-yl]amino]spiro[1H-indole-3,4'-piperidine]-2-one N-cyclobutylsulfanyl-4-[(3,4,5-trifluorophenyl)methoxy]aniline 5-(4-bromophenyl)-3,3a-dihydro-1H-pyrrolo[2,3-b]pyridine-2-thione 6-[2-amino-1-(4-tert-butylcyclohexyl)ethenyl]-3-hydroxy-4H-naphthalen-2-ide-1-carboxylic acid;rubidium(1+) 2-(3,4-dimethylphenyl)quinoline 2-[1-(dimethylamino)propan-2-yl]-3,5-difluoropyridine-4-carbonitrile 4-[(E)-2-azido-3,3-dimethylbut-1-enoxy]pyridine 2-[4-(difluoromethoxy)phenyl]-N-[3-(4-ethyl-6-oxo-1H-pyrimidin-2-yl)phenyl]cyclopropane-1-carboxamide (2S)-2-acetamido-3-[4-(4-chlorophenyl)phenyl]propanoic acid (3R)-4,6-dichloro-1'-(2,5-dimethylbenzoyl)spiro[2H-indole-3,2'-pyrrolidine]-5'-carboxamide 4-[2-(1H-benzimidazol-2-yl)ethoxy]-3,5-dimethoxyaniline;hydrochloride [(2S)-2-methoxycyclohexyl]-(7H-pyrrolo[3,4-b]pyridin-6-yl)methanone (3S,4R)-N-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-oxooxolane-3-carboxamide 2-cyclopropyloxy-4-(methylamino)benzoate (E)-N,5-dimethoxy-2-phenylpentanamide 2-(6-methoxynaphthalen-1-yl)-1,3-thiazole 5-[(2R,3S)-2,6-dimethylmorpholine-4-carbonyl]-2,3-dihydroinden-1-one 5-bromo-2,3,6,7-tetrahydroxynaphthalene-1,4-dione 1-(5-ethyl-2,4-dimethoxyphenyl)-3-[(3S,4R)-4-methoxyoxolan-3-yl]propan-1-ol 3-(3,5-dimethyl-1H-pyrazole-4-carbonyl)-7-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-one 4-amino-3,5,6-trichlorobenzenesulfonic acid N-[3-(3-azido-2,4,6-trifluorophenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]acetamide 2-(3,5-dimethylphenyl)-5-propan-2-ylpyrimidine 2-[(6,7-dichloroquinolin-4-yl)amino]-N,N'-dimethyl-3-phenylpropanehydrazide N-[1,2-dioxo-7-(phenylmethoxyamino)heptan-3-yl]acetamide;methane (2E,4Z)-5-[3-[6-(4,5-dihydrobenzo[e]azulen-9-yl)pyridin-2-yl]phenyl]penta-2,4-dienoic acid (E)-3-[4-(4-methylimidazol-1-yl)phenyl]prop-2-enal 7-(dimethylamino)-8-fluoro-3,4-dihydroquinoline-2-carboxylic acid (4-azido-2-methylsulfinylphenyl)methanamine 1-[6-(5-amino-2-chloropyrimidin-4-yl)sulfanylpyridin-3-yl]-3-(difluoromethoxy)pyrrolidin-3-ol N-[1-(2-methylpropyl)-3,4-dihydroisochromen-1-yl]-5-oxo-1,4-oxazepane-3-carboxamide 2-(3,5-dimethylphenyl)-1-[(4S)-6-hydroxy-4-[(4-iodopiperazin-1-yl)methyl]-8-methyl-3,4-dihydro-2H-quinolin-1-yl]ethanone 2-(2,6-dichlorophenyl)-5-[(E)-ethylideneamino]cyclopentane-1,3-dione 5-[(3S,4R)-1-[2-(3-methylphenyl)acetyl]-4-phenylpyrrolidin-3-yl]-3H-1,3,4-oxadiazol-2-one (Z)-N'-(1,3-dihydroisoindol-2-yl)oxy-3,3,3-trifluoro-2-[2-(methoxymethyl)pyridin-4-yl]prop-1-ene-1,5-diamine 3-amino-5-(2,3-dihydro-1H-inden-2-yloxy)-4-methanimidoylbenzonitrile (Z)-2-amino-4,4,6-trimethylhept-1-en-3-one;4-[[cyclobutylidene-[5-methoxy-7-(methylamino)pyrazolo[1,5-a]pyridin-3-yl]methyl]amino]benzonitrile 4-[2,5-dimethyl-3,4-bis(trifluoromethyl)pyrrol-1-ium-1-ylidene]-2-isocyano-6-(propanoylamino)pyridine-3-carbonitrile 1-(4-chloro-2,3,5,6-tetradeuteriophenyl)-3-diazourea 4-ethylpyridine;N,3,4-trimethyl-6-oxo-7H-thieno[2,3-b]pyridine-5-carboxamide N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-methoxy-6-methyl-N-phenyl-1,3,5-triazin-2-amine 2-methyl-N-[3-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl]benzamide N-[1-(1-methoxyethyl)cyclohexyl]-5,6,7,8-tetrahydroquinazolin-4-amine 6-methyl-1H-pyrrolo[3,2-f]quinoline;pyrrolidine N-[2,6-difluoro-3-(propylsulfinylamino)phenyl]-3-nitrobenzenesulfonamide 3-[(4Z)-2,4-dimethylhepta-2,4,6-trienoxy]-1H-indole 4-fluoro-3,5-dimethylbenzo[c]xanthene 3-chloro-5-[7-methoxy-2-(oxan-4-yl)pyrido[2,3-d]pyrimidin-6-yl]benzonitrile 1-[2-(dimethylamino)ethyl]-5,7-bis(trifluoromethoxy)benzo[g]indazole-3-carboxylic acid 3-(2,6-dichlorophenyl)-7-[4-methyl-5-[2-oxoethyl(3-pyrrolidin-1-ylpropyl)amino]pyridin-2-yl]-8H-[1,2,4]triazolo[4,3-b]pyridazine-6-carboxylic acid N-[2,4-dimethyl-6-(2-methylidenecyclopentyl)phenyl]pentanamide 3-[2,5-dichloro-N-(4-hydroxybutyl)anilino]phenol 2,6-difluoro-N-[1-(4-nitrophenyl)-3-pyrrolidin-1-ylpropan-2-yl]benzamide (2Z)-1-phenyl-3-phenylmethoxypenta-2,4-dien-1-one 3,5-dichloro-N-[[1-(4-fluorophenyl)cyclopropyl]methyl]pyridine-2-carboxamide N-(2,3-dihydro-1H-inden-5-ylsulfonyl)-2-phenyl-4-(trifluoromethoxy)benzamide 1-[4-(2,6-dimethylphenyl)pyridin-3-yl]-N,2,2-trimethylpropan-1-imine N-[[(5S)-3-[4-[(Z,2E)-1-chloro-2-ethylidenehex-3-enoxy]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]acetamide 1-methyl-4-(N-octylanilino)anthracene-9,10-dione N'-hydroxy-5,6-dimethyl-3-[methyl(1-pyridin-2-ylcyclobutyl)amino]pyridazine-4-carboximidamide 2-cyclopropyloxy-N,6-dimethyl-N-[(1S)-5-phenylpentyl]pyrimidine-4-carboxamide 3-[4-[(3,5-dimethylphenyl)carbamoylamino]anilino]benzoic acid [3-[5-[2,6-dimethyl-4-(3-morpholin-4-ylpropoxy)phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]urea 2-[3-(2-cyanopropan-2-yl)phenyl]propanenitrile 4-[[(4S)-2,5-dioxoimidazolidin-4-yl]methoxy]naphthalene-1-carbonitrile 1-[2-(4-chlorophenyl)ethyl]-3,6-dimethoxyisoquinoline 2-azido-N,6-dibenzyl-4-phenylpyridine-3-carboxamide 1-(5-chloro-2,4-dimethoxyphenyl)sulfanyl-3-[3-methoxy-4-(1,2-thiazol-3-ylsulfamoyl)phenoxy]thiourea 3-amino-4-chloro-5-(ethylaminomethyl)phenol;2,6-difluorobicyclo[3.1.0]hexane N-[2-bromo-4-(9H-fluoren-1-yl)phenyl]acetamide N-(2,3-dihydro-1H-inden-5-ylsulfamoyl)furan-2-carboxamide N-[1-(2,3-dihydro-1H-isoindol-5-yl)ethenyl]-7-[4-fluoro-2-(trifluoromethoxy)phenyl]-5-methyl-6,8-dihydropyrimido[4,5-d]pyrimidin-2-amine 1,4-dimethyl-2-(trifluoromethoxy)benzene;ethane 5-(4-chlorophenyl)-1,6-dimethylpyridine-2,4-dione;ethane 5-chloro-1-methyl-3-[2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)ethyl]-4H-diazepine N-(4-hydroxyphenyl)-2,4,6-trimethyl-N-prop-2-enylbenzenesulfonamide N-[[(2R,4S)-1-acetyl-2-benzylpiperidin-4-yl]methyl]-5-bromopyrimidine-4-carboxamide 3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl)phenol 2-[3-(4-methyl-1,2,5-oxadiazol-3-yl)-5-(trifluoromethyl)phenyl]acetic acid 1-(2,5-dimethoxyphenyl)-N-[6-(1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl]cyclopropane-1-carboxamide N-[1-(2,4-dimethylphenyl)-3-oxobutan-2-ylidene]piperidine-2-carboxamide (2R)-1-[3-(2,4-difluorophenyl)azetidin-1-yl]sulfonyl-N-methoxy-N'-methylpyrrolidine-2-carboximidamide N-[(4-chlorophenyl)methyl]-2,3-dimethyl-5-(4-oxo-3H-quinazolin-2-yl)-1H-pyrazole-4-carboxamide N-[(3S,5R)-1-acetyl-5-(hydroxymethyl)pyrrolidin-3-yl]-2-amino-6-[3-(trifluoromethoxy)phenyl]pyrimidine-4-carboxamide 2-N,7-dicyclohexylanthracene-1,9,10-triamine 4-[4-(4,6-diphenyl-1,3,5-triazin-2-yl)dibenzothiophen-1-yl]benzene-1,2-dicarbonitrile 5-azidooxy-6-nitronaphthalen-1-amine 1-ethyl-N-methoxyindole-2-carboxamide 6-[(2E)-3,7-dimethylocta-2,6-dienoxy]-4-hydroxy-1H-quinolin-2-one 6-[2-azidoethyl(pentanoyl)amino]naphthalene-1-sulfonic acid (2R)-1-[[6-chloro-5-[4-(2-fluorophenyl)piperazin-1-yl]pyridazin-3-yl]methyl]pyrrolidine-2,5-diol 3-(1H-pyrazol-4-yl)-8,9-dihydro-7H-benzo[h][2]benzazepine 4-N-[1-(2,3-dihydroindol-1-yl)butylidene]benzene-1,4-disulfonamide 1-[6,7-di(propan-2-yl)pyrido[2,3-d]pyrimidin-4-yl]-N-ethyl-3-methylpyrrolidine-3-carboxamide 1-(5-cyclopropyl-3,4-dimethoxyphenyl)octan-2-ol 2-[4-(1,1,2,2,3,3,4,4,5,5,6,6,7,8,9,9a-pentadecafluorononyl)phenoxy]-1H-indole 2-cyclopropyl-4-[(1,5-dimethylpyrazol-3-yl)amino]pyridazin-3-one 5-[(2-bromo-N-octylanilino)methyl]-1,3,4-oxadiazol-2-amine 4-cyclopropyl-3,6,10,13-tetrazatricyclo[7.4.0.02,6]trideca-1(9),2,4,10,12-pentaene 2-[[4-amino-5,6,7,8-tetrahydroquinazolin-2-yl]sulfanylmethyl-(3-chloropyridin-2-yl)amino]acetonitrile 3-(4-cyclopenta-1,4-dien-1-yl-1H-imidazo[4,5-c]pyridin-2-yl)-5-pyridin-3-yl-1H-pyrazolo[3,4-c]pyridine 1-[4-[[7-(aminomethyl)-3-ethylimidazo[5,1-b][1,3]thiazol-2-yl]methoxy]phenyl]ethanone 4-amino-3-[6-(2,5-dimethylphenoxy)-1H-benzimidazol-2-yl]pentanoic acid 2-[5-(3,4-difluorophenyl)sulfanyl-4-propan-2-ylimidazol-1-yl]acetic acid 4-(1H-imidazol-5-yl)-2,3-dihydro-1H-indene 2-chloro-5-iodo-3,4-dihydro-2H-chromene 2-(benzenesulfonyl)quinolin-8-ol 2-amino-1'-[(5S,6R)-3,4,5-trihydroxy-6-methyloxan-2-yl]spiro[indole-3,4'-piperidine]-2-one 2-[4-(2,6-difluorophenyl)-5-methylsulfanyl-1,3-thiazol-2-yl]-1,3-thiazole 5-azido-1,3-dibromoisoquinoline (5R)-5-[4-ethoxy-3-(methylsulfonylmethyl)phenyl]imidazolidine-2,4-dione 4-chloro-2,6-dihydroxybenzenesulfonamide 5-ethenyl-1-[2-(7-methoxyquinolin-4-yl)oxyethyl]pyrazole-3-carboxylic acid 4-amino-2,5-dimethylquinoline-8-carboxylic acid 2-(4,5-dihydro-1,3-thiazol-2-yl)benzenethiol;ethane 4-[2,3-dimethyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrol-4-ylidene]-N'-hydroxy-1-propanoylpiperazine-2-carboximidamide (3-chloro-5,7-dihydro-4H-thieno[2,3-c]pyridin-6-yl)-(1H-pyrrol-2-ylsulfonyl)methanone 2-(1H-indol-3-yl)quinazoline 1-(benzenesulfinyl)-3-[(Z)-2,4-dimethylhex-4-en-3-yl]benzene (3E)-5,5-dimethylhexa-1,3-diene;2-phenylquinoline 5-[[3-hydroxy-2,6-dioxo-4-(trifluoromethyl)pyrimidine-1-carbonyl]amino]pentanoic acid N-benzyl-2,4-dimethyl-5-(pyridin-3-ylmethoxy)aniline 4-(3,5-difluoro-2-methoxyphenyl)-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 1-[2-(4-chlorophenyl)-2,5-diethyl-3-oxomorpholine-4-carbonyl]piperidine-2-carboxylic acid (2S)-1-[(5R)-3,4-dihydro-2H-chromene-7-carbonyl]pyrrolidine-2-carboxamide 5-[5-chloro-2-(oxan-4-yloxy)phenyl]pyridine-3-carboxylic acid 1-[4-(2-ethylphenyl)piperidin-1-yl]-3-(methoxymethoxy)propan-2-amine 1-(3-fluoro-2,6-diiodophenyl)-N,N-dimethylmethanamine 1-[4,5-bis(ethenyl)pyridin-2-yl]-6-methoxyindole 3-(2,5-dioxopyrrol-1-yl)sulfonylpropanedioic acid 2-[(Z)-2-(3,5-dimethylphenyl)propylideneamino]oxyethanamine 5-[(2R)-2-acetylpyrrolidine-1-carbonyl]-4-methoxy-2H-isoquinolin-1-one 1-[1,3-bis(2-bromophenyl)propan-2-yl]pyrazolidin-3-one 5-azido-6,7-dimethoxy-1H-indazole 3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonyl)benzoic acid [4-(4-fluorophenoxy)phenyl]-[2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methanone [(5Z)-2,6-dimethylhepta-1,4,6-trienoxy]sulfonylbenzene 6-[4,5-bis(ethenyl)-1H-imidazol-2-yl]quinoline 2-fluoro-5-[4-methyl-3-[5-(trifluoromethyl)cyclohexa-1,3-dien-1-yl]pyrazole-1-carbonyl]benzonitrile 1-[5-cyclopropyl-2-(3,4,5-trifluorophenyl)pyrimidin-4-yl]azetidine-3-carbonitrile N'-[[4-amino-1-(2,3-dihydroindol-1-yl)cyclohexa-2,4-dien-1-yl]methyl]oxamide (5Z)-5-[[3,4-dichloro-2-hydroxy-6-(trifluoromethyl)phenyl]methylidene]imidazolidine-2,4-dione 6-methylsulfanyl-4,5,7-triphenylisoquinoline 4-(5,6-dihydro-1H-indazole-3-carbonyl)-N-[2-hydroxy-4-methyl-5-(trifluoromethoxy)phenyl]piperazine-1-carboxamide 1-(2,5-difluorophenyl)-4,7,8,9-tetrahydropyrazolo[3,4-f]quinoline 2-azido-7-ethyl-5-[4-(2,2,2-trifluoroethoxy)phenyl]imidazo[1,2-a]pyridine 2-(2,3,4-trifluorophenyl)benzene-1,3-diamine 2-cyclopentyl-1',5,6-trimethoxyspiro[isoindole-3,4'-piperidine]-1-one 2-ethylsulfanyl-N,3-dimethylaniline 4-(3,5-difluoroanilino)-N'-methylpiperidine-1-carboximidamide;ethane N-[(3Z)-5-chloro-2,6-dimethylhepta-1,3,5-trien-4-yl]-2-cyanobenzamide (5Z)-5-[(2,3-dimethoxyphenyl)methylidene]-2-(4-fluorophenyl)imino-1,3-thiazolidin-4-one N-benzyl-3,4-dimethoxy-5-[(Z)-3-oxoprop-1-enyl]thiophene-2-carboxamide 3-ethylsulfanyl-6,8-dimethylquinazolin-4-one 2-[[4,5-bis(ethenyl)triazol-1-yl]methyl]benzoic acid N-cyclobutyl-2,5-dimethoxy-4-(3,4,5-trifluorophenyl)aniline 4-[(2R,3S)-5-[(4-chlorophenyl)methyl]-2-ethyl-2-[5-fluoro-6-(morpholine-4-carbonylamino)pyridin-3-yl]-1,3-dihydropyrrol-4-yl]benzoic acid 5-[3,4-dimethyl-2-[(1S)-3-oxocyclopenten-1-yl]phenyl]-7-fluorospiro[2H-indole-3,1'-cyclohexane]-1,2'-dione 2-[8-[4-chloro-3-(5-methyltetrazol-1-yl)benzoyl]-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]acetic acid 4-[(3,5-diethoxy-2H-1,3-benzoxazol-2-yl)methyl]phenol N-[(1S)-1-(4-chlorophenyl)-2-oxopiperidin-3-yl]pyridine-2-carboxamide 4-(benzenesulfonyl)-N-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-amine 4-[(2S)-2-acetamido-3-[4-(cyclopropylmethoxy)phenyl]sulfonylazetidine-1-carbonyl]piperazine-1-carboxylic acid 2-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-3-ylsulfanyl)-N'-hydroxypyridine-4-carboximidamide 1-[2-amino-6-(azepane-1-carboximidoyl)phenyl]ethanone (1S)-N'-[4-fluoro-5-[2-(methylamino)pyrimidin-5-yl]indazol-1-yl]cyclopropanecarbonyl-2,2-dimethylcyclobutane-1-carbohydrazide (2R)-2,3-dihydroimidazo[1,2-c]quinazoline-5-carboxamide 3-(dimethylamino)-1H-indole-5-carbonitrile (2S)-3-[[5-chloro-6-(1,1,1,2,3,3,3-heptafluoropropan-2-ylamino)pyridazin-4-yl]methyl]-2-[3-(cyclopentylmethoxy)-4-(difluoromethoxy)phenyl]-N'-hydroxy-2H-imidazole-1-carboximidamide 2-(3,4-dimethoxyphenyl)-5H-[1]benzothiolo[3,2-c]pyridazine 5-cyclopropyl-3,4-dihydro-1H-isochromene-7-carbonitrile 6-chloro-2-[4-fluoro-2-(trifluoromethyl)phenyl]pyrimidine-4-carboxylic acid N-[2,6-bis(phenylsulfanyl)pyridin-3-yl]-1-phenylmethanesulfonamide 7-[(1S)-2,3-dihydro-1H-inden-1-yl]quinoline 5-(azidomethyl)-7,8-dihydronaphthalene 2-(4-anilino-N-tert-butylanilino)acetonitrile 2-(1,4-dioxaspiro[4.5]decan-3-yl)-6-methoxypyridine;ethane 1-[4-(3,3a,5,6a-tetrahydrofuro[3,2-b]furan-3-carbonyl)phenyl]ethanone (4S)-4-(3,5-difluorophenyl)-2-hydroxy-1-[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]pentan-3-one (2R)-1-benzyl-3-(3,4-dihydroxyphenyl)pyrrolidine-2-carboxamide 7-[(Z)-3-amino-2,5,5,5,6,8,8-heptamethylnon-6-enoxy]-N-phenylquinoline-4-carboxamide 2-[3,6-difluoro-8-[3-methylbutoxy(sulfanyl)amino]naphthalen-1-yl]sulfanylethanol 2-[4-[6-[2-(difluoromethyl)benzimidazol-1-yl]-2-morpholin-4-ylpyrimidin-4-yl]piperazin-1-yl]ethanol 1-[4-(2-ethyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl)-2-methoxyphenyl]pyrrolidin-2-one 2-chloro-4,8-dimethylpyrazolo[1,5-a]quinazoline 2-[4-(cyclohexylcarbamoylamino)piperidine-1-carbonyl]benzamide 5-[2,3-difluoro-4-(trifluoromethyl)phenyl]-2H-tetrazole (E)-3-[4-[2-acetyl-5-(trifluoromethoxy)indole-1-carbonyl]oxycyclohexa-1,3-dien-1-yl]prop-2-enoic acid N-[(1S,5R)-3-[6-cyclopropyl-4-[2-[methyl(pyridin-2-ylmethyl)amino]ethoxy]pyridin-2-yl]oxy-6-bicyclo[3.1.0]hexanyl]benzamide 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-tetradecylaniline N-(2-bromophenyl)-4-(1H-pyrrole-3-carbonylamino)-1,2-oxazole-3-carboxamide (3R)-1-[4-chloro-6-(methylamino)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid N-benzyl-6-[2-(4,5-dimethylimidazol-1-yl)pyridine-4-carboximidoyl]pyrimidin-4-amine (2S)-2-amino-3-methylbutanoate;N,N-diethyl-6-[4-[6-(propylamino)pyrimidin-4-yl]piperazin-1-yl]pyrimidin-4-amine 7-methyl-4,6-dihydro-2H-triazolo[1,5-a][1]benzazepin-5-one (2S)-2-amino-3-[4-[1-cyclopropyl-1-[5-(trifluoromethoxy)pyridin-2-yl]ethoxy]phenyl]propanoic acid 6-chloro-2-methyl-4-[3-(trifluoromethoxy)phenyl]sulfonylpiperazine-1-carboxamide 6-azido-2-(chloromethyl)phthalazin-1-one 1-[3-amino-6-(1H-pyrazol-4-yl)pyrazin-2-yl]ethanethiol (1R)-N,2-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]cyclobutane-1-carboxamide 1-ethyl-N-(4-fluorophenyl)sulfonyl-3,7-dimethylpyrazolo[3,4-c]pyridine-5-carboxamide 5-tert-butyl-3,4-diethoxy-N-[2-(1H-1,2,4-triazol-5-yl)phenyl]thiophene-2-carboxamide 4-methyl-2-[4-[6-(trifluoromethoxy)quinolin-7-yl]oxybutyl]pyrrolidine-1-carboxylic acid N-[1-(2,4-dichlorophenyl)cyclopropyl]-3-methoxyspiro[1,4,5,6-tetrahydropyrrolo[3,2-c]pyridine-7,1'-cyclopentane]-2-carboxamide N-[(5-chlorothiophene-2-carbonyl)amino]carbamate 3-chloro-N-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]-5-[2-[2-hydroxyethyl(methyl)amino]ethoxy]benzamide 3-(2,6-dichlorophenyl)-7-[(4,4-dimethylpiperazin-1-yl)amino]pyrimido[5,4-e][1,3]oxazin-4-one;2,2,2-trifluoroacetic acid [(Z)-4-hydroxyhexylideneamino]sulfonyloxymethylsulfanylbenzene N-[2,4-dihydroxy-3-(5-methylcyclohexa-1,3-dien-1-yl)butan-2-yl]-4-methoxybenzamide 4-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidine-1-sulfonamide N-[(3R)-1,1-dioxothiolan-3-yl]-2-[4-methoxy-3-(2-phenylethynyl)anilino]acetamide 3-(7-chloro-2,4,5-trioxo-1H-3-benzazepin-3-yl)propanenitrile 6-[3-(methoxymethyl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidine-2-carboxylic acid 5-fluoro-2-[(Z)-hydroxyiminomethyl]phenol N-[4-chloro-2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carbonyl)phenyl]-5-fluoroquinoline-8-sulfonamide N-[(2E,4E)-5-(6-methylidenecyclohexa-1,3-dien-1-yl)sulfanylpenta-2,4-dienoyl]-2-phenylacetamide 6-[4-chloro-2-(trifluoromethoxy)phenyl]-1,3-diazinane-2,4-dione 1-[1-(3,4-difluorophenyl)ethyl]-5-methylcyclohexa-2,4-dien-1-ol 3-[2-ethoxy-5-(4-methylpiperazin-1-yl)sulfonylphenyl]-7-ethyl-6-(2-hydroxy-5-nitrosophenyl)-1H-thieno[3,2-d]pyrimidine-2,4-dione 2-(4-methylphenyl)sulfanyl-5H-pyrido[1,2-a]benzimidazol-6-one 2-(2,6-dioxopiperidin-3-yl)-4-[[1-[[(1R,2S)-2-hydroxycyclopentyl]methoxy]isoquinolin-7-yl]methylamino]isoindole-1,3-dione 3-[(2,5-dimethylpyrazole-3-carbonyl)amino]-N-propan-2-ylpiperidine-1-carboxamide 4-methoxy-N-[(3S)-oxolan-3-yl]-2-[4-(trifluoromethyl)phenyl]benzamide (1Z,3Z)-5-methylsulfanyl-4-[2-(trifluoromethyl)phenyl]hexa-1,3,5-trien-1-amine 3-(2,4-dichlorophenyl)-6,7-dimethylisoquinoline 5-bromo-4-(2,3-dihydrothiophen-2-ylmethylamino)-1H-pyrimidin-6-one 2-[4-(3-chlorophenyl)piperazine-1-carbonyl]chromen-4-one (E)-N'-ethenyl-2-methylidenebut-3-enehydrazide;1-[(6Z,8Z)-6-prop-2-enylidenedeca-6,8,10-trienyl]naphthalene 4-amino-6-[1-(4-methylphenyl)pyrazole-3-carbonyl]pyran-2,5-dione N-[(3S)-6-cyano-7-methyl-1,2,3,4-tetrahydrocarbazol-9-yl]benzamide N-[5-[1'-(2,4-dimethylpyrimidine-6-carbonyl)spiro[3H-1-benzofuran-2,4'-piperidine]-4-yl]pyridin-3-yl]acetamide 5-[3,4-dihydroxy-2,6-bis(prop-2-enoyloxy)phenyl]-1H-pyrrole-2,3,4-tricarboxylic acid 2-[(E)-[3,5-dimethoxy-4-[6-(trifluoromethyl)pyridin-3-yl]phenyl]methylideneamino]guanidine N-[5-(hydroxymethyl)-1,3,4-thiadiazol-2-yl]-5-oxo-7,8-dihydro-6H-[1,2,4]triazolo[1,5-a]pyridine-2-carboxamide 1-[(3R)-3-(2,5-difluorophenyl)pyrazolidin-4-yl]ethanone 7-chloro-1,2,3,4-tetrahydroquinoxaline-5,6-dione (2S)-2-[[4-methoxycarbonyl-1,3-bis(phenylmethoxy)naphthalene-2-carbonyl]amino]propanoic acid N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-1,6-dihydropyridazine-3-carboxamide 1-cyclobutyloxy-4-[(Z)-4,5,5-trifluoro-2-iodopent-3-enyl]benzene (Z)-3-[6,7-dihydroxy-2-methyl-5,8-bis(3-phenylpropoxy)-3,4-dihydrochromen-4-yl]but-2-enal;N,N'-dimethylethane-1,2-diamine [(2R)-3-azidopropyl]sulfanylbenzene [4-methyl-1-(4-propan-2-ylphenyl)pentyl]sulfanium N-[5-(4-chlorophenyl)-3-methylpyrazol-1-yl]sulfanyl-4,6-difluoro-1H-indole-2-carboxamide 2-[[2-(4,5-dimethylthiophene-3-carbonyl)-6-hydroxy-1-benzofuran-3-yl]oxy]acetic acid 3-[3-fluoro-4-(1,2,3,6-tetrahydropyridin-5-ylmethoxy)phenyl]pentanoic acid N-(2,5-dimethylphenyl)sulfanyl-5-fluoro-6-iodopyrimidin-4-amine N-(2,6-dichloropyridin-3-yl)-2,4,5-trifluoro-3-methoxybenzenesulfonamide 5-[3-ethoxycarbonyl-6-(trifluoromethyl)quinolin-4-yl]oxy-2-methylbenzoic acid 6-chloro-4-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[(3-fluorophenyl)methyl]cyclohexa-1,5-diene-1-carboxamide N-benzyl-4-[(3S,4R)-4-methoxyoxolan-3-yl]piperazine-1-carboxamide 4-[(3S,5R)-1-[(4-methylthiophen-2-yl)methyl]-5-pyridin-4-ylpyrrolidin-3-yl]-2-pyrrolidin-1-yl-1H-pyrimidin-6-one 2-[4-(1,2-dihydroxypropan-2-yl)-5-fluoropyrimidin-2-yl]benzamide 7-(6,7-dimethoxyquinazolin-4-yl)oxynaphthalene-2-carboxylic acid 2-(3,5-dimethoxyphenyl)-N,4-dimethylpentanamide N-[3-(1H-indole-2-carbonyl)-4-[1-(2,2,2-trifluoroacetyl)piperidin-4-yl]oxyphenyl]cyclopropanesulfonamide 4-[3,5-dimethoxy-2-(4-piperazin-1-ylphenyl)cyclohexa-2,5-dien-1-ylidene]-7H-pyrrolo[2,3-d]pyrimidine 1-(4,5-diphenyl-3,4a-dihydrocyclopenta[b]pyrrole-2-carbonyl)pyrrolidine-2-carboxamide (2R)-2-[2-[4-[3-chloro-4-(trifluoromethoxy)phenyl]piperazine-1-carbonyl]-5,6-dihydroimidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-1-carboxylic acid 2-methyl-6-(5-pyridin-4-ylfuran-3-carbonyl)-7,8-dihydro-5H-[1,3]oxazolo[4,5-g]chromen-9-one 4-(2,6-difluorophenyl)-N-[4-[[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]methoxy]butanoyl]-2-methoxybenzamide 4-(2-aminophenyl)sulfanyl-N,N-dimethylaniline (2S)-6-amino-7-[4-(dimethylaminosulfanyloxy)phenyl]-1,4-dimethyl-2-propyl-3H-quinoxaline-2-carboxylate 6-[(3R)-1-[[5-cyclopropyl-2-fluoro-4-(1H-indol-4-yloxy)phenyl]methyl]pyrrolidin-3-yl]oxy-2,3-dihydrofuro[3,2-c]pyridine 2-[2,6-bis(chloromethoxy)phenyl]naphthalene 6,7-dimethoxy-N-(4-phenylphenyl)-1H-indole-3-carboxamide 3-[(4S,5R)-2-amino-4-hydroxy-1-methyl-6-oxo-5-phenyl-3,4,7,8-tetrahydropyrimido[4,5-d]pyrimidin-4-yl]benzoic acid 4-N-[5-(trifluoromethyl)pyridin-2-yl]-6-N-[3,3,3-trifluoro-2-(methanesulfonamido)propoxy]quinazoline-4,6-diamine 2-[1-(4-methylphenyl)sulfonylindol-3-yl]-N-pyrrolidin-1-ylacetamide 2-[(E)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]oxy-N-phenylacetamide [(3R)-1-azabicyclo[2.2.0]hexan-3-yl]-[4-[(2S)-4,4-difluoro-6-methylmorpholine-2-carbonyl]piperazin-1-yl]methanone;hydrochloride (5R)-3-benzyl-2,4,6-trichloro-7-methoxy-9H-fluoren-1-amine N-benzyl-3-methoxy-4-[(E)-2-methylbut-1-enyl]aniline 2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-5-[(Z)-indazol-3-ylidenemethyl]-1,3-thiazol-4-ol 2-[1,3-dihydroxy-4-(1H-pyrazole-5-carbonyl)piperazin-2-yl]-N'-methylethanimidamide 6-[(3,4-difluorophenyl)methyl]-2-(4-fluorophenyl)-7H-purine N-(2,4-difluorophenyl)-4-[4-(3-phenylbutanoylamino)phenyl]thiadiazole-5-carboxamide [4-(2,6-dimethoxyphenyl)sulfanylpiperidin-1-yl]-imidazo[1,2-a]pyridin-3-ylmethanone 3-bromo-N-(2,5-dichlorophenyl)-1-benzothiophen-6-amine N-(4,6-dimethylpyrimidin-2-yl)-4-[(Z)-N'-hydroxycarbamimidoyl]benzamide N-[3-(2,6-difluorophenyl)cyclobutyl]ethanesulfonamide [(3S)-3-[5-[4-[5-[[4,4-bis(methoxycarbonylsulfanyl)cyclohexen-1-yl]amino]pyrimidin-2-yl]phenyl]pyridin-2-yl]oxypyrrolidin-1-yl]-morpholin-4-ylmethanesulfinate 2-(4-fluorophenyl)imino-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 2-[3,5-bis(trifluoromethyl)phenyl]-N-(4-methoxy-6-phenylpyrimidin-2-yl)acetamide 5-[2-(azetidin-1-yl)ethylamino]-N-[3-chloro-4-fluoro-7-[1,3-oxazol-2-yl(dideuterio)methoxy]phenyl]quinazoline-8-carboxamide;trihydrochloride 1,3-bis(trifluoromethyl)benzene-2-sulfinic acid N-[4-(1-methoxyethenyl)phenyl]-2-morpholin-4-ylpyrimidine-5-carboxamide N-[3-(diethylamino)propyl]-2-[1',4'-dioxospiro[1,2-dihydroindene]-5-yl]acetamide 2-[[1-[(3,4-dichlorophenyl)methyl]piperidin-4-ylidene]amino]ethanol 1-methylsulfanyloxy-6H-benzo[c]chromene 1-methoxy-2,3-dipentylnaphthalene N-(3,3-difluorocyclobutyl)-2-(5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carbonylamino)pyridine-4-carboxamide 5-[2-[4-(3,3-difluorobutyl)phenyl]ethynyl]-1,2-difluoro-3-isothiocyanatobenzene 4-chloro-2,3-dihydro-1H-indene;(E)-3-[[4-(chloromethyl)phenyl]disulfanyl]prop-2-enal 5-[(2R)-3-(3,4-dihydro-1H-isoquinolin-2-yl)-2-hydroxypropoxy]-2,4,7,8-tetramethyl-3,4-dihydrochromen-6-ol 2-[4-(3-methoxycyclobutyl)piperidine-1-carbonyl]-N,N-dipropylbenzamide N-(1,3-benzothiazol-2-yl)-2-[2-[(3R)-piperidin-3-yl]-4-propanoyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-6-yl]acetamide (2S)-1,5-dimethyl-N-(4-pyrazin-2-ylbutan-2-yl)piperidine-2-carboxamide 2-fluoro-6-[[[4-(trifluoromethyl)cyclohexyl]amino]methyl]naphthalene-1,4-dione 2-[4-(4,5,6,7-tetrahydroindazole-1-carbonyl)piperidin-1-yl]quinoline-3-carboxamide N-[(5-fluoropyridin-3-yl)methyl]-1-(4-methylsulfonylphenyl)cyclopropan-1-amine 3,4-bis(2-methoxyethyl)aniline 3-(2,4-difluorophenyl)-1-[6-(furan-2-ylmethylamino)pyrimidin-4-yl]piperidine-3-carboxylic acid 2-[(5R)-6-azidohexyl]-4-methoxypyridine (E)-3-[5-[[2,6-dichloro-4-[3-(4-methyl-1H-pyrazol-5-yl)propoxy]phenyl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]-2-ethoxycarbonylcyclopent-2-ene-1-carboxylic acid 1-(2,6-dimethylmorpholin-4-yl)-2-(5H-imidazo[5,1-a]isoindol-5-ium-10-yl)ethanone;bromide 3-[2-methylpropanoyl(pyridin-4-yl)amino]butanoic acid 3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]-1,4,4a,9a-tetrahydrocyclohepta[b]pyridine 4-(2-azidoethyl)-1,6-dichloroacridine 4-hydroxy-N-(3-methylcyclohexa-1,5-dien-1-yl)-1H-benzimidazole-2-carboxamide 4-tert-butyl-2,6-dipyridin-3-ylpyrimidine N-[3-[(2Z)-2-(1H-benzimidazol-5-ylmethylidenehydrazinylidene)-4-oxo-1,3-thiazolidin-5-yl]phenyl]acetamide N-[4-(3,5-dichloropyridin-2-yl)phenyl]thiohydroxylamine 2-[(3,4-dimethylphenyl)methylamino]pyridine-4-carboxylic acid 4-[2,2-bis(benzylsulfanyl)ethoxy]-N-(3-chloro-2H-indazol-5-yl)-6-methylpyrimidin-2-amine 2-ethoxy-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one 2,5-dimethyl-4-(3-phenylpyrrolidine-1-carbonyl)benzoic acid 3-[2,6-dibromo-4-(1,1,1-trifluoropropan-2-yloxy)phenyl]-N,5-dimethylpyridine-2-carboxamide N-cyclobutyl-4,5-dihydroxynaphthalene-2-sulfonamide N-(2,5-dimethoxyphenyl)sulfonyl-1-[3-fluoro-4-methyl-5-(trifluoromethyl)phenyl]imidazole-4-carboxamide N-[3-[(1Z)-buta-1,3-dienyl]imino-2H-pyrrol-5-yl]-4-fluorobenzamide;ethane 2-(3,5-difluorophenyl)acetaldehyde;N'-[4-[6-methoxy-7-[3-methyl-4-[[(Z)-prop-1-enyl]amino]butoxy]quinolin-4-yl]oxy-3-methylphenyl]-N-(4-phenoxyphenyl)oxamide 2-benzyl-3-methoxyacridine 3-azido-2,4,5-trimethoxybenzaldehyde 1-azidooxy-4-(2-methylphenyl)benzene N-(2,4-dichlorophenyl)-4-methylthiadiazole-5-carboxamide N-[(1R)-1,2-diphenylethyl]aniline;ethane N-[6,7-diamino-1-(4-cyanophenyl)heptyl]-1,3-benzothiazole-2-carboxamide 7-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)heptanoic acid 1-[4-(3,4-dimethoxyphenyl)-1,3-thiazol-2-yl]pyrrolidin-3-amine;ethane 4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]benzoic acid 6-(4,5-diphenylfuran-2-carbonyl)oxyhexanoic acid (3-phenylcyclohexyl)methylidenehydrazine N-[2-chloro-5-(trifluoromethyl)phenyl]cyclopropanecarboxamide 6-methoxy-2,3,3a,4,5,9b-hexahydrofuro[3,2-c]quinoline-8-carboxamide 4-chloro-N-(2-methyl-1,3-benzoxazol-5-yl)-6-pyrrolidin-1-ylpyrimidine-5-carboxamide;(4S)-4-ethoxyheptane 2-methyl-4-[(3R)-4-[1-[6-(trifluoromethoxy)pyridin-3-yl]ethyl]morpholin-3-yl]-1H-pyrimidin-6-one 1-(azidomethoxy)-4-chloro-2-phenylsulfanylbenzene 3-cyclopropyl-2,4,6-trimethoxybenzoic acid N-[2-amino-4-(N'-propan-2-ylcarbamimidoyl)phenyl]-2,5-difluorobenzamide;methoxyethane N-[[2,6-bis(difluoromethyl)pyridin-3-yl]methyl]-5-methoxypyridine-2-carboxamide 3-[2,4-dihydroxy-6-(4-methylphenyl)phenyl]-N-propan-2-ylcyclohexane-1-carboxamide 2-methyl-5-[4-(3-phenylpropanoyl)piperidine-1-carbonyl]benzamide 2-[1-(cyclopropylmethylamino)ethenyl]-6,8-difluoroquinoline-3-carboxylic acid 2-[1-[(4-aminobenzoyl)amino]ethylsulfanylmethylidene]hexanoic acid 5-bromo-4-[(2,3-dichlorocyclohexa-1,5-dien-1-yl)methoxy]pyrimidine 5-[(E)-3-[4-(dimethylamino)phenyl]prop-2-enoyl]-1,3-thiazolidine-2,4-dione 4-chloro-N-(2-chlorophenyl)-6,7-dihydro-5H-cyclopenta[d]pyrimidine-7-carboxamide 1-(2,5-dichlorophenyl)ethane-1,2-dione 4-[(3S)-1,2,3,5,6,7-hexahydro-s-indacen-4-yl]-1H-pyridine;4-phenylbenzenesulfonic acid 2-(3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl)-7-[4-(trifluoromethoxy)phenyl]sulfonyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 1-(4,6-dimethylpyrimidin-2-yl)-3-[5-[hydroxy(quinolin-6-ylsulfonyl)amino]pentyl]urea 2-[5-fluoro-6-(2,4,6-trichloroanilino)pyridin-3-yl]acetate 3-(7,8-dihydrothieno[2,3-e]indol-2-yl)-N-methylpropan-1-amine 2-[(3S,4R)-1-azido-4-chloropyrrolidin-3-yl]oxypyridine 4-[2,4-bis(trifluoromethyl)phenyl]pyrimidine 3-[4-(1H-indole-5-carbonyl)-2-oxopiperazin-1-yl]-N,N-dimethylbenzamide 1-[4-amino-3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-3-benzylthiourea N-[2,6-di(propan-2-yl)phenyl]-1-[5-(9H-fluoren-4-yl)-1H-imidazol-2-yl]methanimine 4-(1,3-benzodioxol-5-yl)-3-[3-chloro-2-[1-(hydroxymethyl)cyclopropyl]-1H-indol-6-yl]butanenitrile ethane;(4E,5Z)-4-ethylidene-3-methyl-1-phenylhepta-1,5-dien-3-ol 4-(2,6-dimethylpyridine-3-carbonyl)-N'-[4-ethyl-3-(trifluoromethyl)phenyl]piperazine-1-carboximidamide;5-(hydroxymethyl)pyrimidine N-[3,5-dimethyl-4-(3-morpholin-4-ylpropoxy)phenyl]pyrimidine-2-carboxamide 2-[4-amino-6-(2-methoxyethylcarbamoyl)pyrimidine-5-carbonyl]oxyacetic acid N-[(2,6-dimethoxyphenyl)methyl]-3-(2-imino-4-oxoquinazolin-1-yl)propanamide (E)-N,3-diamino-3-[4-[2-[3-chloro-5-fluoro-6-(1,1,1-trifluoropropan-2-yloxy)pyridin-2-yl]ethynyl]phenoxy]but-2-enamide 2-[4-(2-azidoethynyl)phenoxy]oxane 1-(2,4-dihydroxyphenyl)octadecan-1-one 3,5-dimethoxy-4-[4-(4-methylpiperazin-1-yl)-3-nitrophenyl]phenol 1-[(3S)-3-ethoxypyrrolidin-1-yl]sulfonylpyrazole 2-[4-(dimethylamino)phenyl]-1-[3,5-di(propan-2-yl)cyclohexa-1,5-dien-1-yl]guanidine 4-(4-methylphenyl)piperazine-1,2-dicarboxylic acid 4-[(2S,3aS)-5-[1-[4-cyano-3-(trifluoromethyl)phenyl]piperidin-4-yl]-10-ethoxy-1,2,3,3a,4,5,6-octahydrobenzo[f]quinoline-2-carbonyl]benzoic acid 4-tert-butyl-N-cyclopropyl-2,6-bis[(2,3,5,6-tetrafluorophenyl)sulfanyl]aniline 5-[[4-(2,3-dihydroindole-1-carbonyl)phenyl]sulfonylamino]-N'-hydroxypyridine-2-carboximidamide (NZ)-N-[1-[4-(3,5-dimethylpyrazol-1-yl)pyridin-2-yl]ethylidene]hydroxylamine (E)-3-(6-chloro-1,2,3,4-tetrahydroacridin-9-yl)prop-2-enamide 5-[1,2-dihydroxyethyl(hexyl)amino]-3H-1,3,4-thiadiazole-2-thione 2-[(3aR,6aR)-5-cyclopentylsulfonyl-3a-(5-methyl-1H-1,2,4-triazol-3-yl)-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrole-2-carbonyl]benzonitrile 2-(1,3-benzodioxol-5-yloxy)-1-(7-chloro-4-phenylquinolin-6-yl)ethanone (E)-N-[4-(3-bromophenyl)-1,3-thiazol-2-yl]-2-[(Z)-(4-fluorocyclohexyl)methylideneamino]-3-hydroxyprop-2-enamide 3-[4-(2,5-dimethylpyrrol-1-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 2-[4-(benzylamino)phenyl]-2-iminoacetic acid (4-chlorophenyl)-diphenylphosphane 4-[(2,6-dimethylmorpholin-4-yl)methyl]benzoic acid ethane;6-[3-(4-methylphenyl)sulfonylpyrrolidin-1-yl]-4,5-dihydropyrimidine N-(2-chloroacetyl)-4,6-dimethylpyrimidine-5-carboxamide 2-[4-(3,4-dihydroisoquinolin-7-yl)phenoxy]-2-methylpropanoic acid 4-[(8,9-dimethoxy-2,3-dihydro-[1,4]oxazino[2,3-c]quinolin-5-yl)methyl]phenol 5-bromo-N-[(3R)-1-cyclopentylpyrrolidin-3-yl]pyrrolo[2,1-f][1,2,4]triazin-4-amine 3-[(3S,4R)-1-tert-butyl-4-hydroxypyrrolidin-3-yl]-N-phenylpropanamide 3-bromo-4,5-diethoxybenzoic acid 4-[4-(1-aminoethenyl)phenyl]-5-methylidene-3,4-dihydropyridazine-6,7-diamine;ethane 2-(3,5-dimethoxyanilino)-4-fluoropyridine-3-carboxylic acid 4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-iodopyrimidine 4-[(Z)-(4,6-dihydroxy-3-methoxy-2-oxochromen-8-yl)methylideneamino]benzenesulfonic acid [2-chloro-5,7-dimethyl-3-(trifluoromethyl)imidazo[4,5-b]pyridin-6-yl]-phenylmethanol 1-[2,3-bis(ethenyl)cycloprop-2-en-1-ylidene]-N',2,5,6-tetramethyl-N-naphthalen-2-ylindole-4-carboximidamide (2-aminoethylamino)-(4-bromophenyl)methanol 2,4-difluoro-N-[6-(1H-imidazole-5-carbonylamino)pyridin-3-yl]benzamide 1-[5-bromo-4-(3,5-dimethylanilino)pyrimidin-2-yl]pyrazole-4-carboxamide 2-[2-ethyl-4,5-di(propan-2-yl)pyrazol-3-yl]-6-propan-2-ylpyridine 5-[6-(2,4-difluorophenoxy)pyridin-3-yl]-N-(1-hydroxyethyl)-4-methoxy-2-nitrobenzamide 1-[2-(dimethylamino)ethyl]-3-propyl-8,9,10,11-tetrahydrocycloocta[b][1,5]benzothiazepin-6-one 3-[(E)-1,2-diaminoprop-1-enyl]-N-phenylazetidine-1-carboxamide 3-(cyclopropylmethoxy)-N-[2-(difluoromethoxy)ethyl]benzamide 2-ethoxy-8-methylquinoline 2,3-bis(2-bromopyridin-4-yl)propane-1,1-diol 1-methoxy-4-propan-2-yloxyphthalazine 3-amino-2-[4-(diethylamino)piperidine-1-carbonyl]-N'-hydroxypyridine-4-carboximidamide;2,2,2-trifluoroacetic acid 2-azido-5-tert-butylbenzenesulfonic acid 1-[(1R)-5-chloro-2,3-dihydro-1H-inden-1-yl]pyrrole 2-amino-4-[5-bromo-2-(trifluoromethoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile (E)-N,3,4,4-tetramethyl-5-[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazol-4-yl]hex-2-en-1-imine 4-[4-(4-hydroxy-3-methylphenoxy)piperidine-1-carbonyl]oxane-4-carboxamide [3-(4-carbamoylphenyl)sulfinylthiophene-2-carbonyl]-[4-[2-cyclopropylethyl(methoxy)amino]phenyl]azanium N-[4-(trifluoromethyl)pyridin-2-yl]spiro[2.5]octane-6-carboxamide [1-azidooxy-3,5-bis(2-chlorophenyl)pentan-3-yl]benzene 4-cyclopropyl-5-iodo-1H-pyrimidine-2,4-diamine (E)-N'-[4-(aminomethyl)cyclohexa-1,5-dien-1-yl]-3-(3-ethoxyphenyl)prop-2-enimidamide 3-[6-amino-2,4-dioxo-1-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]propanamide 3-[2-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]azetidine 1-(6,7-dimethoxyquinolin-4-yl)-3-[3-(trifluoromethyl)pyridin-2-yl]urea 6-tert-butyl-4-(1-methylpyrazol-3-yl)-2H-pyrazolo[3,4-c]pyrazol-3-amine 2-cyclohexa-1,3-dien-5-yn-1-yl-4-(trifluoromethyl)benzonitrile 2-[1,3-benzodioxol-5-yl(hydroxy)methylidene]cyclohexan-1-one [3-[1,4-bis(2-methylpropyl)cyclohexa-2,4-dien-1-yl]sulfonyl-5-methoxyphenyl]-pyridin-2-ylmethanone 2-[[3-methylbutoxy(phenyl)phosphoryl]amino]ethanol 1,4-bis[3-(trifluoromethyl)phenoxy]butan-2-one N-[2,6-difluoro-4-(1H-pyrazol-5-yl)phenyl]-3-[(3S)-oxolan-3-yl]oxyazetidine-1-carboxamide (4E)-2,2-dimethyl-5-oxo-N-[2-phenylsulfanylethyl]-4-(3-piperidin-1-ylpropylidene)furan-3-carboxamide [4-(methoxymethyl)-8,9-dihydro-7H-thieno[3,2-f]quinazolin-6-yl]-pyrrolidin-1-ylmethanone 3-(6,6-dioxo-1,4-oxazepan-4-yl)benzoic acid;hydrochloride 5-(1,2-dihydropyridin-4-yl)-3-pyridin-3-yl-2H-pyrazolo[3,4-b]pyrazine 2-(4-fluorophenyl)-7,8,9,10-tetrahydrobenzo[b][1,8]naphthyridine 1-[3,4-dimethoxy-5-(trifluoromethyl)phenyl]azetidine 2-amino-6,7-dimethoxy-3H-quinazolin-4-one N-[(Z)-2,3-dihydroinden-1-ylideneamino]-4-phenylsulfanylpyridine-2-carboxamide 3-(4-bromo-5-methyl-1H-pyrazol-3-yl)azetidine N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-hexylethanesulfonamide 3-(4-aminophenyl)cyclohexane-1,2-dione N-cyclopropyl-1-methanimidoyl-7-[1-(4-fluorophenyl)cyclopentyl]oxy-3-oxo-2,6-dihydroazepino[4,5-b]indole-8-carboxamide 3-[4-(dimethylamino)phenyl]benzene-1,2,5-tricarboxylic acid 2-[1-[4-(5-cyclopropyl-3-fluoropyridin-2-yl)piperazine-1-carbonyl]pyrazol-3-yl]acetamide 2-N-(4-bromophenyl)-4-N,6-dimethyl-1H-pyrimidine-2,4-disulfonamide 4-(2,3-dihydro-1H-indol-5-yl)-6-(methanesulfonamido)-N-[(4-methoxyphenyl)methyl]quinoline-7-carboxamide 3-[(2,4-diaminopteridin-6-yl)methoxy]propane-1,2-diol 2-[4-[(5-chloropyridin-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N-[cyclopropylidene-[5-fluoro-6-methoxy-8-(oxan-4-ylamino)quinazolin-4-yl]methyl]acetamide 1-(4,6-dimethylpyrimidin-2-yl)-3-[3-(1,5,7,10,11-pentazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-12-yloxy)cyclobutyl]urea 5-[(3Z)-4,6-dimethylhepta-1,3,5-trien-3-yl]sulfonyl-2-(3,7-dimethyloctoxy)benzonitrile 4-[5-(1,3-benzodioxol-5-yl)-2H-triazol-4-yl]-3,6-bis(difluoromethoxy)-9H-pyrido[2,3-b]indole 4-[[2,6-difluoro-4-(5-hydroxy-3-methylpent-1-enyl)phenyl]methylideneamino]benzenesulfonamide 4-[3,5-dimethyl-1-(2,2,2-trifluoroethoxy)cyclohexa-2,4-dien-1-yl]benzoic acid 4-[(Z)-[7-cyclopropylimino-5-[2-(3,3-difluoropyrrolidin-1-yl)ethoxy]pyrazolo[1,5-a]pyrimidin-3-ylidene]methyl]-5-hydroxy-1,3-dihydroimidazol-2-one 2-[[5,6-bis(4-methoxyphenyl)pyridazin-3-yl]amino]ethanol N-[4,5-difluoro-2-(hydroxymethyl)phenyl]-5-iodo-1H-pyrrolo[2,3-b]pyridine-3-carboxamide (2R)-N-[4-fluoro-3-[1-(6-iodoquinazolin-2-yl)piperidine-4-carbonyl]phenyl]-2,5-dimethylpyrrolidine-1-carboxamide (E)-2,3-diamino-3-[2-amino-3-(4-ethoxyphenyl)quinolin-6-yl]prop-2-enenitrile ethane;8-ethyl-N,N-dimethylnaphthalen-1-amine 2-[(3,4-dimethoxyphenyl)carbamoylamino]benzamide 1-azidosulfanyl-3-(3,4-dichlorophenyl)sulfanylbenzene 4-(3-azidophenoxy)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine N-(4-cyclopentylphenyl)-2,6-dimethoxypyridine-3-carboxamide 3-hydroxy-2,6-dimethyl-8-[4-(trifluoromethoxy)phenyl]naphthalene-1,4-dione 4-cyclopropylsulfonylmorpholine;N-[3-(difluoromethoxy)phenyl]-2-methylpyrimidine-5-carboxamide 1-[(3R)-1-azabicyclo[2.2.0]hexan-3-yl]-8-benzamidopyrene-2-carboxylic acid N-benzyl-2-bromo-N',5-dimethoxybenzohydrazide N-[(2S)-1-hydroxybutan-2-yl]-1-methoxy-7,8-dihydro-6H-isoquinoline-3-carboxamide 3-[N-(4-hydroxybutyl)-2,6-dimethoxyanilino]propane-1,2-diol (4Z)-2-methyl-4-[(4-pyrazol-1-ylphenyl)methylidene]-1,3-oxazol-5-one [6-(2,4-difluorophenyl)sulfanylimidazo[1,5-a]pyridin-8-yl]methanethiol [2-(3,5-difluorophenyl)pyrrolidin-1-yl]-(4-pyrrolidin-1-ylpyrimidin-2-yl)methanone 3-(3,4-dichlorophenyl)-N'-hydroxypropanimidamide N-methyl-4-[[(2S)-1-[5-(trifluoromethyl)pyridin-3-yl]oxypropan-2-yl]amino]quinazoline-8-carboxamide 4-(3,5-dimethylphenoxy)butane-1-sulfonic acid 2-[(1-azidocyclopropyl)methoxy]-3,4,5,6-tetrafluorophenol N-(4-bromobutan-2-yl)-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridin-2-amine 2-tert-butyl-N-[(4,5-dichlorothiophen-3-yl)methyl]-6-methoxypyrimidin-4-amine 3-[4-(1-benzylpyrazol-4-yl)pyridin-2-yl]-3,4-dihydroquinoline 3-[2-(6,7-dimethoxyquinolin-4-yl)ethynyl]-5-fluoro-N-methoxyaniline 3-bromo-2,5-dichlorobenzoic acid;propanoic acid 1-(1H-indol-3-yl)pentan-2-one N-[1,2-bis(3,4-difluorophenyl)ethyl]formamide 1-[[5-(4-aminophenyl)-2,3-dihydrofuran-2-yl]methylsulfanyl]propan-2-ol 1-[2-(3,4-dimethoxyphenyl)-1H-tetrazol-5-yl]ethanone (E)-3-(4-chlorophenyl)sulfanyl-N,2-dimethylprop-1-en-1-amine 3,5-dichloro-N-[(E)-[4-(2-methylphenyl)piperazin-1-yl]iminomethyl]benzenecarboximidate 4-[5-(difluoromethyl)pyrazine-2-carbonyl]-N'-(6-ethoxypyridin-3-yl)piperazine-1-carbohydrazide N-(4,5-dihydro-1H-imidazol-2-yl)-7-[6-methoxy-5-[(3S)-piperidin-3-yl]pyridin-3-yl]imidazo[1,2-a]pyridine-3-carboxamide 2-[[4-(azetidin-1-yl)piperidin-3-yl]methoxy]-6,7-dihydro-5H-cyclopenta[d]pyrimidine N-[4-fluoro-3-(5-methoxypyridin-3-yl)phenyl]-6-oxo-1H-pyrazine-3-carboxamide 2-[4-[2,6-dimethyl-5-(3-sulfopropanoylamino)phenyl]phenyl]acetic acid N-(2,4-dichloropyrimidin-5-yl)-N-[4-methoxy-6-methyl-1-[2-(2-phenylethynyl)benzoyl]indole-3-carbonyl]acetamide (2S)-1,3-difluoro-N-[4-methyl-5-(trifluoromethyl)pyridin-2-yl]cyclobutane-2-carboxamide 2,3-dimethyl-5-[[(1R)-1-phenylethyl]amino]sulfanylbenzonitrile 5-chloro-4-[2,6-difluoro-3-(trifluoromethyl)phenyl]pyrimidine 7-[(2-chlorophenyl)methyl]-8a-ethyl-2-methylsulfonyl-4a,5,6,8-tetrahydro-3H-pyrido[3,4-d]pyrimidin-4-one 4-(2,3-dihydro-1H-inden-5-yloxy)cyclohexan-1-one 3-[(4-aminocyclohexyl)sulfamoyl]benzoic acid 1-ethyl-3,4-difluoro-2-propan-2-ylidene-5-(trifluoromethoxy)benzene 2-ethyl-4-[[(1R)-1-(4-fluorophenyl)ethoxy]methyl]pyrimidine N-[2-azidosulfanylethyl(methylamino)amino]aniline N-[2-(1-methyl-6,7,8,9-tetrahydroimidazo[4,5-c]isoquinolin-2-yl)ethyl]acetamide;hydrochloride 1-ethyl-6-fluoro-7-(4-methoxyphenyl)-4-oxoquinoline-3-carboxylic acid 4-[5-(1H-indol-3-yl)-4,5-dihydro-1,2-oxazol-3-yl]benzoic acid 1-(4-methoxyphenyl)-7-propyl-2,6-dihydropyrazolo[5,1-c][1,2,4]triazine 1-ethyl-5-(4-fluorophenyl)-3,3,4,7-tetramethylquinolin-2-one 3-[(2S)-1,2-dimethyl-5-oxopyrrolidin-2-yl]oxybenzonitrile 1-amino-3-[(2,5-dichlorothiophene-3-carbonyl)amino]thiourea 4-[5-fluoro-2-(2,2,3,3-tetrafluoropropoxy)phenyl]-7-oxo-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-2-carbonitrile 2-fluoro-1,3-diphenylpropan-1-ol N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[5-ethylsulfonyl-6-[1-oxo-6-(trifluoromethyl)phthalazin-2-yl]pyridin-3-yl]acetamide 3-(9-fluoropyrido[1,2-a]benzimidazol-10-yl)propanenitrile 2-cyclohexa-1,5-dien-1-yl-5-phenyl-2H-[1,3]thiazolo[4,5-b]pyridine 6-(4-cyanobenzoyl)-2-methoxybenzoic acid 5-[4-[3-(4,6-dimethylpyrimidin-2-yl)oxy-1,2,4-oxadiazol-5-yl]butyl]thiophene-3-carboxylic acid 3-(4-ethenylphenyl)bicyclo[1.1.1]pentan-1-amine 2-chloro-5-(chloromethyl)imidazo[1,2-a]pyridine 6-[(4-fluorophenyl)methyl]-1H-indole N-benzylsulfanylcyclohexanamine 1-[2,5-dimethyl-4-(3,3,3-trifluoropropoxy)pyridin-3-yl]ethenol 6-[3-(2,4-diaminopyrimidine-5-carbonyl)oxypropyl]pyridine-2-carboxylic acid 2-[4-ethoxycarbonyl-N-(4-hydroxybutyl)anilino]decanoic acid 3-[(2E)-6-chlorohexa-2,4-dienyl]sulfanyl-5-methoxybenzamide (5R)-6-[3-ethyl-4-[6-[methyl(propan-2-yl)amino]pyridin-3-yl]phenyl]-1,8-diazaspiro[4.5]decane-2,9-dione (2R,6S)-4-[3-(dimethylamino)propoxy]-2,6-bis(2-methylbutan-2-yl)-4-phenylsulfanyloxane 2-[(4-methylphenyl)methylamino]-3H-[1,3]thiazolo[5,4-b]pyridine-6-thione 2-(azidomethyl)-1,4-dichlorobenzene 2-[(6S)-5-amino-4-methyl-6,7-dihydro-1,3-benzothiazol-2-yl]-4-fluorophenol N-azido-2-chloro-6,7,8,9-tetrahydrobenzo[b]fluoren-1-amine 2-fluoro-1,4-bis(isocyanatomethyl)-3-methylbenzene 2-[2,3,6-tris(trifluoromethyl)phenyl]phenol 2-methoxy-6-[4-[2,3,5,6-tetrafluoro-4-(trifluoromethyl)phenoxy]cyclohexa-1,3-dien-1-yl]naphthalene 2-bromo-1-[4-(methoxymethyl)phenyl]ethanone 2,4-dichloro-5-[2-(2-methylphenyl)ethynyl]aniline N-azido-1-[4-(difluoromethoxy)phenyl]cyclopropan-1-amine 1-[2,6-di(propan-2-yl)phenyl]imidazolidine N-[4-(3,4-dihydroisoquinolin-1-yl)phenyl]-N'-[2-[[5-fluoro-2-hydroxy-6-(trifluoromethoxy)cyclohepta-1,4,6-trien-1-yl]sulfonylamino]ethyl]methanimidamide N-ethyl-3,4-dimethoxy-2-methylaniline 4-[1-(8-amino-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)ethenyl]benzoic acid 5-bromo-4-ethoxycarbonyl-3-methyl-2,6-dinitrobenzoic acid 3-[5-bromo-4-(hydroxymethyl)-1H-indole-2-carbonyl]-N,N-diethylcyclohexane-1-carboxamide 5-bromo-N-butyl-2-ethenoxy-3-methylpyridine-4-carboxamide 2-hydroxy-6-(4-methylphenyl)-1,3,8,12-tetrazatricyclo[7.3.0.03,7]dodeca-9,11-dien-8-ol 4-[[2,6-difluoro-3-(trifluoromethyl)benzoyl]amino]butanoic acid 4-[1-(2,4-dichlorophenyl)ethyl]-1H-pyrimidine-2,4,5-triamine 4-amino-N'-(1-hydroxynaphthalen-2-yl)sulfanylpyridine-3-carboximidamide 4-[6-chloro-3-(pyridin-2-ylmethoxy)naphthalen-2-yl]benzaldehyde (3Z,5E)-1-(4-ethylphenyl)-7-[2-fluoro-6-(trifluoromethoxy)phenyl]hepta-3,5-dien-3-ol N-(4,6-dimethylpyrimidin-2-yl)-4-[ethylsulfonyl(phenacyl)amino]benzenesulfonamide 1-(4,6-dimethylpyrimidin-2-yl)sulfanylpyrrolidine-3-carboxylic acid 1-methyl-3-[2-(4-phenylbutyl)pyrrolidin-1-yl]pyrazin-2-one 2-[3-(hydroxymethyl)anilino]-1,7-dihydropurin-6-one N-(2,4-dimethylpyridin-3-yl)-5-propan-2-ylpyridine-2-carboxamide [2-amino-5-(trifluoromethyl)-3,4-dihydropyridin-6-yl]-[1-[(2S,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrrolo[2,3-b]pyridin-3-yl]methanone [(Z)-2-(2,3-dihydroxyphenyl)ethenyl]sulfonylazanium 6-[6-(2,2,2-trifluoroethoxy)pyridin-3-yl]-1H-benzimidazole 2-(5-azidoindol-1-yl)-N,N-dimethylethanamine 3-[(2,4-difluorophenyl)methyl]-5H-pyrrolo[3,2-d]pyrimidine N-(5,7-dichloro-1-phenyl-3H-2,1-benzoxaborol-6-yl)-2-(methanesulfonamido)acetamide 2-[4-(2,3-dihydropyridin-5-yl)naphthalen-1-yl]-4,6-diphenyl-1,3,5-triazine 3-[2-ethyl-5-(4-fluorophenyl)pyrrol-1-yl]propanenitrile 4-(3,5-dimethylphenyl)-7-hydroxychromen-2-one 4-hydroxy-2-[(E)-[(1,3,5-trimethylpyrazole-4-carbonyl)hydrazinylidene]methyl]benzenecarboximidamide 1-(2,3-dimethylphenyl)-N-[3-(4-ethoxypiperidine-1-carbonyl)phenyl]cyclopropane-1-carboxamide 2-[(3S,4R)-1-[5-amino-6-[5-(dimethylcarbamoyloxy)pyridin-2-yl]pyrazin-2-yl]piperidin-3-yl]acetic acid 2-(1,3-dioxol-4-yl)-4H-[1,3]thiazolo[5,4-b]pyridine 4-[1-(5-methoxy-3,4-dihydro-2H-1-benzothiepin-8-yl)ethyl]benzaldehyde 1-(2,4-dimethoxyphenyl)-3-(oxolan-2-yl)propan-2-ol 3-benzyl-N-[(2S)-1-aminobutan-2-yl]-5-butoxy-4,7-dioxo-6H-triazolo[4,5-d]pyrimidine-2-carboxamide 1-[4-(5-aminopyrazin-2-yl)piperazin-1-yl]prop-2-en-1-one N-[2-(2,6-dichlorophenyl)propyl]butanamide 5-(2,6-diphenylpyrimidin-4-yl)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-1,2-benzoxazol-3-amine 2-methyl-5-[3-(trifluoromethoxy)phenyl]pyridine 3-(4-aminopiperidin-1-yl)-6-azidosulfanyl-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine 2-(5-hydroxy-4-iminocyclohexa-1,5-dien-1-yl)-3-methylbenzimidazole-5-carbonitrile 4-[2-(3,5-dimethylpyridin-1-ium-4-yl)-5-propan-2-ylpyridin-4-yl]-N,N,5-trimethylaniline;ethane 6-[3-[2-(4,4-difluorocyclohexyl)oxypyridin-4-yl]phenyl]-1H-indene 2-[3,4,5-trimethyl-6-(2-phenylethoxy)cyclohexa-1,5-dien-1-yl]pyridine 2-(4-methoxy-N-methylsulfonylanilino)acetic acid 5-(3,6-dihydro-2H-pyran-4-yl)-N-[6-[4-[(2S)-1-hydroxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]furan-2-carboxamide N-[4-(1,3-benzothiazol-2-yl)phenyl]-7-(dimethylamino)-N'-[2-(ethylaminosulfanyl)-5-fluoro-6-propanoylpyrimidin-4-yl]-9H-fluorene-2-carboximidamide 5-methyl-2-(trifluoromethyl)pyrrolo[2,3-b]pyridine-1-carboxamide 4-(2,3-dimethylphenyl)-5-ethoxycarbonyl-1-(3-fluoropyridin-4-yl)pyrrole-2-carboxylic acid 4-[(2Z)-4-methylpenta-2,4-dienoyl]benzamide N-[4,4-difluoro-1-(hydroxyamino)-3-methyl-1-oxobutan-2-yl]-4-[[6-ethoxy-5-(4-hydroxypiperidine-1-carbonyl)pyridin-2-yl]amino]-3-methylbenzamide 2-[[4-(difluoromethoxy)phenyl]iminomethyl]-6-propan-2-ylphenol 2-[(Z)-but-1-enyl]-4,6-dimethylnaphthalene 1-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]spiro[2H-indole-3,7'-6H-furo[2,3-f][1,3]benzodioxole] 3,6-difluoro-4-[(E)-2-iodoethenyl]benzene-1,2-dicarbonitrile 6-[3-(2,5-difluorophenyl)imidazo[1,5-a]pyridin-8-yl]-2-(trideuteriomethyl)quinoline N-[(3R)-1-[2-cyano-4,6-bis(trifluoromethyl)phenyl]pyrrolidin-3-yl]formamide 5-bromo-4-[2-(4-fluorophenyl)ethylamino]-1H-pyrimidin-6-one 2-[2-[[4-[2-(1,3-benzoxazol-6-yl)ethynyl]phenyl]methylideneamino]propoxy]acetic acid (2R)-3-[4-[2-methoxyethyl(propan-2-ylsulfamoyl)amino]phenyl]-N-methylsulfonyl-2-(2,2,2-trifluoroethoxy)propanamide N-(4-chlorophenyl)sulfonyl-2-[5-cyano-3-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]-2-methoxyacetamide 2-[(1S,3R)-5,6-dimethoxy-3-methyl-2-phenylmethoxycarbonylcyclohexa-2,4-dien-1-yl]acetic acid (1R)-N,2-dimethyl-4-[methyl(6-piperazin-1-ylpyrimidin-4-yl)amino]cyclopentane-1-carboxamide 2-chloro-3,5-difluoro-N'-hydroxybenzenecarboximidamide 6-amino-2-(5,6-dimethoxypyridin-3-yl)-N-methyl-1H-indole-4-carboxamide (3R)-3-[[2,3,4-tris(fluoromethyl)phenyl]methoxy]azepane [(3S,5R)-4-(2,6-dimethoxyphenyl)-5-propylpyrrolidin-3-yl]azanide N-methyl-2-(7-morpholin-4-ylquinazolin-5-yl)oxypyridine-3-carboxamide (2E,4Z)-N-[3-[(4aS)-8a-methyl-1-oxo-6,7-dihydro-5H-imidazo[1,5-a]pyrazin-4a-yl]-5-fluorophenyl]-4-phenylhepta-2,4,6-trienamide 1-N',2-N'-bis[4-(4-tert-butylphenyl)phenyl]ethanedihydrazide 2,4-dichloro-5-(3,5-dimethylphenyl)pyrimidine;2-[(1S)-6-(ethoxycarbonylamino)-2,3-dihydro-1H-inden-1-yl]acetic acid (1R)-2-[4-bromo-5-[5-(dimethylamino)pyridin-3-yl]oxybenzimidazol-1-yl]-N,N-dimethyl-1-phenylethanamine 3-(1,3-benzothiazol-2-yl)-7-chlorochromen-4-one 1-[4-(cyclohexa-2,4-dien-1-ylmethoxy)phenyl]propan-1-amine;propane 4-(4-amino-6,7-dimethoxyquinazolin-2-yl)benzenesulfonamide 6-(3,5-dimethylphenyl)sulfanylcyclohexa-1,4-diene-1,3-diamine 2-cyclohexa-1,5-dien-1-yl-4-phenylbutan-1-amine N'-[4-[(Z)-[(5E,6E)-2,3-bis(ethenyl)-6-ethylidenecyclohexen-1-yl]methoxyiminomethyl]pyridin-1-ium-1-yl]propane-1-sulfonamide N-[2-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl(phenyl)sulfamoyl]propanamide 5-[[4-(3,5-dichloropyridine-2-carbonyl)piperazin-1-yl]methyl]-1-benzofuran-7-carboxylate N-cyclohexyl-5-methoxy-3,4-dihydroisochromen-1-imine (E)-3-[2,5-dimethyl-1-[3-[[2-(4-methylphenyl)benzoyl]amino]propyl]pyrrol-3-yl]-N-hydroxyprop-2-enamide [[2-(aminomethyl)cyclohexyl]amino]-[(4R,8aS)-3-cyclopropyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-4-yl]methanone 3-[(4R)-2-ethyl-1-[1-(4-methoxyphenyl)ethenyl]-6,7-dihydro-5H-pyrrolizin-3-yl]propanenitrile N-(3-hydroxypropyl)-2-methoxy-N-octylbenzamide 2-[(3E)-penta-1,3-dien-3-yl]-N-propan-2-ylidenecyclopropane-1-carboxamide;yttrium 5-[2,3-difluoro-4-(hydroxymethyl)phenyl]pentanoic acid [(3aR,7aS)-2-benzylsulfonyl-1,3,3a,4,5,6,7,7a-octahydroisoindol-1-yl]-morpholin-4-ylmethanone 1-(4,5-dimethylthiophene-2-carbonyl)piperidine-3-carboxylic acid 5-tert-butyl-3-[(E)-1-(4-chlorophenyl)prop-1-en-2-yl]cyclohepta-1,3,5-triene;ethane [3-[2-aminoethyl(ethyl)amino]pyrrolidin-1-yl]-[4-[5-(trifluoromethoxy)pyridin-2-yl]phenyl]methanone (5Z)-4-[[1-(4-fluorophenyl)pyrazol-3-yl]methylidene]-2,7,9,10-tetrahydro-1H-pyrimido[4,5-b]quinoline 7-chloro-4,8-dimethylquinoline-3-carboxylic acid 4-[[2-(3,5-dimethylphenyl)sulfanylpyrimidin-5-yl]methoxy]aniline 2-azido-3,4,5,6,7,8-hexachloronaphthalene (5-bromoindol-1-yl)-[4-hydroxy-2,3,5-tri(propan-2-yloxy)phenyl]methanone (2S)-1-[2-hydroxyethyl(methylaminomethyl)amino]-3-thiophen-2-ylpropan-2-ol (4S,5R)-N-benzyl-4-[2-[3-fluoro-4-(trifluoromethoxy)phenyl]pyridin-4-yl]-7-(2H-tetrazol-5-yl)heptanamide 4-[(E)-2-[1-[(Z)-3-hydroxybut-2-enoyl]piperidin-3-yl]ethenyl]-N-(5-imidazol-1-ylpyridin-2-yl)benzamide 1-[(3S)-3-methylpiperazine-1-carbonyl]-2H-quinoline-4-carboxylic acid 4-(6-aminopyridin-2-yl)benzene-1,3-diol 3-[4-(3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-2-carbonyl)phenyl]-N-cyclopropyl-5-oxopiperazine-1-carboxamide N-(5,6-dimethyl-[1]benzofuro[2,3-b]pyridin-8-ylidene)hydroxylamine 4-methyl-3,5-bis(2-phenylethoxy)benzamide 5-bromo-3,4-difluoronaphthalene-1,2-dione 6-bromo-2,3-difluorobenzenesulfonic acid 3-[6-(2,5-dimethylphenyl)pyridin-1-ium-2-yl]-9,11-bis(2,2,6,6-tetramethylpiperidin-4-ylidene)indeno[2,1-a]fluorene 2-[4-cyano-3-(trifluoromethyl)phenyl]-8-(5,6-diethoxypyrimidine-4-carbonyl)-N,N-dimethyl-2,8-diazaspiro[4.5]decane-4-carboxamide 5-methyl-1-[(2R)-2-phenylpropyl]imidazole 3-(4-chlorophenyl)-2,5-dihydrothiaphosphol-1-ium-4-amine;ethane 2-[(2-bromophenyl)methyl]-4-[3-(2,5-dichlorothiophen-3-yl)-1H-pyrazol-5-yl]morpholine N-[(3S,7R,8aS)-3-(4-chlorophenyl)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-2-(1,5,6-trimethylpyrazolo[3,4-b]pyridin-3-yl)acetamide 2-methyl-4-[3-(trifluoromethoxy)anilino]butanamide N-[4-(2,3,5,6-tetrafluorophenoxy)butyl]benzenesulfonamide 2-[6,8-bis(4-chlorophenyl)imidazo[1,2-a]pyrazin-3-yl]acetic acid 2-fluoro-1-[4-(triazol-1-ylmethoxy)phenyl]ethanone (3-bromophenyl)-[2-(hydroxymethyl)piperidin-1-yl]methanone (E)-3-aminooxy-1-[4-[7-chloro-6-fluoro-8-methyl-2-(2,2,2-trifluoroethoxy)quinolin-4-yl]piperazin-1-yl]prop-2-en-1-one 3-cyclopropyl-2,5-dimethoxy-1H-pyridine-4-thione 4-amino-N'-[4,6-bis(ethenyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-5-carboximidamide;N'-(2-methoxyphenyl)methanediamine N-[(1R)-2,3-dihydro-1H-inden-1-yl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxamide 2-N-[4-(1H-indazol-5-ylamino)pyrimidin-2-yl]-2-N-propan-2-ylbenzene-1,2,4-triamine (3S)-2-[(1,5-dimethylpyrazole-4-carbonyl)amino]-3-hydroxybutanoic acid 5-[3,4-dimethoxy-5-(2H-tetrazol-5-yl)phenyl]-1-methylpyrrole-2-carboxamide 2-[4-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]quinoline 4-[[3,5-difluoro-2-(methoxymethyl)phenyl]methylideneamino]pyridine-2-carbonitrile 3-[1-methyl-5-oxo-4-(pyridine-3-carbonyl)pyrazol-3-yl]benzonitrile 3-[2-(3,4-dimethoxyphenyl)ethynyl]-5-(6-fluoro-1H-indol-3-yl)piperidine-1-carboxylate 6-(8-ethylnaphthalen-1-yl)oxy-3,4-dihydro-2H-naphthalen-1-one 2-(4-aminobutyl)-3,7-difluorobenzimidazole-5-carboxylate 2-[3-cyclopropyl-1-(4-methoxyphenyl)pyrazol-4-yl]oxyacetic acid 2-[7,8-difluoro-6-(trifluoromethoxy)isoquinolin-3-yl]-1-pyridin-4-ylethanone N'-ethyl-4-(5-methyl-3-oxo-1H-2-benzofuran-1-yl)piperazine-1-carboximidamide 1-[(2R,6S)-4-azido-6-cyclopropylmorpholin-2-yl]-3-phenylpyrazol-4-amine N-[(2S,3R)-4-[2-chloro-4-(trifluoromethylsulfanyl)anilino]-1-(3,5-dihydroxyphenyl)butan-2-yl]-2-methoxybenzamide 2-[4-fluoro-3-(methoxymethyl)phenyl]-1,3-thiazole N-methyl-2-(1,3-thiazol-4-yl)benzenesulfonamide 2-N,7-N-bis(3-aminopropyl)naphthalene-1,2,4,6,7-pentamine (E)-1,3-dimethoxyprop-2-en-1-ol;6-methyl-4-[(3R)-pyrrolidin-3-yl]oxyquinazoline 2-(1H-pyrazol-5-yl)-4-[3-(trifluoromethoxy)phenyl]piperazine N-[5-chloro-2-(1H-indole-3-carbonyl)phenyl]-4-methoxybenzenesulfonamide 1-[(Z)-2,5-dimethylideneoct-3-enoxy]-4-fluorobenzene 2-[3-(1,4-dioxaspiro[4.5]decan-8-yl)phenyl]benzamide 2-[4-[5-(2,4-difluorophenyl)-3-methylimidazol-4-yl]triazol-1-yl]ethanesulfonic acid N-[(Z)-1H-indol-3-ylmethylideneamino]-2,2-diphenylacetamide 2-amino-5-[(3E,5Z)-hepta-1,3,5-trien-4-yl]benzaldehyde 1-cyclohexa-2,4-dien-1-ylbutylbenzene (E)-1-(4,5-dihydro-1H-imidazol-2-ylamino)-3-[2-methoxy-6-[[2-methyl-7-(trifluoromethyl)quinolin-4-yl]amino]phenyl]prop-2-en-1-ol 1,2-bis(4-chlorophenyl)-7-nitroquinazoline-4,6-dione 1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-3-(dimethylamino)propan-2-ol 1-(4-azidophenyl)-2,3,5-trichlorobenzene 2-[5-[3-(1,7-dioxo-6H-pyrrolo[3,4-d]pyridazin-2-yl)-4-methylphenyl]pyridin-3-yl]-N'-methanimidoyl-N-propan-2-ylideneacetohydrazide 2-[(E)-[[1-[3,5-bis(trifluoromethyl)phenyl]pyrrolidin-3-ylidene]hydrazinylidene]methyl]-4,6-diethoxyphenol 4-(5-azidosulfanylbenzotriazol-2-yl)phenol 4-[(3aR)-2,2-dimethyl-5-oxo-1,3,3a,6a-tetrahydrocyclopenta[c]pyrrole-4-carbonyl]benzoic acid 2-tert-butyl-4-propan-2-yl-5,6,7,8-tetrahydroquinazoline (E)-2-cyano-3-(2,3-dihydro-1H-inden-5-ylamino)sulfanylprop-2-enoic acid 2-(4-chlorophenyl)-N-[3-(3,5-dimethoxyphenyl)-1H-pyrazol-5-yl]acetamide [3-(cyclopropylmethoxy)phenyl]-spiro[1,4-dihydroquinoline-3,5'-oxolane]-2-ylidenemethanamine 5-(diethylamino)-2-[[4-[(E)-2-(2,6-difluorophenyl)ethenyl]benzoyl]amino]benzoic acid 1-[4-(N'-tert-butylcarbamimidoyl)phenyl]-2,3,6,7-tetrahydroazepine-4-carboxamide 3-methoxy-4-[(5Z,7E)-6-methylideneundeca-1,5,7,9-tetraen-2-yl]phenol N-(8-bromoquinoxalin-5-yl)-2,4,6-trimethyl-N-propylbenzenesulfonamide 4-[1-(5,6-dichloro-2-hydroxypyridin-3-yl)ethylamino]thieno[2,3-d]pyrimidine-6-carboxylate N-[(3,4-difluorophenyl)methyl]-2-iodoacetamide 1-[(5-bromo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3-(5-propan-2-yl-1H-pyrazol-3-yl)urea;hydrochloride 4-hydroxy-6-methyl-3H-naphtho[2,1-h]quinoline-2-sulfonate 7-(6,8-dimethylimidazo[1,2-a]pyrazin-3-yl)-5,10-difluoro-2,7-diazatricyclo[6.3.1.04,12]dodeca-1,3,5,8,10-pentaene 2-[4-(1,3-benzodioxol-5-yl)-3-phenylbutanoyl]cyclohexane-1-carboxylic acid 5-amino-2-[3-chloro-4-(trifluoromethoxy)phenyl]-6,6-diethylcyclohexa-1,3-diene-1-carboxamide N'-[2-(dimethylamino)pyrimidin-4-yl]thieno[3,2-d]pyrimidine-2-carbohydrazide (Z)-1,2-dicyanoethene-1,2-dithiolate;2-[3-methylbutan-2-yl(prop-2-enyl)amino]benzoate;titanium(4+) N-[3-(2,4-dimethylpentanoyl)phenyl]prop-2-enamide 2-amino-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-ylmethyl)cyclopentane-1-carboxamide;hydrochloride 3-N-[3-(cyclopropanecarboximidoyl)phenyl]benzene-1,2,3-tricarboxamide;ethane 1-azido-3,4-dimethyl-5-nitropyrazole 1-[(3R)-5,7-dichloro-2,3-dihydro-1H-inden-4-yl]-3-(1-pyridin-2-ylcyclopropyl)urea 2-methoxyimino-N,3-diphenylbutanamide (2R)-3,3-dimethyl-5-phenyl-4H-naphthalene (4R)-7-[[(2S,3S)-2-[[4-(3-fluorophenyl)phenyl]methylamino]pentan-3-yl]oxymethyl]-3,4-dihydro-1H-1,8-naphthyridin-2-one 2-[2,4-dichloro-5-(6,7-dimethylquinolin-3-yl)oxyphenyl]-N-ethylbutanamide 2-[(1S,3R)-5-amino-3-ethylcyclohexyl]oxycarbonylbenzoic acid 1-[5-methyl-4-(2,4,6-trifluorophenyl)hexanoyl]pyrrolidine-2-carboxamide N-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-3-yl]acetamide 3-[4-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine N-(4-methoxyphenyl)sulfonylspiro[1,2-dihydroindene-3,3'-pyrrolidine]-1'-carboxamide 1-azidooxy-2,4-dichlorobenzene 2-ethyl-5-(2H-azirin-1-ium-1-ylmethoxy)-4,6-difluoropyridine;5-[4-(5-oxo-3-phenyl-1,2-oxazolidin-2-yl)phenyl]pyrazin-2-amine 6-(2,4,4-trimethylpentan-2-yl)naphthalene-1,3-diamine N-[(Z)-(5,6-dichloro-2,3-dihydroinden-1-ylidene)amino]-N-phenylbenzamide N-[2-fluoro-5-(1H-indole-2-carbonyl)phenyl]-4-(methylsulfamoyl)thiophene-3-carboxamide 1-[3-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]phenyl]piperidine 1-azido-3-ethylsulfinylnaphthalene ethane;5-[(3E)-hexa-1,3,5-trien-3-yl]-2-[3-[methyl-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]amino]phenyl]pyridine-3-carbonitrile 2-[(E)-[4,6-dioxo-1-phenyl-2-sulfanylidene-5-[[2-(trifluoromethyl)phenyl]hydrazinylidene]-1,3-diazinane-5-carbonyl]amino]acetic acid 2-(4,5-dimethyl-1H-imidazol-3-ium-3-yl)quinoline (E)-4-(5-amino-2,3-dihydroindole-1-carbonyl)oxybut-3-enoic acid 2-chloro-3,4,6-trimethoxybenzoate 3-[4-(5-oxo-1H-tetrazol-4-yl)phenyl]-1,2,3-benzotriazin-3-ium-4-one ethane;2-methoxy-4-[3-(8,9,10,11-tetrahydrobenzo[b][1]benzazepin-5-yl)propyl]phenol (4-methoxyphenyl)methylcarbamodithioic acid 2-cyclopropyl-4,4-difluoro-1,3-dihydroisoquinoline;methanamine 2,6-dimethyl-5-[4-(1H-pyrazol-4-yl)phenyl]-[1,2,4]triazolo[3,4-a]pyrimidin-8-one 3-[1,3-dimethyl-5-(2-thiophen-2-ylacetyl)indol-6-yl]benzoic acid 1-(azidomethyl)-4-(difluoromethoxy)benzene N-[4-(cyclohexen-1-yl)phenyl]-N-phenylnaphthalen-2-amine;6-methylidenecyclohexa-2,4-diene-1,1-dicarbonitrile N-[(2R)-5,7-difluoro-1,2,3,4-tetrahydronaphthalen-1-yl]-3-hydroxy-8-[(1-methylpyrazol-3-yl)methoxy]-3H-furo[3,4-c]quinoline-1-carboxamide 2-[3,5-bis(2-aminophenoxy)phenyl]ethanol 1-[4-(4,6-dimethoxypyrimidin-2-yl)piperazin-1-yl]-2-[2-(ethylamino)phenyl]ethanone;ethane (4S)-2,5-dihydroxy-N-[(1S,2R,3S)-2-phenylcyclopropyl]-4,6-bis(phenylmethoxy)hexanamide 3,4-difluoro-2-N-(1H-pyrazolo[4,3-d]pyrimidin-5-yl)benzene-1,2-diamine 2-[4-(1,3-benzodioxol-5-yl)butyl]-N-(1H-pyrazol-4-ylmethyl)-6-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine (2S)-1-[(3,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylic acid 1-[3-(2,4-difluorophenyl)-1-bicyclo[1.1.1]pentanyl]-N,N-bis(pyridin-2-ylmethyl)methanamine 4-[2,5-dimethyl-3-(trifluoromethyl)pyridin-1-ium-1-yl]benzonitrile N-[4-chloro-2-(1,3-thiazol-5-ylcarbamoyl)phenyl]-4-(4-methoxybutan-2-ylsulfamoyl)benzamide 2-[2-(2,4-dichlorophenyl)ethoxy]pyridine 3-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenoxy]-1-(4-fluorophenyl)propan-1-ol;ethane (6S)-4,4,8,11,14,15,17-heptamethyltetracyclo[7.7.0.02,6.010,15]hexadeca-1(9),2,10,12,14-pentaene 1-(4,5-dimethylthiophen-2-yl)ethanethiol N-benzyl-4-[5-(3,6-difluorocarbazol-9-yl)-1-iodophosphanylpentyl]-3,5-dimethoxyaniline 3-(4-carbamimidoylphenyl)-2-[1-oxo-5-(pyrrolidin-1-ylmethyl)-2H-1,3-benzothiazol-3-id-6-yl]propanoic acid 1-[5-bromo-6-(2,3-dihydro-1H-benzimidazol-2-yl)pyridin-3-yl]pyrrolidin-2-one 4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]-N-[3-methyl-1-[2-oxo-3-(propanoylamino)pyridin-1-yl]butyl]benzamide 2-(cyclohexylamino)-N',1-diphenylpyrazolo[3,4-d]pyrimidine-3-carboximidamide N-[5-cyclopropyl-2-(1,3,4-trimethylpiperazin-2-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide 1-[2-(5-bromopyrimidin-2-yl)oxyethyl]cyclopropan-1-amine 2-[4-[(3R,5S)-3-amino-5-fluoropiperidin-1-yl]pyridin-3-yl]-1-[6-[5-chloro-2-(oxan-4-ylmethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]ethanone 1,4-bis[2,6-di(propan-2-yl)phenyl]imidazolidine;palladium(2+);dichloride 3-[4-(1,1-difluoroethyl)phenyl]propan-2-amine;(E)-5-methylidenehept-6-ene (Z)-2,4-diamino-7-[(2S)-1-oxo-1-(5,6,7,8-tetrahydronaphthalen-1-yloxy)propan-2-yl]oxyhept-2-enoic acid N-[6-chloro-1-[(2R)-2-methylmorpholine-4-carbonyl]indol-7-yl]-1-phenylcyclopropane-1-sulfonamide 5-(2,6-dichlorophenyl)-6-oxo-3-[4-(trifluoromethyl)pyridin-3-yl]pyridazine-1-carboxylic acid 2-[3,5-dichloro-N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)anilino]octanoic acid N-[3-(methylamino)butyl]-6-(6,7,8,9-tetrahydrodibenzofuran-4-ylamino)hexanamide 5-[2,3,4-tris(prop-1-enoxy)phenyl]-2H-tetrazole 5-methyl-N-[(1R)-6-methylcyclohexa-2,4-dien-1-ylidene]-3,6-dihydro-2H-pyridine-1-carboxamide N-(3-aminophenyl)sulfanyl-4-(1,3-benzodioxol-5-ylmethoxy)-2-tert-butyl-6-chloroaniline N-[(1R,2S)-2-hydroxycyclohexyl]-4-methoxypyrimidine-5-carboxamide 5-ethyl-2,3-bis[(3-methylphenyl)imino]-1H-imidazo[4,5-c]pyridin-3-ium-7-carboxylic acid 4-azidooxy-2,6-di(propan-2-yl)benzenesulfonate 1-(2-methoxyethyl)-N,3,5-trimethylpyrazolo[4,3-d]pyrimidin-7-amine 4-methyl-N-(2-oxopropyl)benzamide 2-(aminomethyl)-4-[3-(4-hydroxy-3,5-diiodophenyl)prop-2-enoyl]oxybutanoic acid 5-ethyl-4-methoxy-6-[2,3,5,6-tetrafluoro-4-(4-propylcyclohexen-1-yl)phenyl]pyrimidine 2-[3,5-dimethyl-1-(2-pyrrolidin-1-ylethoxy)indol-2-yl]phenol 5-azidosulfanyl-4,8-dihydroxynaphthalene-2-sulfonic acid (5-cyclopropyl-1,2-oxazol-3-yl)-[2-(furan-2-ylmethyl)piperazin-1-yl]methanone;formic acid (1R)-N-benzyl-2,3-dihydro-1H-inden-1-amine N-[4,5-dimethoxy-2-(3-pyrrolidin-1-ylpropoxy)phenyl]acetamide 5-methyl-3-phenylmethoxycarbonylhexanoic acid 2-azidooxy-4-methylsulfonyl-1,3-oxazole N-[5,6-dimethyl-2-(2-phenylethynyl)pyridin-3-yl]methanesulfonamide 7-[3,5-bis(trifluoromethyl)phenyl]-6-oxo-2-piperidin-1-yl-N-[4-(trifluoromethoxy)phenyl]-1H-pyrimidine-4-carboxamide N-ethyl-1'-(oxan-4-yl)spiro[7,8-dihydroimidazo[2,1-c][1,4]benzoxazine-6,3'-pyrrolidine]-2-carboxamide;2,2,2-trifluoroacetic acid 2-[3-(3,4-dichlorophenyl)cyclopentyl]oxyacetic acid 1-butan-2-yl-7,8-dimethoxy-4H-chromeno[3,4-c]pyrazole (3R)-4-ethyl-5-hydroxy-N-(2H-triazol-4-ylmethylsulfanyl)-7-oxaspiro[4.4]nonane-3-carboxamide 3-hydroxy-4-methyl-5-[(1E)-1-(5-methylidenecyclopenta-1,3-dien-1-yl)buta-1,3-dien-2-yl]thiophene-2-carboxylic acid N-ethyl-3,5-dimethoxy-2-methylbenzenesulfonamide N-[(2S)-1-cyclopropyl-4-methoxybutan-2-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxamide 2-(3,5-dimethylpyrazol-1-yl)-7H-purine 3-[(Z)-2-ethyl-6-fluorohex-1-enyl]-4,7-dihydroxy-5H-chromen-2-one 2-[2-(6,7-dichloroquinoxalin-5-yl)oxyethoxy]benzonitrile 1-(3-aminopropylamino)anthracene-9,10-dione 5-(2,5-dichlorophenyl)-4-(2-ethoxyphenyl)-N-(4-methyl-3-nitrophenyl)-1,3-thiazol-2-amine 2-methyl-4,5-diphenyl-6H-[1]benzofuro[3,2-e]indole N-butanoyl-2,3,4,5,6-pentafluorobenzenesulfonamide 6-[2,4-bis(trifluoromethyl)phenyl]-N-[5-chloro-1-(1H-imidazol-5-ylmethyl)pyrazol-3-yl]pyridine-3-carboxamide (Z)-2,3-dichloro-4-[(2E,5S)-2,6-dimethylocta-2,6-dienoxy]imino-2-phenylbut-2-enoic acid N-[2-(dimethylamino)ethyl]-2-(1H-indol-3-yl)-5-oxopentanamide 4-[3,5-dichloro-2-methoxy-6-(trifluoromethyl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile N-(4,5-dihydro-1H-imidazol-2-yl)-N-[3-(dimethylamino)propyl]-6-methoxy-5-nitropyridine-3-carboxamide N-[5-(2-azidoethynyl)pyridin-3-yl]-2,6-difluorobenzamide 4-[(2,5-dimethoxyphenyl)methylideneamino]-3-[(E)-furan-2-ylmethylideneamino]benzenesulfonamide 5-[[2-methoxyethyl(naphthalen-1-yl)amino]methyl]furan-3-carboxylic acid 1,3-bis(4-ethenoxybutyl)benzene 1-chloro-2,6-difluoronaphthalene N-[(1R)-2,4-dihydropyrano[3,2-c]pyridin-1-yl]benzamide 5-bromo-4-tert-butyl-2-(1,1,1-trifluoropropan-2-yl)-1H-pyrimidin-6-one [5-tert-butyl-2-methoxy-3-(trifluoromethyl)phenyl]-methylidyneazanium (E)-3-[4-(5-propan-2-yl-1,4-dihydropyrrolo[2,3-d]pyridazin-6-yl)phenyl]-N-(2,2,2-trifluoroethoxymethyl)prop-2-enamide N-[5-(7-bromoquinolin-4-yl)oxypyridin-2-yl]acetamide 5-[1-(2,3-dichlorophenyl)sulfonyl-6-fluoroindol-4-yl]pyrimidin-2-amine 2-[1-[3-(2,5-dichloropyridin-4-yl)-4-oxophthalazin-1-yl]butoxycarbonylamino]acetic acid N'-[4,5-dichloro-2-(3,5-dimethylphenoxy)phenyl]methanimidamide 2-[1-(diethylamino)propyl]-4-(pyridin-3-ylmethoxy)benzenediazonium 1-[4-(benzenesulfonyl)piperazine-1-carbonyl]-3,4-dihydroquinolin-2-one [3-(3,5-dimethyl-1H-pyrazol-4-yl)morpholin-4-yl]-(2,4-difluoro-6-methoxyphenyl)methanone 1-[3-(hydroxymethyl)piperidin-1-yl]-2-pyridin-4-ylethanone 1-(difluoromethyl)-3-[4-[2-[4-(4-pentan-2-ylidenecyclohexyl)phenyl]ethynyl]phenyl]benzene 2-azido-5,6-difluoronaphthalene (3E)-6,8-dimethoxy-3-[5-oxo-2-sulfanylidene-1-[4-(trifluoromethylsulfonylamino)phenyl]-3H-pyridin-4-ylidene]chromene-7-carboxylic acid N-(3,4,5-trifluorophenyl)furan-2-carboxamide 2-azido-4,5-dimethylthieno[3,2-b]thiophene 3-[[5-chloro-4-(methoxymethyl)pyrimidin-2-yl]amino]benzonitrile 3-azido-2-[(1S)-2,3-dihydro-1H-inden-1-yl]furan 5-azido-2,3-dihydrothieno[3,4-b][1]benzothiole 2-(2,4-dimethylphenyl)sulfonyl-N'-(2,5-dioxopyrrol-3-yl)-2-ethoxybutanehydrazide 2-[4-(7H-purin-6-yl)piperazin-1-yl]ethanol N-[2,4-dichloro-3-(5H-pyrrolo[2,1-c][1,2,4]triazol-7-yl)cyclohexa-1,3-dien-1-yl]oxybenzenesulfonamide 1-(1,3-benzodioxol-5-ylmethyl)piperazine;2,4-bis(2-fluorophenyl)pyrrole 6-(azidomethyl)-1,3-dihydroindol-2-one 4-[3-(2,5-dioxopyrrolidin-1-yl)propanoylamino]benzenesulfonic acid N-[2-(3,4-dichlorophenyl)propyl]-5-ethyl-6H-1,3,4-thiadiazin-2-amine 3-[4-[[4-hydroxy-1-methyl-5-oxo-2-(1,1,3-trioxoisoindol-2-yl)pyrazol-3-yl]diazenyl]phenyl]benzoic acid 2-[(1R)-5,6-difluoro-3-methyl-2,3-dihydro-1H-inden-1-yl]-4-fluoroaniline 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;6-ethyl-8-fluoro-4-(methyliminomethyl)-2H-isoquinolin-1-one 1-[6-(2-bromoethyl)imidazo[4,5-b]pyridin-3-yl]propan-2-one 2-[5-bromo-2-[(Z)-[4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazolidin-5-ylidene]methyl]phenoxy]acetic acid (2R)-3,4-difluoro-1-phenylmethoxycarbonylpyrrolidine-2-carboxylic acid ethane;2-(4-methylphenyl)sulfonyloxyacetic acid 2-[(2,6-dichlorobenzoyl)amino]-3-[5-[4-[ethoxycarbonyl(sulfino)amino]piperidine-1-carbonyl]pyridin-2-yl]propanoic acid (2-amino-4,5-diethoxyphenyl)-[1-(6-chloroquinazolin-8-yl)piperidin-4-yl]methanone 2-[(4S,5R)-5-acetyl-3-methylideneoxolan-2-yl]-N-[(2-chlorophenyl)methyl]-6-fluoropyrimidine-4-carboxamide 4-[2-(5-methyl-1H-indol-3-yl)ethylideneamino]cyclohexa-2,5-diene-1-carboxylic acid 3-azidooxy-2,4-dipropylphenol 6-ethylsulfonyl-3-methoxycarbonylbenzoic acid 6-[(E)-1,2-dibromoethenyl]pyridine-3-carbonitrile 1-benzyl-2-[(1R,5S)-3-bicyclo[3.2.0]heptanyl]imidazole (7R)-7-[2,3-dichloro-6-(hydroxymethyl)phenyl]-4,5,9,13-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-triene-8,10-dione 1-(5-amino-4-chlorothiophen-2-yl)sulfonylpiperidine-4-carboxylic acid 2-[[5-chloro-3-methyl-1-(4-pyrimidin-2-yloxycyclohexanecarbonyl)indol-7-yl]amino]ethanimidate (2-methylsulfonylpyrrolidin-1-yl)-[6-methylidene-3-[4-(trifluoromethoxy)phenyl]pyridazin-1-yl]methanone 2-[(4,6-dimethoxy-1H-indole-2-carbonyl)amino]-9-(5,6,7,8-tetrahydroquinolin-3-yl)nonanoic acid N-(2,3,4-trichlorophenyl)carbamate 2-[3-[6-(4-aminobutyl)pyridin-3-yl]phenyl]propan-1-amine 2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)-3H-thieno[3,2-d]pyrimidin-4-one 1-[5-(3,4-dimethoxyphenyl)pentyl]piperidine 4-chloro-2,3,5-trimethylbenzenesulfonate 2-(1,3-dihydrobenzo[de]isoquinolin-2-yl)acetonitrile 4-(2,3,6,7-tetramethyl-4H-benzo[d][1]benzazepine-5-carbonyl)oxane-4-carboxylic acid 5-[2,4-bis(trifluoromethyl)phenyl]-2-propan-2-ylpyrazole-3-carboxylic acid 5-methyl-N-[2-(oxolane-3-carbonylamino)ethyl]thiophene-2-carboxamide 3,4-difluoro-5-[2-(methoxymethyl)pyrrolidine-1-carbonyl]benzoic acid;hydrochloride 3-[(4-methoxyphenyl)methyl]-1H-indole N-[3-chloro-5-(2,4-dimethylphenyl)sulfanylpyridin-2-yl]-4-methoxypyridine-2-carboxamide [2-(1,3-benzodioxol-5-ylmethoxy)naphthalen-1-yl]hydrazine;ethane [6-(2-aminopyrimidin-5-yl)-1H-pyrrolo[3,2-c]pyridin-4-yl]methanol (Z)-2-[3,5-bis(trifluoromethyl)phenyl]-3-[7-[(3,4,5-trimethoxybenzoyl)amino]heptan-2-yl]prop-2-enoic acid 1-(4-ethenoxyphenyl)sulfonylpiperidine N-[(Z)-3,5-dimethylhex-2-en-4-yn-2-yl]-1-phenyl-4-propanoylpiperidine-4-carboxamide N-ethyl-3-(2-methylpiperidine-1-carbonyl)benzamide 1-[5-chloro-6-fluoro-2,3-dimethyl-4-(6-methylidene-7H-pyrrolo[2,3-d]pyrimidin-3-yl)phenyl]ethanone;propane 7-[4-(3,5-dichloro-N-methylanilino)phenoxy]thieno[2,3-b]pyridine-5-carbonitrile 4-cyclopropyl-5-iodo-2-(1H-pyrazol-5-yl)-1,3-thiazole 2-[(2,3,4,5-tetrahydroxybenzoyl)amino]-1,3-thiazole-4-carboxylic acid N-butyl-2,4-dinitro-N-(2-phenylethyl)aniline 3-(methylamino)-6-[4-(trifluoromethyl)phenyl]sulfanylquinoline-2-carboxylic acid 5-bromo-2-(difluoromethoxy)quinoline N-[2-(5-phenyltetrazol-1-yl)ethyl]-4,6-dihydropyrrolo[3,4-d][1,3]thiazole-5-carboxamide N-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-7-carboxamide 2-[(3R)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]pyrrolidin-3-yl]oxypyridine 4-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyrimidine [4-[[(3R)-1-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridine-7-carbonyl)piperidin-3-yl]amino]piperidin-1-yl]-phenylmethanone (6-fluoro-2,3-dihydroindol-1-yl)-[4-[3-(6-methoxypyridin-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl]methanone 4-(azidomethyl)-2,3,5,6-tetrafluorobenzonitrile 3-(2,6-dichlorophenyl)sulfanyloxypentan-1-ol (3-methyl-2,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-4-yl)-pyrrolidin-1-ylmethanone (E)-N-methyl-3-[4-[4-(4,4,5,5-tetrafluoropentoxy)benzoyl]phenyl]prop-2-enamide [3-(cyclopropylmethyl)morpholin-4-yl]-[6-(ethoxymethyl)imidazo[1,2-b]pyridazin-3-yl]methanone 3-[(1R)-1-fluoroethoxy]benzoic acid 2-(4-methoxypyridine-3-carbonyl)-9-phenyl-6-oxa-2,9-diazaspiro[4.5]decan-8-one N-[(2R)-1-hydroxypropan-2-yl]benzamide N-(2,5-dimethylphenyl)-6-[4-(piperidine-1-carbonyl)pyrazol-1-yl]pyridine-3-carboxamide 1-[2,3-bis(trifluoromethyl)phenyl]-2,4-dihydroxy-6-oxopyrimidine-5-carbonitrile 5-[2-(5,5-dimethyl-1,3-dioxan-2-yl)ethynyl]-2-[2-fluoro-4-(trifluoromethoxy)phenyl]pyridine ethane;[4-(2,4,6-trimethylphenyl)pyrimidin-5-yl]boronic acid (E)-3-[5-tert-butyl-2-(methanesulfonamido)phenyl]-N-[4-chloro-3-[[3-oxo-3-[4-(trifluoromethoxy)phenoxy]propyl]amino]phenyl]prop-2-enamide N-[(3R)-3-[(2-acetyl-6,7,8,9-tetrahydro-5H-carbazol-4-ylidene)amino]pentan-3-yl]benzamide 2-(2,4-dichlorophenyl)-6-[4-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]phenyl]pyridine N-benzyl-1-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)phenyl]pyrazole-3-carboxamide;hydrochloride 4-N-(2-chloropyridin-3-yl)benzene-1,4-disulfonamide 2-[4-methylsulfanylbutyl(propyl)amino]-1H-benzimidazole-4,5-dicarbonitrile 2-azido-6-benzyl-5-methoxy-1,3-benzothiazole 2-[3,5-bis(trifluoromethyl)phenyl]-1,6,7-trimethoxy-N-pyridin-3-ylphthalazin-4-amine ethane;3-[2-(4-methoxyphenyl)cyclohexen-1-yl]-N,5-dimethylbenzenesulfinamide N-(cyclopentylmethyl)-2,4-difluoroaniline 2-N,3-N-bis(1H-indol-3-ylmethylideneamino)thiophene-2,3-dicarboxamide 6-benzyl-2,3,4,9a-tetrahydrocarbazole 4-hydroxy-1-methyl-5-[(2R)-2-(6-nitro-1H-indole-3-carbonyl)cyclopenten-1-yl]pyrrole-2-carboxylic acid 1-chloro-2,3-diethylbenzene;N'-[2-(cyclobutanecarbonylamino)pyridin-4-yl]-N,N-dimethylmethanimidamide 2,3-dibromo-4,6-bis(2-methylpropoxy)phenol (2S)-N,3-dimethyl-2-[(4-propoxyphenyl)sulfonylamino]butanamide 1-[3-(ethylideneamino)-2-(3-methylbutan-2-yloxy)phenyl]propan-1-one 2-(3,4-dimethoxyphenyl)-N-[(3S,7R,8aS)-3-(2-hydroxyethyl)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]acetamide (6R,7R)-3-[[5-(dipropylcarbamoyloxymethyl)-1H-indole-2-carbonyl]amino]-8-oxo-7-[(2-phenylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-[[2-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonylamino)phenyl]acetyl]amino]oxolane-3-carboxamide N-[2,3-dihydroxypropyl(3-methylbutyl)amino]benzenesulfonamide (2R,3S)-N'-cyclohexyl-6-methoxy-2,3-dihydroxy-4-oxochromene-8-carbohydrazide 1-N,4-N-bis(3-iodophenyl)benzene-1,4-dicarboxamide 1,2-diphenyl-6-(trifluoromethyl)-4H-pyrimidine;N'-(4-methoxyphenyl)methanediamine 1-azido-2-(4-methylphenyl)sulfanylpiperazine 7-bromo-4,8-dichloro-1H-3-benzazepine 6-N,4-N,6-trimethyl-2-N-[4-(3-phenylmethoxyphenoxy)cyclohexa-1,5-dien-1-yl]pyrimidine-2,4,6-triamine 4-[2-ethyl-5-(1,1,3-trifluoropropoxy)phenoxy]-7-methoxyquinoline 3-chloro-N-(4,6-dimethylpyrimidin-2-yl)pyridine-2-carboxamide (Z)-3-hydroxy-2-[5-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-3-yl]but-2-enenitrile N-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-methoxy-5-pyridin-4-ylbenzamide (3R)-4-[2,6-dimethyl-3-(2-methylpropoxycarbonylamino)benzoyl]-3-methylpiperazine-1-carboxylic acid 4-(4-ethoxy-3,5-dimethylphenyl)pyridine 2-(4-cyclohexyloxyphenyl)-3,7-dihydroindole N-[4-(2,5-dimethylphenyl)pyrimidin-2-yl]acetamide 1-benzyl-4-(2,4-dichlorophenyl)sulfanylpyridin-1-ium 4-[4-[6-[3-(diethylamino)azetidine-1-carbonyl]pyridin-2-yl]piperazin-1-yl]benzonitrile 5-[2,3-dichloro-4-(trifluoromethoxy)phenyl]-1H-indole 2-amino-N'-(4-methylphenyl)benzenecarboximidamide 5-[(Z)-3,4-dihydroxyhept-2-en-2-yl]-1-methylpyrazole-3-carboxylic acid N-[(Z)-1-amino-3-hydroxy-4,4-dimethylpent-2-enylidene]-3-cyclohexyloxy-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)thiophene-2-carboxamide 1-azido-2-(3,4-difluorophenyl)-4-methoxybenzene N-[3-bromo-7-methoxy-4,5-bis(phenylmethoxy)naphthalen-2-yl]acetamide N-methyl-2,3-dihydro-1H-pyrrolo[2,1-b]quinazoline-5-carboxamide 6-(azidomethyl)-3,4-dichloro-1H-quinolin-2-one 2-azido-3,5-diethyl-4-hydroxybenzenecarboximidamide 2-(1,3-benzoxazol-5-yl)-4-cyclopropyl-1H-pyrimidin-6-one 6-butyl-2,4-bis(4-methoxyphenyl)pyridine-3-carboxylic acid N-[(4-methylpyridin-2-yl)-phenylmethyl]benzamide 3-(1H-pyrrolo[2,3-b]pyridine-3-carbonyl)hexanoic acid 2-(4,4-dichlorobutoxy)-6-(trifluoromethyl)pyridine 3-(dipropylamino)benzamide N-butylsulfanylpyrimidin-2-amine 4-N-[5-methyl-4-(1-propylbenzimidazol-2-yl)pyridin-2-yl]cyclohexane-1,3-diamine [3-(oxan-4-yl)phenyl]methanesulfonamide 3-(dimethylamino)propane-1,2-disulfonic acid;ethane 7-methylsulfonylquinazoline (3S)-1,3-dimethyl-5-[2-[5-[3-(oxan-4-yloxy)propyl]pyridin-2-yl]ethynyl]-3H-indol-2-one 2-tert-butyl-3-ethoxy-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-N-(diaminomethylidene)benzamide 3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)cyclohexan-1-one 2-azidosulfanyl-4-(1,2,3,4-tetrahydronaphthalen-2-yl)-5H-pyrrolo[3,2-d]pyrimidine N-(3,4-dihydro-2H-chromen-4-yl)-2-methyl-N-(pyridin-3-ylmethyl)pentanamide 4-[2-(3,5-dimethylphenyl)iminoethanehydrazonoyl]benzenecarboximidamide ethane;8-[5-fluoro-6-(3,4,4-trifluorobutyl)pyridine-2-carbonyl]-7H-pyrazino[2,3-d]pyrimidin-6-one 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-hexadecylamino]benzenesulfonic acid N-[4-[3-(difluoromethyl)pyrrolidine-1-carbonyl]phenyl]-6-methoxy-1,2,3,4-tetrahydroacridine-9-carboxamide 2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-7-ethylsulfonylspiro[6,8-dihydropyrrolo[2,1-c][1,2,4]triazine-5,3'-oxetane]-1'-one 2-(4,5-dimethylfuran-3-carbonyl)-9-[(3-fluorophenyl)methyl]-6-oxa-2,9-diazaspiro[4.5]decan-8-one N-[(Z)-1H-benzimidazol-2-ylmethylideneamino]-4-(piperidin-1-ylmethyl)benzamide;hydrochloride 4-(4-chlorophenyl)-2,3,5-trimethylthiophene N-[(E)-[1-cyclohexa-2,4-dien-1-ylsulfonyl-5-hydroxyindol-3-yl]methylideneamino]-5-nitropyridine-2-carboxamide 1-[5-tert-butyl-2-(1,3-dioxoisoindol-2-yl)phenyl]-N-diazomethanesulfonamide 3-N-[2-(cyclopropanecarbonyl)-7,7-diethyl-3,4-dihydropyrano[4,3-c]pyrazol-5-yl]benzene-1,3-dicarboxamide 2-methylsulfinyl-5-propan-2-yl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine (2S)-3,4-dimethyl-2-[(5S)-4-oxo-2-propanoyl-6-phenyl-5H-pyrrolo[1,2-b]pyridazin-5-ium-5-yl]pentanoic acid 2-[4-[(2S)-4,5-dimethoxyheptan-2-yl]oxyphenyl]acetic acid 2-(azidomethyl)-5,6-dichlorobenzimidazole 2-[5-(3-cyclobutylphenyl)pyrimidin-2-yl]propan-1-imine;methanamine N-benzyl-1,3-thiazolidin-2-imine;hydrobromide 5-[(Z)-1-amino-3-methyliminoprop-1-en-2-yl]-N'-hydroxypyridine-2-carboximidamide;ethane ethane;N-[2-(3-fluorophenyl)phenyl]formamide N-cyclopropyl-5-(4,4-difluoro-3-methoxypiperidine-1-carbonyl)pyrazine-2-carboxamide N-[1-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)piperidin-4-yl]-2-fluorobenzamide [2-(6-aminopyridin-3-yl)-4,5,7,8-tetrahydro-1H-pyrazolo[3,4-d]azepin-6-yl]-(3,6-dichloroimidazo[1,2-b]pyridazin-7-yl)methanone 2-(dimethylamino)-1',3',6'-trihydroxyspiro[isoindole-3,9'-xanthene]-1-one 1-[(3R,4S)-3-hydroxypiperidin-4-yl]-5-thiophen-2-ylpyrazolo[3,4-c]pyridine-7-carboxamide;hydrochloride 2-(2,3-dimethoxyphenyl)-7H-purine N-[(3S)-8,10-difluorodecan-3-yl]benzenesulfonamide 5-[8-(dimethylamino)-2,3-bis(ethenyl)-4-ethoxybenzo[e]indol-1-ium-1-ylidene]pentanoic acid 1-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]benzimidazole;hydrochloride (2R)-1,3-bis[(3-methoxyphenyl)methyl]-4-oxoazetidine-2-carboxylic acid 2-bromo-N-(2,6-dichloro-4-nitrophenyl)-N-[4-[2-(oxolan-2-ylmethylamino)-1,3-thiazol-4-yl]phenyl]benzamide N-[3,4-difluoro-2-(2-fluoro-6-methylphenyl)phenyl]acetamide 4-methoxy-1-(5-phenylhexyl)benzimidazole N-(1-aminoethyl)-4-[[3-[2-[3-aminopropyl(methyl)carbamoyl]phenyl]-5-fluoroanilino]-hydroxymethoxyphosphoryl]oxypentanamide [2-(3,4-dihydropyridine-2-carbonyl)phenyl]-oxo-sulfidoazanium 2-azido-N,3-dimethyl-1H-imidazo[4,5-b]pyridine-6-carboxamide 2-[(4R)-1-benzhydryl-3-methylideneazepan-4-yl]benzenesulfonate 3-chloro-5,6,7,8-tetrafluoro-9H-fluoren-1-amine N-[(3Z)-4-methylidene-5,6-dioxohepta-1,3-dien-2-yl]-4-phenoxybenzamide 1-benzyl-3,4-dinitro-2H-imidazole 5-hydroxy-N'-[4-(2-methoxyphenyl)sulfanylthieno[3,2-d]pyrimidin-6-yl]thiophene-2-carboximidamide 5-[2,3,4-triethoxy-6-(methylamino)phenyl]pentanal 2-benzyl-2,4-dimethoxy-N-methylbutanamide 4-tert-butyl-2-[(1S)-2-phenylcyclopropyl]-1,3-oxazole 3-fluoro-5,6,8-trihydroxynaphthalene-2-carboxylic acid 3-hydroxy-4-[2-[2-(4,6,7,8-tetrahydrofuro[3,2-c]azepin-5-yl)ethoxy]ethyl]pyrrolidine-1-carboxylate (2S)-2,5-bis[2-chloro-4-(3,3-difluorocyclobutyl)phenyl]pyrrolidine-1,2,3-trione 4-(2,3-dihydrothieno[3,4-b][1]benzofuran-1-yl)phenol (E)-N,4,5-trimethyl-6-oxo-2-[(2R)-1-phenyl-3-pyrrolidin-1-ylpropan-2-yl]hept-2-enamide (3-chlorophenyl)-[4-(trifluoromethoxy)phenyl]phosphane 4-[3,6-bis(sulfanylidene)-2H-1,4-benzoxazin-7-yl]-2-methoxy-N,N-dipropylbenzamide N'-[(E)-(6-oxo-2-phenylcyclohexa-2,4-dien-1-ylidene)methyl]methanimidamide N-[(3R,4S)-1-methyl-4-(2-oxo-3H-1,3,4-thiadiazol-5-yl)pyrrolidin-3-yl]pyrazine-2-carboxamide (4R)-1,5-dimethyl-3,4-bis(phenylmethoxy)-6-[3-(trifluoromethyl)phenyl]-3a,6a-dihydropyrrolo[3,4-c]pyrrole-2,7-dione 2-bromo-5,6-dimethoxy-3H-thieno[3,2-d]pyrimidin-4-one (6S)-2,2-diethyl-9-[4-[4-[1-methoxy-6-(4-methoxyphenoxy)hexan-3-yl]phenoxy]butoxy]-6-(phenylmethoxymethyl)-5,6-dihydro-4H-triazolo[1,5-a][2,7]naphthyridine N-ethenylmethanimine;4,5-dihydro-1H-imidazo[2,1-c][3]benzazepine 6-chloro-3-[2-(4,6-dimethylpyrimidin-5-yl)iminopropyl]-1H-indol-2-ol 2-(2,2-dimethylcyclopropyl)-5-fluoro-3H-quinazolin-4-one N-[2,4-dimethyl-6-(3-morpholin-4-ylpropyl)phenyl]-5-fluoropyridine-3-carboxamide (2S)-2-[3-fluoro-4-(methanesulfonamido)phenyl]-1,4-oxazepane-4-carboxylate 5-(2,3-dimethylpentan-2-ylamino)-N'-hydroxypyrazine-2-carboximidamide N'-[4-[(3,5-dichlorophenyl)methoxy]-2-fluorophenyl]oxamide [5-chloro-3-(pyridine-2-carbonyl)quinolin-8-yl]methanediol 1-benzyliodanuidyl-3-[(2R,4S)-1-cyclohexyl-4-[(3-methoxyphenyl)methoxy]pentan-2-yl]urea 1-(5-azidopentoxy)naphthalene 3-(2,5-dimethylpyrrol-1-yl)-N'-hydroxypyridazine-4-carboximidamide 1-[5-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)furan-2-yl]ethanone 1-(2,2-difluoropropyl)-4-[3-(trifluoromethoxy)phenyl]sulfonylbenzene 2-[(E)-3,4,5-trimethylhex-1-enyl]phenol 5-[6-(3,4-dimethylphenyl)naphthalen-2-yl]-2H-triazole-4-carboxylic acid 2,2-difluoropropanal;4-N-methyl-6-(2-phenylethoxy)-2-N-prop-1-en-2-ylpyridine-2,3,4-triamine 5-amino-N-[4-(cyanomethyl)phenyl]pyrazine-2-carboxamide 2-(1,3-benzoxazol-5-yl)-N-[4-(3H-benzimidazol-5-ylamino)pyrimidin-2-yl]acetamide 1-[(Z)-(5-chloro-2-hydroxyphenyl)methylideneamino]-3-methylthiourea 2-(benzenecarboximidoyl)-4,6-dimethylaniline (3-aminophenyl)-phenylmethanol N'-[2,5-dimethyl-3-(4-methylphenyl)sulfinylphenyl]-N,N,N'-trimethylpropane-1,3-diamine 4-ethyl-5-(3-hydroxyphenyl)thiophene-2-carboxylic acid 4-(6,8-dichloro-2-sulfanylidenechromene-3-carbonyl)piperazine-1-carboxylic acid 5-[(E)-1,2-difluoro-2-phenylethenyl]-6-ethyl-4-[4-(3-piperidin-1-ylpropoxy)phenyl]pyrimidin-2-amine 3-[2,3-bis(methylsulfonyl)phenyl]-2-oxopropanoic acid 2-(5,7-difluoro-1H-indole-3-carbonyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-hydroxybutanamide 2-[(4,5-dimethyl-1H-imidazole-2-carbonyl)amino]spiro[3.3]heptane-6-carboxylic acid 3-[4-methoxy-2-(trifluoromethyl)phenyl]propan-1-amine 1-[2,4-difluoro-6-(5-pentylpyrimidin-2-yl)phenyl]cyclobutan-1-amine 1-[2,3-dihydroxypropyl(phenacyl)amino]propan-2-one N-[3,5-dichloro-4-(6-methoxyquinolin-4-yl)oxyphenyl]-1-(2-hydroxyethyl)cyclopropane-1-carboxamide (4R)-3-[hydroxy(phenylmethoxycarbonylamino)methyl]piperidine-1-carboxylic acid 1-[4,5-bis(trifluoromethyl)pyrimidin-2-yl]-N,N-diethylpiperidine-3-carboxamide [(3aR,8aS)-2-[[4-fluoro-6-methoxy-7-[1-(trideuteriomethyl)cyclopropyl]-1H-benzimidazole-2-carbonyl]amino]-1-oxospiro[5,6,8,8a-tetrahydroimidazo[1,5-a]pyrazine-3,4'-oxane]-7-ylidene]oxidanium N-(5-fluoro-1H-indazol-3-yl)piperidine-4-carboxamide N-[(1R)-5,6-difluoro-2,3-dihydro-1H-inden-1-yl]-4-hydroxy-2-oxopyrrolidine-3-carboxamide 2-[4-[[(1S)-1,3-diphenylpropyl]amino]-6-oxo-1H-pyrimidin-2-yl]sulfanyl-N'-(2,2,2-trifluoroacetyl)benzohydrazide N-methyl-4-[2,3,7-tris(sulfanylidene)azepane-1-carbonyl]benzamide 3-[4-[[2-(1H-indazol-6-ylamino)pyrrolo[2,1-f][1,2,4]triazin-4-yl]methyl]piperazin-1-yl]propanoic acid 3-hydroxy-5-phenyldiazenylnaphthalene-2,7-disulfonic acid 1-(2,4-dichlorophenyl)sulfonylpiperidine-3-carbonitrile 2-(4-cyanophenoxy)benzenesulfinate 6-[4-(2-aminoethoxy)-3,5-difluorophenyl]-N-cyclopropylsulfonyl-1-methylpyrazolo[3,4-b]pyridine-4-carboxamide 4-[5-(2,6-difluorophenyl)-3-oxopentanoyl]morpholine-3-carbonitrile (2-iodophenoxy)-[4-methyl-2,6-dinitro-3-[(E)-3-phenylprop-2-enoxy]benzoyl]phosphinic acid 2-[(5S,10bR)-9-chloro-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol [4-[3-[4-(1,3-benzothiazol-2-yl)phenyl]propoxymethyl]phenyl]phosphane;2-[4-[(2Z,5E)-octa-2,5,7-trienyl]piperazin-1-yl]ethanamine 7-amino-6-(2-methoxyphenyl)sulfanyl-5,6,7,8-tetrahydronaphthalene-1,3,4-tricarbonitrile 2-methylsulfinyl-1,3-benzothiazole 2-[(3S,7R)-6-[4-chloro-3-[[4-(1H-pyrazol-5-yl)phenyl]methyl]phenyl]-2-oxo-8-oxa-3,4-diazabicyclo[4.2.0]octan-3-yl]acetaldehyde;ethane 1-[4,5-difluoro-2-(hydroxymethyl)phenyl]-3-[4-(triazol-1-yl)butanoylamino]urea 1-(3,5-dimethylpyrazol-1-yl)-2,2-bis(hydroxyimino)ethanone N-(8-bromoquinoxalin-5-yl)-N-ethenylsulfonylbenzamide 5-chloro-6-[2-[(Z)-1-methoxybut-1-enyl]iminocyclopentyl]naphthalene-1,3-dione 4-azido-N-[3-chloro-2-fluoro-6-(trifluoromethyl)phenyl]benzenesulfonamide 3-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-piperidin-4-yl-1H-indole;hydrochloride 1-[3-(4,7-dichloroquinolin-2-yl)phenoxy]ethanol;1-methylpiperidine N-(2,4-dioxopentan-3-yl)-3-oxobutanamide;2-[(Z,2E)-2-ethylidenehex-3-enyl]aniline 2-[3-fluoro-4-methyl-5-(trifluoromethyl)phenyl]acetic acid 5-[3-(cyclopropylmethoxy)-4-fluorophenyl]-1H-indazole 1-amino-3-ethoxycarbonylindazole-5-carboxylate N-(1,3-dioxoisoindol-2-yl)carbamate 3-(1H-pyrrole-2-carbonylamino)propanoic acid;hydrate 7-(2,3-difluorophenyl)-1-methyl-8-(5-propan-2-yl-1H-pyrazol-4-yl)pyrido[3,4-b]indole 4-bromo-1-iodo-3,5-dimethylpyrazole [5-(5-bromo-2,3-dihydro-1H-pyrazol-4-yl)pyridin-3-yl]boronic acid 4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperazine-2-carbonitrile 2-[5-(aminomethyl)-1,2,4-oxadiazol-3-yl]-3H-indol-5-ol 3-(2,4-dichlorophenyl)-3H-pyrrole 7-phenyl-N,4,5,6,7,8-hexahydrocyclohepta[d]triazol-3-amine 4-[3,5-bis(2-phenylethynyl)thiophen-2-yl]-1,4-diazepane 2-[[4-[(3E,5Z)-7-chlorohepta-1,3,5-trien-4-yl]phenyl]methoxy]ethanol (Z)-4,4,5-trimethyl-1-(6-methylidenecyclohexa-2,4-dien-1-yl)-3-phenylpent-2-en-1-imine N-[3-[3-(4-methylphenyl)phenyl]propylidene]hydroxylamine 3-(3,4-dihydroxyphenyl)-1-phenylpropan-1-one 2-[1-hydroxy-4-(5,6,7,8-tetrahydroquinolin-4-ylmethoxy)cyclohexyl]-N-[2-[3-(trifluoromethoxy)phenyl]ethyl]acetamide [4-(azidomethyl)piperidin-1-yl]-phenylmethanone N-ethyl-N'-[(2S)-2-(4-ethylphenyl)-1,3-dihydropyrrolo[3,2-b]quinolin-7-yl]-N'-methylpropane-1,3-diamine 2-(4-azidophenyl)-6,7-dimethoxy-3H-quinazolin-4-one 3-(2,2-dimethylpropanoyl)-7-fluorochromen-2-one 4-[3-(cyclopropylmethoxy)-4-fluorophenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 4-[3-(aminomethyl)phenyl]-2H-phthalazin-1-one N-[3-[5-ethenyl-4-(methylideneamino)-6-(pyrrolidine-1-carbonyl)pyridin-2-yl]prop-1-en-2-yl]-4,5-dihydrofuro[3,2-d][1]benzazepine-2-carboxamide N-azido-N-(benzenesulfonyl)carbamate 2-[5,6-difluoro-1'-(5-fluoropyridin-3-yl)spiro[2H-indole-3,4'-piperidine]-1-yl]-N,N-dimethylacetamide;formic acid 1-[4-(2,6-dimethylpyridin-3-yl)piperazin-1-yl]-4-[4-[2-ethoxypropyl(methyl)amino]piperidin-1-yl]butan-1-one 6-[2,6-dichloro-4-(4-propan-2-ylpyrazole-1-carbonyl)phenyl]-8-methoxypyrido[3,4-d]pyridazin-5-one 3-(4,5-dimethylthiophene-2-carbonyl)pyridine-2-carboxamide 1-[(3-methylpyridin-4-yl)methyl]spiro[2H-pyrrolo[3,2-b]pyridine-3,3'-oxetane] 6-bromo-1,4-dimethylpyrrolo[3,2-c]pyridine 4-[(1E)-1,2-diphenylpenta-1,4-dien-3-yl]aniline 3-benzyl-6,7-dihydro-4H-[1,2]oxazolo[5,4-c]pyridine;hydrochloride 2-[2,4-dioxo-1-propyl-5-(trifluoromethyl)pyrimidin-6-yl]sulfanyl-N-[5-(4-methoxyphenyl)pyridin-3-yl]acetamide 1-azido-3-methyldibenzothiophene (7R)-3-(4,5-dihydropyrimidin-2-yloxymethyl)-9-ethyl-8-[4-fluoro-2-(trifluoromethyl)phenyl]-7H-imidazo[1,2-f]purin-6-one N-[(2S)-1-oxo-3,4-dihydro-2H-pyrazino[1,2-a]indol-6-yl]carbamate 1-[1-(1,3-dioxoisoindole-2-carbonyl)azetidin-3-yl]-N-[[4-(trifluoromethoxy)phenyl]methyl]triazole-4-carboxamide 2-[(3R)-1-(cyclopropanecarbonyl)piperidin-3-yl]-6-(thiophen-2-ylmethyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (E)-N-[2-(4-chlorophenyl)ethyl]-3,3-dimethoxy-1-(1H-pyrrol-2-yl)prop-2-en-1-imine 2-amino-N'-(2,5-dichlorophenyl)-2-[4-(3-hydroxypropoxy)cyclohexyl]ethanimidamide (1S)-3-methylsulfonyl-4-azatricyclo[6.2.0.02,7]decane 5-[2-(2,3-dihydro-1H-inden-4-yl)ethynyl]-N-methylpyridine-2-carboxamide N-[(2S)-1-ethoxy-4,4-dimethylpentan-2-yl]-3-pyrazol-1-ylpyrrolidine-1-carboxamide 2-(cyclohexen-1-yl)-7-[(4,5-dimethoxythiophen-3-yl)methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 4-tert-butyl-1-[2,5-difluoro-3-(trifluoromethyl)phenyl]triazole 2-tert-butyl-5-(6,8-dihydrothieno[3,2-c]pyrrole-5-carbonyl)-7-methyl-4H-1,4-benzoxazin-3-one N-(6-bromopyridin-3-yl)benzenesulfonamide 3-(2-hydroxyethoxy)-5-methylbenzenesulfonic acid ethane;N-[[3-methyl-6-(2,4,5-trifluorophenyl)imidazo[1,2-a]pyridin-2-yl]methyl]formamide 2-[3-chloro-4,5-dimethoxy-N-[(4-nitrophenyl)carbamoyl]anilino]acetic acid 3-[(3,5-dichlorophenyl)sulfanylmethyl]-5-[3-(trifluoromethyl)pyrazol-1-yl]pyridine 5-[2-(methylamino)ethyl]-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one (2R,3S)-N-cyclopropyl-2-(methoxymethyl)-5-oxo-1-[2-phenyl-4-(trifluoromethyl)benzoyl]pyrrolidine-3-carboxamide 6-(dimethylsulfamoylamino)pyridine-2,3-dicarboxylic acid 5-(azidomethyl)-2,3-dibromothiophene 1-[2-[6-chloro-2-[(E)-3,3-dimethylbut-1-enyl]-4-oxoquinazolin-3-yl]ethyl]piperidine-3-carboxamide 3-(4-fluoro-N-nonanoylanilino)butanoic acid 5-butyl-2,4-dimethoxybenzoic acid N'-[(3Z,5E)-6-methylhepta-1,3,5-trien-2-yl]benzohydrazide N-(cyclopropylmethyl)-2,3-diethynylbenzamide;2-(4-fluorophenyl)-1H-pyrrole 5-(2,4-dichlorophenyl)-N-[1-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]-3-methyltriazole-4-carboxamide 2-methyl-4-(3,5,6-trichloropyridin-2-yl)sulfanylbutanoic acid 5-bromo-1-(4,6-dimethylpyrimidin-2-yl)oxypentane-3-sulfonic acid 2-[4-[2-(4-hydroxypiperidine-1-carbonyl)thiophen-3-yl]triazol-1-yl]acetic acid [2-[(6-chloropyridine-3-carbonyl)amino]-4,5-dihydropyrazolo[1,5-a]pyrimidin-7-yl]boronic acid 3-amino-4-cyano-5-[2,6-difluoro-4-(trifluoromethyl)phenyl]-1H-pyrrole-2-carboxamide 5-chloro-3-[1-(2,4-dimethylphenyl)cyclopropyl]-2H-isoindol-1-one N-[5-(3,4-dichlorophenyl)-6-ethoxypyridin-2-yl]-1H-indole-7-carboxamide 1-[4-[(4-bromophenoxy)methyl]phenyl]sulfonylpiperazine 7,8-dihydroxynaphthalene-2,3-disulfonate 4-(1H-benzimidazole-2-carbonyl)-7-[[6-[(4-methylpiperidin-1-yl)methyl]pyridin-3-yl]amino]-3,5-dihydro-2H-1,4-benzoxazepine-8-carbonitrile N-(4-bromobutan-2-yl)-2,6-difluoro-N-octylaniline N-[2-(1-methylpyrazol-4-yl)ethyl]spiro[1,3,5,6-tetrahydro-1,5-benzodiazocine-2,4'-piperidine]-4-carboxamide N-[(3S,5R)-1-(2,3-dimethyl-1H-pyrrolo[2,3-b]pyridine-4-carbonyl)-5-(5-methyl-1,3,4-oxadiazol-2-yl)pyrrolidin-3-yl]benzamide 6-tert-butyl-3-[5-(2,4-dimethylphenyl)furan-2-yl]-4H-1,2,4-triazin-5-one 2-(5-acetylpyridin-3-yl)-N-[5-cyano-4-[6-(difluoromethoxy)spiro[2.5]octan-2-yl]pyridin-2-yl]acetamide 1-[4-azido-2-(trifluoromethyl)phenyl]-3-ethoxyazetidine N-[5-[3-(4,6-dimethyl-1H-benzimidazol-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]cyclohexanecarboxamide 4-(dimethylamino)-N-[2,5,7,8-tetramethyl-3-(1-methylpiperidine-4-carbonyl)-1,6-naphthyridin-6-ium-6-yl]but-2-ynamide [1-(cyclopropylmethyl)pyrazol-4-yl]-[4-[2-(dimethylamino)pyrimidin-5-yl]piperidin-1-yl]methanone 4-[1,3-bis(2-methylpropyl)imidazolidin-2-ylidene]piperidine;[2-[[4-[2-(2-hydroxyethoxy)ethoxy]phenyl]iminomethyl]phenyl]-dimethylsulfanium 1-(3-hydroxypropyl)indole-6,7-dicarboxamide 3-[3-(1,2-dihydroacenaphthylen-5-yl)phenyl]prop-1-en-2-ol 4-[1-(2,2,3,3,5,5-hexamethylpiperidine-1-carbonyl)-3-[5-(2H-tetrazol-5-yl)thiophen-3-yl]cyclopentyl]benzonitrile 4-[2-(4-ethoxyphenyl)ethynyl]-1,3-difluoro-5-(trifluoromethyl)pyrazole 5-chloro-4-hydroxy-N-[(3S)-piperidin-3-yl]benzamide;dihydrochloride 1-[2,3,4-tri(propan-2-yloxy)phenyl]ethanethiol 1-N',2-N'-dimethyl-2-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethane-1,1-diamine N-(4-cyclohexyloxypyridin-3-yl)-5-methoxypyrimidine-2-carboxamide N-[(1S)-1-[6-chloro-8-fluoro-7-[(2R,3R)-2-methyl-4-(5-methylfuran-2-carbonyl)morpholin-3-yl]oxy-2H-chromen-3-yl]ethyl]acetamide 1-[[5,6-difluoro-2-(3-methylphenyl)benzimidazol-1-yl]methoxymethyl]cyclopropane-1-carboxylic acid N-[(2,6-dimethylpyridin-4-yl)methyl]-1-[(3R)-1-propanoylpiperidin-3-yl]triazole-4-carboxamide 2-hydroxy-N-[(4-nitrophenyl)methyl]-6-oxo-1H-pyrimidine-5-carboxamide [(E)-[1,3-benzothiazol-2-yl(ethyl)hydrazinylidene]methyl]methanol 2,6-difluoro-N-[(E)-(5-methylfuran-2-yl)methylideneamino]benzamide 5-benzylsulfanyl-2-methoxy-1,3-thiazole 5-azido-2-(4-tert-butylphenyl)pyrimidine N-(cyclobutylmethyl)-4,5-difluoro-2-[(2S,3R)-1-methyl-2-(4-phenylphenyl)azetidin-3-yl]benzenesulfonamide (E)-4-[5-cyano-2-cyclobutylsulfanyl-6-methylidenepyridin-1-yl]-N,N-diethylhept-3-enamide 1-ethyl-4,5-difluoro-6-(1H-pyrrolo[2,3-b]pyridin-4-ylamino)cyclohexa-2,4-diene-1-carboxylic acid (2S,4R)-N-benzyl-1-[(3R)-7-fluoro-5-methylidene-1H-2,3-benzodiazepine-3-carbonyl]-4-hydroxypyrrolidine-2-carboxamide 2,4-dimethoxy-N-(3-methylbutyl)aniline 6-methoxy-5,8-dihydroacridine-1-carboxylate 5-(4,6-diphenyl-1H-1,3,5-triazin-2-yl)-[1]benzofuro[3,2-c]quinoline 1-[3,5-bis(trifluoromethyl)phenyl]-N-cyclohexa-2,4-dien-1-ylbutan-2-imine 4-(3,5-dimethylpyrazol-1-yl)-N-(3-ethoxyphenyl)-6-morpholin-4-ylpyrimidin-2-amine (4-azidopiperazin-1-yl)-(2,5-dimethoxyphenyl)methanone 2-[3,6-dibromo-4-(trifluoromethyl)pyrazolo[4,3-c]pyridin-1-yl]acetic acid 3-(4-chlorophenyl)-5,8,10-triazatricyclo[7.4.0.02,6]trideca-1(9),2,4,6,11-pentaen-12-one 1-methyl-N-[4-(2,3,5-trifluorophenyl)cyclohexyl]piperidine-3-carboxamide 1-[[2,5-difluoro-4-(trifluoromethyl)phenyl]methyl]-N-hydrazinylideneindole-6-carboximidamide N-(azidomethyl)-2-cyclohexyloxy-6,7-dihydro-5H-cyclopenta[b]pyridin-4-amine 1-(1-azidoethoxy)-3,4,5-triphenylbenzene 1-azido-2-(dimethoxyphosphorylmethoxy)benzene 4-N,6-dimethyl-2-[(3E)-penta-1,3-dien-3-yl]pyrimidine-4,5-diamine 1-(2-azido-5,6,7,8-tetrahydronaphthalen-1-yl)naphthalene 5-[3-(3,3-difluorocyclobutyl)azetidine-1-carbonyl]pyrimidine-2,4-dicarboxylic acid 5-chloro-4-[4-[2-[4-(dimethylamino)phenyl]-1,3-thiazol-5-yl]-5-pyridin-4-yl-1H-imidazol-2-yl]-6-fluoro-1H-pyrimidin-2-one 2-[1-(dipropylamino)phenoxazin-10-yl]ethanethiol N-(6-chloropyridin-3-yl)-5-oxospiro[2H-1-benzofuran-3,4'-piperidine]-1'-carboxamide 4-[1-(benzylamino)ethenyl]-N'-[[4-(trifluoromethoxy)phenyl]iminomethyl]benzenecarboximidamide 6-azido-4-hydroxy-3H-2,1-benzoxaborole 4-[3-(azidomethyl)-5-fluorophenoxy]-1,2-dichlorobenzene (4R)-2,2-dimethyl-N'-[4-nitro-3-(trifluoromethyl)phenyl]octanimidamide 3-(cyclohexylmethoxy)-4-phenylbenzoate 4-bromo-5-(2,6-difluorophenyl)-N-[1-(methylaminosulfanyl)piperidin-4-yl]pyridin-3-amine 2-[4-hydroxy-N-(3-methylbutyl)anilino]acetic acid 1-(4,6-dimethoxypyrimidin-2-yl)pyrrolidin-3-amine;dihydrochloride N-[4-(1,3-benzothiazol-2-yloxy)phenyl]-3-chloro-5-nitropyridine-2-carboxamide 6-[3-(4-fluorophenyl)propanoyl]-5,7,8,9-tetrahydro-1H-pyrimido[4,5-d]azepine-2,4-dione 4-(N-tert-butyl-4-propanoylanilino)benzenesulfonic acid 4-(difluoromethyl)-2,5-bis[(2-ethenoxyphenyl)methylidene]furan 2-[4-chlorobutyl(hexyl)amino]benzoic acid N-[2-(3,4-dichlorophenyl)ethyl]-1-[[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]methyl]cyclopropane-1-carboxamide 6-(3,4-dihydropyridin-2-yl)-3-methylidenehexan-2-one 2-tert-butyl-4-[(E)-2-[2,3,6-trichloro-4-hydroxy-5-[(propan-2-ylideneamino)methyl]phenyl]ethenyl]-N-[4-(trifluoromethyl)pyridin-3-yl]benzamide 2-[(1S)-6-chloro-4-fluoro-3,4-dihydro-1H-isoquinoline-2-carbonyl]cyclohexan-1-one (2S)-1-[4-chlorobutyl-(2,6-difluorophenyl)sulfonylamino]-N-hydroxyazetidine-2-carboxamide (2R)-4-benzyl-3-oxo-N-phenylmethoxyiminomorpholine-2-carboxamide ethane;N-(2-hydroxy-2-naphthalen-1-ylacetyl)azetidine-3-carboxamide N-[3-cyano-6-(1-methylpyrazol-4-yl)pyrazolo[1,5-a]pyridin-4-yl]-2,2-difluorocyclopropane-1-carboxamide 2-amino-4-[5-bromo-2-(3-phenylmethoxypropoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile [5-(3,4-dichlorophenyl)pyrazin-2-yl]methylideneazanium 6-(azidomethyl)-4-(3,4-difluorophenyl)sulfanylimidazo[1,2-a]pyridine [1-(1,5-dimethylpyrazole-4-carbonyl)piperidin-4-ylidene]-[4-(trifluoromethoxy)phenyl]sulfonylazanium 2-cyclopropyl-3-[(2E)-2-[1,3-dimethyl-6-nitro-4-oxo-7-[[(2S)-pentan-2-yl]amino]quinolin-5-ylidene]ethoxy]benzoic acid (2S,4R)-4-hydroxy-1-[2-methyl-6-[5-methyl-3-[7-(trifluoromethoxy)quinoxalin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]pyridine-4-carbonyl]pyrrolidine-2-carboxylic acid N-(4-bromophenyl)-2,6-difluorobenzohydrazide 3-[4-(1,2-benzothiazol-6-ylsulfonyl)piperazine-1-carbonyl]-5-methoxybenzonitrile 2-N,6-N-bis(4-bromophenyl)-4-N-butylpyrimido[5,4-d]pyrimidine-2,4,6-triamine (3aR,8bS)-N-[(1S)-2-amino-4-methylsulfonylcyclohexa-2,4-dien-1-yl]-2-[3-fluoro-5-(trifluoromethoxy)phenyl]-7-(2-pyridin-3-ylethynyl)-3,3a,8b-trihydro-1H-pyrrolo[3,4-d]azepine-6-carboxamide 4-methyl-2-(4-pyridin-3-yl-1H-pyrrolo[3,2-c]pyridin-2-yl)-1H-imidazo[4,5-b]pyridine 3-(1H-benzimidazol-2-yl)-6,7-dimethoxy-1H-quinolin-4-one 2-(4-bromophenyl)-1-cyclopropylbenzimidazole;ethane 6-[[1,4-bis(ethenyl)cyclohexa-2,4-dien-1-yl]methoxy]naphthalene-2-sulfonic acid 1-[2-methylpropyl(pentyl)amino]-3,4-dihydro-2H-naphthalen-1-ol 5-(3,5-dimethyl-1H-pyrazole-4-carbonyl)-2,6,7,8-tetrahydro-1H-pyrrolizin-3-one 2-(dimethylamino)-3,4,5-trifluorobenzoic acid 3-[(6,7-difluoroquinoxalin-2-yl)amino]propan-1-ol 1,4-diiodoindazole 1-cyclohexyl-N-[2-[(3-methoxyphenyl)methoxyimino]propoxy]-4,5-dihydroimidazole-2-carboxamide 2-[(1Z)-buta-1,3-dienyl]-5-chlorochromene;ethane 4-[4,7-dimethyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]quinoxalin-2-yl]benzonitrile;ethane 1-[(3E)-4-methylpenta-1,3-dien-2-yl]oxy-N-phenylpropan-2-amine 5-bromo-4-N-[(1R)-2,3,3a,4,5,6,7,8,8a-octahydro-1H-inden-1-yl]pyrimidine-2,4-diamine [2-(1,3-benzodioxol-5-yl)quinolin-4-yl]hydrazine 4-(3,5-dimethylpiperazin-1-yl)-6-[(E)-2-(4-ethoxyphenyl)ethenyl]-N'-[5-(furan-2-yl)-2-methylpyrazol-3-yl]pyridine-2-carboximidamide N-(6-bromo-4-methylpyridin-2-yl)acetamide 2-(7,9-difluorobenzo[e][1]benzofuran-10-yl)-6-pyridin-4-ylpyridine 2-(2,3-dihydro-1H-inden-5-ylmethoxy)-6-[1-(disulfanylamino)-3-oxopent-4-enyl]benzenesulfinic acid 4-[1-hydroxy-2-(oxan-4-ylamino)ethyl]pyridine-3-carbonitrile 2-methyl-1-[6-[4-(2,2,5,5-tetrafluorocyclohexyl)phenyl]naphthalen-2-yl]isoquinolin-2-ium (7S)-8-benzyl-2-(4,6-dimethoxypyrimidin-5-yl)-7-ethyl-[1,3]thiazolo[4,5-e][1,2,4]triazin-3-one 2-(4-chlorobutyl)-6-(1,3-difluoropropan-2-ylamino)-5,6,7,8-tetrahydronaphthalene-1,2-diol 1,5-bis[(4-bromophenyl)methylidene]piperazine 3-[4-[(4-chlorophenyl)carbamoylamino]-1,3-dioxoisoindol-2-yl]piperidine-1-carboxylate 6-fluoro-2-[4-(trifluoromethoxy)phenyl]-3,10b-dihydropyrimido[5,4-d][1,3]benzoxazin-4-one 2-[(3R)-2,7-dioxoazepan-3-yl]sulfanyl-6-hydroxy-5-iodo-1H-pyrimidine-4-thione N-(2,6-difluorophenyl)-3-methoxypyridine-4-carboxamide N-[(4-fluorophenyl)methyl]-2-methylidene-3,7-dihydrobenzimidazole-1-carboxamide 1-(3-chloropyridin-4-yl)oxypiperidine-2,6-dione 2-hydroxy-6,6,7,7-tetramethylbenzo[g]pteridine-5,8-dione 2-bromo-N-(4,5-dichloropyrimidin-2-yl)benzamide 1-[5,7-dimethyl-2-(4-methylphenyl)imidazo[1,2-a]pyrimidin-3-yl]ethanone;N-[3-[6-(ethylaminomethyl)-7-oxooctoxy]phenyl]formamide 5-amino-2-(4,5-dimethylhexan-3-yl)phenol [(1R,5S)-3-phenyl-9-oxatricyclo[6.4.1.02,7]trideca-2(7),3,5-trien-5-yl]methanamine ethane;2-methylbutanamide;N-[(E)-1-morpholin-4-ylpropylideneamino]-4-piperidin-1-ylaniline 2-[4-(dimethylamino)anilino]-5,6,7,8-tetrahydro-3H-quinazolin-4-one 4-(6,7-dihydronaphthalen-2-yl)benzoic acid 4-N,4-dimethyl-5-(methylideneamino)-2-N-[4-[[(Z)-prop-1-enyl]sulfonylamino]phenyl]pyrimidine-2,4-diamine (Z,2E)-N'-[1-[3-methoxypropyl(methyl)amino]ethenylsulfanyl]-2-[1-[4-(trifluoromethoxy)phenyl]ethylidenehydrazinylidene]but-3-enimidamide N-(3,4-dihydroxyphenyl)-2-[(1E)-1-(4-oxo-3H-quinazolin-2-yl)buta-1,3-dien-2-yl]sulfanylacetamide 4-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophen-2-yl)-2-methoxyphenol 1-(2,3-dihydro-1H-inden-5-yl)isoquinoline 2-chloro-3,5-difluoro-4-(methoxycarbonylamino)benzoic acid 2,7-diphenylfluoren-1-one 1-azido-3,5-difluoro-2-methylbenzene N'-[4-[3,5-bis(trifluoromethyl)anilino]-1H-pyrrolo[2,3-b]pyridin-6-yl]-N,N,N'-triethylpropane-1,3-diamine N-[1-(3-methoxyphenyl)ethyl]-4-[4-(trifluoromethyl)phenoxy]aniline 3-[6-amino-4-[2,5-difluoro-4-(trifluoromethyl)phenyl]pyridin-2-yl]propanal (2-bromophenyl)methyl-diethylphosphane N-azido-4-chloro-3,5-diethoxyaniline N-[1-[4-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridin-7-ylmethoxy)phenyl]cyclohexyl]pyrrolidine-2-carboxamide (4E)-2,6-dimethylhepta-1,4-diene;ethane;5-ethenyl-3-[(Z)-prop-1-enyl]-N-phenylaniline 6-chloro-3-(2,2-difluoroethyl)-7H-purin-2-one 4-(1,3,5-trimethylpyrazol-4-yl)spiro[cycloheptane-1,9'-fluorene] 1-azidooxy-2,3,5-triethylbenzene 2-hydroxy-4-(2-methoxyethyl)-6-phenylbenzaldehyde 2-bromo-5,6-diethylpyrazine [4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]-thiomorpholin-4-ylmethanone N-(2,3-dihydroimidazo[1,2-c]quinazolin-8-ylmethyl)cyclobutanamine 4-[8-amino-3-[(E)-2,5-dimethylhex-1-enoxy]imidazo[1,5-a]pyrazin-1-yl]-N-pyridin-2-ylbenzamide 2-[[3,5-diethyl-4-(pyrrolidine-1-carbonyl)pyrazol-1-yl]methyl]-N-[5-(methoxymethyl)pyrazin-2-yl]benzamide 1-[3-chloro-2,6-di(propan-2-yl)phenyl]ethanethiol 4-[(5Z)-5,8-difluoro-1,7,8-trimethylnona-3,5,7-trien-4-yl]pyridine (2R)-6-fluoro-N',1-dimethylspiro[2H-indole-3,4'-piperidine]-1'-carbohydrazide (2S,3R)-1-[(1S,6S)-8-methyl-3,4-dihydro-1H-isochromene-1-carbonyl]-N-phenylazepane-2-carboxamide (2R)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-ethynyl-10-(5-fluoro-2-hydroxyphenyl)-11-oxo-1,2,4,7-tetrahydropyrido[4,3-a]quinolizine-8-carboxamide N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-6-[4-(3-fluoropropoxy)phenyl]-2,7-naphthyridin-8-amine N'-[5-[[6-(methoxyiminomethyl)pyridin-2-yl]disulfanyl]-1,3-thiazol-4-yl]methanethiohydrazide 5-(3-azido-4,5-dimethylphenyl)pyridine-2-carbonitrile (2S)-4,5-dimethyl-1-[3-(trifluoromethoxy)phenyl]sulfonylpyrrolidine-2-carboxylic acid 2-[4-bromo-N-(3,3,3-trifluoropropyl)anilino]acetic acid 1-[5-(4,4-difluorocyclohexyl)oxypyrimidin-2-yl]-N,N-bis[(6-methoxypyridin-3-yl)methyl]azetidine-3-sulfonamide [4-[5-(1H-indole-2-carbonyl)-7,8-dihydroimidazo[1,2-c]pyrimidine-2-carbonyl]piperazin-1-yl]-phenylmethanone [6-hydroxy-3-(4-phenylbutanoyl)-1H-indazole-5-carbonyl]azanium 3-hydroxy-N-methylbutanamide;2-[4-(2-methoxyethoxy)phenyl]-5-pyridin-4-yl-1,3-benzoxazole 3-[2-hydroxyethyl(2,4,6-trimethylphenyl)sulfonylamino]butanoic acid 2-[(3,4-dichlorophenyl)methylsulfanyl]-6-oxo-4-propan-2-yl-1H-pyrimidine-5-carbonitrile 5-[(E)-2-bromopent-1-enyl]-3,4-dimethoxycyclohexa-1,3-diene N-(2,4-dinitrophenyl)-N-octylbenzamide 2-[1-[(2-bromophenyl)sulfonylamino]cyclopropyl]acetic acid 7-(4-chlorophenyl)-2-[3-methoxy-5-(4-nitrophenoxy)phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrimidine 2-[(3,4,6-triethyl-5-methylidenecyclohexa-1,3-dien-1-yl)amino]-1,4,8-triazacyclotetradecan-9-one 2-(4,5-dimethyl-1,3-thiazol-2-yl)-N-[5-(furan-2-yl)-1H-pyrazol-3-yl]piperidine-1-carboxamide 2-(4-azidophenyl)-5-ethyl-1,3-benzothiazole 1-(2,6-dimethoxypyridine-3-carbonyl)-N-[4-(3-methylbutanoylamino)phenyl]piperidine-2-carboxamide N-[(3S,4R)-1-[2-[5-methyl-6-[4-(2-pyrrolidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-7-yl]pyridin-3-yl]piperidin-4-yl]cyclopropanesulfonamide 5-N-[(3,4-dimethoxyphenyl)methyl]-2-N-[[7-fluoro-6-(3-morpholin-4-ylpropoxy)pyridin-2-yl]methyl]pyrazine-2,5-dicarboxamide ethane;(5Z)-5-[[4-[(E,3R)-3-hydroxybut-1-enyl]phenyl]methylidene]imidazolidine-2,4-dione (5R)-5-[4-(cyclopropylmethoxy)phenyl]-2,3-dihydropyrano[3,2-g]chromen-7-one 2-(2,3-dichloro-4-hydroxyphenyl)sulfonylpropanamide 6-(trifluoromethyl)-3H-imidazo[1,2-a]pyridine-4-carbonitrile 5-bromo-2,4-dimethyl-N-[(3R)-1-[(1S)-2-oxocyclohexanecarbonyl]piperidin-3-yl]thiophene-3-carboxamide 6-methylsulfonylnaphthalene-2,3-diamine N-cyclopropyl-2,4-difluoro-3-[5-(1-methoxycarbonyl-6,7-dihydro-4H-triazolo[4,5-c]pyridin-5-yl)tetrazol-2-yl]benzamide 4-(4,5-dimethylpyridin-2-yl)oxy-N-ethylaniline N-[3-(1,2,4-oxadiazol-5-yl)cyclohexa-1,5-dien-1-yl]benzamide N-[(1S)-3-oxo-3-phenylmethoxypropyl]carbamate 2-[3-methoxy-5-(4-nitrophenyl)pyridine-4-carboximidoyl]aniline 6-methyl-2,5-bis(4-pentoxyphenyl)furo[3,2-b]thiophene 4-[[5-(3,4-dimethylphenyl)-4-propanoylimidazol-1-yl]methyl]benzenesulfonamide N-(3-cyano-4-fluorophenyl)-1-methyl-2,5-dioxopyrrolidine-3-carboxamide 1-[3-(4-azidophenyl)pyridin-4-yl]piperidine-4-carbonitrile [(2R,5S)-4-chloro-5-hydroxy-6-(phenylmethoxycarbonylaminomethyl)oxan-2-yl]carbamic acid N-[(2S)-1-oxopropan-2-yl]benzenesulfonamide 3-chloro-4-[(E)-2,5-dimethylhex-2-enoxy]-6-propan-2-ylidenecyclohexa-2,4-diene-1-carboxamide N-(2,4-difluorophenyl)-N'-[4-[6-[4-methoxybutyl(propanoyl)amino]pyridazin-3-yl]-2,5-dimethylphenyl]oxamide 2-ethoxy-N-[4-(3-fluoropyridin-2-yl)phenyl]pyrimidine-5-carboxamide 2-fluoro-4-[(E)-3-(3-methylphenyl)prop-1-enoxy]phenol [4-amino-2-(3,5-dimethyltriazol-4-yl)phenyl]-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]methanone 3-[(Z)-(1,3-dimethyl-2,6-dioxopyrimidin-4-ylidene)amino]benzonitrile 5-cyclobutyloxy-4-methyl-1H-pyrazole-3-carboxylic acid [2-azidooxy-1-[(4-methylphenyl)sulfonylamino]-1,3-dihydroindene-2-carbonyl]azanium 6-[4-(4-aminophenyl)piperidin-1-yl]pyridine-3-carbonitrile 3-(1,2-diphenylethenyl)naphthalen-2-ol 3-[4-bromobutan-2-yl(ethenylsulfonyl)amino]benzoic acid (2R,3S)-N-[(Z)-1-aminoethylidenecarbamothioyl]-3-methyl-2-phenyloxolane-2-carboxamide (2R)-1,5-bis(3-chlorophenyl)pentan-2-ol N-[1-(2,2-difluoroethyl)pyrazol-4-yl]-2-(1H-indazol-5-ylamino)thieno[3,2-d]pyrimidine-7-carboxamide 4-[(Z)-1,3-diamino-2-[4-(azetidine-1-carbonyl)anilino]but-1-enyl]benzonitrile 1-azido-5,6-diethyl-2H-pyrazolo[3,4-b]pyridine N-[2,4-difluoro-3-(3-methoxypropylsulfanyl)phenyl]propane-1-sulfinamide;ethane 2-(8-azabicyclo[3.2.1]octan-8-yl)quinoline 2-ethoxy-N,3,5,6-tetrafluoropyridine-4-carbothioamide 2-(1H-indol-3-yl)-N,N-bis(prop-2-ynylsulfanylmethyl)ethanamine 2-[4,5,6-tris(4-chlorophenyl)pyrimidin-2-yl]oxyacetamide 3-(1-ethylcyclopropyl)-5-fluoropyridine-2-carboxamide N-[(1R)-1-(3,5-dichloropyridin-2-yl)ethyl]-2-[6-(2,2,2-trifluoroethoxy)pyridin-3-yl]acetamide 6-tert-butyl-3-chloro-8-fluoroquinoline 3-(1H-benzimidazol-2-yl)-2-(3-fluorophenyl)iminopropanoic acid 3-(3,4-dihydroxyphenyl)-2-[[4-[(Z)-[[5-(1,3-thiazol-2-yl)-1H-indol-3-yl]methylideneamino]carbamoyl]benzoyl]amino]propanoic acid N-(2,6-dichloro-4-nitrophenyl)-N-(2-methylpropanoylamino)sulfonylbenzamide 3,5-dichloro-N-ethylsulfonyl-4-fluorobenzamide (E)-2-amino-3-hydrazinyl-3-[3-methoxy-4-(6-oxohept-1-enyl)phenyl]prop-2-enenitrile 3-[2-(4-propan-2-yloxyphenyl)iminoethanehydrazonoyl]phenol [(4R)-2,6-diaminohexyl]carbamic acid;ethane;1-methoxynaphthalene;N-[(Z)-[(5Z)-3-methylidenehepta-5,7-dien-2-ylidene]amino]methanamine 2-azido-1,4-dibutylbenzene (2S)-3-methyl-N,2-diphenylpentanamide 2-amino-3-[[4-(5,6-dimethylpyridine-2-carbonyl)phenyl]methoxy]propanoic acid;ethane [2-(5-aminopyrazin-2-yl)piperidin-1-yl]-cyclopropylmethanone;ethane N-(1H-benzimidazol-2-ylmethyl)-N,5-diethoxy-3-methoxypyrazine-2-carboxamide N-[1-(2-chlorophenyl)propyl]-6-cyclohexa-2,4-dien-1-ylidene-7H-benzo[a]quinolizin-5-ium-10-amine 2-[(3,5-dimethylimidazol-4-yl)sulfonylamino]-N-ethylpropanamide 2-[(1R,5S)-3-acetyl-8-methyl-3-azabicyclo[3.2.1]octan-9-yl]-N-cyclobutylpyridine-4-carboxamide [(2-carboxyphenyl)-(4,6-dihydroxy-7-methylnaphthalen-1-yl)methylidene]azanide 5-[2-chloro-3-(trifluoromethyl)phenyl]-N-methylpyrazin-2-amine 2-[(3R,4S)-3-benzyl-1-(dimethylamino)pyrrolidine-3-carbonyl]-7-ethoxy-9-hydroxypyrido[1,2-a]pyrimidin-4-one;hydrochloride 2-[1-(4,4-dimethylcyclohexen-1-yl)ethenyl]-6,7-dimethoxy-3,4-dihydroisoquinolin-1-one 3-[5,7-dichloro-2-[1-(2-fluoroethyl)pyrazol-4-yl]thieno[3,2-b]pyridin-3-yl]-N,N-dimethylbenzamide 3-[2,6-bis(trifluoromethyl)phenyl]-5-[3-(9H-fluoren-1-ylmethyl)piperidine-4-carbonyl]-1,3,4-oxadiazol-2-one (4R)-2,5-dimethyl-4-[2-oxo-3-propan-2-yloxy-6-(trifluoromethyl)pyridin-1-yl]heptanedioic acid (2R,6S)-4-benzyl-N-[4-[1-(1H-imidazole-5-carbonyl)piperidin-3-yl]phenyl]-2,6-dimethylmorpholine-4-carboxamide 2-(4-fluorophenyl)-2-[[5-(1H-indol-3-yl)-4-(oxolan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide N-[2-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-6-azaspiro[2.5]octan-6-yl]benzamide 5-fluoro-4-[4-(2,2,2-trichloroethyl)-1H-imidazol-5-yl]pyrimidine (3E,5E)-1-[1-methyl-4-(4,4,6-trifluorocyclohexa-2,4-dien-1-yl)pyrrol-3-yl]hepta-1,3,5-trien-4-amine (2R,3S)-N-[4-fluoro-3-(trifluoromethyl)phenyl]piperidine-2-carboxamide 4-[3-methylbutyl(phenacyl)amino]benzenesulfonic acid N-[(2S)-3-(1H-indol-3-yl)-1-[4-methoxy-7-(2-methylpropyl)-1,4-diazepan-1-yl]-1-oxopropan-2-yl]benzamide 1-chloro-4,4a,6,8-tetramethyl-3,4-dihydroquinolin-2-one 2-azido-4,6-ditert-butylpyrimidine 1-(7-aminoheptyl)-5,6-dimethoxyindazole-3-carboxylic acid 3-[3-[4-chloro-2,6-di(propan-2-yl)phenyl]-2H-pyrrol-5-yl]benzamide N-(3-chloro-2H-indazol-5-yl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide 3-[4-(1,3-benzodioxol-5-ylmethylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-fluoro-N,N-dimethylbenzamide 4-[(1R,2S)-6,15-dibromo-13-chloro-4-azatricyclo[9.5.0.03,8]hexadeca-3(8),4,6,11-tetraen-2-yl]piperazine-1-carboxylic acid;ethane 2-azido-N,N-dimethylaniline 6-(4,5-dihydrothieno[3,2-d][1]benzazepine-2-carbonyl)-1-methylpyrimidine-2,4-dione 7-bromo-2,3,4a,10a-tetrahydroindeno[1,2-b][1]benzofuran 1-(2,5-dimethoxyphenyl)sulfonyl-N-hydroxyimidazole-4-carboxamide 4-(5,6-dimethylbenzimidazol-1-yl)-N'-hydroxypyridine-2-carboximidamide 5-fluoro-7-[4-(3-iminocyclopentyl)sulfonylpiperazin-1-yl]quinoline-3-carbonitrile N-(3,5-dimethylphenyl)-1-[4-nitro-3-(trifluoromethoxy)phenyl]-5-piperidin-4-ylpyrazole-4-carboxamide N-[3-(5-chloropyridin-2-yl)oxypropyl]-1,2,4-triazol-4-amine 1-[(5-tert-butyl-2-hydroxyphenyl)methyl]piperidine-4-carboxylic acid 5-chloro-6-hydroxy-N-[(1-methylpyrazol-3-yl)methoxy]naphthalene-2-carboxamide N-[6,8-dimethoxy-2-(4-oxopentyl)imidazo[1,2-a]pyridin-3-yl]cyclopropanecarboxamide 2-(7-fluoroimidazo[1,2-a]pyridin-3-yl)-N-phenylpyrimidine-4-carboxamide 2-azidosulfanyl-1,3,5-trichlorobenzene (5Z)-2-(4-bromophenyl)imino-5-[(6-methoxynaphthalen-1-yl)methylidene]-1,3-thiazolidin-4-one (1S)-2,2-difluoro-N-[6-[(3R)-3-methylmorpholin-4-yl]pyridin-3-yl]cyclopropane-1-carboxamide 3-methyliodanuidylbenzaldehyde 2-fluoro-4-[(3E)-hepta-1,3,5-trien-4-yl]phenol 1-[5-(4-chlorophenyl)sulfanyl-2,3-dihydrothieno[3,4-b][1,4]dioxin-7-yl]piperidine (1-diphenylphosphorylsulfanylethylsulfonylmethoxy)benzene 2,4-bis(2-methylbutan-2-yl)-N-phenylaniline ethane;2-methylbutanoic acid;[4-(6,7,8,9-tetrahydro-5H-pyrido[3,2-b]indole-7-carbonyl)piperazin-1-yl]methanone 3-(2,4-dimethylphenyl)-5-methoxy-1H-indole;ethane 4-[5-(2,3-dihydro-1H-inden-5-yl)thiophen-2-yl]-2-propanoylbenzoic acid 3-[(2,4-dichloropyrimidin-5-yl)-(1,3-thiazol-5-yl)amino]phenol N-cyclopropyl-4,6-difluoro-3-[(Z)-1-hydrazinylethenoxyiminomethyl]benzamide 1-(4-ethoxyphenyl)-2,3,4a,5,6,7,8,9,10,10a-dodecahydropyrimido[4,5-b]quinoline 2-(5-methyl-4-phenylmethoxypyrimidin-2-yl)oxyethanol 1-(4,5-dimethylpyridin-2-yl)cyclohexane-1-carboxylic acid 2-(1,3-benzothiazol-6-ylmethoxy)-4,7-dihydropyrrolo[3,4-b]pyridine 2-amino-6-[(Z)-1-amino-3-methyliminoprop-1-en-2-yl]-5-methanimidoyl-N-[3-(4-propan-2-ylpiperazin-1-yl)pyridin-2-yl]pyrimidine-4-carboxamide 3-(4,6-difluorocyclohepta-1,3,5-trien-1-yl)-5-[1-(2-methylpropyl)piperidin-4-yl]-1H-indole 4-(2-aminopropylamino)-1H-pyrrolo[3,2-c]pyridine-7-carboxylic acid 2-[4-(5,6-diethoxy-4-oxo-3H-quinazolin-2-yl)phenyl]-1-[1-(2-methoxyacetyl)piperidin-4-yl]guanidine;hydrochloride 1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one [2-[3-(dimethylamino)phenyl]-1,3-oxazol-5-yl]-[3-methoxy-4-(1H-pyrazol-5-ylamino)phenyl]methanone N-(5,6-difluoro-1H-indol-3-yl)-4-fluorobenzamide;ethane (3S,6S)-6-(1H-indazol-5-ylmethoxymethyl)oxane-3,4,5-triol 5-(4-tert-butylcyclohexen-1-yl)oxycarbonyl-2,6-dimethyl-1,4-dihydropyridine-3-carboxylic acid 3-[7-(2,4-difluorophenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-ethoxy-N-(3-piperazin-1-ylpropylsulfonylmethyl)-1H-indazole-6-carboxamide N-[(3S)-1-[(6R,7aS)-4a-methyl-2-oxo-1,5,6,7,8,9-hexahydropyrrolo[1,2-a]quinoline-6-carbonyl]piperidin-3-yl]naphthalene-1-carboxamide [2-[5-fluoro-1,7a-dimethyl-3-(trifluoromethyl)-6H-cyclohepta[b]pyrrole-2-carbonyl]-1,3-thiazol-4-yl]-phenylmethanone 3-[5,6-bis(4-chlorophenyl)pyrazin-2-yl]oxypyrrolidine-1-carboxylate 7-azido-1,2,3-triphenylimidazo[4,5-c]pyridine (2-chloro-4,6-difluorophenyl)-[(3R)-3-cyclopropylpiperidin-1-yl]methanone 2-[(3S,4R)-3-amino-4-azidopyrrolidin-1-yl]benzenethiol (2S,6R)-4-(azidomethyl)-N'-(5-fluoropyrimidin-2-yl)-3,6-dimethylpiperazine-1-carboximidamide 2-[1-(4-methoxyphenyl)-2,3-dihydrotetrazol-5-yl]-1H-indole 6-(difluoromethyl)-N-[3-oxo-3-[4-[5-[(propanoylamino)methyl]pyrimidin-2-yl]piperazin-1-yl]propyl]pyridine-3-carboxamide 5-[3-(2,4-dichlorophenyl)phenyl]-N'-ethyl-1H-imidazole-2-carboximidamide N'-[3-[1,2,6-trimethyl-4-(oxan-4-yl)-8-(oxetan-3-ylsulfonyl)naphthalen-2-yl]oxypropyl]ethane-1,2-diamine (E)-N-[2-amino-4-chloro-6-[3-(ethylcarbamoyl)phenyl]phenyl]pent-2-enamide N-benzylsulfanyl-3-nitro-1,2,4-triazol-1-amine [4-chloro-2-hydroxy-3-(2,4,6-trimethylphenyl)sulfanylphenyl]carbamic acid [3-chloro-4-(dimethylamino)phenyl]azanide 5-[(4R)-7-fluoro-2,3,10-trimethoxy-9-oxoacridine-4-carbonyl]benzimidazole-1-carboxylic acid N'-(2,3-dimethylindazol-5-yl)-2-(1H-indol-3-yl)acetohydrazide 2,6-ditert-butyl-4-[(7-methoxy-1,3-benzothiazol-2-yl)iminomethyl]phenol 1-azidooxy-4-butyl-2,3,5,6-tetramethylbenzene 2-(3,5-dichlorophenyl)-N-[2-(dimethylamino)-4-methoxypyrimidin-5-yl]acetamide 4-amino-1-[(2R,5S)-5-azidooxolan-2-yl]pyrimidin-2-one 3-(4-tert-butylphenyl)-5-[2,6-difluoro-4-(2-hydroxypropan-2-yl)phenyl]-N-ethoxy-N-methyltriazole-4-carboxamide N-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-3-(4-hydroxyphenyl)-4H-chromene-8-carboxamide 5-(1-methylcyclobutyl)-1,3-diphenylpyrazole (2R)-N-[(Z,3S)-1-amino-2-methylpent-4-en-3-yl]-3-[4-(4-chlorophenyl)phenyl]sulfonyl-2-methylpropanamide 2-[(1R)-1-azidopropyl]-3,4-dichloropyridine 5-benzyl-3-tert-butyl-1H-1,2,4-triazole N-[3-(2-aminoethyl)phenyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide;hydrochloride (4-chloro-2,5-difluorophenyl)-[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)spiro[6H-imidazo[1,5-a]pyrazine-8,4'-piperidine]-1'-yl]methanone 1-(2,4-dimethylphenyl)-3-[(Z)-4-[4-[5-ethoxypentyl(2-hydroxyethyl)amino]piperidin-1-yl]-2-fluorobut-2-enyl]urea 4-[(3,5-dichloropyridine-4-carbonyl)amino]piperidine-1-carboxylate 2-(4,5-dihydroindazol-1-yl)-5,6-dimethoxypyrimidine 5-azidooxy-4-cyclopropyl-2,3,6-trifluoroaniline 1-(2,3-dimethylbutan-2-yl)-5-methylindole (5R)-3,3,4,7-tetramethyl-5-pyridin-2-yl-1,9b-dihydro-[1]benzothiolo[3,2-e]benzimidazol-6-one (E)-3,4-dihydroxy-6-[[4-(trifluoromethyl)phenyl]methoxy]hex-5-enoic acid (3aR,5S,7aS)-1-(4-methoxyphenyl)sulfonyl-N-propan-2-yl-3,3a,5,6,7,7a-hexahydro-2H-pyrano[3,2-b]pyrrole-5-carboxamide [4-(8-aminoimidazo[1,2-a]pyrazin-3-yl)-6-methoxypyridin-2-yl]methanol;dihydrochloride 2-(5-butan-2-yl-1H-pyrazol-4-yl)-N-[6-(prop-2-enoylamino)hexyl]pyridine-4-carboxamide 4-[2,3-dihydroxypropyl([1,2,4]triazolo[4,3-a]pyrazin-5-yl)amino]benzenesulfonamide [2-azido-5-(trifluoromethyl)phenyl]urea 5-chloro-2,3-dimethyl-1H-indole;6-(pyridin-4-ylamino)spiro[1H-indole-3,3'-piperidine]-2-one N-(4-chlorobutyl)-5-nitroquinolin-8-amine N-methylsulfonyl-5-propanoylpyridine-3-carboxamide (1R)-2,3,4-trifluoro-N-[6-(2-methyl-5,6-dihydro-4H-cyclopenta[c]pyrazol-3-yl)pyridin-3-yl]cyclohexane-1-carboxamide 1-[(1R,5S)-3-[3-(trifluoromethoxy)phenyl]-3,6-diazabicyclo[3.2.0]heptan-6-yl]propan-1-one 2-[[6,7-dimethoxy-2-(4-methylphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]ethanesulfonic acid 1-(2,3-dihydropyridin-6-ylmethyl)pyrazolo[4,3-b]pyridine N-benzyl-5-(2,4-dichloro-3-hydroxyphenyl)pentanamide 5-(azetidin-3-yl)pyrazine-2,6-diamine;2,4,6-trimethoxybenzaldehyde (2S)-N-[(4-chlorophenyl)methyl]-5-(methylcarbamoylamino)-5-oxopentanamide (6-azidocyclohexa-2,4-dien-1-yl)oxybenzene 2,4-dimethyl-5-(3-oxobutanoyl)benzenesulfonic acid 5-[(3-bromophenyl)iminomethyl]-6-hydroxy-1,4-dihydropyrimidin-2-amine N-(3,4-dihydroquinolin-2-yl)-5-(2H-tetrazol-5-ylmethoxy)indole-1-carboxamide N-(5-chloropyridin-2-yl)-4-hydroxy-3-methoxybenzamide 5-(1-fluoropropyl)-2,4-dimethoxypyrimidine 4-[5-(9H-fluoren-1-yl)pentanoyloxy]benzoic acid (E)-3-[4-(4-aminophenyl)phenyl]prop-2-enethioamide 2-[2-oxoethyl(pyridin-3-yl)amino]benzoic acid 2,3-bis(1H-imidazol-2-yl)-1H-indole 1-[5-cyano-2-(trifluoromethyl)phenyl]-3-N-cyclopropyl-2,4-dioxopyrimidine-3,6-dicarboxamide (2S,3aS,7aR)-6-[(5-cyclopropyl-1,3-oxazol-4-yl)methyl]-N-methyl-3,3a,4,5,7,7a-hexahydro-2H-furo[2,3-c]pyridine-2-carboxamide 2-[2-methoxyethyl(piperidine-4-carbonyl)amino]quinoline-3-carboxamide;dihydrochloride (3R,4S)-1-[2,6-dimethyl-5-[3-[(4-phenylcyclohexylidene)methyl]pyrazin-2-yl]pyridin-3-yl]pyrrolidin-3-ol 3-[1-[(1R)-6-chloro-4-methylsulfonyl-2,3-dihydro-1H-inden-1-yl]imidazol-4-yl]propanoic acid 1-[3,5-bis(trifluoromethyl)phenyl]-N'-ethylethane-1,2-diamine (4-benzylpiperazin-1-yl)-(7-tert-butylpyrido[2,3-d]pyrimidin-4-yl)methanone 6-[(Z)-2-amino-1-fluoroprop-1-enyl]quinazolin-4-amine 4-[3,5-bis(trifluoromethyl)phenyl]-2,2-dichlorobutanoic acid 2-(2,5-dimethylphenyl)-7H-purine N-(4,5-dihydrobenzo[b]indol-3-yl)-2-sulfanylideneacetamide N-(4-tert-butylphenyl)sulfonyl-2,3-dihydrothieno[3,2-b]pyridine-5-carboxamide 2-(2,3-dihydro-1H-indene-5-carbonylamino)-4-[5-(3-methyloxetan-3-yl)-1,2,4-oxadiazol-3-yl]butanoic acid 3-[(E)-1,2-diphenylethenyl]pyridine;iridium;2-(4-methylbenzene-6-id-1-yl)pyridine 5-methyl-3-[4-(2,2,2-trifluoroethoxy)cyclohexyl]-1,2-oxazole (5E)-3-[(2-fluorophenyl)methyl]-4,7-dioxo-6-piperidin-1-yl-2H-pyrazolo[3,4-b]pyridine-5-carbonitrile 2-[(2,4,6-trimethylphenyl)sulfonylamino]acetic acid 4-[[2-(cyclopropylamino)phenyl]methyl-(3-methoxypropyl)amino]piperidine-1-carboxamide 2-methylpropane;4-(6-phenylpyrazolo[1,5-a]pyrimidin-3-yl)aniline 5-chloro-N-[(2,3-dimethoxyphenyl)methyl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidine-7-carboxamide;ethane 6-[[2-(4-cyanophenyl)cyclopentyl]methoxy]pyridine-3-carboxamide 6-[5-(3-fluorophenyl)sulfonylhexanoyl]pyran-2-one 2-[4-chlorobutyl(2,2-diethoxyethyl)amino]benzenesulfonic acid 1-[6-(4-methylpiperidine-4-carbonyl)pyridin-2-yl]ethanone 1-(4,5-diphenylthiophen-3-yl)ethanone;ethane N-[(Z)-1H-indol-3-ylmethylideneamino]-5-nitropyridine-2-carboxamide [3-amino-6-(2,4-dimethylphenyl)pyridazin-4-yl]-[1-[4-(2-cyclopropylpyrimidin-5-yl)phenoxy]ethyl]azanium N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]ethanesulfonamide 2-[5-(4,4-dimethylcyclohexen-1-yl)pentyl]benzonitrile N-[(2S)-5-hydroxyspiro[1,3-dihydroindene-2,3'-pyrrolidine]-2'-yl]quinoline-4-carboxamide [2-(2,4-dichlorophenoxy)propylcarbamothioylamino]methanesulfonic acid 1,4-diamino-2-[6-(2-ethoxyphenyl)-3-oxo-1H-isoindol-2-yl]anthracene-9,10-dione 3-methyl-1-[2,4,6-tris(methoxycarbonyl)benzoyl]oxyindole-5-carboxylic acid 4-chloro-N-(2,5-dimethyl-1H-pyrazol-2-ium-3-yl)-8-[[4-(trifluoromethoxy)phenyl]methyl]quinoline-7-carboxamide 5-(2-methylpropanoylamino)pyridine-3-carboxamide (Z)-1-[4-[2-methyl-6-(oxetan-3-ylamino)pyrimidin-4-yl]piperazin-1-yl]-4,5-dihydro-2-benzofuran-3-ylidenemethanol N-(2,4-dinitrophenyl)sulfonyl-4-[2-oxo-3-[4-(pyridine-2-carbonylamino)phenyl]imidazol-1-yl]-3-methoxybenzamide 5-bromo-4,7-dimethyl-2H-benzotriazol-1-ium 3-[4-fluoro-2-(oxan-4-yloxy)phenyl]propanenitrile [4-[5-amino-6-[1,2-oxazol-3-yl(propan-2-ylidene)carbamoyl]pyridin-2-yl]-4-fluoropiperidin-1-yl]methanesulfinate 4-[azido(benzyl)amino]phenol N-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-(1-methoxyethyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-2-carboxamide;dihydrochloride 4-amino-2-ethylthieno[3,2-c]pyridine-7-carboxylic acid 1-[3-chloro-4-[(2,5-difluorophenyl)methoxy]-6-methylpyridin-2-yl]-4-methylidenepentan-1-one 2-[1-(4-chlorophenyl)ethylimino]imidazolidine-4,5-dione 1-(4,6-diamino-5-propylpyrimidine-2-carbonyl)azetidine-3-carbonitrile N-[6-(cyclopropylmethoxy)pyridin-3-yl]-3,5-difluoro-1H-pyrrolo[2,3-c]pyridine-7-carboxamide 7-[(2E,4Z)-2-methylhexa-2,4-dienoxy]naphthalene-1,3-disulfonic acid 1-butyl-5-[2-(1H-indol-3-yl)ethoxy]pyrazole-4-carboxylic acid 2-[(3R)-3-methylpiperidin-1-ium-1-ylidene]chromene (4R)-1-[4-chloro-3-(trifluoromethyl)phenyl]-6'-hydroxy-1,3',3'-trimethylspiro[5H-pyrrolo[2,3-c]pyridine]-4-one 2-methyl-5,8a-dihydroquinoline;2-phenylnaphthalene N-[2-(5,6-dihydrophenanthridin-12-yl)ethyl]ethanimine 5-bromo-4-cyclopropyl-2-(1,3-dioxoisoindol-2-yl)sulfanylthiophene-3-carbonitrile 2-chloro-4,5-bis(phenylmethoxy)thiophene 2-[[4-(5-chloropyridine-3-carbonyl)piperazin-1-yl]methyl]-N',N'-diethylbenzohydrazide 1-[(2,5-dichlorophenyl)methyl]piperazine;ethane 2-(5,7-dichloroquinolin-4-yl)sulfanyl-N'-hydroxyethanimidamide N-[6-[4,5-bis(ethenyl)imidazol-1-yl]hexyl]-4-chloropyridine-2-carboxamide 1-(difluoromethoxy)-6-propan-2-ylphenanthrene 5-[[(3S)-1-(cyclopropylmethylsulfonyl)pyrrolidine-3-carbonyl]amino]-2,4-difluorobenzamide 3,5-diamino-N'-(1-methyl-2H-pyridine-4-carboximidoyl)benzenecarboximidamide 2-[4-[(2R)-2,6-dimethylmorpholine-4-carbonyl]anilino]-5,11-difluoropyrimido[4,5-b][1,4]benzodiazepin-6-one 4-[5,5-bis(trifluoromethyl)-1,2,4-oxadiazol-3-yl]-N-cyclohexyl-2-nitroaniline 2-[(6S,9R)-7-(3,4-dichlorophenyl)-5-methyl-6-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]phenol (5R,7S)-7-(3,4-dimethoxyphenyl)-5-(3,4-dimethylphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine 6-[5-(trifluoromethoxy)pyrimidin-2-yl]spiro[3.4]octane 6-methyl-4-[(3R)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]oxypyridine-2-carboxamide 5-methyl-2,3-bis[(4R)-6-nitrocyclohexa-1,5-dien-1-yl]furan 7,8-difluoro-3-methyl-1H-quinolin-4-one (6R)-8-oxo-3,4,5,6-tetrahydro-2H-pyrido[1,2-h][1,7]naphthyridine-9-carbonitrile 1-[2,3-difluoro-4-(trifluoromethyl)phenyl]-N-(oxan-4-ylsulfamoyl)piperidine-3-carboxamide (7R)-2-[3-methoxy-4-[(2-nitrophenyl)methoxy]phenyl]-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide 2-(4,6-dichloropyrimidine-2-carboximidoyl)propanedioic acid 3-[2-(4-chloro-2-fluorophenoxy)acetyl]-7,9-dimethoxy-5,6,8a,9a-tetrahydropyrimido[4,5-b]quinoline-4-thione (2S,3R)-3-(3-chlorophenyl)-4-[(4-methyl-1H-pyrazole-5-carbonyl)amino]butanoic acid 4-[1-(methylamino)propan-2-yl]phthalazine-1,6-diamine 2-[(1-methylsulfanylpiperidine-4-carbonyl)amino]-3H-benzimidazole-5-carboxamide 2-[1-(4-tert-butylphenyl)sulfanylamino]-3,4,6,7-tetrahydrothieno[3,2-c]pyran-5-ol;ethane ethane;3-[2-(4-fluoro-1H-indol-6-yl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl]cyclobutan-1-amine 1-(5,6-dihydronaphthalene-2-carbonyl)piperidine-4-carboxylic acid 2-[3-(3-aminopyridin-1-ium-4-yl)propyl]isoindole-1,3-dione 1,3-dimethyl-5-[1-(2-phenylacetyl)piperidin-4-ylidene]piperidin-2-one 5-ethylsulfanyloxy-1,2,3-trimethylbenzene N-[4-(dimethylamino)-3,5-difluorophenyl]pyridine-2-carboxamide [4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]-phenylmethanone;ethane N-[5-chloro-2-hydroxy-3-(trifluoromethyl)phenyl]thiophene-2-sulfonamide 1-(2,3-dihydrothiophen-2-yl)-4-fluoroindazole 4-fluoro-3-N-methyl-2-(1H-pyrazol-4-yl)benzene-1,3-diamine ethane;2-methylbutanal;1,2,3-trifluoro-5-[4-(4-propylcyclohexen-1-yl)phenyl]benzene N-[5-chloro-2-(4-methoxyanilino)pyrimidin-1-ium-4-yl]-3,4-dihydro-2H-chromene-7-sulfonamide N-[4,5-difluoro-2-(1H-indol-4-yloxy)phenyl]-6-methylidene-8-azaspiro[3.5]nonane-8-carboxamide 3-(2,3-dihydro-1H-inden-1-yl)-1H-benzimidazole 3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]benzonitrile 5-[2-(5,6-dichlorobenzimidazol-1-yl)ethoxy]pyridine-3-carboxylic acid;hydrochloride N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethoxy]acetamide 2-(2,3-dihydroindol-1-yl)ethanol;5-[(E)-4,4-bis(methoxyphenyl)but-2-enoyl]-1H-pyridin-2-one 1-[4-(1H-indole-2-carbonyl)phenyl]cyclopropane-1-carboxylic acid 3-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-1H-imidazo[4,5-b]pyridin-2-one 3-methyl-2-(naphthalen-1-ylamino)benzenesulfinamide 3-[N'-(cyclopropylmethyl)carbamimidoyl]-4-hydroxy-5,6-dihydronaphthalene-1-carboxylic acid N-[1-(3,5-dimethoxyphenyl)ethenyl]-4-ethylaniline (2Z)-4,6-dimethylhepta-2,5-dienal;3-methoxypropanoic acid;1-[2-(pyrrolidin-1-ylamino)phenyl]ethanone N-methyl-1-[2-[(Z)-5,5,5-trifluoro-4-iminopent-2-en-3-yl]imidazo[1,2-a]pyridin-6-yl]ethanamine 2-amino-N-[(4,6-dimethylpyridin-3-yl)methyl]thieno[3,2-d]pyrimidine-7-carboxamide 4-[(2,3-dichloro-5-methoxyphenyl)sulfonylamino]-N-hydroxybenzamide 4-amino-N'-(2,6-dichlorophenyl)-1-(3-hydroxypropyl)pyrazolo[3,4-d]pyrimidine-3-carbohydrazide 2-(3-acetamidophenyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid 1-(2,6-dichlorophenyl)piperidine (2E,5Z)-4-ethylhepta-2,5-diene;2,3,7-trimethoxynaphthalene (2S,4R)-1-[(2R)-2-amino-3-phenylpropanoyl]-N-hydroxy-4-methoxypyrrolidine-2-carboxamide;hydrochloride ethane;7-[3-(2,4,5-trimethyl-3,6-dihydro-1H-pyridazine-3-carbonyl)phenyl]octanal 4-chloro-2,5-dimethyl-6,8-bis[(1R)-3-phenylcyclopenta-2,4-dien-1-yl]quinoline 1-(3,4-dihydro-2H-quinoxalin-1-yl)-N'-methoxy-N-(thiophen-2-ylmethylideneamino)ethane-1,2-diamine 2-[azido-(4-fluorophenyl)methyl]-1,3-dihydroindazole 2-azido-5-methoxy-4,6-bis(trifluoromethyl)pyrimidine 4-benzylimino-2,5-dimethoxypyrrolo[3,2-c]quinoline-1,7-dione 2-hydroxy-3-(6-methyl-1,4-dihydrobenzimidazol-5-ylidene)propanenitrile 2-[5-(4-fluorophenyl)-2-methylpyrazol-3-yl]oxy-1-phenylpropan-2-amine N-[[6-methyl-2-(oxan-4-yl)indazol-5-yl]methyl]-3-oxocyclopentane-1-carboxamide 1-butan-2-yloxy-4-[(E)-prop-1-enyl]benzene 4-(4,4-difluoropiperidin-1-yl)-5-propylpyrimidine;2-methoxy-N-methylethanamine 2-amino-6,7-difluoro-N-[4-(2-fluorophenyl)oxan-4-yl]quinoline-3-carboxamide;methane 5-(2,4-dihydroxyphenyl)-N-propan-2-ylpentanehydrazide 2-[5-bromo-4-(1,1,1-trifluoropropan-2-ylamino)pyridine-3-carbonyl]cyclohexane-1,3-dione 1-[2-[(4Z)-4-(aminomethylidene)piperidin-1-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]ethanone;ethane (6-methoxynaphthalen-2-yl)sulfamic acid 2-(N-[4-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]sulfonyl-3-nitroanilino)acetic acid 2-[4-chlorobutyl(1,3-thiazol-5-yl)amino]phenol 3-[4,5,13-triazatetracyclo[7.6.0.02,6.010,14]pentadeca-1(9),2,5,7,10,12-hexaen-8-ylmethoxycarbonyl(propan-2-yl)amino]butanoic acid 2-[5-amino-6-oxo-4-(4-phenylmethoxypiperidine-1-carbonyl)pyrimidin-1-yl]acetaldehyde;N,3-dimethylaniline N-methyl-4-[(2S)-2-methylpyrrolidine-1-carbonyl]-3H-imidazo[4,5-c]pyridine-7-carboxamide (E)-4-methyl-N,2-diphenylhex-5-enamide 2,5-dibromoterephthalaldehyde;methanol [4-(difluoromethyl)cyclohexa-2,5-dien-1-ylidene]sulfonylmethanimidamide 2-methylsulfonyloxyethylbenzene [4-[5-[4-(2,6-difluorophenyl)piperazine-1-carbonyl]pyridin-3-yl]phenyl]methanimidamide 2-[4-(3,5-dichlorophenyl)triazol-1-yl]-N-ethylpentanamide 1-[3,5-bis(trifluoromethyl)phenyl]-2-methoxyethanone 1,4-bis[2-(1,3-dioxolan-2-yl)ethyl]indole 4-[(2,6-difluorobenzoyl)amino]piperidine-1-carboxylic acid (3R)-N,4-dimethyl-1'-propanoylspiro[1H-indole-3,4'-5H-pyrazolo[3,4-b]pyridine]-2-carboxamide 5-[4-methyl-3,5-di(propan-2-yl)phenyl]-1,10-phenanthroline 4-fluoro-2-[3-(4-hydroxyphenyl)propanoylamino]butanoic acid 2-(cyclopropylmethoxy)-5-[(4,4-difluoropiperidin-1-yl)sulfonylamino]benzoic acid;2,2,2-trifluoroacetic acid 2-[4-chloro-3-(trifluoromethyl)phenyl]-1,4-dihydropyrimidine 4-amino-6-[(1-oxo-2,3-dihydroinden-5-yl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 2-(6-azidopyridin-3-yl)oxyacetonitrile 5-[(2,4-dioxo-1H-pyrimidin-6-yl)methylideneamino]-1,3-thiazole-2-carboxylic acid 1-[3-[4-(benzenesulfonamido)phenyl]propanoyl]piperidine-2-carboxylic acid 4-N-ethyl-6,7-bis(3-methoxypropoxy)quinazoline-2,4-diamine 5-fluoro-3,4-dihydroxy-6-[1-[[(2S)-pyrrolidin-2-yl]methoxy]butylamino]naphthalene-2-carboxamide 3-[2-(4-methylphenyl)ethynyl]-N-propan-2-ylidenebenzamide (1-azido-2,3,5,6-tetrachloronaphthalen-2-yl)methanol 1-[3,4-difluoro-2-(trifluoromethyl)phenyl]sulfonylpiperidine-4-carboxylic acid 2-[[(Z)-4-amino-3,5-dimethoxyhept-1-enyl]-methylamino]benzamide 2-[(3Z,5E)-hepta-1,3,5-trien-2-yl]-6-methylidenebenzo[c]chromene;9-propan-2-ylphenanthrene 4-(4,4-difluoroazepane-1-carbonyl)-3,6-dihydro-2H-pyridine-1-carboxylic acid;trihydrochloride 2-[(3S,5R)-5-methyl-1-(4-propan-2-ylbenzoyl)piperidin-3-yl]-7-(pyridine-2-carbonyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one N-[2-[(4-chlorophenyl)methyl]-3H-benzimidazol-5-yl]-4-methoxybenzenesulfonamide 3-[4-chlorobutyl(hexadecanoyl)amino]benzenesulfonic acid 2-chloro-6-(methylsulfanylamino)benzoic acid [(2R)-1-methoxypropan-2-yl]oxymethylsulfonylbenzene N-[3,5-bis(trifluoromethyl)phenyl]-6-chloro-4H-1,2,4-benzothiadiazin-3-imine 4-[3-(4-aminophenoxy)propyl]-2,6-diethoxyphenol 1-(4,5-dimethylfuran-2-yl)sulfonylpiperidine 1-[2,3-bis(ethenyl)phenyl]cyclobutan-1-amine 6-(1,2,3,5,6,7-hexahydro-s-indacen-4-ylcarbamoylsulfamoyl)pyridine-2-carboxylic acid 6-(4,4a,5,7,8,8a-hexahydropyrano[3,2-c]pyridine-2-carbonyl)-1H-quinolin-2-one 2-tert-butyl-1,3-dimethylindole;ethane N'-hydroxy-6-[methyl(thiophene-2-carbonyl)amino]pyridine-3-carboximidamide [(4R)-4-azido-2,5-dimethylhexan-3-ylidene]benzene 1-[4-(2,3-dihydroxypropyl)piperidin-1-yl]-3-phenylbutan-1-one;ethane N-[3,5-bis(4-fluorophenoxy)phenyl]acetamide (3S,4R)-1-[(5R,7R)-2-chloro-5-phenyl-6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-8-yl]piperidine-3,4-diol 3-(2,6-dioxopiperidin-4-yl)-N-[5-[hydroxymethyl(iodo)amino]pentyl]-1-methyl-1-propan-2-yloxyurea (7-methoxy-5,6,8,9-tetrahydrocarbazol-3-yl)oxyboronic acid 4-[5-(hydroxymethyl)pyrrolo[2,3-b]pyridin-1-yl]benzonitrile [5-azidooxy-1-(3,4-difluorophenyl)-2-methyl-9H-fluorene-3-carbonyl]carbamic acid N'-methyl-1-[2-(trifluoromethoxy)phenyl]pyrrole-3-carbohydrazide N'-[5,5-difluoro-2-hydroxy-4-[1-methyl-6-oxo-3-(trifluoromethoxy)pyridazin-4-yl]oxycyclohexa-2,4-dien-1-ylidene]methanimidamide 2-fluoro-6-(5,8,10-trimethyl-7,9-dihydro-6H-pyrido[3,2-h]quinazolin-2-yl)benzonitrile 2-[[1,3-dimethyl-5-(2-phenylethynyl)pyrazole-4-carbonyl]amino]ethanolate (5R,7S)-N-[2-(4-chlorophenyl)ethyl]-3-(2-methoxypyridin-4-yl)-5-(trifluoromethyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide 4-[(3,5-dimethoxyphenyl)methylamino]-2-morpholin-4-ylpyrimidine-5-carboxamide 2-cyclohexylethanamine;1,4-dihydroxy-3-nitrosoindole-5-carboxamide 2-[3-[3-(1,2,4-triazol-1-yl)phenoxy]phenyl]ethanamine ethane;1-[(E)-2-iodoethenyl]sulfonylpyrrolo[3,2-c]pyridine N-[2-(azidomethyl)phenyl]-3,4-dihydronaphthalene-1-carboxamide 4-(4-methylpiperazin-1-yl)-1H-indazole 5-[3,4-bis(4-methylphenyl)pyrrole-2-carbonyl]-1-[(1S)-1-phenylethyl]pyrrolidine-2,4-dione 5-[3,5-dichloro-4-(4-propanoylpiperazine-1-carbonyl)phenyl]-3H-1,3,4-oxadiazol-2-one [4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-[3-methoxy-2-(triazol-2-yl)phenyl]methanone 1-[[2-fluoro-4-[6-(methylamino)pyridin-3-yl]phenyl]methyl]-N,5-dimethylpyrazole-4-sulfonamide N-methyl-2-[2-(3-pentan-3-yloxyphenyl)ethenyl]aniline 4-amino-2,5-dichloro-N-[1-(3,4-difluorophenyl)cyclobutyl]benzenesulfonamide [3-methoxy-4-(2-pyridin-3-ylethynyl)phenyl]azanide 6-[[6-(4-chlorophenoxy)pyridine-3-carbonyl]amino]spiro[2.5]octane-7-carboxylic acid 1-[(2S,4R)-4-methyloxolan-2-yl]imidazo[4,5-c]pyridine (4S,5S)-3-ethyl-6,9-dimethoxy-2-oxatricyclo[8.1.12,7]hexadeca-1(16),5,7-triene 1,4-bis[(E)-3-(2,5-dihydroxyphenyl)prop-2-enoyl]piperazine-2,6-dione N-[(3S)-5,8-dioxo-2-(4,4,4-trifluorobutyl)-3,6,7,9-tetrahydro-1H-pyrazolo[3,4-b]quinolin-3-yl]acetamide 4-[(2R)-3-[1-(hydroxymethyl)cyclopropyl]-2-methoxypyrrolidin-1-yl]sulfonylbenzoic acid 1-[(2S)-2-ethenylpyrrolidin-1-yl]-3,3-dimethyl-6-[4-[[4-(trifluoromethoxy)phenyl]sulfonylamino]cyclohexyl]heptan-1-one N-cyclopropylsulfanyl-1-[(3,5-difluorophenyl)methyl]-6-methoxyindole-2-carboxamide N-azido-1-phenylpyrazol-3-amine 2-(6-chloro-1,3-benzothiazol-2-yl)cyclohexa-1,3-diene-5-sulfonamide N-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethyl)-3-hydroxypropanamide 7-(methyliodanuidylamino)spiro[3H-chromene-2,1'-cyclohexane]-4-one 2-[4-(aminomethyl)phenyl]benzoate 2-[[3-(5,6-diphenylpyridin-3-yl)benzene-4-id-1-yl]methyl]-4,6-dipyridin-3-ylpyrimidine;platinum(2+) 3-amino-4,5-dihydroxynaphthalene-1,2-disulfonic acid 6-(4-methoxy-3,5-dimethylpyridin-2-yl)-4H-1,4-benzoxazin-3-one 4-[6-methoxy-5-(2-methylpropoxy)pyridin-3-yl]-N,1-dimethylpyrazolo[3,4-b]pyridine-6-carboxamide 2-chloro-N-[(5-methylimidazo[1,2-a]pyridin-2-yl)methyl]benzamide 3-[(E)-2-(aminomethyl)-3-fluoroprop-2-enoxy]-N-[(1R,2S)-4-fluoro-2-hydroxycyclopentyl]benzamide N-methyl-1,2-bis[(4-methylpiperazine-1-carbonyl)oxy]-3-propan-2-ylsulfonylimidazole-4-carboxamide (5-methylpyrazin-2-yl)-[3-[6-(trifluoromethyl)pyridin-3-yl]piperidin-1-yl]methanone 5-benzylsulfanyl-1,4-dimethylpyridin-2-one 3-(5,6-dimethylcyclohexa-1,3-dien-1-yl)-2-N,4-N-bis(4-ethoxyphenyl)naphthalene-2,4-diamine 5-(4,6-dimethylpyrimidin-2-yl)-3a-benzoyl-3-methyl-1,2,4,6-tetrahydropyrrolo[3,4-c]pyrrole-6a-carboxylic acid N-[(3S,4R)-1-benzyl-4-methoxypyrrolidin-3-yl]-2-(5-ethyl-1,3,4-oxadiazol-2-yl)acetamide 3-[[5-azido-2,6-dimethyl-4-[[(1R)-1-phenylethyl]amino]pyridine-3-carbonyl]amino]propanoic acid 6-[2-(4,4-difluorocyclohexyl)ethynyl]-7H-purine (Z)-3-[2,6-dichloro-4-[4-(trifluoromethylsulfanyl)phenoxy]phenyl]-3-hydroxyprop-2-enal 3-[(3-bromo-4-methoxyphenyl)sulfonylamino]cyclobutane-1-carboxylic acid 5-[2,3-dihydroxypropyl(1,1,1,2,3,3,3-heptafluoropropan-2-yl)amino]naphthalene-2-sulfonic acid 6-azido-5,11,14-triazapentacyclo[10.7.0.02,10.04,8.013,18]nonadeca-1(12),2,4(8),9,13,15,17-heptaene (E)-2-(benzenesulfonyl)-3-[(4-methylphenyl)methyl]but-1-en-1-amine 2-(2-azidocyclopropyl)-1,3-dichloro-5-methoxybenzene N-[5-(1,3-benzodioxol-5-yl)-2-[4-(hydroxymethyl)piperidin-1-yl]phenyl]-6-ethoxypyridine-2-carboxamide;hydrochloride 1,3-bis(3-chlorophenyl)urea N-[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-(4-methylpiperidin-1-yl)pyrido[3,4-d]pyrimidin-2-yl]azetidine-2-carboxamide [(3S,4R)-1-benzyl-4-methoxypiperidin-3-yl]-[4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone 6-[(6-aminopyrimidin-4-yl)amino]spiro[3.5]nonan-2-one N-butyl-2-(5-ethynylpyridin-3-yl)propanamide 2-cyclopropyl-4,5-dimethoxybenzamide N-(4-acetylphenyl)-2,2-dimethoxyacetamide 2-methyl-1',7-dipyridin-4-ylspiro[3H-isoquinoline-4,5'-azepane] 5-(1,3-benzothiazol-2-yl)-6-methoxypyridine-3-carbonitrile 4-[N-(4-bromobutan-2-yl)-2,5-dichloroanilino]benzenesulfonic acid 7-(4-chlorophenyl)-2,5,7-trimethyl-N-[3-methyl-1-(oxan-4-ylamino)-1-oxobutan-2-yl]-6H-pyrazolo[1,5-a]pyrimidine-3-carboxamide (2S,3aS,7aS)-6-[(1-methylpyrazol-4-yl)methyl]-N-pyrimidin-2-yl-3,3a,4,5,7,7a-hexahydro-2H-furo[2,3-c]pyridine-2-carboxamide;2,2,2-trifluoroacetic acid 3-N,6-dimethylbenzene-1,2,3,4,5-pentamine;N-hydroxypyridine-2-carboxamide N-[5-chloro-1-(2,4-difluorophenyl)imidazole-4-carboximidoyl]-3,6-dihydro-2H-pyran-4-carboxamide (2S,4R)-4-phenylmethoxypentane-1,2,3-triol 3-azidooxysulfonylbenzamide 5-chloro-2-fluoro-N-[3-(4-oxo-1-phenyl-5H-pyrazolo[3,4-d]pyrimidin-6-yl)pyrrolidin-1-yl]benzamide 4-[3-chloro-2,6-dimethyl-8-(trifluoromethoxy)imidazo[1,2-a]pyridin-7-yl]oxy-2-ethyl-2-methylbutanenitrile 7-[(E)-1,4,4-triaminobut-2-enylidene]naphthalene-2,8-dicarbonitrile N-[4-(cyclopropylamino)sulfanylphenyl]acetamide 1-[(2R,4S)-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-5-methylpyrimidine-2,4-dione 4-[(2,5-dimethylimidazo[1,2-a]pyridin-6-yl)sulfamoyl]-N-hydroxybenzamide [3-(2-aminoanilino)piperidin-1-yl]-phenylmethanone 1-[3-(4-chlorophenyl)-2H-cyclopenta[b]naphthalen-1-ylidene]propan-2-one 4-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide 3-[4-(aminomethyl)phenoxy]cyclopentan-1-one;hydrochloride (3S,4R)-N-[[6-methyl-5-[3-(trifluoromethyl)phenyl]pyridin-2-yl]methoxy]-4-[1-(oxan-4-ylamino)ethenyl]pyrrolidin-3-amine (2R)-1-acetyl-N-[4-[6-[3-[2,3-bis(methoxymethyl)phenyl]-5-[(3S)-oxolan-3-yl]oxyphenyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl]pyrazol-1-yl]azetidine-2-carboxamide 1-cyclopentyl-3-[4-(2H-tetrazol-5-yl)phenyl]thiourea 5-butanoyl-3,3-diethyl-1-methylindol-2-one N-ethenyl-1,2-dimethoxybenzenesulfinamide 2-methoxypropane;4,9,10-trihydroxyphenanthrene-3,6-dione N-[(3R,4S)-1-benzyl-4-(2H-triazol-4-ylmethylcarbamoyl)pyrrolidin-3-yl]-5-cyclopropyl-1,3-oxazole-4-carboxamide 2-(6,11-dihydro-5H-benzo[b][1]benzazepin-3-yl)-N-oxoacetamide N-[2-(3,5-difluorophenyl)-1-hydroxy-3H-isoindol-1-yl]benzamide 6-azidooxynaphthalene-2-sulfonic acid 3-(4-chloro-2-fluorophenyl)-1-[1-(4,5,6,7-tetrahydro-1H-indazole-6-carbonyl)piperidin-4-yl]imidazolidin-2-one 1-[3-(2,4-dimethylphenyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylic acid 3-ethyl-6,8-diphenylimidazo[1,2-a]pyrazine 4-(diethylaminomethyl)-2-methylisoindole-1,3-dione 1-(3-benzoylanilino)butane-2,3-dione [2-(1,3,4-oxadiazol-2-yl)phenyl]carbamodithioic acid 5-[4-(dimethylamino)cyclohexyl]-3-phenylmethoxypyridine-2-carboxylic acid N-azido-1,3-benzodioxol-5-amine 7-chloro-4-(3,5-dimethylanilino)chromen-2-one 2-bromo-N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-(2,2-dimethoxyethyl)benzamide 3-(2,6-dichlorophenyl)-7-[4-(5-methyloxolan-2-yl)anilino]-2H-pyrimido[5,4-e][1,3]thiazin-4-one 6-[3,5-difluoro-2-(1H-indol-4-yloxy)phenyl]-N-[(3E)-hexa-1,3,5-trien-3-yl]pyrimidin-4-amine 2-azido-1,4-difluoronaphthalene 2-(4-bromo-3,5-dimethoxyphenyl)morpholine 3-amino-2,4,5,6-tetradeuterio-N-(2-methylbutan-2-yl)benzamide 2-methyl-4,5-bis[3-(trifluoromethoxy)phenyl]thiophene 3-amino-N,6-dimethylbenzenesulfonamide;7H-1,4-benzodioxine 3-(3,5-dimethylphenyl)-6-fluoro-7-(4-iodopiperazine-1-carbonyl)-9H-pyrido[2,3-b]indole-1-carboxamide 2-[6-(4-chlorophenyl)pyridin-3-yl]-N,N'-bis[(E)-1-hydroxybutan-2-ylideneamino]ethanimidamide N-[4-(1,2-benzoxazol-3-yl)piperidine-1-carbothioyl]-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-3-carboxamide (2S)-3,4-dimethyl-2-(methylamino)-N-[5-(propanoylamino)naphthalen-1-yl]pentanamide 2-benzylsulfanyl-3,6-dihydropyrido[2,1-a]isoindole 4-[[8-methyl-2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-7-yl(propanoyl)amino]methyl]benzoic acid 1-[2-(dimethylamino)ethyl]-3,4-bis(phenylmethoxy)pyridin-2-one 2-amino-6-[4-[(dimethylamino)methyl]phenyl]-7,8-dihydro-5H-1,6-naphthyridine-3,4-dione 6-(2,3-dichlorophenyl)-8-methoxy-N-[4-[(2R)-oxolan-2-yl]butan-2-yl]quinazolin-4-amine N-(4,6-dimethyl-2H-pyrazolo[3,4-c]pyrazol-3-yl)-1H-benzimidazole-5-carboxamide 2-methyl-6-[1-[4-(3,5,5-trimethylcyclohexa-1,3-dien-1-yl)phenyl]imidazol-2-yl]quinoline N-[4-(2-aminopyrimidin-5-yl)-3-cyanophenyl]-5-(1,5-dimethylpyrazol-4-yl)pyridine-3-carboxamide 1-[4-[(3,4-difluorophenyl)methyl]-5-fluoro-6-oxo-1H-pyrimidine-2-carbonyl]piperidine-4-carboxylate N-[3-(2,6-dioxopiperidin-1-yl)phenyl]aziridine-2-carboxamide;hydrochloride 2-(3,5-dichloropyridin-4-yl)acetamide 3,5-dimethylhexane;N-(4-ethenylphenyl)-2-(3-methylphenyl)aniline 1-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-3-sulfonamide 1-(2,2-dimethylchromene-6-carbonyl)-3,4-dihydro-2H-quinoline-8-sulfonamide 7-azidooxy-1-[(3S)-piperidin-3-yl]benzimidazole 1-[1-[(5S)-4,7-dioxo-2-[[4-(trifluoromethylsulfanyloxy)phenyl]carbamoylamino]-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]-3-methylbutylidene]-3-pyridin-4-ylurea 4-(5,7-dimethylquinoxalin-6-yl)oxyaniline 3-(dimethylamino)-1-[4-[7-morpholin-4-yl-2-(4-pyridin-3-ylanilino)thieno[3,2-d]pyrimidin-4-yl]pyrazol-1-yl]propan-1-one 2,6-dimethyl-1-[(2R)-3-methylidene-2-propanoylcyclopenten-1-yl]benzimidazole-5-carboxamide 2-[(1S)-1-[2-methyl-4-(trifluoromethoxy)phenyl]ethyl]propanedinitrile 2,4-dichloro-1-[2-(3,5-dichlorophenyl)-1-hydroxyethoxy]-6-fluoro-10H-acridin-9-one 1-(3,4-difluorophenyl)sulfonyl-N-(2-oxospiro[6H-furo[2,3-f]chromene-3,4'-oxane]-5-yl)piperidine-4-carboxamide 2-[4-(3,5-dimethylpyrazol-1-yl)-3,6-dihydro-2H-pyridine-1-carbonyl]benzoic acid 7-(4,5-dihydro-1H-imidazol-2-yloxy)naphthalene-2-carboxylic acid (2R)-2-amino-3,3-dimethylbutanoic acid;1-[4-[4-[2,6-bis(trifluoromethoxy)phenyl]benzoyl]piperazin-1-yl]prop-2-en-1-one (2-ethylpyrrolidin-1-yl)-[4-methoxy-5-methyl-6-[(7R)-7-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]pyridin-3-yl]methanone 3-[2,5-dimethyl-4-[2-(oxan-2-yloxy)ethylamino]phenyl]-3-[5-[(4R)-6-hydroxy-1,3-thiazepane-4-carbonyl]pyridin-3-yl]propanoic acid 3-methyl-N-[2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)ethyl]pyridine-4-carboxamide;dihydrochloride 3-[(2R,4R)-6-fluoro-2-phenyl-1-propanoylpiperidin-2-yl]propanoic acid 4-[2,4-bis(sulfanyl)phenyl]butanenitrile 4-[4-[2-(6,7-difluoronaphthalen-1-yl)ethynyl]phenyl]benzonitrile N-(3,4-dichlorophenyl)-2-[1-(4-methoxyphenyl)-4-oxo-5H-pyrazolo[3,4-d]pyrimidin-6-yl]acetamide [2-(aminomethyl)piperidin-1-yl]-[4-methoxy-3-(1H-pyrazol-5-yloxy)phenyl]methanone;dihydrochloride (2S)-2-[3-chloro-5-fluoro-6-(4-fluoropyridin-2-yl)oxy-9,10-dihydroanthracen-2-yl]propanoic acid 2-[(3,4-dichlorophenyl)sulfonyl-(2-oxoethyl)amino]acetic acid 2-[4-[(3R)-1-benzylpiperidin-3-yl]phenyl]propanal (2R)-3-[4-[6-[(3S,5R)-3,5-dimethylpiperazin-1-yl]pyridin-3-yl]pyrazol-1-yl]sulfonylpropan-2-ol 2-N,4-N-dibenzylcyclohexane-1,4-diimine 7-chloro-3,4-dihydro-1H-benzo[h]quinoxalin-2-one N-[6-chloro-1-(2,3-dihydro-1H-inden-1-yl)benzimidazol-2-yl]-2-methoxybenzamide 2-[4-bromo-N-(3-methylbut-2-enyl)anilino]phenol N-(3,4-dihydro-1H-isochromen-1-yl)-6-morpholin-4-ylpyridine-2-carboxamide 2-[3,5-dichloro-4-(3-cyano-4-methylsulfonylphenoxy)phenyl]acetamide 3-[1-(2-methoxyethyl)piperidin-4-yl]-6-methylimidazo[1,2-a]pyridine 2-[5-chloro-4-ethyl-1-(6-methoxypyridin-3-yl)pyrazole-3-carbonyl]butanedioic acid 3-[4-(2,6-dimethylphenoxy)piperidine-1-carbonyl]thiophene-2-carbonitrile N-[1-(4-methoxyphenyl)ethyl]-3-oxobutanamide 2-(azidomethyl)-6-ethylsulfonylpyridine (2-ethoxypyridin-3-yl)-[3-(1H-imidazol-5-ylmethyl)piperidin-1-yl]methanone 3-[(3,4-dichlorophenyl)methyl]-7H-purine-2,6-dione (4R)-1-[4-[3,5-bis(trifluoromethyl)phenyl]butanoyl]-N-cyclopropyl-4-hydroxypyrrolidine-2-carboxamide 2-[3-chloro-5-(1H-indol-3-yl)phenyl]-6,8-dimethoxy-2-methyl-1,3-dihydroquinazolin-4-one 6-[2,4-dichloro-3-(trifluoromethyl)phenyl]-2H-pyran 1-(2,3-dihydropyridin-4-yl)-2-methyl-5-phenylindole 1,5-dichloro-2-[(3-fluorophenyl)methyl]pentan-3-amine (E)-1-(5-chloro-2,4-dihydroxyphenyl)-3-[5-chloro-6-[(Z)-prop-1-enyl]pyridin-2-yl]but-2-ene-1,4-dione ethane;4-[(4E,7Z)-6-methylidene-4-propan-2-yl-2-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)octa-1,4,7-trienyl]-5-phenyl-2,6-bis(trichloromethyl)pyridine 3-[4-[2-(aminomethyl)-5,6-difluoroindole-1-carbonyl]piperazin-1-yl]benzonitrile;hydrochloride 3-ethyl-5,7-dimethoxy-N'-(1H-pyrrolo[2,3-b]pyridin-4-yl)isoquinoline-8-carbohydrazide (3S)-4-(7,8-dihydronaphthalene-1-carbonyl)-N-methylmorpholine-3-carboxamide 3-[(2,4-difluorophenyl)methyl]-5-methoxy-1H-indole 2-chloro-5,6,8,9-tetrahydropyrido[2,3-d]azepine 4-azido-3-methoxy-2H-benzotriazole 2-[(1R)-5-bromo-2,3-dihydro-1H-inden-1-yl]propanoic acid (2R)-2,3-dihydroxy-1-(2H-indol-4-ylmethyl)piperidine-4-carboxylic acid 1-ethyl-3-[4-methoxy-2-[5-[1-(6H-pyrrolo[2,3-b]pyrrole-1-carbonyl)cyclobutyl]pyridin-2-yl]phenyl]urea N-[2-(2,3-dihydroindol-1-yl)ethyl]-1-(4-oxo-1H-pyridine-2-carbonyl)piperidine-4-carboxamide 2-(4-methoxyphenyl)-N-[2,4,6-trichloro-3-[(4-sulfanylidenepyrido[1,2-a]pyrimidine-3-carbonyl)amino]phenyl]acetamide (Z)-N'-[2,4-bis(5-methoxypentylsulfanyl)phenyl]-3-hydroxyprop-2-enimidamide 2-[(1R,5S)-3-(4,6-difluorocyclohexa-2,4-dien-1-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-6-methoxypyridine-4-carboxylic acid N-(5-tert-butyl-2,3-dihydro-1H-inden-1-yl)-6-oxo-4-phenyl-1H-pyrimidine-5-carboxamide 2-[(4-methylphenyl)iminomethyl]-N,N'-diphenylethane-1,2-diamine 3-[4-amino-7-methyl-6-[4-(2,2,6,6-tetramethylpiperidin-4-yl)oxyphenyl]pyrrolo[2,3-d]pyrimidin-5-yl]benzaldehyde 6-hydroxy-4,5-dimethyl-1H-benzo[f]indole-3-carboxylic acid 4-(3,5-dibromophenyl)-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 2-(9H-fluoren-1-yl)-3-[(3S,4R)-3,4,5-trihydroxyoxan-2-yl]oxypropanenitrile [(2S)-1-hydroxy-3-phenylpropan-2-yl]-diphenylphosphane 1-[4-(2-methoxyethoxy)phenyl]-5H-pyrazolo[3,4-d]pyrimidin-4-one 1-[2-methyl-4-(morpholine-3-carbonyl)phenyl]-1,5-naphthyridin-2-one 1-(2,3-difluorophenyl)pentan-3-ol;2-ethylpyridine-4-carboxylic acid 3-(2-methoxyphenyl)-N,N-dimethylpyrrolidine-1-sulfonamide 4-[1-(6,7-dihydrothieno[3,2-d]pyrimidin-4-ylamino)ethyl]phenol 3-(hydroxymethyl)-1-(5H-pyrrolo[2,3-b]pyrazin-2-yloxy)pentan-2-ol 2-(1,3-dihydroisoindol-2-yl)-N'-methoxyacetohydrazide N-[5-cyclopropylsulfonyl-4-(6,7-dimethoxyquinolin-4-yl)sulfanylthiophen-2-yl]acetamide (2S)-1-(6-methylpyridine-3-carbonyl)pyrrolidine-2-carboxamide 1-[3,4-dichloro-5-(trifluoromethyl)phenyl]ethanol N-[4-amino-3,4-dioxo-1-(1H-pyrrol-2-yl)butan-2-ylidene]-4-pyrazin-2-ylbenzamide (4-butylcyclohexyl)benzene 7-(2,4-dihydroxy-5-propan-2-ylphenyl)-2-[3-[[4-[[6-(methylamino)pyridine-3-carbonyl]amino]piperidin-1-yl]methyl]anilino]-N,N-dimethylacetamide;dihydrochloride 4-(2-methyl-5,6,7,8-tetrahydropyrido[3,2-d]pyrimidin-4-yl)morpholine 2-(8-azaspiro[4.5]decan-8-yl)-6-(3,5-dimethoxyphenyl)-N,N-dimethylpyrimidin-4-amine 2-[5-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]phenol N-[4-(trifluoromethoxy)phenyl]sulfanylpentanamide N-cyclohexyl-2,4,6-trimethylaniline 5-azido-3-(4-bromophenyl)thiophene-2-thiol 2-tert-butyl-7-[(2,5-dimethoxyphenyl)methyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 5-[(E)-2-(4-tert-butylphenyl)ethenyl]-N-[3-hydroxy-4-methoxy-1-(6-methoxypyridin-3-yl)butan-2-yl]-2,3-dihydroindole-1-carboxamide 6-[3-(5-chloropyridin-2-yl)-1,2,4-oxadiazol-5-yl]-4H-1,3-benzoxazin-2-amine [2-(aminomethyl)-4-phenylpiperazin-1-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone;dihydrochloride 4-[5-amino-6-(methylamino)pyridin-3-yl]-N,2-dimethylbutanamide;cyclohexane 3-[2-(3,5-dimethylcyclohexen-1-yl)ethynyl]pyridine 4-azido-2-methylsulfonylpyrimidine N-[(3R,4S)-1-(8H-cyclohepta[b]pyridin-5-ylsulfonyl)-4-methoxypyrrolidin-3-yl]acetamide 4-[2-(2,3-difluorophenyl)pyrrolidin-1-yl]-5-methoxypyrimidine (5Z)-2-cyclopentylimino-5-[[4-ethoxy-3-methoxy-5-[(3S,5R)-3,4,5-trimethylpiperazine-1-carbonyl]phenyl]methylidene]-1,3-thiazolidin-4-one 3-(2,5-dihydroxyphenyl)-4,5-dihydro-1H-pyridazin-6-one (7R)-5-methyl-N-phenyl-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide (4-fluorophenyl)methyl-diphenylsulfanium;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide 4-[2-[1-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidine-2-carbonyl)piperidin-4-yl]propoxy]benzoic acid [4-[[8-(3-chloropyridin-2-yl)-1,4-dioxaspiro[4.5]decan-8-yl]methoxymethyl]-2-fluorophenyl]methanethiol 1-cyclohexyl-2,4-dimethylbenzimidazole;6-(dimethylamino)pyrimidine-4-carboxamide 2-(ethoxymethyl)-4-[5-methoxy-6-(2,2,3,3,4,4,4-heptafluorobutoxy)pyridin-2-yl]-1H-pyrimidin-6-one 4-[2-aminoethyl(3,3-dimethoxypropyl)amino]-N'-hydroxypyridine-2-carboximidamide [4-(2,6-dimethylanilino)pyrazole-1-carboximidoyl]-[5-[[(3Z,6E)-6-fluoroocta-1,3,6-trien-2-yl]amino]-2-piperidin-1-ylpyridin-3-yl]azanium 7-[(6,7-dimethoxyquinolin-4-yl)amino]-N-hydroxy-3H-benzimidazole-5-carboxamide 1-[(E)-4-(diethylamino)but-2-enyl]-N,5-dimethoxypyrazole-3-carboxamide N-(2,3-dichlorophenyl)-3-[1-ethylsulfonyl-4-(trifluoromethyl)pyrrolidin-2-yl]imidazo[1,5-a]pyrazine-1-carboxamide 1-ethyl-2,4-difluorobenzene;6-[5-methoxy-3-[(3S)-oxolan-3-yl]-4-oxoquinazolin-7-yl]-1H-pyrrolo[3,2-c]pyridine-3-carboxamide N-(3,3,3-trifluoro-2-methylpropyl)pyrido[4,3-d]pyrimidin-8-amine (1R)-2,3,4,9-tetrahydro-1H-carbazole-1-carboxylic acid 3-[N-(2,3-dihydroxypropyl)-4-hydroxyanilino]butanoic acid (1S)-2,2-dimethyl-N-[5-[6-[5-methyl-6-[2-(3-morpholin-4-ylpropoxy)ethyl]pyridin-2-yl]thieno[3,2-d]pyrimidin-4-yl]oxy-1,3-thiazol-2-yl]cyclohexane-1-carboxamide 3-[4-(3,4-dichlorophenyl)piperazin-1-yl]propanal 2-[1,3-dioxo-4-(pyridine-2-carbonyl)isoindol-2-yl]acetamide N-(2,6-difluorophenyl)sulfanylformamide;N-[1-(4-methoxypyridin-3-yl)ethyl]formamide 1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-[6-(1H-pyrazol-5-ylmethylamino)pyrimidin-4-yl]ethanone (1R,2S)-2-[7-chloro-3-[5-chloro-3-fluoro-4-[6-(oxetan-3-ylmethoxy)pyridin-3-yl]phenyl]cinnolin-4-yl]cyclopropane-1-carboxylate 5-(2,6-dichlorophenyl)-3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-N-methyl-1,2-oxazole-4-carboxamide 1-(2,5-dimethoxyphenyl)sulfonyl-2-fluoropyrrolidine 2-(3,4,5-triethoxyanilino)ethanol 2-tert-butyl-5-(phenyliminomethylamino)benzenesulfonic acid;chromium(3+);dichloride N-[(1R,5S)-6-bicyclo[3.2.0]heptanyl]-4-methylbenzamide 2-[(1R,3S)-1-benzyl-4-chloro-3-methylnaphthalen-2-yl]acetate 3-(8,9-dimethoxy-5H-benzo[c]phenanthridin-6-ylidene)propanal 3-[5-bromo-4-(4,4,5,5-tetramethyloxaborolan-2-yl)pyrazol-1-yl]benzonitrile 3-[(2R)-1-(1,1-difluoropropylsulfonylamino)butan-2-yl]-5-fluoro-N'-hydroxybenzenecarboximidamide N-(4-bromophenyl)sulfonyl-2,3-difluorocyclohexane-1-carboxamide 1,4-dichloro-3-methoxy-2-(trifluoromethyl)benzene 2-[3,6-bis(9H-fluoren-1-yl)-1-benzothiophen-2-yl]aniline N-[3-(1H-benzimidazole-2-carbonyl)-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl]-3-cyanobenzamide 2-[3-fluoro-4-(trifluoromethyl)phenyl]-5-hexoxypyrimidine 2-[[(Z)-1-cyano-3-cyclopentylprop-2-enylidene]amino]naphthalene-1,4-dione 1-azido-2,4-difluoro-5-methoxynaphthalene 4-[2-(5,6-dihydronaphthalene-1-carbonylamino)-4-(4-fluorophenyl)thiophen-3-yl]benzoic acid N-[(E)-(4,6-dichlorocyclohexa-2,4-dien-1-ylidene)amino]-3-methyl-1H-pyrrolo[2,3-c]pyridine-7-carboxamide 3-amino-N-(1,2-oxazol-5-yl)-4-(pyrrolidin-1-ylmethyl)benzamide ethane;1-(6-fluoro-3,4-dihydro-2H-chromen-5-yl)propan-1-one 4-[(1R,2S)-1-aminospiro[2,3-dihydronaphthalene-4,4'-piperidine]-1-yl]benzoic acid N-[5-(methoxymethyl)-1H-pyrazol-3-yl]naphthalene-2-carboxamide 2-azido-4-phenyl-1H-indole 7-[5-(4,6-diphenylpyridin-2-yl)oxypentoxy]-1H-indazole;ethane (E)-3-[1,2-bis(ethenylsulfanyloxymethoxy)propoxy]-N-propanoylbut-2-enamide;4,7-diamino-5-bromonaphthalene-2-sulfonic acid;(Z)-1,4-dimethylhept-4-ene 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]propanoic acid ethane;2-[4-(methoxyamino)phenyl]-1H-indole-5,6-diol [4-amino-2,5-di(propan-2-yl)phenyl]-cyclohexylmethanethione;1-formamidoformamide 2-amino-4-methyl-5-(thiophene-3-carbonyl)thiophene-3-carbonitrile 2-[5-(1,3-benzothiazol-6-yl)pyridin-2-yl]-N-(4-cyanophenyl)acetamide 1-(3,4-diethylphenyl)-4-methoxypiperidine N-[2,5-dimethyl-1-(4-phenoxyphenyl)cyclohexa-2,4-dien-1-ylidene]hydroxylamine (2S)-4-methylsulfanyl-N-(1,3-thiazol-5-yl)pyrrolidine-2-carboxamide 3-(5,6-difluoro-1H-indole-2-carbonyl)-4H-[1,2]oxazolo[4,5-d]pyrimidin-7-one N-[(3R)-piperidin-3-yl]quinolin-5-amine 5-[(3,4-dichlorophenyl)methyl]thiophene-2-sulfonamide (4R)-1-[5-chloro-2-methoxy-6-(trifluoromethylsulfanylamino)pyrimidin-4-yl]piperidine-4-carboxylic acid 4-[(2,6-difluorophenyl)methyl]benzenesulfinate 2-methylsulfonyl-N-[6-(1,3-oxazol-5-yl)cinnolin-3-yl]acetamide N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)cyclopentanecarbonyl]propanamide ethane;1-[4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]oxyphenyl]butan-2-one (2R)-2-[3-oxo-1,4-diphenyl-5-(trifluoromethyl)-2H-pyrazin-6-yl]propanoate N-(5,6-dimethylpyridin-3-yl)-4-ethoxybenzamide 3-[1-[4-(aminomethyl)phenyl]ethenoxy]-5-fluoro-6-[2-[2-(1-fluorocyclopropyl)ethyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]pyridine-2-carboxylic acid;ethane N-[[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)phenyl]methyl]acetamide;hydrochloride (2S)-6-amino-2-[4-chloro-3-[(5-methylsulfanylpyrimidin-2-yl)carbamoyl]anilino]hexanoic acid 5-tert-butyl-3-ethynyl-1H-pyrrolo[2,3-b]pyridine 1-[5-cyano-2,6-dimethyl-3-(1H-pyrazol-4-yl)indol-1-yl]propane-2-sulfonic acid 1-(2,6-dimethylpyridin-4-yl)-3-[[(3R)-pyrrolidin-3-yl]amino]piperidin-2-one;dihydrochloride 2-ethoxy-6-methyl-5,6-dihydroimidazo[1,2-b]pyridazine [4-(1,3-benzoxazol-2-ylmethoxy)cyclohexa-1,5-dien-1-yl]-piperidin-1-ylmethanone 2-[[4-[2-(1,3-benzodioxol-5-ylamino)propyl]-3-fluorophenyl]methoxy]ethanimidamide N-[5-tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide 4-[(3R)-1-azidopiperidin-3-yl]oxyaniline 5-ethyl-2,4-dimethoxybenzenesulfonate 2-[(6,7-dimethoxyquinolin-4-yl)amino]oxy-3H-pyrido[3,4-d]pyrimidine-4,7-dione [3-[(1S)-2,2-dimethylcyclohexyl]cyclopenta-1,4-dien-1-yl]benzene 2-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-5-yl)-N,N-dimethylacetamide;ethane 2-(1H-indole-3-carbonylamino)-3,4-dihydro-1H-isoquinoline-5-carboxylic acid 2-[(3S)-3-hydroxy-1-methylpiperidin-4-yl]oxypyridine-3-carboxamide 2-[4-[5-chloro-6-(3,3,3-trifluoropropylamino)pyridin-2-yl]-1H-pyrazol-5-yl]-N-[(1S)-1-naphthalen-1-ylethyl]acetamide 2-cyclohexyl-1-[3-(dimethylamino)-4-methoxyphenyl]ethanesulfonic acid 4-[2,3-dimethoxy-5-(trifluoromethyl)phenyl]-1-propan-2-ylpyrazole N-azido-6,11-dihydrobenzo[c][1]benzazepine-5-carboxamide 2-ethylsulfanyl-6-(2-pyridin-4-ylphenyl)phenol 3-(4,5-dimethylcyclohexen-1-yl)-1-[4-(dimethylamino)phenyl]prop-2-yn-1-one 2-(4-fluorophenyl)-N-methyl-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine-3-carboxamide 1-(2,3-dimethoxy-1H-inden-1-yl)piperidine N-azido-N-benzyl-2-[(5-cyanopyridin-3-yl)methoxy]acetamide 5-amino-6-[(3Z)-2-fluorohexa-1,3,5-trien-3-yl]pyridine-3-carboxamide 2-amino-9-[1-[4-(cyclopropylmethoxy)-3,5-di(ethoxy)phenyl]-5-oxopentan-2-yl]-1H-purin-6-one 2-[4-[1,2-bis(4-methylphenyl)ethylideneamino]phenoxy]-2-methylpropanoic acid N-[(2S)-4,4-difluoro-1-[[5-(trifluoromethyl)pyrimidin-2-yl]amino]butan-2-yl]-1,2-oxazole-3-carboxamide 7-[(3S)-3-hydroxypyrrolidine-1-carbonyl]spiro[3H-pyrido[2,3-d]pyrimidine-4,1'-cyclobutane]-2-one 3-[5-fluoro-2-(hydroxymethyl)phenyl]imidazo[4,5-b]pyridine-7-carboxylic acid 2-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-N-(2,4-dichloro-5-nitrophenyl)acetamide 4-N-[2-(dimethylamino)ethyl]-1-ethanimidoylnaphthalene-2,4-diamine 3-[2-methoxyethyl(propyl)amino]pyrazine-2-carboxamide N-[[4-(1,1-difluoroethyl)phenyl]methyl]-2-[2-[3-fluoro-4-(trifluoromethoxy)phenoxy]propanoylamino]quinoline-6-carboxamide N-[2,6-di(propan-2-yl)phenyl]-1-[5-hydroxy-4-methoxy-2-(oxidoamino)phenyl]methanesulfonamide 2-(3,5-dihydroxyphenyl)sulfanylbenzenethiol 4-(cyclohexylamino)-3-[6-(3,5-dimethylphenoxy)pyrimidine-4-carbonyl]-1-methylidene-2H-isoquinoline-7-carbonitrile 2-[6-fluoro-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonyl)indol-1-yl]acetaldehyde 5-[2,3-dimethylbutanoyl(propan-2-yl)amino]-2-(furan-2-carbonylamino)benzoic acid 4-(methylideneamino)-6-(2,3,5-trifluorophenyl)pyrimidin-5-ol 6-[4-amino-1-[(2,5-difluorophenyl)methyl]pyrazolo[3,4-d]pyrimidin-3-yl]-1H-benzimidazole-4-carboxamide 5-[3-(2-methylpyridin-4-yl)phenyl]imidazolidine-2,4-dione N-(4-chlorophenyl)-7-(2,6-difluorophenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide 4-bromo-1-chloro-2,3,5,6-tetrafluorobenzene;ethane 5-(3-chlorophenyl)-2,4-dihydroxypyrrole-1-carboxylic acid N-[(3E)-2,6-dimethylhepta-1,3,5-trien-4-yl]ethanethioamide;1-[5-ethynyl-3-ethoxy-2-[[3-hydroxypropyl(pyridin-2-ylmethylsulfanyl)amino]methyl]phenyl]ethanone 2-[4-(1H-indazole-3-carbonylamino)pyrazol-1-yl]acetic acid (Z)-2-cyano-3-[4-(4-methylimidazol-1-yl)phenyl]prop-2-enamide 1-[3,4-bis(ethenyl)cyclohexa-1,5-dien-1-yl]-2-methylbenzene;ethane 2-[[5-(cyclopropylamino)-3-ethyl-1,6-dimethylpyrazolo[4,3-g]quinoxalin-7-ylidene]amino]oxyethanol 2,6-dichloro-4-phenyl-N-[1-(3-piperidin-1-ylpropoxy)indol-5-yl]aniline 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-6-fluoroquinoline 1-methyl-N-(1,3-thiazol-2-yl)-4-[2-[4-(trifluoromethoxy)phenyl]ethynyl]pyrrole-3-carboxamide 1,2-dimethyl-9H-carbazole-3-carbohydrazide 5-(2,6-dioxopiperidin-3-yl)-N-[1-[4-fluoro-2-[1-[[2-(methylamino)ethylamino]methyl]pyrazol-4-yl]phenyl]ethenyl]pentanamide 6-[3-(2,4-dimethylphenyl)-5-nitrophenyl]hexanoic acid 2-(3-fluorophenyl)-N-[(3R,4S)-3-hydroxypiperidin-4-yl]-3H-benzimidazole-5-carboxamide N-[[4,5-bis(difluoromethyl)furan-2-carbonyl]amino]propane-1-sulfonamide 2-(N,5-dimethyl-3-oxo-1H-isoindol-2-yl)-N-[1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl]acetamide 3-[3-(4,4-dimethylpentanoylamino)pyrrolidine-1-carbonyl]-N-phenylpiperidine-1-carboxamide 7-[3,5-dimethoxy-4-(4-phenylpiperazine-1-carbonyl)phenyl]-6-oxo-2-thia-5,7,11-triazatricyclo[6.3.1.04,12]dodeca-1(11),8(12),9-triene-3-carboxylic acid 7-ethoxy-N-methylquinoline-4-carboxamide 3-(2,5-dimethylthiophene-3-carbonyl)-10H-acridin-9-one N-[(E)-2-[3,5-dimethoxy-4-(trifluoromethyl)phenyl]prop-1-enyl]methanimine 1-methyl-4-[(2,3,5,6-tetrafluorophenoxy)methyl]pyridin-1-ium 3-[1-(4-tert-butylphenyl)ethenoxy]propanoic acid N-(4-ethylphenyl)-2,5-dimethoxy-3H-indole-1-carboxamide (7R)-7-amino-5,6,8-trideuterio-2-[3-hydroxy-4-(hydroxymethyl)anilino]-N-methyl-9-oxo-10H-acridine-4-carboxamide 4-[3-(2,6-difluorophenyl)-7,8-dihydro-1H-cyclopenta[g]quinoxalin-2-yl]morpholine 3-[[4-[(6-chloro-2,3-dihydro-1H-inden-5-yl)amino]pyrimidin-2-yl]methyl]pyridine-2-carboxylate 2-(N-(4-ethoxyphenyl)anilino)-2-methylpropanoic acid (2-ethylnaphthalen-1-yl)phosphonic acid 4-(3-methoxyphenyl)sulfonylpiperidine N-[2-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-5-thiophen-2-ylpyrazol-3-yl]-2,5-dihydroxybenzamide 4-[(1R,3S)-3-(5-oxo-2-sulfanylideneimidazolidin-1-yl)cyclohexyl]oxy-2-(trifluoromethyl)benzonitrile 4-(1,2-oxazol-3-yl)benzene-1,3-diol 1-(1,2,4-triazol-1-yl)naphthalene-2-carbonitrile 4-(2,3,3a,7a-tetrahydro-1H-inden-5-yl)-N-(4-chlorophenyl)-6-methoxy-5-propan-2-ylpyridine-3-carboxamide [2-(azidomethyl)cyclohexyl]oxymethylbenzene 1-[4-(3,5-dimethylphenyl)-2-methoxypyridin-3-yl]butan-1-ol 2,2,3-tributoxy-4-(cyclohexylmethoxy)oxane [3-(carboxymethoxy)phenyl]sulfamic acid N-[[2-(methoxymethyl)phenyl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide [3-(3,4-dichloroanilino)piperidin-1-yl]-[6-methyl-2-(triazol-2-yl)pyridin-3-yl]methanone 5-(2-aminopyrimidin-4-yl)oxy-3,3a,7a-tetrahydro-1H-indol-2-one [2-bromo-4,6-bis(methylamino)phenyl]methylideneazanium N-(2,6-dimethylphenyl)-1H-indole-3-carboxamide;ethane 1-(3,4-dihydro-2H-quinoline-1-carbonyl)-N'-hydroxy-5,6-dimethylindolizine-7-carboximidamide 4-[4,5,6-tribromo-1-(3-methoxyphenyl)sulfonylpyrrolo[2,3-b]pyridin-3-yl]benzamide N-[1-(2,6-dimethoxyethyl)pyrazol-4-yl]-5-nitropyrimidin-2-amine 2-[(1R)-1-azidoethyl]-5-chloro-3H-isoindol-1-one 3-[3,4-dihydroxy-5-(pyridin-2-ylmethylideneamino)phenyl]propanoic acid ethane;N-[2-[4-(1,3-thiazol-5-ylmethoxy)phenyl]propan-2-yl]formamide 1-[5-(4,6-diphenyl-1,3,5-triazin-2-yl)-1-[3-fluoro-4-(trideuteriomethoxy)benzoyl]piperidin-2-yl]ethanone 2-ethyl-1-[3-(trifluoromethoxy)phenyl]butan-1-one N-(2,5-dichlorophenyl)-4-[2-(3,5-dimethylbenzoyl)hydrazinyl]-3-nitrobenzenesulfonamide N-[5-[(Z)-1-aminoprop-1-enyl]pyridin-2-yl]-3-[4-(4-chlorophenyl)phenoxy]-2-hydroxypropanamide N-[2,5-diamino-4-(fluoromethyl)phenyl]sulfonyl-2,6-difluorobenzamide 2-[(4-azidophenyl)methyl]-3,5-dichlorothiophene N-[(6S)-2,4-dichloro-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]benzamide 4-[1,5,7-tris(ethenyl)-3,4-dihydroisoquinoline-2-carbonyl]benzonitrile 1-(5-tert-butylthiophen-2-yl)sulfinyl-3-[4-[7-[[2,6-dichloro-4-[(E)-hydroxyiminomethyl]phenyl]methoxy]-2-oxochromen-4-yl]phenyl]urea 3-[2-(4,5-dihydro-1H-imidazol-2-yl)ethynyl]-N-[2-[(2R)-1-hydroxypropan-2-yl]oxyphenyl]benzamide;dihydrochloride 2-[(5-bromopyridin-2-yl)-ethylamino]decanoic acid (3-fluorophenyl)methyl-(2-hydroxyethylimino)azanium 6-(4-ethylphenyl)sulfonyl-N-hydroxy-2,3-dihydrochromene-4-carboxamide N-(3,4-dimethylphenyl)-2-[[6-oxo-4-(propan-2-ylsulfanylmethyl)-1H-pyrimidin-2-yl]sulfanyl]acetamide [2-[(4-carboxynaphthalene-1-carbonyl)amino]phenyl]methyl-triethoxyphosphanium (2Z,5S)-2-[(Z)-1-(4-methoxyphenyl)ethylidenehydrazinylidene]-5-phenacyl-1,3-thiazolidin-4-one 3-[3,5-di(carbazol-9-yl)phenyl]pyridine-2-carbonitrile 5-(6,7-dihydroxyquinolin-4-yl)oxy-N-[2-oxo-3-phenyl-1-[4-(trifluoromethylsulfanyl)phenyl]butan-2-yl]pentanethioamide 6-azido-3-chloroanthracene-9,10-dione N-[(Z)-but-2-enyl]-N',5-dimethylpyridine-2-carboximidamide 4-(azidooxymethyl)-1,2-diethoxybenzene 3-azido-6,7-dimethylpyrazolo[1,5-a]pyridine (4R)-5-[3,5-bis(trifluoromethyl)phenyl]-4-[1-[2-(4-chlorophenyl)ethenoxycarbonylamino]hexan-2-yl]-4H-1,3-thiazole-2-carboxylic acid 2-(3,5-dimethylpyridin-4-yl)-N-[(5-hydroxy-1,3-dihydroisoindol-2-yl)sulfonyl]acetamide 1-(3,4-dichlorophenyl)-2-pyridin-2-ylethanone;ethane [4-(4-chlorobenzoyl)phenyl]-(4-methylcyclohexyl)carbamic acid N-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophene-2-carboxamide 1-cyclopentyl-3-[4-methoxy-5-(methylideneamino)pyridin-2-yl]urea 2-(2,4-dibromoanilino)-5-[(E)-2-thiophen-3-ylethenyl]phenol 5-(3-aminopropyl)thiophene-2,4-dicarboxylic acid 6-(2,4-dichlorobenzoyl)sulfanylhexanoic acid N-[5-[2-(1H-indol-3-yl)ethyl]-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-2-yl]-4-phenylbenzamide 6-bromo-5-nitropyrazolo[1,5-a]pyrimidine N-[4-chloro-3-(trifluoromethyl)phenyl]-2-(1H-indazole-6-carbonylamino)pyridine-4-carboxamide N-(4,4,4-trifluorobutan-2-yl)furan-3-carboxamide 4-(3-methoxypropoxy)-N,2-bis(sulfanyl)benzamide 3-(5-butoxy-2,4-dimethylanilino)sulfanylbenzoic acid 2-methyl-1'-[(5-phenylpyridin-3-yl)methyl]spiro[6,7-dihydropyrrolo[2,1-c][1,2,4]triazole-8,3'-pyrrolidine]-3,4-dione;2,2,2-trifluoroacetic acid 1-(4,4-dimethylpent-1-en-2-yl)-3-propylbenzene 6-(5-aminopyridin-3-yl)-N-[1,2,4]triazolo[4,3-a]pyridin-3-amine N-methoxy-2-[5-(2,4,6-trimethylphenyl)-1H-imidazol-3-ium-3-id-2-ylidene]-3H-furan-5-carboximidamide 1-amino-3,4-dichloro-6-phenylcyclohexa-2,4-dien-1-amine N-[2-(6,8-dimethylimidazo[1,2-a]pyrazin-3-yl)ethyl]-4-hydroxypyrrolidine-2-carboxamide (5R,7S)-3-bromo-5-[2-chloro-4-(trifluoromethyl)phenyl]-N-cyclopentyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide 2-[4,6-bis(3-methylphenyl)-1,3,5-triazin-2-yl]-4,6-ditert-butylphenol 2-chloro-7-ethyl-6-fluoroquinoline 2,4-dimethyl-N-(3-methylbut-2-enyl)benzamide 2-[(E)-2-[4-(3,5-dimethoxyphenyl)cyclohexyl]ethenyl]-6,7-bis(ethoxymethyl)quinoline 2-(3-fluorophenyl)-6,11b-dihydrobenzo[b]quinolizin-5-one 4-amino-N'-[3-(2,6-dimethoxyphenyl)-1-(7-fluoro-2-hydroxy-1H-indol-5-yl)prop-2-enylidene]benzenecarboximidamide 2,4-dimethyl-6-(3-propoxyphenyl)pyrimidine (2R,4S)-N-[(Z)-(4-hydroxyphenyl)methylideneamino]-5-oxopyrrolidine-2-carboxamide 2-[N-(3-methylbutyl)-4-phenoxyanilino]ethanol 2-[1-benzyl-4-(3-chloro-4-hydroxyphenyl)piperidin-4-yl]oxyethanimidamide;dihydrochloride (NZ)-4,4-dimethylpentanamide;2-[2,4-bis(trifluoromethyl)phenyl]-6,13-diazapentacyclo[12.7.0.03,12.04,9.017,22]henicosa-1(14),3(12),4(9),5,7,10,15,17(21),19-nonaene 1-(2,5-dimethoxyphenyl)sulfonylpiperazine 3-[4-(4-azidopiperidine-1-carbonyl)anilino]-5-methylcyclohexa-2,4-dien-1-one 2-(4-chlorophenyl)-1,3-dihydroindene-2-carboxylic acid N-[(3R,4S)-1-cyclohexyl-4-pyridin-2-ylpyrrolidin-3-yl]-3-methoxy-2-methylbenzamide;hydrochloride N-[(6,7-dimethoxy-4-oxochromen-3-yl)methyl]furan-2-carboxamide [(E)-3-(dimethylamino)-1-methoxyprop-2-enylidene]-[4-[3-[[6-oxo-5-(trifluoromethyl)pyridazin-1-yl]methyl]phenoxy]-7H-pyrrolo[2,3-d]pyrimidine-6-carbonyl]azanium 1-methyl-5-(3-phenylphenyl)pyrazolidine 3-[1-(2,4-dichlorophenyl)propan-2-yl]-N'-hydroxypyridine-2-carboximidamide 2-(3,5-dichlorophenyl)-N-[4-[methyl-[2-[(2S)-2-methylpyrrolidin-1-yl]ethyl]amino]cyclohexyl]acetamide N'-amino-2-[4-(8,9-dihydroxy-6-oxobenzo[c]chromen-3-yl)oxyphenyl]benzenecarboximidamide 1-[2-(2,6-dichlorophenyl)-5-fluoropyrimidin-4-yl]azetidine-3-carboxylic acid [3-[4-(2-pyridin-2-ylethynyl)phenyl]phenyl]boronic acid 2-(5-azidopyridin-3-yl)-4,6-dimethoxypyrimidine N-[(E)-[1-(3,4-dihydroxyphenyl)-2-nitroethylidene]amino]-4-methoxybenzamide 1-[3,5-bis(trifluoromethyl)phenyl]-2,3-dihydroxypropan-1-one 4-(2-oxo-1H-quinoline-3-carbonyl)-1,1-diphenyl-2,5-dihydropyrazole-3-carboxylic acid N-methyl-1-[3-(3-propan-2-yloxyphenoxy)pyrazin-2-yl]methanimine N-(2,3-dihydro-1H-inden-4-yl)-6,7,8-trifluoroquinoline-5-sulfonamide 3-(4,5-dihydrobenzo[g][2]benzazepin-1-yl)piperidine-2,6-dione 7-[(2R)-3-amino-2-hydroxypropoxy]-N-[1-[4-methanimidoyl-2-(oxetan-3-ylsulfamoyl)phenyl]ethyl]quinoxaline-5-carboxamide (3E)-4-amino-3-[(6-morpholin-4-ylpyridin-2-yl)methylidene]azete-2-thione 4-(4-phenylpiperazin-1-yl)quinazoline N-methyl-4-[2-(pyridin-3-ylamino)-5-[3-(pyrrolidin-1-ylmethyl)phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]benzamide 1-[4-(4-azido-6-methoxy-1,3,5-triazin-2-yl)-3-methylphenoxy]-3-morpholin-4-ylpropan-2-ol N-[3-[(4,6-dimethylpyrimidin-2-yl)sulfamoyl]phenyl]-N-ethylsulfonylbenzamide 3-cyclohepta-1,3,6-trien-1-yloxy-1H-1,2,4-triazole-5-carboxylic acid 2-(1H-indazole-3-carbonyl)-4,5-dimethylbenzonitrile N-[3-(4,6-difluoropyridin-2-yl)oxyphenyl]-6-methoxyspiro[1H-indole-3,1'-cyclopropane]-2-imine 4-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazine-3-carbonyl)-1-propan-2-yl-N-[3-(trifluoromethoxy)phenyl]piperazine-2-carboxamide 1-[4-(dimethylamino)phenyl]-3,4,9,11-tetrahydro-2H-benzo[h][1,6]naphthyridine-5,7-dione 2-(4-aminophenyl)sulfinylethyl-butoxyphosphinic acid 4-(azidomethyl)-3,5-dibromoaniline 1-[(E)-4,4,4-trifluoro-3-methoxybut-2-en-2-yl]naphthalene 1-[2-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-1-yl]ethanone 2-[1,6-dimethyl-5-(4-nitrophenyl)cyclohexa-2,4-dien-1-yl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane N-[4-amino-5-(1,2,3,6-tetrahydropyridin-4-yl)-[1]benzofuro[3,2-d]pyrimidin-7-yl]-2-piperidin-4-ylacetamide N-[4-(benzylamino)phenyl]sulfonyl-6-(cyclopentyloxyamino)-2-(2,3,5,6-tetrafluorophenoxy)pyridine-3-carboxamide 1-[(2E,4Z)-hexa-2,4-dien-3-yl]oxyhexan-1-ol;methanamine;2-methylidenebutane;1-methyl-4-[5-(4-phenylphenyl)pentyl]benzene 2-(4-azidophenyl)-1,3,5-trimethoxybenzene 7-(3,4-dimethylphenyl)-2-heptan-4-ylsulfanyl-[1,2,4]triazolo[1,5-a]pyridine 2-[5-[1-cyclohexyl-6-(cyclopropylmethoxy)pyrazolo[3,4-b]pyridin-4-yl]pyrimidin-2-yl]propan-2-ol 6-bromo-2,4-diphenyl-1H-benzimidazole 3-[4-(2,2-diphenylethyl)phenyl]pentanenitrile 1-[(4Z)-hexa-2,4-dienyl]-2-methyl-3-phenylbenzene (2S)-4-(4,5-dimethyl-1H-pyrazole-3-carbonyl)-N-[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]morpholine-2-carboxamide 2-azido-5-methoxy-N,3-dimethylbenzamide N-benzyl-2,6-difluoropyridine-4-carboxamide 1-N-[1-(4-methoxyphenyl)propan-2-yl]-5,6,7,8-tetrahydroimidazo[1,5-a]pyridine-1,6-dicarboxamide N-[2-(1H-indol-3-yl)ethyl]-2,4,6-trimethyl-N-propylaniline (3-methyl-1,1,2-triphenylbutoxy)benzene N-[(4R)-8-ethenyl-7,8-diazabicyclo[5.1.0]octan-4-yl]benzamide 2-amino-4-(5-cyclopentyloxy-3-methoxy-1,6-dimethylindol-2-yl)benzaldehyde 4-(2,3-difluoro-4-methoxyphenyl)-6-[(E)-pent-3-enyl]benzonitrile N-(2,6-difluorophenyl)-5-methyl-2H-1,3-thiazol-4-amine;ethane 7,8-dibromo-2,9-dimethylpurine 2-cyclohexyloxy-1-[5-(4-propan-2-yl-1,3-thiazol-2-yl)-2,3-dihydroindol-1-yl]ethanone 1-[3,5-dimethyl-4-[4-(2,4,5,13,15-pentazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),3,5,7,9,11,15,17-octaen-3-yl)phenyl]phenyl]-N,N-dimethylmethanamine (2E,3Z)-N-[4-chloro-6-(1H-imidazol-5-ylsulfonylamino)pyridin-2-yl]-3-ethylidenehepta-2,4,6-trienenitrilium 5-bromo-4-[(3,6-dichlorocyclohexa-1,5-dien-1-yl)methoxy]pyrimidine N-[2,4-dimethyl-5-(phenylcarbamothioylamino)hexan-3-yl]pyrimidine-4-carboxamide 2-N-[[4-(diethylamino)phenyl]methyl]-7-N,3-diethyl-5-N-(2-piperidin-1-ylethyl)pyrazolo[1,5-a]pyrimidine-2,7-diamine 2-amino-6-[3-(1,4-dihydroquinazolin-2-yl)phenyl]phenol 2-(cyclopentylsulfamoyl)-N,3-dimethoxy-N-[3-[4-(trifluoromethyl)phenyl]propyl]benzamide 6-[(3-ethylphenyl)methyl]-2-thiophen-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one N-(3-chlorophenyl)sulfonyl-4-(2,5-dimethoxyphenyl)piperazine-1-carboxamide 3-[4-(2,2-dimethylpropanoyloxy)phenyl]-4-oxopentanoic acid 3-(cyclohexylmethylsulfonyl)-1,2,4,5-tetrahydropyrrolo[2,3-d]pyridazine N-[5-(4-fluorophenyl)-6-(oxan-2-yloxymethyl)pyridin-3-yl]methanesulfonamide 1-(1,3-benzoxazol-2-yl)-N-cyclopentylpiperidine-4-carboxamide N-cycloheptyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 2,3-dichloro-N-[[3,5-difluoro-4-(methylamino)phenyl]carbamothioyl]benzamide (E)-5,6-diamino-3-methyl-1-(4-methylideneazepan-1-yl)hex-2-en-1-one;7H-purine 4-fluoro-1-[(1R,2R)-2-methoxycyclopropyl]indazole N-(1,5-dimethylpyrazol-4-yl)-2-[2-hydroxyethyl(propan-2-yl)amino]acetamide 6-bromo-2,3-dimethylpyrazolo[1,5-a]pyrimidine 3-[2,6-bis(ethenyl)phenyl]-N-[(Z)-2-(dimethylamino)but-1-enyl]-4-hydroxybenzenesulfonamide 4-(1H-indol-3-ylmethylideneamino)benzonitrile 4-[(6E)-6-ethylidene-5,8a-dimethyl-1H-phthalazin-2-yl]cyclohexan-1-ol N-[1-azido-3,5-bis(trifluoromethyl)pyrazol-4-yl]benzenesulfonamide 3-benzyl-8-(3-bromophenyl)purine 2-bromo-N-(3-nitrophenyl)-N-(1,3-thiazol-5-yl)benzamide 4-[2-methylsulfanyl-6-(trifluoromethoxy)quinazolin-4-yl]-3,5-dihydro-1H-pyrazole-2-carboximidamide (5Z)-2-imino-5-[(4-propanoyloxyphenyl)methylidene]-1,3-thiazolidine-4-carboxylic acid (2R,4R)-2-[3-amino-6-(4-methylphenyl)pyrazine-2-carbonyl]oxy-2-methyl-5-oxa-1-azabicyclo[2.2.0]hexane-4-carboxylic acid [(3S)-1-benzyl-2,5-dioxopyrrolidin-3-yl]carbamic acid N-(4-acetamidophenyl)-2,5-dimethylfuran-3-carboxamide 2-[(3R)-3-(tert-butylcarbamoylamino)-4,4-difluoropiperidin-1-yl]-N-methylbenzamide (6S,11bR)-11b-methylsulfanyl-6-propyl-3,5,6,7-tetrahydro-2H-[1,3]thiazolo[3,2-a]isoquinoline 2-[[2-(4-chlorophenyl)ethylamino]methyl]-3H-quinazolin-4-one N-methyl-2-[(1S)-2-phenylcyclopropanecarbonyl]-3,4-dihydro-1H-isoquinoline-5-carboxamide 1-[3-azido-2,4,6-trimethyl-5-(4-propanoylpiperazin-1-yl)phenyl]ethanone N-[(2R)-3,3-dimethylbutan-2-yl]-4,5-dihydrobenzo[g][1,3]benzoxazol-2-amine 4-[5-(azidomethyl)thiophen-2-yl]-N,N-dimethylaniline 3-[4-(2,6-dichlorophenyl)cyclohexyl]benzamide 6-[(6-cyano-7-fluoro-2,4-dioxoquinazolin-3-yl)methyl]piperidine-1-carboxylic acid N-[5-tert-butyl-2-[3-(1H-pyrrolo[2,3-b]pyridin-4-yl)-2H-pyrazolo[3,4-b]pyridin-6-yl]phenyl]-2-methoxyacetamide 5-chloro-3-[4,6-dimethyl-2-[(2S)-1-methylpyrrolidin-2-yl]pyrimidin-5-yl]sulfanylpyridin-2-amine [2-methyl-4-(3,4,5-trimethoxyphenyl)pyrazol-3-yl]carbamic acid 6-(diethoxyphosphorylmethylidene)cyclohexa-2,4-dien-1-one 2-[(3S)-1-[4-chloro-3-(trifluoromethyl)phenyl]-5-oxopyrrolidine-3-carbonyl]-N,3-dihydro-1H-isoindole-1-carboxamide N-[4,7-bis(ethenyl)imidazo[1,2-a]quinoxalin-3-yl]acetamide (Z)-3-amino-1-[2-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]pyridin-4-yl]but-2-en-1-one 2-azido-5,7-difluoroacridine 1-[4-(3,5-dimethyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]propan-1-one 1-[7-(methylamino)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-2-yl]azetidine-3-carbonitrile;dihydrochloride 6-[4-(2,5-dimethoxyphenyl)piperazine-1-carbonyl]-3H-thieno[3,2-d]pyrimidin-4-one (2E)-N-[4-amino-3,6-bis(4-fluorophenyl)thieno[2,3-b]pyridin-5-yl]-3-ethenoxy-2-methanimidoylpenta-2,4-dienamide N-[(2S)-2-[7-amino-3-(3,4-dimethoxyphenyl)indol-1-yl]pentanoyl]-2-propan-2-ylcyclohexane-1-carboxamide 1-(2,5-diphenylthiophen-3-yl)propan-1-one 2-[4-(1,4-dioxan-2-ylmethoxy)phenyl]-5-thiophen-2-ylthiophene N-(3-nitrophenyl)-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide;hydrochloride 2-[[4,5-bis(ethenyl)pyridin-3-yl]methoxy]-N-[3-fluoro-5-(1H-imidazol-5-yl)phenyl]acetamide 3-(2,4-dichloro-5-ethylsulfonylphenyl)-1-[6-methoxy-7-[1-[2-(trifluoromethyl)pyridin-3-yl]ethylideneamino]quinazolin-2-yl]butan-2-one 2-(4,6-diphenylpyrimidin-1-ium-2-yl)-N'-methanimidoylpyridine-4-carboximidamide 1-[(E)-2,3-dihydro-1H-1,5-naphthyridin-4-ylideneamino]-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepine-3-carboxamide N-[4-chloro-3-(5,6-dihydroquinolin-4-yl)phenyl]-2-methoxyethanimidate (5E)-2-(4,7-dichloro-2-methyl-1-benzofuran-3-yl)-4,4,8-trimethylnona-5,7-dienoic acid 3-bromo-6-[(4E,7Z)-9-chloronona-2,4,7-trien-3-yl]imidazo[1,2-a]pyridine 6-tert-butyl-2-oxo-1,3-dihydroindole-4-sulfonamide 1-[2,3-di(propan-2-yloxy)phenyl]ethanethiol 3-(5-chloropyridin-2-yl)-1-[2-[[1-(4-hydroxy-4-methylpiperidin-1-yl)-1-oxopropan-2-yl]amino]-2-oxoethyl]-N,N-bis(2-methoxyethyl)indazole-6-carboxamide;2-fluoro-N'-phenylacetohydrazide 5-[(2R,3S)-4-[(3,5-dichloropyridin-4-yl)amino]-3-hydroxybutan-2-yl]oxycarbonylfuran-3-carboxylic acid 2-chloro-6-(3,5-dimethylphenyl)-3-fluoroaniline;1-[2-(4-fluoronaphthalen-2-yl)ethynyl]-N,N-bis(2-methoxyethyl)cyclopropane-1-carboxamide 3-amino-4,6-bis(2-phenylpropanoyl)phthalic acid 1-azidosulfanyl-3,5-dimethoxybenzene N-[(2R,3S)-1,1-dioxothiolan-3-yl]-3-[[4-(methoxymethyl)triazol-1-yl]methyl]piperidine-1-carboxamide N-[3-(3,4-dihydroquinolin-8-yl)phenyl]sulfanylacetamide 5-tert-butyl-2,4-dimethylthieno[3,4-c]pyridine 3-(5-chloro-2-cyanophenyl)-1H-pyrrole-2-carboxylic acid 1-[3-fluoro-4-(2H-tetrazol-5-yl)phenyl]ethanesulfonate 1-[4-(8-cyanoquinolin-3-yl)phenyl]ethanolate 5-[4,6-bis(trichloromethyl)pyrimidin-2-yl]-N-tert-butyl-2-(methylideneamino)aniline 2-(6-bromospiro[1,3-dihydroisoquinoline-4,1'-cyclopropane]-2-yl)sulfanylacetic acid 1-chloro-3,3-dimethyl-2H-fluorene 2-methyl-6-nitro-4H-[1,3]thiazolo[5,4-d]pyrimidine 4-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carbonylamino)phenyl]butanoic acid 1-(3-bromophenyl)sulfonylbutane-2,4-diamine 4-[[1-(cyclopropanecarbonyl)azetidin-3-yl]methoxy]pyridine-2-carboxamide N-[3-(cyclopropylmethoxy)oxolan-3-yl]-5,6-difluoro-1H-indole-2-carboxamide (4S)-2-[(3,5-difluorophenoxy)methyl]-8-(2-fluorophenyl)sulfonyl-2,8-diazaspiro[4.5]decan-1-one N-azido-2-(3,5-dimethoxyphenyl)aniline (E)-N-[2-(4-chloroanilino)ethyl]-3,5-dihydroxyhept-6-enamide 2-[(2R,4S)-4-acetamido-1-benzylpiperidin-2-yl]-N-phenylquinoline-4-carboxamide 1-[(2-methylphenoxy)methyl]-3H-pyrazolo[3,4-b]pyridine [2-(4-aminophenoxy)-5-chlorophenyl]-oxidoazanium (3S)-N-ethyl-1-[2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyrrolidin-3-amine N-butyl-4,6-dimethoxy-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide (2R)-N'-[2,6-dimethyl-4-(1H-pyrazol-5-ylamino)phenyl]-N-ethanimidoyl-2-methylpiperazine-1-carboximidamide 3-[2,6-bis(3H-oxadiazol-5-yl)phenoxy]propanoic acid 3-[3-(4,4-dimethylcyclohexen-1-yl)cyclobutyl]-5-(trifluoromethoxy)benzenesulfonamide 5-(4,6-diamino-1H-triazin-2-yl)-8-methyl-7-nitronaphthalene-2-carboxylic acid 3-[(2-chloro-4-fluorophenyl)methylsulfanyl]-6,7,8,9,10,11-hexahydro-5H-cycloocta[b]pyran-2-one 3-[4-(2-methylpropoxy)phenyl]oxirane-2,2-dicarbonitrile N-[3-(2-morpholin-4-ylethoxy)phenyl]-5,6-dihydroquinolin-8-imine 2-tert-butyl-5-(3,5-dimethoxyphenyl)pyrazine 2-[4-(chloromethyl)phenyl]-N-(3,4-difluoro-5-propan-2-yloxyphenyl)imidazo[1,2-a]pyrimidin-7-amine 1-(3,5-dimethylphenyl)-N-[2-(3H-indol-3-yl)ethyl]ethanimine (2S)-1-[4-[8-chloro-6-[2-hydroxyethyl(methyl)amino]isoquinolin-3-yl]phenyl]-5-oxopyrrolidine-2-carboxamide [3-(2,4-difluoroanilino)sulfanylphenyl]-(3-ethoxyphenyl)methanone 2-[6,8-dichloro-3-(3-methylsulfonylpropoxy)quinoxalin-2-yl]-5-fluorophenol 4-(3,4-dimethylthiophen-2-yl)-7-methoxyquinazoline 1-(3,4-dimethoxyphenyl)-2-(8-oxaspiro[4.5]decan-4-ylsulfanyl)hydrazine 2,3-bis(ethenyl)quinoline [(Z)-4-(3-aminophenyl)-1,2-difluorobut-1-enyl]carbamic acid 2-(7-benzoyl-8,11-dihydropyrrolo[1,2-c][4,3]benzodiazepine-5-carbonyl)oxyethanesulfonic acid 2-[(6-nitropyridin-3-yl)oxymethylidene]propanedioic acid 2-[4-(1,3-benzoxazol-2-yl)phenyl]butanoate 3-[(E)-[[4-(diethylamino)phenyl]hydrazinylidene]methyl]-6-fluorochromen-2-one N-[4-chloro-6-(cyclopenten-1-yl)pyrimidin-5-yl]sulfanyl-2,6-difluoroaniline;2-(3,4-dimethoxyphenyl)acetaldehyde 3-fluoro-1-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonyl)piperidin-1-yl]-2H-pyridin-4-one;dihydrochloride 1-[3-[(3R,4S)-4-benzyl-1-pyridin-2-ylpyrrolidin-3-yl]oxypropylsulfanylmethyl]-5,6-dihydronaphthalene ethane;3-[2-(4-morpholin-4-ylphenyl)ethynyl]-1-benzothiophene-2-carboxamide 4-[2-(3,5-diaminophenyl)ethyl]benzenethiol N-[3-[2-(6,7-dimethoxyquinazolin-4-yl)oxyethynyl]phenyl]-2-[2-oxopropyl-[2-(propanoylamino)pyridin-3-yl]amino]acetamide 4-methyl-2,3-dihydrothiochromene;propane 3-[4-(trifluoromethyl)phenyl]benzene-1,2-diamine 3-[5-tert-butyl-3-(2,4-dioxopyrido[3,4-d]pyrimidin-1-yl)pyridin-2-yl]sulfanylpropanenitrile 7-amino-N-[(1S,3R)-3-methylcyclohexyl]quinoline-3-carboxamide;ethane 1-[4-chloro-3-(trifluoromethyl)phenyl]-4,5-bis(2-hydroxyethoxymethyl)pyridin-2-one 1-[2,3-bis(ethenyl)phenyl]-4-ethenylpiperazine (2E)-2-[amino-(4-methylphenyl)sulfanylmethylidene]-3,5-difluorocyclohexan-1-one 2-[N-(4-bromobutan-2-yl)-3-methylanilino]-1-phenylethanone 4-[3-(3,5-dimethylphenyl)phenyl]pyridine;ethane (3Z)-4-[1-benzofuran-2-ylmethyl(ethyl)amino]-4,5,5,6,7,8,9,10-octadeuterioundeca-3,8,10-trienal N-[1,6-di(propan-2-yl)cyclohexa-2,4-dien-1-yl]-2H-acenaphthylen-1-imine 1-[4-(2-ethylsulfanylphenyl)piperazin-1-yl]prop-2-en-1-one (2E,4Z)-3-bromo-1-[3-(2-methoxyethyl)-5-methylidenepyrrol-2-yl]hexa-2,4-dien-1-one 4-[(3S)-3-aminopyrrolidin-1-yl]-N'-isoquinolin-5-yl-2-oxobutanimidamide 2-[2-methyl-4-(trifluoromethyl)pyridin-3-yl]acetic acid 5-cyclopropyl-2-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine N-[(1R)-2-azido-1-phenylethyl]-4,5-dichloropyrimidin-2-amine 5-(3,4-difluorophenyl)sulfonyl-N-[2-hydroxyethyl-[1-(3-methoxypropyl)-6-oxopyridin-2-yl]amino]-N-methylfuro[3,2-b]pyridine-7-carboxamide 3-[5-(benzylamino)pentoxy]propane-1,2-diamine [2-[[(3R)-1-(4-aminocyclohexyl)piperidine-3-carbonyl]amino]-5,6-difluorobenzimidazol-1-yl]boronic acid 2-(4,5-dichlorothiophene-3-carbonyl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-5-carboxylic acid N-(3-hydroxypropyl)-2,4,6-trimethyl-N-phenacylbenzenesulfonamide 2-[(2E)-4,8-dimethylcyclooct-5-en-1-yl]oxy-N'-hydroxypyridine-4-carboximidamide (2R)-3-[4-[(E)-hept-5-enoxy]phenyl]-2-[(2S,3S)-3-hydroxy-4-oxobutan-2-yl]oxypropanoic acid N-[(4,4-dimethyloxolan-2-yl)methyl]-3-(3-phenyl-1H-pyrazol-5-yl)propanamide 2-(5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-ylamino)ethanol N-[3-amino-5-(2,4-difluorophenyl)sulfanylphenyl]acetamide 3-(4-fluorophenyl)sulfonylpropanenitrile 2-(benzimidazol-1-ylmethyl)-4-N,4-N-diethylbenzene-1,4-diamine 1-(2-azidoethyl)-3,5-bis[2-(4-fluorophenyl)ethenyl]benzene 3-[(4,5-dimethylpyridazin-3-yl)oxymethyl]-1-oxa-8-azaspiro[4.5]decane;2,2,2-trifluoroacetic acid 2-chloro-N-[4-(difluoromethoxy)-3-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-ylsulfonyl)phenyl]benzamide 3-(5-fluorothiophen-2-yl)-5-[2-[1-methyl-4-(trifluoromethyl)pyrazol-3-yl]pyridin-4-yl]-2H-1,3,4-oxadiazole N-(2,3-dimethylpentan-3-yl)pyrimidine-4-carboxamide 2-hydroxy-6-[(3R)-3-hydroxypyrrolidin-1-yl]imino-4-N,5-dimethoxy-4-N-phenylpyrimidine-4,7-dicarboxamide 1-[6-(4-chlorophenyl)-2-oxo-1H-pyrazine-3-carboximidoyl]pyrrolidin-3-ol 2-[(4R)-4,5-diphenyl-3-[(2S)-2-phenylpropyl]cyclohexa-1,5-dien-1-yl]-N-methylideneethanimidamide N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-methyl-5-[ethyl(oxan-4-yl)amino]benzamide;ethane N-[1-(1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carbonyl)cyclopropyl]benzamide N-[4-(3,5-dimethylphenoxy)phenyl]-6-methoxypyridine-2-carboxamide 3-(2,4-dichlorophenyl)-6-[4-(4-nitroanilino)piperidin-1-yl]quinazolin-4-one N-[3-(1,2-dihydropyrido[4,3-d]pyrimidine-7-carbonylamino)cyclobutyl]quinoxaline-5-carboxamide 2-[2-(2-methylpropoxy)-5-nitrophenyl]oxolane 1-azido-4-[4-(dimethylamino)phenyl]piperazine (2S)-2-[4-[5,6-bis(sulfanyl)pyrazine-2-carbonyl]piperazin-1-yl]-3-(1H-imidazol-5-ylmethylideneamino)propanoic acid 4-[2-(3,5-dimethylphenyl)acetyl]-N'-hydroxypiperidine-1-carboximidamide N-[3-chloro-4-(2,6-dimethylphenoxy)phenyl]butanamide 1-ethoxy-2,3,4-tris(fluoromethyl)benzene;N-(5-ethynylpyridin-2-yl)formamide 5-amino-2-[4-(methylamino)pentyl]benzonitrile 1-methylsulfonyl-N-[(3R)-piperidin-3-yl]-5,6,7,8-tetrahydroimidazo[4,5-c]azepine-4-carboxamide N-[5,6-bis(4-chlorophenyl)pyridin-2-yl]oxy-2-methylbutanamide 4-amino-2,5-dimethylbenzenesulfonate (6E,10Z)-11-[(3R)-3-benzylpiperazine-1-carbonyl]-16-hydroxyimino-3,5,8,14-tetrazabicyclo[15.4.0]henicosa-1(21),6,10,12,17,19-hexaene-2,16-dione 4-(5-methoxycarbonylpyridine-3-carbonyl)benzoic acid 5-(azidomethyl)-N,4-dimethyl-1H-indazole-3-carboxamide 2-[3-(cyclopropylamino)-1-(2,3,4,5,6-pentafluorophenyl)sulfonylpyrrolo[2,3-b]pyridin-2-yl]acetic acid;ethane 3-(2,4-dichlorophenyl)sulfonyl-1-methyl-5-piperidin-4-ylpyrazolo[4,3-b]pyridine 2-[5-(4-methylthiophen-3-yl)-1H-indazol-3-yl]-4-pyridin-3-yl-1H-pyrrolo[2,3-b]pyridine 1-benzylsulfonyl-4-[2-(3,3-dimethoxycyclobutyl)ethenyl]piperidine [(E)-3-hydroxybut-1-enyl]benzene;(Z)-4,4,4-trifluoro-N,2-dimethylidene-N'-phenylbut-1-ene-1,5-diamine N-(4-cyclopropyl-1,3-oxazol-2-yl)-2,4-dimethylpyrazole-3-carboxamide 2-[(4aS,8aS)-4a-(3,4-dimethoxyphenyl)-2-methylsulfonyl-4,5,6,7,8,8a-hexahydrobenzo[d][1,3]thiazin-9-yl]acetic acid N-[(2S)-3-(1H-indol-3-yl)propyl]-3-(4-methoxyphenyl)-5-oxo-7H-thieno[3,4-b]pyridine-6-carboxamide N-[4,4,4-trifluoro-1-(4-methylphenyl)but-3-en-2-ylidene]hydroxylamine 6-(5-methylfuran-2-yl)-4H-pyrazolo[1,5-a]pyrimidine N-[3-(4-methylphenyl)sulfonyl-2H-1,3-thiazol-5-yl]benzamide 3-[1-(2-bromoethyl)-4-(trifluoromethoxy)benzimidazol-6-yl]propanoic acid N-cyclohexyl-2-(diethylamino)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine-4-carboxamide 1-[1-(cyclohexylmethyl)piperidin-4-yl]triazole-4-carboxamide N-[2-(4-methylpiperazin-1-ium-1-ylidene)ethylidene]-6-phenylpyridine-3-carboxamide;tetrafluoroborate [3-(2,3-dihydroxypropyl)phenyl]phosphonic acid 3-[2,5-difluoro-4-[[[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]amino]methyl]phenoxy]phenol 3-[3,5-dichloro-N-(2,4-dihydroxybutyl)anilino]propane-1,2-diol [4-(2,5-dimethylpyridine-3-carbonyl)piperazin-1-yl]-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methanone N-[3-(2,6-difluorophenyl)oxetan-3-yl]carbamate [3-(2,5-dimethylphenyl)-4-sulfanylidenechromen-2-yl]methylurea 2-(1,3-benzodioxol-5-yl)-6-chlorochromene-4-thione 1-(4-azidophenyl)sulfonyl-5-bromoindole 3-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-5-oxo-4H-pyrazole-3-carbonyl]amino]propanoic acid 4-[(3R)-3-aminopyrrolidine-1-carbonyl]-6-cyclopropylpyridine-2-carboxamide N-[6-(2,3-dihydroindole-1-carbonyl)pyrimidin-4-yl]pyrrolidine-1-carboxamide 3-[(2E,4Z)-hexa-2,4-dien-3-yl]-2,6-bis(trifluoromethyl)quinoline 4-[5-[3-(dimethylamino)propoxy]-1,3-benzoxazol-2-yl]aniline 4-[[3-(cyclohexylmethoxy)phenyl]methyl]-N-hydroxybenzamide;uranium(2+) 3-[4-(2,6-dimethylphenyl)pyridin-2-yl]oxy-5-(5-methylsulfonylpyridin-2-yl)benzonitrile;ethane 2-[1,3-dichloro-6-(4-hydroxy-2,5-dimethoxyphenyl)pyren-2-yl]oxy-N-[2-(3,4-dimethoxyphenyl)ethyl]acetamide 6-[(4E)-2,4-dimethylhepta-2,4,6-trien-3-yl]-2-[5-(pyrrolidin-1-ylmethyl)pyridin-3-yl]-7H-pyrrolo[3,4-b]pyridin-5-one 4-tert-butylbenzenesulfonate;6,7,8,9-tetrahydro-5H-carbazol-2-ylmethanol (2R,3S)-1-(4-ethyl-6-oxo-1H-pyrimidin-2-yl)-N-[(5-methoxypyridin-2-yl)methyl]-2-phenylpiperidine-3-carboxamide 2-[5-carbamoyl-9-[(4-methylphenyl)methyl]-2-propan-2-ylcarbazol-4-yl]oxyacetic acid 7-amino-5,11-dihydrobenzo[d][1]benzazepine-9-carboxamide 7-fluoro-2,3,8,9-tetrahydrobenzo[f]chromene-1,6-dione 4-[5-(aminomethyl)thiophen-2-yl]sulfonyl-N'-hydroxybenzohydrazide 3,5-dibromo-4-[2-(3,7-dimethyloctyl)phenoxy]aniline 4-(3,5-dinitrophenoxy)-2H-triazole [(Z)-1,2-dibromoethylideneamino]benzene N-[6-(hydroxymethyl)quinolin-4-yl]-2-[3-[(4-nitrophenyl)sulfanylamino]propoxy]acetamide N-[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-4-yl]propane-1-sulfonamide 2-[N'-(2,4-dichlorophenyl)carbamimidoyl]pyrrolidine-1-carboxamide 6-(4,4-difluorocyclohexyl)-3H-1,3,5-triazine-2,4-dione N-[4-(difluoromethoxy)phenyl]-2,5-dioxopyrrolidine-1-carboxamide (2R)-3-[2,6-dimethyl-4-(1H-pyrazole-5-carbonylamino)phenoxy]-2-methoxypropanoic acid 4-[3-(2-chlorophenyl)propanoyl]-2,6-dimethylpiperazine-1-carboxylic acid N-[2,3-bis(4-methylphenyl)cyclopropyl]-N'-[2-oxoethyl(pyrimidin-5-ylsulfonyl)amino]ethanimidamide 1-[5-(cyclopropylmethoxy)-2,3-dihydro-1H-inden-4-yl]ethanone;ethane N-[3-[2-(methoxyiminomethyl)-5-phenylphenyl]prop-1-en-2-yl]thiohydroxylamine 1-(4-bromophenyl)-2-hydroxy-4-propan-2-yloxypyridine-3,5-dicarboxylic acid 2,6-bis(trifluoromethyl)-5H-benzo[d][1]benzazepine N-[4-(4-azidobutyl)phenyl]-3,5-dimethoxyaniline 2-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine 1-azidooxyanthracene (3S)-7-(cyclopropylmethoxyimino)-4,6-difluoro-2-methyl-5-oxo-1,2,3,4-tetrahydroquinoline-3-carboxylic acid 3-[2,4-dihydroxy-6-(N-phenylanilino)phenyl]propanoic acid N-[3-(1,3,4,6,7,8,9,10,11-octahydrocyclonona[c]furan-1-yloxy)phenyl]-2-(trifluoromethyl)benzamide 3-amino-4-methyl-6-(2-phenylmethoxyethyl)pyran-2-one 2-(2,6-dimethoxyphenyl)-N-[[(1S,3R,4R)-3-hydroxy-4-(4-pyridin-2-ylpiperazine-1-carbonyl)cyclohexyl]methyl]acetamide 3-[(2-methylpropanoylamino)methylidene]-N-[1,1,1-trifluoro-4-(3-methoxyphenyl)butan-2-yl]piperidine-1-carboxamide 5-ethyl-1-methylsulfonyl-6H-pyrazolo[4,3-d]pyrimidin-7-one 2-[5-methyl-3,4-bis(phenylmethoxy)oxolan-2-yl]acetic acid N-(4-chlorophenyl)sulfonylbut-2-ynamide [3-(3-azidopyrazol-1-yl)piperidin-1-yl]-pyridin-2-ylmethanone 3-(cyclopropylmethoxy)-4-fluoro-N-[5-(6-piperidin-1-ylpyridin-2-yl)-1H-pyrazol-4-yl]benzamide 4-amino-3,6-ditert-butylbenzene-1,2-dicarboxylic acid 1-N,4-N-bis(4-methylphenyl)benzene-1,4-dicarboxamide 4-[6-amino-5-(trifluoromethyl)pyrimidin-4-yl]phenol;ethane N-[1-(2,4-dioxo-1H-pyrimidin-6-yl)piperidin-3-yl]pyrimidine-5-carboxamide N-[5-bromo-2-(3,5-dimethylpiperidin-1-yl)phenyl]pyrimidine-4-carboxamide 4-(4-methoxycyclohepta-1,3,6-trien-1-yl)-3-[3-methanimidoyl-5-(3-pyrrolidin-1-ylpropoxy)phenyl]pyrazin-2-amine 4-tert-butyl-2-phenylmethoxyphenol 3-benzyl-4H-[1,2]oxazolo[5,4-d]pyrimidine;(E)-N-cyclopropyl-N'-ethoxy-N-methyl-4-phenylbut-3-enimidamide (2R)-1,1,1-trifluoro-3-[4-[6-(methylaminomethyl)pyridin-2-yl]oxyphenyl]propan-2-ol 2-chloro-3,5,7,8-tetrahydropyrimido[4,5-d]pyrimidine-6-thione 3-[(4-hydroxypiperidine-1-carbonyl)amino]-2,5,6-trimethylbenzenesulfonic acid ethane;1-[4-(8H-pyrrolo[2,3-f]quinolin-9-yl)phenyl]ethanamine 4-[6-methoxycarbonyl-7-methyl-2-(4-nitroanilino)-1H-benzimidazole-5-carbonyl]benzoic acid 3-[2,4,6-trichloro-N-(1-methoxy-1-oxopropan-2-yl)anilino]butanoic acid (4S)-3,6'-bis(dimethylamino)-2-[2-(4-phenylmethoxyphenyl)ethyl]-1'-propanoylspiro[isoindole-3,5'-azetidine]-1-one (4-tert-butylphenyl)-[4-[5-[5-(1,3-thiazol-2-ylamino)pyridin-2-yl]pyrimidin-2-yl]oxypiperidin-1-yl]methanone 3-(6,7-dimethoxyquinazolin-4-yl)sulfanylpyridine-2-carbonitrile N-(2,3-dihydro-1H-indol-6-yl)-5-fluoro-1,4,5,8-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide 1-(4,5,6,7-tetrahydrothieno[2,3-b]pyridine-2-carbonyl)piperidine-4-carboxylic acid 6-[(E)-1,2-bis(2-hydroxyphenyl)ethenyl]benzene-1,3-diol [3-(1,3-benzothiazol-2-yl)-2-methoxyphenyl]-[3-(cyclopropylamino)azetidin-1-yl]methanone;ethane 2-chloro-4,5-difluoroacridine (NZ)-N-[6-[3-chloro-4-fluoro-5-(trifluoromethoxy)phenyl]-3-cyclopropylpyrimidin-2-ylidene]nitramide 4-methoxy-N-[2-(1-methylpyrazol-4-yl)phenyl]cyclohexane-1-carboxamide 1-(azidooxymethyl)-2,4-diphenylbenzene 5-chloro-N,2-dimethylquinoline-8-carboxamide 4-[(3R)-3-methylpiperazine-1-carbonyl]benzonitrile N-(2,3-dihydro-1H-inden-5-yl)-1-[7-[(E)-1,2-difluoropent-2-enoxy]imidazo[1,2-a]pyridin-2-yl]methanimine N-[2-[(4-methoxyphenyl)carbamoylamino]ethyl]-1,3,5-triazinane-2-carboxamide 2-[4-(2-ethylphenyl)piperazin-1-yl]-N'-hydroxypyrimidine-4-carboximidamide (5R)-3,7,10-trihydroxy-2-oxabicyclo[9.4.0]pentadeca-1(15),11,13-triene-4-thione (3R)-N'-[(Z)-1-[4-(trifluoromethoxy)phenyl]propylideneamino]pyrrolidine-3-carboximidamide N-(6,8-dichlorospiro[4H-quinoxaline-3,4'-oxane]-2-yl)benzamide 2-cyclopentyl-N,N-diethyl-4-phenylpyrazole-3-sulfonamide 4-(2,5-diaminophenyl)benzene-1,3-diamine N-[(6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl)methyl]-N-ethyl-2-[(4-fluorophenyl)sulfonylamino]acetamide (3aR,6aS)-2-methylsulfonyl-5-[2-oxo-2-(4-pyrimidin-5-ylphenyl)ethyl]-1,3,3a,4,6,6a-hexahydrocyclopenta[c]pyrrole-5-carboxylic acid N-[4,5-dichloro-2-(hydroxymethyl)phenyl]cyclopropanecarboxamide N-[(1R)-1-phenylethyl]-2-propan-2-ylidenehexanediamide 1-(2,5-dimethylpyrazol-3-yl)-4-(dimethylsulfamoylamino)benzene 3-amino-2,6-dichloro-N-[(Z)-[4-(diethylsulfamoyl)phenyl]methylideneamino]benzamide N-(4,4-dimethylpent-1-en-2-yl)-5-[3-[4-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-1H-pyrazolo[4,3-b]pyridin-5-yl]pyridin-3-amine N-(4-methylpyridin-3-yl)pyrrolidine-1-carboxamide 4-[(3E,5Z)-hepta-1,3,5-trien-3-yl]oxybenzaldehyde 2-[4-(5,8,10-triazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,11-pentaen-12-yl)cyclohexyl]propan-2-ol 2-(5-fluoropyridin-3-yl)sulfanylacetaldehyde;5-methoxypyrazine-2-carboxamide 1,3-dimethyl-2-[(E)-2-(4-methylphenyl)ethenyl]-5-propanoylbenzimidazol-1-ium N-[6-[2-fluoro-4-(4-fluorophenoxy)phenyl]pyrazin-2-yl]-2,3,7,11-tetramethyldodecanamide 2-[(1E,3Z)-5-azidohexa-1,3,5-trienyl]-4-(2-chlorophenyl)-6-nitrophenol 1-[[2,5-difluoro-4-(4-hydroxybutoxy)phenyl]methyl]-3,4-diethylpyrrole-2,5-dione 3-[2,2-dimethoxyethyl(hexanoyl)amino]benzenesulfonic acid 4-(3,5-difluorophenyl)sulfanyl-7-methoxy-2H-isoquinolin-1-one 2-(dimethylamino)-4-(trifluoromethoxy)benzamide 1-[[2-bromo-4-(trifluoromethyl)phenyl]methyl]imidazole 1-bromo-2,4-dichloronaphthalene N-[(2S)-4,5-dihydroxypentan-2-yl]-2-ethoxy-6-[(Z)-hydrazinylidenemethyl]benzamide 4-[(2R)-5-cyclopropylpentan-2-yl]oxy-2,6-difluorobenzonitrile 3,6-dibromo-7H-purine 1-azido-2,4,6-trifluoro-3-nitrobenzene 1-[[7-(cyclopropylmethoxy)-2,3-dihydro-1H-indene-5-carbonyl]amino]cyclopentane-1-carboxylic acid 6,7-bis[(E)-3-methylbut-1-enyl]-2-propan-2-ylidene-1H-1,4-diazepine 3-[2-(3,4-difluorophenyl)ethyl]-6-(4-propoxycyclohexa-1,5-dien-1-yl)pyridazine 4-[[2,6-dibromo-4-(oxan-2-yloxy)phenyl]methylideneamino]benzenesulfonamide 2-methyl-5-[(4-methylcyclohexyl)carbamoyl]benzoic acid 2-[(4-aminophenyl)methylsulfanyl]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione 5-amino-6-[2-aminoethyl(methyl)amino]pyridine-3-carbonitrile;3-(6,7-dihydrofuro[3,4-b]pyrazin-5-yl)-5-methoxybenzaldehyde 4-[2-(3,5-dimethoxyphenyl)ethynyl]benzoic acid N-[[6-amino-1-[(2-amino-5,6,7,8-tetrahydroquinolin-4-yl)methoxy]naphthalene-2-carbonyl]amino]pyridine-3-carboxamide;methanol 1-(4-hydroxy-3,5-diiodophenyl)-N'-propan-2-ylsulfanylethane-1,2-diol 2-[4-(3,5-dimethoxyphenyl)piperidin-1-yl]-N'-(4-oxo-1H-pyrazolo[3,4-d]pyrimidin-6-yl)ethanimidamide N-[3,5-bis(trifluoromethyl)phenyl]-1-[6-[(E)-3-hydroxyprop-1-enoxy]cyclohexa-2,4-diene-1-carbonyl]piperidine-3-carboxamide 2-(4-methoxyphenyl)iminopropanoate 1-cyclobutyl-3-methoxy-5,6-dihydroindole 3-[4-(2,3,5,6-tetrafluoro-4-methoxyphenyl)pyridin-2-yl]propanoic acid 4-(4-hexoxyanilino)-N'-hydroxypyridine-2-carboximidamide 4-[2-(4-butylphenyl)ethynyl]phenol 2-[3-(difluoromethyl)-4-fluorophenyl]-6-oxo-1H-pyrimidine-5-carboxylic acid 2-[2-(4-ethylpiperazin-1-yl)pyrimidin-5-yl]guanidine 3-[2-(oxolan-2-ylmethylamino)pyrimidin-4-yl]-1H-indole-6-carboxylate 6-amino-2-(3,4-dichloroanilino)-3H-quinazolin-4-one 6-[(E)-2,3,5-trimethylhept-2-enoxy]pyridin-2-amine 2-amino-4,5-dimethylbenzenesulfonate;tetraphenylazanium 5-(3,4-dimethylphenyl)cyclohexa-1,3-dien-1-ol 6-bromo-N-[(3E)-4,5-dimethylhexa-1,3,5-trien-2-yl]pyridine-3-carboxamide 1-chloro-4-[(E)-1,2,3-trimethylundec-1-enyl]benzene 4-[[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl]amino]-6-chloro-8-(2H-tetrazol-5-yl)quinoline-3-carbonitrile 2-(3,4-dimethoxyphenyl)-N-[2-(4-fluorophenyl)-5H-[1]benzoxepino[5,4-b]pyridin-9-yl]acetamide 1-[2,6-di(propan-2-yl)phenyl]-N-methoxymethanamine 4-fluoro-N-[(3S)-2-oxopyrrolidin-3-yl]benzenesulfonamide 5-[(1S)-1-hydroxyethyl]-2,6-dimethoxy-3H-inden-1-ol (E)-3-[4-(diethylamino)phenyl]-1-(5,6-dimethylindolizin-2-yl)prop-2-en-1-one 4-(2,3-dihydro-1H-inden-5-yl)piperidine N-(3,5-difluorophenyl)sulfonyl-6-(2-methoxyphenyl)pyridine-3-carboxamide 6-chloro-N-[2-(diethylamino)ethyl]-3H-indene-1-carboxamide;hydrochloride N-(3,5-difluorophenyl)sulfanyloxy-4-methylaniline 6-[(4,5-dimethyl-2-phenyldiazenyl-1H-pyrrol-3-yl)methylideneamino]oxypyridine-3-carboxylic acid 5-(difluoromethyl)-4-iodopyridine-2,3-diamine 1-(2-azidooxyethyl)-4,5-dibromo-2-methoxybenzene N-(3,4-dimethylphenyl)-2-ethylimino-1,3-dihydrobenzimidazole-5-carboxamide 4-[2-(1H-indol-3-yl)ethenyl]-N-[2-[[(Z)-1-naphthalen-1-ylbut-1-enyl]amino]phenyl]benzamide N-[2-(4-methylphenyl)sulfonylethenyl]-3,5-bis(trifluoromethyl)aniline 2-[4-ethyl-3,5-bis(methoxycarbonyl)piperazin-1-yl]pyridine-4-carboxylic acid N-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-3-ylmethyl)-2,1,3-benzothiadiazol-4-amine 2-(4-tert-butylphenoxy)pyridine 4-N-(1,3-dioxolan-2-ylmethyl)pyrimidine-2,4-diamine;uranium(2+) 4-(4-aminophenyl)-N-[2-(1H-indol-3-yl)ethyl]butanamide (4R)-3,4-bis[2-(2-methoxyethylamino)-1,3-benzoxazol-6-yl]cyclopentane-1,2-dione N-cyclopropyl-1,5,7,10,11-pentazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaene-12-carboxamide 6-(furan-2-ylmethylidene)-3-sulfanylpiperidin-2-one 2-[3-chloro-5-(trifluoromethyl)pyridin-4-yl]-1-(oxolan-3-ylmethoxy)benzimidazole 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-ethyl-N-(5-methylpyridin-3-yl)-1H-pyrazole-5-carboxamide 3-(aminomethyl)-5,7-dihydroxychromene-2,4-dione 2-[6-methyl-8-(1,3-thiazol-4-yl)-9H-fluoren-1-yl]benzenethiol N-[(3S)-2,6-dimethylpiperidin-3-yl]-4-pyridin-2-ylaniline (2S)-4-cyclohexyl-1-[2-[(4,4-difluorocycloheptanecarbonyl)amino]acetyl]-N-(6-methoxypyridin-3-yl)pyrrolidine-2-carboxamide 2-[[5,7-difluoro-6-(3,3,3-trifluoroprop-1-ynyl)naphthalen-2-yl]methylsulfonylamino]butanedioic acid N-[(3,4-dichlorophenyl)methyl]-2-methoxy-6-methyl-8-(thiolan-3-ylamino)pyrido[3,4-d]pyrimidine-7-carboxamide 1-(3,4-dimethoxyphenyl)hept-2-yn-1-one 4-(4,6-dimethoxypyrimidin-2-yl)-2,5-difluorophenol 1-[[5-methylsulfonyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]methyl]imidazole 4-hydroxy-6,11-diazatricyclo[5.3.0.02,4]deca-1(10),2,4,6,8-pentaene-14,18-dione 2-[[1-(methoxyamino)cyclopentyl]methoxy]-5-propan-2-ylbenzoic acid N-[4-[1-[4-(dimethylamino)phenyl]-3,5-dioxo-6H-2,1,3-benzothiadiazol-4-yl]-2-fluorophenyl]acetamide;ethane 3-(2,5-difluorophenyl)-2H-quinolizine N-(6-chloro-3,4-dihydro-2H-chromen-8-yl)-2-methoxyacetamide 6-methylsulfonyl-3-propan-2-yl-1H-imidazo[4,5-c]pyridine 4-N,4-N-bis[(E)-2-chlorobut-1-enyl]benzene-1,4-diamine 1-[4-(2,3-dihydro-1H-indol-6-ylamino)piperidin-1-yl]-2-[4-(trifluoromethyl)phenoxy]ethanone 5-[1-azido-2-(3,4-difluorophenyl)ethyl]-2H-tetrazole 2-[5-fluoro-6-(4-methylpiperazin-1-yl)pyridin-3-yl]propan-2-ol 2-(4-aminophenyl)-6-[(3,5-dibromo-2-hydroxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-chloro-1,3-dimethyl-2-[(2E)-3,7,11-trimethoxydodeca-2,6,10-trienyl]imidazol-1-ium;chloride 2-[6-[(2-phenylethylamino)methyl]-1,4-dihydroquinoxalin-7-yl]acetic acid 2-[4,6-bis(3-pyridin-2-ylphenyl)-1,3,5-triazin-2-yl]-8-methylidene-6H-benzo[c][1,7]naphthyridine 4-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)morpholine [2-(cyclobutylmethoxy)phenyl]-phenyl-pyridin-3-ylmethanol (1S)-2-azido-1-[5-chloro-6-fluoro-3-[(4-methylpyridin-2-yl)amino]pyridin-2-yl]ethanol 3-(2,6-dichlorophenyl)-4-methylsulfonylbenzonitrile 2-(4-fluorophenyl)-6,7-dimethoxy-3H-quinazolin-4-one 1-azido-2-(6-bromohexyl)-4,5-dichlorobenzene N'-[(4-chlorophenyl)methyl]-N-[[4-[4-chloro-3-(trifluoromethyl)phenoxy]phenyl]methyl]oxamide (E)-3-[6-[2,5-dihydroxy-4-methoxy-6-(4-propanoylpiperazine-1-carbonyl)phenyl]pyridin-3-yl]prop-2-enoic acid 2-[(3R,4S)-3-fluoropiperidin-4-yl]oxybenzamide;hydrochloride 1-(4,6-diamino-1H-benzimidazole-2-carboximidoyl)naphthalen-2-ol N-[5-aminosulfanyl-2,4-dihydroxy-3-(oxolan-3-yl)phenyl]benzamide 4-[1-(5-fluoro-2-nitrophenyl)ethyl]morpholine 4-(diethylamino)benzenecarboximidamide 4-[7-(cyclopropylmethylamino)imidazo[1,2-a]pyrimidin-3-yl]phenol N-(2-bromoethyl)-4,6-dimethoxypyrimidine-5-carboxamide 5-(aminomethyl)-6-[5-[2,4-bis(trifluoromethyl)phenyl]furan-3-yl]-3H-quinazolin-4-one 6-methoxy-7-[[4-(1,3-thiazol-5-yl)phenyl]methoxy]quinazoline 1,3-dimethyl-5-[6-(4-pyridin-2-yl-1H-pyrrol-2-yl)naphthalen-2-yl]pyrazole 5-[2-(4-ethylpiperazin-1-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]azepan-2-one 2-[4-azidooxy-3,5-di(propan-2-yl)phenyl]pyridine (Z)-N'-hydroxy-3-[4-[[(1,5-naphthyridin-2-ylamino)methyl-propan-2-ylamino]methyl]phenyl]prop-2-enimidamide N-[3-(4,6-dimethylpyrimidin-2-yl)phenyl]sulfanyl-2-fluoro-5-nitroaniline (4-azidopiperazin-1-yl)-[5-methyl-2-(trifluoromethoxy)phenyl]methanone 4-[3-methylbut-2-enyl(prop-2-enyl)amino]-N-pyrimidin-2-ylbenzenesulfonamide 4-[2,3-dimethyl-5-(trifluoromethyl)indol-1-yl]benzonitrile 5-cyclohexyloxy-1-[(2R)-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]pyrimidine-2,4-dione 1-azido-4-[3-(dimethylamino)phenyl]butan-2-one 4-cyclopentyloxybenzaldehyde N-[4-methoxy-2-nitro-5-(trifluoromethyl)phenyl]-N'-[1-oxo-3-[4-(trifluoromethyl)anilino]-2H-isoquinolin-6-yl]oxamide (2R)-1-[[4-(2,3-dichloroanilino)quinoline-7-carbonyl]amino]propane-1-sulfonic acid 3-[2-(3-fluorophenoxy)pyrimidin-5-yl]oxan-4-ol (1R,2S)-2-[(4-methylphenyl)carbamoylamino]cyclopentane-1-carboxylic acid 2-[5-[[4-(5,5-dimethylcycloocten-1-yl)-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]indol-1-yl]acetic acid 2-hydroxy-4-(1H-pyrrolo[2,3-b]pyridine-5-carbonylamino)butanoic acid 3,5-diamino-4-chloro-1H-pyrrole-2-carboxamide (2R)-2-amino-1-[4-(3,5-dimethyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-3-phenylpropan-1-one 4-(3-aminophenyl)-5,6-dihydronaphthalen-1-amine 4-methoxy-N,2-dimethyl-3-(3-methyl-5-oxopiperazine-1-carbonyl)benzenesulfonamide 2-tert-butyl-5-[1-(3-tert-butyl-5-iodo-4-methoxyphenyl)ethyl]-1,3-dimethoxybenzene 2-(4-bromo-3-fluorophenyl)-6-(4,5-dihydro-1H-imidazol-2-ylmethylamino)quinoline-4-carbonitrile N-[4-[(3Z)-2,7-dimethylcycloocta-1,3,5,7-tetraen-1-yl]phenyl]-4-methoxybenzenesulfonamide 1-(2,5-dimethylpyrrol-1-yl)-3-[5-ethoxycarbonyl-4-methyl-6-oxo-1H-pyrimidin-2-yl]urea (3E)-N'-(5,6-dihydroindolo[1,2-a]quinoxaline-4-carbonyl)-3-hydroxy-3-(3-methylfuran-2-yl)iminopropanimidamide 2-fluoro-N,4-dimethylbenzenesulfonamide 3-ethyl-5,6-dimethoxy-2-phenyl-1H-indene 2-(4-chlorophenyl)-6,7-dimethoxyisoquinolin-1-one 2-[3-azido-1-(3,4-difluorophenyl)propyl]tetrazole N-(4,6-dimethylpyrimidin-2-yl)oxy-2-phenylacetamide 3-[(4Z)-7-fluoroocta-2,4-dienyl]naphthalene-1,8-dione ethane;3-[(4Z,6E)-7-hydroxy-5-methyl-2-oxohepta-4,6-dienoxy]-5-[(3S)-1-methylpiperidine-3-carbonyl]benzonitrile N-(3-azidopropyl)-5-methoxy-4,6-dimethylpyrimidin-2-amine N-(4-chlorobutyl)-N-cyclohexylnaphthalen-2-amine 6-methoxy-7-(2-phenoxyethyl)-1,3,4,5-tetrahydro-1-benzazepin-2-one 5-[(Z)-1-methylsulfanylprop-1-en-2-yl]-4-prop-1-ynylpyrimidin-2-amine 3-(4,5-dimethylthiophene-2-carbonyl)-1-(7H-purin-6-yl)-1,8-diazaspiro[4.5]decan-2-one 4-[1-(2,6-dimethylcyclohexa-1,5-dien-1-yl)sulfonylindole-3-carbonyl]oxybenzenesulfonic acid 4-[1-[(2R,6R)-2-methyl-6-propan-2-ylmorpholine-4-carbonyl]cyclobutyl]oxypyridine-3-carboxamide 3-(4-chlorophenyl)sulfonyl-2-[4-(1H-indol-5-yloxy)piperidin-1-yl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine (2R,3S)-1-[1-[4-[(4-chlorophenoxy)methyl]cyclohexanecarbonyl]piperidin-4-yl]-N,N-dimethyl-5-oxo-2-phenylpyrrolidine-3-carboxamide N-(3,4-dimethylphenyl)-6,7-difluoro-2-hydroxynaphthalene-1-carboxamide N-benzyl-N',2-diethoxypentanimidamide N-(3,5-dichloropyridin-4-yl)-2,3,7,9,14-pentazatricyclo[8.4.0.03,8]tetradeca-1(10),4,6,8,11,13-hexaen-16-imine 4-chloro-2-[4,7-bis(ethenyl)-3-thia-5,7,10,11-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-10-yl]benzonitrile 4-[(3S)-3,5-dihydroxypentyl]benzene-1,2-diol (2S)-1-[2-(4-acetylpiperazine-1-carbonyl)-3-(4-hydroxyphenyl)benzimidazol-5-yl]oxypyrrolidine-2-carboxamide 3-(2-methylprop-1-enoxy)-6,7-dihydroquinoline 4-[[2-(ethylaminomethyl)pyrrolidine-1-carbonyl]amino]pyridine-3-carboxylic acid;hydrochloride 2-[3,5-dichloro-N-(cyanomethyl)anilino]ethanol (2S)-1-[4-hydroxy-3-[1-[3-(hydroxymethyl)phenyl]sulfonylindol-5-yl]phenyl]pyrrolidine-2-carboxylic acid 2-[7-(difluoromethyl)-6-[4-(hydroxymethyl)piperidin-1-yl]-3,4-dihydro-2H-quinoline-1-carboximidoyl]benzamide 2-(5-ethyl-4,6-dihydroxy-1H-indole-3-carbonyl)-3-phenylprop-2-enoic acid 4-(3,5-diamino-2,6-dimethylphenyl)-2,2,5,5-tetramethylheptanoate 1-[[5-(5-bromo-2,4-dihydroxyphenyl)-3-hydroxypyridin-2-yl]methylideneamino]propan-2-one 2-[(4S)-5,7-dimethyl-3,4-dihydro-1H-isochromen-4-yl]ethanol;propane 1-azido-4,5-dimethyl-3-phenylpyrazole 1-(2,3-dichlorophenyl)-4,5-bis[2-[di(propan-2-yl)amino]ethoxy]penta-1,4-dien-3-one 7-[3-[(5-fluoro-2,4-dimethylphenyl)sulfonylamino]azetidine-1-carbonyl]-N-methylpyrazolo[1,5-a]pyridine-3-carboxamide 5-[4-(hydroxymethyl)-6,6-dimethoxycyclohexa-1,3-dien-1-yl]pyrimidine-2,4-diamine 2-[4-(methylamino)-3-[(Z)-pent-1-enyl]pyridin-2-yl]cyclobutane-1,3-dione 1-[5-(3,4-difluorophenoxy)pyrimidin-2-yl]-4-ethylazepane 5-(2,5-dimethoxyphenyl)-3-ethylimidazole-4-carboxylic acid 4-[(1R)-1-hydroxypropyl]-3-methylidene-5,6,7,8-tetrahydrochromen-2-one 4-[3-(3,4-dihydropyridin-5-yl)propanoylamino]-N-hydroxy-2,3-dihydrochromene-7-carboxamide 2-(3,5-dimethyl-1H-pyrazol-4-yl)-6-[4-(4-fluorophenyl)piperidine-1-carbonyl]pyridazin-3-one 3-fluoro-N,2-dimethyl-5-(prop-1-en-2-ylamino)aniline 4-[[1,3-dimethyl-2-oxo-6-(trifluoromethoxy)benzimidazole-5-carbonyl]amino]pyridine-3-carboxylic acid 3-chloro-5-[4-hydroxy-2,6-dioxo-1-(pyridine-3-carbonyl)-1,3-diazinan-5-yl]oxybenzonitrile 4-azido-2-[(4-methylphenyl)methoxy]pyrimidine 2-[3-(4,5-dimethylimidazol-1-yl)propyl]-4-pyridin-3-ylphthalazin-2-ium 2-[(3,5-dimethoxyphenyl)methyl]propanedioate N-[6-(1,3-benzothiazol-2-yl)-5-methoxypyridin-2-yl]pyridine-4-carboxamide 1,3-dihydroxy-4-methyl-2H-benzo[f]isoindole-6,7-disulfonic acid 1-[5-(3,4-dihydro-2H-chromen-6-yl)pyrazin-2-yl]ethanone (Z)-3-amino-N'-[4-[(5-methylthiophen-2-yl)sulfanylmethyl]-6,7-dihydro-1H-pyrrolo[2,3-b]pyridin-2-yl]prop-2-enimidamide 6-[2-(2,4-dichlorophenyl)pyridin-3-yl]-3-methylidene-1H-indol-2-one 2-[(4R,5S)-1-(3-fluorophenyl)-3-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridine-4-carbonyl]benzoic acid 5-(4-chlorophenyl)-7-methylsulfanylquinoline 6-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]pyridine-3-carboxamide (4-chlorophenyl)methyl-methanimidoyl-[4-morpholin-4-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-2-yl]azanium N-[2,4-difluoro-3-(6-methylquinazolin-4-yl)phenyl]-N',5-diethoxypyridine-3-carboximidamide N-[2,2-dimethyl-1-(4-sulfamoylphenyl)propylidene]-1-(3-hydroxy-5-oxo-7H-thieno[3,4-b]pyridine-6-carbonyl)piperidine-4-carboxamide 2-(4-propan-2-ylphenyl)quinoline 5-fluoro-2-[(4-formylcyclohexanecarbonyl)amino]benzoic acid 4-[N-(3-nitrophenyl)anilino]benzenesulfonic acid N-[1-(2,6-difluorophenyl)ethyl]-4,5,7,8-tetrahydro-1H-oxepino[4,5-c]pyrazole-3-carboxamide N-[5-chloro-4-(1H-indole-3-carbonyl)-2-methyl-6-phenylpyridin-3-yl]-3,4-dimethoxybenzamide N-benzyl-2,3-dimethoxy-4-phenylpyridine-3-carboxamide N'-[2,5-dichloro-4-(3,6-dicyanocarbazol-9-yl)phenyl]-N-propan-2-ylidenemethanimidamide [5-[2-(cyclopropylmethoxy)ethylamino]-1,3,4-thiadiazol-2-yl]-[2-(pyridine-3-carbonyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-yl]methanone;2,2,2-trifluoroacetic acid (3S)-5-[2-(1,3-benzodioxol-5-ylamino)pyrimidin-4-yl]oxy-3-ethylspiro[3H-chromene-2,4'-piperidine]-1'-carboxamide 2-[4-[2-(6,7-dimethoxy-3,4-dihydroisoquinolin-1-yl)ethynyl]phenyl]-N'-(2H-tetrazol-5-ylmethylidene)ethanimidamide 1-[4-(1,1-difluoroethyl)phenyl]-3-[2,5-dimethyl-4-[7-(trifluoromethoxy)quinolin-4-yl]oxypyrazol-3-yl]urea [2-ethylsulfanyl-6-[(4-fluorophenyl)methoxy]pyrimidin-4-yl]carbamic acid 5-chloro-N-[3-(4-fluorophenyl)sulfonylpropyl]pyrimidine-2-carboxamide 6-[4-(4-aminobutylamino)butyl]pyridine-3,5-diol 2-chloro-N-[5-(1H-pyrrol-3-yl)pentan-2-ylidene]aniline 3-[(4,4-dichlorocyclohexyl)methoxy]-5-hydroxybenzamide 2-[3-azidooxypropylsulfanyl(benzylsulfanyl)methylidene]oxane 2-(4-bromo-3,5-dimethoxyphenyl)-7-[2-(4-nitroimidazol-1-yl)ethoxy]-3H-quinazolin-4-one 5-fluoro-4-[3-(trifluoromethyl)phenyl]pyrimidine 6-(2-ethylphenyl)iminocyclohexa-2,4-dien-1-amine (5-amino-2-pyrimidin-4-yl-1,3-thiazol-4-yl)-(3-tert-butylphenyl)methanone 2-tert-butylsulfanyl-N'-hydroxypyrimidine-4-carboximidamide (1S,3R)-2,2,3-trimethyl-N-[(1-pyridin-4-ylpiperidin-4-yl)methyl]cyclopropane-1-carboxamide 2-(4-hydroxyphenyl)-5H-pyrrolo[3,2-d]pyrimidine-7-carboxylate (E)-3-[4-chloro-2-fluoro-3-(trifluoromethylsulfanyl)phenyl]-N-(1,3,5-triazin-2-ylmethoxy)propan-1-imine 2,6-diethylaniline;N,N',2,3-tetraphenylcyclohexa-1,5-diene-1-carboximidamide 5-(2-azidoethyl)-7-(trifluoromethyl)-1,3-dihydroindol-2-one (3-tert-butylphenyl)-[3-[(1-methylpyrazol-4-yl)methyl]azetidin-1-yl]methanone N-(5-bromopyrimidin-2-yl)-N'-phenylsulfanylethane-1,2-diamine 3-[2-[[1,6-dimethyl-2-oxo-4-(trifluoromethoxy)quinoline-3-carbonyl]amino]ethylamino]propanoic acid 1,2-bis[(2Z)-2-[1-(2,4-dimethylphenyl)ethylidene]hydrazinyl]ethane-1,2-dione (E)-N-[2-[4-[(3,5-dimethylpyrazol-1-yl)methyl]phenoxy]ethyl]prop-1-ene-1-sulfonamide (2S)-3-[(4R)-5-(6,7-dimethoxyquinazolin-4-yl)oxy-2,4-dihydroxypentanoyl]-N-[3-[[3-(trifluoromethyl)phenyl]sulfonylamino]propyl]pyrrolidine-1-carboxamide 2-methyl-5,7-dihydropyrimido[4,5-d]pyrimidine-6-thione 4-N,6-bis[(4-methoxyphenyl)methyl]pyrimidine-2,4-diamine 2-[(4S)-1-methyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]benzonitrile 3-[1,3-bis(2-ethoxyphenyl)-4-hydroxy-6,7-dimethylisoquinoline-8-carbonyl]benzoic acid N-[1-(6-phenylpyridine-2-carbonyl)pyrrolidin-3-yl]propane-1-sulfonamide (3-fluorophenyl)-[4-(1H-indazole-6-carbonyl)-1,4-diazepan-1-yl]methanone N-[6-(2,4-dihydroxyphenyl)pyrido[3,4-d]pyrimidin-2-yl]propanamide 2-[[1-(4,6-dimethylpyrimidin-5-yl)sulfonylpiperidin-4-yl]methoxy]-1-pyrrolidin-1-ylethanone 6-(1,3-benzothiazol-2-ylsulfanyl)pyridine-2,3-diol 3-[1-(1,2-benzoxazol-3-yl)piperidin-4-yl]-1H-quinazoline-2,4-dione N-[2-(5,6-dihydro-4H-cyclopenta[c]pyrazol-1-yl)phenyl]-5-methoxypyridine-3-carboxamide N-[5-(3-nitrophenyl)-1H-pyrazol-4-yl]pyridine-2-carboxamide 4-amino-3-[6-(2,2-dimethylpropanoyloxy)hexyl]-7-phenylmethoxychromen-2-one 4-(5,6-difluoro-2-methoxypyridin-3-yl)-7H-pyrrolo[2,3-d]pyrimidine N-(3-chlorophenyl)sulfonyl-2-[4-[3-(dimethylamino)propoxy]phenyl]acetamide 1-N,2-N,6-trimethyl-3-phenylbenzene-1,2-diamine ethane;(3E,5Z)-3-ethenyl-6-methoxyhepta-1,3,5-triene;N-methyl-2-[[(2S)-pentan-2-yl]amino]pyridine-4-carboxamide (4S,5R)-5-azido-1-[(1S)-1-phenylethyl]-2,2-dipropylpiperidine 2-ethoxy-4-(1-ethylpyrazol-3-yl)benzoic acid (3-bromo-2,4,6-trimethylphenyl)phosphane N-[(1S)-2,3-dihydro-1H-inden-1-yl]-3-methylimidazo[1,2-b]pyridazine-7-carboxamide (3R,4S)-1-benzyl-N-[(2-methoxyphenyl)methylidene]-3-nitropiperidine-4-carboxamide 4-(2,4,6-trimethylphenyl)-2,3-dihydrofuran (1S)-2,3-dihydro-1H-indene;4-fluorobenzaldehyde 4-chloro-6,8-dimethylquinoline-2,3-dicarboxamide 4-azidooxy-7,8-difluoroquinoline 2-[(2,4-dimethylphenyl)iminomethyl]-6-ethoxyphenol (2S)-3-methoxy-1,9-diphenyldecan-2-ol (1-azido-2-nitrocyclopentyl)benzene (Z)-1,3-bis[4-chloro-3-(dimethylamino)phenyl]prop-2-en-1-one N-(3,4-difluorophenyl)-1,2,5-trimethylpyrrole-3-carboxamide 5-[1-(3,4-dimethoxyphenyl)ethenyl]pyrimidine 1-(2-oxo-3H-indol-1-yl)pyrrole-2,5-dione ethane;1-[2-(3,4,5-trimethoxyphenyl)quinolin-7-yl]oxybutan-2-one 2-(1-azidooxy-4-hydroxycyclohexyl)benzonitrile 4-bromo-5-iodobenzaldehyde 1-N'-[1-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethoxymethyl]cyclopropane-1,1-dicarboxamide 2-(5-iodopyridin-3-yl)sulfonyl-N-methylsulfanylacetamide 2-(1,3-dihydropyrazol-2-yl)quinoline 1-azidooxy-4-methylsulfanylnaphthalene 2-[azido(methoxy)amino]sulfanylbenzoic acid 4-chloro-2,3,5,6-tetrafluoro-N'-hydroxybenzenecarboximidamide (4Z,5E)-1-methoxy-4-[2-(4-pyridin-3-ylpyridin-1-ium-1-yl)ethylidene]hepta-5,7-dien-2-one 3-(2-bromo-5-methoxyanilino)-4H-1,2,4-triazin-5-one 4-[(2-aminoethylsulfonylamino)methoxy]benzenesulfonic acid 2-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[5-ethyl-2-(trifluoromethoxy)phenyl]quinoline-7-carboxamide 2-[4-[4-(3-chlorophenyl)piperazin-1-yl]butoxy]acetic acid N-[1-(2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl)propan-2-yl]-2-(4-ethoxyphenyl)acetamide (2S)-4,5,5-trideuterio-3-[1,7-dimethyl-6-oxo-8-[(E)-3-phenylprop-2-enyl]-3H-imidazo[1,5-c]pyrimidine-2-carbonyl]-N-methyl-2-[4-(2-morpholin-4-ylethoxy)phenyl]pyrrolidine-1-carboxamide 3-(2,6-dimethylpyridin-4-yl)-5-[7-[ethyl(sulfino)amino]-6-fluoro-2,3-dihydroimidazo[1,2-a]pyridin-3-yl]-2H-pyrazolo[3,4-b]pyridine 4-[[1-cyclopentyl-3-(methylamino)-5,6-dihydropyrrolo[2,1-c][1,2,4]triazol-7-yl]oxy]benzenesulfonamide 7,8-difluoro-2,3-dimethylimidazo[1,2-a]pyridine 5-[3-chloro-4-(difluoromethoxy)phenyl]imidazolidine-2,4-dione (2R,6S)-4-[4-chloro-3-[1-[(4-ethylphenyl)methyl]piperidin-4-yl]oxyphenyl]sulfonyl-N-hydroxy-2-methyl-3-oxo-5-thia-1,7,11-triazatricyclo[6.4.0.02,6]dodeca-8,10-diene-12-carboxamide 4-(4-bromophenyl)sulfanyl-5-(2,5-difluorophenyl)-3-methoxycarbonyl-1,4-dihydropyridine-2-carboxylate N-ethylpropan-2-amine;(3E)-6-[4-methoxy-5-[2-(1,3-thiazol-2-yl)ethynyl]-1H-indol-3-yl]hexa-3,5-dienal 5-[(2,3-difluorophenyl)methyl]-N-[(1R)-1-(4-ethylsulfonylphenyl)-2-hydroxyethyl]-6-oxo-1H-pyrimidine-4-carboxamide 1-[(3Z,5E)-6-[4-[2-[4-fluoro-N'-(methylideneamino)carbamimidoyl]phenoxy]phenyl]oxyhepta-3,5-dienyl]piperidine-2-carboxylic acid 2-[3,5-bis(trifluoromethyl)anilino]-7-morpholin-4-yl-1H-pyrimido[4,5-d]pyrimidine-4,8-dione (4R)-1'-ethyl-7,10-dimethoxyspiro[1,3-dihydrobenzo[h]isochromene-2,4'-piperidine] 1-(3,5-dimethoxyphenyl)indole 2-[4-(cyclopenten-1-yl)phenyl]acetamide N-cyclopropyl-2-[4-[3,5-dichloro-4-(3-hydroxybutoxy)phenyl]sulfonylphenoxy]acetamide 7-chloro-3-[(E)-2-(5-chlorofuran-2-yl)ethenyl]quinazolin-4-one 1-azidooxy-4-(3,3,4,5,5-pentafluorocyclopenten-1-yl)benzene 6-fluoro-3-(1H-imidazol-2-yl)-1-methylquinoline 6-[(2,5-dimethylphenyl)sulfamoyl]pyridine-3-carboxylic acid 4-(3-azido-2-ethyl-6,7-dimethoxyquinolin-4-yl)morpholine 2-[4-(aminomethyl)phenyl]-6-[2,3-difluoro-4-(trifluoromethoxy)phenoxy]aniline N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]-1-formylcyclopropane-1-sulfonamide 5-N,6-N-bis(1,3-benzoxazol-2-yl)pyrimidine-4,6-diamine 3-amino-5,6-dimethoxynaphthalene-1,7-disulfonate 2-(2,4-dimethylphenyl)-N-(2-hydroxyethylsulfonylcarbamoyl)cyclopropane-1-carboxamide [(E)-1-benzyl-3-methyliminoindol-2-ylidene]-phenylazanium (1S,2R)-2-(4-fluorophenyl)-N-[6-(6H-pyrrolo[3,2-f]isoquinolin-5-yl)hexa-1,3,5-trienyl]cyclopropan-1-amine 2-[3-(6-methoxypyrimidin-4-yl)phenoxy]propanoic acid N-[(1R,2S)-4-methoxyimino-2-(6-oxo-4-phenyl-1H-pyrimidin-2-yl)cyclobutyl]furan-3-carboxamide 1-methyl-2-oxo-N-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)pyridine-4-carboxamide 3-fluoro-4-[6-methyl-7-(2-methylpyridin-4-yl)oxyimidazo[1,2-a]pyrimidin-3-yl]aniline 2-[3-(3,5-difluorophenyl)propyl]triazole 3-(3,4-diethoxyphenyl)-2-[(2-fluorophenyl)methyl]prop-2-enoic acid (2-cyclopentylpyrrolidin-1-yl)-[2-(3,4-difluorophenoxy)phenyl]methanone 1,3-bis(3-chlorophenoxy)propan-2-one 4-[3-(4,5-dihydro-1H-imidazol-2-ylmethoxy)-4-(trifluoromethylsulfonylamino)phenyl]benzoate 3-(2,5-dimethylphenyl)-1-ethenoxy-1,3-diazinane-2,4-dione 1-butyl-2,3,4,5,6,7,8-heptamethoxyanthracene 2-[4-[1-(3,4-dichlorophenyl)ethyl]piperazin-1-yl]acetamide ethane;5-[1-(2-methylpropoxy)ethenyl]pyridine-3,4-dicarbonitrile 2,3-dimethyl-5-[5-(6-phenylpyridin-3-yl)pentoxy]pyrazine 4-[5-(1,3-dioxolan-2-yl)pentyl]aniline 4-ethylsulfonyl-5,6,7,8-tetrahydronaphthalene-1-thiol 5-[3,6-bis(2-phenylphenyl)pyrazin-2-yl]pyrido[4,3-b]indole 3,5-diphenyl-6H-cyclopenta[b]thiophene N-[(1R)-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl]-4-(4-methoxyphenyl)piperazine-1-carboxamide 3-(1,3-benzodioxol-5-yl)-2,7-dihydropyrrolo[2,3-c]pyridazine 3-(4-bromocyclohexyl)naphthalene-1,2-dione N-(2,3-dihydro-1H-inden-2-yl)-3-hydroxybenzonitrilium 4-amino-3,5,6-trichloro-N'-hydrazinylpyridine-2-carboximidamide (2R)-2,3-dihydroxy-1,2,5-triphenylpentan-4-one 5-methyl-N-(2-morpholin-4-ylphenyl)furan-3-carboxamide 2-chloro-7-(cyclohexylmethyl)-4,5,6,8-tetrahydropyrazolo[1,5-d][1,4]diazepine;3-methylbut-1-ene 2-(4,5-dihydropyrimidin-2-yl)-N-[1-(3-methoxyphenyl)ethylideneamino]aniline 1-[6-(3,5-dichloropyridin-4-yl)-7H-purin-2-yl]-N'-hydroxypyrrole-2-carboximidamide N-[2,4-difluoro-3-(propanoylamino)phenyl]-4,5-bis(ethenyl)-1H-pyrrole-3-carboxamide N-[1,6-diethyl-3-(2-methoxyphenyl)-8-oxo-7H-imidazo[1,5-a]pyrazin-4-yl]cyclopropanecarboxamide N-[3,4-difluoro-2-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-5,6-dimethyl-4-oxofuro[2,3-d]pyrimidine-7-carboxamide [(5aS,8aR)-4-methyl-3,5,5a,6,8,8a-hexahydro-2H-pyrrolo[3,4-f][1,4]oxazepin-7-yl]-(1H-imidazol-5-yl)methanone;formic acid 1-(2,3-dihydro-1H-indol-5-yl)-N-methoxy-7-(1,4,5-oxathiazepan-4-yl)naphthalene-2-sulfonamide N-(2,6-difluorophenyl)-3-[methyl-[4-(4-methylpiperazine-1-carbonyl)phenyl]sulfamoyl]benzamide (4S)-2,5-dimethyl-N-[5-oxo-2-phenyl-1-(trifluoromethyl)pyrrolidin-3-ylidene]-6,7-dihydro-4H-1-benzothiophene-4-carboxamide 3,5-dimethoxy-N'-[[(E)-1-phenylpropan-2-ylideneamino]carbamothioyl]benzohydrazide 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[3-(propan-2-ylamino)butylsulfonyl]urea 2-[4,6-bis(trichloromethyl)-1H-benzimidazol-3-ium-5-ylidene]propanedinitrile;tetrakis(2,3,4,5,6-pentafluorophenyl)boranuide 1-(3-ethylpyridin-2-yl)-6,7-dimethoxy-3-sulfanylidene-4H-quinoxaline-2-thione 1-[(2S)-3,7-dibromoheptan-2-yl]oxy-4-[(1R,2R)-2-(4-methoxyphenyl)cyclobutyl]benzene N-[(1E)-3,4-dimethyl-2-[6-[4-methylidene-5-[(propan-2-ylamino)methyl]pyrazol-1-yl]pyridin-3-yl]penta-1,3-dienyl]ethanimine 1-(3,5-dimethylphenyl)-4-[2-ethyl-6-[2-fluoro-N-methyl-4-[(Z)-prop-1-enoxy]anilino]pyridin-3-yl]butane-2,3-dione;(Z)-pent-2-ene (2S)-N,3-dimethylbutan-2-amine;formaldehyde;4-methyl-1H-1,5-benzodiazepin-2-one (Z,4R)-4-[5-chloro-2-[1-(1H-indole-6-carbonyl)azetidin-3-yl]oxyphenyl]-N-methylpent-2-enamide N-[2-(2,4-dimethylphenyl)-3H-benzimidazol-5-yl]piperidine-1-carboxamide 1-cyclohexyl-2,5,5-trimethyl-3-[4-(2-methylphenyl)sulfonylpiperazin-1-yl]heptan-4-one N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-6,7-dihydro-1H-indazole-4-carboxamide N-[5-(1-ethyl-3,6-dihydro-2H-pyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-4-yl]cyclobutanecarboxamide ethane;5-fluoro-2,7-di(propan-2-yl)carbazole 7-bromo-3-(2,6-dichlorophenyl)-2-methylsulfonyl-5H-pyrido[4,3-b]indole [2-(3,5-difluorophenyl)pyrrolidin-1-yl]-(6-methoxypyridin-3-yl)methanone 2-(4-fluorophenyl)-N-[3-[5-(methylamino)-1,3,4-oxadiazol-2-yl]prop-1-en-2-yl]quinazoline-6-carboxamide;2,2,2-trifluoroacetic acid 2-[5-(1H-indol-3-yl)-6-(methylamino)pyrimidin-4-yl]oxyacetic acid 1-[(3S)-5-methyl-2,3,4,10-tetrahydropyrano[3,2-h][1]benzoxepin-9b-yl]ethanone;uranium(2+) N'-(4-hydroxyphenyl)octanediamide (4E)-5,8-dibromo-N-[3-[1-[2-(diethylamino)-1-phenylethyl]piperidin-4-ylidene]prop-1-en-2-yl]-6H-thieno[2,3-f][1,7]naphthyridine-2-carboxamide 3,6-diethyl-N'-methylidenebenzenecarboximidamide;5,5-diphenyl-1H-pyrrole (4R)-3-[hydroxy-(1H-indol-2-ylmethoxyamino)methyl]oxolane-2,4-dione [2-(2-methylpyrazol-3-yl)piperidin-1-yl]-(2-propan-2-ylpyrimidin-5-yl)methanone 2-[4,6-difluoro-3-(trifluoromethyl)phenyl]benzo[g][1,3]benzothiazole 1-[4-methyl-3-(2H-tetrazol-5-yl)phenyl]-N,N-dipropylpiperidine-4-carboxamide 5-fluoro-N-(3-oxo-2,5-diphenylcyclohexen-1-yl)pentanamide 2-[4-(1H-indol-3-yl)phenyl]benzoic acid ethane;N-(3-methylbutanoyl)-2,6-dinitrobenzamide 2-[5-(2,3-dihydro-1H-inden-5-ylmethylideneamino)pyridin-2-yl]oxyacetohydrazide 3-[4-(pyridine-2-carbonyl)phenoxy]propanoic acid 4-[2-(dimethylamino)ethoxy]benzamide N-(4-chlorophenyl)-5,7-dimethyl-3-[4-[4-(trifluoromethoxy)phenoxy]phenyl]-4,6,8,9-tetrahydropyrazolo[1,2-a]azepine-2-carboxamide (2S)-3-[4-chloro-5-methoxy-2-[2-[(2-methylpropan-2-yl)oxy]ethoxycarbonylamino]phenyl]-2-(pyrimidin-2-ylcarbamoylamino)propanoic acid 1-[4-(2-azidoethoxy)phenyl]cyclohexan-1-ol N-(4-fluorophenyl)-1-[4-(3-methylsulfonylpropoxy)phenyl]cyclopentane-1-carboxamide 2-[4-[(2E)-2-[3,5-bis(trifluoromethyl)phenyl]sulfonyliminopropanoyl]cyclohexyl]ethoxymethanesulfonic acid 2-azidooxy-4,6-ditert-butylphenol 5-ethylsulfanyl-6-fluoronaphthalene-2-carboxylic acid 4-[5-bromo-2-(cyclopropylmethoxy)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile 1-[2,3-dimethyl-4-(1H-pyrazole-5-carbonyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone 6-amino-2-[(2,4,5-trichlorophenyl)methylsulfanyl]-3H-quinazolin-4-one 5-cyclopropyl-2-[(4S)-1-(4-methoxybenzoyl)-6-phenylpiperidin-3-yl]oxypyridine-3-carboxylic acid 2-[4-(2,2-dimethylpropanoyl)piperazine-1-carbonyl]-3H-quinazolin-4-one (2S,4R)-N-[5-amino-6-(6-ethynyl-1H-benzimidazol-2-yl)hex-5-enyl]-4-fluoropyrrolidine-2-carboxamide 2-[3-methylbut-1-en-2-yl(pentan-2-ylidene)azaniumyl]benzenesulfonate N-[5-(furan-2-yl)pyridin-3-yl]sulfanyl-1,4-dioxane-2-carboxamide 2-methyl-N-[4-(oxiran-2-ylmethoxy)phenyl]butanamide 2-[3,5-di(propanoyloxy)phenyl]-2-oxoacetic acid 4-[2-hydroxy-3-(3,3,3-trifluoro-2-methylpropoxy)phenyl]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 6-(4-cyclopropylphenyl)-N,5,7-trimethylimidazo[1,2-a]pyrimidine-2-carboxamide (5E)-2-imino-5-[(2,4,6-trimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 3-[2-(3,4,5-trimethoxyphenyl)ethynyl]benzamide N-butan-2-yl-1-(3,4-difluorophenyl)sulfonylpiperidine-3-carboxamide 1-cyclohexyl-4-[4-(trifluoromethoxy)phenyl]imidazole 1,2-bis(methoxycarbonyl)perylene-3,4-dicarboxylic acid 5-amino-7-(3,4-dihydro-2H-1,5-benzodioxepine-7-carbonyl)-1H-indole-2-carbonitrile 3-bromo-6-(4-chlorophenyl)sulfonylquinoline N-[5-[[5-(3,4-dimethoxyphenyl)-3-hydroxypyrazolo[1,5-a]pyrimidine-7-carbonyl]amino]pyridin-2-yl]carbamate N-ethylpropan-2-amine;3-methoxy-5-methylphenol 2-[1,1,1,3,3,3-hexafluoro-2-(4-nitrophenoxy)propan-2-yl]benzenesulfonic acid 5-azido-2,3,4-tri(propan-2-yl)benzonitrile (2S,4R)-1-[3-(2,6-dimethoxyphenyl)benzoyl]-N-methyl-N'-(5-methylpyrazin-2-yl)-4-sulfanylpyrrolidine-2-carboximidamide N-[(E)-1,2-bis(phenylmethoxy)pent-3-enyl]-4-ethynylbenzamide (4-aminophenyl)-[3-(1,3,4-oxadiazol-2-yl)piperidin-1-yl]methanone 7-[(4-methoxyphenyl)methyl]-N,5-dioxopyrrolo[3,4-b]pyridine-6-carboxamide 1,2-dimethylpiperidine;ethane;6-(2-fluoro-4-methylanilino)-3-(trifluoromethyl)pyridine-2-carboxylic acid 1-benzyl-4,5-dimethoxyindole 4-benzyl-N'-[1,1-dihydroxy-6-[(2R)-2-pyridin-3-ylpyrrolidin-1-yl]-1,2,3,4-tetrahydronaphthalen-2-yl]morpholine-2-carboximidamide 3-[3-[4-(dimethylamino)phenyl]phenyl]-3-oxopropanamide N-[(E)-2,4-dimethylpent-1-enyl]propan-1-imine;ethane;2-[(5R)-3-ethoxy-6-oxo-5H-phenanthridin-8-yl]acetaldehyde N-(3-chlorophenyl)-2-[(6S)-5,7-dioxo-3-thiophen-2-yl-4H-pyrazolo[1,5-a]pyrimidin-6-yl]acetamide 5-(2,3-dihydropyrrole-1-carbonyl)pyrazine-2-carboxylic acid 1-[2-(1,3-dioxolan-2-yl)ethoxy]-4-(2,6-dimethylphenyl)triazole 4-N-[3-(7,8-dimethyloctyl)phenyl]-2-N-[4-(4-propan-2-ylpiperazin-1-yl)sulfonylphenyl]pyrimidine-2,4-diamine 1-cyclopentyl-2-[(4-fluorophenyl)methoxy]propan-1-ol 3-[[4-(6-methoxypyridine-2-carbonyl)piperazin-1-yl]methyl]pyrrolidin-2-one 1-N,3-N,3-N-triethylbenzene-1,3-dicarboxamide 3-[(1Z)-buta-1,3-dienyl]-5-methyl-8H-cyclohepta[b]pyridine 2-[(3S)-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione (E)-N'-[[2-(1,3-benzodioxol-5-yloxy)pyridin-4-yl]methyl]-2-ethenyl-3-propan-2-ylidenehex-4-enimidamide N-[1-[3-(4-ethylphenyl)propanoyl]piperidin-2-yl]acetamide N-butyl-2,6-dimethoxy-3H-benzimidazole-5-carboxamide;hydrochloride N-[(2E)-1-cyclopentyloxypenta-2,4-dien-2-yl]-1-(4-methylphenyl)ethanimine 5-amino-2,4-dimethylquinazoline-8-carboxylic acid 3-(4-chlorophenyl)-4-methylsulfanylmorpholine 5-ethyl-3,6-di(propan-2-ylidene)isoindol-1-one 1-(2,3-dihydroindol-1-yl)-2-(2,4-dimethoxyphenyl)ethane-1,2-dione;hydrochloride 1-methylsulfonyl-2-(pyridin-3-yloxymethyl)pyrrolidine-2,5-dicarboxylic acid (5S,6R)-3-[4-[1-(2-hydroxypropan-2-yloxymethoxycarbonylamino)-3-iminopropoxy]-3-methoxyphenyl]-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid N-(2,3,3a,4,5,6,7,7a-octahydro-1H-inden-1-yl)-4-[(2,6-difluorobenzoyl)amino]pyrazole-1-carboxamide N-(2,3-dihydro-1H-inden-5-yl)-4-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)piperidine-1-carboxamide N'-[(3R)-1,2,3,4-tetrahydroquinoline-3-carbonyl]benzohydrazide N-[5-fluoro-3,4-dioxo-6-(trideuteriomethyl)spiro[1H-quinoxaline-2,4'-oxane]-8-yl]carbamate 2-(1,4,5,6-tetrahydropyrimidin-2-yl)benzimidazole 2-amino-6,7-dimethoxy-4,5-diphenylheptanoate N'-(3-anilino-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-yl)pentanehydrazide (2S)-2-[(2R)-6,7-dichloro-1-fluoro-3,4-dihydronaphthalen-2-yl]-N-[(3R,4S)-3-methoxyoxan-4-yl]propanamide N-[(E)-butanoyl]-4-methyl-5-nitrosofuran-3-carboxamide 7-[4-(2,3-dihydro-1H-inden-5-yl)piperazine-1-carbonyl]-8-methylpyrido[2,3-d]pyrimidin-6-one 5-[4-(4-cyclopentylbutoxy)phenyl]-3-fluoro-2,7-dimethylpyrazolo[1,5-a]pyrimidine 3-[1-(4-fluorophenyl)cyclobutyl]-5-(2,2,2-trifluoroethoxymethyl)-1,2,4-oxadiazole 5-(4,8-dimethylnonyl)pyrimidine 1,2-dihydroxy-N-phenylcyclohexane-1-carboxamide (2S)-2,5,7,8-tetrahydroxy-6,9-dioxo-2H-benzo[c]chromene-3-carboxylic acid N-methyl-2-[(3E,5Z)-2-oxohepta-3,5-dienyl]-4-phenylbutanamide 5-chloro-4-[(3R)-4-ethyl-1,4-oxazepan-3-yl]-1H-pyrimidin-6-one;hydrochloride N-[2-[4-[(2,6-dichlorobenzoyl)amino]phenyl]ethyl]-1H-indazole-3-carboxamide N-[4-(3,5-dimethylphenyl)-1,2,4-triazol-3-ylidene]formamide;oxan-2-amine N-[4,6-difluoro-1'-(1H-indole-2-carbonyl)spiro[2,3-dihydrochromene-4,4'-piperidine]-7-yl]methanesulfonamide N-[3,4-difluoro-2-(1H-pyrazolo[3,4-b]pyridin-5-yl)phenyl]formamide 6-ethyl-2,4-dimethoxybenzenesulfonate 2-[(1R)-6,7-dimethoxy-4-oxo-3H-quinazolin-2-yl]-N-propan-2-ylacetamide 2-[2,6-dichloro-N-(3,3-dimethylbutyl)-4-nitroanilino]acetonitrile 3-bromo-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]benzaldehyde N-(1,3-thiazol-2-yl)-1H-indole-2-carboxamide N-[3-[3-(2,4-dioxopyrimidin-1-yl)propylamino]phenyl]-2H-triazole-4-carboxamide 1-[(2Z,4E)-hepta-2,4,6-trien-3-yl]-5H-imidazo[1,2-a]quinoxaline 5-(3,4-dimethoxyphenyl)-1,2,5-oxadiazolidine-6-carbonitrile;(2R,4S)-2,4-dimethylpiperidine 2-[3-(3,6-dihydro-1H-cyclopenta[c]pyrazol-5-yl)piperidin-1-yl]quinoxaline (3R)-5,5-difluoro-3-[2-[4-methoxycarbonyl-1-(4-propan-2-ylphenyl)sulfonylpyrrolidin-3-yl]ethynyl]-6-oxohexanoic acid 3-[4-(2,2,3,5,5-pentadeuteriopentyl)piperazin-1-yl]aniline 6-(4-chlorophenyl)-3-phenyl-2,5,7,11,13-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,10-trien-8-one 4-[4-(benzenesulfonyl)piperazin-1-yl]-7-methoxyquinoline 4-(2-tert-butylphenyl)-1-cyclopropylideneisoindole 6-chloro-1H-indole;5,9-dimethylpyrido[2,3-b]indole 6-[(5R)-2,5-dimethylpyrrolidin-1-yl]-4-N-[(Z)-(3-nitrophenyl)methylideneamino]-2-N-propylpyrimidine-2,4-diamine 4-[(2,6-dichlorophenyl)methyl]quinazoline 2-[6,7-difluoro-1'-(3-methylphenyl)sulfonylspiro[3H-chromene-2,4'-piperidine]-4-yl]acetic acid 2,3-dimethoxy-N-[(4-propan-2-ylphenyl)methyl]aniline 2-[4-(cyclobutylmethylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile;hydrochloride 4-[5,6-bis(ethenyl)pyridin-3-yl]-2-methanimidoyl-5-N,5-N-dimethylpyridine-1,5-diamine (E)-2-[amino(methyl)amino]-1-phenylbut-2-en-1-one 2-(6-fluoro-5-pyridin-3-ylindazol-1-yl)oxyethanol 4-amino-3,5-dimethyl-N-[(E)-(2-methylidenenaphthalen-1-ylidene)amino]benzamide (2S)-3-[4-[3-(4-chlorophenoxy)phenyl]sulfonylpiperazin-1-yl]propane-1,2-diol 3-[(1Z)-3-[4-(2-methylpyridin-4-yl)oxypiperidin-1-yl]buta-1,3-dienyl]pyridine N-(4,6-dimethylpyrimidin-2-yl)oxy-1-benzofuran-3-carboxamide 3-(N-hexadecyl-4-methoxyanilino)propane-1,2-diol 2-amino-4-[1-(pyridin-3-ylmethoxy)cyclohexyl]-6H-pyrrolo[3,4-d]pyrimidine-5,7-dione 3-cyclopropyl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole-6-carbonitrile;ethane 3-[4-[3-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyrrol-1-yl]phenyl]sulfonylpyrrolidine-2,5-dione (5-amino-3,4-dihydroxy-2-methylphenyl)urea 6-chloro-2,3,4-trifluoropyridine;N-[(1S)-1-[1-methyl-5-(2,2,2-trifluoroethoxy)benzimidazol-2-yl]butyl]formamide 1-methylsulfanyl-2-[(Z)-prop-1-enyl]xanthen-9-one N-[(1R)-3-hydroxycyclohexyl]-6-pyridin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide 7-[2-methoxyethyl(pentanoyl)amino]-6,8-dihydro-5H-4,1-benzoxazepine-3-carboxamide 3-[(4R,5R)-3-amino-5-fluoro-2,7,10-triazabicyclo[9.4.0]pentadeca-1(15),11,13-trien-9-yl]benzaldehyde N-[(1R)-3-aminocyclopentyl]pyrazolo[1,5-a]pyridine-2-carboxamide 3-(5-chloropyridin-2-yl)-4-cyano-N,N,4-trimethylpyrrolidine-1-carboxamide 3,9,13-triazatetracyclo[7.6.0.02,6.010,14]pentadeca-1(15),2(6),4,8,10(14)-pentaene 2-amino-6-borono-3-[(1,3-dioxoisoindol-2-yl)oxy]hexanoic acid 3-[(2-amino-4,5-dimethylphenyl)carbamoyl]-6-oxocyclohexa-2,4-dien-1-olate 1-[(3,5-difluorophenyl)methyl]-4-[4-(trifluoromethoxy)phenoxy]piperidine 2-[(Z)-2-(aminomethyl)-3-fluoroprop-2-enoxy]-4-[7-[1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]quinolin-5-yl]oxyaniline 7-chloro-N-ethyl-3,4-dihydro-2H-1,5-benzoxazepine-5-carboxamide 2-[4-(3,5-dimethylpyrazol-1-yl)butyl]-6-methoxy-1H-benzimidazole (4S)-3,4-dimethyl-1-[5-phenyl-6-(trifluoromethyl)pyridazin-3-yl]-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one [3-(1H-pyrazole-5-carbonyl)piperidin-1-yl]-[4-(5,6,7,8-tetrahydroquinazolin-2-yl)phenyl]methanone 7-(5-ethylpyridin-3-yl)oxy-1,3-dimethyl-8-[4-(1H-pyrazol-4-yl)anilino]imidazo[4,5-c]quinolin-2-one 5-(3,4-dimethoxyphenyl)-N-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethyl-formamidoamino]ethyl]pentanamide 2-(3,5-dimethylphenyl)-4-(prop-1-en-2-ylsulfanylmethyl)pyridazin-3-one ethane;N-(2-ethylbutyl)-4-[(3-methyl-1,2-thiazol-5-yl)sulfonylamino]benzamide (4Z,6E)-8-ethenyl-N-methoxy-1-[(4-methoxyphenyl)methoxy]-2-methylsulfanyl-7-morpholin-4-ylocta-4,6-dien-3-imine 1-(2,3-difluorocyclobutyl)-4-(4,6-difluoro-5H-pyrrolo[3,4-d]pyrimidin-7-yl)azepane N-[1-(4-methylphenyl)ethenyl]-5-piperidin-3-ylpyridine-2-carboxamide (2E,4Z)-5-methoxyimino-N-methyl-1-[2-(1H-pyrrole-3-carbonyl)-2,10-diazatricyclo[6.3.0.03,6]undeca-1(11),2,4,7,9-pentaen-8-yn-12-ylidene]pentan-2-imine 4-[6-(2-chloroanilino)pyridin-3-yl]-1H-pyridin-2-one 5-amino-4-[4-[(2,3-difluorophenyl)methoxy]-3-methoxyphenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 2-(3,4-dimethylbenzo[g]indol-7-ylidene)propanedinitrile 1-[2-methoxy-4-[(3R)-pyrrolidine-3-carbonyl]phenyl]ethanone 4-[1-(4-fluorophenyl)ethenyl]-N-(3-methoxypropylsulfanyl)-2H-chromene-7-carboxamide 4-[(4,5-dichloro-1H-imidazole-2-carbonyl)amino]-3-ethoxybenzoic acid 2-(4,6-dimethylpyrimidin-5-yl)oxy-N'-[(2R)-1-hydroxypentan-2-yl]pyridine-3-carboximidamide (4S)-1-ethyl-3,3-dimethyl-4-[2-nitro-5-(trifluoromethoxy)phenyl]pyrrolidine 6-(4-fluorophenyl)-3-[2-oxo-2-[2-[1-(trifluoromethyl)cyclopropyl]piperidin-1-yl]ethyl]sulfanyl-4H-1,2,4-triazin-5-one 2-[5-(4,6-dimethoxypyrimidin-2-yl)sulfanylpentyl]isoindole-1,3-dione (2R)-N-[[3,4-bis(phenylmethoxy)phenyl]methyl]pyrrolidine-2-carboxamide;dihydrochloride [[4-(difluoromethyl)phenyl]sulfonylamino]carbamic acid (2E,4Z)-N,3-diethyl-2,5-bis[(1S)-1-(6-methoxynaphthalen-2-yl)-2-oxopropyl]hexa-2,4-dienamide;ethane 1-[3,5-bis(trifluoromethyl)phenyl]-4-[(1R)-3-(dimethylamino)cyclopentyl]butan-2-one 1-[2,6-dichloro-4-(2-hydroxypropan-2-yl)phenyl]-3-[[5-ethoxy-2-methyl-4-(trifluoromethyl)pyrazol-3-yl]sulfamoyl]urea N-[5-(dimethylamino)naphthalen-1-yl]-2,5-dihydro-1H-pyrrole-3-carboxamide 5-methyl-N-(2,2,2-trifluoroethyl)-3H-indene-1-carboxamide N-[(5R)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl]-1-(4-fluorophenyl)pyrazole-3-carboxamide 2-(2,4-dimethoxyphenyl)-N'-hydroxy-1H-imidazo[4,5-b]pyridine-7-carboximidamide (3S,4R)-1-[5-(3-chlorophenyl)-6-methoxypyridin-2-yl]-N-ethyl-3-(hydroxymethyl)piperidine-4-carboxamide (E)-4,5-diamino-N'-[1-(2,3-dihydro-1H-inden-5-yloxy)ethyl]oct-7-enediamide 1-azido-4,5-diphenylbenzene [2-chloro-3,5-dimethyl-6-(1,2,4-triazol-1-yl)pyridin-4-yl]urea N-[2-chloro-5-(4,6-diethoxypyrimidine-5-carbonyl)phenyl]-1H-imidazole-2-carboxamide [1-[2,5-dimethyl-4-(5,6,7,8-tetrahydroquinolin-3-yloxy)phenyl]cyclopropyl]carbamic acid 2-[(2S,3aS)-1-(cyclopropanecarbonyl)-10,10-dimethyl-5-methylidene-6-methylidene-3-oxo-4H-imidazo[1,5-b]isoquinolin-2-yl]acetaldehyde 3-[2-methoxy-5-[1-(1-piperidin-4-ylpiperidin-4-yl)benzimidazol-2-yl]phenyl]prop-2-enamide 2-[4-[2-[4-(aminomethyl)phenyl]ethyl]pyrimidine-5-carbonyl]guanidine;hydrochloride 2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3-propan-2-yl-5H-pyrrolo[3,2-d]pyrimidine 2-ethoxy-N-[(3-imidazol-1-ylphenyl)methyl]acetamide 1,2-diamino-4-(3-butylphenyl)-6-oxopyridine-3,5-dicarbonitrile N-(4,5-dimethyl-2H-pyrazolo[3,4-b]pyridin-6-ium-7-ylidene)hydroxylamine 7-[3-(2,6-dimethylphenyl)imidazol-4-ium-1-yl]thieno[3,2-c]pyridine;(Z)-3-hydroxy-1,3-thiazolidine-2-thione;iridium 4-[1,2-bis(3-cyanophenyl)ethyl]piperazine-1-carboxylic acid 2-azido-N,N,1-triphenylpiperidin-4-amine 4-tert-butyl-1-methoxy-2,3-dihydroisoquinoline N-[2-fluoro-5-(2-hydroxypropan-2-yl)phenyl]methanesulfonamide 1-[2-(4-fluorophenyl)ethyl]-3-methyl-2-sulfanylideneimidazolidine-4,5-dione 2-[1,4-bis(ethenyl)piperidin-4-yl]oxypyridine 2-amino-4-(3,5-dihydroxyphenyl)-2H-pyran-6-carbonitrile 2-[(1S)-1-[[3-(trifluoromethoxy)benzoyl]amino]ethyl]benzoic acid N-[(E)-1-(2,6-dihydroxyphenyl)ethylideneamino]-2-methylsulfanylacetamide 2-tert-butyl-7-[4-(cyclohexylamino)piperidine-1-carbonyl]-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one (3S)-2,3,4a,5-tetrahydroindeno[1,2-b]pyridine (2Z,4E)-3-[4-amino-5-(4-phenoxyphenyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-N'-methanimidoylpenta-2,4-dienimidamide 3-[1-[(E)-2-ethenylbut-2-enoxy]ethenyl]-N,4-dimethylaniline;(E)-4-fluoropent-3-ene 6-(2-chlorophenyl)-8-N-[4-fluoro-3-(trifluoromethyl)phenyl]pyrido[1,2-a]pyrimidine-2,8-dicarboxamide 1-[(E)-2,3-dimethylbut-1-enyl]-5,6,7,8-tetrahydroisoquinoline 1-methyl-3-[2-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]thiourea 2,6-dimethyl-N-(4-pyrazin-2-yloxyphenyl)pyridine-3-carboxamide 5-(2,4-dihydroxyphenyl)-N'-methylfuran-2-carbohydrazide 3-(2,6-difluorophenyl)sulfonyl-5-(4-methyl-1,2,4-triazol-3-yl)pyridine 2-amino-N-[2,3-bis(ethenyl)quinoxalin-6-yl]acetamide 2-amino-9-[(3R,4S)-1-methyl-5-oxopyrrolidin-3-yl]-7-phenyl-1H-purine-6,8-dione (4-bromo-3,5-difluorophenyl)-[(2S)-3-methylbutan-2-yl]azanium (3aR,7aR)-2-[3-(3,5-dimethylpyrazol-1-yl)propanoyl]-1,3,4,6,7,7a-hexahydropyrano[3,4-c]pyrrole-3a-carboxylic acid 1-[(3S,7R,8aS)-3-cyclopropyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-3-pyridin-4-ylurea;formic acid (2R)-1-acetyl-N-[4-chloro-3-(trifluoromethoxy)phenyl]pyrrolidine-2-carboxamide 3,4-difluoro-N'-hydroxybenzenecarboximidamide;hydrochloride 5-azidooxy-2,6-difluoroindazole 6-(hydroxymethyl)-N-[1-[4-(trifluoromethoxy)phenyl]propan-2-yl]pyridine-3-carboxamide 1-[5-(benzylamino)sulfanylnaphthalen-1-yl]sulfinyl-N,N-dimethylpiperidine-4-carboxamide 3-fluoro-N'-methyl-4-pyrrolidin-1-ylaniline 3-aminosulfanylnaphthalene-1,6-disulfonic acid [5-methyl-4-(2-naphthalen-1-ylamino)pyrimidin-2-yl]cyanamide 4-[3-chloro-6-(2,3-difluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-N-[3-(5-hydroxypyridin-2-yl)butan-2-ylidene]piperidine-1-carbothioamide N-[(4S)-4-benzylimino-2,8-dioxo-3,4-dihydrochromen-7-yl]-5-chloro-6-methoxypyridine-3-sulfonamide 2-[4-[(7-oxo-1,6-dihydropurin-8-yl)amino]phenyl]acetic acid 2-amino-5-(3,5-difluorophenyl)-3-[6-hydroxy-4-methoxy-8-[2-oxo-4-[4-(1,3-oxazol-5-yl)phenyl]butyl]-7,8-dihydrobenzo[e]benzimidazol-1-yl]pentanoic acid 2-(1,4-dimethylpiperazine-2-carbonyl)-8-oxa-2-azaspiro[4.5]decane-4-carboxylic acid N-(cyclopropylmethoxy)-5-(4-ethylsulfinylphenyl)pyrazine-2-carboxamide 6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-ethylsulfanylpyrido[4,3-d]pyrimidin-7-imine 1-[2,2-bis(4-methoxyphenyl)ethyl]-3-cyclopentyl-5-nitroimidazol-2-one ethane;2-phenyl-3,4-dihydro-1H-isoquinoline 4-(6-azidooxyhexyl)benzonitrile ethane;(2E,4Z)-hepta-2,4-diene-3-thiol;methanol;2-[5-[2-[[6-phenyl-3-[(Z)-prop-1-enyl]-5,6,7,8-tetrahydroisoquinolin-1-ylidene]amino]phenyl]pyridin-2-yl]acetonitrile 1-[3,5-difluoro-4-(2-morpholin-4-ylethoxy)phenyl]-3-[[5-(3-methoxypropyl)-1-methylpyrazol-4-yl]amino]-5H-pyrazolo[4,3-c]pyridin-4-one 1-butanoyl-N-[5-(2,4-difluorophenyl)sulfonyl-7a-methyl-3H-1,3-benzoxazol-2-ylidene]pyrrolidine-2-carboxamide 3,4-dimethylpentanal;4-(ethylamino)-3-[6-formamido-4-(hydroxyamino)-7-oxothieno[2,3-b]pyridin-2-yl]benzaldehyde [(2R)-4-ethyl-6-(4-methoxycarbonyl-3,5-dihydro-2H-1,4-benzoxazepine-7-carbonyl)-6-azaspiro[2.4]heptan-2-yl]carbamic acid N-(2,3-dihydropyridin-5-yl)-2-[methoxy(sulfanyl)amino]acetamide;N-[4-(1-piperidin-1-ylethenyl)phenyl]cyclopropanecarboxamide 4-(4,6-dimethoxypyrimidin-2-yl)-2-[5-(6-methylcyclohexa-1,3-dien-1-yl)pentanoylamino]thiophene-3-carboxylic acid 3-[5-[4-(benzenesulfonyl)phenoxy]-6,7-dihydroindazol-2-yl]-N-methyl-3-phenylpropanamide 2-[4-(2-hydroxyphenyl)-6-methyl-1,3,5-triazin-2-yl]phenol 5-(2,4-dimethylphenyl)-2-[1-[4-ethoxybutyl(methyl)amino]ethenyl]-3-methylaniline (7S)-4,8-dimethyl-2-[[1-(piperidine-4-carbonyl)piperidin-3-yl]amino]spiro[5H-pteridine-6,3'-pyrrolidine]-2',7-dione;dihydrochloride 1-[2-[(3-amino-5-methyl-1H-pyrazol-4-yl)diazenyl]-4,5-dibromothiophen-3-yl]ethanone 4-(7-hydroxyimidazo[1,2-a]pyridine-3-carbonyl)piperazin-2-one N-(2-fluoropyridin-4-yl)-1H-imidazo[4,5-b]pyridin-7-amine 2,6-dimethyl-4-[4-[2-methylidene-1-(3-nitrophenyl)-8-oxoimidazo[4,5-g]phthalazin-5-yl]piperazin-1-yl]benzonitrile 2,3-dimethyl-4-(2,3,5,6-tetrafluorophenyl)pyridine 4-methoxy-N,1-diphenyl-2-phenylmethoxybutan-1-imine N-[(Z)-1H-indol-3-ylmethylideneamino]-4,5-diphenylfuran-2-carboxamide 2-methyl-3,4-bis(prop-1-en-2-yl)-5-pyrimidin-4-ylpyridine 3-[1,4-dimethyl-2-(2-methylphenyl)-5-methylsulfanyl-8H-cyclohepta[d]pyrimidin-7-ylidene]-2,2-bis(sulfanylidene)propanenitrile (E)-N-[(2S,3R)-1-(3,5-difluorophenyl)-4-hydroxy-3-pyrrolidin-1-ylbutan-2-yl]-3-(3-methoxyphenyl)prop-2-enamide 2-(1H-indol-3-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole 5-[4-(1,2,3,6-tetrahydropyridin-4-yl)phenyl]pentanoic acid 2-(2,6-dichloroanilino)-N-ethyl-5-oxo-7H-pyrrolo[3,4-b]pyridine-6-carboxamide 1-(2,3-dihydro-1H-inden-2-yl)-6-[5-(3,4-dimethoxyphenyl)pentanoyl]piperidin-2-one (2E,4Z)-5-[5-amino-6-(N,4-dimethylanilino)pyrazin-2-yl]hepta-2,4,6-trienal;cyclohexane 4-[3-(2,6-diamino-5,8-dioxonaphthalen-1-yl)phenyl]naphthalene-1,7-disulfonic acid 4-[(6,8-dimethoxyquinazolin-4-yl)amino]-2-(1-methylpiperidin-3-yl)phenol 6-(2,4-dimethoxyphenyl)-1-ethylbenzimidazole 1,2-diamino-4-(3-hydroxyphenyl)-6-oxopyridine-3,5-dicarbonitrile 2-(3-iodocyclohexa-1,5-dien-1-yl)pyrimidine 2-[5-carbamoyl-9-(cyclobutylmethyl)carbazol-4-yl]oxyacetic acid 6-cyclopentyloxy-N-[1-(cyclopropanecarbonyl)pyrrolidin-3-yl]pyridine-2-carboxamide 2-amino-4-[3,5-bis(trifluoromethyl)phenyl]quinoline-6-carbonitrile ethane;2-ethyl-1-(3,4,5-trimethoxyphenyl)butan-1-one 5-[(E)-3,6-dimethyloct-2-enoxy]carbonylthiophen-2-olate N-[(2S,3R)-1-(1H-indole-6-carbonyl)-2-methylpyrrolidin-3-yl]-5-phenyl-1,3,4-oxadiazole-2-carboxamide 5-[3-[4-(3,4-dimethoxyphenyl)piperazin-1-yl]propoxy]-6-piperidin-1-ylsulfonyl-2H-indole 3-[2-(cyclopropanecarbonylamino)imidazo[1,2-b]pyridazin-6-yl]benzoic acid 2-[(4R)-3,3-difluoroazetidine-1-carbonyl]-7-(trifluoromethyl)-10H-thieno[3,4-b][1,5]benzodiazepine-4-carbonitrile 2-(cyclobutylmethyliminomethyl)-4,6-diiodophenol 4-[2-(dimethylamino)ethyl-methylamino]-N'-hydroxypyridine-2-carboximidamide (3Z)-1-(4-chlorophenyl)-3-[2-(furan-2-ylmethylamino)-5-nitropyrimidin-4-yl]iminopropan-1-one 2-[4-fluoro-5-methyl-3-(trifluoromethyl)pyrazole-1-carbonyl]pentanal 6-chloro-N-[4-[3,5-dimethyl-1-(4-nitrophenyl)pyrazol-4-yl]but-1-en-2-yl]-3-methylpyridin-2-amine N'-[5-(difluoromethyl)pyridin-3-yl]sulfanyl-2,4-dinitrobenzohydrazide 5-(disulfanyl)-N,2-dimethoxy-N-phenylpyridine-3-carboxamide 5-[(2,4-dimethylphenyl)diazenyl]-2-hydroxy-1-propan-2-yl-6-(pyridin-3-yliminomethyl)pyrimidin-4-one 2-[(5,6-dichloro-1H-benzimidazol-2-yl)methoxy]pyridine-3-carboxamide 5-[1-(2,4-dimethylphenyl)butan-2-yl]-4H-1,3-benzothiazine;ethane (1-azidoazetidin-3-yl)-[2-cyclohexyl-5-(2,6-dimethoxyphenyl)-4-hydroxypyrazol-3-yl]methanone 1-(2,2-dimethylpropanoyl)oxycarbonylanthracene-9,10-dicarboxylic acid 2-(4,6-dimethylpyrimidin-2-yl)oxy-N-(1H-indazol-6-ylcarbamoyl)-3-phenylpropanamide 3-amino-N-[2-(4-chloro-6-methylpyrimidin-5-yl)ethyl]-6-phenylpyrazine-2-carboxamide 4-azidosulfanyl-6,7-diphenylthieno[3,2-d]pyrimidine N-[5-[3-(7-pyridin-4-yl-1H-imidazo[4,5-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]propanamide N-benzyl-4-oxo-4-[(3S)-1-(4-phenylphenyl)pyrrolidin-3-yl]butanamide 4-fluoro-3-methyl-N'-[(2E)-2-methyl-5-oxopenta-2,4-dienimidoyl]benzenecarboximidamide 4-azidooxy-N,N-diethylaniline N-(3,4-dimethylphenyl)sulfonyl-1,2,3,5,6,7-hexahydropyrrolizine-8-carboxamide 6-methyl-2-(4-propan-2-ylphenyl)-3,4-dihydropyrrolo[1,2-a]pyrazine-1,7-dione 3-bromo-N-cyclopropyl-5-(trifluoromethoxy)benzamide 3-[2-(3,4,5-trifluorophenyl)ethyl]azetidine 1-[4-(1,3-benzoxazol-2-yl)phenyl]cyclopropan-1-amine [2,6-diamino-5-(cyclohexyliminomethyl)pyrimidin-4-yl]-[4-[(3S)-oxolan-3-yl]piperazin-1-yl]methanone 1-[5-(3-methylsulfonylphenyl)pyrazolo[4,3-b]pyridin-1-yl]ethanone 3-[(2E,4Z)-5-tert-butylhexa-2,4-dien-2-yl]-N-propan-2-ylidenebenzenecarboximidamide 3-[4-(2,2-difluoroethoxy)phenyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine 1-(6-chloroquinoline-3-carbonyl)piperidin-4-one 1-phenyl-4-pyridin-3-ylindole 3-[(4-aminobenzoyl)amino]-5-phenylbenzoic acid 4-methoxy-N-[(2S,3R)-1-methyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]pyridine-2-carboxamide N-[(3E)-4,6-dimethylhepta-1,3-dien-2-yl]-2-methylaniline 3-[4,5-bis(ethenyl)imidazol-1-id-2-yl]propan-1-amine;propane;uranium(2+) 2-(2,3-dichloroanilino)-N-[[4-(trifluoromethylsulfanyl)phenyl]methyl]pyridine-4-carboxamide 2-ethyl-4-[5-(4-fluorophenyl)pyrazin-2-yl]benzoic acid 2-[2,4-dibromo-6-(5-nitropyridin-3-yl)phenoxy]acetonitrile N-[4-(2,5-dimethylphenyl)piperazin-1-ium-1-ylidene]hydroxylamine;bromide 2,5-dimethyl-4-(2,4,6-trichlorophenyl)-1H-pyrimidin-6-one (E)-3-phenylhept-2-enal [1-methylsulfonyl-3-(1,2,4-triazol-4-yl)pyrazol-4-yl]-[3-(1H-pyrrol-2-yl)pyrrolidin-1-yl]methanone 6-(4-bromophenyl)sulfonyl-9,10,16-triazatetracyclo[8.7.0.02,8.011,16]heptadeca-1(17),2,4,6,11(16),12-hexaene 4-[5-[1,3-bis(ethenyl)pyrrol-2-yl]furan-2-carbonyl]benzamide 4-N,8a-dimethyl-1-[3-(trifluoromethoxy)phenyl]sulfonyl-2,3,4a,5,6,7,8-hexahydro-1H-naphthalene-2,4-diamine 2-amino-4-methyl-6-[3-(trifluoromethoxy)phenyl]benzene-1,3-dicarbonitrile N-[3,5-dimethyl-1-(oxan-4-yl)pyrazol-4-yl]-2-oxo-1,5,6,7,8,9-hexahydrocyclohepta[b]pyridine-3-carboxamide (3S)-N'-cyclopentyl-2-oxo-1-phenylpiperidine-3-carbohydrazide ethane;2-(5-hydroxyspiro[3H-1-benzofuran-2,4'-piperidine]-4-yl)acetonitrile 4-azido-6,7-dichloronaphthalene-2-sulfonic acid 3-[(1S)-2,4-dimethylcyclohexa-2,4-dien-1-yl]sulfanylpyridine (2S)-N,N-dimethyl-3-[4-[5-phenyl-1-(pyridine-3-carbonyl)pyrazol-3-yl]phenyl]sulfanyloxolane-2-carboxamide 2-amino-9H-indeno[1,2-b]pyridine-3-carboxamide 2-(4-fluorophenyl)-1,4-dimethylbenzene;(Z)-3-(5-methoxy-6,7-dihydro-1H-indol-3-yl)but-2-enal N-[(1R)-2,3-dihydro-1H-inden-1-yl]propanehydrazide 2-(5,6-dichloropyridin-3-yl)oxy-4-(trifluoromethyl)benzamide 6-[(2R,4S)-2-azido-1-fluorooctan-4-yl]oxyquinoline N-[(1S)-2,2-dimethylcyclopropyl]formamide;N-[[3-(6-ethoxypyridazin-4-yl)-5-fluorophenyl]methyl]cyclopropanecarboxamide 4-(azidomethyl)-N,1-dibenzylpiperidine-3-carboxamide 2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.3]hexane 2-[(3S)-1-[(1R)-cyclohexa-2,4-dien-1-yl]sulfonyl-7b-hydroxy-2,3a,5,6-tetrahydro-1H-pyrrolo[2,3-b]indol-3-yl]acetic acid 1-(3-ethylphenyl)-6-methoxynaphthalene 3-[5-(difluoromethyl)pyridine-2-carbonyl]-1H-pyrido[2,3-d]pyrimidine-4,7-dione 5-azido-4-tert-butyl-2-(trifluoromethyl)benzenethiol 1-chloro-4-(4-cyclopropylphenyl)benzene 5-(azidomethyl)-6,7-dihydropyrrolo[2,3-b]pyridine 5-phenylmethoxyquinazoline N-[3,5-bis(trifluoromethyl)phenyl]-1-propan-2-ylpiperidine-4-carboxamide (3E)-4-amino-3-[(2,3-dimethoxyphenyl)methylidene]azete-2-thione (6-ethyl-3-methylideneheptyl)benzene (6S)-7-acetyl-3-butylsulfanyl-6-(5-propan-2-ylthiophen-2-yl)-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-one 6-[3,5-bis(trifluoromethyl)phenyl]-3-(1H-pyrazol-4-yl)-8-[[4-(trifluoromethyl)piperidin-1-yl]methyl]pyrido[2,3-d]pyrimidin-4-one 1-[5-(furan-2-yl)-4,5-dihydro-1H-pyrazol-3-yl]indole (2R)-N-[5-chloro-4-(trifluoromethyl)pyridin-3-yl]-1-(2,6-difluorobenzoyl)piperidine-2-carboxamide 2-azido-4,6-dichlorobenzene-1,3-diamine 1-[(3,4-dimethoxyphenyl)methylamino]-3-[2-(dimethylamino)ethyl]urea 1-[2,6-diethoxy-4-[(E)-2-nitroethenyl]phenyl]pyrrolidine [[7-[[3-(chloromethyl)phenyl]methoxy]-2H-chromene-3-carbonyl]amino]carbamodithioic acid 2-(cyclohexylmethyl)-3,5,7,8-tetrahydrothiopyrano[4,3-d]pyrimidin-4-one 2-(cyclopropylmethoxy)-3-(4-fluorophenyl)sulfonylpropanamide 1-[(2R)-5-cyclopropylsulfonylspiro[2H-indole-3,4'-piperidine]-1'-yl]ethanone N-[(2,4-difluorophenyl)methyl]-5,6,7,8-tetrahydroquinazoline-8-carboxamide N-benzyl-2,2,4,4-tetramethylpentan-1-amine 1-(7,8-dihydronaphthalen-2-yloxy)-3-phenylpropan-2-ol N-[2-(5,6-dimethylcyclohexa-1,3-dien-1-yl)ethyl]-2-(3-phenyl-1H-pyrazol-5-yl)acetamide 1-cyclopenta-2,4-dien-1-ylethylbenzene;dichlorozirconium(2+) (E)-2-[(3R,5S)-7-chloro-5-phenyl-1,2,4,5-tetrahydro-3-benzazepine-3-carbonyl]hept-2-enamide 5-[(3R)-1-methylpiperidin-3-yl]oxy-6-quinolin-3-ylthieno[2,3-d]pyrimidine 4-[2-(oxan-4-ylmethylamino)quinoline-3-carboximidoyl]phenol (5E)-6-hydroxyimino-4,7-dimethyl-1H-quinoline-2-thione [2-(2-diazohydrazinyl)phenyl]methanol 3-chloro-N'-hydroxy-2-(4,5,6,7-tetrahydro-1H-indazol-3-ylsulfanyl)pyridine-4-carboximidamide (2S)-N,1-ditert-butyl-2,3-bis(4-chlorophenyl)cyclopropane-1-carboxamide 6-[(4S)-4-aminoazepan-1-yl]-5-[(2,3-difluorophenyl)methyl]-N'-hydrazinylpyridine-2-carboximidamide 4-[5-(3,4-dihydro-2H-quinoline-1-carboximidoyl)pyridin-2-yl]-N'-pyrrolidin-3-ylpiperazine-1-carboximidamide (2R)-3-[4-[(1R)-1-aminoethyl]pyridin-3-yl]-N-hydroxypropanamide 3-azido-N,N-diethyl-6-pyridin-2-ylpyridine-2-carboxamide 2,4-diamino-6-[(3,5-difluorophenyl)methyl]phenol 1-[(4aR,10aS)-9-chloro-10a-methyl-10H-phenanthren-2-ylidene]piperidin-4-amine 3-[3,5-dimethyl-4-[2-oxo-2-(2-piperidin-4-ylethoxy)ethoxy]phenyl]-1H-pyrrole-2-carboxylic acid 1-cyclopropyl-6-fluoro-7-[4-(2,3,4,5-tetrahydropyridin-6-yl)piperazin-1-yl]quinazoline-2,4-dione 2-(3,5-dimethylpyrazol-1-yl)-N-[(Z)-5-methylsulfanylpent-1-en-4-ynyl]acetamide N-[1,6-bis(2-methoxyethyl)-4-oxo-5H-pyrazolo[3,4-d]pyrimidin-7-yl]-2-(4-methylphenoxy)acetamide (Z)-1-[amino(methylsulfanyl)amino]-1-phenylprop-2-en-1-amine 2-chloro-N,N-bis(2-bromoethyl)aniline 2-(1,3-dioxoisoindol-4-yl)-2-[[4-ethoxy-3-hydroxy-5-(hydroxymethyl)phenyl]methylideneamino]acetonitrile 1-(2,4-dichlorophenyl)-6-fluoro-8-methyl-7H-pyrido[3,2-d]pyrimidine-2,4-dione 4-[(1S)-5-azidooxy-2,3-dihydro-1H-inden-1-yl]morpholine 6-(2,4-dimethoxyphenyl)-5-ethynylpyridine-3-carboxylic acid 2-[4-fluoro-1'-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl)spiro[2H-indole-3,3'-pyrrolidine]-1-yl]-N,N-dimethylacetamide 4-N-methyl-2-N,2-N-bis[4-(5-propan-2-yloxypent-1-ynyl)phenyl]pyrimidine-2,4-diamine 2-tert-butyl-6-[(6-chloropyrimidin-4-yl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one (4aS,8aR)-6-[3-(1H-indol-3-yl)propanoyl]-N-[2-methoxy-2-(oxan-4-yl)ethyl]-3,4,5,7,8,8a-hexahydro-1H-2,6-naphthyridine-4a-carboxamide;hydrochloride N'-(benzenecarboximidoyl)-1,3,5-trimethylpyrazole-4-carboximidamide (E)-2,3-diaminoprop-1-en-1-ol;8-[4-(cyclobutylmethoxy)phenyl]-6-N-ethyl-5-(methylideneamino)-4,9-dihydropyrimido[4,5-c]azocine-2,6-diamine 6-[5-(4-butoxy-3,5-dimethylphenyl)furan-2-yl]hexanoic acid 4-N,6-bis(benzenesulfonyl)-1H-pyrazolo[3,4-d]pyrimidine-4,5,7-triamine 2-[4-[2-(1H-indazole-3-carbonylamino)ethyl]phenyl]sulfanylacetic acid [4-(5,6,7,8-tetrahydropyrido[3,2-d]pyrimidin-4-yl)piperazin-1-yl]-(5H-pyrrolo[3,2-b]pyridin-2-yl)methanone 7-tert-butylpyrido[2,3-b]pyrazine 2-chloro-3-(3,5-difluorophenyl)-1H-indole 1-[(2R,3S)-2,3-bis(4-methoxyphenyl)-5-oxopyrrolidin-1-yl]-5-methylpyrazole-4-carboxylic acid 4-[4-(4,5-diphenyl-1H-imidazol-2-yl)pyridin-2-yl]pyridine 1-[(2S,4R)-4-benzylsulfanylpyrrolidine-2-carbonyl]-N-methoxyazetidine-3-carboxamide 1-amino-3-[1-(2,4-dichlorophenyl)ethyl]thiourea 6-(4-methylphenyl)sulfonyloxynaphthalene-2-carboxylic acid 2-[azido(methylsulfanyl)methyl]-5,8-dichlorochromen-4-one 1-(2-fluorophenyl)-3-[5-methyl-4-[(E)-prop-1-enyl]cyclohepta-1,3,6-trien-1-yl]-1,3-diazinan-2-one 2-[3-methyl-N-(2-oxopropyl)anilino]decanoic acid 1-(3,4-dimethoxyphenyl)-4-fluoropiperidine;ethane (5S,7R)-5-phenyl-7-[4-(trifluoromethoxy)phenyl]-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine N-[1-(4-fluoro-3,5-dimethylphenyl)ethyl]-6-(4-hydroxybutylamino)pyrimidine-4-carboxamide 6-[(3-fluorophenoxy)methyl]cyclohexa-2,4-dien-1-one 4-[5-(diethylamino)-2-(1,3,4-oxadiazol-2-yl)pyrimidin-4-yl]oxybenzoic acid 3-(1,1-difluoroethyl)-N'-hydroxypyridine-2-carboximidamide (3S)-3,4-dimethyl-N'-[2-methylsulfonyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazine-1-carboximidamide [(1S,3R)-4,6-diphenyl-2,3-dihydro-1H-inden-1-yl]urea (5S,7R)-2-ethylsulfanyl-N-[(4-methoxyphenyl)methyl]-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 2-[4-(cyclohexylmethoxy)-3,5-dimethoxyphenyl]benzo[g][1,3]benzothiazole N'-[4-(2-phenylhydrazinyl)butyl]ethane-1,2-diamine;hydrobromide 5-bromo-4-[2-methoxyethyl(propanoyl)amino]-1H-pyrimidin-6-one N-[2-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]but-2-ynamide 4-tert-butyl-2-[(6-morpholin-4-ylpyridin-3-yl)methyl]piperazine-1-carboxylic acid 3-[2-[(1R,3S)-3-methylcyclohexyl]oxyphenyl]-5-pyridin-4-yl-1H-imidazo[4,5-b]pyrazin-2-one 2-azidooxy-6-[1-(methylamino)ethyl]phenol 3,5-dichloro-4-phenylmethoxybenzoic acid 2-[(3,5-dichlorophenyl)sulfonylamino]-4-hydroxybutanoic acid 1-cyclohexa-2,4-dien-1-ylpropan-1-amine;(3R)-5-[(3-propoxyphenyl)methoxy]pent-1-yn-3-ol 2-chloro-1,3-difluorobenzene;N-cyclohexyl-5-methoxy-2,3,4a,6,7,8,9,10,11,11a-decahydrobenzo[b]fluoren-1-amine 6-chloro-4-N-(2,2-dimethoxyethyl)-2-N,4-N-dimethylpyrimidine-2,4-diamine 5-chloro-N-(4,6-dimethylpyridin-2-yl)sulfonyl-1-benzofuran-2-carboxamide 2-[1,3-dioxo-5-(2,4,6-triiodophenyl)isoindol-2-yl]acetic acid 5-(2-cyclobutylpyrazole-3-carbonyl)-N,4,6,7-tetrahydropyrazolo[1,5-a]pyrazine-3-carboxamide 2-[(4-methyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)amino]ethanol 2-[(4R,5S)-4,5-dihydroxy-6-oxooxan-3-yl]oxybenzonitrile 2-[3,5-bis(trifluoromethyl)anilino]-6,7-dihydro-1H-pyrrolo[2,3-d]pyrimidine-4-thione 4-(aminomethyl)-6-chloro-3-cyclopentylsulfanylpyridine-2,5-dicarbonitrile [4-(2-aminophenyl)sulfonylpiperazin-1-yl]-[5-methyl-6-(quinolin-3-ylamino)pyridin-3-yl]methanone (4R)-1,4-dimethyl-N-[6-(trifluoromethylsulfanyl)pyridin-2-yl]pyrrolidine-3-carboxamide 5-bromo-2,4-dichloro-N-[(E)-1-(3,5-dinitrophenyl)ethylideneamino]aniline (2E)-2-[[3-cyano-6-cyclopropyl-5-ethoxy-4-(2,4,4-trimethylpentan-2-ylamino)pyridine-2-carbonyl]-propylhydrazinylidene]acetic acid (3S,4R)-1-[3-amino-6-(3-methoxyphenyl)pyrazine-2-carbonyl]-4-hydroxypyrrolidine-3-carbonitrile N-(1H-indol-4-ylsulfonyl)-2,3-dihydro-1-benzofuran-7-sulfonamide 1,2-diamino-4-[3-[(5-fluoropyridin-2-yl)methoxy]phenyl]-6-oxopyridine-3,5-dicarbonitrile N-[5-methyl-4-(2-phenoxyanilino)pyrimidin-2-yl]-3,7-diazabicyclo[3.3.1]nonane-3-carboxamide 2-[4-hydroxybutyl(1,3-thiazol-5-yl)amino]acetonitrile (4-chlorophenyl)sulfanylcarbamodithioate;nickel(2+) 2-[4,6-bis(sulfanyl)triazin-5-ylidene]propanedinitrile 4-(1H-indazole-6-carbonyl)-3,5-dimethylpiperazin-2-one 4-(2,3-dihydro-1H-inden-5-yloxymethyl)pyridine N-[(3R,4S)-1-benzyl-3-hydroxypiperidin-4-yl]-2-pyridin-3-ylacetamide;hydrochloride 2-(4-aminophenyl)-6-[(5,8-difluoronaphthalen-1-yl)methyl]pyrimidine-4-carboxamide 2,4-dinitro-N-(2-propanoylimino-1H-pyrimidine-6-carbonyl)benzenesulfonamide 4-(2,5-dioxoimidazolidin-1-yl)-N-[(2-fluorophenyl)methyl]butanamide 1-(2,4-difluorophenyl)sulfonyl-N-[5-(2-methoxypyrimidin-5-yl)pyridin-2-yl]piperidine-4-carboxamide 4-bromo-3-methyl-N'-[2-oxo-2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]benzohydrazide (3-ethoxycarbonylphenyl)methylcarbamic acid N-benzylspiro[1H-indole-3,4'-piperidine]-2-imine 1-[4-fluoro-3-(trifluoromethyl)phenyl]-4-[5-(trifluoromethyl)pyridin-2-yl]piperidine-4-carboxamide 2-(7,8-dihydroisoquinolin-6-yl)-N-methanimidoyl-N-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]pyrimidine-5-carboximidamide 3-(1,4-dioxaspiro[4.5]decan-8-ylmethoxy)benzenecarbothioamide 2-methyl-4-[(3R)-3-(3-oxocyclopenten-1-yl)oxypyrrolidin-1-yl]benzonitrile 5-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-ethyl-4-[3-fluoro-5-[[4-methyl-4-(4-methylpiperazin-1-yl)cyclohexa-1,5-dien-1-yl]amino]pyridin-2-yl]-1,2,4-triazole-3-carboxamide 5-bromo-4,8-dihydrothieno[3,2-c]quinoline 3-[4-(3-hydroxyphenyl)butyl]benzenecarboximidamide N-[4-(7,8-dihydronaphthalene-2-carbonylamino)phenyl]pyridine-3-carboxamide 3-[2-(1,4-dioxin-2-yl)ethynyl]pyran-4-one 7-[[(1S,3R)-3-aminocyclopentyl]methyl]-4-fluoroisoquinolin-5-amine 2-methyl-5,6-dinitrobenzimidazole N-[(2S)-1-oxo-1-[[3-phenylmethoxy-4-[(3,4,5-trimethoxybenzoyl)amino]butan-2-yl]amino]pentan-2-yl]morpholine-4-carboxamide 4-[(6R)-7-[3-[cyclopropanecarbonyl-(2,6-dichlorobenzoyl)amino]propanoylamino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-2-yl]benzoic acid (1S)-1-[5-cyclobutyloxy-2-fluoro-4-(1,3-oxazol-5-ylamino)sulfanylphenyl]ethanethiol 1-[2,4-bis(trifluoromethyl)phenyl]-6-cyclopropyl-5H-pyrazolo[3,4-d]pyrimidin-4-one N-(4,5-dimethyl-2-phenyldiazenylphenyl)-4-nitro-N-octylbenzamide 4-methoxy-2-phenyl-N'-[4-(2-piperidin-1-ylethoxy)quinolin-8-yl]benzenecarboximidamide 2-amino-3-phenyldiazenylnaphthalene-1,4,7-trione 4-[2-amino-6-[5-(2,6-difluorophenyl)-1H-imidazol-4-yl]pyridin-3-yl]cyclohexan-1-ol 2-(3,5-difluorophenyl)-4H-pyrido[1,2-a]pyrimidine (6R)-8-oxo-3-propanoylsulfanyl-7-[[2-[2-(trifluoromethyl)phenyl]acetyl]amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid N-[5-fluoro-4-(2,4,5-trichlorophenoxy)pyrimidin-1-ium-2-yl]-2-methyl-3H-benzimidazol-5-amine 2-[2,4-difluoro-N-(3-methylbut-2-enyl)anilino]-1-phenylethanone [4-(3,5-difluorophenoxy)phenyl]-[4-(1H-imidazole-2-carbonylamino)phenyl]sulfanium 2-[4-(4-methoxy-1H-triazin-2-yl)phenoxy]acetic acid 4-[(2-fluoro-6-methoxyphenyl)methylamino]-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione N'-methanimidoyl-4-(propylsulfanylamino)benzenecarboximidamide 2-(aminomethyl)butanal;5-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-3-[6-[4-[(4-ethylpiperazin-1-yl)methyl]anilino]pyridin-2-yl]-1H-indole-7-carboxamide 2,3-bis(ethenyl)naphthalene (1R)-5,7-dimethoxy-2-[[4-[2-methyl-3-[2-methyl-6-(trifluoromethyl)phenyl]anilino]piperidin-1-yl]methyl]-1-pyridin-2-ylpentan-1-ol (4-azidooxyphenyl)methylphosphonic acid [4-methylsulfonyl-3-(trifluoromethoxy)phenyl]-[3-[[6-(triazol-2-yl)pyrazolo[1,5-a]pyridin-2-yl]amino]piperidin-1-yl]methanone 2-[4-(azidooxymethyl)piperidin-1-yl]-N,N-diethylpyrimidin-5-amine 2-azido-5-methylsulfonylbenzamide 1-[2-(2,4-difluorophenyl)ethyl]-4-oxo-3-pyridin-2-ylmethoxypyridine-2-carboxylic acid N-[1,1-di(butanoyloxy)propyl]-4-(1H-indol-3-yl)butanamide 4-hydroxy-1,3-bis(4-methoxyphenyl)-2H-benzo[f]isoindole-5,8-dione 5-[2-(2-chlorophenyl)pyrrolidine-1-carbonyl]-N,N-dimethylpyridine-3-sulfonamide 1-(2,5-diaminophenyl)propan-2-one N-[(2S)-1-cyclohexyloxypropan-2-yl]-3,4-dihydro-2H-chromene-6-sulfonamide 2-(4-propanoylphenyl)sulfinylcyclopentane-1,3-dione 5-[4-(N'-tert-butylcarbamimidoyl)phenyl]-2,3-dimethylbenzenesulfonamide (2S)-1-[4-[4-amino-3-(cyclopropylmethoxyiminomethyl)phenyl]piperidin-1-yl]-2,5-dihydroxypentan-1-one 2-(hydroxymethyl)but-3-enal;methanol;[(3R)-oxolan-3-yl]methoxymethylbenzene (1S,2R)-4-[2-hydroxy-3-[6-(oxolan-3-yloxy)pyridin-3-yl]propanoyl]cyclopentane-1,2,3-tricarbonitrile 2-[(2,3-dihydroxyphenyl)methylideneamino]pentanoic acid 2-[(4Z,6E)-5-fluorononaa-1,4,6-trien-3-yl]-N'-hydroxypyridine-4-carboximidamide 1-[5-methyl-2-(3,4,5-trifluorophenyl)-1H-imidazole-4-carbonyl]pyrrolidine-2-carboxamide 3-amino-N'-(4,5-dihydro-1H-imidazol-2-yl)pyrazine-2-carboximidamide 1-(3,4-dihydroxyphenyl)-2-[2-(3-morpholin-4-ylpropoxyiminomethyl)phenyl]ethanone 4-fluoro-2-[3-[(5-fluoro-2-methylphenyl)methoxy]pyridin-1-ium-2-yl]benzaldehyde 4-(2-fluoro-5,6,7,8-tetrahydroquinazolin-4-yl)piperazine-1-carboxylate 4-[2-(3,4-difluorophenyl)morpholine-4-carbonyl]-N,N-dimethylbenzenesulfonamide 2-[4-methyl-6-oxo-2-(1H-pyrrol-3-yl)-1H-pyrimidin-5-yl]acetic acid 4-[(3R)-3-[(1,5-dimethylpyrazol-4-yl)methylamino]pyrrolidin-1-yl]pyrimidine-2-carboxamide 5-(3,4-dihydropyridin-2-yl)-N-[[4-fluoro-2-(trifluoromethoxy)phenyl]methyl]pyridine-3-carboxamide 1,5-dimethyl-4-[(E)-pent-3-enoxy]benzene 3-(2,3-dimethoxybenzoyl)-4-hydroxychromen-2-one 1-benzyl-4-(3,5-dimethoxyphenyl)piperazine (2-benzyl-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-1-yl)-pyridin-3-ylmethanone 4-chloro-2,5-dimethylbenzenesulfonic acid 2,4-ditert-butyl-6-[(E)-[[5-(diethylamino)naphthalen-1-yl]hydrazinylidene]methyl]phenol N-[(1E,3Z)-2-methylpenta-1,3-dienoxy]-5-phenylpentanamide 2-[5-bromo-4-[(E)-[2-(3-chloro-2-methylphenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]-2-ethoxyphenoxy]propanoic acid 4-[2,5-difluoro-3-(trifluoromethyl)phenyl]-1H-tetrazol-5-one 4-[2-(2,6-dimethylphenyl)imidazo[1,2-a]pyrimidin-7-yl]morpholine (4R)-1-(2,6-dichlorophenyl)-6-methyl-3-pentyl-4-phenyl-5H-pyrazolo[3,4-d]pyrimidin-7-one 2-azidooxy-6,7-dibromoquinazoline (2-azidopyridin-3-yl)-(2,3-dihydro-1H-isoindol-5-ylamino)methanol 4-bromo-2-chloro-6,8-difluoroisoquinolin-1-one 3-[5-bromo-1-(2,4-difluorophenyl)sulfonyl-4-methoxycyclohexa-2,4-dien-1-yl]-N-fluorosulfonylpropanamide 4-[2,5-dimethyl-4-(3-oxo-1H-isoindol-2-yl)cyclohexa-2,4-dien-1-ylidene]butanoic acid 4-[4-(4,4-dimethylpiperidin-1-yl)-5-(1H-indazol-7-ylamino)pyrido[3,2-d]pyrimidin-8-yl]cyclohexane-1-carboxylic acid (2R)-2-[4-amino-3,5,6,7,8,9-hexahydropyrido[2,3-d]azepine-2-carbonyl]pyrrolidine-1-carbonitrile 4-(3,5-dimethylpyrazol-1-yl)-2-fluoro-6-(trifluoromethoxy)benzamide 2-[[(1R,3S)-3-azidocyclohexyl]methoxymethyl]naphthalene 1-(5,6-dimethyl-2-pyridin-3-ylpyrimidin-4-yl)ethanone N-[(1R,2S)-4-(imidazol-1-ylmethyl)-2-propoxycyclopentyl]oxane-4-carboxamide (7R)-N-(4-chlorophenyl)-5-methyl-7-[2-(3,4,5-trifluorophenoxy)acetyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide N-[1-(3,4-dimethoxyphenyl)ethyl]-5-propylpyridine-2-carboxamide 2-(3,4-dimethoxyphenyl)-N-(1H-imidazol-5-ylmethylideneamino)-2,8-diazaspiro[4.5]decan-3-imine;dihydrochloride 3-(4-azido-2-butoxyphenoxy)propane-1,1,2-triol 4-(1,3-benzodioxol-5-yl)-N-[1-[2-[[ethyl(methyl)amino]methyl]phenyl]ethenyl]aniline 7-(2,4-dimethoxyphenyl)-N-[3-(oxolan-3-ylamino)propyl]quinoxalin-5-amine [4-(azidomethyl)piperidin-1-yl]-[3,5-bis(trifluoromethoxy)phenyl]methanone N-[1-[2-(3,5-dimethylphenoxy)acetyl]azetidin-3-yl]-N-(2-morpholin-4-ylethyl)cyclopentanecarboxamide 6-tert-butyl-8-ethenyl-N,2,5,9,11-pentazatetracyclo[10.4.0.02,7.08,10]hexadeca-1(12),3,6,13,15-pentaene-5-carboxamide [2-(dimethylamino)-6,7,8,9-tetrahydro-5H-pyrido[3,4-b]azepin-4-yl]-(1,7,11-triazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-12-yl)methanone;dihydrochloride 4-(azidomethyl)-2-bromo-N-[(3,5-dimethoxyphenyl)methyl]aniline 7-amino-5-(4-cyanophenyl)-2,3-dihydro-1H-1,4-benzodiazepine-8-carboxylic acid 2,3-dihydrofuro[3,4-b][1,4]oxazin-5-yl-[6-(2H-pyridin-2-id-3-yl)-3-azabicyclo[3.1.0]hexan-3-yl]methanone;yttrium 4-(difluoromethyl)-3,5-diiodothiophene 4-(1H-benzimidazol-2-yl)-3-ethylsulfonylphenol (2-cyclobutylpyrazol-3-yl)-[4-methoxycarbonyl-1-(oxan-4-ylmethyl)piperidin-4-yl]carbamic acid 2-(1-azidocyclopentyl)phenol 4-ethoxy-N'-[(Z)-1H-indol-3-ylmethylideneamino]benzenecarboximidamide 3-[2-[4-(5,6-dihydronaphthalen-1-yl)piperidine-1-carbonyl]-4-oxo-4a,9a-dihydro-5H-1,10-phenanthrolin-9-ium-3-ylidene]azetidine-1-carboxylic acid 6-[(2Z,4E)-5-aminohepta-2,4,6-trienyl]-N-[(3S,4R)-1-[2-[1-(dimethylsulfamoyl)ethylideneamino]ethoxy]-4-hydroxypiperidin-3-yl]naphthalene-2-carboxamide 2-[(6,6-dioxo-1,4,5,7-tetrahydrothiopyrano[3,4-c]pyrazol-3-yl)sulfanylamino]-N-propan-2-ylacetamide N-[4-(3-amino-1,2-oxazol-5-yl)pyridin-2-yl]cyclobutanecarboxamide;hydrochloride 2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-N'-hydroxypyrimidine-4-carboximidamide 1-[2,3-dihydroxypropyl(ethenylsulfonyl)amino]-4a,9a-dihydroanthracene-9,10-dione N-[2-(3,5-dichlorophenyl)-2-morpholin-4-ylethyl]-2-oxopiperidine-3-carboxamide N-[2-(1H-benzimidazol-2-yl)ethyl]-3,5-dimethoxycyclohexa-2,4-dien-1-imine 5-(1H-benzimidazol-2-yl)imidazolidine-2,4-dione 6-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-1-phenyl-5H-pyrazolo[3,4-d]pyrimidin-4-one [2-(3-methoxyphenyl)pyrrolidin-1-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)methanone;dihydrochloride (2Z,4E)-3-ethylsulfonyl-2-[5-methoxycarbonyl-6-oxo-1-(1H-pyrazol-4-yl)pyridazin-4-ylidene]-3-methyl-5-sulfanylpentanenitrilium 4-(1,3-benzodioxol-5-ylmethoxy)-2H-chromene-3-carbonitrile 2-[4-(5-azido-2,6-dimethylpyrimidin-4-yl)piperazin-1-yl]ethanol (7R)-3-methyl-5-oxo-N-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide (3R)-1',2'-diaminospiro[2H-indene-3,5'-imidazolidine]-4'-one 2-(1,4-dimethylpyrrol-3-yl)-5,6-dihydrothieno[2,3-d]pyrimidine N-[4-[(5-methylpyrazine-2-carbonyl)amino]phenyl]quinoline-2-carboxamide 3,4-dimethoxy-N-(3-oxo-2-propan-2-ylspiro[5.5]undecan-9-ylidene)benzamide 4-[2,6-dichloro-N-(4-methoxybutyl)-4-nitroanilino]butan-1-ol 1-[5-(cyclopentylmethyl)-3,4-dihydro-2H-quinoline-1-carbonyl]piperidine-3-carboxylic acid 5-[3-(3,4,6,7,8,9-hexahydrobenzo[f][2]benzazepine-11-carbonyl)pyridin-1-ium-1-yl]-2-[[(E)-prop-1-enoxy]methyl]benzonitrile (2E)-2-[(Z)-5,6-dimethylidenehept-4-enylidene]-3H-1-benzofuran-6-ol 2,4-dichloro-5-fluoroquinoline 1-[4-(dimethylamino)phenyl]pyrrole-2,5-dione ethane;N-methylformamide;6-methylidene-1,3-di(propan-2-yl)quinoline 2-[4-methyl-3-(trifluoromethyl)phenyl]benzotriazole N-[3-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-3H-benzimidazol-5-yl]cyclobutanecarboxamide;ethane N-[(1S)-2,3-dihydro-1H-inden-1-yl]-7-methoxy-6,11-dioxo-5H-benzo[b][1,4]benzothiazepine-9-carboxamide 1-[5,6-dihydroxy-9,10-bis(4-hydroxyphenyl)anthracen-2-yl]oxyethanol 2-(5-chlorobenzimidazol-1-yl)cyclopentan-1-ol ethane;6-[2-(4-hexyl-3,5-dimethoxyphenyl)phenoxy]hexan-1-ol 5-(2,4-difluorophenyl)-1-[(Z)-3,7-dimethyloct-5-enoyl]pyrrolidine-2-carboxylic acid [4-(2,6-diphenylpyrimidin-4-yl)piperazin-1-yl]-[(3R,4S)-4-methoxypyrrolidin-3-yl]methanone;formic acid 1-[(5S)-3-tert-butyl-2,4,6-trioxo-1,3-diazinan-5-yl]-1-[4-[4-(trifluoromethyl)phenoxy]phenyl]urea N-[(1R,2S)-6-bromo-2-ethyl-3-oxo-1,4-dihydronaphthalen-1-yl]carbamate 2-(2,3-difluoro-4-propoxyphenyl)-6-[4-(trifluoromethyl)cyclohexyl]-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene N-[2,5-bis(trifluoromethyl)phenyl]sulfonyl-1-[[4-fluoro-3-(trifluoromethoxy)phenyl]methyl]-1,2,4-triazole-3-carboxamide 3-ethylsulfanyl-6,7-dimethoxy-1H-quinoline-2,4-dione N-azido-6-(2,3-dimethoxyphenyl)pyrido[3,4-d]pyrimidin-8-amine 2-fluoro-4-[(1R,5S)-3-methylsulfonyl-6-azabicyclo[3.2.0]heptan-6-yl]benzoic acid 2-[N-(2,3-dihydroxypropyl)-4,5-dimethyl-2-phenyldiazenylanilino]acetic acid 2-[8-chloro-1-(3,3-difluorocyclobutyl)imidazo[4,5-c]quinolin-7-yl]propan-2-ol 3-[8-amino-1-(2,6-difluorophenyl)imidazo[1,5-a]pyrazin-3-yl]cyclohexane-1-carboxylic acid 2-[(1S)-6-bromo-4,5,7-trifluoro-3-oxo-1H-isoindol-2-yl]acetic acid (E,3S)-N-hydroxy-3-[4-[2-(2,5,6-trimethylbenzimidazol-1-yl)ethylamino]phenyl]but-2-enamide 3-cyclohexyloxy-1H-1,2,4-triazol-5-amine 1-chloro-2,4-difluorobenzene;1-methoxypropane 5-(aminomethyl)-N-[[6-chloro-2-(4,5-dihydro-1H-pyrazol-3-yl)pyridin-4-yl]methyl]-1,3,4-thiadiazol-2-amine;ethane 1-chloro-4,5,10-trimethoxynaphtho[2,3-f]indazole-7,12-dione (4R)-4-[3,5-bis(trifluoromethyl)phenyl]-1,2,4-triazolidine 2-(4,7-dioxo-3H-imidazo[5,1-f][1,2,4]triazin-2-yl)-N-phenylacetamide 4-azidooxy-3,5-dichlorobenzoic acid 7-chloro-5-[(2R)-4-ethylazepan-1-yl]-3H-pyrido[2,3-d]pyrimidin-4-one [5-[5-[4-(2,3-dihydropyridin-5-yl)-6-phenyl-1,3,5-triazin-2-yl]naphthalen-1-yl]-2-methylpyrazol-3-ylidene]hydrazine (4Z)-2-methyl-3,5-bis[(4-phenylmethoxyphenyl)methyl]hepta-4,6-dien-1-ol N-[(3-ethyloxan-4-yl)methyl]-6-iodothieno[2,3-b]pyridine-5-carboxamide 5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid (4R)-2-amino-N'-(1,3-benzothiazol-6-ylmethyl)-4-(3,4-dichlorophenyl)-5-methoxypentanimidamide 4-[3,5-bis(trifluoromethyl)anilino]piperidine-1-carboxylate 2-azido-6,7-dimethoxy-1,3,4,9-tetrahydropyrido[3,4-b]indole 4-chloro-6-(difluoromethyl)-3-ethynylpyridazine 1-(2,3-dihydro-1H-inden-5-yl)-N-[(5,6-dimethylpyridin-3-yl)methoxy]ethanimine 2-(dibutylamino)-3,4-di(cyclooctyl)phenol N-[2,3-difluoro-4-(6-propoxypyridin-1-ium-3-yl)phenyl]-1H-indole-5-carboxamide 2-[1,3-dioxo-2-(propan-2-ylamino)isoindol-4-yl]-3H-isoindol-1-one 2-[4-(3,6-dimethylpyridin-2-yl)piperazin-1-ium-1-ylidene]acetaldehyde (5-fluoropyridin-2-yl)-[4-(1H-pyrazol-5-ylmethyl)piperazin-1-yl]methanone N-ethyl-3-[6-methyl-5-oxo-7-(4-piperidin-1-ylbut-1-ynyl)imidazo[1,2-a]imidazol-3-yl]benzamide 3-[6-(2,4-difluorophenyl)-1H-benzimidazol-2-yl]-N-propan-2-ylidenecyclohexane-1-carboxamide;1,3-oxazolidine 5-(6,7-dimethoxyquinolin-4-yl)oxypyridine-2-carboxylic acid 5-chloro-4-[1,2,3,6-tetradeuterio-7-fluoro-3-[1-(trideuteriomethyl)piperidin-4-ylidene]-5H-[1,4]dioxepino[6,5-b]pyridin-9-yl]pyridine-2-carbonitrile 2-(azidomethoxy)-3,5-dibromobenzoic acid (E)-4-[2,6-dichloro-4-(trifluoromethylsulfanyl)phenoxy]but-2-enoic acid 2-[5-(1,3-benzoxazol-2-ylmethoxy)-4-chloro-1H-indol-3-yl]acetate (6R)-5-phenylspiro[3H-1,3-thiazole-2,3'-indole]-2'-one N-(4-chlorobutyl)-2,6-difluoro-N-(1,3-thiazol-5-yl)aniline (1S)-N,N,4-triethyl-2-methoxycyclohexan-1-amine;hydrochloride 2-[[5,6-dimethyl-3-(trifluoromethyl)pyridazine-4-carbonyl]amino]-6-phenylbenzoic acid 3,5-dimethyl-4-propan-2-yloxybenzenesulfinate 4-[(E)-2-(3,5-difluorophenyl)ethenyl]-N'-methoxybenzenecarboximidamide;hydrochloride N-[6-(1,3-benzodioxol-5-yl)pyridazin-3-yl]-2-chloro-N-methylbenzamide 3,4-dimethoxy-N-[[(2S)-4-methylpyrrolidin-2-yl]methyl]benzamide 2-[N-acetyl-4-(dimethylamino)anilino]decanoic acid 1-(7,8-dihydronaphthalen-2-yl)piperidine N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-5-(1-methylpyrazol-4-yl)benzamide 2-chloro-3-[3,5-difluoro-6-[1-(4-hydroxyphenyl)ethyl]pyrazin-2-yl]-N'-methanimidoyl-4-propan-2-yloxybenzenecarboximidamide 3-amino-1-(5-methylthiophen-2-yl)sulfonylindole-2,4-dione 1-(3-aminopropoxy)-7-[(2E,4Z)-hexa-2,4-dien-3-yl]oxy-8,9,10,11-tetrahydrocycloocta[c]quinoline-6-carboxylic acid (5Z)-2-(3,4-dichlorophenyl)imino-5-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-1,3-thiazolidin-4-one 3-[2,6-dimethoxy-4-(3-nitrophenyl)phenyl]-1-hydroxypiperidine 2-(1,5-dimethylpyrazole-3-carbonyl)cyclopropane-1-carboxylic acid 2-(4-hydroxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 6-benzyl-7-oxo-5,8-diazaspiro[3.4]octane-2-carboxylic acid 1-(3,4-dichlorophenyl)-2,3,6,7-tetramethylimidazo[4,5-b]pyridin-1-ium ethane;1-methoxybutylbenzene;2-[4-[(3E,5Z)-3-(trifluoromethylsulfonylmethylidene)octa-1,5,7-trien-4-yl]phenyl]acetaldehyde 3-[(1R)-1-(4,5-dimethyl-2H-pyridin-1-yl)ethyl]aniline 1-[3-fluoro-4-(2,3,6-trimethylpyridin-4-yl)oxyphenyl]-2-(6-oxopiperidin-3-yl)guanidine 4-[[[(2S)-1,4-dioxan-2-yl]methylamino]methyl]benzamide 2-[4-(ethylamino)piperidine-1-carbonyl]-6,7-dimethyl-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one 1-(3-chloro-2-fluorophenyl)-5-methylpyrrolidine N-[2,6-di(propan-2-yl)phenyl]-3,4-bis(pyridin-2-ylmethoxymethyl)aniline 2-cyclopropyl-1'-(6,7-dihydro-5H-pyrrolo[3,4-b]pyridine-1-carbonyl)spiro[5,6-dihydro-3H-cyclopenta[d]pyrimidine-7,3'-piperidine]-4-one 3-methyl-4-[(5E)-6-[(Z)-2,7,8-trimethylnon-5-en-5-ylidene]cyclohexa-1,3-diene-1-carbonyl]benzamide 2-azido-4,5-diphenyl-3H-1,2-oxazole 2-methylsulfonylethyl-[5-(trifluoromethyl)pyrimidin-4-yl]azanium 5-[4-chloro-3-(trifluoromethyl)phenyl]-2-[[5-methoxy-6-(trifluoromethyl)pyridin-3-yl]methyl]-1,3-dioxane-5-carboxylic acid (5-bromo-1H-indol-2-yl)-(3,4-dimethoxyphenyl)methanone N-[(2R,3S)-1-methyl-5-oxo-2-pyridin-4-ylpyrrolidin-3-yl]butanamide 1-(2,4-diethylphenyl)-N'-[2-(3-methoxy-2H-pyridin-3-id-6-yl)-2-oxoethyl]cyclopropane-1-carbohydrazide;uranium(2+) 4-(8-bromo-2,3-dihydro-1H-pyrrolo[1,2-a]indole-5-carbonyl)-N'-hydroxybenzenecarboximidamide 4-chloro-N-ethyl-N-methylaniline;(3Z)-3-[(5-fluoro-2-formamidophenyl)-(methylideneamino)methylidene]-1,2-dihydropyrrole-5-carboxamide N-[(2S)-5-hydroxypentan-2-yl]-4-methoxy-3-(2-oxo-1,4-dihydroquinazolin-3-yl)benzamide 2-[4-bromobutan-2-yl(propanoyl)amino]benzenesulfonic acid 1-(3-nitro-5-thiophen-2-ylthiophen-2-yl)ethanone 2-[(4-oxo-1-phenyl-5H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-(4-phenoxyphenyl)acetamide 4-(1H-indol-2-yl)benzene-1,3-diol 3-[2-(4-chlorophenyl)ethyl]-1H-indole 4-[4-hydroxybutyl(2H-tetrazol-5-yl)amino]benzenesulfonic acid 5-[4-amino-6-(4-methylpiperidin-1-yl)pyrimidine-5-carboximidoyl]-3H-indol-2-amine 3-[3-(2,4-dichlorophenyl)propanoyl]-1-hydroxyindole-6-carboxylate (2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-1-(6-methoxypyridine-3-carbonyl)pyrrolidine-2-carboxamide 2-[2,6-di(propan-2-yl)phenyl]-N-[1-methyl-5-(methylaminosulfanyl)pyrazol-4-yl]imidazo[1,2-a]pyridin-7-amine N-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-methylpyrimidine-4-carboxamide 2-[(4R)-1,4-dimethyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]thiophene-3-carbonitrile 7-hydroxy-8,8-dimethyl-4-(3,4,5-trimethoxyphenyl)pyrano[4,3-h]chromene-2,9-dione 2-methyl-3-phenyl-5-[4-(2-pyridin-2-ylphenyl)buta-1,3-dienyl]-2H-benzimidazole N-(2,6-dichloropyrimidin-4-yl)nitramide (Z)-2,4-dimethyl-3-methylidenehept-1-ene;ethane;8-[(E)-5,6,7,11-tetrahydrobenzo[d][1]benzazocin-12-yl]-9H-carbazole 2-[3,4-dihydroxy-6-(3-oxocyclohexen-1-yl)oxan-2-yl]benzoic acid [[3-[4-(dimethylamino)piperidin-1-yl]benzoyl]amino]thiourea 2-tert-butyl-4-[2,6-dimethoxy-5-[(3R)-3-methylpiperazine-1-carbonyl]pyrimidin-4-yl]piperidine-1-carboxylate 2-[(3,5-dichloropyridin-4-yl)carbamoylamino]acetic acid (4-aminophenyl)-[4-[2-[(5S)-5,7-dimethyl-4-oxo-6,8-dihydrofuro[3,2-c]azepine-5-carbonyl]pyridin-4-yl]oxy-3-fluorophenyl]carbamic acid 2-[3,4-dichloro-5-(1H-pyrrol-2-yl)pyridin-2-yl]-1-ethoxypropan-2-ol 2-methylsulfanyl-4-[5-(trifluoromethoxy)indol-1-yl]pyridine-3-carboxylic acid 5-chloro-2-(chloromethyl)-3,4-difluorobenzaldehyde 4-(6,8-dibromo-3-methylimidazo[1,2-a]pyridin-2-yl)benzoic acid 1-(2,4,5-trichlorophenyl)propan-1-one 2-[5-(azidomethyl)thiophen-3-yl]pyrazine N-[2-(dimethylamino)ethyl]-4-fluoro-3-[1',7'-dioxospiro[3H-furo[3,4-b]pyridine-1,4'-5,6-dihydro-1,3-benzothiaze]-6-yl]benzamide 3-[[1-[4-(trifluoromethyl)phenyl]benzimidazole-2-carbonyl]amino]benzamide 3-[5-[3,4-bis(ethenyl)cyclohexa-2,4-dien-1-ylidene]piperidin-3-yl]oxypyridine 1-[4-(2,6-difluorophenyl)piperazin-1-yl]propan-2-ol;uranium (4R)-6,6-dimethyl-8-phenylmethoxy-N-[(1S)-1-pyridin-2-ylethyl]-4H-imidazo[5,1-d][1,2,3,5]tetrazin-7-imine 5-(2,3-dihydrofuran-4-yl)-N-[4-(trifluoromethylsulfanylamino)butyl]pyridine-3-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]-2-(cyclohepta-1,4,6-trien-1-yloxyamino)ethanone 6-chloro-N-[(2,4-dimethoxyphenyl)methyl]-4H-1,3-benzoxazin-8-amine 3-(4-cyanophenyl)-N-[(Z)-4,5-difluorohex-2-enyl]propanamide N-[1-(4-methylcyclohexanecarbonyl)piperidin-3-yl]-2,3-dihydrofuro[2,3-b]pyridine-5-carboxamide N-[3-[[4-(methylamino)cyclohexyl]methoxy]phenyl]methanesulfonamide 2-[(2S)-4-bromobutan-2-yl]sulfanyl-5-methoxybenzenecarboximidamide 1-[4-(6-cyclopropylpyridine-2-carbonyl)piperazin-1-yl]-2,3,3a,5,6,7,7a-octahydropyrazolo[3,4-b]pyridin-4-one 5-(diethylaminomethyl)-N,6,7-trimethoxynaphthalene-2-carboxamide 2-[2-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethoxy]-1-[2-[2-methanimidoyl-5-(propylamino)anilino]pyrimidin-5-yl]butan-1-one N-(2,4-difluorophenyl)-2-[methyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]propanamide (5Z)-2-(4-bromophenyl)imino-5-[(3-ethoxy-4-hydroxy-5-iodophenyl)methylidene]-1,3-thiazolidin-4-one 2-hydroxy-N,3-dimethyl-5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)benzamide 4-[3-(benzenesulfonyl)propanoylamino]-2,5-dichlorobenzoic acid N-[(4S)-5,6-dihydro-1H-benzimidazol-2-yl]-9-methoxy-8-(3-methylbutyl)-5-oxospiro[3.5]nonane-7-carboxamide N-(4-chlorophenyl)-N'-[3-(1H-pyrrolo[2,3-b]pyridin-3-yl)prop-1-en-2-yl]ethane-1,2-diamine 3-[[2,4-bis(phenylmethoxy)benzoyl]amino]-3H-thiophene-2-carboxylic acid 1-azido-2,4,5-trifluoro-3,6-di(propan-2-yl)benzene 2-[4-bromobutan-2-yl-(8-chloro-6,11b-dihydro-5aH-chromeno[3,4-d]pyrimidin-4-ylidene)amino]ethanol 2-[5-(trifluoromethyl)pyridine-3-carbonyl]-8-oxa-2-azaspiro[4.5]decan-1-one 6-chloro-2-[4-(1,3-dioxolan-2-yl)phenyl]-7-fluoroimidazo[1,2-a]pyridine N-[3-methoxy-4-(morpholine-4-carbonyl)phenyl]pyridine-4-carboxamide 2-[(1S,6R)-7-ethyl-2-(oxane-4-carbonylamino)-3-azabicyclo[4.1.0]heptan-3-yl]-N-methyl-1H-benzimidazole-5-carboxamide 3-fluoro-5,6-dimethoxy-7,8,9,10-tetrahydroimidazo[1,2-d][1,4]benzodiazepine N-[(2S,4R)-2-methyl-1-prop-2-enoylpiperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide 1-N-[2-(3,5-dimethylphenyl)ethyl]-4-N-[5-[2-methoxy-5-(propanoylamino)phenyl]pyridin-2-yl]benzene-1,4-dicarboxamide 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-1,3-dioxolane 2-(4,6-diamino-1,3,5-triazin-2-yl)acetic acid;1-ethoxypyridin-1-ium 6-methyl-3-phenylmethoxy-2-[(3,4,5-trichlorophenyl)sulfanylmethyl]pyridine 4-(4-fluorobenzoyl)-1H-pyrrole-2,3-dicarboxamide 4-amino-N-[(1Z,3E)-1-[methyl(propan-2-yl)amino]penta-1,3-dien-3-yl]benzamide 4-[8a-(hydroxymethyl)-2,3,5,6-tetrahydroimidazo[1,2-a]pyrazin-7-yl]benzonitrile;dihydrochloride 1-(3-azidophenyl)-2,4-dichlorobenzene [4-(2-cyclobutyloxyanilino)piperidin-1-yl]-[6-methyl-3,4-bis(sulfanylidene)-2H-pyridin-5-yl]methanethione 5-(furan-2-yl)-4-methylidene-1,3,6-triphenylpyrrolo[3,4-c]pyrrole N-[(3,5-dimethoxyphenyl)methyl]-2-oxo-1H-pyridine-4-carboxamide N-[[4,5-bis(ethenyl)furan-3-yl]methyl]-2-(4-fluorophenyl)-N-methylethanamine 1-bromopyrrolo[2,3-b]pyridine-2-carboxylic acid 1-[3,4-dichloro-5-(4-ethoxycarbonylpiperidine-1-carboximidoyl)phenyl]-2H-pyridine-4-carboxylic acid N-[(1S,3R)-2,2-dichloro-3-[4-fluoro-3-(trifluoromethyl)phenyl]cyclopropanecarbonyl]-3-ethyl-N-[2-hydroxy-5-[1-(4-propan-2-ylbenzoyl)piperidin-4-yl]phenyl]benzamide 5-(3-benzylsulfanyl-2,5-dichlorophenyl)-1,5,6,8-tetrahydropyrimido[4,5-d]pyrimidine-2,4,7-trithione 4-tert-butyl-2-[(2,6-dimethoxyphenyl)methylsulfanyl]-5-iodo-1H-pyrimidin-6-one ethane;N-[4-(2-fluorophenyl)cyclohexyl]propanamide 5-[3-amino-4-(trifluoromethoxy)anilino]sulfanyl-6,7-dihydro-1H-indole-2-thiol;hydrochloride N-[2-chloro-3-(1,5,7,10,11-pentazatricyclo[6.4.0.02,6]dodeca-2(6),3,7,9,11-pentaen-12-ylmethyl)phenyl]methanesulfonamide 1-[3-(3,4-dihydropyrido[2,3-b]pyrazine-8-carbonyl)pyrrolidin-1-yl]ethanone 7-[(2,4-dimethoxyphenyl)methyl]-2-(3-fluoropyridin-4-yl)-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 2-(4-acetamido-N-(3,4-dimethoxyphenyl)sulfonylanilino)-N-[(Z)-(2-hydroxyphenyl)methylideneamino]butanamide 2-[2,6-difluoro-4-(trifluoromethylsulfanyl)phenyl]-5-phenylfuran 5-[(Z)-1-amino-3,3,4,4-tetrafluorobut-2-enyl]-N-methylpyridine-2-carboxamide (2R)-3-(4-fluorophenyl)-2-[2-[4-methyl-6-oxo-2-(1-phenylethylamino)-1H-pyrimidin-5-yl]acetyl]oxypropanoic acid 2-[3,5-dichloro-4-(7-cyano-6,8-difluoroquinoline-3-carbonyl)oxyphenyl]propanoic acid 5-(6,7-dihydro-1H-benzimidazol-2-yl)-4-N,8-N-dimethylisoquinoline-3,4,8-triamine 6-[4-(4,5-dihydro-1H-imidazol-2-yl)piperidin-1-yl]pyrimidine 4-(2,6-dichlorophenyl)-5-methyl-1H-pyridine-2-thione 1-bromo-2,4,5,6-tetramethylpyrene 2-N,3-N,4-N-triethylbenzene-1,2,3,4-tetramine 1-(2,4-dichlorophenyl)-3-[5-[4-(trifluoromethyl)pyrimidin-2-yl]oxolan-2-yl]urea 3-amino-5-[2,6-dichloro-4-(trifluoromethyl)phenyl]sulfonylphenol N-[4-[8-amino-6-(8-methylnaphthalen-2-yl)imidazo[1,5-a]pyrazin-3-yl]cyclohexyl]propane-1-sulfinamide 1-[4-(hydroxymethyl)phenyl]sulfonylbutan-2-ol 5-[3-(4,6-diphenyl-1,3,5-triazin-2-yl)phenyl]-15,16-diazaheptacyclo[14.9.0.02,10.03,8.011,23.012,17.022,25]hexacosa-1(26),2(10),3(8),4,6,11(23),12,14,17,19,21(24),23-dodecaene 2-[(4-methylphenyl)methoxy]-1H-quinoline [3-amino-5-methoxy-4-(2-methylpropyl)phenyl]boronic acid (3,5-difluorophenyl)sulfonyl-[2-hydroxy-6-[[4-(1H-pyrazol-5-yl)piperazin-1-yl]methyl]spiro[3.3]heptan-2-yl]azanium 4-[6-(4-fluoroanilino)-2,4-dioxo-1H-quinazoline-3-carbonyl]piperazine-1-carboxylic acid 4-chloro-3,5-diphenylpyrazole (4S,5R)-5-ethyl-3-[1-(2-methoxyphenyl)isoquinolin-6-yl]imidazolidine-2,4-dione 2-[4-bromo-N-(2,3-dihydroxypropyl)anilino]guanidine (5Z)-2-(2,6-dichlorophenyl)imino-5-[[3-ethoxy-4-[(4-fluorophenyl)methoxy]naphthalen-1-yl]methylidene]-1,3-thiazolidin-4-one 5-[4-(6,7-dihydro-1H-benzimidazole-2-carboximidoyl)piperidin-1-yl]-3-[4-methoxy-3-(trifluoromethyl)phenyl]sulfonylpentanoic acid 2-(1,3-benzothiazol-2-yl)-5-chlorophenol;zinc 2-[4,5-diethyl-3-(phenylmethoxycarbonylamino)pyrazol-1-yl]acetic acid 4-(3,5-dimethylphenyl)-N'-hydroxypyridine-2-carboximidamide 2-(4-azidophenyl)-N,N-dimethyl-1H-inden-5-amine N-[3,5-dichloro-4-(2,6-dioxopiperidin-3-yl)phenyl]-2-(7-fluoro-3-methyl-1H-isoindol-2-yl)acetamide 6-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(prop-2-enyl)amino]-4-hydroxynaphthalene-2-sulfonic acid (1R,2S)-N-[8-amino-6-[4-[3-[ethyl(methyl)carbamoyl]-5-methoxyphenyl]pyridin-3-yl]isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide ethane;(3Z,5E)-1-(4-methyl-2-propan-2-ylphenyl)octa-3,5-dien-7-one 3-(2,4-dichlorophenyl)-5-fluorobenzamide [[3-(3,4-difluorophenyl)-2H-tetrazol-5-yl]hydrazinylidene]methanamine N-[2-(2-ethoxyphenoxy)propyl]formamide 6-[4-(2,2-dimethylpropoxy)-3-(trifluoromethyl)phenyl]pyridine-3-carboxamide 2-methyl-5-[1-(2,3,4-trihydroxyphenyl)ethyl]benzene-1,4-diol 3-[5-(2,4-dimethylpentan-3-ylidene)cyclohexa-1,3-dien-1-yl]-2-propan-2-ylpyridine 6-[(5-chloro-2-oxo-1H-indol-3-ylidene)methyl]-N,4-dimethyl-7-(1-propanoylpiperidin-4-yl)oxy-8,9-dihydropyrimido[4,5-e][1,4]oxazepine-2-carboxamide 3-amino-N',2-dimethylbenzimidazole-5-carboximidamide 2-(5,6-diphenylpyrimidin-4-yl)-3-phenylbenzene-1,4-diamine N'-(2,3-dihydro-1H-indene-5-carbonyl)pyridine-4-carbohydrazide 3-[2-oxo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-1-yl]benzoic acid N-[4-(hydroxymethyl)oxan-4-yl]-6-methoxypyridine-3-carboxamide 6-[(E)-2-cyclohexylethenyl]-3-fluorobenzonitrile (6R)-5,7-dihydroxy-6,8-bis[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]octanoic acid 3-(9H-fluoren-2-ylmethoxy)benzenecarboximidamide (2S)-N-methyl-N-[4-(3-methylbutan-2-ylideneamino)phenyl]-1-[[4-[4-(trifluoromethyl)phenoxy]cyclohexyl]methoxymethyl]propan-2-amine 3-benzylsulfanyl-N'-hydroxypyrazine-2-carboximidamide 6-chloro-3-N,4-N-dimethyl-2-(trifluoromethyl)pyridine-3,4-diamine 4-[5-(1H-benzimidazol-2-yl)-6-chloropyridin-3-yl]oxy-3,5-dimethyl-N-phenylaniline (6R)-2,7-bis[(3S)-oxolan-3-yl]-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one 2,4-dichloro-N-[5-chloro-6-(4-methylpiperazine-1-carbonyl)pyridin-3-yl]benzenesulfonamide [4-[(5-fluoropyridin-2-yl)methoxy]phenyl]methanimine 6,7-dibromo-1-propanoylnaphthalene-2-carbonitrile 3-[1-(4-chlorophenyl)-2,5-dioxopyrrolidine-3-carbonyl]-1H-pyrrolo[3,2-b]pyridine-6-carboxylic acid 3-(4-acetylpiperazine-1-carbonyl)-N-methylidenebenzenecarboximidamide N-[(3R)-1-cyanopyrrolidin-3-yl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide 1-[6-(6,7-dihydroquinolin-2-ylmethoxy)naphthalene-2-carbonyl]pyrrolidine-3-carboxylic acid [(2S)-4-[7-(8-chloronaphthalen-1-yl)-2-methoxy-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]piperazin-2-yl]-pyrrolidin-2-ylmethanol (7S)-N,2-dimethyl-3-(propan-2-ylamino)-5-[4-(trifluoromethoxy)phenyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-6-carboxamide N-(3-cyclohexyl-5-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)butanamide 3-(4-azidophenyl)-5-(2,6-dimethylmorpholine-4-carbonyl)-1H-pyridin-2-one 3-methyl-1,2-bis(2,4,6-trimethylphenyl)imidazolidine 4-azido-1-methylquinoline-2,6-dione N-(cyclopropylmethoxy)-2,4-difluoro-5-[[[5-oxo-7-(trideuteriomethylamino)-[1,3]thiazolo[3,2-a]pyridine-3-carbonyl]amino]methyl]benzamide 1-[4-(2,2-dimethoxyethyl)phenyl]-5-[(3R)-pyrrolidine-3-carbonyl]piperidin-2-one;hydrochloride [4-(6,7-dihydro-5H-cyclopenta[b]pyridin-3-ylamino)piperidin-1-yl]-(2-methoxyphenyl)methanone 6-(3,5-difluorophenyl)-2-(4-ethylsulfonylpiperidin-1-yl)-N-methoxyquinazolin-4-amine 2-(1,5-dimethylpyrazol-4-yl)-N-[1-[4-(trifluoromethoxy)phenyl]pyrrolidin-3-yl]acetamide 2-(4-bromophenyl)-3,10,12,14-tetrazatetracyclo[6.6.1.02,7.011,15]pentadeca-1(15),2,4,6,8,11,13-heptaene;hydrochloride 3-[(4-chlorophenyl)methylamino]-5-methyl-1H-pyridine-2,6-dione;3-hydroxycyclobutan-1-amine 3-(4-nitrophenyl)-1-oxidopyridin-1-ium 5-(3-chloroanilino)-N-[(Z,2S)-2-methylpentylideneamino]-4H-azepine-7-carboxamide 2-[(5S)-3,4-dimethyl-7,11-dioxo-5H-benzo[d][1]benzazepin-6-ylidene]propanenitrile;N-(2,5-dimethylphenyl)acetamide 1-(3,4-dichlorophenyl)sulfonyl-4-ethyl-N'-methylsulfanylpiperidine-4-carbohydrazide 3-[(2-chloro-4,5-dimethoxyphenyl)methyl]-1H-pyrido[3,2-b]indole 4-[3-(2,3-dihydropyridin-4-yl)phenyl]butanoic acid 2-cyclobutylidene-5,7-dimethylquinazolin-4-one ethane;N-(2,3,4,5,6-pentafluorophenyl)aniline 2,3-bis(ethylsulfanyl)benzo[g]pteridine-4,9-dione 2-(1H-benzimidazol-2-ylsulfanyl)-N-[5-bromo-2-methoxy-4-[(E)-2-phenylethenyl]phenyl]butanamide N-(3-bromophenyl)pyrrolidine-2-carboxamide N-[3-[(E)-2-[4,5-bis(ethenyl)-1H-imidazol-2-yl]ethenoxy]propyl]acetamide 3-[3-methylbut-2-enyl(prop-2-enyl)amino]phenol 3-[(2,5-dimethoxyphenyl)sulfonylamino]-4-[(4-ethylpiperazin-1-yl)methyl]benzoic acid;2,2,2-trifluoroacetic acid N-(4-azidobutyl)-2-[5-[(2,3,4,5,6-pentafluorophenoxy)methyl]pyridin-2-yl]acetamide N-[(Z)-1H-indol-3-ylmethylideneamino]-2-(2,4,6-trichlorophenoxy)acetamide 1-N,2-N,3,6-tetramethylnaphthalene-1,2,8-triamine (E)-3,4-dimethyl-N-[[1-[(3,4,5-trifluorophenyl)methyl]piperidin-4-yl]methyl]oct-2-enamide N-[2-(1,3-benzodioxol-5-yl)ethyl]spiro[1H-2-benzofuran-3,4'-piperidine]-1'-carboxamide 2-(3-bromopyridin-2-yl)-N,N'-di(propan-2-yl)ethane-1,2-diamine 5-[[4-(methylamino)phenyl]methylsulfanylmethylideneamino]pentan-2-one 2-[(3-butoxyphenoxy)methyl]benzenethiol N-(2,4-difluorophenyl)-2-methoxy-5-[5-(2-oxopyrrolidin-1-yl)sulfonylpyridin-3-yl]benzamide 4-amino-N,N-dimethyl-2-propylbenzamide;6-(methoxymethyl)-1H-indole 1-ethyl-4-[(E)-3-methylidenepent-1-enoxy]benzene 4-[(2R)-2-[2,5-bis(difluoromethoxy)phenyl]pyrrolidin-1-yl]-3-methylquinazoline (Z)-2-methoxycarbonyl-3-phenyl-3-phenylsulfanylprop-2-enoic acid ethane;2-(3-methylphenyl)-N,N-dipropylbutan-1-amine 5-[[7-(4-methylpiperazine-1-carbonyl)imidazo[1,2-c]quinazolin-3-yl]methyl]-1H-indole-2-carbonitrile (6-ethylpyridine-3-carbonyl)carbamic acid (6R,9S)-6-(furan-2-yl)-9-thiophen-3-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one (2E)-3,4-dimethoxy-1-phenyl-2-[(E)-[3-(trifluoromethyl)phenyl]methylidenehydrazinylidene]butan-1-one 2-[4,6-bis(dimethylamino)-1-methylpyridin-1-ium-3-yl]acetic acid 4-[(3S)-1,2-dioxo-5-phenylpentyl]benzoic acid N-[2-azido-1-(3,4,5-trimethoxyphenyl)ethyl]propanamide 6-cyclopentyl-2-[1-(2,3-dihydro-1H-indene-4-carbonyl)piperidin-4-yl]pyridazin-3-one 6-benzyl-2-[(3S,4R)-4-ethoxypiperidin-3-yl]-1H-benzimidazole;dihydrochloride 4-azidooxy-3-(oxolan-2-yl)pyridine N-[2-(5,6-dimethylpyrimidin-4-yl)oxyethyl]-1,3-benzothiazol-7-amine ethane;N-methylcyclopropanamine;2-[1-[4-methyl-3-(trifluoromethoxy)phenyl]ethylamino]-4,8-dioxo-7H-pteridine-6-carbonitrile 3-[5-(2-aminopyrimidin-4-yl)-1,3-dihydroisoindole-2-carbonyl]-N-[(6E,10Z)-10-ethylidenedodeca-6,8,10-trienoyl]benzamide N-[3-[(2E)-2-[(Z)-prop-1-enyl]penta-2,4-dienoxy]phenyl]-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-2-carboxamide 4-(5,6-dihydroisoquinolin-1-yl)-2H-phthalazin-1-one 3-[(2,6-dichlorophenyl)methyl]-5-[2-(1H-imidazol-2-ylmethoxy)propan-2-yl]-4-methyl-1,2,4-triazole 3-[2-(4-azidobutyl)-5-fluorophenyl]pyridine 3-ethyl-4,5-dimethoxythiophene-2-carboxylic acid N-(2,3-dihydroxypropyl)-N-methylbenzenesulfonamide 6-(4-hydroxy-5-propan-2-yl-3-propanoylphenyl)hexanoic acid 1-N,2-N,4-N-trimethyl-1-N-(4-methylphenyl)benzene-1,2,4-triamine 2-[1-[2,3-bis(ethenyl)naphthalene-1-carbonyl]piperidin-4-ylidene]acetic acid 2-[[5-[(Z)-2-(2,3-dihydro-1H-inden-4-ylamino)-4-oxobut-2-enyl]pyrazin-2-yl]amino]acetic acid;hydrochloride 2-(2,6-dioxopiperidin-3-yl)-4-[2-methoxyethyl-[4-(1H-pyrazol-5-yl)cyclohexyl]amino]isoindole-1,3-dione N-[(2S)-3-(4,6-dimethoxypyrimidin-2-yl)-1H-indol-2-yl]carbamate 1-(1,3-benzodioxol-5-ylsulfonyl)pyrrolidine 2-[4-(2,6-difluorobenzoyl)piperazine-1-carbonyl]-3H-quinazolin-4-one 4-[3,5-dimethyl-1-(propanoylamino)pyrazol-4-yl]sulfonylpiperazine-1-carboxylic acid (2S)-4-amino-N-[(4-methoxyphenyl)methyl]-3,3-dimethylbutanamide 4-(6-bromothieno[3,2-d]pyrimidin-4-yl)-N,1-dimethylpiperazine-2-carboxamide 4-[5-(furan-2-ylmethylamino)-1,3,4-thiadiazol-2-yl]phenol N-[(3,4-dimethylphenyl)methyl]-2-[3-ethoxy-4-(2H-tetrazol-5-yl)phenyl]ethanamine 2-aminoacetaldehyde;N'-[1-(5,6-dichloropyridin-3-yl)ethenyl]methanimidamide N-(2,4-dioxo-1H-pyrimidin-5-yl)-N-hexylmethanesulfonamide (Z)-1-[4-hydroxy-2-oxo-3-phenyl-5-(trifluoromethyl)imidazolidin-1-yl]-N'-phenylprop-1-ene-1,3-diamine N-[(3R)-1-(5-amino-2,4-difluorobenzoyl)piperidin-3-yl]-7,8-dihydrothieno[3,4-b][1,4]dioxine-6-carboxamide 1-[[(2R)-oxetan-2-yl]methoxy]isoquinoline 1-(azetidin-3-yl)-N-[(3,5-difluorophenyl)methyl]-4-[(E)-3-fluoroprop-2-enoxy]piperidine-4-carboxamide N-[2-(N-methylsulfonylanilino)ethyl]acetamide 3-cyclopentyl-1,7-dimethylpurine-2,6-dione (3R)-4-ethoxy-1-[6-methyl-5-[2-methylpropyl-[[4-(trifluoromethyl)phenyl]methyl]amino]pyrazine-2-carbonyl]pyrrolidine-3-carboxylic acid N-[2-(4-cyanophenyl)ethyl]-6-(3,5-dimethoxyphenyl)-8-[4-hydroxy-3-(trifluoromethyl)anilino]imidazo[1,2-b]pyridazine-3-carboxamide (E)-N-[2-[(1S,3R)-3-(aminomethyl)cyclohexyl]oxypyridin-4-yl]-3-cyclopropyl-N'-[5-fluoro-6-(2-methoxyethoxy)-1H-indazol-3-yl]prop-2-enimidamide (3Z)-7,8-difluoro-N-methyl-2-oxo-3-[[4-(trifluoromethoxy)phenyl]methylidene]quinoline-6-carboxamide 1-azido-4,5,8-trimethylnaphthalene 6-(1,3-benzodioxol-5-yl)-2,7-bis(4-methoxyphenyl)quinoxaline 1-[2-(4-methoxyphenyl)ethyl]-6-(6-methylidene-2,3-dihydropyran-4-yl)imidazo[4,5-c]pyridine 1-(4-methoxyphenyl)sulfonyl-2-[2-methyl-6-(5,6,7,8-tetrahydroquinolin-3-yl)pyridine-4-carbonyl]piperidine-3-carboxylic acid 2-amino-6-[4-(dipropylamino)phenyl]quinoline-5,8-dione N-[2-(1,5-dimethylpyrazol-4-yl)ethyl]prop-2-enamide 6-(4-fluorophenyl)-2-[1-(5-methylsulfanylpyridine-3-carbonyl)piperidin-4-yl]pyridazin-3-one 1-N,3-N-diphenylnaphthalene-1,3-disulfonamide N-[1-cyclopropyl-2-(4-fluorophenyl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide 3-[4-(6-methoxynaphthalen-2-yl)sulfonylphenoxy]propanoic acid 2-[4,6-bis(3H-azepine-7-carbonyl)benzimidazol-1-yl]acetic acid 2-[4-[(2S)-1-tert-butylsulfonylpropan-2-yl]-6-(4,4-dimethylcyclohexen-1-yl)pyridin-3-yl]-5-chloropyrimidine [(2S)-1-(2,6-difluorophenyl)pyrrolidin-2-yl]methanol N-[[4-chloro-3-(6,7-dihydroquinoline-2-carbonyl)phenyl]methyl]-2-methoxyacetamide N-(azidomethyl)-6-chlorospiro[1,4-dihydroquinoline-3,4'-oxane]-2-imine 2-chloro-7-methoxy-8-nitro-4,6-dihydropyrido[3,4-d]pyrimidine 4-amino-6-[(3,5-dibromo-2-fluorophenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 1-[5-(azepan-4-ylmethyl)thiophen-2-yl]ethanone 4-hydroxy-2,3-dihydrothiochromene-4-carbothioate 4-[(2,2-dimethylpropanoylamino)methyl]-N-phenylbenzamide N-[4-[(4S)-4-methylcyclohexa-1,5-dien-1-yl]phenyl]-2,3-dihydropyridine-2-carboxamide 3-chloro-2-(3,4-dimethylpyridin-2-yl)oxy-5-fluorobenzonitrile N-[5-cyclopropyl-2-(4,6-dimethylpyrimidin-2-yl)pyrazol-3-yl]pyrazine-2-carboxamide 1-N',2-diphenylethene-1,1-diamine;4-methyl-7H-naphthalene 2-[(5E)-4-methylidene-5-[(E,3Z)-3-(6-pyridin-2-yl-1H-benzimidazol-2-yl)but-2-enylidene]-1H-pyrazol-3-yl]-4-thiophen-2-yl-1H-pyrrolo[3,2-c]pyridine 4-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-N'-methylbenzenecarboximidamide N-[4-(dimethylamino)phenyl]-N'-ethyl-N'-(3-fluorophenyl)methanediamine [5-(4-chlorophenoxy)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxyphosphane 4-[2,3-bis(ethenyl)-4-hydroxyphenyl]-5-(3-methoxyphenyl)-1H-1,2,4-triazole-3-thione 5-[2-(4-chlorophenyl)ethoxymethyl]pyrrolidin-3-one 7-azido-3,5-dichloro-2H-1,8-naphthyridine 6-(azepan-1-yl)-4-tert-butylpyridazine 6-[7-(3,4-dichlorobenzoyl)-2-piperazin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-1-(oxan-4-yl)-3,4-dihydroquinolin-2-one (3S)-2-[4-fluoro-6-[(1R,5R)-3-oxabicyclo[3.1.0]hexan-1-yl]pyridine-2-carbonyl]-N'-hydroxy-2-methylspiro[3H-chromene-4,4'-piperidine]-1'-carboximidamide 5-chloro-2-methyl-N'-(2,4,6-trimethoxyphenyl)benzohydrazide 1-[3-[(4R,6R)-2-amino-8-hydroxy-4-phenylmethoxy-7,8-dihydropyrano[4,3-d]pyrimidin-5-yl]-5-ethynylcyclohexa-1,3-dien-1-yl]ethanone [6-chloro-2,3-difluoro-4-(trifluoromethyl)phenyl]boronic acid 2-(4-amino-1,3,5-triazin-2-yl)benzene-1,3-diol 3-butyl-2,7-dichloroquinoline 2-[3-(2,6-dichlorophenoxy)-5-oxocyclohexylidene]acetic acid N-[2-chloro-3-(trifluoromethoxy)phenyl]-2-hydroxyethanesulfonamide 5-(2,6-dimethoxyphenyl)-1-ethyl-4-iminoimidazolidin-2-one N-[2,4-bis(trifluoromethyl)phenyl]-6-[4-[2-[butanoyl(cyclopropyl)amino]ethoxy]piperidin-1-yl]-5-cyano-3,4-difluoropyridine-2-carboxamide 1-[4-[2,5-dimethyl-2,3,7-tris(sulfanylidene)pyrido[4,3-e]thiazin-4-ium-4-yl]phenyl]-3-(pyridin-3-ylmethyl)urea;bromide N-[(3R,4S)-3-fluoropiperidin-4-yl]-5-methylsulfonyl-2-phenylbenzamide;hydrochloride N-(cyclopentylmethyl)-2-[4-(cyclohexanecarbonylamino)-3-fluorophenyl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 2-[(6S)-6-[(1,1-dioxothiolan-3-yl)amino]-5,6,7,8-tetrahydronaphthalen-2-yl]cyclohexan-1-amine 3-bromo-6-(methoxyamino)-5,8-diphenylnaphthalene-2,7-disulfonic acid 4-[(1R)-3,6-difluorocyclohexa-2,4-dien-1-yl]sulfonyl-N-methylaniline 7-bromo-1,2-diethylindole 4-[[(3S)-pyrrolidin-3-yl]amino]-1H-pyrimidin-6-one 3-(4-chlorophenyl)-N',N'-diethylbenzohydrazide 6-methyl-3,5-dinitrobenzene-1,2,4-tricarboxylic acid 2-hydroxy-5-[(4-methylphenyl)sulfonylamino]benzoic acid ethane;1-(2-methoxynaphthalen-1-yl)-N-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]methanimine 2-azido-1,3-difluoro-5-[2-(4-propan-2-ylcyclohexa-2,4-dien-1-yl)ethynyl]benzene (3S,4R)-1-[2-(5,7-difluoro-3H-indol-3-yl)ethyl]-4-ethenylpyrrolidin-3-amine [6-(trifluoromethyl)pyridin-2-yl]urea 4-(2,3-dimethylphenyl)-1H-pyrrole-2-carboxylic acid 3-[2,6-dichloro-4-nitro-N-(2H-tetrazol-5-yl)anilino]propane-1,2-diol (6S)-5-[2-(3,5-dimethylphenyl)pyrrolidine-1-carbonyl]-6-(4-fluorophenyl)piperidin-2-one 1-(3,4-dihydro-2H-quinolin-1-yl)-2-[4-(ethylaminomethyl)phenyl]sulfanylpropan-1-one 2-[4-[6-(2,3-dimethylimidazol-4-yl)pyrazolo[1,5-a]pyridin-4-yl]pyrazol-1-yl]propan-2-ol N-(2,6-dichloro-3,5-dimethoxyphenyl)-7-fluoro-2H-4,1,3-benzoxadiazole-5-carboxamide 4-chloro-7-methyl-1-(2-phenoxyethoxy)isoquinoline 5-(6,7-dihydroquinolin-4-yl)pyridine-3-carbonitrile [4-(2-aminophenyl)piperazin-1-yl]-spiro[2H-indole-3,7'-6H-furo[2,3-f][1,3]benzodioxole]-1-ylmethanone 5-[(3S)-6-aminohexan-3-yl]oxy-2-chlorophenol (2S)-N-[(1R)-1,7-dihydroxy-1H-pyrrolo[3,4-c]pyridin-6-yl]-1-methylsulfonylpyrrolidine-2-carboxamide (2S)-4,4,4-trifluoro-3-methoxy-2-[(4-nitrobenzoyl)amino]butanoic acid 2-chloro-N-(cyclohexa-1,5-dien-3-yn-1-ylmethyl)aniline 7-[3,5-bis(trifluoromethyl)phenyl]heptanoic acid 6-methyl-4-[(5-propan-2-ylthiophen-3-yl)amino]-1H-pyrido[3,2-d]pyrimidine-8-carboxamide 3-[[4-(2-methoxyethyl)phenyl]sulfonylamino]-N,N,2-trimethylbenzenesulfonamide 1-[3,4-dichloro-2-(trifluoromethyl)phenyl]propan-2-one 2-(2,4-difluorophenyl)-N-[3-(methanesulfonamido)pyridin-4-yl]piperidine-1-carboxamide N'-[(2Z)-3,4-dimethylpenta-2,4-dien-2-yl]sulfanyl-1H-indole-2-carboximidamide;ethane 4-(cyclopropanecarbonyl)-N'-[5-fluoro-6-(triazol-2-ylmethoxy)pyridin-3-yl]piperazine-1-carboximidamide 5-bromo-4-cyclobutyl-2-(1,3-thiazol-2-yl)-1H-pyrimidin-6-one 1-[(1S)-2,3,4,9-tetrahydro-1H-fluoren-1-yl]pyrrolidine 2,4-dichloro-N-[(Z)-(2,4-dimethoxyphenyl)methylideneamino]benzamide 1-(5-cyclopentylsulfonylthiophene-3-carbonyl)piperazine N-[2,6-di(propan-2-yl)phenyl]-1H-imidazol-3-ium-5-carboxamide [(1R)-2-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-yl]methanol 2-(4-fluorophenyl)sulfonyl-N,1H-benzimidazole-4-sulfonamide 3-(2-nitro-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]anilino)propanoic acid 5-[6-(3,4,5-trichlorophenyl)-4,5-dihydropyridazin-2-ium-2-yl]pyrimidine 1-[7-(trifluoromethyl)pyrazolo[4,3-b]pyridin-2-yl]butane-2,3-dione 1-[2-(4,7-dimethoxyquinolin-6-yl)ethyl]pyrrolidine-3-carboxylate 2,4-dichloro-6-(2,2-dimethylpropyl)phenol 4-[(3R)-3,5-dimethylpiperazine-1-carbonyl]benzenesulfonamide 2-(1H-benzimidazol-2-ylsulfanyl)-N,3-dimethoxypropan-1-amine 6,8-diaminopurine-9-carboxylic acid 2-cyclopropyl-4,7-dioxo-3,6,8,9-tetrahydropyrido[1,2-a]pyrimidine-9-carbonitrile (3Z)-1,2,4-trichloropenta-1,3-diene;5H-chromeno[2,3-b]pyridine 3-[5-(4-chlorophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2,4-dimethoxybenzaldehyde 2-[N-ethylsulfonyl-4-(thiophen-2-ylsulfamoyl)anilino]decanoic acid 2-[2-(1-cyclopropyl-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)phenyl]acetamide 4-[3-(difluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine-2-carbonyl]benzenesulfonamide 4-[2-[4-(1,3-benzodioxol-5-ylsulfonyl)piperazin-1-yl]ethyl]-7-fluoropyrido[3,2-b]indole 4-[(2S)-1,2-dihydroxyethyl]benzaldehyde;3-[[(2S)-4-methyl-2-methylidenepentanoyl]amino]thiophene-2-carboxylic acid N-(2,3-dihydrofuro[3,4-b]quinolin-1-yl)benzamide [4-(2,3-dihydroindole-1-carbonyl)piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone N-[6-methyl-5-(2,3,4,6-tetrafluorophenoxy)pyridin-2-yl]methanesulfonamide 1-[(2,5-difluorophenyl)methyl]-3-phenylimidazol-2-imine 1-[[4-(4,5-dichloroimidazol-1-yl)phenyl]methyl]-4-propanoylpiperazine-2-carboxamide 1-[(2,3,4,5,6-pentafluorophenoxy)methyl]naphthalene 1-[2,5-bis(trifluoromethyl)phenyl]-3-methylurea 6-methoxy-1-[(5-nitrofuran-2-yl)methylidene]indene N'-[(3R,5S)-3,4,5-trihydroxy-6-methyloxan-2-yl]thiophene-2-carbohydrazide 4-[1-azido-2-(4,5-dimethylcyclohexa-1,3-dien-1-yl)ethyl]phenol 1-[2-(dimethylamino)ethyl]-4-(3,5,7,10,12-pentazatricyclo[7.3.0.02,6]dodeca-1,3,6,8,11-pentaen-13-yl)piperidine-4-carbonitrile 6-[[2-(3,4,5,6,7,8-hexahydro-1H-isoquinolin-2-yl)acetyl]amino]pyridine-2-carboxamide 1-(5-amino-4,6-diethylpyrimidin-2-yl)-3-(cyclopropanecarbonylamino)urea 4-chloro-N'-[(2,3-difluorophenyl)methyl]benzohydrazide 2-[(1S,4R)-3-benzoyloxy-3-oxo-4-phenylmethoxycyclopentyl]acetic acid N-[2,5-dimethoxy-4-(trifluoromethyl)phenyl]-3-(propanoylamino)benzamide 2-[3-[4-[(5R)-1-(5-bromopyridin-2-yl)-2-azabicyclo[3.1.0]hexan-2-yl]butoxymethyl]phenyl]acetamide [(2S,3aS)-2-phenyl-1,4-dioxa-8-azaspiro[4.5]decan-8-yl]-(4-methoxypyrazolo[1,5-a]pyridin-7-yl)methanone [5-methyl-2-(oxan-4-ylamino)pyrimidin-4-yl]boronic acid (2-aminopyridin-3-yl)-[4-(4-propan-2-ylanilino)piperidin-1-yl]methanone 3-[[4-(1,2-benzoxazol-6-yloxymethyl)piperidin-1-yl]methyl]-5-(trifluoromethyl)-1,2,4-oxadiazole 2-cyclohepta-1,4,6-trien-1-yl-N-(5-methylfuran-2-yl)imidazo[1,2-a]pyridine-3-carboxamide 2-[4-[6-chloro-8-fluoro-7-(12-methyl-7,11-dihydropyrido[3,2-a]carbazol-5-yl)isoquinolin-3-yl]piperazin-1-yl]ethanol ethane;4-[4-(5-methyl-1H-indazol-3-yl)triazol-1-yl]butanoic acid 6-amino-4-(3,5-ditert-butyl-2-hydroxyphenyl)-4-methyl-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile N-[(1S)-4-fluoro-6-phenylmethoxy-2,3-dihydro-1H-inden-1-yl]pyridine-3-carboxamide 1-azidooxy-5-chloro-2,3-dihydroindene 5-hydroxy-3,7-dimethyl-4H-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid 3-[2,4-dimethyl-6-(4-morpholin-4-ylanilino)benzimidazol-1-yl]propanal 1-[(2Z)-2-methylsulfanylpenta-2,4-dienyl]-5-(pyridin-3-ylmethoxy)benzotriazole 7-chloro-6-(4-hydroxyphenyl)-3,5-dihydro-1H-imidazo[2,1-b]quinazolin-9-one 2-(5,6-dichloropyridin-3-yl)-1H-indole 4-[(3Z,5E)-5-methylhepta-1,3,5-trien-2-yl]oxycarbonylbenzoic acid 2-[6-fluoro-5-[(2E,4Z)-hepta-2,4,6-trien-3-yl]oxypyridin-3-yl]-8-methyl-N-propan-2-ylquinazolin-4-amine 3-methyl-1-(2,4,6-trichlorophenyl)pyrazole 3-[1-(dimethylamino)ethoxy]quinoxalin-2-amine 3-azido-2-methylsulfanylfluoren-1-one 2-(4-chlorophenyl)-2-[5-[3,5-dimethyl-1-(1H-pyrazol-4-yl)pyrazol-4-yl]pyridin-2-yl]oxyethanol (2R,3S)-1-(azidomethyl)-N-[2-(cyclopropanecarbonylamino)imidazo[1,2-a]pyridin-6-yl]-N'-(4-chlorophenyl)-5-oxopyrrolidine-3-carboximidamide N-[2,4-dimethyl-5-(6-morpholin-4-ylpyridine-3-carbonyl)phenyl]-2-fluorobenzamide 1-(2-azidoethyl)-3-[4-(trifluoromethoxy)phenyl]urea (2S)-N-[1-cyclohexyl-2-oxo-2-[4-(2,2,3,3,4,4,5-heptadeuteriopyrrolidine-1-carbonyl)anilino]ethyl]-2-(methanesulfonamido)pentanamide N-(2,2-difluoroethyl)-1'-[(5-methylfuran-3-yl)methyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 4-chloro-N'-(2-cyano-6-fluoro-3-methylbenzoyl)-3-[(E)-3-(1,3-dioxoisoindol-2-yl)propoxyiminomethyl]benzohydrazide 6-methylsulfonyl-2-piperidin-1-ylquinazoline N'-amino-4-(3,5-diethoxyphenyl)-N-methylbenzenecarboximidamide (7-methoxyspiro[chromene-2,4'-piperidine]-1'-yl)-[4-(1,3-thiazol-4-yl)phenyl]methanone N-methyl-2-oxo-N-[4-[(2E,3Z)-penta-2,3-dien-2-yl]oxycyclohexyl]-1H-pyridine-3-carboxamide 3-[(E)-[(1S,5R,6S)-7,9-dihydroxy-9-oxo-3-oxa-7-azabicyclo[4.2.0]octan-10-yl]iminomethyl]chromen-2-one 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-[2-methyl-4-[(2-methylphenyl)diazenyl]phenyl]amino]decanoic acid ethane;2-(1,4-oxazepane-4-carbonyl)indole-1-carboxamide 1-(2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-fluoropyrrolidine-3-carbonitrile 3-methoxy-2,5-dimethyl-1-[4-[(2S)-pentan-2-yl]phenyl]pyrrole (4S,5R)-3-[(E)-1-cyclohexylprop-1-enyl]-2-ethoxy-5-phenyl-4,5-dihydro-1H-azepine [1-[1-[2,6-dimethyl-4-(oxan-4-ylamino)phenyl]ethenyl-ethylamino]cyclopropyl]methylideneazanide 2-[(3,5-dimethoxyphenyl)-morpholin-4-ylmethylidene]propanedioic acid 2-cyclopentyl-1-[4-(4-ethenyl-5-methyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]propan-1-one 1-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-5,6-dihydro-4H-cyclopenta[c]pyrazole 2-[(1S)-1-[4-[3-hydroxy-5-(trifluoromethyl)phenoxy]pyridin-2-yl]propyl]-6-morpholin-4-yl-3,4-dihydroisoquinolin-1-one N-cyclopropylsulfonylspiro[4,5-dihydrothieno[2,3-c]pyran-7,1'-cyclopentane]-3-carboxamide 4-(cyclopentylmethoxy)-3-hydroxy-1,7-dioxopyrrolo[2,3-d]pyrimidine-6-carboxylic acid 5-[2,6-difluoro-4-(methoxymethyl)phenyl]spiro[1H-indene-3,2'-cyclohexane] (2S)-2-methyl-N-[[4-(3-methylpyridin-4-yl)phenyl]methyl]piperidine-1-carboxamide (1R,3S)-N-[2-amino-5-[4-(difluoromethoxy)phenyl]-6-methylpyrimidin-4-yl]-2,2-dimethylcyclopentane-1-carboxamide;formic acid 5-[2-cyclopentylethoxy(2,6-difluorophenyl)phosphanyl]-1H-pyrazole-4-carbonitrile 6-(difluoromethoxy)-1H-indole N-[1-(4-methoxyphenyl)ethylideneamino]acetamide (3E)-4-amino-3-[(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yloxymethyl)imino]azete-2-thione 5-(3,4-dihydro-2H-chromen-6-yl)-1,2-oxazol-4-amine 6-[2,4-bis(trifluoromethyl)phenyl]-5-N-[1-[5-chloro-6-(3,4-dihydro-2H-pyridin-1-yl)pyridin-3-yl]ethenyl]-7-methoxy-3-(oxan-4-yl)pyrazolo[1,5-a]pyrimidine-5,7-diamine;ethane (2R)-2-[6,7-dichloro-4-[3-fluoro-5-(hydroxymethyl)phenyl]quinazolin-2-yl]sulfanylpropanedioic acid 5-methyl-2-(2H-triazolo[4,5-b]pyridin-6-ium-3-ylidene)pentanamide 3-chloro-N-[1,3,4-oxadiazol-2-yl(phenyl)methyl]-5H-pyrrolo[3,2-d]pyrimidin-6-imine (NE)-N-[amino-(4-chloro-3,5-dimethylpyrazol-1-yl)methylidene]nitramide 4-(1,3-dioxan-2-yl)-N-[2-[2-(1H-imidazol-5-ylmethoxy)ethyl]phenyl]benzamide 3-[3-(1,2-difluoroethyl)phenyl]-4H-1,2,4-oxadiazol-5-one 3-azido-2-(2,4-dimethoxyphenyl)oxane 4-[(Z)-1-cyanopent-2-en-3-yl]-N-(2-methoxyphenyl)benzamide 2-[(4-aminophenyl)methyl]-1,3-thiazole-4-carboxylic acid 2,6-dimethyl-4-[4-[(3E)-penta-1,3-dien-3-yl]phenyl]phenol N-[5-(3,4-dimethoxyphenyl)-1H-pyrazol-3-yl]-7-methylthieno[2,3-d]pyridazine-6-carboxamide 6-[(1S)-1-methoxyethyl]-2,3-dihydrofuro[3,2-c]pyridine 2-(3-acetylcyclohexa-1,5-dien-1-yl)-N,N-bis[1-(cyclohexylmethyl)pyrazol-4-yl]acetamide (5R,7S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2,7-difluoro-6,9-diazatetracyclo[8.8.0.02,7.012,17]octadeca-1(10),11,13,15,17-pentaene-16-carboxamide 3-[4-amino-2-[(1S)-6-ethoxycarbonyl-7-methyloctan-5-ynyl]-6-oxo-1H-pyrimidin-5-yl]propanoic acid 6-[(1R)-1-azidobutyl]-2,3-dihydrochromen-4-one N-[6,7-bis(4-chlorophenyl)quinoxalin-2-yl]hydroxylamine [5-chloro-2,3-di(propan-2-yl)phenyl]boronic acid (2R,3S,4S)-3-amino-4-[[(2R)-5-amino-2-methyl-4-oxopentanoyl]amino]-4-phenylbutanoic acid 2-[(E)-but-1-enyl]-5,6-diethylpyridine;6-propan-2-ylidenecyclohexa-2,4-diene-1-carboxylic acid 3-[(4,6-dimethylpyrimidin-2-yl)amino]benzamide N-[(E)-(3,5-dichloro-2-hydroxyphenyl)methylideneamino]-5-nitrofuran-2-carboxamide N-[6-chloro-1-(cyclopropanecarbonyl)indol-3-yl]acetamide 1-[2-(3,4-dimethoxyphenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]propan-2-one 4-(4-chloro-2-methoxyanilino)-6,7-diethoxy-1H-quinazoline-2-thione [3-(hydroxymethyl)-1,2,4,9-tetrahydrocarbazol-1-yl]azanide 2-[3,5-bis(trifluoromethyl)phenyl]ethanol;N,N'-diaminoethane-1,2-diamine 2-[3-(difluoromethoxy)anilino]-5,7-dihydrocyclohepta[d]pyrimidin-6-one 4-[7-(2-methyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl)-9-oxoindeno[2,1-c]pyridin-10-yl]benzonitrile N-(4,6-dimethylpyrimidin-2-yl)sulfanyl-3-methylazetidine-1-carboxamide 3-[(Z)-1-amino-2-(1,5-dimethylpyrazol-4-yl)ethenyl]phenol 4-[2-methyl-5-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-[1]benzofuro[3,2-d]pyrimidine 1-[2,6-di(propan-2-yl)phenyl]pyrrolidine 2-[3,5-ditert-butyl-4-(methanesulfonamido)phenyl]acetic acid 2-[2-(5,6-difluoropyridin-3-yl)-1H-inden-4-yl]-N-ethylethanamine 1-[(2S,3R)-2-(morpholin-4-ylmethyl)-3-pyridin-2-ylmorpholin-4-yl]ethanone 3-azido-4,5-diphenyl-1H-pyrrole 2-[[1-(2,6-dioxopiperidin-3-yl)-5-methoxy-4-oxo-2H-quinazoline-7-carbonyl]amino]propanoic acid 5-(2,4-difluorophenyl)pent-3-ynylboronic acid 5-(2,4-difluorophenyl)-6-methylsulfonylimidazo[1,5-a]pyridine 1-(4-chlorophenyl)sulfonyl-5-methoxy-3,6-dihydro-2H-pyridine 5-amino-N-methyl-6-[3-[(E)-2-phenylethenyl]quinoxalin-5-yl]hexanamide;ethane 4-[2-(4-chlorophenyl)-1,3-thiazol-5-yl]pyridine-2-carbonitrile (2S,4R)-N-[(Z)-(3-ethoxy-4-hydroxyphenyl)methylideneamino]-1-(4-fluorobenzoyl)-4-methylpyrrolidine-2-carboxamide 1-[(5S)-5-[3-[4-(7-chloroquinazolin-4-yl)piperazin-1-yl]propoxy]piperidin-2-ylidene]ethanol 2-(2,4-difluorophenoxy)-N'-hydroxypyrimidine-4-carboximidamide 4-chloro-1,2-difluorobenzene;N-[5-[(Z)-1-methylsulfanylprop-1-enyl]pyridin-3-yl]cyclopentanecarboxamide 3-[(2-azidooxyethylsulfonylamino)methylidene]-5,6-dihydroimidazo[4,5-c]pyridine-7-carboxylic acid 2,6-dichloro-3,4-bis(trifluoromethyl)pyridine 3-[5-(2,6-dimethylphenyl)pyrimidin-4-yl]phenol N-[1-[(4-chlorophenyl)methyl]benzimidazol-2-yl]carbamate 1-N,3-N,6-trimethylbenzene-1,3-diamine;1H-pyrrolo[2,3-c]pyridine-5,7-diol 3-[2-chloro-4-(8,9-dihydroxy-7-methylnonoxy)phenyl]propanoic acid 2-[2,4-dimethyl-5-(1H-pyrazol-4-yl)phenyl]acetic acid 4-[2-(3,5-ditert-butylphenyl)propan-2-yl]phenol [2-ethyl-4-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]urea (3R,5S)-N-[4-chloro-2-methyl-6-(propanoylamino)phenyl]-7-(3-fluorophenyl)-5-methyl-1-benzothiophene-2-carboxamide (3R,5S)-2-[6-fluoro-7-(8-methylnaphthalen-1-yl)-4-morpholin-4-ylpyrido[3,4-d]pyrimidin-2-yl]-5-methyloxolane-3,4-diol 2-[(4-amino-1,3-dioxoisoindol-2-yl)methyl]quinoline-8-carbonitrile 2-[4-(cyclopropanecarbonylamino)phenyl]-5,6-difluoroindole-1-carboxamide 4-[1-(2,6-difluorophenyl)ethyl]-5-iodo-N-pyrimidin-2-yl-1,3-thiazol-2-amine 2-azido-1-butan-2-yloxy-4-[(E)-3-chloroprop-2-enoxy]benzene 2-(5-azido-1H-pyrazol-4-yl)-N,N-dimethyl-3H-benzimidazole-5-carboxamide 7-hydroxy-4,5-dimethoxy-2-(3-methylbut-1-ynyl)naphthalene-1,8-disulfonic acid 5-[2-ethyl-4-(methoxymethoxy)phenyl]-N-hydroxypentanamide 5-methyl-N-[1-(1,3-oxazole-4-carbonyl)piperidin-3-yl]-2-pyridin-3-ylpyrazole-3-carboxamide (2S)-3-[[4-[2-[(4-chlorophenyl)methyl]pyridin-3-yl]-1,3-thiazol-2-yl]amino]-1-phenylpropan-2-ol 1-cyclopropyl-6,7,8-trimethoxy-N-(4-methylphenyl)isoquinoline-3-carboxamide 6-[2,4-bis(phenylmethoxy)phenyl]-3H-thieno[3,2-d]pyrimidin-4-one 2,3-dimethyl-7-propanoyl-4H-pyrazolo[1,5-a]pyrimidin-5-one N-[5-(3,3-difluoropyrrolidine-1-carbonyl)-2-methylphenyl]propanamide 4-(3,5-dimethylpyrazol-1-yl)-2-oxo-6-pyridin-2-yl-1H-pyridine-3-carbonitrile N-(3,5-dichlorophenyl)sulfonyl-N-ethyl-2-[4-(3-methoxypropoxymethoxy)phenyl]acetamide 3-[(4R,5S)-2-hydroxy-4,5-dimethylheptan-2-yl]-7-phenylmethoxy-1H-quinoxalin-2-one 4-(2-aminoethyl)-N-azido-1,3-thiazol-2-amine 2-[[6-(4-chlorophenyl)pyridin-3-yl]methoxyimino]butanoic acid N-[2,4-difluoro-3-[(Z)-1,3-thiazolidin-3-yliminomethyl]phenyl]-4-(5-methylpyridin-3-yl)-3-(trifluoromethoxy)benzamide (5R)-1,4-dimethyl-5-[2-[5-(pyridin-3-ylmethoxymethyl)imidazo[2,1-b][1,3]oxazol-6-yl]ethynyl]imidazolidin-2-one 6-amino-5,5-dimethyl-2,3-dihydroimidazo[1,2-c]quinazoline-8-carboxylic acid N-[4-(1,3,4-oxadiazol-2-yl)phenyl]-2-[(6R)-2-oxo-5-propan-2-ylidene-4,6-dihydroimidazo[1,2-b]pyrazol-6-yl]acetamide 1-[2,4-dichloro-3-(trifluoromethyl)phenyl]propan-1-one 2-[3,4-dihydroxy-5-(2-methylbutanoyl)oxyphenyl]acetic acid (3-phenyl-1,2-oxazol-5-yl)-[4-[4-(trifluoromethoxy)benzoyl]piperazin-1-yl]methanone N-[2-(6-chloropyridin-3-yl)ethyl]-2-iodoacetamide 1-cyclopropyl-6-fluoro-7-[4-(2-fluoroethylcarbamoylamino)phenoxy]-N,2-dimethylbenzimidazole-5-carboxamide 6-N,8-N-diethyl-3H-imidazo[4,5-c]quinoline-2,6-diamine (4R)-6-(4-chlorophenyl)-1,3,4-trimethyl-7H-pyrazolo[3,4-b]pyridine 3-[(2Z)-2,7-dimethylocta-2,6-dienoxy]-4-propanoylbenzaldehyde 2-(2,6-difluorophenyl)-5-[4-hydroxybutyl-[(1S)-1-phenylethyl]amino]-3H-pyrido[2,3-d]pyrimidin-4-one 2-[(3S)-1-[4-(trifluoromethylsulfanyl)phenyl]pyrrolidin-3-yl]acetic acid N-[[4-(trifluoromethyl)cyclohexyl]methoxy]benzenesulfonamide 3-[5-(6-ethylsulfonylpyridin-2-yl)pyridin-2-yl]oxy-N,N-dimethylpropan-1-amine 2-(3,4-dihydropyridin-6-yl)benzene-1,4-dicarboxamide N-[5-(dimethylamino)thiophen-2-yl]sulfonyl-2-(1,3,4-trimethylcyclohexa-2,4-dien-1-yl)acetamide N-[3-(diethylamino)propyl]-5,6-bis(4-fluorophenyl)imidazo[1,2-a]pyridine-8-carboxamide;hydrochloride 3-azido-5,6-dichloro-2-methylimidazo[1,2-a]pyridine 7-hydroxy-2-(4-methylcyclohexa-1,5-dien-1-yl)chromene-6,8-dione (2E)-5-[(4,6-dimethoxypyridin-3-yl)methyl]-N-ethyl-4-methylhepta-2,6-dienamide;ethane;1-methyl-2-[(2Z)-penta-2,4-dienoxy]benzene 4-[[2,5-dimethyl-4-(4-methylphenyl)sulfanylpiperazin-1-yl]sulfinylmethoxy]benzonitrile (5S,7R)-N-[2-(6-bromopyridin-3-yl)ethyl]-7-fluoro-1,5,10,11-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaene-12-carboxamide 1-(4-azidophenyl)sulfonylpiperidine (2E)-2-[[4,6-dioxo-2-(thiophen-3-ylmethylimino)-1,3-thiazinane-5-carbonyl]amino]penta-2,4-dienoic acid 2-(5-aminothiophen-3-yl)sulfonylphenol 1-[4-(3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl)phenyl]ethanone N-[3-(difluoromethoxy)phenyl]-1,2,4-triazol-1-amine 1-[(2,6-dichlorophenyl)methoxy]-2-piperidin-4-ylpropan-2-ol 4-[5-[(3,5-ditert-butyl-4-hydroxyphenyl)methylidene]hepta-1,6-dien-2-yl]benzenesulfonamide (NE)-N-[6-amino-3,3,5-trimethyl-1-[2-[4-(trifluoromethoxy)phenyl]ethynyl]hexan-2-ylidene]hydroxylamine [(3Z)-4,5,5,6,6,7,7,8,9,10,11,12,12a-dodecafluoro-2-methoxydeca-1,3,7,9-tetraenyl]benzene 5-(5-chloro-3-propan-2-ylimidazo[1,2-a]pyridine-2-carbonyl)-4-methoxy-N-methyl-N-(oxolan-2-ylmethyl)pyridine-2-sulfonamide (4Z)-2,5-diphenyl-3H-1,3-oxazole N-cyclopentyl-1H-indazol-6-amine N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-propanoylpyrrolidine-1-carboxamide 1-(5-cyanopyridin-2-yl)-3-[6-hydroxy-2,4-dioxo-1-[3-(trifluoromethylsulfanylamino)propyl]pyrimidin-5-yl]urea 4-chloro-N,5-dimethyl-N'-(3,3,3-trifluoropropanoyl)pyrazole-1-carboximidamide 2-[(3S)-1-(2,5-difluorobenzoyl)piperidin-3-yl]-7-(pyridine-4-carbonyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 4-[3-(4-fluorophenyl)-2H-imidazol-1-yl]butanenitrile 2-(4-ethylsulfonylphenyl)-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-4-one 6-(4,5-diaminocyclohexa-1,3-dien-1-yl)hexanamide;N-ethylhydroxylamine 5-[(2,4-dimethoxyphenyl)methyl]-1,3,4,6-tetrahydropyrano[4,3-c]pyrazole (2R,4S)-5-hydroxy-N-methyl-2,3,3a,6,7,7a-hexahydrofuro[3,2-b]pyridine-4-carboxamide;2-methoxy-N-phenylacetamide [6-[5,8-bis(ethenyl)naphthalen-1-yl]oxyhexyl-methylamino]phosphonic acid 5-[(1R)-1-[[4-[6-amino-2-methylsulfanyl-7-oxopyrido[2,3-d]pyrimidin-8-yl]cyclohexanecarbonyl]amino]ethyl]-N-phenylpyridine-3-carboxamide 4-[(4-amino-2-chlorophenyl)iminomethyl]-5-ethoxy-1,3-dihydroimidazole-2-thione (1R)-N-[5-cyano-4-methyl-2,6-dioxo-1-[3-(trifluoromethoxy)phenyl]pyridin-3-yl]-1,2,3,4-tetrahydronaphthalene-1-carboxamide 1-amino-N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-2-ylmethyl)cyclohexane-1-carboxamide 4-(4-butylpiperazine-1-carbonyl)-2,3-dimethyl-N-phenylbenzenesulfonamide 3-amino-2-(1,4-dioxaspiro[4.5]decan-8-yl)benzoate N-[(3R,4S)-1-[2-methyl-6-(1H-pyrazol-4-ylamino)pyrimidin-4-yl]piperidin-4-yl]propane-1-sulfonamide N-[1-(4-methoxyphenyl)pyrrolidin-3-yl]-2-(methylamino)thieno[3,2-d]pyrimidine-4-carboxamide 1-[2,3-dibromo-5-(2-nitrophenyl)imidazol-4-yl]-N-methylmethanimine 1-[4-[6-fluoro-3-[(2R,6S)-1,2,6-trimethylpiperidine-4-carbonyl]quinolin-4-yl]-2,5-diphenylpyrazol-3-yl]butane-1,3-dione 1-[3-(2,2-difluorocyclopropyl)phenyl]pyrazole 2-[[4-[(3S)-1,3-dimethylcyclohexa-1,5-dien-1-yl]-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]furan-3-carbonitrile N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-[[2-hydroxyethyl(methyl)sulfamoyl]amino]benzamide 4-[(E)-3-fluorobut-2-enoxy]-1,5-dihydropyrrolo[3,2-c]quinoline 2-[3-(4-methoxyphenyl)propanoylamino]-4,5-dihydro-1H-imidazole-5-carboxylic acid 3-chloro-N-[2,4-di(propan-2-yl)phenyl]benzamide (2R,3S)-2-[3-(7H-benzo[d][1]benzazepin-6-ylmethoxymethylamino)propyl]piperidine-3-carboxylic acid 1-benzyl-3,4-dihydro-2H-1,6-naphthyridine 4-[(Z)-[4,6-dioxo-2-sulfanylidene-1'-[3-(trifluoromethyl)phenyl]spiro[5.5]undecane]-3-ylidene]methyl]benzoic acid 5-[3-(tert-butylamino)sulfanylphenyl]-2,4-dimethyl-1H-pyrimidin-6-one 1-azido-3-(6-chloropyrimidin-4-yl)indole 3,5-dihydroxy-2-propoxybenzenesulfonic acid 3,5-dichloro-N-(2-fluorophenyl)sulfanylaniline 3-[5-(dimethylamino)naphthalene-1,2-diylidene]indol-4-amine 2-(N-methylanilino)ethanol;(E)-3-[2,4,6-tris(trifluoromethoxy)phenyl]prop-2-enal 2-[4-bromobutan-2-yl(pyridin-3-yl)amino]ethanol [2-(3-fluorophenyl)pyrrolidin-1-yl]-[4-[4-[4-(hydroxymethoxy)phenoxy]cyclohexa-1,5-dien-1-yl]piperazin-1-yl]methanone 4-[(2S)-butan-2-yl]-5-[2-chloro-6-methoxy-4-(1,1,2,2,3,3-hexafluoropropyl)phenyl]-N-cyclohexyl-1-ethylpyrazole-3-carboxamide 5-(azepane-1-carbonyl)-2-[2-(2,3-dihydro-1H-inden-4-yloxymethyl)phenyl]benzamide 2-[(4-methylbenzoyl)amino]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxylate 1-methyl-N-[2-(5-phenyl-1,3-oxazol-4-yl)ethyl]pyrazole-3-carboxamide [(2S)-1-[4-(5-fluoropyridine-3-carbonyl)piperazin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamic acid (4Z)-2-phenyl-3,6-dihydrocycloocta[d]pyrimidine 4-[[[(1R)-1-phenylethyl]amino]methyl]benzamide N-[(E)-1-[3-chloro-4-(3,3-dichloroprop-2-enoxy)phenyl]ethylideneamino]acetamide 4-[6-methylsulfanyl-2-(2,3,4,5-tetrahydropyrido[1,2-a]benzimidazol-7-ylamino)pyrimidin-4-yl]benzonitrile 3-[4-chlorobutyl(2,2-dimethoxyethyl)amino]phenol 7-[2-(2,6-dimethylmorpholine-4-carbonyl)phenyl]-N-ethyl-5H-pyrrolo[3,2-d]pyrimidine-4-carboxamide 1-[(4-chlorocyclohexa-2,5-dien-1-ylidene)methylsulfonylmethyl]-3-phenylurea [6-amino-2,3-dihydroxy-5-(4-methylphenyl)phenyl]-phenylmethanone 2-(3,4-dimethylphenyl)-6-[[5-methyl-1-(4-nitrophenyl)pyrazol-4-yl]methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 5-[3,3-bis(sulfanyl)propoxy]-1H-benzimidazole 4-ethenyl-1,2-dimethoxybenzene;(Z)-3-[6-(2-phenylethynyl)quinolin-5-yl]prop-2-enethial N'-[amino(methyl)amino]-5-[(2,4-dichlorophenyl)sulfonylamino]pyridine-2-carboximidamide 1-[(3S)-7-bromo-2,3-dihydro-1-benzofuran-3-yl]-N-butoxy-N-methylmethanamine;ethane N-[6-(1,4-diazepane-1-carbonyl)pyridin-2-yl]cyclopropanecarboxamide 1,5-dimethoxy-2-[(4-methylsulfonylphenyl)methyl]-3-propan-2-ylbenzene 4-(1,2,3,5,6,7-hexahydropyrrolizin-8-yloxy)benzaldehyde 2-(N-octyl-4-phenoxyanilino)decanoic acid N-[(2R,3R)-1-[3-fluoro-4-(2-oxopyridin-1-yl)phenyl]-4-[(4-methylphenyl)methoxy]-5-oxo-2-phenylpyrrolidin-3-yl]-4-(trifluoromethoxy)benzenesulfonamide (4S)-2-amino-9-[2,3-bis(ethenyl)naphthalen-1-yl]-3,4-dihydropyrido[1,2-a]pyrazine-1,6-dione 3-bromo-2,6-dichlorobenzenesulfonamide 1-(6,8-dichloronaphthalen-2-yl)ethanone 4-[2,6-difluoro-4-(1-phenylbutyl)phenyl]-N'-hydrazinylidenebenzenecarboximidamide N-[1-(2,6-dimethylphenoxy)-4H-pyrimidin-5-ylidene]nitramide 2-[(1-acetylpiperidin-4-yl)amino]-3,5-dichloro-N-(4-methylphenyl)benzamide 2-[3-(5-chloro-2-methoxyphenyl)pyrazol-1-yl]propanenitrile 1-ethyl-7,12-diphenylphenanthridine N-[2,3-di(propan-2-yl)phenyl]imino-4-hydroxy-5,6-dihydro-1H-indole-2-carboxamide 2-bromo-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N-propylbenzamide N-[1-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-yl)cyclobutyl]-5,6,7,8-tetrahydroquinoline-8-carboxamide N-[3-(4-chlorocyclohexa-1,5-dien-1-yl)phenyl]methanimine 3-[4-bromo-2-fluoro-5-(2,2,2-trifluoroethoxy)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 3-(2,4-dimethylphenyl)-1,3-oxazolidine 2-[4-azido-5-(2,3-dihydropyridin-6-yl)furan-2-yl]ethanamine 6-[(2,5-dihydroxyphenyl)methyl]-2-pyridin-4-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-[4-(5,7-dimethoxyquinazolin-4-yl)pyrazol-1-yl]-3-fluorophenol 5-(9H-fluoren-1-yl)oxane-2,6-dione 1-[(2E,4Z)-4-methylhepta-2,4,6-trien-3-yl]-4-pyridin-4-ylpiperazine 2-[(1S)-5,7-dimethoxy-2,3-dihydro-1H-inden-1-yl]acetic acid N-(3,5-dimethylphenyl)-2-[(4-oxo-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-2-yl)sulfanyl]propanamide 5-(azidomethyl)-1,2-diethoxynaphthalene N-[2,5-diamino-1-(4-chlorophenyl)sulfanylpyrrol-3-yl]-4-methylbenzenesulfinamide 1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-2-carboxylic acid 1-ethenyl-3-[2-(4-pentan-2-ylphenyl)propan-2-yl]benzene N-benzyl-4-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]piperazine-1-carboxamide 1-[3,6-bis(trifluoromethyl)carbazol-9-yl]butan-2-one 2-(5-chloro-1,3-dimethylpyrazol-4-yl)-6-fluoro-3H-pyrrolo[3,2-c]pyridine 2-[(Z)-2-(1,3-benzodioxol-5-yl)ethenyl]-4-butyl-6-methoxypyrimidine 2-[[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]methylidene]propanedinitrile 2-azido-N-benzylpyrimidine-4-carboxamide 2-(4-chloroanilino)-N-[(E,3R)-6-hydroxy-1-hydroxyhex-5-en-3-yl]acetamide;ethane 1-[2-methyl-4-(2,3,5-trimethoxyphenyl)sulfanyl-3H-thiadiazol-5-yl]ethanone 2-[[7,8-dimethyl-3-(1-phenylcyclopropyl)imidazo[1,5-a]pyridine-6-carbonyl]amino]ethanesulfonate N-(4,5-difluorocyclohexa-1,3-dien-1-yl)sulfonyl-2-[6-methoxy-2-methyl-4-(pyridin-2-ylamino)benzimidazol-1-yl]acetamide 3-(4-fluorophenyl)-5,6-dimethyl-2H-furo[2,3-d]pyrimidine 2-[1-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]cyclopropyl]ethanesulfonamide 6-(1-benzylpiperidin-4-ylidene)pyridine-2,5-dione 2-[5-(methylsulfonylcarbamoylamino)indol-1-yl]acetamide 3-ethenyl-2,4,5,6-tetramethylbenzenesulfonate 2-[4-chloro-3-(cyclopropylmethoxy)phenyl]-6-(difluoromethyl)pyridine (4-methoxyphenyl)-[4-[3-(5,6,7,8-tetrahydroquinolin-2-yl)propyl]piperazin-1-yl]methanone 4-(2-hydroxyethyl)benzohydrazide;[[6-methyl-5-[(3E,5Z)-octa-1,3,5,7-tetraen-4-yl]pyridin-2-yl]amino]methanol 3-(2-methylcyclohexanecarbonyl)benzenesulfonamide 2-[4-(3,5-dimethylphenyl)piperazin-1-yl]-N'-hydroxypyrimidine-4-carboximidamide 3-[2-(1,4-dioxan-2-yl)ethoxy]-5-ethylbenzoic acid N-(2,6-dimethoxypyrimidin-4-yl)-4-[ethylsulfonyl(propyl)amino]benzenesulfonamide 1-(4,6-diphenylpyridin-2-yl)-5-ethoxycarbonylpyrazole-3-carboxylic acid 3-[4-(cyclopropylmethoxy)phenyl]pyrazine 4-N,6,6-tributyl-2-N,7-N-bis[(2S)-butan-2-yl]benzimidazole-1,2,3,7-tetramine 2-[3-methylbutyl(pyridin-2-yl)amino]decanoic acid N-[3-fluoro-4-(pyridine-2-carbonyl)phenyl]formamide 3-[(4-propan-2-ylphenyl)methyl]benzamide 1,3-di(cyclobutyl)-2-phenylbenzene 6-[(Z)-2,3-difluoro-4-phenylmethoxybut-2-enyl]-1-ethyl-5H-pyrazolo[3,4-d]pyrimidin-4-one 4-[(5,7,9,10-tetraoxo-2H-[1]benzothiolo[6,5-b]quinolin-8-yl)oxymethyl]benzonitrile 2-[6-fluoro-3-(2-piperazin-1-ylethoxy)indol-1-yl]acetaldehyde 1-[3-[(2,5-dichlorophenoxy)methyl]phenyl]pyrrole 3-[4-(pyridin-2-ylmethoxy)phenyl]oxirane-2,2-dicarbonitrile (5Z)-2-imino-1,3-dimethyl-5-[[4-(2-methylpropoxy)phenyl]methylidene]imidazolidine-4,6-dione N'-ethenyl-N-[(4-methoxyphenyl)methylideneamino]-1-(2,3,6-trifluorobenzoyl)piperidine-3-carbohydrazide (2S)-N-[4-(dimethylcarbamoyl)phenyl]pyrrolidine-2-carboxamide 1-azido-4,5,6-triphenyltriazine 2-hydroxy-1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazole-6,7-dione N-[4-(2,6-dimethylmorpholine-4-carbonyl)phenyl]-5-methoxynaphthalene-1-sulfonamide 2-(3,5-ditert-butylphenyl)propan-1-ol N-[4-(3-chlorophenoxy)pyridin-2-yl]-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazin-6-amine 2-bromo-4,5-dimethoxy-N-(3-nitrophenyl)benzenesulfonamide 5-fluoro-2-methoxy-N,4-dimethyl-N-[(1S)-1-pyridin-3-ylethyl]benzamide 2-[4-[(1R,3S)-2,2,3-trimethylcyclopropanecarbonyl]phenoxy]acetate [2-(4-aminobutyl)-1H-imidazol-5-yl]methanesulfonate 4-[2-[[5,6-dimethoxy-3-(1H-pyrazol-4-yl)quinolin-4-yl]amino]ethoxy]benzonitrile 3-[2,4-bis(ethenyl)phenyl]hexanoic acid 6-amino-4-[2,5-dimethoxy-3-(trifluoromethyl)phenyl]-4-methyl-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile 2-[3,5-dichloro-4-(6-methoxynaphthalen-2-yl)phenyl]ethanamine 4-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-N'-[2-[[6-[5-(dimethylamino)-5-oxopentoxy]quinazolin-4-yl]amino]pyridin-4-yl]benzenecarboximidamide 1-(4-chlorophenyl)sulfonyl-2-oxo-5-propan-2-ylpiperidine-3-carboxamide 3-[(2-amino-6,7-dimethoxyquinazolin-4-yl)amino]propanoic acid 2-[6-(cyclohexylmethylamino)pyridin-3-yl]-N-[4-(4-fluorobenzoyl)phenyl]propanamide 4-cyclopropylsulfonylbenzonitrile 1-[3-[2-(dimethylamino)ethoxy]-4-methoxyphenyl]-N',2-dimethyl-N-phenylethenamine;toluene 3-[4-[(3,5-difluorophenyl)methoxy]phenyl]oxirane-2,2-dicarbonitrile 4-methoxy-6,8-dimethyl-1H-quinoline-2,5-dione 2,6-ditert-butyl-4-(10H-phenoxazine-1-carbonyl)phenol 4-[6-(azetidin-3-yloxy)pyridin-2-yl]sulfonyl-2-(2,2,4-trimethylpyrrolidin-1-yl)pyridine-3-carboxamide 2-[4,5-bis(ethenyl)furan-3-ylidene]propanedinitrile (3R)-N'-(2-methylquinolin-4-yl)ethane-1,2-diamine N-(3,4-dichlorophenyl)-5-propanoyl-3,6,7,8-tetrahydro-2H-pyrrolo[1,2-a]pyrazine-1-carboxamide N-[2-amino-4,5-dichloro-3-(pyridine-4-carbonyl)phenyl]benzamide N-(6-chloropyridin-2-yl)-1,5-dimethylpyrazole-3-sulfonamide 1-butyl-3-[4-[2-(4-oxo-7,8-dihydro-6H-pyrrolo[1,2-a]pyrimidin-3-yl)ethynyl]phenyl]urea 2-[3,5-dichloro-4-(4-methylsulfonylphenyl)phenoxy]ethanol 6,8-dihydroxy-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one 2-(1-phenylethyl)-8-[[3-(trifluoromethoxy)phenyl]methyl]-4,5-dihydropyrazolo[1,5-a]quinazoline 1-[3-(2-ethoxyethyl)-4H-quinazolin-6-id-7-yl]-N',N'-dimethylethane-1,2-diamine;uranium(2+) N-[2-(4-amino-6,7-dimethoxyquinazolin-2-yl)sulfanylethyl]-1-azidoethanethiol 3-ethylsulfanyl-N-[2-(4-oxo-5H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl]prop-2-enamide 2-(4,6-dichloropyrimidin-5-yl)oxy-N-ethyl-N-[(3-hydroxyphenyl)methylideneamino]acetamide 3-amino-4-cyano-5-[2,5-dichloro-4-(trifluoromethyl)phenyl]-1H-pyrrole-2-carboxamide 2-(4-benzylphenyl)-1,8a-dihydroquinoxaline 2-[[3-(azidomethyl)azetidin-1-yl]methyl]aniline 2-[4-bromobutan-2-yl(3-methylbutyl)amino]phenol (4E)-1-cyclobutyl-8,9-dimethoxy-3,4-dihydro-2H-pyrido[2,3-b]indole 3-amino-N-[(Z)-3-cyano-4,4,4-trifluorobut-2-enimidoyl]benzamide 3-benzylsulfanyl-6-[4-(dimethylamino)phenyl]pyridazine-4-carboxamide N-[2-(4-fluorophenyl)ethyl]-1,7a-dihydroindazole-6-carboxamide (2R,3S)-1-[4-methyl-3-(trifluoromethyl)benzoyl]-N-naphthalen-1-ylsulfonylpiperidine-2-carboxamide (2Z,4E)-4-methoxy-N-[3-(trifluoromethyl)phenyl]hepta-2,4,6-trienamide 2-bromo-1,3-dichloro-4-(trifluoromethyl)benzene ethane;5-methyl-4-[3-(3-phenoxypropoxy)propyl]pyrimidine (2S)-1-[[5-[1-[4-(2-methylpropoxy)phenyl]heptan-4-yl]thiophen-3-yl]methyl]pyrrolidine 5-benzyl-N-[(2R)-2,3-dihydroxypropoxy]-6-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-2-carboxamide 6-bromo-3-(4,5,8,14,16-pentazatetracyclo[7.6.0.02,7.010,12]pentadeca-1,6,9,11,13-pentaen-5-ylmethylidene)indole 2,5-diphenylpyrazole;molybdenum(3+);methanol 4-[(2R)-2,4-dimethylpiperazin-1-yl]-10H-thieno[2,3-b][1,5]benzodiazepine;dihydrochloride 1-[2-(4-ethylcyclohexyl)propoxy]-5,6-difluoronaphthalene 2-[3,4-bis(ethenyl)phenyl]-6-methylquinoline 1-azido-3,5-dinitro-2H-indole 1,2-dimethoxybenzene;N-(3,6-dihydro-2H-pyran-4-yl)-2,2-dimethylbutanamide 2-bromo-4-(3,5-dimethylphenyl)butanoic acid 2-[(3R)-1-[2,4-dimethyl-1-[(4-oxo-3H-quinazolin-2-yl)methyl]pyrrole-3-carbonyl]piperidin-3-yl]acetamide 2-[2,6-dibromo-4-(5-methoxypyridine-3-carbonyl)phenoxy]-1-(3-methylpiperazin-1-yl)ethanone (Z)-2,3-dihydroindene;N-[[6-(trifluoromethyl)pyridin-3-yl]methoxymethyl]pyrazin-2-amine 3-(7-oxobenzo[a]phenalen-1-yl)prop-2-enoic acid 4-(3-ethynylanilino)-6-propanoylquinoline-3,8-dicarboxylic acid 5-[4-[[(2S)-3-cyclohexyl-3-methoxy-1-oxopropan-2-yl]carbamoylamino]phenoxy]pyridine-3-carboxamide N-[1-[(4aS)-3,4a,5,6,7,8,8a-octahydro-2H-benzo[b][1]benzazepine-11-carbonyl]cyclopentyl]cyclopropanecarboxamide N-methyl-N-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)phenyl]pyridine-3-carboxamide ethane;1-[(3Z,5E)-2,4,5-trimethylhepta-1,3,5-trien-3-yl]pyrrole 1-[2-(2,4-dichlorophenyl)ethenyl]indazole 4-tert-butyl-2-(4-methylphenyl)pyrimidine 1-(2,3-dihydro-1H-inden-1-yl)naphthalene 3-[(2E)-1,4-diaminopenta-2,4-dienyl]-N-ethylnaphthalene-1-carboxamide 6-methyl-N-[1-(pyridine-2-carbonyl)piperidin-3-yl]pyrimidine-4-carboxamide 2-ethyl-5-[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]pyrimidine-4,6-diamine 3-cyclobutyl-N-[1-[4-(hydroxymethyl)phenyl]ethyl]benzamide N-[3-(2,5-dimethylphenoxy)phenyl]-1H-indole-6-carboxamide 3-methyl-5-[2-(4-methylphenyl)-1,3-dioxan-2-yl]-1-tritylindazole N-[2,3-diamino-5-(trifluoromethyl)phenyl]-4-hydroxybutane-1-sulfonamide 5-(4-phenylbutoxy)bicyclo[2.1.0]pentane 4-[2-(trifluoromethyl)phenyl]sulfonylbenzenethiol 6-(2-chloro-3,5-dimethoxyphenyl)-N-[4-[(1R)-1-ethylcyclopropyl]pyridin-2-yl]pyridine-2-carboxamide 1-azidooxy-4-(2,6-difluorophenyl)benzene 1-[(4R)-3,3-dimethylpiperidin-4-yl]oxy-2H-benzimidazole N-[(5-methoxyfuran-2-yl)methyl]-4,7-dioxo-6-phenyl-2-propylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 3-(azidomethyl)-1H-quinazoline-2,4-dione (4-azido-2,3,5,6-tetrafluorophenyl)methanamine 1-[4,5-dichloro-2-(6-oxopyridazin-1-yl)phenyl]-3-methoxyurea 5-chloro-4-N-[(E)-1,3-diaminoprop-2-enylidene]-6-N-ethylpyridine-2,4,6-triamine (3-ethyl-1H-indol-2-yl)-[4-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridine-2-carbonylamino)phenyl]azanium [5-(2,3-dihydro-1H-inden-5-yl)pyridin-2-yl]urea (4R,5S)-1-benzyl-2,3,3a,4,5,6,7,8,9,10,11a,12b-dodecahydroindeno[2,1-f]indolizine 2-(furan-2-ylmethylimino)imidazolidine-4,5-dione N-[2-(dimethylamino)ethyl]-5,5-difluoro-N-phenylhexanamide (5E)-2-imino-5-[(4-methoxy-3-nitrophenyl)methylidene]-1,3-thiazolidin-4-one [4-amino-2,6-bis(1H-indol-5-yl)phenyl]methanol N-[(Z)-3-aminobut-2-enyl]-2,3-dichloroaniline 4-[2,3-bis(ethenyl)pyridine-4-carbonyl]-1H-pyrazole-5-carbonitrile N-[2-azido-1-(4-pyridin-3-yloxyphenyl)ethylidene]hydroxylamine 2-[(4S,6R)-8-bromo-4-[2-methoxy-3-(2H-tetrazol-5-yl)phenyl]-1-oxo-3,6-dihydro-2H-pyrazino[1,2-a]pyrimidin-6-yl]-N,N-dimethylacetamide 6-[2-(4-butylphenyl)ethynyl]-1-fluoronaphthalene 1-(2,5-difluoro-4-methoxyphenyl)-7-methyl-3-(2-methylpropylamino)-5H-pyrazolo[3,4-d]pyridazin-6-one [4-[3-cyano-6-(2,5-dimethylpyrrol-1-ium-3-ylidene)-4H-pyrrolo[2,3-b]pyrrol-1-yl]phenyl]urea 4-[2-fluoro-6-methyl-5-(2,2,3,3,3-pentadeuteriopropoxy)pyridin-1-ium-3-yl]-N-[(2R)-2-hydroxybutylidene]-2-propan-2-ylbenzenecarboximidate 4-(3,5-dimethylphenyl)imino-5-[2-hydroxy-4-(trifluoromethoxy)phenyl]pyrrolidine-3-carboxylic acid 4-azido-1-(4,6-dimethylpyrimidin-2-yl)azepane N-[4-(2,3-dihydropyridin-6-yl)phenyl]-1,3,5-trimethylpyrazole-4-carboxamide 2-[5-(4,6-diphenylpyrimidin-1-ium-2-yl)pyridin-3-yl]-9,9-dimethylfluorene 3-(1,5,7a-trimethyl-2-oxo-3,4,7,8,9,10-hexahydropyrimido[4,5-b]quinolin-6-yl)propanoic acid 2-[(1R,5S)-3-acetamidobicyclo[3.1.0]hexanyl]-N-methylidenebenzamide 1-(5,6-dichloro-2-methylpyrimidin-4-yl)-7-methoxy-2H-quinoline 5-bromo-3,3a-dihydro-2H-pyrazolo[1,5-a]pyrimidine;hydrochloride (2-benzylpiperidin-1-yl)-phenylmethanol (2S)-3,4-dihydro-2H-chromene;ethane 1-[2-methyl-4-[(1,5R)-3-oxabicyclo[3.1.0]hexan-6-yl]phenoxy]-2-[2-(trifluoromethoxy)phenyl]ethanone N-(2,6-dichloro-4-nitrophenyl)-2,4,6-trimethyl-N-prop-2-enylbenzenesulfonamide N-cyclohexylacetamide;4,4,5,6,7,8,9-heptamethyl-2,3-dihydrochromene [6-(methoxymethyl)-2,2-dimethylmorpholin-4-yl]-(3-propan-2-yloxyphenyl)methanone (3R)-N-[2,6-difluoro-4-(1H-pyrazol-5-yl)phenyl]morpholine-3-carboxamide 7-chloro-1,2,3,4,5,6-hexahydro-[1]benzothiocino[5,4-d]pyrimidine N-ethylformamide;2-[(3R)-1-[3-[[(5Z,8E,11Z,14Z,17E)-icosa-5,8,11,13,15-pentaenoyl]amino]propanoyl]pyrrolidin-3-yl]oxy-6-methylpyridine 5-(cyclohexylmethoxy)quinazoline N-[3-[2-(4-fluorophenyl)ethenyl]thiophen-2-yl]-N',N'-dimethylpropane-1,3-diamine (5E)-2-cyclopentylimino-5-[[5-(dipropylamino)furan-2-yl]methylidene]-1,3-thiazolidin-4-one 1-[4-amino-6,7-dichloro-8-(2,3-dimethoxyphenyl)pyrimido[5,4-b]pyrrolizin-9-yl]ethanone 2-amino-3-[4-[(4,4-difluorocyclohexyl)methoxy]naphthalen-1-yl]propanoic acid 3-[(4S)-1-(1,3-benzodioxol-5-ylmethyl)-2',6-dioxospiro[3H-pyrido[2,3-b][1,4]thiazine-4,3'-pyrrolidine]-4-yl]-N,N-diethylpropanamide 4-[4-[(Z,3S)-3,5-bis(hydroxymethyl)hex-4-enoxy]phenyl]phenol N-[2,3-dihydroxypropyl(1,2,4-triazol-4-yl)amino]benzenesulfonamide 4-[(E)-2-aminooxy-1-fluoroethenyl]aniline 2-[4-[3-[(E)-2-[7-chloro-1,8-naphthyridin-2-yl]ethenyl]phenyl]cyclohexyl]propan-2-ol N-[3-(dimethylamino)propyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane-2-carboxamide 4-(3,4-dichlorophenyl)-2H-1,2,5-oxadiazol-3-one 2,4-ditert-butyl-6-(1H-imidazo[1,2-a]benzimidazol-9-yl)phenol 5-[2-(3,4-dimethylphenyl)pyrrolidine-1-carbonyl]-N-piperidin-4-yl-N-propan-2-yl-2,3-dihydroindole-1-carboxamide N-(2,5-dichlorophenyl)-2-[6-ethyl-7-(4-methoxyphenyl)-2-oxo-1,3-dihydroimidazo[1,2-b]pyrazol-3-yl]acetamide 3-[(1S)-1-aminoethyl]-5-(2,4-dichlorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine 6-(3,4-dichlorophenyl)-5,8-dihydropyrimido[4,5-d]pyrimidine-7-thione 1,3-dibromo-5-(4-tert-butylcyclohexa-2,4-dien-1-yl)benzene N-[6-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]hexan-2-yl]-2-(trifluoromethoxy)benzamide [4-(4-carbamoylpyridin-2-yl)oxynaphthalene-1-carbonyl]oxidanium 2-[1,3-benzodioxol-5-ylmethyl(propan-2-yl)amino]pyrimidine-4-carboxylic acid N-[2-bromo-6-(4,5-dimethyl-1H-imidazole-2-carbonyl)phenyl]acetamide 4-[(2,3,3a,8b-tetrahydro-1H-cyclopenta[b]indol-6-ylamino)methyl]benzoic acid [2-azidooxysulfanyl-1-[4-(trifluoromethyl)phenyl]ethyl]benzene 4-[(3S)-3-aminopiperidine-1-carbonyl]-3,5-dimethylthiophen-2-ol;hydrochloride N-[4-(5-chlorothiophen-2-yl)sulfonyl-1,4-thiazepan-6-ylidene]hydroxylamine N-[(2S)-1-cyclohexa-1,5-dien-3-yn-1-ylpropan-2-yl]-N-methyl-5H-pyrazolo[3,4-d]pyrimidine-4-sulfonamide 3-[2,5-dihydroxypentyl(ethyl)amino]-5-nitro-6-phenyl-1H-pyridin-2-one 3-ethoxycarbonylnaphthalene-1,6-dicarboxylic acid 6-[3-(2,5-difluorophenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]spiro[3.4]octane-7-carboxylic acid 6-(2,5-dimethoxyphenyl)-3-[2-fluoro-4-(2,2,6,6-tetramethylpiperidin-1-ium-1-yl)anilino]pyrazine-2-carboxamide 2-[2,4-difluoro-3-(propan-2-ylsulfonylamino)phenyl]acetamide [4-(1H-pyrazol-5-ylmethylideneamino)phenyl]methanamine 4-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-nonanoylamino]benzenesulfonic acid 5-[[4-fluoro-3-methoxy-2-(trifluoromethyl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione (2S)-3-methoxy-1,2-diphenylpropan-1-one 2-[4-fluoro-3-(trifluoromethyl)phenoxy]phenol N-butyl-4-[2-hydroxyethyl(2,3,5,6-tetrafluorophenoxy)phosphoryl]oxyoxyaniline (Z)-2-(4-butoxy-3,5-dimethylphenyl)sulfonylpent-2-enedioic acid N-[3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)propyl]acetamide 3-[4-(benzylamino)-3-fluorophenyl]propanal;2,2,2-trifluoroacetaldehyde (4-azidooxy-3-cyclopropylphenyl)methanamine 2-[(3Z)-6-chloro-2,5-dimethylhexa-1,3,5-trien-3-yl]oxyacetic acid;6-[[4-fluoro-3-[4-(trifluoromethoxy)phenyl]phenyl]methyl]-7H-pyrrolo[3,4-b]pyridin-5-one 5-[3-methylbut-2-enyl(1,3-thiazol-5-yl)amino]-1H-pyrimidine-2,4-dione 2-bromo-5-[1-(methoxymethyl)cyclobutyl]pyrazine N-(2,5-dimethylphenyl)-4-methoxy-6-methylcyclohexa-1,3-diene-1-carboxamide 1-[4-[(2-bromophenyl)methoxy]phenyl]-N,N-diethylpyrrolidine-3-carboxamide 3-(6,7-dihydroxyquinolin-4-yl)oxybenzamide (4aR,8aS)-N-[2-chloro-5-(2H-tetrazol-5-yl)phenyl]-1-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-2-carboxamide (NZ)-N'-[3-(4-methoxyphenyl)-1,2-dihydropyrido[1,2-a]benzimidazol-4-ylidene]-N'-methylethane-1,2-diamine 2-[(E)-3-[amino(methyl)amino]prop-1-enoxy]-6-[4-(trifluoromethyl)phenyl]cyclohexan-1-one 3-(5,6-dihydroisoquinolin-1-yl)benzamide 1-[4,5-difluoro-2-(triazol-2-yl)benzoyl]-N-propan-2-ylpiperidine-3-carboxamide (5R)-3,3-dimethyl-5-[2-[4-(3-propan-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-2-one 5-bromo-2,3,4-trimethyl-1H-indole 4-[3-(1,1-dioxothiolan-3-yl)-5-methoxycarbonylphenyl]-2,6-difluorobenzoic acid 4-(1H-indazol-5-yl)-N,N-dimethylbenzamide 2-[(3S)-1-benzylpyrrolidin-3-yl]imino-5-methyl-3-[(4-nitrophenyl)methyl]-6H-pyrimidin-4-one 7-chloro-N-(1H-indazol-3-yl)imidazo[1,2-a]pyridine-5-carboxamide 3-[4-(2,6-dimethoxyphenyl)phenyl]oxirane-2,2-dicarbonitrile 2-[4-(aminomethyl)phenyl]-6-thiophen-3-ylpyridazin-3-one 2-[4-(4,7-dimethylnaphthalen-1-yl)oxybutoxy]ethanol 5-ethylsulfinylpyridine-2,3-diamine 5-(3-bromo-2H-indazol-4-yl)-3,6-diethylpyrazine-2-carboxamide 2-[(7R)-5-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-7-yl]pyridine-3-carbonitrile;N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]formamide 6-[2,4-difluoro-N-(3-methylbutyl)anilino]sulfanyl-5H-furo[3,2-b]pyridine-7-carbonitrile 2,3-dimethylpentanoic acid;ethane;7-(8-ethyl-7,9,10,11-tetrahydronaphtho[2,1-g][1]benzofuran-2-ylidene)-5-methyl-4H-tetrazolo[1,5-a]quinoline 4-[(1R,2R)-2-hydroxycyclopentyl]sulfanyl-N'-hydroxybenzenecarboximidamide 3-[6-[1-(7H-purin-6-ylamino)ethyl]pyrazin-2-yl]benzenecarboximidamide 4-amino-2-[4-[(1E,3Z)-1-(methylideneamino)penta-1,3-dienoxy]anilino]pyridine-3-carboxylic acid 2-(4-methylthiophen-3-yl)-5,6,7,8-tetrahydroquinazoline 2-[4,6-difluoro-5-(6-methylpyridin-3-yl)-1H-benzimidazol-2-yl]-5-methoxyphenol (3R)-N-cyclopentyl-4,7,8,10-tetrazatricyclo[6.4.0.02,6]dodeca-1,6,9,11-tetraen-3-amine;dihydrochloride 2-[4-(azidomethyl)phenyl]-5,6-dimethoxy-1H-benzimidazole 5-[(3-chlorophenyl)methyl]-N,6-dimethylthieno[2,3-d]pyrimidine-4-carboxamide 3-(4-oxo-1,2,5,6-tetrahydrobenzo[h]quinolin-9-yl)propanoic acid 3-[2,6-di(propan-2-yl)phenyl]-1-phenyl-2H-imidazole 4-[3,5-bis(trifluoromethyl)phenyl]-2-chlorobenzoic acid [2-[(6-bromopyridin-3-yl)methylidene]-4,5-dihydroxyfuran-3-ylidene]oxidanium 4-amino-6-(2,2-diphenylethoxy)quinoline-3-carbonitrile N-[(3R)-1-(azetidine-1-carbonyl)piperidin-3-yl]-5-chloropyridine-2-carboxamide 4-[3-(2,6-difluorophenyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylaniline (E)-3-[1-[2,5-difluoro-4-(trifluoromethyl)phenyl]-4-oxopyridazin-3-yl]prop-2-enoic acid 3-[4-(dimethylamino)phenyl]-5,6,7,8-tetrahydro-1H-quinoline-2,4-dione N-(4,6-dimethylpyrimidin-2-yl)-4-[1,3-thiazol-5-yl(2H-tetrazol-5-yl)amino]benzenesulfonamide 3-[3-[(3,4-difluorophenyl)methyl]-2-oxoimidazolidin-1-ium-1-yl]benzoic acid 2-(3,4-dichlorophenyl)imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one 5-[3,4-dihydroxy-6-(methylamino)oxan-2-yl]-2,8-dimethylbenzo[e][1,2,4]triazine-6,7-dione N-[5-(7-cyanoquinolin-4-yl)oxypyridin-2-yl]cyclopropanecarboxamide 5-methoxycarbonyl-4-[3-oxo-2-(1H-pyrrol-2-yl)-3a,6a-dihydro-1H-pyrrolo[3,4-c]pyrazole-5-carbonyl]furan-2-carboxylic acid N-[(4-methoxyphenyl)methyl]-2,3-dihydroimidazo[1,2-b]pyrazole-6-carboxamide 5-chloro-2,3-dimethoxy-1H-indole;hydrochloride 1-[(2E,4Z)-2-methylhexa-2,4-dienyl]-2-[1-(4-methylphenyl)ethylidene]hydrazine [4-(7,8-dihydronaphthalene-1-carbonyl)morpholin-2-yl]methanone 1,2-dichloro-4-[(Z)-3-methylpent-2-en-2-yl]benzene;ethane [2-(2,3,4,5-tetrafluorophenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]methanamine 1-[2-(cyclopropylmethoxy)-5-fluoropyridin-3-yl]propan-2-ol 2-[[1-(4-methylphenyl)sulfonylpiperidin-3-yl]methoxy]pyridine [3-[1,5-dimethyl-2-(trifluoromethyl)indol-6-yl]propanoylamino]carbamodithioic acid 3-(7,8-dihydrodibenzofuran-4-yl)-2H-1,3-thiazole 3-(4-chlorophenyl)-1-methyl-2-oxopyrrolidine-3,5-dicarboxamide 5-amino-4-[3-(cyclopropylmethoxy)phenyl]-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione 5-(3,4,6,7,8,9,9a-hexahydro-1H-pyrido[2,1-c][1,4]oxazin-3-ylsulfonyl)-N-ethylfuran-2-carboxamide 6-chloro-N-ethylnaphthalene-2-carboxamide 1-amino-4-benzylidene-3H-quinoline-2,6-dione (E)-N-[2-methyl-1-[4-(6,7,8,9-tetrahydro-5H-pyrido[3,2-b]indol-10-yloxy)butanoylamino]propylidene]-6-thiophen-2-ylhex-4-enamide 3-(6-methoxynaphthalen-2-yl)-4-[(5R)-5-methyl-1H-pyrazol-4-yl]butanoic acid N-[2,4-difluoro-3-[7-(thiophen-2-ylmethylamino)quinazolin-2-yl]phenyl]propane-1-sulfonamide 1,3-dichloro-5-(fluoromethyl)benzene;N'-(2-methoxyethanimidoyl)-4-[methyl(oxolan-3-yl)amino]benzenecarboximidamide 1-[4-(6-aminohexyl)phenyl]propan-2-ol 4-[2-(difluoromethoxy)benzoyl]piperazine-1-carboxylic acid (2-methylpyridin-4-yl)-(2-pyridin-3-ylpyrrolidin-1-yl)methanone N'-(3,5-dichlorophenyl)sulfanyl-1H-imidazo[4,5-b]pyridine-6-carboximidamide 2-amino-6-[[2-(4-chloro-3,5-dimethylphenoxy)acetyl]amino]pyridine-3-carboxylic acid (3Z,5E)-4-amino-7-[3-[cyclopropylmethoxy(phenyl)methyl]phenyl]hepta-1,3,5-triene-2,8-dione 4-[1-(2-aminoethyl)piperidin-3-yl]-6,7-dichloroquinoline-5-carbonitrile 6-[2,3-difluoro-4-(2-iodoethynyl)phenoxy]hexanal [5-(4-fluorophenyl)spiro[1H-2-benzofuran-3,3'-azetidine]-1'-yl]-(6-methoxypyridin-3-yl)methanone 3-[6-(5,8-dichloroquinolin-6-yl)cyclodeca-1,4,7,9-tetraen-1-yl]propanal 5-[[5,7-dioxo-6-(4-pyrrolidin-1-ylphenyl)pyrrolo[3,2-c]thiazin-4-ylidene]amino]pyridine-3-carbonitrile 3-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]cyclopentane-1-carboxylic acid 2-[1,3-benzodioxol-5-yl(phenyl)methoxy]-N-methylethanamine [2-(3,5-dimethoxyanilino)pyrimidin-4-yl]urea 6-(3,4-dimethylphenyl)-5-isocyanofuro[2,3-d]pyrimidine 2-[3,5-dichloro-4-(1H-pyrrol-2-yl)phenyl]acetic acid N-[2-chloro-5-(1H-pyrazol-4-yl)phenyl]-3-ethoxy-2-fluorobenzamide 2-[2,6-diethyl-4-(6-methoxypyrimidin-4-yl)piperazine-1-carbonyl]benzonitrile (2R,3S)-1-[2-[4-[2-[ethyl(propan-2-yl)amino]ethoxy]phenyl]-3H-benzimidazole-5-carbonyl]pyrrolidine-2,3-dicarboxylic acid 5-methoxy-4,8-dihydrofuro[3,2-g]chromen-7-one 6-bromo-3H-1,2,4-triazolo[4,3-a]pyridine;difluorobenzene 2-[4-(4-tert-butylphenyl)phenyl]-N,1,3-trimethyl-4H-quinazolin-2-amine 3-(2-chlorophenyl)-4-(4,5-dimethyl-1H-pyrazol-3-yl)morpholine ethane;2-methyl-7,8-dihydro-1H-imidazo[4,5-c]azepine;5-[3-(trifluoromethoxy)phenyl]imidazolidine-2,4-dione 1-azido-4-(2,3-dihydro-1H-indene-5-carbonyl)piperidine-4-carboxylic acid 2-methyl-N-[5-(3-methylphenyl)-3-oxopentanoyl]cyclohexane-1-carboxamide 5-(4-methylpiperazin-1-yl)sulfanyl-2-phenylmethoxybenzaldehyde 5-(9H-fluoren-1-yl)-2,3,4,5-tetrahydrofuran-2-ide;titanium(2+) 2,5-dichloro-N-[4-(1H-imidazol-3-ium-5-yl)butyl]benzenesulfonamide 5-cyclopropyl-3-[1-(2,6-difluorobenzoyl)piperidin-4-yl]oxy-N-methyl-N-phenyl-2H-1,3-thiazole-2-carboxamide 3-amino-N-(7-hydroxyquinazolin-4-yl)propanamide N-[[2-(4-methoxyphenyl)pyridin-3-yl]methyl]-N,6,7-trimethylquinoline-8-carboxamide 1-[1,3-bis(trifluoromethyl)pyrazolo[4,3-c]pyridin-6-yl]-2-[4-ethoxy-N'-[(5Z)-5-ethenyliminocyclopenta-1,3-dien-1-yl]carbamimidoyl]propan-2-one 5-[2-methyl-3-(trifluoromethoxy)phenyl]imidazolidine-2,4-dione 3-[4-(diaminomethylideneamino)phenyl]furan-2-carboxylic acid 1,3-bis(2-methylbutan-2-yloxy)benzene;5,7-dichloroquinoline 5-[(2S,3R)-4-benzoyl-3-methylpiperazin-2-yl]-1-(2-chlorophenyl)pentan-1-one 2-[4,5,6,7-tetrachloro-2-(2-methyloctanoyloxy)quinolin-3-yl]acetic acid 2-(3,5-dihydro-2H-1,4-benzothiazepine-4-carbonyl)-N'-phenyl-1H-imidazole-5-carboximidamide 4-(1H-pyrazol-5-yl)-6,7,8,9-tetrahydro-3H-pyrimido[5,4-b]azepin-2-one (2E)-3,7-dimethyl-6-methylidene-1H-4,8-benzodioxecine 5-chloro-N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2,4-dihydroxybenzamide 2-(3,4-dimethoxyphenyl)-2H-[1,3]thiazolo[5,4-c]pyridine 2-[(2Z)-4-oxo-2-[(E)-(3,5,6-trimethyl-1H-benzimidazol-2-ylidene)hydrazinylidene]-1,3-thiazolidin-5-yl]acetic acid 4-(7,8-dihydroimidazo[1,2-a]pyridin-5-yl)phenol 4-bromo-2,6-dichloro-N-[(1S)-5-(5,7-dimethoxyimidazo[1,5-a]pyridin-3-yl)cyclohexa-2,4-dien-1-ylidene]benzamide 2,6-dibutyl-4-(6-methoxypyridin-3-yl)pyridine 1-[4-(6,7-dimethoxyquinazolin-2-yl)-3-fluorophenyl]-N-[5-[(5-methyltetrazol-2-yl)methyl]pyridin-2-yl]methanesulfonamide 2-chloro-6-[(3R)-2,3-dihydrofuro[3,2-b]pyridin-3-yl]-4-fluorophenol 4-(2,5-dioxopyrrolidin-1-yl)-3-[[4-methoxy-3-[(E)-2-(7H-purin-6-ylamino)ethenyl]benzoyl]amino]benzoic acid 2-(4-butoxyphenyl)-1,3-benzothiazole N-(2-cyanoethyl)-3-[(4,6-dichloropyrimidin-5-yl)amino]benzamide 2-[4,5-bis(ethenyl)pyrazol-1-yl]acetaldehyde 4-(3,5-dimethylbenzenecarboximidoyl)pyridin-2-amine N-[(4-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 4-(3,5-dichloropyridin-2-yl)-N-methanimidoyl-6-[(3R)-3-prop-1-en-2-ylpiperazin-1-yl]pyrimidin-2-amine 6-chloro-3-methyl-4-propan-2-ylchromen-2-one 2-[3-(hydroxymethyl)phenyl]-3,4,6,7,8,9,10-octahydropyrazino[1,2-a]pyrimidin-1-one (4R)-3-[2-(2,6-dimethoxyphenyl)-5-(6-fluoropyridin-3-yl)-1,2,4-triazol-3-yl]-4-(4-hydroxybutylsulfonylamino)piperidine-1-carboxylic acid 5-[2-(3,4-dimethoxyphenyl)ethyl]-2-(dipropylamino)-4H-1,3-thiazole-4-carboxylic acid 2-(3,5-dibromothiophen-2-yl)-7,8-dihydro-6H-pyrido[1,2-a]pyrimidine 1,6-bis(2-methoxyethyl)naphthalene (E)-N-[5-(methoxyamino)-4,5-dihydrothiepin-2-yl]-3-pyridin-2-ylprop-2-enamide 1-[4-(dimethylamino)piperidin-1-yl]-2,3,7-trimethoxyanthracene-9,10-dione N-[(2S)-3-(3,4-dihydro-1H-isoquinolin-2-yl)-2-hydroxypropyl]-6-[2-[5-methanimidoyl-4-(methylamino)-1,3-thiazol-2-yl]ethynyl]imidazo[1,2-a]pyridine-2-carboxamide 3-[2-cyclopenta-1,4-dien-1-yl-5-(2,6-diphenylpyridin-4-yl)-9-methylidenefluoren-3-yl]-5,7-dimethoxyquinoxaline 6-[(3R)-4-azido-3-methylpiperazine-1-carbonyl]-N-tert-butylpyrimidine-4-carboxamide 5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-N-ethyl-2-fluorobenzenesulfonamide 1-(3,4,5-trimethoxyphenyl)heptane-2,3-dione 4-[2-(4-aminophenyl)ethynyl]benzaldehyde 6-cyclobutyloxy-4,5,7-trifluoro-2-(2H-tetrazol-5-yl)benzimidazole (5R)-5,7-dimethyl-2-[2-[3-(4-methylpiperazin-1-yl)phenyl]ethynyl]-N-(oxan-4-yl)-6H-indolo[2,3-b]quinoline-9-carboxamide 3-[2-(4-ethylphenyl)ethenyl]-5,6,7,8-tetrahydrocyclopenta[b]naphthalene 2-[(3R,4S)-3-fluoropiperidin-4-yl]oxybenzaldehyde (5R,7S)-N-[2-(5-bromothiophen-3-yl)ethyl]-1,3,5,7-tetramethyl-5,8-dihydro-4H-pyrazolo[3,4-d]azepine-6-carboxamide 3-amino-1-[4-(4,5-dihydrotriazin-2-yl)piperazin-1-yl]-2,3-dihydroisoquinoline-7,8-diol 2-methyl-4-[4-(3,4,5-trifluorophenoxy)phenyl]butanoic acid 2-(4-fluorophenyl)-6,11-dioxo-3-propan-2-yl-1,8-diazatricyclo[7.3.0.03,7]dodeca-9,11-diene-12-carboxamide 2-fluoro-N'-[4-(morpholine-4-carbonyl)phenyl]benzenecarboximidamide N-[(3,5-dichlorophenyl)methyl]-1-[(4E)-2,6-difluorohepta-2,4,6-trienyl]-5-ethoxy-8-methyl-4H-chromeno[4,3-c]pyrazole-3-carboxamide 3-[4-(1,2,6-trimethylcyclohexa-2,4-dien-1-yl)oxyphenyl]cyclopropane-1,1,2,2-tetracarbonitrile (4S)-3,4-dihydro-2H-chromene;ethane;formaldehyde;2-[7-methyl-5-oxo-4-[3-(trifluoromethoxy)phenyl]-1,4-dihydroimidazol-2-yl]acetamide 2-(4-azidophenyl)-6-ethoxycarbonylbenzoic acid 2-[2-aminoethyl(methyl)amino]-3,5,6,7,8,9-hexahydrocyclohepta[d]pyrimidin-4-one 4-N,6-dimethyl-2-(2-propan-2-ylpyrazol-3-yl)pyrimidine-4,5-diamine 2-(3,4-dichlorophenyl)-3-fluorocyclohexa-1,5-diene 2-[(5-ethoxycarbonylfuran-3-yl)methyl]butanoic acid (3S)-N,5'-dimethyl-2-(5-oxopyrrolidin-2-yl)-3-phenylmethoxy-2'-(6H-triazolo[4,5-d]pyrimidin-7-ylsulfanylmethyl)spiro[1H-indole-3,1'-cyclohexane] [3-(1H-imidazol-5-yl)phenyl]-(2,4,6-trihydroxyphenyl)methanone 2-(azidomethyl)-7-[5-fluoro-3-(4-fluorophenyl)pyridin-2-yl]heptanoic acid 1-[(4aR)-6,7-dimethyl-2,3,4a,5,11b-hexahydro-1H-pyrido[4,3-b]carbazole-8-carbonyl]pyrrolidine-3-carboxylic acid;hydrochloride 2-cyclobutyloxy-N'-[5-(4-hydroxyphenyl)pyrazin-2-yl]acetohydrazide 2-benzylsulfanyl-3,4-di(propan-2-yl)phenol 1-(4-azidobutyl)-2,5-dimethoxybenzene (3S)-3-azido-2-benzylpyrrolidine [3-(1,4-dioxan-2-ylmethoxy)phenoxy]boronic acid 2-[N-(carboxymethyl)-4-methoxycarbonylanilino]decanoic acid 4-fluoro-N-[(1R)-3-[2-fluoro-5-(6-methoxypyridin-3-yl)phenyl]-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethyl)phenyl]propyl]-3-methylbenzamide 3-[1-amino-2-(3,5-dichlorophenyl)ethyl]pyridine-4-carboxamide 6-[[5-chloro-2-(3-ethoxyanilino)pyrimidin-4-yl]amino]-1-methylcyclohexa-3,5-diene-1,3-dicarboxylic acid N-(3,4-dichlorophenyl)-2-[ethylsulfonylmethyl-(4-phenylbenzoyl)amino]-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide N-(1,3-benzothiazol-5-yl)-4-(difluoromethoxy)benzenesulfonamide 3-[7-(2-fluorophenyl)-1H-imidazo[4,5-b]pyridin-2-yl]-5-pyrazin-2-yl-1H-pyrazolo[3,4-c]pyridine 3-(1H-imidazol-2-yl)-N-[[6-oxo-4-(trifluoromethyl)-1H-pyrimidin-2-yl]methyl]-5-phenyl-1,2-oxazole-4-carboxamide 5-(4-chlorophenyl)-1-methyl-N-[[(3S,6R)-6-(4-propan-2-yloxyphenyl)oxazepan-3-yl]methyl]pyrazole-4-carboxamide 2-[2-(3,5-dichlorophenyl)propanoylamino]cycloheptane-1-carboxylic acid 1-(4-azidocyclohexyl)oxyanthracene 4-[3-(4-hydroxyphenyl)-5-oxo-4H-1,2,4-triazin-6-yl]butanoic acid 4-[[1-(5-chlorothiophene-2-carbonyl)pyrrolidin-3-yl]amino]-2,2,6,6-tetramethylpiperidine-1-carboxylic acid 2-azido-1,3-dibromo-4-phenylmethoxybenzene 2-[4-(dimethylamino)phenyl]-N-[(Z)-(5-ethoxy-3,4-dihydroxyoxan-2-yl)methylideneamino]acetamide 3-[4-[(E)-2-[5,8-bis(ethenyl)naphthalen-1-yl]prop-1-enyl]phenyl]-N,N'-dimethylcyclopentane-1-carboximidamide 2-(2-hydroxynaphthalen-1-yl)cyclohexane-1,3-dione 5-amino-1,3-dimethylimidazole-2-thione;3-(4-cyano-3-propan-2-ylphenyl)-2-[6-(2,2-difluoroethoxy)pyridin-3-yl]propanoic acid 1-[4-fluoro-3-(trifluoromethyl)phenyl]propane-2,3-diamine 2-methyl-1-(4-pyridin-3-yloxyphenyl)butan-1-one (2-azidosulfanyloxyphenyl)-phenylmethanol 2-[(1,4-dioxin-2-ylmethylamino)methyl]prop-2-enamide;ethane N-(3,4-dimethyl-1,2-oxazol-5-yl)-2-[6-fluoro-3-(trifluoromethyl)pyridin-2-yl]acetamide 1,1-dimethylcyclopropane;1-ethenyl-4-[1-(3-fluorophenyl)butan-2-ylidene]benzene 5-fluoro-N-methyl-2-(pyridin-3-yloxymethyl)benzamide 3-(4,5-dimethylpyridin-2-yl)oxypyridine 5-[4-(3,4-difluorophenyl)triazol-1-yl]-6-ethoxypyrimidine-2,4-diamine (2S,3R)-1-cyclohexyl-N-[(2S)-2-hydroxy-3-phenylpropyl]-N-methyl-2-phenylpiperidine-3-carboxamide 7-[(2S,3R)-3-amino-5-chloropentan-2-yl]oxy-2-butylisoquinolin-1-one;hydrochloride 1-[2,4-dimethoxy-3-(methylamino)phenyl]ethanone;methanol 2-(N,2-diaminoanilino)ethanol (2R,3S)-2-amino-5-[3-(5-hydroxypentyl)phenyl]-1,1,6,2,3-pentamethyl-3H-indene-4,6-diol 4-[3-(8,9-dimethoxydecyl)phenyl]phenol N-(cyclopropylmethyl)-3,6-difluoro-2-[4-methoxy-1-[[4-phenylmethoxy-3-(trifluoromethyl)phenyl]methylamino]pentan-3-yl]oxybenzamide 5-[(4-methoxyphenyl)sulfonylamino]-2-(3-propan-2-ylpiperazin-1-yl)pyridine-3-carboxylic acid;2,2,2-trifluoroacetic acid 6-[3,5-difluoro-4-(trifluoromethyl)phenyl]hexanamide 5-(furan-2-yl)-7,8-dihydroimidazo[1,2-c]quinazoline 6-[5-(3,4-dichlorophenyl)tetrazol-2-yl]-3H-1,3-benzoxazol-2-one (1R)-N-[1-amino-6-(azepan-4-yloxy)isoquinolin-3-yl]-2-fluorocyclopropane-1-carboxamide 6-chloro-5-[4-(1H-indol-2-yl)piperidin-1-yl]pyridazine-3-carbonitrile 2-[(1R,3S)-3-hydroxycyclopentyl]-7-methoxychromene-4-thione (2R)-1,3-dimethoxy-2-propyl-2H-naphthalene 5-bromo-N,3-dimethylpyrazolo[1,5-a]pyridine-2-carboxamide;ethane N-azido-6,6,6-trifluoro-4-oxo-5H-1,7-naphthyridine-3-carboxamide 6,7-dihydro-5H-pyrazolo[3,4-b]pyridin-3-ylmethanesulfonamide 1-[(3,5-dichloro-4-hydroxyphenyl)methyl]pyrrolidine-2,5-dione N-[1-(3-chloropyridin-2-yl)pyrrolidin-3-yl]ethanesulfonamide 3-[(4R)-6,6-difluoro-7,10,11-trimethyl-2-oxa-5,8,12-triazatricyclo[6.4.0.02,6]dodeca-1(11),9,12-trien-4-yl]propan-1-ol 5-(4-fluorophenyl)-7H-thieno[2,3-b]pyridine 1-methylsulfonylpyrazole-4-carboxamide 1-(3,4-dichlorophenyl)-2-[1-(2-methylpyrimidin-5-yl)piperidin-4-yl]ethanone 1-[2,4-bis(methoxymethoxy)phenyl]-4-iodobenzene 1-[2-[(4,5-diphenyl-1,3-thiazol-2-yl)amino]ethylcarbamoyl]cyclopropane-1-carboxylic acid N-[2-(methylcarbamoyl)phenyl]-3,4-dihydroisoquinoline-1-carboxamide 5-amino-3-(3-chloro-4-hydroxyphenyl)-2,3-dihydro-1,2-oxazole-4-carbonitrile 2-[(2R)-butan-2-yl]sulfanyl-6-methoxy-4H-pyrido[3,2-b][1,4]oxazin-3-one 3-[2-[(1S)-5-fluoro-8-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]ethynyl]pyridine 2-(3,4-dichlorophenyl)-N-[2-fluoro-5-methyl-4-(trifluoromethyl)phenyl]acetamide 4-methyl-5-[(2E,3Z)-2-propylidenehexa-3,5-dienoxy]-2-(trifluoromethyl)phenol (7E)-1-[2,5-dimethyl-4-(trifluoromethyl)phenyl]-2,3-bis(ethenyl)-7-ethylidene-6,8-dihydro-5H-indolizine;ethane 5-methyl-N,2-diphenylaniline 1-[[4-(3,5-dichlorophenyl)oxan-4-yl]methyl]-3-(6-methoxypyridin-2-yl)urea 4-[(E)-2-(1,3-benzodioxol-5-yl)ethenyl]pyridine 3-[4-[5-(1H-indol-6-yl)pyrimidin-2-yl]morpholin-2-yl]benzonitrile 3-[3-(2,4-difluorophenyl)propanoyl]-7-oxa-3,10-diazaspiro[5.6]dodecan-11-one 3-[4-[4-[2-chloro-5-(trifluoromethoxy)phenyl]phenoxy]piperidine-1-carbonyl]azetidine-1-carbonitrile 4-[(3R)-3-amino-2,5-dioxopyrrolidin-1-yl]-6-fluoropyrazolo[1,5-a]pyridine-3-carboxylic acid (3-aminopyridin-2-yl)-[4-[5-(2,6-difluorophenyl)-1H-imidazol-2-yl]piperidin-1-yl]methanone;ethane [3-[(dimethylamino)methyl]piperidin-1-yl]-phenylmethanone 4-[3-(dimethylamino)phenyl]-3,5-dioxohexanal [6-(2,4-dimethylanilino)-9-propan-2-ylpurin-8-yl]-(3-methoxyphenyl)methanethione 1-[4-(2,5-dimethylhexan-3-yl)phenyl]buta-1,3-dien-1-ol 1-cyclopentyl-3,3-dimethyl-2H-indene-1-carboxamide 2-[[4-(trifluoromethoxy)phenyl]carbamoyl]pyrrolidine-1-carboxylic acid (6S)-7-[[2-amino-3,3-dideuterio-3-(4-fluorophenyl)propyl]amino]-8-oxo-3-(4-phenoxyphenoxy)-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid N-(2,4-dichloropyrimidin-5-yl)-1H-pyrrole-3-carboxamide N-[1-[4-methoxy-3,5-bis(phenylmethoxy)phenyl]ethyl]-2-methylcyclopropane-1-carboxamide [2-bromo-4,6-di(propan-2-yl)phenyl]phosphane 3-methoxy-5-(4-propanoylphenyl)benzamide 2-(benzylamino)oxyethanol 2-(4-bromophenyl)-3,5,6,7-tetrahydropyrrolo[3,4-d]pyrimidin-4-one 1-(2-propan-2-yloxyphenoxy)-3-(pyrimidin-5-ylmethylamino)propan-2-ol 5-[(3R)-1-(2,4-difluorophenyl)sulfonylpyrrolidin-3-yl]-3-pyrazin-2-yl-6H-triazolo[4,5-d]pyrimidin-7-one 3-[(4,5-dimethylthiophene-2-carbonyl)amino]cyclobutane-1-carboxylic acid 2-[(7R,8aS)-2-[1-oxo-5-phenylmethoxy-3-(4-propan-2-ylphenyl)isoindole-2-carbonyl]-1,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-7-yl]acetamide 2-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]oxirane 3-[5-[4-(2-azidoethoxy)phenoxy]pentylsulfanyl]propanoic acid 2-[[2-amino-4-(dimethylamino)-6,7,8,9-tetrahydro-5H-cyclohepta[d]pyrimidine-7-carbonyl]amino]-3-cyclohexylpropanoic acid 3-(2-methylphenoxy)-1-[4-[4-(trifluoromethoxy)phenyl]sulfonylpiperazin-1-yl]propan-1-one 2-(6,7-dimethoxyquinolin-4-yl)oxy-N-methylcyclohexan-1-amine [1-(4-fluorophenyl)sulfanylpyrrolidin-2-yl]methanetriol 2-cyclopropyloxy-N-(3,4-dimethylphenyl)-6-[(Z)-N'-hydroxycarbamimidoyl]benzamide N-(3,5-dichlorophenyl)sulfonyl-2-(1H-indol-7-yl)propanamide N-[5-(1,3-benzothiazol-2-yl)pyridin-2-yl]-4,6-bis(4-methoxyphenyl)pyrimidine-2-carboxamide (4S,5R)-2-ethylsulfanyl-6,11-dioxo-9-[[1-[4-(trifluoromethylsulfonyloxy)phenyl]cyclopropyl]amino]-3-azabicyclo[4.2.0]octa-1(7),8-diene-4-carboxylic acid 1-(3,4-dimethoxyphenyl)-3,5,6-trimethylpyrrolo[2,3-b]pyridine N-[5-bromo-2-(4-hydroxyphenyl)-1,3-benzoxazol-6-yl]formamide;1H-indole 2-(3,4-dimethoxyphenyl)-7-iodoquinoline N-(4-aminophenyl)sulfonyl-5-methylisoquinoline-7-carboxamide 4-amino-6,7-diethoxyquinoline-3-carbonitrile N-[3-(4,5-dihydropyrimidin-6-yl)phenyl]-2-(4,7,10,13-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,5,10,12-pentaen-8-ylsulfanyl)acetamide 4-[1-(2,6-difluorophenyl)propan-2-ylamino]-3-methoxy-N-methylsulfanylbenzamide 2-methylsulfanyl-3-[(E)-2,5,5-trideuteriopent-1-enyl]pyrazine 2-hydroxy-3-[(4S)-4-methyl-1,2,5-oxadiazol-3-yl]benzaldehyde N-[3,5-bis(trifluoromethyl)phenyl]-2-cyclopropyl-5H-pyrrolo[3,2-d]pyrimidine-7-carboxamide (5Z)-5-[[2,4-dihydroxy-6-methyl-3-(phenyliminomethyl)phenyl]methylidene]imidazolidine-2,4-dione N-(2-butylsulfonylethyl)-4,6-dihydroxy-7-oxo-1H-indole-3-carboxamide 2-[4-methoxycarbonyl-N-(3-nitrophenyl)anilino]octanoic acid N-[2-(5-chloro-3,4-dihydropyrazole-2-carbonyl)phenyl]-N',N'-dimethyloxamide 5-[5-[1,4-bis(trifluoromethyl)cyclohexa-2,4-dien-1-yl]furan-2-yl]-1H-pyrazole 4-[4-fluoro-3-(trifluoromethyl)phenyl]sulfanylmorpholine N-(4,6-dimethylpyrimidin-2-yl)-3-[ethyl(propanoyl)amino]pyrrolidine-1-carboxamide (5-fluoro-3,4-dihydro-2H-quinolin-1-yl)-[1-[2-[(4-methoxyphenyl)methyl]indazole-7-carbonyl]piperidin-4-yl]methanone 1-methyl-3-(3,4,5-trifluorophenyl)cyclohexa-2,4-diene-1-carboxamide 1-(2,4-difluorophenyl)-6-[1-[(3S)-piperidin-3-yl]indazol-5-yl]-7H-cyclopenta[d]pyridazine 2-bromo-5-[(3Z)-hexa-1,3,5-trien-2-yl]benzenesulfonic acid 2-azido-6,6-dimethyl-4-phenylpiperidine 5-[1-[(2,4-dichlorophenyl)methyl]piperidin-3-yl]-2-(pyridine-4-carbonylamino)pentanoic acid 3-(azidomethyl)-7-chlorobenzo[g]chromene-2,4-dione 5-(2,4-difluorophenyl)-6-methyl-5H-tetrazolo[1,5-a]pyrimidine 2-(2,4-difluorophenyl)-1H-indole 1-[4-(2,5-difluorophenyl)pyridin-3-yl]ethenamine 3,5-bis(trifluoromethyl)benzaldehyde;N-[2-(3-chlorophenyl)ethyl]-4-cyclobutyl-2-cyclopentyloxyaniline;N,N-dipropylbutan-1-amine 4-amino-1-[[2,4-bis(trifluoromethyl)phenyl]methyl]indazole-3-carboxylic acid N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-[(6,7-dimethoxy-1,5-naphthyridin-4-yl)oxy]benzamide 4-[3-(2,6-difluorophenyl)imidazo[1,5-a]pyridin-8-yl]benzonitrile 2-[(6S)-5-oxo-3-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-6-carbonyl]sulfanyl-N-(2-phenylethyl)benzamide 4-(3-amino-2,6-difluorophenyl)-2-chloro-6-methoxycarbonylpyridine-3-carboxylic acid 3-[(2-methoxyphenyl)-(oxolan-2-ylmethylamino)methyl]phenol N'-[(Z)-(2,5-dimethylphenyl)methylideneamino]-N-[4-(trifluoromethoxy)phenyl]ethanimidamide 1-azido-5-benzylindole 3-methoxy-1-[2-(4-methoxyphenyl)ethyl]pyrrolidine;2,2,2-trifluoroacetic acid N-[2,6-dichloro-4-(methoxymethyl)phenyl]-3-sulfamoylbenzamide 2-amino-4-(6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-3-yl)benzenecarboximidamide N-[2,3-difluoro-4-(1,1,1,3,3,3-hexafluoropropan-2-yloxy)phenyl]formamide (2S)-3-[8,9-dimethoxy-2-(4-methylphenyl)-5,6-dihydropyrrolo[2,1-a]isoquinolin-11-yl]-2-ethenylpyrrolidine-1-carboxylic acid [4-(5-ethylbenzotriazol-2-yl)phenyl]-trimethylazanium N-[(2S)-6-amino-2-[(3,4-difluorophenyl)methyl]-1,2,3,4-tetrahydronaphthalen-1-yl]cycloheptanecarboxamide (2R)-1-[4-[6-chloro-8-fluoro-7-(2-fluorophenyl)quinazolin-4-yl]piperazin-1-yl]propane-1,2-diol (5-chloro-2,3-dihydroindol-1-yl)-[3-(1H-imidazol-2-yl)phenyl]methanone 2-[(6S)-3-methylsulfanyl-7-oxo-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-5-ium-1-yl]-N-phenylacetamide 3-azido-4-hydroxychromen-2-one 4-[2-(5-bromoindol-1-yl)acetyl]morpholine-3-carboxylic acid [4-[(4-azidopyridin-2-yl)methyl]morpholin-2-yl]methanol N-[3-amino-4-(2-hydroxyethylcarbamoyl)phenyl]-6-methoxynaphthalene-2-carboxamide 2-[[1-[(4-methylpyrazol-1-yl)methyl]cyclopropanecarbonyl]amino]pyridine-3-carboxylic acid 1-[(3S)-3-phenylpiperazine-1-carbonyl]cyclopentane-1-carbonitrile N-(5,8-dimethylquinoxalin-6-yl)benzamide 2-[(5-bromopyridin-3-yl)amino]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidin-5-one 1-[4,5-dimethyl-2-(1,3-thiazol-2-yl)phenyl]sulfonyl-N-(2,6-naphthyridin-3-yl)piperidine-4-carboxamide 2-fluoro-3-[4-(1H-imidazole-2-carbonyl)phenyl]benzoic acid [(4aS,6S)-1-methyl-2,3,4a,5,6,7,8,9,10,11a-decahydropyrido[3,2-b]azocin-6-yl]-pyridin-3-ylmethanone 6-methoxy-2-phenyl-7H-purine 2-[3-(oxiran-2-ylmethoxy)phenyl]sulfonylaniline (2S)-1,6-bis[5-chloro-3-(difluoromethyl)pyrazol-1-yl]-4-phenylsulfanylsulfanylhexane-2-thiol 2-[(3R)-5-(4-chlorophenyl)-1-ethanimidoyl-7,8,9,10-tetrahydrophenanthridin-6-yl]acetaldehyde;N,N-dimethylmethanamine 4-[(E)-2-[3,5-bis[2-methoxyethyl(methyl)amino]phenyl]ethenyl]-N,1,6,7-tetrahydroindol-5-amine 4-azido-N-[2-chloro-6-(difluoromethoxy)phenyl]pyrimidin-2-amine (2S)-2-[3,4-dimethyl-5-(trifluoromethyl)phenyl]sulfanyloxane (4R)-1,3,4-trimethyl-6-pyridin-2-yl-4H-[1,2]thiazolo[5,4-d]pyrimidine-7-thione 1-[2,6-di(propan-2-yl)phenyl]-3-methylsulfanylurea 2-[(4R)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]quinoline 2-[(4-nitrophenoxy)carbonylamino]pentanoic acid N-benzyl-6-(2,4-difluorophenyl)sulfanylpyridine-3-carboxamide 6-chloro-7,8-dimethoxy-N,N,5,5,9,11-hexamethylacridin-3-amine;hydrochloride (2R,3S)-3-[(4-chlorophenyl)sulfonylamino]-N-hydroxy-1-methylpyrrolidine-2-carboxamide 2-cyclohexyl-N-(2,4-difluorophenyl)-5-methylsulfonyl-1H-imidazole-4-carboxamide N-(6,7-dihydro-5H-cyclopenta[b]pyridin-3-yl)-4-methoxy-2,3,5,6-tetramethylbenzamide 3-ethyl-7-[4-(methoxymethyl)-2H-azet-1-ium-1-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine 2-[[(2R)-1-methylpiperidin-2-yl]methoxy]-8-propan-2-yl-7H-purine 2-N,4-N-bis(4-methylphenyl)acenaphthylene-1,2,4-triimine;cobalt N-(6-methylpyridin-2-yl)-4-[1,3]dioxolo[4,5-f][1,10]phenanthroline-7-carboxamide N-[6-(2,3-dihydro-1,4-benzodioxin-6-yl)imidazo[1,2-a]pyrazin-8-yl]-2-methoxy-4-(oxolan-3-yl)benzamide 2-[(E)-2-nitroethenyl]naphthalene 1-(4,7-dioxo-2-thiophen-2-yl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-ium-6-yl)hexane-1,5-disulfonic acid 3-[(3R)-1-tert-butylpyrrolidine-3-carbonyl]benzamide N-[1-[4-(cyclopropylcarbamoyl)phenyl]ethylideneamino]pyridine-2-carboxamide (2S)-3,6-difluoro-N-[1-[4-methyl-3-[(E)-prop-1-enyl]phenyl]ethylidene]spiro[2.5]octane-2-carboxamide 4-[3,5-bis(trifluoromethyl)phenyl]sulfanyl-N'-(7-phenylheptyl)benzenecarboximidamide 4-(3-phenyl-2H-pyrrol-5-yl)benzoic acid 1-[3-[2-(6,7-dihydro-5H-imidazo[1,5-a]imidazol-2-yl)ethynyl]phenyl]piperidine-4-carboxamide ethane;N-methyl-1-(2-pyridin-3-ylacetyl)piperidine-4-carboxamide (6R,7S)-3-(dihydroxymethylcarbamoyl)-8-oxo-7-[(2-phenylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 6-(2-diazohydrazinyl)naphthalene-1,4-disulfonic acid 6-amino-3,5-diethyl-1,8-naphthyridine-2-thione N-[1-(5-methylimidazo[1,2-a]pyridine-3-carbonyl)azetidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)cyclobutanecarboxamide 2-[4-[2-(2,6-difluorophenyl)-7H-purin-6-yl]piperazin-1-yl]pyrimidine 5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-2-methylpyran-4-one 5-[2,3-difluoro-4-(trifluoromethyl)phenyl]-6-oxo-1H-pyrazine-3-carboxylate 2-(1,3,3a,4,5,7a-hexahydroisoindole-2-carbonyl)cyclohexan-1-one N-(2,6-difluorophenyl)-4-[[(E)-1,3-dipyridin-2-ylprop-1-enoxy]methyl]-5-hydroxyfuran-2-carboxamide 2-[6-amino-5-(1,3-benzothiazol-7-ylmethoxy)pyridin-3-yl]acetamide 4-[5-[2-fluoro-6-(trifluoromethyl)phenyl]-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide N-[(1R)-6,7-dihydro-5H-cyclopenta[c]pyridin-3-yl]-7-methoxy-4-methylidenepyrido[1,2-a]pyrimidine-2-carboxamide 4-bromo-2-[(E)-3,6-dimethylhept-1-enyl]phenol [3-fluoro-4-(2-phenylethynyl)phenyl]methanol N'-hydroxy-4-methoxy-3-[(2S)-2-(piperidine-1-carbonyl)morpholin-4-yl]benzenecarboximidamide 2-(3,4,6,7,8,9-hexahydrobenzo[g]quinolin-1-yl)benzaldehyde 2,5-bis[(4-nitrophenyl)diazenyl]-6H-1,3-thiazin-4-amine N-[[3,5-dimethyl-1-[(E)-2-phenylethenyl]pyrazol-4-yl]methyl]-6-(3-fluoropyrrolidin-1-yl)pyridazin-3-amine 2-[(3S,4R)-1-(cyclopropanecarbonyl)piperidin-3-yl]oxy-6-hydroxybenzamide;hydrochloride 2-methoxy-N,N'-dimethyl-N-[(1R)-2-[4-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)phenyl]cyclopropyl]ethanimidamide 3,4-diphenylbutane-1,1,2-tricarboxylic acid (7S)-5-[3-bromo-4-methoxy-2-(2,2,2-trifluoroethylsulfanyl)phenyl]-6,7-dihydro-5H-pyrrolo[1,2-b][1,2,4]triazole 1-(3-methylphenyl)-N-[2-[2-[(2S,4R,6R)-6-(4-methylphenyl)oxan-2-yl]ethoxy]ethyl]methanesulfonamide 6-[(5,6-dimethyl-1H-indol-3-yl)methyl]-2-propan-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 3-[(6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-2-ylamino)methyl]benzenesulfonamide 2-[[6,8,10,11,12-pentamethyl-4-(morpholine-4-carbonyl)-3,5-dioxoindolizino[1,2-b]quinolin-9-ylidene]amino]acetaldehyde (2-hydroxy-1,3-benzothiazol-6-yl)-(4-nitrophenyl)methanone 6-azido-3,4-bis[(2-chlorophenyl)methoxy]pyridine 1-[3,4-difluoro-2-(triazol-2-yl)phenyl]-N-methoxymethanimine [(Z)-1-bromo-2-methylpent-3-en-2-yl]benzene;ethane 1-[[4-(2,6-dimethoxyphenyl)pyridin-3-yl]amino]-3-(4-ethyl-2,5-diphenylpyrazol-3-yl)urea 2,3-difluoro-1-N-[(E)-4-nitrobut-3-enyl]benzene-1,4-diamine N-(1H-indazol-6-yl)-1,3-benzothiazol-2-amine N-azido-3,5-dichloro-4-fluorobenzamide (5R)-3-(3-bromophenyl)-2,7-diazaspiro[4.5]decan-1-one 5-(1H-pyrazol-4-yl)-3,6-dihydro-2H-1,4-thiazin-5-amine N-[3,4-difluoro-2-(propylamino)phenyl]sulfanyl-1,3-thiazol-5-amine 4-[2,6-dimethyl-4-(4,5,6,7-tetrahydrobenzimidazol-1-yl)phenyl]benzoic acid 4-[(1R)-2-hydroxycyclopropyl]benzoic acid 2,4-bis[4-(trifluoromethyl)phenyl]-6-[3-[3-(trifluoromethoxy)phenoxy]piperidin-1-yl]-1H-1,3,5-triazine 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[1H-indole-3,4'-piperidine]-2-one 7-(1,3,5-trimethylpyrazole-4-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 2-[4-hydroxybutyl(methoxycarbonyl)amino]benzenesulfonic acid 2-(6-methyl-5,6,7,8-tetrahydronaphthalen-2-yl)-6-propan-2-yldibenzofuran 4-fluoro-N-[3-(5-pyridin-2-yl-1,3,4-thiadiazol-2-yl)-4,5,6,7-tetrahydrothieno[2,3-c]pyran-2-ylidene]benzenesulfonamide 3-[(E)-2-[4-(5-fluoro-6-methoxypyridin-2-yl)phenyl]ethenyl]aniline 1-[2,3-difluoro-4-(trifluoromethyl)phenyl]-2-fluoronaphthalene 4-(2,1,3-benzoxadiazol-5-yl)-N-methylpyrimidin-2-amine 1,3-diethyl-6-[(E)-1-hydroxy-2-[4-[2-[methyl(methylideneamino)amino]phenyl]phenyl]ethenyl]indol-5-ol 1-azido-3-(2,2-dibromoethenyl)-5-phenylbenzene (5E)-2-(4-iodophenyl)imino-5-[(1,3-thiazol-2-ylamino)methylidene]-1,3-oxazolidin-4-one 5-[1-(6-aminopyridin-3-yl)piperidin-4-yl]oxypyrazine-2-carboxamide 2-[(4-chlorophenyl)methylsulfanylamino]-5,7-dihydro-3H-thieno[3,4-d]pyrimidin-6-one ethane;3-(3-ethylphenyl)-1,2,4,6-tetrahydrotriazolo[4,5-d]pyridazine N-[(1S)-6-(2,5-difluorophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]-1,3-benzothiazol-2-yl]acetamide 2-[(3aR,6aS)-5-methylsulfonyl-1,2,3,3a,4,5,6,6a-octahydropentalen-2-yl]-N-[4-amino-3-(trifluoromethoxy)phenyl]acetamide (3S)-1-[4-[2-[5-[4-(1,1-difluoroethyl)phenyl]-7-fluoroimidazo[4,5-b]pyridin-3-yl]ethynyl]pyridin-2-yl]pyrrolidine-3-carboxamide 2-amino-8-(1H-imidazol-5-ylmethyl)-1,7-dihydropurin-6-one (3S)-N,5-dimethyl-1-[(2S)-1-[[(Z)-4-(methylideneamino)but-3-enoyl]amino]-3-phenylpropan-2-yl]-N-propylpiperidine-3-carboxamide 3-[4-(5,5,6,6,8,10,11,13,14,15,16,17-undecafluorononoxy)phenyl]cyclopentan-1-one [6-(4,6-diphenylpyrimidin-2-yl)naphthalen-1-yl]boronic acid [3-(2-chlorophenyl)piperidin-1-yl]-(1-propan-2-yltriazol-4-yl)methanone N-[(4,5-dimethyl-1H-pyrazol-3-yl)carbamothioyl]pentanamide 2-(1H-indol-3-yl)-N-[4-(5,6,7,8-tetrahydroquinoline-4-carbonylamino)phenyl]acetamide 2-[1,3-dioxo-4-(thiophene-2-carbonyl)isoindol-2-yl]-5-[[5-ethyl-6-(methylaminomethyl)pyridin-2-yl]methyl]benzonitrile [2-(4,5-diphenyl-1H-imidazole-2-carbonyl)-1,3-thiazolidin-3-yl]methanol (1R,3S)-2,2-dichloro-N-[4-chloro-3-[2-[5-fluoro-6-methyl-3-(trideuteriomethoxy)pyridin-2-yl]acetyl]phenyl]-3-(3,4-dichlorophenyl)cyclopropane-1-carboxamide (5Z)-2-sulfanylidene-5-[[4-[(3,4,5-trifluorophenoxy)methyl]phenyl]methylidene]imidazolidin-4-one 2-[2-oxo-3-(thiophene-2-carbonyl)chromen-8-yl]oxyacetate N-butyl-6-methoxy-2,3-dihydro-1H-indene-4-carboxamide ethane;5-methyl-2,3,4,7,8,9-hexahydro-1H-carbazole 2-[3-(1,4-dihydropyrimidin-5-yl)phenyl]quinazoline 1-ethyl-4-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxybenzene N-[[2-(dimethylamino)phenyl]methyl]-2-ethoxy-N,3-diethyl-6-imidazol-1-ylpyridine-4-carboxamide 2-(1H-indol-3-yl)-N-[3-methoxy-4-(1,3-thiazol-4-ylsulfonylamino)phenyl]acetamide (E)-1,3-dichlorobut-2-ene;methoxyethane;4-methylhexanamide;4-[3-methyl-5-(6-methylideneheptanoyl)phenoxy]pentanal;pentane N-(2,4-dimethylphenyl)-1-(4-oxo-3H-quinazolin-2-yl)piperidine-4-carboxamide N-[(E)-1H-indol-3-ylmethylideneamino]-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxamide 2-ethoxy-5-methyl-N-[3-(4-propan-2-ylphenoxy)phenyl]pyridine-3-carboxamide 6-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-1,2,3,4,6,7,8,9-octahydropyrido[4,3-b]indole 2-[4-(4-chlorophenoxy)piperidin-1-yl]-6-methoxyquinoline 5-methyl-N-[2-oxo-1-(4,6,7,8-tetrahydrofuro[3,2-c]azepine-5-carbonyl)piperidin-3-yl]-2,3-dihydro-1H-indene-2-carboxamide 3-[(5-chlorothiophene-2-carbonyl)amino]cyclobutane-1-carboxylic acid 4-(4-aminobutylamino)-5-chloro-1H-pyrimidin-6-one N-[(4S)-5,8a-dimethyl-2,3,4,9-tetrahydrochromen-4-yl]-1-aminocyclopropane-1-carboxamide;hydrochloride N-[(4-phenylphenyl)methyl]propane-2-sulfonamide 5-[3-(4-methylpiperazin-1-yl)propoxy]quinoline 1-(3,5-dichlorophenyl)-2,4-diethylpentane-2,3-diol 6-(4-bromophenyl)-2-methoxy-1,2-dihydronaphthalene 6-[(4R)-5-chloro-2,2-difluoroethyl]quinoline 3-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)cyclopentan-1-ol 3-[5-methoxy-2,4-bis(phenylmethoxy)phenyl]propanamide 4-(azidomethyl)-5-chloro-2,3,6-trimethoxypyridine 1-[2,4-dihydroxy-3-(5-thiophen-2-ylfuran-2-carbonyl)phenyl]pentane-1,6-dione 1,4-dimethylcyclohexane;(Z)-4-methoxy-2,3-dimethylidenepent-4-ene;4-[5-[(E)-2-pyridin-4-ylethenyl]thiophen-2-yl]butanal 4-[2-(3,5-dimethoxyphenyl)ethylamino]-1H-pyrimidin-6-one 6-chloro-5-(2,3-dimethylphenyl)-1-ethylpyrazolo[4,3-c]pyridine 4-N-(1,3-benzodioxol-5-yl)-2-methylsulfanylpyrimidine-4,6-diamine;cyclopropanecarboxylic acid 1-(2,3-dihydro-1H-inden-1-yl)-6-[5-methoxy-4-[2-(6-methylpyridin-3-yl)ethyl]pyrimidin-2-yl]indole 2-[(3,4-dichlorophenyl)methyl]sulfanylacetic acid N-[(2S)-1-amino-3,3-difluoro-1-oxobutan-2-yl]-4-(6-methoxypyridine-3-carboximidoyl)benzamide N-[3-bromo-4-[(Z)-(2,5-dioxoimidazolidin-4-ylidene)methyl]phenyl]thiophene-2-carboxamide 1-[3-[5-(5,6-dihydroquinoline-7-carbonylamino)pyridin-2-yl]oxycyclobutyl]triazole-4-carboxylic acid N-[2,3-difluoro-5-[4-(1H-indole-6-carbonyl)piperazin-1-yl]phenyl]acetamide 1-(4-bromophenyl)sulfonyl-3-methoxypyridin-2-one N-[4-(3-chlorophenyl)butan-2-yl]-7,8-dihydro-6H-furo[3,2-e]indole-1-carboxamide N-[2-(1,1a,6,6a-tetrahydrocyclopropa[a]inden-4-yl)ethyl]-N'-(3,5-dimethoxyphenyl)-N-ethyl-N-methylethanimidamide 1-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-2-hydroxy-N'-methyl-4-oxo-6,7-dihydro-5H-indole-3-carbohydrazide 3-[3-(1H-benzimidazol-2-yl)benzenecarboximidoyl]quinoxalin-6-amine 4-[2,5-difluoro-3-(trifluoromethoxy)phenyl]-1H-tetrazol-5-one 2-(methoxymethyl)-N-(3-pyrazin-2-ylpropyl)aniline 1-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexan-1-one 2-[(1E,3Z)-5-[N'-(4-chlorophenyl)carbamimidoyl]penta-1,3-dienyl]-4,7-bis(sulfanylidene)-3,6,8,9,10,11-hexazatetracyclo[8.7.0.02,7.012,17]heptadeca-1(17),2,4,6,8,11,13,15-octaene-14-carboxamide 4-[4-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethoxy)phenyl]benzamide N-[4-[2-[(3,5-dichloropyridin-4-yl)amino]ethyl]cyclohexyl]carbamate 1-[(5,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)amino]ethylideneazanium 3-[4-(4,4-dimethylcyclohexen-1-yl)piperidin-1-yl]-5-fluorosulfonyloxypyridine 1-benzyl-3,5-dimethoxybenzene;cyclohexanamine 5-[[7-(3,4-dichlorophenyl)-2-methylpyrazolo[1,5-a]pyrimidin-5-yl]amino]piperidine-2,6-dione 2,3-difluoro-1-[(E)-3-[4-(trifluoromethyl)phenyl]but-2-en-2-yl]benzene 3-(4-bromophenyl)-2-(dimethylamino)propanal 2-[(3S,4S)-1-(2,6-difluorobenzoyl)piperidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one (2Z,5Z)-3-[1-[4-ethylsulfanylbutyl(methyl)amino]ethenyl]-6-fluoro-8-methoxyiminodeca-2,7-dienimidamide;(4R)-4-hydroxyoxolan-2-one 4-[1-[(2E)-2-(1,3-benzodioxol-5-ylmethylidene)hydrazinyl]ethoxy]benzenesulfonamide 2-(methoxymethyl)-7,8-dihydrobenzo[g]quinoline 2-chloro-N-[4-(1,3-dioxolan-2-yl)phenyl]acetamide;1-ethylpyrrolidine N-[2-amino-3-[(2S)-1-propan-2-ylpyrrolidine-2-carbonyl]quinolin-7-yl]acetamide;ethane N-[3,4-dihydro-2H-chromen-7-yl-(1-methylpyrazol-4-yl)sulfamoyl]-2-(5-ethyl-6-oxo-1,4-diazepan-1-yl)acetamide 5-N-azido-2,4,6-trimethylpyrimidine-5,7-diamine 1-[(2S)-4,5-bis(4-chlorophenyl)morpholin-2-yl]-N,N-dimethylpyrrolidine-3-carboxamide 2-(3,5-dichlorophenyl)-N-[4-hydroxy-5-(trifluoromethyl)cyclohepta-1,3,6-trien-1-yl]acetamide 3-[1-(3-fluorobenzoyl)piperidin-4-yl]-8-methylpyrido[1,2-a]pyrimidin-4-one [4-amino-5-(2H-benzotriazol-5-yl)-1,3-thiazol-2-yl]-(4-hydroxypiperazin-1-yl)methanone 2-[1,3-dioxolo[4,5-f]isoindol-2-yl(4-phenylbutanoyl)amino]acetic acid 6-chloro-N-(4,5-dihydropyrimidin-2-yl)imidazo[1,2-b]pyridazine-3-carboxamide 3-bromo-6-[4-(3,7-dimethyloctyl)thiophen-2-yl]-1H-pyrrolo[2,3-b]pyridine N-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluorobenzamide;methane (NE)-N-[[3-chloro-1-ethyl-5-(trifluoromethoxy)pyrazol-4-yl]-phenylmethylidene]hydroxylamine 4-cyclopentyloxy-N'-hydroxypyridine-2-carboximidamide 4-[(1E,3Z)-hexa-1,3-dienyl]-N-methoxy-2,6-dimethylaniline 5-[(1R)-2,3-dihydro-1H-inden-1-yl]-4,6-dimethoxy-7-(oxan-2-ylmethoxy)quinazoline N-[(5-chlorothiophen-2-yl)methyl]-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxamide;hydrochloride 2-[3-chloro-5-ethylsulfonyl-4-(5,7,8,10-tetrahydropyrimido[4,5-b]quinolin-6-ylamino)phenyl]propan-2-ol 2-[4-(2,3-dihydroindole-1-carbonyl)piperidin-1-yl]-5-methylpyrimidin-4-amine (5S,7R)-N-[2-(dimethylamino)ethyl]-N-methyl-1-propan-2-yl-5,7-dihydro-4H-pyrano[3,4-c]pyrazole-3-carboxamide (2-chloro-6-ethylphenyl)-dimethoxyborane 4-[3,5-difluoro-2-(methylamino)phenyl]-N'-ethenyl-6-methylidenecyclohexa-2,4-dien-1-imine 3-[2-(4-benzoylphenyl)sulfanylethoxy]pyrrolidine-1,3-dicarboxylic acid 2-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]oxyacetic acid N-[2-(dimethylamino)pyrimidin-4-yl]-N'-(1H-indazol-6-ylcarbamoyl)-2-oxopyrrolidine-1-carboximidamide N-[(Z)-N'-(1H-benzimidazol-2-ylmethoxy)carbamimidoyl]-3,4-difluorobenzamide;ethane N-[(1S,3R)-3-cyanocyclopentyl]-4-[(6-methoxypyridin-2-yl)amino]-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide 1-[5-chloro-2-[1-(4-methoxyphenyl)ethylcarbamoyl]pyridine-3-carbonyl]azetidine-3-carboxylic acid 1-[2,6-bis(2-methylbutan-2-yl)phenyl]-3-(5-tert-butyl-1H-pyrazol-4-yl)-7-hydroxyimidazo[1,5-a]pyridin-8-ium N-(4,5-dimethylpyrimidin-2-yl)-N-phenylbenzamide [5-cyano-2-hydroxy-6-methyl-3-(3-methylbut-2-enoxy)phenyl]urea 7-[4-(difluoromethoxy)phenyl]-2,3-dihydrothieno[3,2-b]pyridine 1-[2,3-bis(4-tert-butylphenyl)cyclopropyl]imidazole 2-[(4S)-4-(3,4-dimethoxyphenyl)-1-ethyl-6-oxopiperidin-3-ylidene]acetate N-[2-(2,5-dimethylphenyl)ethenyl]-1-[4-[(6S)-1,3-dimethyl-5-oxo-7,8-dihydroimidazo[1,2-a]pyrazin-6-yl]phenoxy]ethanimidate;manganese(2+) 1-[(2S)-3,3-difluoro-2-hydroxypropyl]-N-[(2R)-6-[(4-ethynoxycyclohexa-2,4-dien-1-yl)amino]spiro[2.5]octan-2-yl]indole-3-carboxamide 2-ethylimino-5,7,8-trimethylquinoline-3-carboxylic acid 1-(cyclohexen-1-yl)-3-[[4-methoxy-2,6-di(propan-2-yl)phenyl]carbamoylamino]thiourea N-(4,4-difluorocyclohexyl)-3-methoxy-1-methylpyrazole-4-carboxamide (2R)-1-[4-(difluoromethylsulfonyl)anilino]-N,N-dimethyl-2-phenylcyclopropane-1-carboxamide 1-[2,6-di(propan-2-yl)phenyl]-3-[(Z)-4-(2,6-dimethylcyclohexa-1,5-dien-1-yl)but-1-enyl]thiourea 2-[(4R)-4,7-dimethyl-1-oxo-2,3-dihydropyrrolo[3,4-b]indol-3a-yl]-N,5-bis(4-fluorophenyl)-6-propan-2-ylpyrimidine-4-carboxamide 2-[2,4-di(piperidine-1-carbonyl)anilino]acetonitrile 5-amino-3-[4-methoxy-3-(pyrrolidine-1-carbonyl)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile 1-(2-benzoyloxyethyl)-4-(4-hydroxyphenyl)sulfonylpiperazine-2,3-dicarboxylic acid ethane;2-fluoro-1-[4-[2-methoxy-5-(2,2,2-trifluoroacetyl)phenyl]phenyl]ethanone 4-(3,5-difluorophenyl)sulfonyl-1-(1H-pyrrolo[2,3-c]pyridine-7-carbonyl)piperidine-4-carbonitrile (4S)-2,2,3,4-tetramethyl-8-nitro-4H-chromene (3S,4R)-3-[[2-(dimethylamino)-5-fluoropyrimidin-4-yl]amino]-1-methylpiperidin-4-ol;formic acid N'-(3,5-dimethylphenyl)-2,6-dipyridin-4-ylpyrimidine-4-carbohydrazide [1-(aminomethyl)piperidin-3-yl]-[4-[5,7-difluoro-2-(4-fluorophenyl)indol-1-yl]piperidin-1-yl]methanone N-[(1E,3Z)-2,4-dimethylpenta-1,3-dienyl]-5-[4-fluoro-3-[4-(furan-3-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-1H-indazol-5-yl]pyridin-3-amine N-[4-(2,3,3a,5,6,7,7a-octahydro-1H-isoindole-4-carbonyl)phenyl]quinoline-8-sulfonamide 2-(4-chlorophenyl)sulfonyl-2,9b-dihydro-1H-benzo[f]isoindol-3-one N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-4,5-difluoropyridine-2-carboxamide 1-[7,10b-dimethyl-2-(4-methylphenyl)sulfanyl-6H-benzo[c]chromen-5-yl]propan-1-ol (3R,4S)-4-[3-fluoro-4-(2-methylphenyl)sulfonylphenoxy]piperidine 5-(2-fluorophenyl)-1-[2-methoxyethyl(methyl)amino]pentan-3-one 4-methyl-2,6-bis(trifluoromethyl)-1H-pyrimidine-4-carbonitrile 2-[4-[5-(3,6-dihydro-2H-pyran-4-yl)benzimidazol-1-yl]phenyl]benzenethiol 3-[5-(2,6-difluorophenyl)pentyl]-4H-1,2,4-oxadiazol-5-one 2-(1,3-benzodioxol-5-yl)-5-bromo-4-methyl-1H-pyrimidin-6-one 5-(2,3-dimethylbutan-2-yl)-1H-pyridine-4-thione 1-[3,5-bis(trifluoromethyl)phenyl]-2,4-dioxopyrimidine-5-carboxylate 2-[5-(3,4-dichlorophenyl)furan-2-yl]propanoate N-[(3S,4R)-1-benzyl-2-oxopiperidin-4-yl]-1H-pyrrolo[2,3-b]pyridine-6-carboxamide 2-(6,7-difluoro-1-methylnaphthalen-2-yl)propanoic acid 2-(2,4-dimethoxyphenyl)pyridine;ethane N-(1,3-benzodioxol-5-yl)-6-[[[(2Z)-2-ethylidenehexa-3,4-dienoxy]-phenoxyphosphoryl]methyl]pyrimidin-4-amine;formaldehyde 6-[6-bromo-2,3-bis(ethenyl)phenyl]naphthalene-1,7-diamine 5-[6-(4-methylsulfonylphenyl)-2,3-dihydropyridin-4-yl]pyrazin-2-amine N-[4-(2,6-dimethoxyphenyl)-5-pyridin-3-yl-1,2,4-triazol-3-yl]-3,3-bis(sulfanylidene)propanethioamide N-ethylacetamide;4-[2-(8-methoxy-3-propan-2-ylpyrazolo[1,5-a]pyridine-6-carbonyl)-2-azaspiro[3.3]heptan-6-yl]benzonitrile 2-(2-chlorophenyl)-N,N-dimethylethanamine;2-[3-hydroxypropyl(propyl)amino]pyridine-4-carboxylic acid N-[3,5-bis(trifluoromethyl)phenyl]-N-[2-[4-(difluoromethoxy)anilino]-1-hydroxyethyl]-2-oxochromene-3-carboxamide 2-azido-1,3,4,5-tetrafluoro-6-propan-2-ylbenzene N-[2-(2-aminoethoxy)-4-[butan-2-yl(pentan-2-ylidene)amino]phenyl]acetamide;1,3-difluoro-5-methylbenzene 5-chloro-4-[[(2S)-1-(3,4-dimethoxyphenyl)sulfonylpyrrolidine-2-carbonyl]amino]-1-methylpyrazole-3-carboxamide 6-azido-5-methoxy-N,N-dimethylpyridine-3-carboxamide 4-amino-2-[[1-[(4-fluorophenyl)methyl]piperidin-3-yl]methyl]-5-propan-2-yl-1H-pyrimidin-6-one 1-[2-hydroxy-4,6-bis(trifluoromethyl)phenyl]-3-(7-oxodecan-8-yl)urea 4-(2,6-difluorophenyl)-N-methyl-5-(1H-pyrrole-3-carbonyl)-1,2,4-triazole-3-carboxamide N-[(3S,4R)-1-(2-phenylacetyl)-4-(5-propan-2-yloxyfuran-2-carbonyl)pyrrolidin-3-yl]benzamide N-[3-(1,6a-dihydrocyclopropa[a]inden-4-yl)-5-(difluoromethyl)phenyl]-2,3,3a,4,5,7,8,9,10,10a-decahydro-1H-pyrrolo[3,4-g]isoquinoline-6-carboxamide 4-amino-3,6-difluoronaphthalene-1,7-disulfonic acid 6-chloro-N-(4,4,4-trifluorobutyl)pyridine-3-carboxamide 3,5-dimethyl-2H-1,4-benzothiazin-7-amine 5-amino-N-[(Z)-4-[1-(3-butan-2-ylanilino)ethenyl]-2-methylidenepent-3-enyl]thiophene-2-carboxamide N-(5-chloro-2,3-dihydro-1H-inden-1-yl)-2-imidazol-1-yl-6-methoxypyrimidine-4-carboxamide 6-[4-(benzenesulfonamido)phenyl]-2-(3,5-dimethoxyanilino)-N-phenylpyridine-3-carboxamide N-[[4-(2-diazohydrazinyl)phenyl]methyl]methanesulfonamide 3-[(2R)-4,6-dihydroxy-1-methoxy-5-propanoyl-3,4-dihydro-2H-naphthalen-2-yl]propanoic acid N-[2-[4-(3,5-dimethyl-1H-pyrazol-4-yl)piperidin-1-yl]ethyl]-1-phenylpropan-1-amine (1S,3R)-1-methyl-3-(6-methylidene-7H-purin-8-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole 1-(1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-3-[5-[1-(trifluoromethyl)pyrazol-4-yl]-1H-1,2,4-triazol-3-yl]urea 1-[4-[3,5-bis(trifluoromethyl)phenyl]phenyl]ethanone 7-(cyclopropylmethoxy)-2,3-dihydrochromen-4-one N-[3-(tert-butylamino)sulfanylphenyl]-3,6-dichloropyridazine-4-carboxamide N-[(1S)-2-(dimethylamino)cyclohexyl]-6,7-bis(4-fluorophenyl)heptanamide 6-[3-(4,4-difluorocyclohexyl)-4-ethoxyphenyl]-2-ethyl-1H-benzimidazole 2-(3,5-dimethylphenyl)-1H-imidazo[4,5-f]benzimidazole;hydrobromide [4-(2,3-dimethylphenoxy)thieno[2,3-c]pyridin-6-ium-5-yl]methanamine N-(4,6-dimethylpyrimidin-2-yl)-4-[3-ethoxypropanoyl(methyl)amino]benzamide 4-[2-[(3-fluoropyridine-2-carbonyl)amino]propanoyloxymethyl]piperidine-1-carboxylate 2-(3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl)-N'-hydroxypyrimidine-4-carboximidamide (2S,4R)-2-azido-1-[3-cyclopropyl-4-(pyridin-2-ylmethoxy)phenyl]-4-methylsulfonylpyrrolidine N-[3-[2-(5-tert-butyl-1,2-oxazol-3-yl)ethynyl]phenyl]-4-chlorobenzamide 5-(4-chlorophenyl)sulfanyl-2-[3,5-dimethoxy-4-(methylamino)pyridin-1-ium-1-yl]pyridine-3-carbonitrile 1-N-(2,5-dichlorophenyl)-4-N,4-N-dipropylbenzene-1,4-disulfonamide N-[2,4-difluoro-3-(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)phenyl]-1,1-difluoromethanesulfonamide 3,5-dibromo-N'-[6-(methylsulfanylamino)pyridin-3-yl]benzenecarboximidamide N-[2,3,5,6-tetrafluoro-4-(hydroxyiminomethyl)phenyl]cyclopropanecarboxamide 1-(4-aminophenyl)-2,3,6,7,8,9-hexahydro-[1]benzofuro[2,3-d]azepine-4-thione;dihydrochloride 4-(3,4-dichlorophenoxy)-1-[(2E)-penta-2,4-dienyl]piperidine N-[3-[2-amino-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)propan-2-yl]-4,5-dihydroxyphenyl]acetamide N-[3,5-dichloro-4-(2H-quinolin-1-yl)phenyl]-4-methoxybenzamide 3-(4-bromophenyl)sulfanyl-6,7-dimethoxy-1H-indole 3-azido-4-benzylsulfinylphenol 4-[2-[4-(dimethylamino)phenyl]ethynyl]-5,6-difluoroquinazoline-8-carboxamide 4-[4-amino-2,3-bis(ethenyl)imidazo[1,5-a]pyrazin-8-yl]-N-(pyridin-3-ylmethyl)benzamide 6-bromo-2-[4-(difluoromethyl)phenyl]-N-(3,3-dimethylbutanoyl)quinoline-4-carboxamide 3-(3,6-dihydro-2H-pyran-4-yl)-1-[(2E,4Z)-hepta-2,4,6-trien-3-yl]pyrazole 2-(4,5-diethoxy-1H-pyrazole-3-carbonyl)piperidine-1-carboxylic acid (Z)-2,2,4-trifluoro-3-(7H-purin-6-yloxymethyl)pent-3-enoic acid (2S)-4,4,5,5,6,7,8,9,10,10a-decahydrophenanthrene-1,2,3-triol 6-methoxycarbonyl-7,8-dihydronaphthalene-2-sulfonate 5-(2,4-dichlorophenyl)-3-(pyridin-3-ylmethylamino)-1H-pyrrole-2-carboxamide 7-[(3S)-1,2-dihydroxyhexan-3-yl]oxy-8-fluoro-4-oxochromene-6-carboxylic acid 2-bromo-N-(9,10-dioxo-4a,9a-dihydroanthracen-1-yl)-N-(3-methylbut-2-enyl)benzamide 7-[4-(azidomethoxy)phenyl]-1,2-benzothiazol-3-one N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(6R)-5-oxo-3-phenyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-6-carbonyl]benzamide 5-cyclohexyl-2,4-dimethylthiophene 5-bromo-N-[(2R)-1,1-dihydroxy-6-oxoheptan-2-yl]-4-(trifluoromethoxy)pyridine-2-carboxamide N-[2,4-dimethyl-5-(1-piperidin-1-ylethylidene)cyclohexa-1,3-dien-1-yl]-8-fluoro-2-propan-2-ylpyrazolo[4,3-c]quinolin-9-amine ethane;2-methyl-4-(4-phenylcyclohexyl)phenol [1-(3,5-dimethylbenzoyl)piperidin-4-yl]-[(7S)-2,7-dimethyl-3-(3,4,5-trifluorophenyl)-6,8-dihydro-5H-pyrido[3,4-b]pyrazin-5-ium-7-yl]methanone 2-amino-4-(1-ethylindol-5-yl)-6-methylbenzene-1,3-dicarbonitrile 4-[1-(3,5-ditert-butyl-4-hydroxyphenyl)decylsulfonyl]benzenesulfonate (Z)-2-[6-(3,5-dichlorophenyl)pyridine-2-carbonyl]-1,3-bis(methylsulfanyl)prop-2-en-1-one 6-hydroxy-N,2,3-trimethyl-9H-xanthene-1-carboxamide N-methyl-4-[[6-[4-(trifluoromethoxy)phenyl]quinazoline-4-carbonyl]amino]benzamide 2-(4-chloroanilino)-N,N-bis[(4-methoxyphenyl)methyl]-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidine-5-carboxamide 5-chloro-4-[(2R,3S)-1-ethyl-3-hydroxy-7-oxononan-2-yl]sulfonylbenzenesulfonate [[3-chloro-6-[[4-(trifluoromethyl)phenyl]carbamoylamino]pyridazine-4-carbonyl]amino]methanediol 1-[3,5-bis(trifluoromethyl)phenyl]piperazine 3-methyl-6-[[2-(pyrrolidine-1-carbonyl)phenyl]methoxyiminomethyl]-5,7-dihydropyrrolo[2,3-d]pyrimidin-4-one 1-[2-(2,5-dimethylphenyl)ethynyl]cyclohexane [3-bromo-5-(trifluoromethyl)phenyl]-dicyclopropylmethanol N'-[2,6-di(propan-2-yl)phenyl]cyclopropanecarboximidamide 5-[(3S)-2,4-dimethylpentanoyl]-1-phenylpyrazole-4-carboxylic acid 4-[2,5-difluoro-4-(methylamino)phenyl]-1H-pyrrole-3-carboxylic acid 2-(N-ethenylsulfonyl-4,5-dimethyl-2-phenyldiazenylanilino)acetic acid 6-[5-chloro-2,4-bis(phenylmethoxy)phenyl]hexanoic acid 4-azidooxy-6,7,8-trifluoronaphthalene-2-sulfonic acid N-cyclohexyl-N-(2-phenylpropanoyl)nonanamide 3-amino-4-cyano-5-(2,6-dibromophenyl)-1H-pyrrole-2-carboxamide (4S,5R)-4-methyl-5-phenylhexan-3-one (2R)-1,1-diphenylpentan-2-amine;methanol N-[3-cyano-4-(trifluoromethoxy)phenyl]-8-(1,5-dimethylpyrazole-4-carbonyl)-2-oxo-6,7,9,10-tetrahydro-5H-cycloocta[b]pyridine-3-carboxamide 1-[3,5-bis(trifluoromethyl)phenyl]pyrazole ethane;2-methylbuta-1,3-diene;N-(5-methylpyridin-3-yl)acetamide 4-[(4-chlorophenyl)methylamino]-5-fluoro-1H-pyrimidin-6-one 6-[4-amino-3-(trifluoromethyl)piperidine-1-carboximidoyl]-N-pyridin-2-ylpyrimidin-4-amine 3-[(1S)-2,6-diamino-4-methylcyclohexa-2,4-dien-1-yl]oxyphenol (2S)-N-cyclohexyl-5,7-dihydroxy-2-[4-(1-methoxypropan-2-yloxy)phenyl]-8-[(5-nitrothiophen-3-yl)methyl]-1,6-naphthyridine-6-carboxamide (7S)-8-cyclopentyl-2-[1-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]ethylamino]pyrido[2,3-d]pyrimidine-7-carboxamide (2R)-4,8-dimethoxy-N-[(1S)-1-(3-phenylphenyl)ethyl]decan-2-amine 1-[4-(dimethylamino)cyclohexyl]-2-[5,6,7,8-tetrahydroquinolin-3-yl(triazolo[4,5-b]pyridin-3-ylmethylsulfonyl)amino]benzimidazole-5-carboxamide 2-[5-methyl-4-(3-pyrrolidin-1-ylpropoxy)pyrimidin-2-yl]phenol 4-[(4R,5S)-5-ethenyl-2,3,4-trihydroxy-6-[(4-methoxyphenyl)methoxycarbonyl]oxan-4-yl]benzoic acid 2-[1-(6,7-dimethoxyquinazolin-4-yl)pyrrolidin-3-ylidene]-6-iminocyclohexan-1-one 5-[3-(azetidin-2-ylmethoxy)phenyl]imidazolidine-2,4-dione 1,2-diamino-4-[3-methoxy-4-(2,2,2-trifluoroethoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile N-methyl-2,6-dioxo-5-phenylmethoxypyran-3-carboxamide 2-bromo-6,7,8,9-tetrahydro-5H-imidazo[1,2-d][1,4]diazepine-3-carboxamide 6-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-N-ethyl-9-propan-2-ylpurine-2,8-diamine 4-chloro-2-(1,3-dioxoisoindol-2-yl)-5-phenylmethoxybenzenesulfonate 3-methyl-N-[(1R,2S)-2-phenylmethoxycyclopentyl]benzamide 5-bromo-2-(4-chlorophenyl)pyridine 4-[(1S)-3-cyano-1-(2,6-dimethylphenyl)propoxy]-N-ethylidenebenzenecarboximidamide (Z)-4,5-dimethoxy-1-[4-[2-[4-[1-(3-phenoxypropyl)piperidin-4-yl]phenoxy]ethyl]phenyl]hex-5-en-1-one N'-[(Z)-(3-chloro-4-hydroxyphenyl)methylideneamino]-N-(thiophen-2-ylmethyl)oxamide 5-[5-chloro-2-[(4-methylsulfonylpiperazin-1-yl)methyl]phenyl]-7-(2,3-dihydro-1H-inden-5-ylamino)imidazo[1,2-c]pyrimidine-8-carboxylic acid [2-[amino-[(Z)-1-aminobut-1-enyl]amino]phenyl]-piperidin-4-ylmethanone;ethane 5-[(4,6-dimethoxypyrimidin-2-yl)carbamoylamino]naphthalene-1-sulfinic acid 4-[1,3-bis(4-hydroxyphenyl)propan-2-yl]cyclohexane-1-carboxylic acid 3-azido-4,5-dichlorobenzaldehyde 4-[3,5-bis(trifluoromethyl)phenyl]-1-(2,6-diethoxypyridin-4-yl)sulfonylpiperazine N-(2,3-dihydro-1H-inden-5-yl)-4-methoxy-6-methylpyrimidine-5-carboxamide 1-[2,3-bis(methoxymethyl)phenyl]-4-methylpiperazine 3-[4-[(3R)-pyrrolidin-3-yl]oxyphenyl]sulfanylpyridine 3-(N-(2,4-dichloropyrimidin-5-yl)anilino)propanoic acid 2-[N-(4-chlorobutyl)-3,5-difluoroanilino]acetamide 5-N,9-N-diethyl-2,3,4,7,8,10-hexahydrobenzo[h][1,4]benzoxazine-5,7-dicarboximidamide (3R)-N,N-dimethyl-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-3-carboxamide;ethane (2R)-2-amino-3-phenyl-N-[2,4,5-trifluoro-3-(1-pyrimidin-4-ylindazol-6-yl)oxyphenyl]propanamide (E)-2-[1-[5-chloro-6-[[4,6-dimethyl-5-(trifluoromethoxy)-1H-benzimidazol-2-yl]methyl]pyridine-3-carbonyl]piperidin-4-ylidene]ethenesulfinate 2-[5-(6-methoxynaphthalen-2-yl)tetrazol-1-yl]acetic acid N-(2,4-dichloropyrimidin-5-yl)-N-[1-(2H-tetrazol-5-ylmethylsulfonyl)piperidin-3-yl]acetamide 1-benzylsulfonyl-3-tert-butyl-6-chloroindole 1-[(2R)-1-aminopyrrolidin-2-yl]pyrimidine-2,4-dione;hydrochloride 2-[(4-bromophenyl)sulfanylmethyl]thiophene 3-azido-5-chloro-2-(1H-indol-2-yl)phenol 1-[(3S)-5,7-dihydroxy-3-methylhept-6-enoyl]indole-2,3-dione N-[3-[5-methyl-4-[(2Z)-penta-2,4-dienyl]sulfanyltriazol-1-yl]propyl]-6-phenoxypyridine-2-carboxamide 3-[5-[2,4-bis(methoxycarbonyl)phenyl]pyridin-3-yl]-N,1-diethylpyrazole-4-carboxamide N-[[2,5-difluoro-4-(methylsulfamoyl)phenyl]methyl]-6-morpholin-4-ylpyridine-3-carboxamide 2-[5-(3,4-dichlorophenyl)-1H-imidazol-4-yl]pyridine 5-(4-chlorophenyl)-3-ethoxy-1,2-thiazole 2-amino-N-[(4,6-dimethyl-1H-benzimidazol-2-yl)methyl]quinoline-4-carboxamide 2-[3,5-dichloro-N-(2,2-dimethoxyethyl)anilino]-4-nitrophenol 2-[[4-(pyridine-3-carbonylamino)piperidin-1-yl]methyl]benzoic acid 1-(4-methylpiperazin-1-yl)-2-pyridin-3-ylbutan-1-one [2-amino-4-(methyliminomethyl)phenyl]-[3-[6-chloro-7-fluoro-1-[2-[3-(4-methylpiperazin-1-yl)propoxy]ethyl]indol-3-yl]azetidin-1-yl]methanone 2-methyl-6-(1H-pyrrolo[3,2-b]pyridine-5-carbonyl)-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one 3-[4-(2,2-dimethylpropoxy)anilino]butan-2-one 1-[5-(2-aminopyridine-4-carboximidoyl)-6-methylpyrimidin-4-yl]-N,N-dimethylpiperidine-3-carboxamide 3-methylsulfanyl-N-[(2S)-1,1,1-trifluoropropan-2-yl]-5-(6H-pyrrolo[3,4-c]pyrrole-1-carbonyl)thiophene-2-carboxamide 2-[(4,5-dimethyl-1H-pyrazole-3-carbonyl)amino]pentanoic acid 2-(9H-fluoren-1-yl)cyclopentan-1-one 4-[(4R)-3-methylsulfanylpiperidin-4-yl]oxy-1H-indazole N-[3,5-bis(trifluoromethyl)phenyl]-6-chloropyridine-2-carboxamide 2-azido-3,5-ditert-butylbenzaldehyde N-[(3E)-2-methoxyhexa-1,3,5-trien-3-yl]-1,3-benzoxazol-2-amine 5-(cyclopropylmethoxy)-4-iodopyridine N-cyclohexyl-2-(7,8-dimethyl-1-oxo-3,4-dihydroisoquinolin-2-yl)acetamide 1-[2,6-difluoro-4-(6-methoxyheptyl)phenyl]pyrazolidine 4-[(4S)-3-ethyl-2,5-dioxoimidazolidin-1-ium-4-yl]-N-[[2-fluoro-6-(trifluoromethoxy)phenyl]methyl]benzamide 2-bromo-5-[(E)-2-(4-hydroxyphenyl)ethenyl]phenol N-[6-amino-5-(4-chlorobenzoyl)pyrazin-2-yl]-4-(4-methylpiperazine-1-carbonyl)benzamide 3-(6,8-dimethyl-[1,2]oxazolo[5,4-f][1,3]benzothiazol-4-yl)benzenesulfonic acid 1-[5-fluoro-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl]pyrrolidin-2-one 2-[5-bromo-6-[(4-hydroxyphenyl)methylamino]-1H-benzimidazol-2-yl]phenol 4-[4-[(6-methylpyridin-3-yl)amino]phenoxy]-1H-triazole-5-carboxylic acid;hydrochloride 1,3-dichlorobenzene;1-[1-[4-fluoro-2-(trifluoromethyl)phenyl]ethyl]piperidine (2Z)-N-[5-(7-methyl-1H-indol-3-yl)pentyl]-6,8-dihydro-5H-oxocine-7-carboxamide N-(1,3-benzothiazol-2-ylmethylideneamino)-4-methylbenzenesulfonamide (4E,5Z)-2-methyl-1,3-diphenylocta-2,5,7-trien-4-ol 2-bromo-N-(4-hydroxybutyl)-N-[4-(pyridin-2-ylsulfamoyl)phenyl]benzamide 6-[1-(2,3-dihydroindole-1-carbonyl)cyclobutyl]pyridine-3-carboxamide 1-[5-(4-bromophenyl)-1,2,4-oxadiazol-3-yl]butan-1-ol (2R)-1,4-bis[2-methoxy-5-(3-phenylpropyl)thiophen-3-yl]pentan-2-amine N'-(6-cyclohexyloxypyridin-3-yl)oxamide N-[(3-imidazol-1-ylphenyl)methyl]imidazo[4,5-b]pyridine-3-carboxamide N-ethyl-1,3-dihydroisoindole-2-carboxamide N-[5,7-difluoro-6-(3,4,5-trimethoxyphenyl)isoquinolin-8-yl]-3,4-dihydro-1H-2,4-benzoxazine-6-sulfonamide [2-(3,4-dihydropyridin-5-yl)phenyl]methanethiol 2-[2-oxo-1-(thiophene-3-carbonyl)pyrrolidin-3-yl]sulfanylacetamide 2-(1-methylcyclopentyl)oxypyridine 4-[6-(2,3-difluorophenyl)pyridin-2-yl]pyridine-2,3-diamine 2-[[2,4-bis(difluoromethoxy)phenyl]methyl]-N-cyclopropylideneimidazo[1,5-a]pyridine-8-carboxamide;cyclohexane 2-methoxy-N-[5-methyl-3-(2,4,6-trichlorophenyl)pyrazol-1-yl]benzenesulfonamide N-[5-chloro-2,4-bis(phenylmethoxy)phenyl]formamide 2-methyl-N,3-diphenylbutanamide 3-[1-(2,6-difluorophenyl)-2-[4-(1H-indol-5-ylmethoxy)anilino]-4-oxopyrimidin-5-yl]benzamide N-[4,6-dimethyl-2-(1H-pyrazol-5-yl)pyrimidin-5-yl]-N'-ethenylsulfonylpropanimidamide 1-[4-(9,10-diiminophenanthridin-6-yl)phenyl]ethanone;2-phenylpyridine 3-[(2S)-5,7-dihydroxy-8-methoxy-2-(4-morpholin-4-ylphenyl)chromene-2-carbonyl]-N-phenylbenzamide 2-[1-(8-fluoroquinolin-3-yl)ethenyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-6-ol 5-amino-N-[4-(1,2-dihydroimidazo[4,5-b]pyridin-3-yl)phenyl]pentanamide (2R)-2,6,8-trihydroxy-7-(4-methoxyphenyl)octanal N-[(6S)-8-chloro-10-oxo-2-phenyl-3,4-dihydro-1H-pyrimido[1,2-b]indazol-6-yl]-2,5-bis(trifluoromethyl)pyrazole-3-carboxamide N-[1-azidooxy-2,3-di(propan-2-yl)phenyl]benzamide N-(2,3-dihydro-1H-inden-5-yl)-4-fluoro-9H-pyrimido[4,5-b]indole-7-carboxamide (2R)-1-[4-(2,6-dimethylphenyl)-1,3-thiazol-2-yl]pyrrolidine-2-carboxylic acid N-(6-methylheptan-3-yl)aniline (2-chloroquinolin-3-yl)boronic acid N-[4-amino-1-(1,3-thiazol-2-yl)piperidin-3-yl]-2-chloro-5-oxopyrido[4,3-d]pyrimidine-8-carboxamide N-[(2S,3R)-1-amino-5-cyclopropyl-4-oxo-2-phenylpentan-3-yl]-2-[2-(4-methoxyphenyl)ethynyl]benzamide 2-[4-[5-[2-ethyl-3-[(5-methylthiophen-2-yl)sulfonylamino]phenyl]pyridin-2-yl]piperazin-1-yl]-2-oxoacetamide 4-N,4-N-dimethylbenzene-1,2,4,5-tetramine;2-[3-(4-methylphenyl)propanoylamino]benzoic acid [2-methoxyethyl(phenyl)phosphoryl]benzene 4-tert-butyl-N-[4-(1H-imidazol-5-ylmethoxy)cyclohexa-2,4-dien-1-ylidene]benzenesulfonamide 3-[(1S)-2,2-dimethylcyclopentyl]oxy-5-fluorobenzenesulfonamide 4-[(6-tert-butylpyridin-2-yl)amino]-N-ethanimidoyl-3-methoxybenzenesulfonamide 4-[(2Z,5R)-3,7-dimethylocta-2,6-dienoxy]-N,N-bis(4-fluorophenyl)benzamide N-[(2R)-4-[2-(4-chlorophenyl)pyrrolidin-1-yl]butan-2-yl]-5,6-dimethoxy-1H-indole-2-carboxamide 1-(4-bromophenyl)-2-[methyl(1,3-thiazol-5-ylmethyl)amino]ethanone N-[(4,5-dimethyl-1H-pyrazol-3-yl)methyl]-6-oxo-2-phenyl-1H-pyrimidine-4-carboxamide [2-hydroxy-5-[3-(4-hydroxyphenyl)propyl]phenyl]azanium 2-(2,4-dichloropyrimidin-5-yl)sulfanyl-4,7-bis[3-(trifluoromethoxy)phenyl]pyrido[2,3-d]pyrimidine N-(2,4-dichloropyrimidin-5-yl)-3-methoxybenzamide 4-(aminomethyl)-N-[2-[(3R,5S)-3,5-dimethoxypiperidin-1-yl]ethyl]benzamide;dihydrochloride 2-amino-4-methylpentanamide;(Z)-but-2-ene;7,8-difluoro-N-heptan-3-ylidene-6-piperidin-1-yl-1H-isoquinoline-4-carboxamide (3E)-1-cyclopentyl-N-[2-(2,4-difluorophenyl)ethyl]-3-ethylidenepyrrolidine-2-carboxamide 2-[4-(1,3-benzothiazol-6-ylsulfonyl)piperazin-1-yl]-N-ethyl-N-(2-methoxypyridin-4-yl)acetamide N-[2,4-difluoro-3-(5-methylpyrazolo[1,5-a]pyrimidin-7-ium-3-yl)phenyl]formamide 1-benzyl-4,7-dihydroxy-3-phenylmethoxyquinolin-2-one N-[1-(2,3-dihydropyridin-4-yl)-5-fluoro-7-methoxy-2,3-dihydroindol-6-yl]-1H-pyrrolo[2,3-b]pyridine-4-carboxamide N-[2,6-dimethyl-4-(1H-pyrazol-4-yl)phenyl]-3-fluoro-5-(triazol-2-yl)benzamide 2-(3,4-dibromophenyl)-5-methylfuran 3-[1,2-diamino-4-(furan-2-yl)-6-oxopyrimidin-5-yl]propanoic acid 6-[3-(4,5-dihydro-1H-imidazol-2-yl)benzoyl]-N-[2-methoxy-5-methyl-4-(4-methylpiperazin-1-yl)phenyl]-7,8-dihydro-5H-2,6-naphthyridine-3-carboxamide 1-[2-(3,5-difluorophenyl)acetyl]-N-(4-methoxypyridin-2-yl)pyrrolidine-2-carboxamide 2-[2-hydroxyethyl(2H-tetrazol-5-yl)amino]ethanol (3S,4R)-4-azido-1-(2,6-difluorobenzoyl)pyrrolidine-3-carbonitrile 6-[3-(trifluoromethyl)anilino]-1H-pyrimidine-2,4-dione 6-N-[(4,5-dichloro-1H-imidazol-2-yl)methyl]-1H-indole-3,6-diamine 5-fluoro-N-(2,3,6-trifluorophenyl)pyrazine-2-carboxamide 4-chlorobutanal;N,2-dimethylpyridine-3-carboxamide;ethane;1-methoxypent-3-enylcyclopropane 4-[(2,6-difluorophenyl)methyl]-1H-tetrazol-5-one N-[4,6-difluoro-1-[(3R)-pyrrolidin-3-yl]indazol-5-yl]-2-(1H-indol-3-yl)acetamide N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-5-[4-[2-methoxyethyl(methyl)amino]phenyl]benzamide 2-[(4-chloro-5,7-difluoroquinazolin-2-yl)methylideneamino]-3-sulfanylidenepropanoic acid (2S,4R)-1-[5-chloro-3-fluoro-6-oxo-7-(trifluoromethyl)thieno[3,2-b]pyridine-2-carbonyl]-4-hydroxypyrrolidine-2-carboxamide 1-[5-(4-chlorophenyl)-2-methylfuran-3-carbonyl]-N-(3,5-difluorophenyl)piperidine-4-carboxamide 2-[4-(dipropylamino)butanoyl]-N-(3-fluorophenyl)-1,3-thiazole-5-carboxamide N-[(E)-(5,7-dimethoxyimidazo[4,5-b]pyridin-3-yl)methylideneamino]pyridine-2-carboxamide 3-[5-fluoro-2-(2-methylpropyl)phenyl]piperidine 2-N,8-N,3-trimethyl-5-N-[6-(2-phenylethyl)pyrimidin-4-yl]imidazo[1,2-b]pyridazine-2,8-diamine 5-chloro-6-methyl-1-[1-(3-phenylmethoxypropanoyl)piperidin-4-yl]indole-2,3-dione (2R)-N,3,3-trimethyl-2-[(4-phenylpiperazine-1-carbonyl)amino]butanamide N-[4-fluoro-3-(6-oxo-1H-pyridin-2-yl)phenyl]propanamide N-methyl-5-(1-methylpyrazol-3-yl)pyridine-2-carboxamide 1-[4-bromobutan-2-yl(hexadecyl)amino]-3a,9a-dihydrobenzo[f]isoindole-5,10-dione 3-(3-azidocyclobutyl)-N,4-dimethoxybenzamide 2-[4-chlorobutyl(naphthalen-1-yl)amino]propanoic acid N-[(4-chlorophenyl)methyl]-7-hydroxy-3,6-dioxoheptanamide N-[(Z)-(2,3-dichlorophenyl)methylideneamino]-4-methyl-1H-pyrrole-3-carboxamide 3-amino-5-[4-bromo-2-(trifluoromethyl)phenyl]-4-cyano-1H-pyrrole-2-carboxamide 4-N-[6-methyl-2,3-bis(4-nitrophenyl)cyclohex-2-en-1-ylidene]benzene-1,4-dicarboxamide 6-(2-methylsulfanylethylamino)-4-phenylthieno[3,2-b]pyridine-7-carboxylic acid 7-benzyl-5-(3,4-dichlorophenyl)-2,3-dihydrothieno[3,4-b][1,4]dioxine;N-cyclohexyl-N'-methanimidoylmethanediamine (E)-N',3-dihydroxy-2-[5-[4-(piperidin-1-ylmethyl)phenyl]furan-2-yl]but-2-enediamide 4-[2-(1,3-benzothiazol-2-yl)phenyl]benzenesulfonic acid 3-[2,6-di(propan-2-yl)phenoxy]oxolane 1-(3,4,6,7,8,9-hexahydro-1H-pyrimido[5,4-b]indolizin-2-yl)butan-2-one 3-(2,6-dichlorophenyl)-7-[(4-methoxyphenyl)methylamino]-1-(2-methylpyridine-4-carboximidoyl)-1,8-naphthyridin-2-one N-benzylsulfanyl-4-(3-chlorophenyl)aniline N-azido-2,4-bis(3-ethenylanilino)pyrimidine-5-carboxamide 2-methyl-N-[5-(oxan-4-yl)-1H-pyrazol-3-yl]benzamide 6-[2-[1-(4-ethylphenyl)cyclopentanecarbonyl]-3,4-dihydro-1H-isoquinolin-5-yl]pyridine-2-carboxylic acid 1-(4,6-dimethylpyrimidin-2-yl)-3-[2-(6-oxopyridin-2-yl)ethoxy]pyrazole-4-carboxamide 6-[3,5-di(propan-2-yl)phenyl]iminocyclohexa-2,4-dien-1-imine N-[4-chloro-6-(2-fluoro-5-methoxyphenyl)pyrimidin-1-ium-2-yl]acetamide 5-[2,6-difluoro-3-methyl-4-(2H-pyrimidin-1-yl)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 1-[(4S)-6,11-dihydroxy-2-methyl-8-oxa-3,10-diazatricyclo[7.4.0.02,7]trideca-1(13),9,11-trien-12-yl]ethanone (Z)-2,3-bis[4-amino-5-(dimethylamino)-1H-pyrimidin-2-ylidene]prop-2-enethioamide N-[4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]-N'-(2-iodopyridin-3-yl)-4-oxobutanimidamide N-[(3,4-dimethylphenyl)-phenylmethyl]-6-oxo-2-propan-2-ylidene-1,3-oxazinane-4-carboxamide 5-[1-(3,4-difluorophenyl)ethoxy]quinazoline 2-[(6S)-8-cyclopentyl-5-hydroxy-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]benzoic acid 6,8-dimethyl-2-(trifluoromethoxy)quinoline 2-chloro-N-[4-(3,5-dimethylpyridin-2-yl)phenyl]benzamide 5-(difluoromethyl)-2-[[3-[6-[4-[1-(oxetan-3-yl)piperidin-4-yl]phenyl]pyridin-3-yl]oxycyclobutyl]amino]pyrimidine-4-carbonitrile 5-[4-(2,3-dichloroanilino)phenyl]sulfinyl-N-hydroxypentanamide (2R,3S)-N,3-dihydroxy-5-oxo-8-[4-(piperidine-1-carbonyl)piperazin-1-yl]-2-thiophen-2-yloctanamide 6-fluoro-5-[2-(4-methoxycyclohexyl)ethylsulfamoyl]pyridine-3-carboxylic acid 2-[[4-(methylamino)phenyl]iminomethyl]phenolate;nickel(2+);1,3,5-triaza-7-phosphatricyclo[6.4.0.02,6]dodeca-2(6),4,8,10-tetraene 5-[5-(2,4-difluorophenyl)-4H-1,2-oxazol-3-yl]benzene-1,3-diamine 7-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-hydroxyethyl)-8-[(4-methoxyphenyl)methyl]-6-iminopurine-3-carboxamide 2,3-dihydroxy-6,7-dimethylchromene-4-thione 2-(3,4-dihydroxyphenyl)-7-methoxychromene-5,8-dione 3-(2,4-difluorophenyl)sulfonyl-5-propan-2-yl-1H-imidazole-2-thione 1-ethyl-5,6-difluoro-2,3-dihydrobenzimidazole-4-carbonitrile 2-[3-bromo-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenol 2-N,4-N-bis[(E)-1H-indol-3-ylmethylideneamino]pyrimidine-2,4-diamine 2-(benzylamino)-5-hydroxypentanoic acid (1S,2R)-N-benzyl-2-[(4-methoxyphenyl)sulfonylamino]-3,3a,4,5,6,6a-hexahydrocyclopenta[b]furan-2-carboxamide (1R,2S)-N'-[[4-chloro-3-fluoro-5-(trifluoromethyl)phenyl]methoxy]-2-isoquinolin-6-ylcyclopropane-1-carboximidamide N-[(3S,4S)-1-(benzenesulfonyl)-3-methylpiperidin-4-yl]-2-phenylacetamide N-[[1-(3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl)isoquinolin-3-yl]methyl]cyclohexanamine 4-chloro-N'-(1-chloropropyl)benzenecarboximidamide;hydrochloride 3-[2,6-dimethyl-4-[1-(oxiran-2-yl)ethyl]phenoxy]-1,5-bis(4-hydroxyphenyl)pentane-1-thione N-[1,5-bis(4-fluorophenyl)pyrazol-3-yl]-2-methylpyridine-3-carboxamide 4-(3-bromo-5-chlorophenyl)-2,6-dioxo-1,3-diazinane-5-carbonitrile 2-[4-(3,4-dihydronaphthalen-1-yl)-2-phenylimino-1H-pyrimidin-6-ylidene]propanedinitrile N-(5,6-dichloropyridin-3-yl)sulfanylmethanamine N-[(3R)-1-[[4-[ethyl(2-methoxyethyl)amino]quinazolin-2-yl]methyl]pyrrolidin-3-yl]prop-2-enamide 5-ethyl-6,7-dimethoxy-3H-quinazolin-4-one 2-[6,7-dimethoxy-4-[(1E)-1-(3-propan-2-ylphenyl)buta-1,3-dien-2-yl]quinazolin-8-yl]-N-ethylsulfanylethanamine 4-(3-chloro-2,5-dimethoxyphenyl)-6-methylidene-1H-pyrimidine 6-(N,4-dimethylanilino)-2-[4-[4-(propan-2-ylsulfonylamino)phenyl]pyridin-3-yl]-1H-benzimidazole-4-carboxylic acid 3-[4-(6,7-dihydroquinolin-4-yl)piperazine-1-carbonyl]benzonitrile [6-(4-chloroanilino)-7-fluoroquinolin-5-yl]boronic acid 4-[[5,6-dichloro-1-(2-pyridin-3-yloxyethyl)benzimidazol-2-yl]methyl]benzoic acid 6-azido-1,2,3,4,5-pentafluoroanthracene 3-[(2S,4R)-4-amino-1-(2-chlorobenzoyl)pyrrolidin-2-yl]-5-phenylthieno[3,4-d]pyrimidin-4-one [3-[2,6-bis(propanoylamino)pyridin-4-yl]oxy-4-(dimethylcarbamoyl)phenyl]carbamic acid 4-[[5-(2,3-dihydro-1H-inden-5-yl)-6-phenyl-1H-pyrrolo[2,3-b]pyridin-4-yl]oxymethyl]-N,N-dimethylbenzamide 1-cyclopentyl-N,N-dimethyl-3,4-dihydro-2H-naphthalen-1-amine [[2-(4,5-dimethylpyrazol-1-yl)phenyl]-hydroxyphosphinothioyl]oxidanium N-[3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclohexyl]thiophene-2-sulfonamide [7-chloro-3-(2,6-dichlorophenyl)-5H-pyrido[4,3-d]pyrimidin-4-yl]hydrazine;ethane (5S)-2-(3-chloroanilino)-N-(4-methoxyphenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide [(5-chlorothiophene-2-carbonyl)amino]carbamodithioic acid 2-N-benzyl-1,3-benzothiazole-2,6-diamine (1-ethoxy-2,3-dihydroindol-5-yl)-[(4R)-4-methoxy-7-azaspiro[3.5]nonan-7-yl]methanone (2R)-3-[4-[5-fluoro-2,6-dioxo-1-propan-2-yl-8-(trifluoromethyl)quinazolin-7-yl]phenyl]-N,N',N'-trimethylpropanehydrazide 3-[4-methoxycarbonyl-N-(1,2,4-triazol-4-yl)anilino]butanoic acid 2-[2-amino-5-(4-ethoxy-3,3-dimethylbut-1-ynyl)phenoxy]propanal;formaldehyde N-[6-chloro-5-(trifluoromethoxy)naphthalen-1-yl]-4,5-dihydro-1H-imidazol-2-amine 3-fluoro-N,4,6-trimethylimidazo[1,5-a]pyridine-7-carboxamide 4-[2-(3,5-dichlorophenyl)pyrrolidin-1-yl]sulfonyl-N'-methylbenzohydrazide (2S)-1-[4-[4-[3-chloro-5-methyl-4-[(4-nitrophenyl)methoxy]anilino]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]piperazin-1-yl]propan-2-ol N-[2-amino-5-(1-methylpyrazol-4-yl)phenyl]-6-azidooxypyridine-3-carboxamide 2,4-diaminopyrimidine-5-carbonitrile;1-ethyl-3-phenyl-8-[2-(1H-pyrazol-4-yl)ethynyl]isoquinoline 2-methylsulfanyl-3-(4-phenylcyclohexa-1,5-dien-1-yl)-6H-pyrazolo[1,5-a][1,3,5]triazin-4-one N-(2,6-dichlorophenyl)-1H-pyrrole-3-carboxamide 2,6-dibromo-4-[(4R)-1,8-dichloro-7H-quinazolino[2,3-a]benzimidazole-2-carbonyl]phenolate 2-[4-[(3,5-dichloropyridin-4-yl)carbamoyl]phenyl]acetic acid;hydrochloride 4-amino-N'-[(4-fluorophenyl)methyl]-1,2,5-oxadiazole-3-carboximidamide [1-(1,5-dimethylbenzimidazole-2-carbonyl)piperidin-4-yl]-(1H-pyrrol-3-yl)methanone 2-azido-N',1-dimethyl-6H-pyrrolo[3,4-c]pyridine-4-carbohydrazide 7-cyclopropyl-8-(6-cyclopentyloxypyridin-3-yl)-5-methylpyrrolo[1,2-a]quinoxaline 4-[3-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]benzonitrile 5-[3-(4-methylphenoxy)pyrrolidine-1-carbonyl]-1H-pyrrole-2-carbonitrile 2-ethyl-4,6-bis[(3-hydroxyphenyl)sulfanyl]phenol 5-chloro-N-[2-(1-pyridin-3-ylpiperidin-4-yl)ethyl]pyrimidine-4-carboxamide [3-(2-chlorophenyl)iminospiro[1,4-dihydroquinoxaline-2,3'-pyrrolidine]-5'-yl]-pyridin-2-ylmethanone N-[2-(2-aminoethyl)phenyl]-1H-benzimidazole-4-carboxamide N-[2,6-difluoro-4-(1H-1,2,4-triazol-5-yl)phenyl]-3-methoxy-4-phenylpyrrolidine-1-carboxamide N-cyclopropylsulfonyl-2,3-dimethoxybenzamide 5-(2-methoxyethyl)-6,8-dihydro-[1]benzothiolo[3,2-c]pyrazole 4-(2,6-diamino-3,5-dicyano-4H-pyran-4-yl)benzenesulfonamide 3-(difluoromethoxy)-2-(3,5-difluorophenyl)benzoic acid 1-[4-(4-aminophenyl)butoxymethyl]pyrazole-3,5-diamine (E)-3-[5-butanoyloxy-2-fluoro-4-methyl-6-prop-1-en-2-yl-3,4-dihydronaphthalen-1-yl]prop-2-enoic acid N-[2,6-di(propan-2-yl)phenyl]-1-pyridin-3-ylmethanimine 3-[(4-fluorophenoxy)methyl]-N'-hydroxypyridine-2-carboximidamide (2E)-N-(2,3-dihydro-1H-inden-5-ylmethyl)-2-[(1-ethylquinolin-4-ylidene)hydrazinylidene]propanamide (5Z)-5-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-2-(2,3-dichlorophenyl)imino-1,3-thiazolidin-4-one 6-(2,4-difluorophenoxy)-5-methylpyridazine-3-carboxylic acid N-[4-(2,3-dimethylphenyl)pyridin-3-yl]-1H-benzimidazole-4-carboxamide 4-[2-(5-fluoropyridin-3-yl)oxypropanoyl]piperazine-1-carboxamide 2-[5-(4-methoxy-6-methylcyclohexa-1,3-dien-1-yl)imidazo[2,1-b][1,3]thiazol-3-yl]ethanamine 2-(4-acetyl-N-prop-2-enoylanilino)octanoic acid (2S,3R)-3-azido-1-[4-(1,1-difluoroethyl)anilino]butan-2-ol 2-[4-(1,3-benzothiazol-2-yl)pyridin-1-ium-1-yl]-N-(3,5-dimethoxyphenyl)acetamide 1-[2,6-difluoro-4-(5-propylpyrimidin-2-yl)phenyl]ethanamine;dihydrochloride 3-(4-methylphenyl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole 4-[3,5-dimethyl-N-(2-oxopropyl)anilino]butanoic acid N-(3,4-dimethylphenyl)-1-azabicyclo[2.2.2]octan-5-imine 3-cyclobutyl-6-(4,5-dimethyl-1H-imidazol-2-yl)-1,2-benzoxazole (5E)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[(2,4-diethoxyphenyl)methylidene]-1,3-thiazolidin-4-one (4R)-3,4-dimethyl-1-phenyl-6,7,8,9-tetrahydro-5H-pyrazolo[4,3-b]quinoline 1-[4-(7,8-dihydroxynaphthalen-2-yl)sulfonylpiperazin-1-yl]propan-1-one 2-amino-3-[(4R)-3,8,12-triazatricyclo[6.5.0.02,7]trideca-1,6,9,11-tetraen-8-yl]propanal 5-[(4-azidophenyl)diazenyl]benzene-1,2,3-triol N-[3,5-bis(trifluoromethyl)phenyl]-2-[4-[(3-chloro-1,4-dihydroxycyclohexa-2,4-dien-1-yl)methylideneamino]phenyl]acetamide 4-[5-chloro-6-(2,5-dimethylpyrrol-1-yl)pyridin-3-yl]-N-[4-(trifluoromethoxy)phenyl]pyrimidin-2-amine;2-formamido-2-propan-2-yloxyacetic acid 2-[5-(ethylaminomethyl)pyridin-3-yl]-4-phenyl-6,7-dihydropyrrolo[1,2-a]pyrimidine-8-carboxamide;hydrochloride 4-(azetidine-1-carboximidoyl)-3-methylaniline;5-chloro-3,6-dimethylpyrazin-2-amine N-[2-(2,6-dichlorophenyl)ethyl]-5-fluoro-4H-thiopyran-3-carboxamide [4-methyl-3-(trifluoromethyl)phenyl]-spiro[5,6-dihydrocyclopenta[d]pyrimidine-7,3'-piperidine]-1'-ylmethanone 4-(4-acetylphenyl)benzenecarboximidamide;1,2-dimethoxy-5-propan-2-ylidenecyclopenta-1,3-diene 6-[4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-2H-azepine 4-(2,3-dihydro-1H-imidazo[1,5-a]pyridine-8-carbonyl)piperazin-2-one 4-(2,3-dichlorophenyl)-5-[5-methoxy-1-(4-sulfamoylphenyl)imidazol-4-yl]pyrimidine 5-[1,3-dimethyl-5-(trifluoromethyl)pyrazol-4-yl]-2H-tetrazole 2,6-bis[5-chloro-1-(4-methoxyphenyl)sulfonylpyrrolo[2,3-b]pyridin-2-yl]benzaldehyde 5-(2,6-dimethoxyphenyl)sulfanyl-1-(4-fluorocyclohepta-1,3,7-trien-1-yl)pyrazole 2,3-dimethyl-5-[(4-propan-2-ylphenyl)methylidene]bicyclo[5.1.0]oct-1-ene 3-[5-(2,4,6-trichlorophenyl)tetrazol-2-yl]benzenesulfonic acid 6-[(4,5-dimethoxy-2-nitrophenyl)iminomethyl]-1H-indole-3-carbonitrile 5-bromo-2-[(2S)-4,4-dimethyloxolan-2-yl]pyridine N-[3,4-dioxo-1-(2H-triazol-4-yl)butan-2-ylidene]benzamide 2-(5-propan-2-ylthiophen-2-yl)propanedioate 2-bromo-N-(4-chlorobutyl)-N-pyridin-3-ylbenzamide 7-(azidomethyl)-2-butanoyl-3,4-dihydroisoquinolin-1-one N-cyclohexyl-N-(4,5-dimethyl-2-phenyldiazenylphenyl)benzamide N-(2,4-dimethoxyphenyl)sulfonyl-3-hydroxy-5-[[3-methyl-1-(oxan-4-yl)pyrazol-4-yl]amino]pyridine-2-carboxamide 1-[4-(2,3-dihydro-1H-indene-5-carbonyl)piperazin-1-yl]propan-1-one (2S)-3-amino-1-[2,4-bis(4-chlorophenoxy)phenyl]propan-2-ol 2-aminopyrazolo[1,5-a]pyridine-3-carboxamide;4-[1-(3,4-dimethylphenyl)propan-2-yl]morpholine 2-(6,7-dimethoxy-4-oxoquinazolin-3-yl)-N-[(4-hydroxyphenyl)methylideneamino]acetamide 6-(4,5-dimethylpyrimidin-2-yl)-N-[1-[[3-(oxan-4-yloxy)phenyl]methyl]pyrrolidin-3-yl]pyridazin-3-amine 3-[(2S)-2-[[methyl(2,2,2-trifluoroethoxymethyl)amino]methyl]morpholine-4-carbonyl]benzoic acid (3R,4S)-1-[2-[3-(difluoromethoxy)phenyl]ethyl]-3-(hydroxymethyl)piperidine-4,6-diol 2,3-dibutylanthracene 1,2-difluoro-3-[4-(3-isothiocyanatopentan-3-yl)phenyl]benzene 1,2-diamino-4-(5-bromo-2,3-dichlorophenyl)-6-oxopyridine-3,5-dicarbonitrile 5-(cyclopropanecarbonylamino)-N-[2-methyl-5-[1-(methylsulfamoyl)piperidin-4-yl]phenyl]indazole-1-carboxamide 1-[5-(3,4-difluorophenyl)-3,6-dihydro-2H-pyridine-1-carbonyl]cyclopropane-1-carboxylic acid N'-(3,5-dichloropyridin-4-yl)-2-(1H-pyrrolo[2,3-b]pyridin-6-ylmethyl)propanediamide 2-[2,4-dichloro-N-(1,3-thiazol-5-yl)anilino]ethanol 5-bromo-4,6-dimethylpyrimidine;ethane N-(6,7-dihydrobenzo[c]chromen-3-ylmethyl)-5-ethoxypyrazine-2-carboxamide 2-azido-6-(1,3-benzodioxol-5-yl)-N-benzyl-8-methoxyquinazolin-4-amine 5-[(3,4-dimethylphenyl)iminomethyl]-1-pentan-2-ylidenepyrrole-3-carboxamide 1-[6-(5-butan-2-yloxypent-1-ynyl)pyridin-3-yl]prop-2-en-1-one 5-[4-[(E)-2-cyclopropylethenyl]piperidin-1-yl]-6,7-dimethoxy-2-methylidene-3H-quinazoline (3S)-7-chloro-N-[1-[2,5-difluoro-4-(trifluoromethyl)phenyl]ethyl]spiro[3H-pyrido[2,1-c][1,4]oxazine-4,3'-pyrrolidine]-1'-carboxamide 3-[4-(2,5-dimethylthiophene-3-carbonyl)piperazin-1-yl]propanenitrile N-cyclohexyl-2-(3,5-dichloropyridin-4-yl)-6,7-dihydropyrrolo[1,2-a]imidazol-4-amine 3-[3-oxo-6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]hexyl]cyclobutane-1-carboxylic acid 4-(3,5-dichlorophenyl)-1,3,6,7,8,9-hexahydropyrimido[4,5-b]quinoline-2,4-dione 1-[4-methyl-6-[(3S)-3-methylmorpholin-4-yl]pyrimidin-2-yl]piperidine-4-carboxylic acid 5-amino-3-[4-fluoro-2-(trifluoromethyl)phenyl]-2,3-dihydro-1,2-oxazole-4-carbonitrile 5-[3-[(3,5-dichloropyridine-4-carbonyl)amino]phenyl]pentanoic acid N-(3,3-difluorocyclobutyl)-2,6-dimethoxy-4-[6-(1H-pyrazol-5-ylamino)pyrimidin-4-yl]benzamide 3-[3,5-dimethyl-2-(trifluoromethyl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 1-[2,5-bis(trifluoromethyl)phenyl]-3-[4-[(7R)-4-oxo-3,6,7,8-tetrahydropyrazolo[1,5-a][1,3]diazepin-7-yl]cyclohexyl]urea [4-(methylamino)phenyl]-(3-pyrimidin-2-yloxypiperidin-1-yl)methanone 4-[1-(5,6-dichloropyridin-3-yl)ethylamino]butan-2-ol 2-(1H-pyrazol-5-yl)-N-[2-propan-2-ylidene-7-[4-(trifluoromethoxy)phenyl]sulfonylheptyl]acetamide N-[2-[(1E)-2-[4-[2-(6,7-dihydro-5H-cyclopenta[c]pyridin-3-ylamino)ethoxy]phenyl]buta-1,3-dienyl]iminobut-3-enylidene]hydroxylamine 6-(4-aminophenyl)-2,5-dimethyl-N-[(E)-1-pyridin-2-ylethylideneamino]pyridazin-3-imine (6E)-N-[2-[4-(1H-indazole-3-carbonylamino)piperidin-1-yl]ethyl]-3,7,11-trimethoxy-5,8-dihydrocycloocta[b]thiophene-2-carboxamide 3-(1-ethylsulfanylethenyl)thiophene 6-(2-chlorophenyl)-3-methyl-1-sulfanylidene-5,7-dihydroimidazo[4,5-c]pyridine-2,4-dione ethane;N-[[2-[(3E)-hexa-1,3-dien-3-yl]oxyphenyl]methyl]-2-sulfanylidene-3H-imidazo[4,5-c]pyridine-7-carboxamide (2R)-3-benzamido-4,4-dimethylpentanedioic acid 3-(4-butylphenyl)-6,8-difluoro-7-[4-(trifluoromethoxy)cyclohexa-1,5-dien-1-yl]-1,2-dihydronaphthalene 5-[2-[(2-fluoro-6-methoxyphenyl)sulfonylamino]ethylcarbamoyl]pyridine-3-carboxylic acid 3-(1,2,4-oxadiazol-5-yl)-6-thiophen-2-yl-1H-quinazoline-2,4-dione N-(2,6-difluorophenyl)-2,4,7-trimethyl-1H-indole-3-sulfonamide 3-(1,3-benzodioxol-5-ylmethyl)-1H-pyridazine-2-carboxamide (5Z)-5-[[1-[[4-fluoro-2-(trifluoromethyl)phenyl]methyl]indazol-6-yl]methylidene]-3-methyl-1,3-thiazolidine 2-[(4-butoxyphenyl)iminomethyl]phenol 2-[(E)-1-amino-3-(methylamino)prop-2-enyl]-4-[4-(4-piperidin-1-ylanilino)pyrimidin-5-yl]benzamide 2,4-dichloro-6-[(E)-(quinolin-3-ylhydrazinylidene)methyl]phenol (Z)-1-(3,6-dimethylthieno[2,3-b]pyridin-2-yl)-N'-ethenyl-N-prop-1-en-2-ylbut-1-ene-1,4-diamine 4-[[(2S)-1,3-dihydroxypropan-2-yl]amino]-N'-hydroxypyridine-2-carboximidamide N-(2,4-dimethylphenyl)-3-[(1E)-2-ethenylbuta-1,3-dienyl]iminopentanamide (Z)-3-[4-[(2,5-dichlorophenyl)methoxy]-3-ethoxyphenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile 2-(1H-benzimidazol-4-yl)imidazo[1,5-a]pyridine 7-(4-chlorophenyl)-3-methylsulfanyl-1,5-dihydroimidazo[1,2-b]pyrazol-6-one N-[1-(4-chlorophenyl)ethenyl]pyridine-3-carboxamide 6-chloro-N-[[2-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]pyrimidine-4-carboxamide 6-(2,3,3a,4,5,7a-hexahydroindole-1-carbonyl)-2,4,5,7,8,9,10-octamethylphenanthren-3-ol (E)-2-[3-tert-butylsulfanyl-5-(trifluoromethyl)pyridine-2-carbonyl]but-2-enoic acid 1-[(2E)-2,7-dimethylocta-2,6-dienoxy]-4-ethoxybenzene N-[(2R,3S)-1-(cyclopropylmethoxy)-5-oxo-2-phenylpyrrolidin-3-yl]benzamide 4-[(E)-3,3-dimethylpent-1-enyl]benzaldehyde 2-(6-bromohexyl)benzoic acid (2R)-1-[4-methoxy-3,5-bis(phenylmethoxy)benzoyl]pyrrolidine-2-carboxylic acid 4-[(3S)-6,7-dichloro-1-(4-methoxyphenyl)sulfonyl-2-oxo-4,5-dihydroindol-3-yl]butanoic acid 5-(2,4-difluorophenyl)-3-[2-[4-(6-methylcyclohexa-1,3-dien-1-yl)piperazin-1-yl]ethyliminomethyl]-1H-indol-2-ol 6-(2,2-diphenylhydrazinyl)-N'-ethenylhexanimidamide 4-[3-(6-hydroxyquinolin-2-yl)-1H-pyrazole-5-carbonyl]piperazine-2-carboxylic acid [4-(methoxymethyl)oxan-4-yl]-spiro[1,3-dihydroisoquinoline-4,1'-cyclopropane]-2-ylmethanone 2-benzyl-2-(4-bromophenyl)pyrrolidine 5-(2,4-dimethylphenyl)-N-propanoyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 2-(4,6-dimethylpyrimidin-5-yl)oxy-3-[(1E)-3-ethoxybuta-1,3-dienyl]-N-[4-fluoro-3-[(2Z)-penta-2,4-dien-2-yl]phenyl]-6-[2-(2H-tetrazol-5-yl)phenyl]pyridine-4-carboxamide (2-cyclobutylpyridin-4-yl)-[5-methyl-7-(1H-pyrazol-4-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone 3-[5-ethyl-6-[3-(7-fluoro-1H-indol-4-yl)phenyl]pyridin-2-yl]propanenitrile 1-[(1Z)-buta-1,3-dienyl]-4-methoxy-2-methylbenzene;(E)-3-[5-ethenyl-6-methylidene-9-[3-(trifluoromethyl)phenyl]nonan-5-yl]sulfanylpent-3-enal 2-bromo-6,7-dichloroquinoline 2-chloro-N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]pyrimidine-5-carboxamide 5-[4-(cyclopropylmethoxy)piperidine-1-carbonyl]pyridine-2-carboxamide 4-[(3S)-1-[2,5-difluoro-4-(2,4,6-trifluorophenyl)phenyl]piperidin-3-yl]oxy-N-methylsulfonylbenzamide N-(4,5-dichlorothiophen-2-yl)sulfonylpyridine-3-carboxamide 6-[3-methyl-2-[[(E)-4-(methylideneamino)but-1-enoxy]iminomethyl]phenyl]-N-(2,2,2-trifluoroethylsulfanyl)quinazolin-8-amine N-[(Z)-1H-indol-3-ylmethylideneamino]-2-[[4-phenyl-5-(piperidine-1-carbonyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide 1-[6-(3-aminopropylsulfanylamino)hexyl]-4,5-dihydrothieno[2,3-c]quinolin-9-one [4-(4,5-dihydrobenzo[e]benzimidazol-2-yl)phenyl]-[5-hydroxy-3-(4-methoxycyclohexa-1,3-dien-1-yl)-5-methyl-4H-pyrazol-1-yl]methanone 5-bromo-3-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]pyridine-2-carboxylic acid 1-[4-[6-[[(3R)-5-fluoropiperidin-3-yl]amino]-2H-pyrazolo[1,5-a]pyridin-3-yl]phenyl]ethanone 1-(cyclopropylmethylamino)-3-[1-(2,4-difluorophenyl)ethoxy]propan-2-ol 1-(6,7-dihydronaphthalene-2-carbonyl)-N-ethylpiperidine-4-sulfonamide 4-[1,3-benzodioxol-5-ylmethyl(ethoxy)amino]piperidine-1-carboxylic acid 4-chloro-N-[(5S)-2-oxo-1,3-oxazolidin-5-yl]naphthalene-1-carboxamide 4-fluoro-3-N,5-N,2,6-tetramethylbenzene-1,3,5-triamine (2S)-4-cyclopropyl-1,4-dimethyl-3-[3-(5-methylpyridin-2-yl)phenyl]pentan-2-ol 1-methyl-3-[(2-nitrophenyl)methylidene]quinoxaline-2,4-dione 1-[(3S)-6-ethylsulfonyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]cyclobutane-1-sulfonamide 3-[(2R)-2-[4-[3-[6-methoxycarbonyl-5-methyl-1-(oxan-4-yl)benzimidazol-2-yl]phenyl]pyrazol-1-yl]propyl]benzoic acid 5-(3-fluorophenyl)sulfanyl-2,6-dimethyl-N-(1H-pyrrolo[2,3-b]pyridin-4-ylsulfonyl)pyrimidin-4-amine 4-amino-5,7,8-trihydroxynaphthalene-1-sulfonic acid N-[(Z)-1,3-diaminobut-2-enylidene]-6-methoxy-4-[[7-(methylcarbamoylamino)quinoline-2-carbonyl]amino]pyridine-2-carboxamide 1-[(3R)-3,4-bis[2-(dimethylamino)ethoxy]pyrrolidin-1-yl]-2-[4-fluoro-7-[8-methoxy-5-(trideuteriomethoxy)quinolin-7-yl]-9H-fluoren-2-yl]propan-1-one 2-tert-butyl-6,8-dichloropyrimido[5,4-d]pyrimidine 2-[(5R)-1,3-dimethyl-7-oxo-4,5,6,8-tetrahydropyrazolo[3,4-b]azepin-5-yl]benzoic acid 4-[3-(1,2-dibromoethyl)phenyl]phenol 1-[(3,4-difluorophenyl)methyl]-3,4,6,7-tetrahydropyrido[2,3-b]pyrazine N-[1-(6,7-dimethoxyquinazolin-4-yl)piperidin-3-yl]-2,5-difluorobenzamide 1-[3-ethenyl-5-(1H-pyrazol-4-yl)phenyl]-3-[3-(trifluoromethoxy)phenyl]urea 2,6-ditert-butyl-4-[5-(trifluoromethoxy)cyclohepta-1,3,6-trien-1-yl]pyridine 2-azido-5,6-dimethylimidazo[1,2-a]pyridine (2S)-1-azido-3,4-dihydro-2H-quinoline-2-carboxylic acid (4-fluorophenyl)methylsulfinylmethanol 2-[4,5-dichloro-3-(2-phenylethynyl)pyrazol-1-yl]acetic acid 3-[2,4-dinitro-N-(1,3-thiazol-5-yl)anilino]butanoic acid N-[2-(cyclopropylamino)ethyl]-4-[(1S,5R)-3-(2-fluoropyridine-3-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]benzamide;dihydrochloride 2-azido-4,6-diphenylbenzene-1,3-diol 4-[[5-chloro-4-[3,6-dimethyl-1-(2H-tetrazol-5-yl)indol-6-ium-2-yl]pyridin-2-yl]amino]cyclohexan-1-ol 4-[5-[2-[methyl(2,3,4,9-tetrahydro-1H-carbazol-2-yl)amino]ethylcarbamoyl]pyridin-2-yl]piperazine-1-carboxylic acid N-[(E)-3,5-dimethylhex-2-enyl]-4-(phenylcarbamoylamino)benzamide 4-ethylsulfanyl-N'-hydrazinylidenebenzenecarboximidamide N-(4-fluorophenyl)-5-methyl-2-pyrimidin-5-ylpyrimidine-4-carboxamide 2-[4-[3-(2,6-dimethylpyridin-4-yl)propoxy]phenyl]-N-ethanimidoyl-1H-imidazo[4,5-b]pyridine-7-carboximidamide N-[4-methyl-3-(5H-pyrido[3,2-b]indol-6-ylidenemethyl)phenyl]morpholine-4-carboxamide 6-(difluoromethoxy)-2,3,4-trihydroxybenzenesulfonamide 1-[3-ethoxy-2,5-difluoro-4-(hydroxymethyl)phenyl]propan-2-ol 2-[(4-methyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N-[(Z)-(3,5,7-trihydroxyquinolin-2-yl)methylideneamino]acetamide N-[(1S,2R)-2-hydroxycyclohexyl]-4-methylpyridine-3-carboxamide 1-benzylsulfanylpiperidine-2,6-dione 1-(3,4-difluorophenyl)-6-[3-(trifluoromethyl)anilino]hexan-2-one 1-(2,5-dichlorophenyl)sulfonyl-4-(4-ethylbenzoyl)piperazine-2-carboxamide N-[2-hydroxy-1-(3-thiophen-2-ylpropanoyl)indol-5-yl]-6-methoxypyridine-3-sulfonamide 1-(3,4-dimethylphenyl)sulfonylpiperazine 4-(azidomethyl)-N-[2-chloro-6-[2-fluoro-3-[6-methoxy-5-[(1E,3Z)-penta-1,3-dienyl]pyridin-2-yl]phenyl]phenyl]sulfanylbenzamide 2,7-dimethyl-10H-phenoxazine (3R)-7-amino-4-(4-bromophenyl)sulfonyl-N,2-dimethyl-5,6,8,9-tetrahydrooxepino[4,5-d]pyrimidine-3-carboxamide N-[5-[4-fluoro-3-(4-thiophen-2-yl-1H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]cyclohexanecarboxamide 2-[(Z)-2-[2-[3,5-dimethyl-4-[(E)-prop-1-enyl]phenyl]ethenyl]-4-methylidenehex-2-enoxy]ethanamine 4-[5,6-diamino-2-(deuteriomethyl)pyrimidin-3-ium-4-yl]oxypiperidine-1-carboxylic acid 1-[(5-tert-butyl-2-methoxyphenyl)methyl]pyrazole 7-bromo-5-methyl-1H-pyrazolo[4,3-c]quinoline N-[2-(diethylamino)ethyl]-1'-(2,5-dimethylbenzoyl)spiro[4,7-dihydropyrano[3,4-c]pyrazole-6,3'-pyrrolidine]-2-carboxamide (1S,3R,4R)-N-[2-[methyl-[[4-(trifluoromethoxy)phenyl]methyl]amino]ethyl]-3-propan-2-ylbicyclo[2.1.0]pentane-1-carboxamide 1-[4-(trifluoromethoxy)phenyl]heptan-2-one [2-(2,3-dihydro-1H-inden-2-yl)-6-methoxy-1-benzofuran-4-yl]methanamine 4-[(4-fluorophenyl)methoxy]-N,2,5-trihydroxybenzamide 2-methylpropane;1-phenyl-3-[1-(pyridin-4-ylamino)ethenyl]pyrazolo[3,4-d]pyrimidin-4-amine 2-(5-bromopentoxy)-6-methoxynaphthalene N-[[5-chloro-2-methoxy-4-(trifluoromethyl)phenyl]methylideneamino]-1,3-benzothiazol-2-amine N-[(1E,3Z)-2-methylsulfanylpenta-1,3-dienyl]-4-phenoxybenzamide 4-benzyl-1,2-dimethylpiperazine;ethane N-(5-bromonaphthalen-2-yl)sulfonylcyclopropanecarboxamide 3-[1-(2-amino-6,7-dihydropurin-9-yl)-4-methoxybutyl]oxetan-2-one;ethane 3-(3,4-dichlorophenyl)sulfanyl-N'-hydroxypyridine-2-carboximidamide 1-[2,2-difluoro-4-(methanesulfonamido)butyl]-N-[[5-[6-(trifluoromethyl)pyridin-3-yl]pyridin-2-yl]methoxy]pyrazole-4-carboxamide N-[2-(methoxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-yl]oxane-4-carboxamide 2-[4,5-diphenyl-3-(1-pyridin-4-ylethylidene)pyrazol-2-yl]-2-iminoacetaldehyde N-[2-amino-4-(3,5-dimethylanilino)pyrimidin-1-ium-6-yl]imino-N',2-difluoroethanimidamide 3-chloro-5-[(1E)-3-fluoro-2-methylbuta-1,3-dienyl]pyrazolo[1,5-a]pyridine N-(4-tert-butylphenyl)-6,7-dihydro-2H-[1,3]thiazolo[5,4-e]benzimidazole-5-carboxamide;hydrobromide 1-[(2S,4R)-4-phenylmethoxypyrrolidine-2-carbonyl]pyrrolidine-3-carbonitrile N-[(2S)-1-[4-(3,4-dimethylphenyl)-5-oxotetrazol-1-yl]propan-2-yl]-4-fluorobenzenesulfonamide N'-methyl-N,2,4-triphenylbenzenecarboximidamide 4-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8,11-pentaene 2-chloro-6-(1,3-dioxolan-4-ylmethoxy)benzaldehyde 6-bromo-2,3-dimethyl-1-[(4-pyridin-3-ylphenyl)methyl]imidazo[4,5-b]pyridin-2-ium 3-[4-(dimethylamino)cyclohexyl]oxypyridine-2,6-diamine (2S)-5-amino-1-[(2R)-4,7-difluoro-3,3,5-trimethyl-6-phenylmethoxy-2H-indole-1-carbonyl]pyrrolidine-2-carboxylic acid;hydrochloride N-[5-(2,4-difluorophenyl)sulfonyl-6,6-dimethylhept-1-en-3-yl]piperidine-1-carboxamide (Z)-1-[3-(2-methoxypyridin-4-yl)-6,8,9,10-tetrahydrocyclohepta[b]indol-5-yl]prop-1-en-1-amine 2-(2,6-dichlorophenyl)-N-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]acetamide 2-[(5S)-6,9-dimethyl-5H-[1]benzoxepino[5,4-b]pyridin-3-yl]ethanol (5R)-6-amino-3-[4-[2-hydroxy-3,5-dimethyl-N-(2,2,2-trifluoroacetyl)anilino]cyclohexa-1,5-dien-1-yl]-7-methoxy-1-phenyl-4H-pyrimido[4,5-d]pyrimidin-2-one 4-[(3,5-dimethylphenyl)iminomethyl]phenol;dichlorotitanium 2-[2-(3,5-dichloropyridin-4-yl)phenyl]-N-methoxyacetamide 6-[5-(3,4-dihydroquinolin-7-yl)-1H-pyrazol-3-yl]pyridine-2-carbonitrile;ethane 3-(1,2-diphenylethyl)-4H-quinazoline 5-chloro-6-(4,6-diazaspiro[2.5]octan-7-yl)pyrimidine-4-carboxamide 1-[2-bromo-5-methoxy-4-(trifluoromethyl)phenyl]ethanone 2-N,3-N-bis(prop-2-ynyl)benzene-1,2,3-tricarboxamide [4-(8-methoxy-7H-imidazo[1,2-a]azepin-2-yl)phenyl]-piperidin-4-ylmethanone 6-methoxyspiro[1,2-dihydro-4H-quinoline-3,4'-piperidine] 2-(5-bromo-1H-pyrazole-3-carbonyl)-8a-ethyl-N-pyridin-4-yl-3,4,6,7,8-pentahydro-1H-pyrrolo[1,2-a]pyrazine-9-carboxamide 3-methoxy-1,2,5-tris(trifluoromethyl)benzene ethane;1-(4-methylphenoxy)propan-2-one 4-bromo-3,5-dichloropyridine-2-carboxylic acid 4-[[1-(2,6-dioxopiperidin-3-yl)-3-methylideneisoindol-5-yl]oxymethyl]piperidine-1-carboxylic acid N-[(3S)-1-ethylpyrrolidin-3-yl]-4,5-dimethylthiophene-2-carboxamide 3-[7-(3,5-dimethyl-1H-pyrazol-4-yl)-5-fluoro-3,4-dihydro-2H-quinoline-1-carbonyl]-N,N,6-trimethylpyridine-2-carboxamide N-[2-(2,3,4,5-tetrafluorobenzenecarboximidoyl)phenyl]cyclohexanecarboxamide 1-(cyclopropylmethoxy)-4-propan-2-yl-2-[4-(trifluoromethyl)phenyl]benzene 4-(1H-indol-3-yl)-2,5,6-trimethoxycyclohepta-1,3,6-trien-1-ol 5-methyl-1-(oxan-2-yl)indazole 1-[[(2S)-1,4-dioxan-2-yl]methyl]-3-(5-methoxypyrazin-2-yl)urea 1-(3,5-dimethylbenzene-6-id-1-yl)-6-ethoxyisoquinoline;iridium;2-methanidylpropane-2,3-diol 6-[(4-chlorophenyl)methyl]-1H-pyrido[2,3-d]pyrimidine-2,4-dione;ethane 2,4-dichloro-3-[(6S)-6-[5-[3-[3-(3,3-difluoroazetidin-1-yl)propoxy]phenyl]pyridin-3-yl]-4,7-dioxo-6,8-dihydropyrimido[5,4-c]pyridazin-3-yl]benzaldehyde N-(2-azidooxyethyl)quinoline-3-carboxamide 4-[(3R)-1-(2,2,2-trifluoroethyl)piperidine-3-carbonyl]-1,3-dihydroquinoxalin-2-one 1-(1H-inden-4-yl)naphthalene 3-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-N-phenyldibenzothiophen-8-amine 1-[4-chlorobutyl(2,3-dihydroxypropyl)amino]-4a,9a-dihydroanthracene-9,10-dione 5-chloro-3-[4-(cyclohexylamino)-1H-pyrrolo[2,3-b]pyridin-2-yl]-1H-pyridazin-6-one 2-[3,5-di(propan-2-yl)phenyl]ethyl-trimethylazanium 3-[5,7-difluoro-6-(2-fluorophenyl)naphthalen-1-yl]cyclopentan-1-amine 1-[3-(2,5-dichlorophenyl)-4H-azepin-6-yl]ethanone N'-[(3S,5R)-7-fluoro-5-pyridin-2-yl-3,4-dihydro-2H-chromen-3-yl]oxamide 2-[4-(dimethylamino)phenyl]-N'-[(E)-[5-[(Z)-ethylideneamino]pyridin-2-yl]methylideneamino]benzenecarboximidamide;propane 4-(3-methylcyclobutyl)oxy-2-[(4-methylidene-2,3-dihydrophthalazin-1-ylidene)amino]benzaldehyde (2S)-2-[[4-(N-acetylanilino)phenyl]sulfonylamino]-3-methoxypropanoic acid 3-methyl-1-[4-(2,3,5,6-tetrafluoropyridin-4-yl)phenyl]butan-2-one (2E,3Z)-4-[2-aminoethyl(methyl)amino]-N-[[1-[4-[(4-aminocyclohexyl)amino]quinazolin-2-yl]benzimidazol-5-yl]methyl]-2,3-di(ethylidene)hepta-5,7-dienamide 1-(6-azido-2,3-difluorophenyl)propan-2-one N-[(2S)-1-[4-[2-chloro-6-fluoro-4-[[(3R)-piperidin-3-yl]amino]phenoxy]-7-methoxyquinazolin-6-yl]pyrrolidin-2-yl]prop-2-enamide 2-[4-[2-(cyclopropylamino)ethyl]phenyl]guanidine (4-ethylphenyl)-[5-[2-(4-ethynylphenyl)ethenyl]-1,3,3a,6a-tetrahydrocyclopenta[c]furan-3-yl]methanone 2-(3-azidocyclohexyl)-N,N-dibenzylacetamide 2-chloro-N-[(Z)-(3,5-dibromo-4-hydroxyphenyl)methylideneamino]benzamide 4-fluoro-2-[3-[[3-(4,5,6,7-tetrahydro-1-benzofuran-2-yl)piperidin-1-yl]methyl]pyrrolidin-1-yl]pyridine 1-[3,5-bis(trifluoromethyl)phenyl]-2,2,2-trifluoroethanol 3-[(4-methylpyrazole-1-carbonyl)amino]-2,3-dihydro-1H-indene-5-carboxylic acid N-ethenylsulfonyl-2,4,6-trimethylbenzenesulfonamide ethane;[(3S)-5-fluoro-2,6,9-trimethyl-4,9-dihydroxanthen-3-yl]hydrazine (1R)-5-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carbonylamino)propyl]-N-[(E)-[(Z)-prop-1-enoxy]diazenyl]-1H-indene-1-carboxamide 5-azido-2,3-dichloro-4-propoxyaniline 2-azido-4-(4,5-dihydropyrimidin-2-yl)phenol 3,5-dichloro-4-[6-(methylamino)pyrazin-2-yl]oxyphenol N-butyl-3-[7-cyclopropylidene-8-methoxy-1-(3-morpholin-4-ylpropyl)pyrrolo[2,3-c]quinolin-5-yl]benzamide;2-methoxyethanol ethane;(4-methoxyphenyl)urea 3-(4-ethoxy-2,6-dimethylphenyl)cyclopropane-1,1,2,2-tetracarbonitrile 6-methyl-2-phenylpyrrolo[3,4-f]isoindole-1,3,5,7-tetrone 4-amino-6-(4-ethoxyanilino)-5-nitropyridine-2-carboxamide 2-[7-(4,6-dimethylcyclohexa-1,3-dien-1-yl)-5-[4-(2-hydroxyethoxy)phenyl]-1-benzofuran-4-yl]acetic acid N-[3-(3,4-dichlorophenyl)propyl]-4H-pyrimido[5,4-h]quinazolin-8-amine N-(1,2-benzoxazol-3-yl)-4-cyclohexa-2,4-dien-1-yloxy-5-(trifluoromethyl)pyrimidin-2-amine (5S,7R)-N-[2-(2-hydroxyethoxy)pyridin-3-yl]-1,5,6,7-tetrahydropyrazolo[4,3-g]quinoline-8-carboxamide 2-[4,6-dimethyl-5-[(1Z)-3-methylbuta-1,3-dienyl]pyridin-2-yl]phenol 2-[1-(furan-2-carbonyl)piperidin-4-yl]-N,3,4-trimethoxybenzenesulfonamide 1-[2,3-dihydroxypropyl(hexyl)amino]-4a,9a-dihydroanthracene-9,10-dione N-[3-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)phenyl]thiophene-2-carboxamide;ethane [(2S)-5,7-diethyl-3,4-dihydro-2H-chromen-2-yl]carbamic acid N-ethyl-3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-2-carbonyl)benzenesulfonamide (Z)-2-amino-3-[amino-[(2-methylindazol-6-yl)carbamoyl]amino]-N-[5-chloro-4-[4-(dimethylsulfamoyl)phenyl]pyridin-2-yl]but-2-enamide (3R)-3-[2,5-difluoro-4-[5-methyl-6-[[8-oxo-2-(oxolan-3-ylmethyl)-1,7-naphthyridin-9-yl]amino]pyridin-3-yl]phenyl]pentanoic acid 5-(2,4-dichlorophenyl)-3-[(2R)-2-hydroxy-2-methylhexoxy]furo[3,2-b]pyran-7-one 2,2-difluoro-3-[4-(4-methylcyclohexa-1,5-dien-1-yl)oxybenzoyl]oxypropanoic acid 3-[3,5-bis(trifluoromethyl)phenyl]-1-[2-chloro-6-(cyclopropanecarbonylamino)benzoyl]oxysulfonylimidazolidine-4-carboxylic acid 7-chloro-2-[3-(1H-imidazol-5-yl)phenyl]imidazo[1,2-a]pyridine 2-azido-1H-cyclopenta[b]chromene 2-chloro-N-[(4-nitrophenyl)methyl]-N-phenacylacetamide 3-[[2-[ethyl(oxan-4-yl)amino]-6-methoxypyrimidine-4-carbonyl]-propan-2-ylamino]cyclobutane-1-carboxylic acid N-[2-(3,5-dichloropyridin-4-yl)ethoxy]-1-[6-[[(2R,5S)-2,5-dimethylpiperazin-1-yl]methyl]pyrimidin-4-yl]pyrazole-3-carboxamide 4-(2,5-dimethylphenyl)sulfanylpyrimidine;ethane 5-cyclohexyl-3-[(4-methylphenyl)sulfonylamino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-indole-2-carboxamide 2-(1,3-benzodioxol-5-yl)-6-[[4-(methoxymethyl)phenyl]iminomethyl]-3-(phenylsulfanylamino)phenol 7-bromo-2,5-dihydroimidazo[1,2-a]pyrimidine-3-carboxylic acid 6-(aminomethyl)-8-azido-4H-1,4-benzoxazin-3-one N-[5-[4-chloro-6-(methoxymethyl)pyrimidine-5-carbonyl]pyridin-2-yl]acetamide (4-azido-2-methoxyphenyl)-[4-chloro-2-fluoro-5-(trifluoromethyl)phenyl]methanone 1,3-dimethylpyrrole;2-methoxy-N'-[1-[4-(methylideneamino)phenyl]ethenyl]ethanimidamide 4-[(6-chloropyridin-3-yl)methylamino]-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile (2R)-1,5-dihydroxy-4-(2-oxochromene-3-carbonyl)oxy-6-propan-2-yliminohexane-2-sulfonic acid 4-[5-(4,5-dihydro-1H-imidazol-2-yl)pyridin-3-yl]sulfonylaniline 4-[(3R)-3-[1-[2,4-bis(trifluoromethyl)phenyl]ethoxy]-5-oxopyrrolidine-1-carbonyl]benzenesulfonamide 5-azidooxycarbonylpyridine-2-carboxylic acid N-[2,2-bis(4-chlorophenyl)ethyl]cyclohexanamine 1-[4-(5,6,7,8-tetrahydro-1,7-naphthyridin-3-ylmethoxy)phenyl]ethanone;hydrochloride (1R,3S)-N,4-dimethyl-2-(phenylmethoxyiminomethyl)cyclohexan-1-amine 4-hydroxy-3,5-bis(2-methoxyethyl)-N,1-diphenylpyrrole-2-carboxamide 3-[(5R,7S)-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carbonyl]benzoic acid 4-chloro-6,7-dimethoxy-8-[2-(methylamino)ethoxy]chromene-2-thione 1-[6-(3,4,5-trimethoxyphenyl)quinazolin-2-yl]piperidine-4-carbonitrile 4-[6,7-bis(ethenyl)naphthalen-2-yl]-N-methylbutan-1-amine 4-[[3,5-bis(trifluoromethyl)phenyl]sulfanylamino]-3-chlorobenzoic acid N-(2,6-dimethylphenyl)-N-propan-2-ylacetamide;ethane 2-[4-(2,5-dimethylcyclohexen-1-yl)phenyl]propanoate N-azido-3-[2-(4-chlorophenyl)ethenyl]pyridin-4-amine N-methyl-2-(6-propan-2-ylpyridin-3-yl)imidazo[1,2-a]pyridine-5-carboxamide (3S)-6,8-dibromo-2',2'-dimethylspiro[3H-indene-1,3'-azetidine] 4-(5,6-dimethoxypyridin-3-yl)iminoimidazolidin-2-one 2-[(4,5-dimethyl-1,3-oxazol-2-yl)methoxy]-N-[(Z)-[(6Z)-6-hydroxyiminocyclohexa-2,4-dien-1-ylidene]amino]acetamide (4S)-1,3-dimethyl-4-[2-(2,2,2-trifluoroethoxymethyl)pyridin-4-yl]imidazolidin-2-one 2-azido-3-(5,7-dimethoxy-1H-indol-4-yl)chromen-4-one 3-[2,4-dimethyl-1-(5-oxo-6H-benzo[b][1]benzazepine-11-carbonyl)indol-3-yl]-N,N-dimethylpropanamide 1,4-dimethyl-2-[2-(2-phenoxyethoxy)ethyl]benzene (2R,3S)-6-amino-N-[2-(4-fluorophenyl)ethyl]-2,3-dimethyl-2-(piperidine-1-carbonyl)heptanamide;hydrochloride (2Z,4E)-3-[5-(2-methylphenyl)pyridin-1-ium-2-yl]-N-(4-pyrrolidin-1-ylphenyl)hepta-2,4-dienamide (1R,2S)-N-[3-[5-(2,6-difluorophenyl)-3H-isoindol-1-yl]propyl]-2-pyridin-4-ylcyclohexan-1-amine 2-(benzylideneamino)ethenamine;1-methyl-4-propylcyclohexane 1-cyclobutyl-4-(3,5-diphenylcyclohexa-2,4-dien-1-yl)benzene (E)-3-(5,6-dimethylpyridin-2-yl)oxy-4-(prop-1-en-2-ylamino)but-3-en-2-one 5-bromo-N',6-dimethylpyrimidine-4-carbohydrazide (Z)-1-[2,4-bis(trifluoromethyl)phenyl]-N'-methoxyprop-1-ene-1,3-diamine;hydrochloride 4-(2-methoxyanilino)oxypyridine-3-carboxylic acid 3-chloro-N-(6-ethynylquinolin-5-yl)-2,4-difluorobenzamide N-(2,6-dimethylpyridin-3-yl)-2-[4-[5-fluoro-6-(2-morpholin-4-ylethoxy)quinazolin-4-yl]oxyphenyl]acetamide 5-chloro-N-(3,4-dimethylphenyl)benzenesulfonamide (1S)-2-[[8-amino-3-azido-7-methyl-6-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-5-yl]methoxy]cyclohexan-1-ol 2-[3-(5,6-dimethoxypyridin-3-yl)prop-2-ynyl]-5-[4-(trifluoromethyl)phenyl]thiophene-3-carboxamide (5E)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[[6-hydroxy-1,3-dimethyl-2-oxo-8-(trifluoromethylsulfanyl)quinolin-7-yl]methylidene]-1,3-thiazolidin-4-one 2-[(5-chloropyridin-2-yl)-ethenylsulfonylamino]decanoic acid 4-[2-[7-(3,6-dimethylpyridazin-1-ium-4-yl)quinazolin-5-yl]oxyethyl]morpholine 6-[2-(aminomethyl)-3H-benzimidazol-5-yl]-N-ethyl-N-ethylhexan-1-amine 4-chloro-7-methylspiro[1,2-dihydropyrido[2,3-d]pyrimidine-5,3'-oxolane] 2-methylbuta-1,3-diene;4-[5-[(Z)-prop-1-enyl]pyridin-2-yl]oxybenzoic acid 5-(2-methoxyethyl)-1'-[(6-methoxypyridin-3-yl)methyl]spiro[6H-pyrazolo[4,3-d]pyrimidine-7,4'-piperidine];2,2,2-trifluoroacetic acid 1-[(4S)-4-(3-chlorophenyl)-5-(2-methylpropanoyl)-3,4-dihydropyrazol-2-yl]ethanone 5-(6-methoxypyridine-3-carbonyl)-2-phenylpyrazolidin-1-ium-3-one 7-[(1S)-1-[(6R,8aS)-2-methoxycarbonyl-1,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-6-yl]ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxylic acid 2-(difluoromethyl)-N-[6-(5-fluoropyridin-3-yl)cinnolin-3-yl]-1,3-thiazole-4-carboxamide N-methyl-3-[(E)-2-phenylethenoxy]benzamide N-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide (4S)-4,6,9-trimethyl-2-propan-2-ylidene-1,5,7,8-tetrahydrocyclohepta[b]pyrrole 3-[2-(2,6-difluorophenyl)acetyl]azetidine-1-carboxylic acid 4-chloro-N-[2,3-difluoro-4-[[(2R)-1-hydroxypropan-2-yl]amino]phenyl]benzenesulfonamide 2-(1,3-benzodioxol-5-yl)-N-[(4-fluorophenyl)methoxy]ethanimine 2-benzylsulfanyl-8-[(2R)-2-(diethylaminomethyl)pyrrolidine-1-carbonyl]pyrido[3,4-d]pyrimidin-5-one 4-[3-(cyclopentylmethylamino)propyl]benzenethiol 2-[3,5-bis(trifluoromethyl)phenyl]pentanamide ethane;4-[(4E)-4-ethenylhepta-1,4,6-trien-2-yl]oxyaniline 3-bromo-N-[2-[ethenyl(propan-2-ylidene)hydrazinylidene]ethyl]benzamide [5-chloro-2-(5-methoxypentan-2-ylamino)phenyl]-[1-[[1-hydroxy-3-[4-(trifluoromethyl)phenyl]propan-2-yl]sulfamoyl]cyclobutanecarboximidoyl]azanium 6-[4-(2,3-difluoro-4-pentylphenyl)cyclohexyl]-1-fluoronaphthalene 2-[(E)-(2,4-dihydroxyphenyl)methylideneamino]cyclopentan-1-one 3-methyl-7-[5-[4-[(2S)-oxane-2-carbonyl]piperazine-1-carbonyl]pyridin-2-yl]-1H-quinoxalin-2-one 7-(1,2-dimethylimidazol-4-yl)sulfonylspiro[3H-chromene-2,4'-piperidine] 2-chloro-6,7-dimethoxy-4,4a,8,9-tetrahydroacridine 5-[(3,4-dimethylphenyl)methoxy]pentane-2,3-dione N-[2-chloro-3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]-7-[[2-methoxy-6-(trifluoromethyl)benzoyl]amino]indole-1-carboxamide 5-methyl-1,2-dihydronaphthalene;1-phenylpropan-1-ol (5S,7R)-2-cyclopropylsulfonyl-11-(furan-2-ylmethyl)-2,6,9-triazabicyclo[9.4.0]pentadecan-10-one;2,2,2-trifluoroacetic acid 2-(4,5-dihydro-1H-imidazol-3-ium-3-ylmethylamino)benzenesulfonic acid 1-(benzenesulfonyl)-2,3,5,6-tetrafluoro-4-methylbenzene N'-(4-fluorophenyl)sulfanyl-N-methylmethanesulfonohydrazide 3,5-dimethyl-1-(2,4,6-trichlorophenyl)pyrazole 2-(3,5-dibromo-4-methylphenyl)-N'-hydroxy-3H-benzimidazole-5-carboximidamide 5-(1H-indazol-4-yl)-2,3-dihydro-1H-indene-4-carbonitrile N-[1-[4-(trifluoromethoxy)phenyl]ethyl]but-2-ynamide 6-[2,4-dimethyl-5-(piperidin-3-ylamino)phenyl]-1H-pyrrolo[3,2-c]pyridine-7-carboxylic acid 1,2-dimethylcyclopropane;N'-[(3S)-pyrrolidin-3-yl]-N-[4-[(1E)-penta-1,4-dienyl]phenyl]ethanimidamide 1-(3,4-dichlorophenyl)-5-[(2S)-2-methylpyrrolidine-1-carbonyl]pyrazole-3-carboxylic acid 3-(6-aminopyridin-2-yl)sulfanylpyrrolidine-1-carboxylic acid 5-chloro-3,4,8,10-tetramethylpyrimido[4,5-b]quinoline-2,6-dione 2-[5-(4-fluorophenyl)sulfanyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]pyrimidine-4-carboxylic acid 2-(benzenesulfonyl)propanoyliminomethylideneazanide (5Z)-N,3-bis(4-bromophenyl)-2-[(1E)-buta-1,3-dienyl]-5-ethylideneimidazole-4-carboxamide N-[3-(2,5-dihydrofuran-2-yl)quinoxalin-6-yl]-1H-imidazole-5-carboxamide 5-(7H-purin-2-yl)-1,3-dihydrobenzimidazol-2-one N-(diaminomethylidene)-4,5-dinitrobenzenecarboximidamide 5-amino-1-(2,4-dihydroxyphenyl)ethylazanone;but-1-yne;1-[2-(dimethylamino)ethoxy]-3-phenylpropane N-[4,5-dimethyl-2-(morpholine-4-carbonyl)phenyl]prop-2-enamide 2-azidosulfanyl-5,6,7,8-tetrahydronaphthalene 5-bromo-3-[6,7-diethyl-4-(4-fluorophenyl)phthalazin-1-yl]pyridin-2-amine 2-[(1,3-dioxoisoindol-4-yl)methyl]-5-[(3R)-3-fluoropyrrolidine-1-carbonyl]oxyisoindole-1,3-dione 1,3-bis(2,4,6-trimethylphenyl)imidazolidin-2-ide;5-ethynyl-3-[2-(2,4,6-trimethoxyphenyl)ethenyl]-6H-chromen-2-one;iridium N-[2-(3,5-dimethylphenyl)ethynyl]cyclobutanecarboxamide 2-(2,4-dihydroxyphenyl)-3H-benzimidazole-5-carboxylic acid N'-(2,5-dimethylphenyl)-2-[3-ethoxypropyl(methyl)amino]-6-morpholin-4-ylpyrimidine-4-carboximidamide N-[(5,7-dihydroxy-2-methylchromen-4-ylidene)amino]benzamide 3-[2,4-difluoro-5-[[4-(2-phenylethyl)piperidin-1-yl]methyl]phenyl]-N'-hydroxybenzenecarboximidamide 4-[3-methylbutyl(propyl)amino]benzenesulfonamide 2-amino-4,4-dimethoxy-6-(4-phenoxyphenyl)-3-azabicyclo[3.1.0]hex-2-ene-1,5-dicarbonitrile (3R)-1-cyclohexyl-N,2,5,5-tetramethyl-6,7-dihydroindol-4-imine 2-[1,3-bis(ethenyl)indol-6-yl]oxybenzonitrile 2-methoxy-4,6-dinitrophenol;hydrate (2S,3R)-1-benzyl-N-[1-hydroxy-5-(4-methoxyphenyl)pentan-2-yl]pyrrolidine-3-carboxamide 2-[(Z)-6-oxo-5H-benzo[b]carbazol-7-yl]acetamide 4-[2,6-dichloro-4-(hydroxymethyl)phenoxy]butanal;ethane 6-azidooxy-2,4-diphenylpyrimidine 3-[(2Z)-2-[(3,5-diethoxyphenyl)methylidene]hydrazinyl]-6-methyl-4H-1,2,4-triazin-5-one 3-(3,5-difluorophenyl)-4-[2-methyl-4-[1-(oxetan-3-yl)piperidin-4-yl]anilino]butanoic acid;methanol 4-(azetidin-1-ylmethyl)-6,8-difluoro-7-[[3-fluoro-2-(2H-tetrazol-5-yl)phenyl]methylamino]-3,4-dihydro-2H-naphthalen-1-one;2-methylbutane N-[4-chloro-2-(6,7-dimethoxyquinolin-4-yl)-5-fluorophenyl]-1-ethylpiperidine-4-carboxamide 1-[2-(cyclobutylmethoxy)phenyl]azepane (1S)-2-azido-N,1-dimethyl-3H-indene-5-sulfonamide 3-[7-(aminomethyl)-1H-indol-2-yl]-4,5-difluorobenzoic acid (1E,3Z)-N'-(4-acetylphenyl)-2-hydroxypenta-1,3-diene-1,6-disulfonamide 4-(4,4,5,5-tetramethyloxaborolan-2-yl)-1H-indole 2-(1,3-benzodioxol-5-yl)-N-[5-methyl-2-(4-oxo-6,7-dihydropyrano[3,2-d]pyrimidin-3-yl)pyrazol-3-yl]acetamide N-[1,1-diphenyl-3-(quinoline-2-carbonylamino)propyl]piperidine-4-carboxamide 3-[4-(2-hydroxyethoxy)phenyl]pentane-1,5-diol 5-bromo-2-[(Z)-1,3-diaminoprop-1-enyl]benzonitrile 2-azido-N-methyl-6-(trifluoromethoxy)benzamide N-cyclohexa-1,3-dien-1-yl-N'-(naphthalene-2-carbothioyl)-N'-propan-2-ylpropanehydrazide 2-[3-oxo-5-(2,4,6-trimethylanilino)-1H-pyrazol-2-yl]benzoic acid 7-bromo-N-(cyclopropylmethoxy)isoquinoline-1-carboxamide N'-cyclopropylsulfanyl-2-[5-(2-methoxyphenyl)pentylamino]pyrimidine-4-carboximidamide 3-[4-(4-methoxyphenyl)sulfonyloxy-2H-indazol-5-yl]propanoic acid 2-[1-(3,5-difluoropyridine-4-carbonyl)piperidin-4-yl]-7-propanoyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one (4R)-5'-ethyl-1'-[(6-methoxypyridin-2-yl)methyl]-5-methylspiro[1H-indole-3,3'-pyrrolidine]-2-one N-[6-(4,5-dihydro-1H-imidazol-2-yl)-3-oxohexan-2-yl]-5,5-bis(trifluoromethyl)-1,3-benzothiazol-2-amine 2-(3-aminopropyl)-N,4-dicyclohexylaniline 4-N-ethyl-6-(4-nitrophenyl)-2-(pyridin-3-ylamino)pyrimidine-4,5-diamine 2-(azidomethyl)-3,5,7,8-tetrahydropyrano[4,3-d]pyrimidin-4-one 1-[(Z)-(2,4-dihydroxyphenyl)methylideneamino]-3-morpholin-4-ylthiourea 2-[3-[(7-hydroxyquinolin-4-yl)amino]propoxy]-6-methanimidoylbenzoic acid 5-bromo-N,4-dimethyl-2-[4-(trifluoromethoxy)phenyl]-1H-pyrimidine-6-thione 5-fluoro-3,4-dihydroxybenzo[g]chromen-2-one 1-[1-(3,4-dichlorobenzoyl)piperidin-4-yl]-1-methyl-3-[5-(trifluoromethoxy)-2H-triazol-4-yl]urea 7-(3,5-dichlorophenyl)-N-[2-(oxan-4-yloxy)ethyl]thieno[3,2-b]pyridine-5-carboxamide N-[(2,4-dichlorophenyl)methyl]spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 5-chloro-3,4-difluoro-N-(2-methoxyethyl)benzamide 6-(4-methoxyphenyl)sulfinyl-1,2,3,7-tetrahydrocyclopenta[b]pyrazine (2E,4Z)-N-[3-[6-[3-(azetidine-1-carbonylamino)propyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]hepta-2,4-dienamide 5-[4-[2-(azetidine-1-carbonyl)phenyl]anilino]imidazolidine-2,4-dione 1-[(3E)-hexa-1,3,5-trien-3-yl]oxycarbonyl-4-oxo-3H-quinazoline-2-carboxylic acid N-(2,6-dimethylphenyl)-2-[[5-oxo-8-[3-(trifluoromethoxy)phenyl]-4H-pyrazolo[1,5-a]quinazolin-3-ylidene]amino]acetamide N-[3-(4-chloro-1H-indole-2-carbonyl)phenyl]methanesulfonamide (2E)-2,3,4a,5,9b-hexahydro-1H-pyrano[2,3-c]quinoline-6-carboxamide 1-[4-[(2S)-2,3-dihydroxypropyl]piperazin-1-yl]-2-[(6R)-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-6-yl]ethanone;hydrochloride 1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]sulfanyl-3-methoxybenzene;2-methylpropane (E)-3-(1-methylimidazol-4-yl)-N-[[6-oxo-9-propan-2-yloxy-5-(2,2,2-trifluoroethylamino)pyrido[1,2-a]pyrimidin-8-yl]methyl]prop-2-enamide 1-chloro-2,3,5-trifluoro-4-(2-fluoro-3-methylphenyl)benzene;3-[(E)-prop-1-enyl]pyridine 1-(5,6-diaminopyrimidin-4-yl)piperidine-2,5-dione N-[1-cyclohexyl-2,2-dimethoxy-2-(3-morpholin-4-ylphenyl)ethyl]aniline 2-(1-azido-2,2,2-trifluoroethyl)-5-(4-phenoxyphenyl)-1H-imidazole 2-(2,6-difluorophenyl)imino-5-methyl-1,3-thiazolidin-4-one 4-chloro-6-N,1-diphenylcyclohexa-2,4-diene-1,2,3-triamine 2-tert-butyl-6-[(3,5-ditert-butyl-4-hydroxyphenyl)methyl]-4-nitrophenol 6-methoxy-5,7-dipropylquinoline;hydrochloride N-(3,4-dihydroxyphenyl)benzenecarboximidate ethane;N-(4-hydroxynaphthalen-1-yl)-2,5-dimethylpyrazole-3-carboxamide 1,3-dichlorobenzene;ethane 5-chloro-2-[2,4-dihydroxy-3-(3-methylbutanoyl)anilino]benzonitrile 6-methyl-3-[4-(1-methylidene-2H-naphthalen-5-ylium-2-yl)phenyl]-2,3-dihydroisoindol-1-one 3-(methylamino)-1-[3-[2-(4-methylphenyl)propan-2-yl]cyclohexa-1,5-dien-1-yl]propan-1-ol 2-[4,6-bis(dimethylamino)pyridin-3-yl]ethane-1,1-diol 2-[2,5-bis(methylamino)anilino]phenol N-azido-1-(4,6-difluoroindazol-2-yl)methanimine 2-(3,4-dihydroxyphenyl)-7-methylcyclohepta-1,6-diene-1-carboxylic acid (2S)-N,3-dimethylbutanamide;4-[[(1S)-1-[5-fluoro-6-(2-hydroxyethoxy)pyridin-3-yl]propyl]amino]-2-(trifluoromethyl)benzonitrile 1-bromo-3-iodo-5,6-dimethylindazole 2-[1,3-benzothiazol-2-yl(2-sulfanylidenepropyl)amino]acetamide 5-(1,3-benzothiazol-2-yldiazenyl)benzene-1,2,4-triol 4-[4,5-bis(ethenyl)thiophen-2-yl]butanoic acid 2-[(2,5-dichlorophenyl)methylamino]-N'-[3-hydroxybutyl(propan-2-yl)amino]ethanimidamide;hydrobromide 1-(3-ethyl-2,4,6,7-tetramethylheptan-3-yl)-3-prop-1-ynylbenzene 3-[(3,4-dichlorophenyl)methylsulfanyl]piperidine;hydrochloride 2-fluoro-4-(9-iodononyl)benzoic acid 2-[3-(1,4,5,6-tetrahydropyrimidin-2-yl)phenyl]pyridine ethane;4-methyl-6-[1-[1-(oxetan-3-yl)piperidin-4-ylidene]ethylsulfonyl]-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine 1-(2,5-dimethylphenyl)sulfanyl-3-[2-oxo-2-[4-(pyrimidin-2-ylamino)piperidin-1-yl]ethyl]urea 2-N,3-N-bis(2-methoxyphenyl)pyrazine-2,3-diimine (E)-2,3-bis[3,5-dimethyl-4-(2-phenoxyethoxy)phenyl]prop-2-enenitrile 3-(2-chloro-6-methylphenyl)-1,7-naphthyridin-8-ol 2-(1,5-dimethylimidazol-4-yl)sulfanyl-N'-hydroxypyridine-3-carboximidamide 4-azido-2-(5-phenyltetrazol-1-yl)pyrimidine 4-fluoro-N-[3-(2-oxopyrrolidin-1-yl)phenyl]benzamide 4-N-ethyl-2-(5-methoxybenzotriazol-2-yl)benzene-1,4-diamine N-(4,5-dichloropyridin-2-yl)-2,3-dihydroindole-1-carboxamide N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-2,6-dimethyl-1-[(2-methylphenyl)methyl]benzimidazole-5-carboxamide (5Z)-2-(4-bromophenyl)imino-5-[[1,2,2,4]methyl-3-nitro-6-(trifluoromethoxy)indol-3-yl]methylidene]-1,3-thiazolidin-4-one 6-methoxy-N',7-dimethyl-4-oxo-1H-quinoline-3-carboximidamide 2-(3,4-dimethylphenoxy)-1H-pyridine-2-carboxylic acid 2-bromo-3,6-dichloro-N-diazobenzenesulfonamide 4-[(7S)-6,8-dimethyl-5-[1-[(2R)-2-methyloxiran-2-yl]ethoxy]imidazo[1,2-a]pyridin-7-yl]phenol 3-[(5-methylpyrazin-2-yl)amino]sulfanylbenzonitrile N-(2,4-dinitrophenyl)-N-octylbenzamide 4-hydroxy-2-(5-methylthiophene-3-carbonyl)-1H-pyrimidin-6-one 5-methyl-4-nitro-2-[(3R)-piperidin-3-yl]pyrazole 3-[3-(4,6-dimethylpyrimidin-2-yl)phenyl]-5,7-diethoxy-1H-quinolin-2-one N-[(E)-1H-indol-3-ylmethylideneamino]-4-methylbenzenesulfonamide N-[(1S,2R)-1-hydroxy-3-oxo-5-phenyl-1-pyrrolidin-1-ylpentan-2-yl]acetamide 3-[(5E)-4-[(2,6-difluorophenyl)methyl]-3-oxo-1H-pyrazol-5-yl]-N-ethylpropanamide 2-(5,6,7-trimethylnaphthalen-1-yl)hexanoic acid (1R,3S)-3-[2-methyl-6-[4-[5-(trifluoromethyl)pyridin-3-yl]phenyl]pyridine-3-carbonyl]cyclopentane-1-carboxylic acid (Z)-2-cyano-3-[3,5-dimethyl-4-[(2R,3S)-3-(trifluoromethoxy)butan-2-yl]oxyphenyl]prop-2-enamide (1S,2R)-N-[6-(4-fluoropyrazol-1-yl)pyridin-3-yl]-2-methoxycyclohexane-1-carboxamide 7-(2,6-dichlorophenyl)-12-[4-(methyliminomethyl)anilino]-2,5,7,11,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),3,5,9,11-pentaen-8-one 7-amino-5-(3,4,5-trichlorophenyl)-2,4-dioxa-5-azabicyclo[4.1.0]heptane-3,6-dione (4-aminopiperidin-1-yl)-[2-(3,5-dimethoxyphenyl)imidazo[1,2-a]pyridin-7-yl]methanone [3-chloro-4-(trifluoromethyl)phenyl]-[4,7-dimethoxy-2-(methoxymethyl)-1H-indol-5-yl]methanone [1-[2,6-dimethyl-4-(pyrrolidin-3-ylamino)benzoyl]piperidine-4-carbonyl]azanide 2-[1,4-bis(3,5-dimethylphenyl)cyclohexa-2,4-dien-1-yl]-4,6-dinaphthalen-1-yl-1,3,5-triazine 5-amino-3-(2,4-dichlorophenyl)-1-methylpyrazole-4-carbonitrile N-cyclopropyl-4-[2-fluoro-3-(tetrazol-1-yl)phenyl]-7-methoxyquinoline-6-carboxamide (1R,4S)-6-[5-[[1-[2-methyl-5-(trifluoromethyl)pyrazole-3-carbonyl]piperidin-2-yl]methoxy]pyridin-3-yl]-3,4-dihydro-1H-[1,4]oxazino[4,3-a]benzimidazole-9-carboxylic acid N-[(4,6-dimethylpyrimidin-2-yl)carbamoyl]-3,3,3-trifluoropropanamide 5-[3-(4-cyanophenyl)imidazo[1,2-b]pyridazin-6-yl]pyridine-3-carboxylic acid 5-[(1Z)-buta-1,3-dienyl]-6-ethenyl-9H-fluoren-2-amine;(7E,8Z,9Z)-4-cyclopropylidenenona-8,12-diene 3-fluoro-5-[2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indazol-3-yl]-3H-imidazo[4,5-c]pyridin-7-yl]phenol 7-methoxycarbonyl-2,6-diphenylheptanoate N-[4-(2,6-diphenylpyridine-4-carbonyl)phenyl]acetamide 2-(2,5-dimethylpyrrol-1-yl)-N-[3-[4-(4-morpholin-4-ylcyclohexa-1,3-dien-1-yl)phenyl]phenyl]benzamide 3-[3-(4-chlorophenyl)sulfonyl-2-methylpropoxy]pyridine 5-chloro-N-cyclohexylpyrazine-2-carboxamide 5-(3,4-dimethylphenyl)-7-[[1-(2-ethoxyethyl)triazol-4-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amine 1-(2,5-dichlorophenyl)sulfonyl-6,7-difluoro-N'-[(3R,4S)-4-methoxyoxolan-3-yl]indole-3-carbohydrazide 4-amino-N-(4-carbamoylphenyl)-6-fluoro-1H-indole-2-carboxamide 1-methoxy-3-[(2,4,6-trifluorophenyl)methyl]urea 6-amino-4-[2-(cyclopentanecarbonyl)phenyl]-4-methyl-2-sulfanylidene-1,3-dihydropyrimidine-5-carbonitrile 1-amino-6,8-difluoro-7,9-dihydroanthracene-2-carboxylate 6-(2,4-difluorophenyl)-N'-hydroxy-5-oxo-7H-imidazo[1,2-c]imidazole-3-carboximidamide 2-chloro-N-[4-cyano-3-(trifluoromethyl)phenyl]propanamide 5-[3-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrrole-2-carbonitrile 4-methoxy-5,5-dimethyl-1-[(2S)-3,3,3-trifluoro-2-hydroxypropanoyl]pyrrolidine-2-carboxylic acid;1-(7H-purin-6-ylamino)butane-2,3-diol N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)phenyl]-1-(4-methylcyclohexa-1,5-dien-1-yl)cyclopropane-1-sulfonamide 2-(1,4-diphenylbutyl)benzotriazole 1,2-bis(5-bromopentyl)naphthalene 1-butyl-2,3,4,5-tetrafluorobenzene (2R,3aS,6aR)-N-methylsulfonyl-1-[(4-propan-2-ylphenyl)methyl]-5-pyrimidin-5-ylspiro[2-benzofuran-3,4'-piperidine]-1'-carboxamide 3-[7,8-dimethyl-6-(4-methylpiperidin-1-yl)-2H-chromene-3-carbonyl]benzoic acid N-[(3S,5R)-1-[2-(4-fluorophenyl)acetyl]-5-(5-methoxy-1H-1,2,4-triazol-3-yl)pyrrolidin-3-yl]cyclopropanecarboxamide (3Z,5E)-5-[4-chloro-2-[3-methyl-5-(trifluoromethoxy)phenyl]phenyl]sulfanylhepta-1,3,5-triene-2,6-diamine N-cyclopentyl-1'-(pyridine-2-carbonyl)spiro[6,7-dihydrothieno[3,2-c]pyran-4,4'-piperidine]-2-carboxamide 4-[(4R)-3-(cyclohexen-1-yl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl]benzonitrile 5-(dimethylamino)naphthalene-2,7-disulfonate 2-[3,5-bis(trifluoromethyl)phenyl]-N-methyl-1-[6-(4,4,5,5-tetramethyloxaborolan-2-yl)indazol-1-ylidene]ethanamine 3-[2-(2,4-dimethylphenyl)ethyl]-2H-pyrazolo[4,3-c]pyridine [3-amino-4-(benzenesulfonyl)thiophen-2-yl]methanol 1-(azidomethyl)-5-(3,4-dichlorophenyl)-N-[2-hydroxyethyl]triazole-4-carboxamide 1-[(Z)-[3,4-dimethoxy-2-(methylaminomethyl)phenyl]methylideneamino]-3-cyclopropylurea;fluorobenzene 1-(benzenesulfonyl)-3-diazopyrrolidine 2-[(1E,3Z)-4-bromobuta-1,3-dienyl]-3-methylideneindene N-methyl-5-(4-phenoxyphenyl)-1,2,3,6-tetrahydropyridine-2-carboxamide;hydrochloride 1-[3-[4,6-bis(trichloromethyl)-1,2,3,5-tetrazin-3-ium-3-yl]phenyl]cyclopentan-1-ol N-[1-(2-aminoethyl)pyrazol-4-yl]-3,5-dimethoxy-N'-methylbenzenecarboximidamide 5-[4-(diethylamino)phenyl]sulfanyl-2,3-dimethoxyphenol 6-chloro-5-[3-(2,3-dihydroindole-1-carbonyl)phenyl]pyridine-2-carboxamide N-[(3S)-5,7-dimethyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-4-(pyridine-4-carbonylamino)benzamide N-(1,3-benzothiazol-5-yl)propanamide;ethane 4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-7-(4-methylcyclohexa-2,4-dien-1-ylidene)-3,5-dihydropyridazino[4,5-e][1,4]oxazepine 5-[(6,8-dimethyl-9H-fluoren-1-yl)-propoxycarbonylamino]pentanoic acid 2-[6-[(4,5-difluoropyridin-3-yl)amino]-7H-purin-2-yl]benzonitrile N-[4-[5-amino-1-(5-hydroxycyclohexa-2,4-dien-1-yl)pyrazole-3-carbonyl]phenyl]pyridine-4-carboxamide 3-[(1Z)-2,3-diaminobuta-1,3-dienyl]-N'-[4-(cyclopropanecarbonyl)phenyl]-5-fluorobenzohydrazide 6-(2,3-dihydro-1H-isoindol-5-yl)-N-(3,4,5-trimethoxyphenyl)imidazo[1,2-a]pyrazin-8-amine N-[4-(chloromethyl)phenyl]naphthalene-2-sulfinamide 2-[(5E)-4,7-bis(ethenyl)-3-methylidene-1H-2-benzazepin-2-yl]phenol 2-(4-cyclohexylphenyl)-N'-hydroxy-5-methoxy-3-[4-(trifluoromethoxy)phenoxy]benzenecarboximidamide 3-[3-(azidomethyl)phenyl]pyridine 3-[4-(1,2-dihydropyridine-5-carbonylamino)phenyl]propanoic acid 3-[4-(difluoromethoxy)-6,7-dihydropyrrolo[2,1-c][1,2,4]triazol-5-yl]-N,N-bis(sulfanyl)propanamide 3-(diaminomethylideneamino)-5,6-bis[4-(4-hydroxyphenoxy)phenyl]pyrazine-2-carboxamide 2-amino-N'-[(4S)-2,3-dihydro-1H-inden-4-yl]-5-pyridin-3-ylpyridine-3-carboximidamide 1-[2-azidooxy-3,5-bis(4-methylphenyl)cyclopenta-2,4-dien-1-ylidene]ethanol N-[3,5-bis(trifluoromethyl)phenyl]-N',2,2-tris(4-chlorophenoxy)ethanimidamide 6-[[4,5-dimethyl-2-(1,3-thiazol-2-yl)-1H-indol-7-yl]amino]-N'-hydrazinylpyridine-3-carboximidamide 3-cyclohexyl-4-methoxyaniline;3-cyclopentyl-1,4-dihydroquinazolin-2-one 3-[(2,5-difluorophenyl)methyl]-1-hydroxy-1-[4-[2-[4-(methanesulfonamido)piperidin-1-yl]ethoxy]cyclohexa-1,3-dien-1-yl]urea N-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-4-methoxy-6-methyl-N-octyl-1,3,5-triazin-2-amine 1-[2-(4-fluorophenoxy)ethyl]-5-methylpiperidine 5-(2,4-dichlorophenyl)-3-[2-[2-fluoro-4-[1-methyl-7-(2-morpholin-4-ylethoxy)benzimidazol-5-yl]phenyl]acetyl]-1-propan-2-ylpyridin-2-one [3-[(2,4-dimethoxyphenyl)methylcarbamoyl]oxetan-3-yl]carbamic acid 5-[(2,4-dichloropyrimidin-5-yl)-hexadecylamino]naphthalene-2-sulfonic acid (5Z)-1,3-diethyl-5-[[4-hydroxy-3,6-bis(methoxymethyl)-5-methylpyridin-2-yl]methylidene]-1,3-thiazolidine-2,4-dione 1-(3-methylbutan-2-ylideneamino)-4,5,6,7-tetrahydrobenzotriazole-5-carboxylic acid [2-(9H-fluoren-1-yl)ethylamino]methanesulfonic acid N-[5-(3,4-dimethoxyphenyl)-2-(1-propanoylpiperidin-4-yl)pyrazol-3-yl]-N'-(3-methylbutyl)butanediamide ethane;[(5S)-5-hydroxyoxolan-2-yl]-diphenylmethanolate 4-methyl-3,11,11a-trioxoindeno[1,2-c]quinoline-9-carbonitrile 1-[4-[2-chloro-3-(2,5-dimethylhexoxy)phenyl]piperazin-1-yl]ethanone 2-(3-hydroxyphenyl)-5,6,7,8-tetrahydro-3H-pyrido[3,4-d]pyrimidin-4-one N-methylsulfonyl-1,3-benzoxazole-2-carboxamide ethane;6-[5-(methoxymethyl)-1,2-oxazole-3-carbonyl]-N-propan-2-ylpyridine-3-sulfonamide N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-4-hydroxycyclohexane-1-carboxamide 2-(7,9-dihydrobenzo[a]azulen-10-yl)-1,3-diphenylpropan-2-amine 5-(1H-benzimidazol-2-yl)-4-[[(1R,3S)-3-methoxycyclohexyl]amino]pyridine-2,3-diamine 3-[3,5-dimethoxy-4-(phenylcarbamoyl)phenoxy]-1,2-oxazole-4-carboxylic acid 2-chloro-6-methyl-3-(trifluoromethoxy)benzoate [2,3-difluoro-4-(1H-pyrrolo[3,2-c]pyridine-2-carbonyl)phenyl]-piperazin-1-ylmethanone 4-(4-fluorophenyl)-2,5-dimethylfuran 2-[3-(cyclohexylcarbamoylamino)anilino]-4,7-dioxo-N-pyridin-3-yl-1H-pyrrolo[2,3-d]pyrimidine-6-carboxamide (E)-1-[4-amino-5,6-diethyl-3-(4-fluorophenyl)furo[2,3-b]pyridine-2-carbonyl]-N-methoxypyrrolidine-2-carboxamide 2-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-N-ethyl-3-methoxy-N-propan-2-ylaniline 2-hydroxy-N-[2-oxo-1-phenyl-2-(propylamino)ethyl]benzamide 3-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-[[(2R,3S)-2-phenyloxolan-3-yl]methyl]propanamide 2-[[(3S,4R)-1-benzyl-4-methylpyrrolidine-3-carbonyl]amino]-4-[4-(4-methoxyphenyl)piperazin-1-yl]butanoic acid 1-(5,6,7,8-tetrahydronaphthalen-2-yl)pentan-3-one 2,5-dichloro-N-(1H-indol-4-ylmethylideneamino)aniline 6-[(3R)-1-acetylpiperidin-3-yl]-7-(3,4,5-trimethoxybenzoyl)-2-thia-5,7,11-triazatricyclo[6.3.1.04,12]dodeca-1(11),8(12),9-trien-3-one (2Z)-5,6-diamino-N'-azido-2-[2-(4-benzylpiperazin-1-yl)ethylidene]-3H-1-benzofuran-7-carboximidamide 4-[[(5Z)-2,3-dimethylocta-1,3,5,7-tetraen-5-yl]amino]sulfanylaniline 1-amino-3-[(3,4-dimethoxyphenyl)sulfonylamino]thiourea 4-[2,3,6-tris(trifluoromethyl)phenyl]-1H-pyrimidine-4,6-diamine 1-[3-(4,5-dihydroimidazol-1-yl)phenyl]hexan-2-ol N-ethyl-2-[4-hydroxy-3-(2,4,5-trimethoxyphenyl)chromen-1-ium-2-yl]benzamide 2-[4-[(2,6-difluorophenyl)methoxy]-1-hydroxy-2-oxopyridin-3-yl]-N-prop-2-enoyl-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridine-3-carboxamide 2-[4-(6-chloropyridazin-3-yl)-2,5-dimethoxyphenyl]-1H-pyrrolo[2,3-b]pyridine 2-[(4R)-1-cyclohexyl-3,4-dimethyl-6-oxo-5H-pyrazolo[3,4-d]pyrimidin-4-yl]propanoic acid N-[4-(1,3-benzodioxol-5-yl)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]acetamide N-[1-(3,4-dimethoxyphenyl)ethyl]-6-[[5-(trifluoromethyl)pyridin-2-yl]amino]pyrazine-2-carboxamide 1-(2,5-dimethylpyrazol-3-yl)-2-[6-[(E)-4,4-dimethylpent-1-enyl]spiro[3H-1-benzofuran-2,3'-pyrrolidine]-1'-yl]ethane-1,2-dione 6-[(5-chloro-2-cyclopropylbenzimidazol-1-yl)methyl]quinoline 4-[(1,5-dimethylpyrazol-3-yl)methyl]thieno[2,3-d]pyrimidine 5-[3,5-dichloro-4-[(2R)-4,4-difluoro-2-methylpyrrolidin-1-yl]phenyl]-1H-indole (Z)-1-N',3-N'-diethylprop-2-enedihydrazide;4-[[4-(dimethylamino)phenyl]methylidene]-5-oxoimidazolidine-2-thione 4-azido-5-bromoquinoline (5Z)-5-[(4-bromo-2,3-dichlorophenyl)methylidene]imidazolidine-2,4-dione 5-[4-(2,6-difluorophenyl)phenyl]-3-(oxolan-3-ylmethoxy)pyridine 2-[1-(4-fluorophenyl)sulfonylpiperidin-3-yl]-N,N-dimethylacetamide (5Z)-3,6-dimethylocta-1,5,7-triene;5-ethynyl-2-methoxypyridine 2-(4,5-dimethylthieno[3,2-b]pyrrole-6-carbonyl)-1H-pyrrole-3-carboxylic acid 5-[2,3-bis(ethenyl)phenyl]-1H-pyrrole 3-azidooxy-N',2-dimethylbenzenecarboximidamide 2-methyl-6-[(3R)-3-methylpyrrolidin-1-yl]-N-[4-(2-oxopyridin-1-yl)phenyl]pyrimidine-4-carboxamide [4-(methoxymethyl)-2,5-dihydropyrrolo[3,2-d]pyrimidine-1-carbonyl]-pyridin-3-yl-pyrrolidin-3-ylazanium 5-chloro-3-(2,4-dihydroxy-6-methylphenyl)-N-[(1S)-2-hydroxy-1-naphthalen-2-ylethyl]thiophene-2-carboxamide N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2,8-dioxo-7H-purine-9-carboxamide N-[4-(2,3-difluorocyclohexa-1,5-dien-1-yl)pyrimidin-2-yl]-6-methoxy-7H-quinolin-8-imine 2-[3-(2,5-dioxopyrrolidin-1-yl)phenyl]acetic acid;ethane 1-[(3-chloropyridine-4-carbonyl)amino]cyclohexane-1-carboxylic acid 2-[(1,3-diethoxy-1,3-dioxopropan-2-yl)-(4-hydroxy-6-methyl-1H-inden-5-yl)amino]acetic acid 2-[(3,5-dimethoxyphenyl)methyl]-3-phenylspiro[4,6-dihydropyrrolo[1,2-a]pyrazine-8,3'-pyrrolidine];2,2,2-trifluoroacetic acid 2-(1H-benzimidazol-2-ylmethylamino)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 5-[2-[1-(pyridine-4-carbonyl)piperidin-3-yl]propan-2-yl]-3H-1,3,4-oxadiazol-2-one ethane;(4E)-4-[2-[methyl-[[3-methylidene-1,1-bis(sulfanyl)azetidin-1-ium-1-yl]methyl]amino]-7,8-dihydro-6H-cyclopenta[g]quinazolin-4-ylidene]butan-2-one (3S)-2,3-dimethyl-1,3,4,5-tetrahydropyrido[4,3-b]indole-8-carbonitrile N-[2,3-diamino-4-(3-chloro-2-fluorophenyl)phenyl]acetamide 2-(4-cyclopropylphenyl)-1,1-difluoro-5-nitro-3H-indene 2-[azido-(2,4,6-trimethylphenoxy)sulfanyloxyamino]-3-methylphenol 6-azido-N,N-dimethyl-2-phenylpyridazin-3-amine N-[(E)-3-(2,5-dichlorophenyl)prop-2-enyl]-6-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-8-amine 3-[3-(5-hydroxypyrimidin-2-yl)phenoxy]-2,6-dimethylphenol 1-[(4-hydroxy-3,5-diiodophenyl)methyl]-N-[(4R)-1-propanoylazepan-4-yl]pyrrolidine-2-carboxamide 1-[[6-[4-hydroxy-3,5-di(piperidine-1-carbonyl)phenyl]pyridin-2-yl]amino]ethanesulfinic acid 4-(1,2-oxazol-3-ylmethylamino)thieno[3,2-c]quinoline-7-carboxylic acid 3-(1,2,4-oxadiazol-5-yl)-1-[3-(2H-tetrazol-5-ylmethyl)piperidin-1-yl]butan-1-one 4-[2-azido-1-(4-methylphenyl)ethyl]pyridine 1-azido-3-[(4-bromophenyl)methyl]-2,6-dichlorobenzene 3-(2-chloro-6-methyl-4-phenylphenyl)propanoic acid N-[2-bromo-4,6-dichloro-3-(2-chloroanilino)phenyl]acetamide 2-[3-(2,4-dimethylimidazol-1-yl)propyl]isoindole-1,3-dione;hydrochloride 1-[3-(2,6-dichlorophenyl)propyl]cycloheptane N-[4-[2,3-dichloro-5-(1H-pyrazol-4-yl)phenyl]butan-2-ylidene]hydroxylamine 7-(5-methoxypyridin-3-yl)-4,5-dihydropyrazolo[1,5-a]pyrimidine 1-(5,6-dihydronaphthalen-2-yl)-N-ethylnaphthalene-2-carboxamide 4-[3-(2,3-dihydro-1H-isoindole-5-carbonyl)phenyl]-7-ethoxypyrido[3,4-d]pyridazin-1-one N-[4-amino-6,8-bis(2,3-dimethoxyphenyl)imidazo[1,2-a]pyrazin-5-yl]acetamide 5-phenylmethoxybenzene-1,2,3,4,6-pentol (2E)-N'-[1-benzyl-5-[(4-fluorophenyl)methyl]imidazol-2-yl]-2-hydrazinylideneethanimidamide 4-fluoro-3,6-dimethoxy-2-[(E)-2-nitroethenyl]benzaldehyde 2-(azidooxymethyl)naphthalene 3-[(2E)-2-[1-cyano-1-[4-(4,5-dihydroimidazol-1-yl)phenyl]ethylidene]hydrazinyl]benzonitrile 4-[2-(4-hydroxyphenyl)-5,6-dimethyl-1H-benzimidazol-4-yl]phenol 2-cyclopentyl-3-[4-[4-(2-methoxyethyl)piperazine-1-carbonyl]anilino]-7H-pyrrolo[2,3-c]pyridazin-6-one 2-hydroxy-5,6-dimethyl-1H-indole-3-carboxylic acid 3-[4-(2,5-difluorophenyl)-1H-benzimidazol-2-yl]-5-[(1E,3Z)-penta-1,3-dienyl]-2H-pyrazolo[3,4-b]pyridine 4-(2,3,5,6-tetramethyl-1H-pyridin-4-ylidene)cyclohexa-2,5-dien-1-one N-[4-(1-amino-3-methyliminoprop-1-en-2-yl)-3-chlorophenyl]-5,7-difluoro-2,3-dihydroinden-1-imine;ethane 4-(2,6-difluorophenyl)-7-[4-[[methyl(methylamino)amino]methyl]phenyl]-N-(3-morpholin-4-ylpropyl)pyrido[3,4-d]pyridazin-1-amine;methanol (NZ)-N-[[1-[2-fluoro-4-(trifluoromethyl)phenyl]sulfonylazetidin-3-yl]methylidene]-2,5-dimethylbenzenesulfonamide N-(5-tert-butyl-1,2-oxazol-3-yl)-4,7-dimethylthieno[2,3-d]pyridazine-6-carboxamide 1-[(E)-3-(3,4-dichlorophenyl)prop-2-enoyl]-N-[3-fluoro-5-(trifluoromethyl)phenyl]piperidine-4-carboxamide 3,5-bis(trifluoromethyl)cyclopenta[a]fluorene (5-methoxy-3,4-dihydronaphthalen-2-yl)azanide 4-[2-(2-diazohydrazinyl)ethyl]benzenesulfonic acid [1-(2,6-dichlorobenzoyl)piperidin-4-yl]-(7H-pyrrolo[3,2-d]pyrimidin-4-yl)methanone 6-butyl-2,3-dimethoxyphenol N-(2,6-dioxopiperidin-3-yl)-5-iodo-4-[4-(trifluoromethoxy)anilino]thiophene-2-carboxamide 4-[3,3-dimethyl-6-(1-phenylbenzimidazol-2-yl)indol-5-ium-2-yl]benzenesulfonate [(3R,5S)-3,5-dimethylpiperidin-1-yl]-phenylmethanone 4-methylbenzenesulfonate;oxygen(2-);triphenylphosphanium [2-methyl-4-(3-methylbutan-2-yloxy)phenyl]methanamine 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]-1-phenylethanone (5R)-3,3,4,4,5-pentadeuterio-5-[7-[[4-[dideuterio-[3-(morpholin-4-ylmethyl)phenyl]methoxy]cyclohexa-2,4-dien-1-ylidene]amino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione 3-methyl-2-(4-propan-2-ylphenyl)aniline 6-[2-(2,4-dichlorophenyl)ethoxy]-3-ethyl-1H-quinolin-2-one 3-azido-4-(2,3,6-trimethylphenyl)pyridazine 2-[5-(6-butoxypyridin-3-yl)pyridin-3-yl]-1,5,5-trimethylimidazolidine (4S)-N'-[3,5-bis(trifluoromethyl)phenyl]-2-oxo-1,3-oxazolidine-4-carboximidamide N-cyclopropyl-2,3-bis(ethenyl)aniline;4-[[1-[2-[4-(3-cyclopropylidenehexan-2-yloxy)phenyl]-6-fluoroquinolin-4-yl]-3-hydroxyazetidin-3-yl]methyl]benzonitrile 3-methylbutane;5-phenylcyclohepta-1,3,6-triene 1-(5-tert-butylthiophen-2-yl)sulfonyl-N-[[4-fluoro-3-(1,3-oxazol-5-yl)phenyl]methyl]piperidine-4-carboxamide 2-[2,3-dihydropyrrolo[1,2-a]indole-1-carbonyl(methyl)amino]acetic acid 2-[(E)-[[6,7-dimethoxy-1-(3-morpholin-4-ylpropyl)isoquinolin-3-yl]-hydroxyhydrazinylidene]methyl]benzene-1,4-disulfonic acid 1-[5-azido-2-(4,4-difluorocyclohexyl)oxyphenyl]pyrrole 2-[(2S)-4,5,6,7-tetrahydroxy-3-(2-methoxyphenyl)-1,2,3,9b-tetrahydrodibenzothiophen-2-yl]acetic acid 4-[2,6-dichloro-N-[(3-fluorophenyl)methyl]-4-nitroanilino]butan-1-ol 2-[(1,3,5-trimethylpyrazole-4-carbonyl)amino]-9H-pyrido[3,4-b]indole-1-carboxamide 6-methoxy-4,4a-dihydroindeno[1,2-d][1,3]thiazol-2-one 4-[(Z)-(3,5-dimethyl-1H-pyrrol-2-yl)-hydroxyiminomethyl]benzene-1,2,3-triol 3-[(1S)-6-fluoro-2,4-dioxocyclohexyl]-5-hydroxy-2H-isoindole-1,3-dione 3-[1-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)pyrrolidine-2-carbonyl]-1,3-thiazolidin-2-one (2R)-1-[4-[bis(4-methoxyphenyl)methyl]piperazin-1-yl]propan-2-amine 1-(3,5-dimethoxyphenyl)sulfonyl-6-hydroxy-2-[4-(methanesulfonamidomethyl)phenyl]indole-3-carboxylic acid 3-methyl-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazole 2-[(3S,4R)-4-benzylpyrrolidin-3-yl]oxybenzonitrile 6-[2-[(4R)-2,4,5-trihydroxycyclopentyl]oxyphenyl]pyridine-3-carboxamide N-[1-[2-(3,5-dimethoxyphenyl)ethyl]piperidin-4-yl]-N-propanoylmethanesulfonamide N-[4-methylsulfanyl-2-(propylamino)pyrimidin-5-yl]acetamide N-(2,4-dichloropyrimidin-5-yl)-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]methanesulfonamide 4-[4-(azidomethyl)phenyl]sulfanylmorpholine 5-methylsulfonyl-2-propyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine (2R)-1-[4-cyano-3-(trifluoromethyl)phenyl]-N-[5-[1-[2,6-di(propan-2-yl)anilino]ethyl]pyridin-2-yl]pyrrolidine-2-carboxamide 2-tert-butyl-5,6-diphenylpyridine ethane;N-[[4-[3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)propoxy]phenyl]methylidene]hydroxylamine 2-(3,5-difluorophenyl)-N'-[(Z)-1H-indol-3-ylmethylideneamino]ethanimidamide 2-methyl-N,3-bis(4-phenylphenyl)benzenecarboximidate N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-prop-2-enylbutanamide N-[1-(2,5-dimethylpyrazol-3-yl)ethenyl]-4-[5-fluoro-6-methoxy-4-[(1-methylpiperidin-4-yl)amino]pyridin-3-yl]pyridin-2-amine (4R,5S)-5-[4-(4-chlorophenyl)-2-fluoro-6-methoxyphenyl]-1,3-dioxan-4-ol 2-(1,3-benzodioxol-5-yloxy)-N-methyl-N-[3-(4-pyridin-2-ylpiperazin-1-yl)propyl]acetamide 5-[(1S)-3-amino-2,2,4-trimethylcyclobutyl]pyridine-3-carboxylic acid 6-cyclohexa-1,3-dien-1-yl-4-(2-phenylethenoxy)pyridine-3-carbonitrile 3-[1-(4-cyclopropylphenyl)ethenylamino]pyridine-2,6-dicarboxylic acid 3-[4-[1-(2,2-difluoropropyl)pyrazol-4-yl]triazol-1-yl]thiophene-2-carboxamide N-[5-(diethylaminomethyl)pyridin-3-yl]imidazo[1,2-a]pyrazine-8-carboxamide 3-cyclopentylsulfanyl-5-(4-ethylphenyl)-N'-hydroxypyridine-2-carboximidamide 6-[4-chlorobutyl(cyclohexyl)amino]-2-sulfanylidene-1H-pyrimidin-4-one 5-[(2E,4Z)-hepta-2,4,6-trienyl]-1-hexan-3-ylpyrazole (5S,7S)-N-[2-(4-chlorophenyl)ethyl]-1-methyl-3-propanoyl-6-oxabicyclo[3.2.0]heptane-7-carboxamide N-[(E)-1-cyclopenta-2,4-dien-1-ylprop-1-enyl]aniline 6-(1,3-benzothiazol-2-yl)-4-propan-2-yloxypyran-2-one 5-azidooxy-N-tert-butyl-2,3-dichlorobenzenesulfonamide 2-[1-(3,4-dimethylphenyl)butyl]-N-methyl-5-nitroaniline 7-fluoro-2-[(4E,5Z)-4-ethylidene-1,6-dimethyl-2-oxo-3-propan-2-ylidenepyridine-5-carbonyl]-3H-isoindol-1-one 2-[3-(dimethylamino)propylimino]-5-[2-hydroxyethyl-(6-oxo-4-phenyl-1H-pyrimidin-2-yl)amino]imidazolidin-4-one 2-(4-methylpiperazin-1-yl)-5-[(3R,6S)-3-methyl-6-propanoyloxyheptyl]benzoic acid 1-[3,5-diamino-4-(2,6-dichlorophenyl)phenyl]ethanone;hydrochloride 2,5-difluoro-4-[3-methyl-6-[(7H-purin-6-ylamino)methyl]cyclohexa-1,5-dien-1-yl]benzaldehyde (4aS)-8-[5-(2,6-difluorophenyl)pyridin-3-yl]-4a-methoxy-2,12-dihydro-1H-naphtho[2,1-f]isoquinoline N-[[4,5-bis(ethenyl)furan-2-yl]methoxy]-1,6-diiodo-3-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide 2-(4-chlorophenyl)-7,8-dihydroquinoxaline [(3S,4R)-1-[(2-aminopyridin-4-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methanol 6-(3,5-dimethoxyphenyl)-4-methoxypyrazolo[1,5-a]pyridine 5-amino-6-phenyl-3-(1,2-oxazol-3-ylmethoxy)pyrazine-2-carboxamide 3-[3-(2,5-dihydroxyphenyl)phenyl]propyl-triethylazanium;4,6-dimethoxynaphthalene-2-sulfonate (2R)-2-[7-(4-chlorophenyl)-5-methyl-2-(1,3-oxazol-2-ylamino)-1,3-benzothiazol-6-yl]-2-propoxyacetic acid;2-methoxypyridine 2-N,3-N-dibenzylfuran-1,2,3,4-tetramine 4-[[(2Z,5E)-3,7-dimethylocta-2,5,7-trienoxy]methoxymethyl]benzaldehyde 2-methoxy-3,6-di(propan-2-yl)benzonitrile 3-[1-(5-chloro-6-fluoropyrimidin-4-yl)piperidin-4-yl]-2H-1,3-thiazole 1-[3,5-dimethyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]propan-2-one 2-[2-[5-(4-bromophenoxy)pentyl]phenoxy]acetic acid (2R)-1,3-dihydroxy-2-phenylpropane-2-sulfinic acid 2-hydroxy-1-[2-(6,7,8,9-tetrahydropyrido[3,2-b]indolizin-11-ylmethoxy)-5-thia-1-azatricyclo[6.4.0.02,6]dodeca-2(6),3,7-trien-9-yl]ethanone 4-[2,6-difluoro-3-(pyridin-2-ylmethoxy)benzoyl]piperazine-1-carboxylic acid 2-(3,5-dibromo-4-fluorophenyl)sulfanyl-N'-hydroxypyrimidine-4-carboximidamide 3-[4-[5-(2,6-dimethylpyridine-3-carbonyl)pyrazin-2-yl]oxyphenyl]-1-pyrrolidin-1-ylpropan-1-one 3-[[2-butyl-4-(trifluoromethyl)imidazol-1-yl]methyl]pyridine 3-chloro-6-fluoro-4-methylthieno[2,3-b]pyridine;6,8-dimethoxy-5,7-dimethylquinoline 5-(2-bromo-4,6-dihydroxyphenyl)-N'-[(Z)-(3-ethoxy-4-hydroxyphenyl)methylideneamino]-1H-pyrazole-4-carboximidamide 4-azido-2,3,5-triphenylfuran 2-(8,10-diphenyl-1,3,11-triazatricyclo[7.4.0.02,7]trideca-2,4,6,8,12-pentaen-4-yl)-5-phenylpyrido[3,2-b]indole 3-(4,6-dichloropyrimidin-5-yl)oxy-1-ethynylazetidine 1-[(4-cyanophenyl)methyl]-3-[(2S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl]urea 5-chloro-4,6-dimethoxypyrrolo[3,4-b]pyridine-1-carboxylic acid 3-[5-methoxy-1-(2,2,2-trifluoroacetyl)indol-4-yl]piperazine-1-carboxamide 2-(1-methylpiperidin-4-ylidene)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine 2-azidooxy-4,5-dichloro-3-(3-ethyl-6-fluoropyridin-2-yl)-6-methylsulfanylpyridine 2-azido-5,6-dibromo-3-ethylpyridine 1-(2-aminophenyl)-3-[2-[5-(4-chlorophenyl)sulfanylthiophen-2-yl]ethyl]thiourea N-[[1-(3,3a,4,5,6,6a-hexahydro-2H-cyclopenta[b]pyrrole-1-carbonyl)pyrrolidin-2-yl]methyl]benzamide (2S)-N'-hydroxy-2,3-diphenylpropanehydrazide 4-fluoro-2-methyl-N-[1-(5,6,7,8-tetrahydroquinazolin-4-yl)piperidin-3-yl]benzamide 1,2-diamino-4-[3-(3-hydroxyphenoxy)phenyl]-6-oxopyridine-3,5-dicarbonitrile N-[3-(2,3-dihydropyridin-4-yloxy)-5-fluorophenyl]-1H-pyrrolo[3,2-c]pyridine-6-carboxamide 1-[4-(2-methylpyrrolidine-1-carbonyl)phenyl]imidazolidin-2-one (2S)-N-[2,6-difluoro-4-(1H-indol-3-yl)phenyl]-2,4-dihydroxy-3-methoxybutanamide [(4E)-1,3-bis(4-methylphenyl)-6,7-dihydroindazol-5-ylidene]-dimethoxyazanium;chloride N-[6-[4,5-dihydroxy-2-(1H-indol-3-ylmethylidene)piperidin-1-yl]pyridin-3-yl]-5-(furan-2-yl)pyridine-2-carboxamide 4-[4-[(2R)-2-cyclopropylpiperidine-1-carbonyl]phenyl]benzonitrile 1-[2,6-di(propan-2-yl)phenyl]-4-[3-fluoro-5-(trifluoromethyl)phenyl]sulfinyl-N-iodoimidazole-2-carboxamide 3,5-diamino-6-[(E)-2-[6-bromo-1H-indol-2-yl]ethenoxy]cyclohexa-1,5-diene-1-carboxylic acid 3-[(4Z)-2-cyclooctyloxyimino-4-propylidene-1,3-thiazol-3-ium-5-yl]-N'-hydrazinyl-N-methylidenebenzenecarboximidamide 4-ethylpyridine;[5-methyl-6-[2-methyl-3-(oxan-4-yl)imidazol-1-ium-1-ylidene]cyclohexa-2,4-dien-1-yl]methanethiol 2-[3,5-bis(trifluoromethyl)phenyl]-N-methyl-3,4-dihydropyridin-6-amine (2-methylnaphthalen-1-yl)oxy-oxidosulfanium 2-azido-5-(4-chlorophenyl)pyridine 3-[[4-(2,5-dimethylphenyl)imino-1,3-thiazolidin-2-ylidene]amino]benzamide 4-[6-(1-azidocyclopropyl)pyridin-2-yl]sulfonylphenol 2-[(3S)-4,5-dimethyl-6-oxoheptan-3-yl]isoindole-1,3-dione 5-methylsulfanylpyrimidine;N-[3-(1,2,4-triazol-1-yl)phenyl]formamide 1,2-bis[(3-methylphenyl)imino]guanidine;hydrate 1-methyl-3-[3-(pyridin-2-ylamino)phenyl]thiourea 2-(3,4-dichlorophenyl)-7-[1-(oxan-2-ylmethyl)piperidin-4-yl]pyrido[2,3-d]pyrimidine 4-chloro-5-fluoro-2,3-dihydro-1H-indole-6-carbonitrile;ethane 5-methyl-2-(5,6,7,8-tetrahydronaphthalen-1-yl)-1H-indole [4-(dimethylamino)phenyl]-bis(2,4,6-trihydroxyphenoxy)phosphanium N-[1-(2,4-dimethyl-6-oxocyclohexa-1,3-dien-1-yl)-5-(4-methylphenyl)pyrazol-3-yl]thiophene-3-carboxamide (Z)-3-[2,4-difluoro-5-[3-(fluoromethyl)pyridin-2-yl]phenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile 2-[(E)-3-chloro-2,6-dimethylhept-1-enyl]quinoline;ethane;ethene (1S,3R)-6-chloro-3-[(2-fluorophenyl)methyl]-N-(4-methoxyphenyl)-1-phenyl-3a,4-dihydro-1H-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide N-[1-[3-(benzenesulfonamido)phenyl]ethyl]-2-[[4-[ethoxymethyl(methyl)amino]cyclohexyl]methylsulfonyl]acetamide 4-[2-(6,7-dihydrodibenzofuran-3-yl)phenyl]pyridine 1-[4-[2,6-difluoro-3-(4-hydroxyphenyl)phenyl]piperazin-1-yl]ethanone 2-amino-N,3,4,5,6-pentadeuteriobenzenesulfonamide (3E,4Z)-2-(4-chlorophenyl)sulfonyl-3-ethylidenehepta-1,4-diene-5-sulfonamide 4-[(2S)-5,7-dichloro-2-methyl-3-oxo-1H-isoindol-1-yl]piperidine-2-carboxylate 2-[1,4-dimethyl-6-(trifluoromethoxy)indol-2-yl]-3H-benzimidazole-5-carboxylic acid 3-[4-(ethoxymethyl)phenyl]-6,6-dimethylpyrano[2,3-d]pyrimidine-1,2,4-trione N-[2-fluoro-3-(2-methoxy-5,6,7,8-tetrahydronaphthalen-1-yl)phenyl]methanimine (4-azidooxyphenyl)-pyrrolidin-1-ylmethanone 6-[2-(difluoromethoxy)phenyl]imidazo[1,2-a]pyridine;N,N-dipropylformamide N-(4-bromophenyl)-1,2,4-triazol-3-amine 2-[(2E)-4,5-dimethylhepta-2,6-dien-3-yl]oxy-N'-hydroxypyridine-4-carboximidamide 5-[(Z)-aminomethylideneamino]-2-(methylamino)pyridine-3,4-dicarbonitrile 3-[7,8-dideuterio-5-(2-fluorophenyl)pyrido[4,3-b]indol-3-yl]-9-methoxycarbazole 4-methoxy-6,8-dimethylquinoline-3-carbonitrile 4-(2,6-dichloropyridin-4-yl)oxy-3-ethanimidoylbenzonitrile (3-butyl-1,2-benzoxazol-6-yl)methanol 7-[(2,4-dihydroxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one (5Z)-2-cyclopentylimino-5-[(1,3-dimethoxy-1,3-dioxopropan-2-yl)amino]-4-imino-7-thiophen-3-yl-3H-azepine-6-carbonitrile N-[(3-aminophenyl)methyl]-5-chlorothiophene-2-carboxamide 5-cyclopropyl-N-(2-methylpyrazol-3-yl)-1,2-oxazole-4-carboxamide 2-[[3,5-bis(trifluoromethyl)phenyl]iminomethyl]quinolin-8-olate;cobalt(3+);tetrachloride 5-(4-iodophenyl)sulfinylpentanal (1R,2S)-N-[3,5-bis[2-methyl-4-[methyl(2-pyridin-2-ylethyl)amino]pentan-2-yl]oxyphenyl]-2-phenylcyclopropane-1-carboxamide 2-bromo-5-(3,4-dihydro-1H-isoquinoline-2-carbonyl)benzenecarboximidamide 2,5-dimethyl-6-nitro-3,4,4a,9b-tetrahydro-1H-indeno[1,2-c]pyridine N-[1-[2,3-bis(ethenyl)phenyl]ethenoxymethyl]acetamide [2-[6,7-bis(ethenyl)quinoxalin-2-yl]azaniumylidene]methylazanide 2-(4,5-diphenyl-1H-imidazol-2-yl)phenol N-[4-[6-(2-fluoroethoxy)pyrazolo[1,5-a]pyridine-3-carboximidoyl]phenyl]propanamide 4-[5-cyclopropyl-3-(methylamino)pyrazol-1-yl]-N'-hydroxybenzenecarboximidamide N-[(4R)-5-amino-5-sulfanylpentyl]-3,4-dichlorobenzamide N-[4-(azidomethyl)-1,3-thiazol-2-yl]-3H-benzimidazole-5-carboxamide 2-[(4S,8aR)-4-benzhydryl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-N-(6-fluoroimidazo[1,2-a]pyridin-8-yl)acetamide 1-(2,4-dichlorophenyl)-6-hydroxy-5-[5-[3-methoxy-4-(2-phenylethyl)phenyl]-4,5-dihydro-1H-pyrazol-3-yl]pyrimidine-2,4-dione 4-bromo-1,2-dihydronaphthalene;ethane N-[1,3-bis(4-methoxyphenyl)propan-2-yl]acetamide 4-(1,3-dioxolan-2-yl)-5-ethyl-7H-pyrrolo[2,3-d]pyrimidine 1-[(2R,4S)-3-hydroxy-2-[[methyl-[5-methyl-6-(triazol-1-yl)pyridin-3-yl]amino]methyl]piperidin-4-yl]-N,N-dimethyltriazole-4-carboxamide 6-[1,2-difluoro-2-(4-hexylphenyl)ethenyl]-1-fluoronaphthalene 3-methyl-5-phenylsulfanyl-2H-1,4-benzoxazine 2-[4-(oxiran-2-ylmethoxy)phenyl]pyridine 5-[(2R)-butan-2-yl]sulfonylpyridine-3-carboxylic acid 7-amino-5-[3,5-bis(trifluoromethyl)phenyl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile 4-(azidomethyl)-3-chloro-2,6-dimethoxypyridine 1-[(2E)-1,3-benzothiazol-2-yl]-3-benzyl-5-(4-butoxyphenyl)sulfanylindole N-[5-fluoro-6-(2,3,4,5-tetradeuteriopyrrol-1-yl)pyridin-2-yl]-4-methoxypyrrolo[1,2-a]pyrimidine-8-carboxamide 4-[2-[3,5-dichloro-4-[[6-(trifluoromethyl)pyridin-3-yl]methoxy]anilino]cyclopenten-1-yl]sulfonylmorpholine (4-diphenoxyboranyl-3,5-dibromophenyl)-methoxyazanium N-[4-(5,6-dihydropyrido[2,3-b]pyrazin-7-yl)butyl]-1,2-benzothiazole-3-carboxamide 3-methyl-N-[2-[(E)-3-oxo-3-(5-pyrimidin-4-ylthiophen-2-yl)prop-1-enyl]phenyl]butanamide 5-bromo-3,4-difluorofuran-2-carboxylic acid (E)-3-(2-fluorophenyl)-N-[2-[6-methyl-7-(oxan-4-yloxy)quinazolin-4-yl]ethyl]prop-2-enamide 2-[4-(3,5-dimethylpyridin-2-yl)phenyl]benzonitrile 4-azidooxynaphthalene-1,3-dicarbonitrile 2-[2-(3,4-dimethoxyphenyl)ethyl]-8-[[2-(5-hydroxy-1H-indol-6-yl)ethylamino]methyl]quinolin-7-ol (2R,3S)-N-[3,5-bis(trifluoromethyl)phenyl]-1-cyano-N'-methyl-2-phenylpiperidine-3-carboximidamide 2-amino-1-[4-methyl-3-(trifluoromethyl)phenyl]ethanol;ethane 2-[(3,5-difluorophenyl)methyl]-N-[(4,6-dimethyl-2-oxopiperidin-3-yl)methyl]-1-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide [2-(1,3-dioxolan-2-yl)piperidin-1-yl]-[5-methoxy-6-(2H-tetrazol-5-yl)pyridin-3-yl]methanone 2-[(7S)-9,10-bis(trifluoromethylsulfonyloxy)-3-thiatetracyclo[12.4.0.02,6.08,13]octadeca-1(18),2(6),4,8(13),14,16-hexaen-11-yl]acetic acid 2-[(5R,10bR)-9-chloro-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-yl]phenol 2-(7-methyl-2,4-dihydropyridazino[9,8-b][1,4]benzoxazin-3-ylidene)propanedinitrile 1-[4-(4-bromoanilino)phenyl]sulfinylpyrrolidine 3-[(5S,6R)-8-chloro-1-(3-chlorophenyl)-2,7-dimethyl-5,6-dihydroazonine-9-carbonyl]piperidine-1-carboxylic acid 4-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-(1,3-thiazol-5-yl)amino]benzenesulfonic acid N-cyclopropyl-3-[(7S)-6,8-dihydroxy-2-methoxy-11,12-dioxo-1,4,5,10-tetrahydronaphtho[2,3-f]quinolin-7-yl]benzenesulfonamide (1R)-3,7-bis[(2-methylphenyl)methoxy]-1,2,3,4,5,6,8a-octahydroisoquinoline 2-azido-4,6-bis(2-methoxyethyl)thieno[3,2-d]pyrimidine N'-hydroxy-2,5-dimethyl-4-[(3R)-oxolane-3-carbonyl]furan-3-carboximidamide N-[(Z)-N-aminocarbamohydrazonoyl]-2-[5-methoxy-6-oxo-3-(trifluoromethyl)pyridazin-1-yl]acetamide 2-[(4R)-4,5-diphenylhexanoyl]oxyethylsulfonic acid 2-[(1,4-dimethylpiperazin-2-ylidene)amino]-1-[1-(3-ethoxyphenyl)azetidin-2-yl]ethanone 2-[3-(3,5-dimethylphenoxy)propoxy]butanoic acid N-[2-(2-cyclopentylbenzimidazol-1-yl)ethylidene]hydroxylamine N-ethyl-5,6-difluoroquinoline-8-carboxamide 3-[(4-aminobutylamino)methyl]naphthalen-2-ol;propane N'-(4,5-difluorocyclohexa-1,5-dien-1-yl)-1H-indole-6-carboximidamide N'-cyclohexyl-N-[3-[(2,5-dioxoimidazolidin-4-ylidene)methyl]phenyl]-2-(dipropylamino)ethanimidamide 2-[3-fluoro-5-(1-methylpiperidin-4-yl)phenyl]indazole 1-[4-(2-aminoethyl)piperidin-1-yl]-5,5,5-trifluoropentan-1-one;ethane 2-[3-[2,6-di(propan-2-yl)phenoxy]phenyl]acetic acid N-[3-(N'-ethylcarbamimidoyl)phenyl]formamide;methanol 3-[1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-6-ylmethyl)pyrrolidin-2-yl]pyrazine;dihydrochloride 1,2,4-triethyl-3-(2-methoxyethyl)naphthalene (2S,4R)-1-[3-chloro-4-[[1-(4,6-dimethylpyrimidin-5-yl)cyclopropyl]amino]benzoyl]-N-[1-(cyanomethoxy)-2,2,2-trifluoroethyl]-4-fluoropyrrolidine-2-carboxamide 3-(2,6-dimethoxyphenyl)-5-[(2E)-4,6-dimethylocta-2,7-dienyl]-N-[4-(4-methylpiperazin-1-yl)pyridin-3-yl]-1H-pyrazole-4-carboxamide (2R)-N,3,3-trihydroxy-4-(4-propan-2-ylphenyl)butanethioamide 3-(4,4-difluoropiperidine-1-carbonyl)-6,7-difluoro-2H-chromene-2,3-diol ethane;1-(3-methoxypropyl)cyclobutan-1-amine;5-methoxy-N,4-dimethyl-2-[6-oxo-8-(pentan-2-ylamino)purin-9-yl]pyridine-3-carboxamide N-azidosulfanyl-3-chloroaniline 4-amino-3,5-dinitrobenzamide 4-(3-azido-2,6-difluorophenyl)-1H-imidazole 1-methyl-2-[(3R)-6-oxo-1,7-dihydroimidazo[4,5-f]benzimidazol-7-ium-3-yl]benzimidazole-5-carboxamide 4-ethoxy-N'-[(3-fluorophenyl)methyl]-N,N-dimethylpyrimidine-5-carboximidamide 3-[1-(8-bromoquinoline-2-carbonyl)pyrrolidin-3-yl]oxybenzonitrile 1-[3,5-bis(trifluoromethyl)phenyl]piperidine;methane 2-[4-(benzoylsulfamoyl)-N-(3-nitrophenyl)anilino]-2-methylpropanoic acid 1-(3-fluoropyridin-2-yl)oxypropane-2,3-diol 1-[2-methoxy-4-(trifluoromethyl)phenyl]-3,3,5,7,7-pentamethyloctan-4-one 4-methoxy-N,2-dimethyl-5-[(3Z)-penta-1,3-dien-2-yl]pyrazole-3-carboxamide N-[2,2-bis(4-fluorophenyl)ethyl]-3-methoxypyrazine-2-carboxamide 1-[5-amino-2-(propylcarbamoyl)phenyl]pyrrole-3-carboxylic acid 4-[1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-6-one 3-cyclohepta-1,4,6-trien-1-yl-5-methoxy-N-(methylideneamino)aniline [2-amino-4-[5-chloro-3-(cyanomethyl)indol-1-yl]-6-fluorophenyl]methylideneazanium (2S)-N-[(3R,4S)-3,4-dihydroxy-5-[4-(6-pyridin-4-ylhexoxy)phenyl]pentyl]pyrrolidine-2-carboxamide 3-(4-methoxyphenyl)-4-(2-oxochromene-5-carbonyl)pyrrolidin-2-one 2-[(3R)-1-ethylpiperidin-3-yl]oxy-5-(2,4,6-trifluorophenyl)aniline N-[2,3-bis(ethenyl)imidazo[1,2-a]pyridin-7-yl]-2,2-dimethoxyacetamide 4-[5,6-bis(ethenyl)pyridin-3-yl]-1H-benzimidazole 1-[4-amino-5-(4-chlorobenzoyl)-3,6-dihydro-2H-pyridin-1-yl]-3-methoxypropan-1-one 2-(3-amino-1H-pyrazol-5-yl)-4-bromo-6-methoxyphenol 5-(azidooxymethyl)naphthalene-2-carboxylic acid 3-[1-[4-(dimethylamino)phenyl]sulfonylpiperidin-4-yl]oxy-N,2-bis[(4-fluorophenyl)methyl]benzamide (3E)-4-amino-3-[[2-fluoro-5-methoxy-6-(trifluoromethyl)phenyl]methylidene]azete-2-thione 4-[4-(benzylamino)phenyl]benzamide [4-amino-3,5-di(propan-2-yl)cyclohexa-1,5-dien-1-yl]-phenylmethanone N-[(E)-(3,5-dibromo-2,4-dihydroxyphenyl)methylideneamino]-3-(4-oxoquinazolin-3-yl)propanamide 3-(cyclohexylamino)pyrazine-2-carboxylic acid 1-(3,4-dimethoxyphenyl)piperazine;formic acid N-(3,5-dichlorophenyl)-2-[(6-oxo-4-propyl-1H-pyrimidin-2-yl)sulfanyl]butanamide (2S)-1-[4-(cyclopropanecarbonyl)piperazine-1-carbonyl]-N-methoxy-5,5-dimethylpyrrolidine-2-carboxamide;ethane 1-(2,4,6-tribromophenyl)imidazole 1-(5,6-dihydropyrrolo[2,3-b]pyridin-1-yl)propan-1-one 1-(4-hydroxyphenyl)-2-morpholin-4-ylbutan-1-one 5-tert-butyl-2-hydroxy-3,4,6-triiodobenzenecarboximidamide 2-[1-(6,7-dimethoxyquinazolin-4-yl)piperidin-4-yl]acetic acid 2-[3-fluoro-4-(trifluoromethyl)phenoxy]propanoic acid N-[(3S)-9,10-difluoro-2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl]carbamate (2S)-N,2-dihydroxy-4-methylsulfanyl-1-(3,4,5-trifluorophenyl)butanamide 5-[(2S)-5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]thiophen-2-amine 2-(4-chlorophenyl)-3,5,7-trimethylcyclohepta-1,3,6-triene 2-N,2-N-bis(propan-2-yloxy)acenaphthylene-1,2-diimine ethane;4-methyl-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-2-yl]benzamide [(Z)-1-[2,6-difluoro-4-[5-(methoxymethyl)pyrazol-1-yl]phenyl]-3,3,5,5,8,8-hexamethyloct-7-en-2-ylideneamino]thiourea (1S,3R)-3-[[(2R)-1-(3,4-dimethylphenyl)propan-2-yl]amino]cyclohexane-1-carboxylic acid [(2S)-6-chloro-4,5,10,12-tetrahydroindolo[3,2-c]carbazol-8-yl]-phenylmethanone N-[(2,5-dimethylphenyl)methyl]-3-(imidazol-1-ylmethyl)benzamide N-(4-bromobutan-2-yl)-4,5-dichloro-N-(3-methylbutyl)aniline N-[(Z)-N'-diphenylphosphanyl-N-methylcarbamimidoyl]acetamide N-[(4S)-2-cyclopropyl-1-[5-[[4-(trifluoromethoxy)benzoyl]amino]pyridine-3-carbonyl]piperidin-4-yl]ethenesulfonamide 3,5-dichloro-6-[2-(1-methyltriazol-4-yl)ethyl]pyridazine 2-[4-methoxy-3-(trifluoromethyl)phenyl]oxan-4-ol N-[(1S,2R)-2-methoxycyclohexyl]-2-pyrimidin-5-ylpyrimidine-4-carboxamide [3-hydroxy-5-[2-(1H-imidazol-2-yl)ethyl]pyridin-2-yl]methanediol 5-[[4-[2-(2,3-dimethoxyphenyl)ethynyl]benzoyl]amino]pyridine-3-carboxylic acid [3-[[4,6-bis(3-cyanophenyl)-1,3,5-triazin-2-yl]amino]phenyl]boronic acid 3-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)cyclobutanecarbonyl]oxypropanoic acid 3-(4,5-dichloro-2-hydroxyphenyl)cyclopropane-1,1,2,2-tetracarbonitrile 2-[4-(1,3-dioxoisoindol-5-yl)oxybutoxy]propanoate 1-[4,5-dimethoxy-3-(2-pyrrolidin-1-ylethoxy)indol-1-yl]propan-2-ol 4-[[3-[6-(1,2,3,5,6,7-hexahydropyrrolizin-8-yl)pyridin-2-yl]propanoylamino]methyl]cyclohexane-1-carboxylic acid 4-(3,5-ditert-butylphenyl)-2H-azirine 2-hydroxyethyl(dimethyl)azanium;N'-[[1-(trifluoromethoxy)naphthalen-2-yl]iminomethyl]benzenecarboximidamide 6-[(1Z)-buta-1,3-dienyl]-2-methylidene-5,7-dihydrobenzimidazol-1-ol [2-(methylamino)phenyl]-(4-morpholin-4-yl-1H-pyrrolo[3,4-c]pyridin-6-yl)methanone 3-[4,5,6-trimethyl-2-(1-piperidin-1-ylbutan-2-ylideneamino)pyrimidin-4-yl]benzenesulfonic acid 3-[(1S)-6,7-dimethoxy-2H-chromen-3-yl]propan-1-ol 2-[3-(cyclopropanecarboximidoyl)-6-hydroxy-1H-indazole-5-carbonyl]-N',4-dimethyl-1,3-oxazole-5-carbohydrazide N-[(1R)-3,4-dihydro-2H-chromen-7-yl]butane-1-sulfonamide 2-[4-ethyl-1-(4-methylphenyl)sulfonylpiperidin-2-yl]acetic acid N-[1-(2,3,4,6,7,8-hexahydrochromen-5-yl)ethenyl]acetamide 1-cyclohexyl-2,3-dimethoxybenzene N-[[4-[2-(dimethylamino)ethyl]phenyl]methyl]-2,2,3,3,5,5,6,6-octafluorocyclohexane-1-carboxamide [3,5-bis(trifluoromethyl)phenyl]-[4-(cyclohexylamino)piperidin-1-yl]methanone N'-[2,5-dimethyl-4-[4-(3-phenoxypropoxy)phenyl]phenyl]sulfonyl-1,3-benzodioxol-4-carboximidamide (4-methylbenzotriazol-2-yl)-naphthalen-1-yldiazene N-[(Z)-1H-pyrrol-2-ylmethylideneamino]pyridine-3-carboxamide 1-(7-azido-2,4-diphenylquinolin-3-yl)piperidin-4-ol 3-[(6R)-3,5-dimethyl-1-octyl-2-oxopyrrolidin-3-yl]-4H-1,2,4-oxadiazol-5-one 3-(2,6-difluorophenyl)-5-[2-fluoro-4-(trifluoromethyl)phenyl]-1-(2H-tetrazol-5-yl)-7,8-dihydroimidazo[4,5-f]quinoline 1-[3-hydroxy-4-(pyridin-4-ylmethoxy)phenyl]ethanone N-(diaminomethylidene)-2,3-bis[(4-nitrophenyl)sulfonyl]benzamide N-[(2-methoxyphenyl)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-7-carboxamide ethane;2-[2-[6-(6-ethynylpyridin-3-yl)oxypyrimidin-4-yl]oxyethoxy]-N,N-dimethylethanamine 3-ethyl-6,7-dimethoxychromene-4-thione N-(3-amino-5H-pyrrolo[2,1-c][1,4]oxazin-7-yl)-2,6-dimethoxybenzenesulfonamide N-[3-(2,4-difluorophenyl)oxetan-3-yl]-4-(oxetan-2-ylmethoxy)piperidine-1-carboxamide 2-[7-[(3-hydroxy-1,2-dihydrobenzotriazol-5-yl)methylideneamino]heptanoylamino]butanedioic acid [4-(3,7-difluoroquinolin-6-yl)oxycyclohexylidene]methyl-ethylcarbamic acid 3-[(3R)-3-aminopyrrolidin-1-yl]sulfonylphenol (1R,2S)-N'-[[4-(4-fluorophenyl)phenyl]methyl]-5,6-dihydroxy-N-methyl-2,3-dihydro-1H-indene-1-carboximidamide 4-[3-(ethylamino)pyrrolidine-1-carbonyl]-N,N-dimethylbenzenesulfonamide 1-[(6S)-3,7-dioxo-1,4-benzoxazin-6-yl]-3-[[3-(trifluoromethoxy)phenyl]methyl]urea 2-[3-chloro-4-(1,5-dihydrotriazol-2-yl)phenyl]ethane-1,1-diol (2S)-1-azido-3-[4-(6-bromopyridin-2-yl)piperazin-1-yl]propan-2-ol [(2S,4R)-1-acetyl-2-methylpiperidine-4-carbonyl]-bis(pyridin-3-ylmethyl)azanium N-(6-chloropyrimidin-4-yl)dibenzofuran-4-amine N-[(1S)-2-oxocyclopentyl]-2H-chromene-7-carboxamide 1,3-bis(4-chlorophenyl)-6-[4-methoxy-5-nitro-2-[4-(trifluoromethyl)phenoxy]phenyl]-4,5-dihydropyrrolo[3,4-c]pyrazole 3-(1,3-dimethylpyrazol-4-yl)-5-[(2R,6S)-6-(5-fluoropyridin-2-yl)piperidin-2-yl]-1H-1,2,4-triazole (4-acetylphenyl)sulfonylazanium 3-[4-(3,5-dimethylphenyl)butoxy]benzamide N-[(2R,3S)-1-azido-4,6-dioxo-2-phenylpiperidin-3-yl]-2-methoxyacetamide N-[(2S,4R)-1-hydroxy-1-(5-thiophen-3-ylindol-1-yl)propan-2-yl]-6-nitropyridine-2-carboxamide N'-ethyl-2,3,4,9-tetrahydroxanthene-1-carboximidamide 2-[4-azido-3,5-dichloro-6-(trifluoromethyl)pyridin-2-yl]oxyethanol 2-[(E)-pent-3-enyl]-6,7-bis(4-pentoxyphenyl)thieno[3,2-f]indole N-[6-(4-ethylpiperazin-1-yl)pyridazin-3-yl]benzamide 2-[(3S)-1-[[6-(2,4-dimethylpyrazol-3-yl)pyridine-3-carbonyl]amino]pyrrolidin-3-yl]acetic acid 6-(8-bromoimidazo[1,2-a]pyridin-5-yl)-3H-indole-4-carboxylic acid 2-[N-benzyl-4-(pyridin-2-ylamino)anilino]ethanol N-[(2R,4S)-1-[2-hydroxyethyl(methylsulfanyl)amino]-3-methyl-1-oxohexan-2-yl]-6-oxo-5H-benzo[b][1,4]benzoxazepine-11-carboxamide (3R)-N,1-dimethyl-4-[3-(2-phenylethynyl)phenyl]sulfonylpyrrolidine-3-carboxamide N-[1-[4,4-difluoro-3-(propanoylamino)piperidin-1-yl]-2-methoxyethylidene]thieno[2,3-b]quinoline-2-carboxamide 2-[4-(3,5-dimethylphenyl)piperidin-1-yl]-N-[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]acetamide 3,4-ditert-butyl-5-octoxybenzoic acid 2,7-ditert-butyl-3-[2-(4-ethenoxyphenyl)ethynyl]fluorene 5-chloro-N-[(2S)-1-[(4,6-dimethylpyrimidin-2-yl)amino]propan-2-yl]thiophene-2-sulfonamide N-[5,6-bis(ethenyl)pyridin-3-yl]-N',2,4-trimethylbenzenecarboximidamide 2-(1H-indol-3-ylmethylideneamino)-N,N,1-tripropylbenzimidazole-5-sulfonamide (2Z)-2-[5-[1-(2,3-dihydro-1H-inden-2-ylamino)-1-oxopropan-2-ylidene]cyclohexa-1,4-dien-1-yl]oxyiminoacetaldehyde N-(3,5-difluorophenyl)sulfonyl-4-[3-ethoxy-2-hydroxypropyl(methyl)amino]butanamide 3-(1H-indol-4-yl)propanamide 6-[2,4-dichloro-N-(3-methylbut-2-enyl)anilino]hexanoic acid 2-(3,4-difluorophenyl)imino-5-[1-[4-methoxy-2-(trifluoromethyl)anilino]ethylideneamino]pentanenitrile 3-methyl-N-(6-nitro-1H-benzimidazol-2-yl)butanamide 2-(azidooxymethyl)-1,4-diethylbenzene 5-bromo-2,3-dimethylbenzenesulfonate [4-(2-phenyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-[6-(trifluoromethyl)pyridin-2-yl]methanone 5-fluoro-6-methyl-2,3,4,9-tetrahydrocarbazole 3-ethyl-N-[1-[3-(1H-pyrrolo[2,3-c]pyridin-2-yl)pyridin-4-yl]butan-2-ylidene]hepta-4,6-dienamide (3-hydroxy-2-methylbutan-2-ylamino)-[4-(trifluoromethyl)phenyl]methanol 2-[1-(4-fluorobenzoyl)piperidin-4-yl]oxy-5-methoxybenzamide 3-hydroxy-2-phenylbenzoic acid;hydrate 2-[(5R)-6,7,8,9-tetrahydro-5H-fluoren-1-yl]propanoic acid N-[4-[3-acetyl-6-(2,3-dihydroxypropoxy)-1H-pyrrolo[3,2-b]pyridin-5-yl]phenyl]-2-oxo-2-pyrrolidin-1-ylacetamide 2-N-[3-(hydroxymethyl)cyclobutyl]-6-propan-2-ylpyridine-2,5-dicarboxamide 4-(4,5-dichlorothiophen-2-yl)sulfanylpiperidine N-[3-(3,4-dimethoxyphenyl)propyl]-5-iodo-1,2,4-oxadiazol-3-amine 5-[3-methyl-4-(trifluoromethyl)phenyl]-1H-pyrrole-2-carbonitrile 5-(3,4-dichlorophenyl)-N-[3-(hydroxymethyl)oxan-4-yl]pentane-1-sulfonamide 3-benzylsulfanyl-5,8-dimethyl-1H-quinoline-2,4-dione;ethane 6-[7-fluoro-2-(1H-indol-3-ylmethyl)-3,4-dihydro-1H-isoquinolin-6-yl]-N-hydroxyhexanamide 2-chloro-5-[(4-methylsulfonylphenyl)diazenyl]thiophene-3,4-dicarbonitrile 4-amino-1-[2,6-dichloro-3-(trifluoromethyl)phenyl]-5-methylpyrazole-3-carboxylic acid 1-[(3S)-6,8-dimethoxy-3-methyl-3,4-dihydro-2H-quinolin-1-yl]ethanone;ethane 4-[(2Z,3E)-2-ethylidenehexa-3,5-dienyl]benzonitrile 7-chloro-3,4-difluoro-2,6-naphthyridine 5-[1,3-dihydroisoindole-2-carbonyl(formyl)amino]pyridine-3-carboxylic acid 4-(1,3-benzodioxol-5-yl)-N,2-bis[(4-methoxyphenyl)methyl]butanamide N-(3-bromopropyl)-2-chloro-4-fluoroaniline 2-ethyl-4-(1,3-thiazol-5-ylmethyl)-7H-pyrrolo[2,3-d]pyrimidine 3-[N-hexadecyl-4-(pyridin-2-ylamino)anilino]propane-1,2-diol 7-cyclohexyloxy-N-[3-(methylaminosulfanyl)phenyl]pyrrolo[2,1-f][1,2,4]triazin-4-amine N-[(3R)-1-methylpyrrolidin-3-yl]-4-propan-2-ylpyridine-2-carboxamide 3-(2,4-dihydroxyphenyl)-4-[6-(3,5-dimethyl-1H-pyrazol-4-yl)-1,5-naphthyridin-3-yl]-1H-imidazol-2-one 2-azido-7-[(4-chlorophenyl)methoxy]chromen-4-one 1-(azidomethyl)-3,7-difluoronaphthalene 3-chloro-6,8-diethylbenzo[c]cinnoline N-[2-chloro-4-[[(5Z)-5-(hydroxymethylidene)furan-2-yl]sulfonylamino]phenyl]furan-3-carboxamide 4-(azidooxymethyl)-2-(trifluoromethyl)pyridine 5-[3,6-bis(trifluoromethyl)carbazol-9-yl]sulfonylbenzene-1,2,4-triol 4-chloro-2-[(Z)-[(1-cyclopropylpyrazol-3-yl)hydrazinylidene]methyl]phenol 4-[5-[4,6-bis(2,3-dimethylphenyl)pyridin-2-yl]benzimidazolo[1,2-a]benzimidazol-9-yl]benzonitrile N-[3-(dimethylamino)propyl]-2,3-diethoxybenzamide (1R)-N,2-dimethyl-2-[4-[methyl-[5-[[3-methyl-2-[[4-(6-oxohexanoyloxy)butan-2-ylideneamino]methyl]phenyl]methoxy]pyrimidine-2-carbonyl]amino]piperidine-1-carbonyl]cyclopropane-1-carboxamide (1S,2R)-2-methyliodanuidyloxy-N-phenyl-1-[4-(tetrazol-1-yl)phenyl]propanamide (2S)-5-acetyloxy-4-oxo-6-[3-(4-piperidin-1-ylphenyl)phenyl]hexanoic acid 2-[3,6-difluoro-5-methyl-1-(4-piperidin-1-ylbutoxy)isoquinolin-8-yl]propanal (2R)-2-[3-oxo-5-(1,3,4-thiadiazol-2-ylsulfanylmethyl)-1H-isoindol-2-yl]-N-[2-(1,4,7,10-tetrazacyclododec-1-yl)ethyl]propanamide 3-[4-(3-methylimidazol-4-yl)sulfonylmorpholin-2-yl]propanoic acid N-cyclopropylsulfanyl-3,5-difluoroaniline 4-methyl-3-[1-(2,3,6-trifluorophenoxy)propan-2-ylamino]-5-(trifluoromethyl)benzoic acid 2-amino-4-[1-(methyliodanuidylsulfonyloxyamino)ethyl]benzoic acid 5-(3-tert-butyl-1,2-oxazol-4-yl)pyridine-2-carboxamide N-cyclohexyl-1,3-benzodioxole-5-carboxamide (2S,3R,4S)-1-[1-benzyl-3-hydroxy-5-(hydroxymethyl)pyrazole-4-carbonyl]-N-(pyridin-3-ylmethyl)-4-[2-[(2R)-2-(trifluoromethoxy)piperidin-1-yl]ethylamino]pyrrolidine-3-carboxamide 2-(3,5-dihydroxyphenyl)quinazoline-4-carbonitrile 2-azidooxyquinoline-7-sulfonic acid N-[(Z)-4-methylpent-2-enyl]-N'-phenylmethanimidamide;3-N,2-N-dipyridin-2-ylquinoxaline-2,3-diamine (Z,2R)-N'-diazenyl-3-ethoxy-2-[(1S)-2-phenylsulfanyl-1-pyridin-4-ylprop-2-ynyl]but-3-enehydrazide 5-chloro-N'-hydroxy-1H-imidazo[4,5-b]pyridine-2-carboximidamide (2R)-3-amino-1-[4-[(2S,4S)-2-hydroxyhexanoyl]piperazin-1-yl]-2-methyl-N'-phenylpropanediamide (2E)-1,3,3-trimethyl-N-[(4-methylphenyl)methoxy]isoquinoline-2-carboxamide 2-(4-methylphenoxy)quinoline 3-[2,5-dimethyl-1-(3-nitrophenyl)pyrrol-3-yl]propanamide (E)-3-[4-[[(2S,5R)-6-amino-5-(4-phenylbutanoyloxymethyl)-1,4-oxazepan-2-yl]methylamino]phenyl]prop-2-enoic acid 2-(4,5-diphenylimidazol-1-yl)ethoxymethanethiolate 3-[3,4,5-trihydroxy-6-(2H-naphthalen-1-yloxy)oxan-2-yl]oxybenzoic acid 4-[(E)-1-(5-fluoropyrimidin-2-yl)-3-methoxy-3-oxoprop-1-enyl]piperidine-4-carboxylic acid 1-[5-(4-fluorophenyl)pyridin-2-yl]-N-methanimidoylazetidine-3-carboximidate 2-chloro-N-[4-(6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl)cyclohexyl]pyridine-3-carboxamide 1-(2,4-dimethoxyphenyl)-6-fluoro-7-[3-[(2-methylpyrazol-3-yl)sulfamoyl]pyrrolidin-1-yl]-4-oxoquinoline-3-carboxylic acid 2-azidooxy-1,3-dimethyl-5-propan-2-ylbenzene N-ethyl-3,5-bis[4-(methoxymethoxy)-2-(trifluoromethyl)phenyl]-N-propanoylthiophene-2-carboxamide 2-amino-1-[6-(4,5-dihydropyrimidin-2-yl)-3-methylindazol-1-yl]ethanone 2-[2-(6,7-dimethoxyquinolin-4-yl)ethynyl]aniline N'-[(2E)-3,7-dimethylocta-2,6-dienoyl]-4-[[6-oxo-5-(phenylsulfanylmethylidene)-1H-pyrimidin-4-yl]amino]benzohydrazide;ethane 1-(2,4-difluorophenyl)-3-[3-hydroxy-4-[(6-morpholin-4-ylpyridin-2-yl)amino]naphthalen-1-yl]urea 2-bromo-1-(4-propan-2-ylcyclohexa-1,3-dien-1-yl)naphthalene N-(2-chloroacetyl)-4-nitro-N-prop-2-enylbenzamide 1-(2,3,5,6-tetrafluorophenyl)pentane-1-sulfonate 5-ethyl-4,6-bis(methoxymethyl)pyrimidine-2-carboxylic acid 2-[4-(ethoxymethyl)phenoxy]-6-propanoyloxybenzenesulfonate (6S,9R)-6-(furan-2-yl)-9-(4-methoxyphenyl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one 2-(6-chloropyridin-2-yl)oxy-N-[(3S,7R,8aS)-3-propan-2-yl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]acetamide 1-cyclopropyl-8-[4-(methylamino)piperidine-1-carbonyl]-6H-pyrano[2,3-b]indol-7-one 6-azidooxy-N,3,4-trimethylpyridine-2-carboxamide 1-[7,8-dimethoxy-2-oxo-4-(1-phenylethyl)chromene-3-carbonyl]azetidine-3-carboxylic acid 2-chloro-4-[(3S,5R)-1-[(E)-hex-2-enyl]-2-oxopiperidin-3-yl]benzonitrile 2-(4-aminophenyl)-1-cyclohexylethanone 1-[3-[4-amino-6,7-dimethoxy-5-(methyliminomethyl)phthalazin-1-yl]oxypropoxy]cyclobutane-1-carbonitrile N-[5-(3,4-dichlorophenyl)-1H-pyrazol-3-yl]-3-(2,5-difluorophenoxy)propane-1-sulfonamide 2-[2,5-bis(trifluoromethyl)phenyl]-N-[4-[2-[5-[(1Z,3E)-hexa-1,3-dienyl]furan-2-yl]propanoylamino]but-1-en-2-yl]acetamide 2-[3,4-dimethyl-5-(trifluoromethyl)phenyl]propanoate 4-azidooxy-3,6-dichlorophthalaldehyde 1-[(2S,3aS)-5-(4,6-dimethylpyrimidin-2-yl)-8a-(hydroxymethyl)-2,3,3a,4,6,7-hexahydrofuro[3,2-c]pyridin-2-yl]ethanone;formic acid [(3S)-6-azido-4,7-dimethoxy-3H-quinoxalin-2-yl]-phenylmethanone 2-[1,2,4-triazol-1-yl(phenyl)methylidene]propanedinitrile (2-aminophenyl)sulfonylformic acid N-[(1R,2R)-2-(4-chlorophenyl)cyclobutyl]-6-propan-2-ylpyrimidine-4-carboxamide N-[(3Z,5E)-6-[5-acetamido-1-[(4,6-dimethyl-1H-indol-2-yl)sulfanyl]pentyl]-8-chloroocta-3,5-dienyl]-2-aminoacetamide;2-(4,7-diazaspiro[2.5]octane 2-(4-methylpiperazin-1-yl)-4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridine [(3S,4R)-1-[2-chloro-5-(trifluoromethyl)phenyl]sulfonyl-4-hydroxypyrrolidin-3-yl]methanone 2-[(4-chlorophenyl)methyl]benzenesulfonate 3-[[1-benzyl-2-(ethylamino)-6,7-dihydroindol-5-yl]oxymethyl]benzonitrile 5-(5-chloro-2,3-dihydrothieno[3,4-b][1,4]dioxin-7-yl)-6,8-dihydroxy-2-propan-2-ylsulfanylnaphthalene-1,4-dione N-(4,4-dimethylpentan-2-yl)-3-phenylsulfanylpropanamide [3-(4-bromophenyl)pyrrolidin-1-yl]-(5,6,7,8-tetrahydroimidazo[2,1-c][1,4]oxazin-2-ylmethoxy)borinic acid 3-[4-[(3-fluorophenyl)methyl]piperazin-1-ium-1-yl]-2,6-dihydro-1H-pyridine N-[4-[5-methyl-2-(pyrimidin-2-ylamino)-1,3-thiazol-4-yl]pyridin-2-yl]acetamide N-(1,1-dioxothiolan-3-yl)-4-pyridin-2-ylbenzenesulfonamide 1-butyl-5,7-dihydroxy-3-methoxy-4,8-bis(piperidine-1-carbonyl)quinolin-2-one 4-[(2S)-1-tert-butylsulfanyl-3,3-dimethylbutan-2-yl]oxy-1-cyclopentyl-5-ethyltriazole 3-[4-[(6S)-2,6-dimethylmorpholine-4-carbonyl]phenyl]benzamide 2-[(2R,4S)-1-[8-amino-6-(3-cyanopyrrolo[1,2-b]pyridazin-7-yl)isoquinolin-3-yl]-4-fluoropyrrolidin-2-yl]ethylcarbamic acid 1-[2,3,4,5-tetrachloro-6-(3,5-dichlorophenyl)sulfanylphenyl]piperidine N-(4-chlorophenyl)-N'-[5-[(2,6-dimethoxybenzoyl)amino]-1H-indazol-3-yl]oxamide ethane;5-hydroxy-N,4-dimethyl-6-oxopyran-2-carboxamide N-[1,4-bis(5-ethylthiophen-2-yl)butan-2-yl]formamide;5-methylidenecyclohepta-1,3,6-triene 7-methyl-N-(4-propan-2-ylphenyl)nonanamide 5-amino-4-[7-(2-imidazol-1-ylethoxy)-3,4-dihydro-2H-quinolin-1-yl]-N-(oxan-4-ylidenemethyl)thieno[2,3-d]pyrimidine-6-carboxamide 5-azido-4,7-diethyl-1H-indazole N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-N-[(4-nitrophenyl)methoxycarbonyl]butanamide 5-[[2-cyclopropyl-4-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)piperazin-1-yl]methyl]thiophene-2-carboxylic acid;dihydrochloride 3-[4-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]piperazine-1-carbonyl]piperidine-2,6-dione N-[3-chloro-4-(trifluoromethyl)phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxamide;hydrochloride (2R)-N-[[4-chloro-3-[[4-oxo-5,6,7,8-tetrahydro-3H-quinazolin-2-yl]sulfanylmethyl]phenyl]methyl]oxirane-2-carboxamide 2-[1-(8-methylquinoline-3-carbonyl)piperidin-4-yl]-4-pyridin-2-yl-1H-pyrimidin-6-one N-methyl-3,5-bis(trifluoromethoxy)benzamide 5-(2,6-difluorophenyl)-4,7-dioxo-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile 5-[(2E,4Z)-hepta-2,4-dien-3-yl]oxy-1H-indazole 3-[(6S)-1-(2,3-difluorophenyl)sulfonylpiperidin-3-yl]-1H-benzimidazol-2-one 4-(2,5-dioxopyrrol-1-yl)-N-phenylbenzenesulfonamide 5-azidooxy-2,3-dimethyl-7-nitroquinoxaline (2R,3S)-N-hydroxy-5-methyl-2,3-diphenylheptanamide (3R,4S)-3-[(1S)-5-fluoro-2-methyl-1H-inden-1-yl]piperidine 1-(4-chlorophenyl)-3-[[5-(trifluoromethyl)-1H-imidazole-2-carbonyl]amino]urea N-[4-(2-azidoethynyl)phenyl]methanesulfonamide 4-[4-(oxan-2-yl)piperidin-1-yl]benzonitrile 2-tert-butyl-4,6,7,8,9,10-hexahydro-[1]benzothiolo[3,2-d]pyrimidine 6-[7-(1,3-dioxol-2-yl)heptoxy]-1H-quinazoline-2,4-dione 2-benzylsulfanyl-N-[4,6-dichloro-5-(4-phenylphenoxy)pyrimidin-1-ium-2-yl]acetamide 6-benzylsulfanyl-N',N'-dimethyl-2H-pyrazolo[3,4-d]pyrimidine-3-carbohydrazide 5-azido-2-(1,3-benzothiazol-6-yl)-1H-pyrimidin-6-one 3-[(2Z,4E)-4,6-dihydroxyhepta-2,4,6-trienyl]-1H-indole-5-carboxylic acid 1-(2,2-difluoroethyl)-5-[4-methyl-3-[(2Z,4E)-6-(4-piperidin-1-ylphenyl)hepta-2,4-dien-4-yl]phenyl]triazole-4-carboxylic acid 2-(N-butyl-2-hydroxy-5-nitroanilino)decanoic acid 2,4-bis(ethenyl)-5-methoxy-3-[(2Z)-penta-2,4-dienoyl]-1H-pyrrole-3-carboxylic acid 3-[6-(2-methylbutoxy)pyrazin-2-yl]cyclohexan-1-ol 2,4-dibromo-1-[(Z)-(3-chloropyridin-2-yl)methylideneamino]guanidine 3-(4-azidocyclohexyl)oxypyridine 4-ethyl-5-fluoro-2,6-dimethoxypyrimidine;formaldehyde 3-(dimethylamino)-5-methoxycarbonylbenzoic acid 2,6-dipyridin-3-ylpyrazine;ethane 4-[4-bromo-3-(1,1-difluoroethyl)anilino]cyclohexan-1-ol 3-(methylamino)-1-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]propan-1-ol 3-(2,6-dimethylphenyl)-1-ethyl-4H-imidazole-3-ium-5-carboxylic acid 3-(5,6-dimethylpyridine-2-carbonyl)oxy-2,2-difluorobutanoate 2-[2-(furan-3-ylmethyl)pyrimidin-4-yl]-1,3,4,5-tetrahydrobenzo[b][1,8]naphthyridin-6-one N-(7,8-dihydronaphthalen-1-ylmethyl)ethanamine 2-[2,4-difluoro-N-(2H-tetrazol-5-yl)anilino]acetonitrile 4-chloro-N-[5-methyl-3-(2,2,2-trifluoroethoxy)pyrazin-2-yl]benzamide N-[3,5-dichloro-2-(4,5-dihydrobenzotriazol-1-yl)phenyl]propanamide 5-azido-3,4,7-trimethyl-2H-1,6-benzothiazine 2-amino-6-bromo-7,8-dimethoxy-3H-quinazolin-4-one 2-(4,5-dimethoxy-2-nitrophenyl)ethanol 1-amino-2-[6-methyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidine-7-carbonyl]butan-1-one N-[(E)-1H-indol-3-ylmethylideneamino]-2,6-diphenylpyrazolo[3,4-d]pyrimidin-4-amine 2-cyclopentylsulfanyl-4-(3,5-dimethylphenyl)-1H-pyrimidin-6-one 4-[2-fluoro-6-(triazol-1-yl)phenyl]pyridine 3-[(2-azidophenoxy)methyl]piperidine 7-hydroxy-3-methyl-6,9-dihydropyrido[1,2-a]pyrazine-8-carbonitrile N-[4-(5-carbamoyl-1H-indazole-7-carbonyl)phenyl]-2,3-difluorobenzamide (7-ethyl-4,9-dimethoxyanthracen-2-yl)oxidanium 2-hydroxy-4,5-dimethoxynaphthalene-1,8-disulfonic acid 3-[5-(cyclopropylmethoxy)pyridin-2-yl]-2-azaspiro[4.4]nonane 5-(3,4-dimethylphenyl)-N'-hydroxypyridine-2-carboximidamide 1-[(3S,4R)-3-hydroxy-4-(1H-imidazol-5-ylmethylamino)pyrrolidin-1-yl]-2-(3-phenylphenyl)ethanone;dihydrochloride 2-ethylsulfonyl-1-[4-(7H-pyrrolo[3,4-b]pyridin-5-yl)cyclohexyl]ethanone 5-[3-(6,7-dihydro-4H-triazolo[1,5-a]pyrazin-5-ylmethoxy)phenyl]-6-fluoroquinoline (3S,4R)-1-[5-[[6-chloro-2-methyl-4-(trifluoromethyl)benzimidazol-1-yl]methyl]pyrimidin-2-yl]-4-[(2-methoxyphenyl)methylamino]piperidine-3-carboxylic acid 5-(2,3-dihydropyridin-6-yl)pyrimidine;ethane 3-[[(6Z)-6-ethylidenecyclohexa-2,4-dien-1-ylidene]amino]aniline 5-[4-[4-(1,3-dithian-2-yl)-6-oxopyridazin-1-yl]butoxymethylideneamino]pyridine-2-carbonitrile 2-chloro-N-(3,5-dimethoxyphenyl)-4-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]benzamide 5-amino-3,4-dimethyl-N-(oxan-4-yl)thieno[2,3-c]pyridazine-6-carboxamide;ethane 3-[4-(2,3-dihydroindole-1-carbonyl)phenyl]-6-methyl-1H-quinolin-2-one 4-[2-(6,7-dimethoxy-3H-imidazo[4,5-c]quinolin-2-yl)pyridin-4-yl]phenol N-[(3R,4R)-1-(6-chloropyridazine-3-carbonyl)-3-fluoropiperidin-4-yl]-5-cyclopropyl-1H-pyrazole-3-carboxamide 3-[4-(trifluoromethyl)phenyl]benzenethiol [4-[2-(1,3-benzodioxol-5-yl)pyrrolidine-1-carbonyl]piperidin-1-yl]-cyclopropylmethanone 6-(4-aminophenoxy)-2-methoxyquinoline-3-carboxylic acid N-methyl-1-[(E)-3-phenylprop-2-enoxy]propan-2-amine 3-(4,5-dimethylthiophen-2-yl)sulfanyl-1,2,4,5,6,7-hexahydropyrazolo[4,3-b]pyridine 5-[3-(oxan-2-yl)benzoyl]oxy-1-azabicyclo[2.2.2]octane-2-carboxylic acid N-[(4-methoxyphenyl)methyl]-8-pyridin-3-yl-5-oxa-2-azaspiro[3.5]nonane-2-carboxamide;2,2,2-trifluoroacetic acid 4-[5-(3,5-dimethylimidazol-4-yl)sulfonyl-1H-indol-2-yl]pyrimidin-2-amine N-[(E)-3-(4-fluorophenyl)prop-1-enyl]cycloheptanamine 2-[[6-[(dimethylamino)methyl]pyridine-3-carbonyl]amino]acetic acid (5Z)-2-imino-5-[(1-methylimidazol-4-yl)methylidene]-3,4-diphenylimidazolidin-4-one 2-[6-ethylsulfanyl-5-(3-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2,5-diazaspiro[3.4]octan-6-one N-[4-(trifluoromethyl)phenyl]sulfonyloxane-2-carboxamide 1,2-diamino-4-[3-(6-methylpyridin-2-yl)phenyl]-6-oxopyridine-3,5-dicarbonitrile (2Z,4E)-N-methyl-5-methylidenehepta-1,6-dien-3-amine;8-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-9-[1-[3-prop-1-ynyl-5-(trifluoromethoxy)pyridin-2-yl]ethylamino]-1H-purin-6-one 2-(3,4-dimethoxyphenyl)-6-[3-(pyridin-3-ylamino)pyrrolidine-1-carbonyl]-9H-fluorene-1-carboxamide N-[5-amino-4-(trifluoromethyl)pyridin-2-yl]-1,3-benzodioxole-5-carboxamide;hydrochloride 2-(4,5-dibromothiophen-2-yl)acetaldehyde;methanamine N-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide 3-[6,8-diamino-7-(1-methylpyrazol-4-yl)quinazolin-4-yl]-N-cyclopropyl-2,5-difluorobenzamide 5-benzyl-2,3-dimethyl-N-(1,2-oxazol-4-yl)thiophene-2-sulfonamide 1-benzyl-6,7,8-trihydroxyquinoline-2-thione 2-(3-nitrophenyl)sulfonyl-8-pyridin-4-yloxy-1,3,4,5-tetrahydropyrido[4,3-b]indole (4S)-N'-[2,6-dimethyl-1-[(Z)-propylideneamino]oxyheptan-3-yl]-5-oxo-4-phenylpyrrolidine-2-carboximidamide 4-(2,3-dihydro-1H-pyrrol-5-yl)-N-[3-[4-[(5-ethylsulfonylpyridin-3-yl)amino]-6-(4-propan-2-ylpiperazin-1-yl)pyrimidin-2-yl]phenyl]benzamide 3-bromo-2-(5,6,7,8-tetrahydroisoquinolin-4-yl)benzamide 4-[1,2,5-trimethyl-3-(4-oxoquinazolin-3-yl)indole-6-carbonyl]piperazin-2-one 1-[(Z)-4,5-difluoronon-2-enyl]-3-ethynylbenzene 2-azido-5,6-dipropoxypyridine 6-[(3,5-dimethoxyphenyl)sulfonylamino]pyridine-2-carboxylic acid 2,6-bis(tert-butylcarbamoyl)benzenesulfonic acid;yttrium N-(4-fluorophenyl)pyridine-2,5-diamine (2S)-1-[(3-methoxypyridine-4-carbonyl)amino]-N,4,5,6-tetrahydrocyclopenta[c]thiophen-7-one 2-benzylsulfanyl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile 3-[(4-azidopyrimidin-2-yl)amino]-N-cyclopropylbenzenesulfonamide 1,2-diphenylhydrazine;ethane [4-(6-oxo-1H-pyridine-3-carbonyl)phenyl]methanesulfonic acid 3-azidooxy-2,5-diphenoxybenzenecarboximidamide 4-[(Z)-2-amino-1,2-diphenylethenyl]benzaldehyde;N-methylpropan-2-amine [3-methoxy-4-(2-morpholin-4-ylethoxy)phenyl]phosphane 3-(1H-imidazol-5-yl)-N-[4-(pyrrolidin-1-ylmethyl)phenyl]propanamide 2-[3-oxo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridazin-2-yl]benzonitrile N-azido-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboxamide (5Z)-2-imino-5-[(4-methoxyphenyl)methylidene]-1,3-thiazolidin-4-one N-[(Z)-1H-indol-6-ylmethylideneamino]-2-methoxybenzamide 2-[4-(2-methoxyethylamino)phenyl]-3H-benzimidazole-5-carbonitrile 2-[4-[(4,5-dihydro-1,3-thiazol-2-ylamino)methyl]phenyl]sulfanylethanimidamide;3-methylpentan-2-one (E)-2-[3-ethoxycarbonyl-6-fluoro-1-methyl-4-phenyl-4H-quinolin-7-ylidene]propanedioate 4-[(E)-2-chloroprop-1-enyl]quinoline (2S)-4-[3-(3,5-dimethylpyridin-4-yl)phenyl]-N,N'-dimethyl-1-(pyridin-2-ylmethylamino)butane-2-sulfonamide 3-[6-(cyclopropanecarbonylamino)-2H-pyridin-1-yl]-N,4-dimethyl-5-oxo-7,8-dihydrothieno[2,3-b]quinoline-6-carboxamide (2R,3R)-2-[(4-methylphenyl)methoxycarbonylamino]-3-[(5-nitrofuran-2-carbonyl)amino]butanoic acid 6-azidooxy-5,7,8-trimethylnaphthalene-1,4-dione 3-[2,5-bis(trifluoromethyl)phenyl]-1-hydroxy-N-methylpropan-2-imine (1S)-1'-[4,5-bis(ethenyl)-2-methoxypyridin-3-yl]spiro[1,3-dihydroindene-2,3'-pyrrolidine];1H-indazol-3-ol 4-[1-(3,3-dimethylbutanoyl)piperidine-4-carbonyl]-2-phenylpyridazin-3-one 4-[1-(4-chlorophenyl)ethylamino]-N,6-dimethylpyrimidine-2-carboxamide 2-(4,6-dichloroquinazolin-7-yl)oxybutanoic acid 1-(2,4-dinitrophenyl)butan-1-one 2-(1,3-benzothiazol-6-yl)-3-chloroquinoxaline 7-(4,6-diamino-1,3,5-triazin-2-yl)-7H-pyrrolo[2,3-d]pyrimidine-4,8-dione 5-bromo-4-cyclopropyl-2-[(1R)-1-cyclohexa-1,3-dien-1-ylethyl]-1H-pyrimidin-6-one (4-propan-2-yloxyphenyl)-[5-(trifluoromethyl)cyclohexa-1,3-dien-1-yl]iodanium (1R,2S)-N'-benzyl-2,3-dihydroxy-1H-indene-1-carbohydrazide (1E)-1-[(3,4-dichlorophenyl)methylidene]-5-phenyl-2H-indole 2-(hydroxymethyl)-N-[4-(trifluoromethoxy)phenyl]-6,7-dihydroquinoline-3-carboxamide N-[4,5-bis(ethenyl)-3-methoxyfuran-2-ylidene]hydroxylamine 1-methyl-4-(2-methylpropyl)-6-(6-piperazin-1-ylpyridin-3-yl)pyrazolo[4,3-c]pyridine 4-(2,5-difluorophenyl)-1H-pyrimidine-2,4-diamine 2-[5-[3,3-dimethyl-6-(2-oxopyrrolidin-1-yl)-1-propan-2-ylindol-2-ylidene]cyclohexa-1,4-dien-1-yl]sulfanylacetic acid N-[(3Z,5E)-1,2-dihydroxy-6-methylhepta-3,5-dien-3-yl]thiophene-2-carboxamide 4-[(Z)-[(Z)-[2-(3,5-dimethoxyphenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]hydrazinylidene]methyl]benzamide 6-methoxy-N-[1-(2,4,5-trifluorophenyl)ethyl]-7H-purin-8-amine (E)-1-[9-chloro-2-[[2-fluoro-5-(trifluoromethoxy)phenyl]methylamino]pyrimido[4,5-b]indol-8-yl]ethanol 2-ethyl-4-methylidenequinazolin-3-amine 4-[(4-aminophenyl)-[[(E)-3,7-dimethyloct-6-enoxy]-hydroxyboranyl]methylidene]cyclohexa-2,5-dien-1-one 5-(2,4-dimethylphenyl)-2H-pyridine-1-carboxylic acid ethene;2-N,5-dimethyl-4-N-[(1E)-3-(trifluoromethoxy)buta-1,3-dienyl]pyrimidine-2,4-diamine 1-butyl-3-ethenoxynaphthalene 1-cyclobutyl-3-[4-(2,6-dimethoxyphenyl)quinazolin-7-yl]urea 5-[2,4-dihydroxy-6-(3-methoxycyclobutyl)-3-oxophenyl]pentanamide 1-[3,4-bis(difluoromethoxy)phenyl]-N-[2-chloro-6-fluoro-4-iodo-5-(3,3,3-trifluoropropylamino)sulfanylphenyl]methanesulfinamide N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)-3-pyrazol-1-ylpropanamide 2-[2-ethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]acetamide 1,2-bis(benzylideneamino)guanidine 3-(2,4-difluorophenyl)-1,2-dimethylcyclobutane-1-carbonitrile [2-chloro-3-[(4-methylpiperazin-1-yl)amino]phenyl]azanium 1-[2-(3,5-dimethylphenyl)ethenoxy]-6-methylnaphthalene N-[1-(2,4-difluorophenyl)ethenyl]-3-methoxypropan-1-amine 1-[[3-(4-chlorophenoxy)phenyl]methyl]azetidine (Z,2S)-N-[(6-chloropyridin-3-yl)methoxy]propan-2-imine;methanol 6-[[2-cyclopropylethyl(methyl)amino]methyl]-1-phenyl-5H-pyrazolo[3,4-d]pyrimidin-4-one 1-azidooxy-2,5,6-trichloro-3-nitrobenzene (2S)-4,7,8-trimethyl-1-phenylnonane-2-thiol 1-phenylundecane-2,7-dione 6-methyl-4-[(2R)-pentan-2-yl]pyridine-3-carboxylic acid 6-N,7-dimethylnaphthalene-1,6-disulfonamide;methanamine 3-(4-chlorophenyl)-6,11-dioxobenzo[c]chromene-2-carboxamide (5Z)-2-[4-chloro-3-(trifluoromethyl)phenyl]imino-5-[[1,6-diethyl-4-(4-fluorophenyl)benzimidazol-2-yl]methylidene]-1,3-thiazolidin-4-one 4-(5-fluorocyclohexa-2,4-dien-1-yl)-5-methoxycarbonyl-2-[4-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxylic acid 4-amino-N-[(1S)-1-phenylethyl]quinazoline-7-carboxamide;cyclohexanol 2-[(5S)-1,4-diphenyl-6,7-dihydroindazol-3-yl]aniline 2-[5-(2,3-dimethylimidazol-4-yl)-1H-indazol-3-yl]-7-piperidin-1-yl-4H-imidazo[1,5-a]pyrazine N-(2,3-dihydronaphthalene-1-carbothioyl)-3,4,5-trimethoxybenzamide N-ethyl-4-(2,3,5,6-tetrachlorophenyl)cyclohexane-1-carboxamide 2-amino-3,4,5-trichloro-6-methoxybenzoate N-(4,5-dimethyl-2-phenyldiazenylphenyl)-1H-indole-3-carboxamide 2-azidooxy-6-chloro-1,3-benzoxazole 1,4-diamino-6-fluoro-7-[(2R)-3,3,5,5-tetramethyloxolan-2-yl]oxyisoquinoline-3-carboxylic acid (2S)-N-[4-[2-(3,5-dimethoxyanilino)pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamide 4-[1,1-bis(2-hydroxyphenyl)ethyl]phenolate;pentan-3-ylidenezirconium(4+) 2-(6-methylpyridin-3-yl)oxy-5-(trifluoromethyl)phenol 2-hydroxy-N,N'-dimethyl-4-[[(1S)-3-oxocyclohexyl]amino]benzohydrazide 3-[4-(2,4-dihydroxyphenyl)butyl]-7-oxa-1,3-diazaspiro[5.6]dodecan-2-one 2-[2,4-bis(trifluoromethyl)phenyl]-3-[3-(trifluoromethoxy)pyridin-2-yl]piperidine-1-carboxylic acid (4S)-3-[5-(3,4,5-trimethoxyphenyl)furan-2-carbonyl]imidazolidine-4-carboxylic acid 5-ethyl-6-phenylindolo[2,3-c]quinoline 4-[2-[(3-methylphenyl)sulfonylamino]acetyl]morpholine-3-carboxamide N-[3-[6-[(dimethylamino)methyl]-2H-pyrimidine-1-carbonyl]phenyl]pyridine-4-carboxamide N-[2-methyl-4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]propanamide 2-amino-9-[(5R)-6,7,8,9-tetrahydro-5H-pyrido[3,4-b]azepin-5-yl]-1H-purin-6-one 7-ethyl-1,2-dimethoxy-3-phenyl-5H-pyrido[2,3-d]pyrimidine-4,6-dione N-butanoyl-2-bromo-N-[4-(thiophen-2-ylsulfamoyl)phenyl]benzamide 1-azidooxy-2,3-dimethylbenzo[g]indole 2-(aminomethyl)-6,7-bis[4-chloro-3-(trifluoromethyl)phenoxy]-1H-quinoline-2-carboxylic acid 5-[(3,5-dibromophenyl)methyl]-4-imino-1-propan-2-ylimidazolidin-2-one N'-hydroxy-5-(2,4,6-trimethylphenoxy)pyridine-2-carboximidamide 5-tert-butyl-N-(4,5-difluorocyclohepta-1,3,6-trien-1-yl)thiophene-2-carboxamide [3-hydroxy-3-(triazol-1-ylmethyl)piperidin-1-yl]-(2-methoxypyridin-4-yl)methanone 2-(1,3-benzodioxol-5-yl)-4-hydroxy-5-[3-oxo-7-[5-(trifluoromethoxy)-6,7-dihydro-1H-pyrrolo[2,3-b]pyridin-3-yl]isoindol-1-ylidene]cyclohexane-1,3-dione 2,2-dimethyl-1-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one;ethane 3-cyclohexyl-6-[(4R)-1-ethylpiperidin-4-yl]pyridine;2,2,5,7,8-pentamethyl-3H-chromen-4-one (2S)-2-acetamido-3,3-dimethylbutanamide;N-[4-chloro-2-[3-(difluoromethyl)piperidine-1-carbonyl]phenyl]methanesulfonamide 7-[6-(2,3-dihydro-1H-pyrrolo[1,2-a]indole-7-carbonyl)pyridazin-4-yl]-7-azaspiro[3.5]nonan-8-one 6-[(2R)-1,3-benzoxazol-2-yl]-3-(4-hydroxyphenyl)thieno[3,2-d]pyrimidin-4-one 4-(6,7-dimethoxyquinolin-4-yl)oxy-3,5-diethyl-N-phenylbenzamide 6-(4-fluorophenyl)-7-hydroxypyrrolo[3,4-g]quinoxaline-5,8-dione ethane;1-(3-methylbutanoyl)-5-phenylpyrrolidine-2,4-dione 2-N,4-N-dimethyl-6-N-[1-(oxan-3-yl)pyrazol-4-yl]pyrimidine-2,4,6-triamine 4-[(3S,5R)-3,4,5-trimethylcyclohexyl]quinoline 3-chloro-2-fluorobenzaldehyde;(6R)-7-methoxy-5,5,8a-trimethyl-4a,6-dihydrocyclohepta[d][1,3]thiazol-2-amine N-[4-[1-(methoxyamino)ethenyl]phenyl]cycloheptanamine;1-methyl-3,5-bis(trifluoromethyl)benzene 1-bromo-4,5-ditert-butyl-2-fluorobenzene 3-(dimethylamino)-N,N-diethylpropanamide;ethane;1-[4-(9H-xanthen-9-ylsulfamoylamino)butyl]piperidine N-[4-methoxy-5-(3-oxomorpholine-4-carbonyl)-2,3-dihydroinden-1-ylidene]benzamide 6-[4-(2,6-dichlorophenyl)piperazine-1-carbonyl]-N-methylpyridine-3-sulfonamide;2,2,2-trifluoroacetic acid N-[4-(methylamino)phenyl]-2-naphthalen-1-ylcyclopropane-1-carboxamide 3-cyclopropyl-N-[(2S)-1,1,1-trifluorobutan-2-yl]pyridine-2-carboxamide 2-azido-1-(3,5-dibromopyridin-2-yl)ethanone N-[4-[(3,6-dimethylthieno[2,3-b]pyridin-4-yl)amino]butyl]-1,5-bis(phenylsulfanyl)pentane-3-sulfinamide (4aS,8aR)-6-[(3R)-3-cyclopropylpiperidine-1-carbonyl]-4a-hydroxy-5,7,8,8a,9,10-hexahydrophenanthrene-2-carbonitrile;hydrochloride N-[3-fluoro-5-(2-methylphenyl)pyridin-4-yl]-N'-propan-2-ylmethanimidamide (5Z)-2-(3,4-dichlorophenyl)imino-5-[(4-morpholin-4-ylphenyl)methylidene]-1,3-thiazolidin-4-one N-[(5S)-6-(5-chloro-2,4-difluorophenyl)-3-bicyclo[3.1.0]hexanyl]isoquinoline-7-carboxamide 1-phenylsulfanylpiperazine;hydrochloride 6-[(4-fluorophenyl)methyl]-2-(trichloromethyl)-7H-imidazo[5,1-c][1,2,4]triazole 6-(8,9,10,11-tetrahydrobenzo[c]phenanthridin-7-yl)carbazole-2,5-dicarbonitrile 4-(2-azidoethyl)-1-(4,5-dimethoxy-1H-benzimidazol-2-yl)triazole (Z)-3,3,3-trifluoro-1-[4-[(E)-prop-1-enyl]phenyl]-2-(1H-pyrazolo[3,4-d]pyrimidin-6-yloxy)prop-1-en-1-amine 1-[4-(2,6-dipyridin-3-ylpyridine-4-carbonyl)piperazin-1-yl]ethanone;formic acid 2,6-dibutoxybenzenethiol 4-[3,5-dichloro-4-(trifluoromethyl)phenyl]sulfanylbenzonitrile;ethane 1-butyl-2,4-dihydroxy-6-oxo-5H-pyrrolo[3,4-c]pyrrole-3-carboxylic acid 1-(8-bromooctyl)-2,3,4,5,6,7-hexahydro-1H-indene 2,7-ditert-butylimidazo[1,2-a]pyridine 3-(4,7-difluorocyclohepta-1,3,5-trien-1-yl)-2H-pyrido[3,2-b][1,4]oxazine N-[2,3-dichloro-4-(trifluoromethyl)phenyl]-3,5-diethoxybenzamide 4-fluoro-2-[3-[(6-methylpyridine-2-carbonyl)amino]pyrazol-1-yl]benzoic acid N-(1H-imidazol-2-yl)-6,7-dimethoxynaphthalene-2-carboxamide 5-[4-(benzylamino)phenyl]imidazolidine-2,4-dione (3S)-5-(3,4-dihydroxyphenyl)-N'-[2-(4-fluoropiperidin-1-yl)ethyl]-N-methylidene-3-phenyl-3,4-dihydropyrazole-2-carboximidamide 2-[2-(2,6-dichlorophenyl)ethyl]aniline (2R)-N,3-dihydroxy-2-[1H-indole-7-carbonyl-[(E)-4-morpholin-4-ylbut-2-enoyl]amino]propanamide (2R)-4-[(2S,3S,5R)-3,5-dihydroxyoxan-2-yl]oxy-1,1-bis(4-methylphenyl)butane-1,2-diol (2R)-3-amino-N-[(5-fluoropyridin-2-yl)methyl]-2-hydroxypropanamide;dihydrochloride (4-amino-3,5-dichloropyridin-2-yl)-[(6S)-1,2,6-trimethylpiperidin-4-yl]carbamic acid 2-[2-(3-methoxyphenyl)ethyl]-1H-pyrrole 3-[5-(5-chloro-2,4-difluorophenyl)-1H-imidazol-2-yl]pentanoic acid 2-[4,5-dimethoxy-2-[(3-methyl-1,2-oxazol-5-yl)carbamoyl]phenyl]acetic acid 1-[(3-chlorophenyl)methyl]-5-iodopyrazole 2,4-ditert-butyl-6-[(2E)-2-[[5-[(3,3,4,7,8-pentamethyl-1-bicyclo[4.2.0]octa-1,3,5-trienyl)sulfanylmethyl]furan-2-yl]methylidene]hydrazinyl]phenol 5-methyl-2,3,4,9-tetrahydro-1H-xanthene 4-(3-aminobutyl)-2,6-bis[[dimethylphosphoryl(phenyl)methylidene]amino]phenol [2-(1,3-benzodioxol-5-yloxy)-6-methylpyridin-4-yl]-[4-[4-[(E)-pent-3-en-2-ylideneamino]phenyl]piperazin-1-yl]methanone 4-chloro-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine-7-carboxylic acid 1-[(1S,3S)-3-methoxycyclopentyl]-N-[(2-phenylpyrimidin-5-yl)methyl]methanamine (1-ethylcyclobutanecarbonyl)-[(2S,4R)-4-fluoro-2-propan-2-yloxy-5-pyridin-3-ylsulfanyloxypyrrolidin-1-yl]methanone 3-fluoro-5-[7-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]sulfanylbenzonitrile 2-[3,5-dibromo-4-(2-hydroxypropoxy)phenyl]ethanol N-[5-[3-(4-pyridin-2-yl-1H-pyrrolo[2,3-b]pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]pyridin-3-yl]benzamide 4-[2-(dimethylamino)ethoxy]-6-(4,5-dihydropyren-1-ylsulfanyl)pyridine-3-carbonitrile (E)-2-[6-[2-(4-fluorophenyl)ethynyl]imidazo[1,2-b]pyridazin-2-yl]-3-(methylamino)prop-2-enamide 4-(1H-indol-2-ylmethoxy)-N,5-dimethylpyrimidin-2-amine 2-[4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxyphenoxy]propanamide 3-(4-nitrophenyl)sulfanyl-4,5-dihydro-1H-pyrrolo[2,3-b]pyridine 4-[2-(1H-indol-3-yl)propyl]phenol 2-[N-cyclohexyl-4-(quinoxalin-2-ylsulfamoyl)anilino]acetamide (4R)-3-[3,5-bis(phenylmethoxy)benzoyl]-1-(furan-2-ylmethyl)pyrrolidine-2,4-dione 2-azido-N'-hydroxy-5,6-dimethylpyrimidine-4-carboximidamide (2R)-1-[6-(2,5-dimethylpyrrole-1-carbonyl)pyridin-3-yl]piperidine-2-carboxamide 6-fluoro-N-(4-fluorophenyl)-1-methyl-N'-[(E)-[[2-(methylideneamino)pyrimidin-5-yl]-pyridin-3-ylmethylidene]amino]benzimidazole-4-carboximidamide 2-(1,3-benzoxazol-5-ylmethyl)-4-pyridin-4-yl-2H-furan-5-one 1-[4-(dimethylamino)phenyl]sulfonyl-2,5-diethyl-3H-pyrazole-5-carboxylic acid 2-[(1R)-1-[[7-fluoro-3-(2-methylpropyl)-1,2-dihydroquinolin-4-yl]amino]ethyl]pyridine-4-carboxamide 4-[4-(2,4-difluorophenyl)-6-fluoropyridin-3-yl]-1-(oxan-4-yl)azepane 3-(9H-fluoren-1-yl)-2,4-dimethylpentane-2-thiol (7S)-2-methylsulfanyl-5,6,7,8-tetrahydropyrimido[4,5-d]pyrimidine 1-[(2R)-4-benzyl-2-ethylpiperazin-1-yl]-2,3-dihydroxypropan-1-one (2E,4Z)-3-[3-methoxy-4-[1-(2-phenoxyacetyl)pyrrolidin-3-yl]oxyphenyl]hexa-2,4-dienoic acid N-[1-(3,5-difluorophenyl)ethyl]-5-methoxy-2-nitroaniline 2-[(E)-[5-amino-4-(3,4,5-trimethoxyphenyl)triazol-1-yl]iminomethyl]-6-fluorophenol 3,4-diethoxycyclohepta[b]naphthalene N-[(2E,4Z)-5-chlorohexa-2,4-dienyl]-5-(1H-pyrazol-4-yl)thiophene-3-carboxamide 2-(disulfanyl)-5,7-dihydrobenzo[d][2]benzazepine ethane;[3-methyl-4-(1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]hydrazine N-[2-(1H-benzimidazole-4-carbonyl)phenyl]-3,4-dichlorobenzamide 2-[(Z)-3-iminoprop-1-enyl]pyridine-4,5-dicarboxylic acid 4-(2,1,3-benzothiadiazol-5-ylamino)-6-[3-[3-methyl-5-[[2-morpholin-4-yl-4-(trifluoromethyl)phenyl]carbamoyl]pyrazol-1-yl]anilino]pyridine-3-carboxamide 1-[5,6-difluoro-4-(2,2,2-trifluoroethoxy)pyridin-3-yl]-N-methylmethanimine 3-amino-5-(5,6-dichloropyridin-2-yl)thiophene-2-carboxamide N-[2-(6-bromo-5-hydroxyimidazo[1,2-a]pyridin-3-yl)ethynyl]benzenesulfonamide;methanol (6R)-2,6-dimethyl-4-[6-(trifluoromethoxy)-1H-benzimidazole-5-carbonyl]piperazine-1-carboxylic acid 3,7-bis(4-propan-2-ylphenyl)phenanthrene 4-azido-3,5-dichloroquinoline 2-(ethylamino)-1-[5-(3-ethynylphenyl)pentyl]-N,4-dimethyl-6-oxopyridine-3-carboxamide 2-[[4-methyl-6-(trifluoromethoxy)pyrimidine-5-carbonyl]amino]-2-(3,4,5-trimethoxyphenyl)acetic acid 6-hydroxy-3-[(4-methoxyphenyl)methyl]-2H-indazole-5-carboxylic acid 3-(2,4-difluorophenyl)-1-iodopyrazolo[3,4-c]pyridine 1-(4-propan-2-ylphenyl)sulfanylpiperidine 2,4-dichloro-N-(3-methylbutyl)pyrimidine-5-carboxamide (4-ethyl-3,5-dimethoxyphenyl)-[2-(4-fluorophenyl)pyrrolidin-1-yl]methanone 5-(3,5-difluorophenyl)-1H-indazole 1-[5-bromo-4-fluoro-2-(2-methoxyethylamino)phenyl]-3-(3,5-dichloropyridin-4-yl)urea N-(1,3-dimethylpyrazol-4-yl)-6,7-dihydro-5H-cyclopenta[d]pyrimidine-4-carboxamide 4-[(3,5-dichlorophenyl)methyl]pyrimidine 3-[[5-bromo-1-(2,4,6-trichlorophenyl)sulfanylindole-3-carbonyl]amino]propanoic acid 2-[3,5-bis(trifluoromethyl)phenoxy]-N-[[4-chloro-5-[difluoro(iodo)methoxy]-2-methoxyphenyl]carbamothioylamino]acetamide 2-azido-5-cyclobutyloxy-4-propan-2-ylaniline 3-[1-(4-azidobutanoyl)piperidin-4-yl]oxy-5,6,7,8-tetrahydronaphthalene-2-carboxylic acid 2-[(5Z)-5-[(4,6-dimethyl-2-oxochromen-3-yl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid 6-[2,2-diethoxyethyl(methoxycarbonyl)amino]-4-hydroxynaphthalene-2-sulfonic acid 2-[3,5-difluoro-4-(3,3,3-trifluoropropylsulfanyl)phenyl]-6,7-dihydro-5H-pyrrolo[1,2-c]imidazole 4-(2,6-dihydroxyphenyl)-2H-pyrimidine-1-carboxylic acid (2S,3R)-5,8-diamino-2-[[1,3-bis(2-chlorophenyl)propan-2-ylcarbamoylamino]methylidene]octanoic acid 1-[(2,4-difluorophenyl)methyl]-3-[1-[5-(3-isocyanophenyl)pyrimidine-2-carbonyl]piperidin-4-yl]-8-[(4-methoxyphenyl)methyl]purine-2,6-dione 4-[3-[2-(2,5-dihydroxycyclohexa-1,5-dien-1-yl)-1-ethylbenzimidazole-5-carbonyl]phenyl]benzoic acid 5-(5-methoxycarbonylpyridin-3-yl)-2-oxopentanoic acid 3-(azidomethyl)-1,2,5-trifluoro-4-nitrobenzene 4-[2-(azetidin-1-yl)ethoxy]-3,5-dichloroaniline (3R,6S)-1-[4-cyano-2,5-difluoro-3-(trifluoromethyl)phenyl]-N-[(2,3-dimethylphenyl)methyl]-6-ethoxypiperidine-3-carboxamide 1-(4-tert-butylphenyl)-2-[3-(2,4-dimethoxyphenyl)propanoylamino]pentane-1-sulfinamide (2S)-1-[(3R,4R)-6-chloro-3-hydroxy-3,4-dihydroisochromene-1-carbonyl]-N-[(2E,4Z)-6-fluorohexa-2,4-dienyl]pyrrolidine-2-carboxamide N-[2-(dimethylamino)ethyl]-3-methylpyridine-4-carboxamide 4-(9H-fluoren-3-yl)-2,6-difluoroaniline 4-(6,7-dimethoxyquinolin-4-yl)oxyaniline (2R)-2-azido-N,4,5-trimethyl-1-phenylpentan-3-amine 3-[2,4,6-tri(propan-2-yl)phenyl]-1H-imidazol-3-ium;bromide 3-(4-ethenylphenyl)-N,2-dimethylpropanamide 6-chloro-7-[(2R)-4,4-difluoro-2-methylpyrrolidin-1-yl]sulfonyl-2H-isoquinolin-1-one 4-N-(2-bromo-3,6-difluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine 4-[(Z)-3-aminoprop-2-enyl]-8-fluoro-1,2,5,10b-tetrahydroisochromeno[3,4-a]indol-7-ol (3-pyridin-4-ylpiperidin-1-yl)-(3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]isoquinolin-7-yl)methanone;hydrochloride N-[4-(6,7-dimethoxyquinolin-3-yl)oxypyridin-2-yl]-2,3,4,5-tetrahydro-1H-azulene-1-carboxamide 4-[(2E,4Z)-1-ethenyliminopenta-2,4-dien-3-yl]-N-hexan-3-ylaniline 2-chloro-N'-[4-(7,8-dimethylimidazo[1,5-a]pyridin-6-yl)pyrimidin-2-yl]ethanimidamide (2R,3S)-4-[bis(dimethylcarbamoyl)amino]-N'-[5-chloro-6-(1,2-dihydropyridin-5-ylamino)pyrimidin-4-yl]-2,3-dihydroxybutanimidamide 5-[1-(3,4-difluorophenyl)ethylamino]imidazo[1,2-c]pyrimidine-8-carboxamide 3-[[4-(2,6-dichlorophenyl)-5-(2H-tetrazol-5-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-N'-hydroxybenzenecarboximidamide 2-amino-9-[(2S,4R)-5-(hydroxymethyl)-3,4-dimethylideneoxolan-2-yl]-8-[(4-morpholin-4-ylphenyl)methoxy]-1H-purin-6-one 3-[(6,8-dichlorospiro[chromene-2,4'-piperidine]-1'-yl)methyl]-7-fluoroindazole 1-[3,4-di(propan-2-yloxy)phenyl]propane-1,3-dione N-benzyl-3,4,6-trimethyl-1-phenylsulfanylnaphthalen-2-amine (3R)-3,4-bis(ethenyl)-7,8-dimethoxy-2-oxo-1,3,5,9b-tetrahydroisochromeno[3,4-c]pyridine-10-carbonitrile N-[(5,7-dimethylimidazo[1,2-a]pyridin-2-yl)methyl]-4-methoxybenzamide 3-[3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-2-ethanimidoylbut-3-enamide 2-amino-4-(3,5-dimethyl-1,2-oxazol-4-yl)benzenethiol 3-(1,1-difluoroethyl)-N'-hydroxypyridine-2-carboximidamide 5-(1,1-difluoroethyl)-N'-hydroxypyridine-2-carboximidamide N-[4-(N'-hydroxycarbamimidoyl)-1H-pyrazol-5-yl]cyclohexanecarboxamide 2-[3-[4-(2,6-difluorophenoxy)piperidin-1-yl]sulfonylphenyl]acetic acid N-[5-(3,4-dihydropyridin-6-yl)-2-oxo-1H-pyridin-3-yl]cyclohexanecarboxamide 5-(azidomethyl)-7-[1-[2,4-bis(trifluoromethoxy)phenyl]pyrazole-3-carbonyl]-N'-hydroxy-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-1-carboximidamide 3-[2-(cyclopropylmethylamino)pyridin-4-yl]-5-[1-(2,3-difluorophenyl)-3,5-dimethylpyrazol-4-yl]pyridin-2-amine ethane;methanol;4-[2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridine-2-carbonylamino)thieno[3,2-b]thiophen-5-yl]benzoic acid 1-(azetidin-3-ylmethoxy)-2,4-dichlorobenzene 1-[4-[3,5-dichloro-2-(1H-pyrazol-4-yl)indole-1-carbonyl]piperazin-1-yl]propan-1-one 2-[[1,3-bis(difluoromethyl)pyrazole-4-carbonyl]amino]-5-(methoxycarbonylamino)pentanoic acid 3-amino-4-cyano-5-[2,6-difluoro-3-(trifluoromethyl)phenyl]-1H-pyrrole-2-carboxamide N-[2-(3,5-difluorophenyl)ethyl]-4-oxospiro[6H-pyrazolo[1,5-a]pyrimidine-7,1'-cyclopentane]-5-carboxamide 6-[4-(2,3-dimethylphenyl)butanoyl]oxyhexanoic acid [4-[1-methyl-5-[4-(6-methylsulfanylpyridine-2-carbonyl)piperidine-1-carbonyl]pyrazol-3-yl]phenyl]-[(2R,4S)-4-methyloxolan-2-yl]methanone 1-[4-(1,3-dimethylpyrazol-4-yl)phenyl]piperazine;ethane 3-azido-2,6-dibromo-N-cyclobutylaniline [3-amino-2-fluoro-5-(1H-pyrazol-4-yl)phenyl]-[2-(2,6-diazaspiro[3.3]heptan-2-ylmethyl)pyrrolidin-1-yl]methanone 7-(4-chlorophenyl)-8-fluoro-3H-imidazo[1,5-a]pyridine 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]-1-phenylethanone 4-(benzenesulfonylmethyl)-5-bromo-2H-phthalazin-1-one 7-chloro-4-(2,5-difluorophenyl)-6-methyl-N-propan-2-yl-1,2,3,4-tetrahydroquinoline-3-carboxamide N'-[(E)-2-aminobut-1-enyl]-4-[2-chloro-3-(4,5,6,7-tetrahydro-1H-indazol-5-ylamino)phenyl]pyridine-2-carboximidamide 5-[2,3-dihydroxypropyl(1,3-thiazol-5-yl)amino]-1H-pyrimidine-2,4-dione (2S,4R)-1-[3-bromo-5-fluoro-6-methoxy-2-(piperidine-1-carboximidoyl)phenyl]sulfonyl-N,4-dihydroxypyrrolidine-2-carboxamide N-azido-1,3,5-trimethylpyrazolo[4,3-d]pyrimidine-7-carboxamide 5-[(2,4-dihydroxyphenyl)methyl]-1,3,7-trifluoroheptane-2,6-dione (3S)-1'-benzyl-2,2-dimethylspiro[2H-furo[2,3-g]chromene-3,4'-piperidine] 2,3-ditert-butylquinoline-6,8-dicarboxylate 2-[(3-methylthiophene-2-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid 3-[(3S)-3-methylmorpholin-4-yl]-1H-quinolin-2-one 2-[4,5-dimethyl-N-(1,3-thiazol-5-yl)-2-phenyldiazenylanilino]acetonitrile 4-[4-(6,7-dihydrodibenzothiophen-2-yl)phenyl]-6-oxo-2-sulfanylidene-1,3-diazinane-5-carbonitrile [(2S,3R)-4-benzoyl-5-fluorospiro[2H-indole-3,1'-cyclopentane]-1-yl]carbamic acid ethane;N-[2-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-5-yl]-N'-phenylsulfanylethane-1,2-diamine 3-(5,6-diethoxypyridin-2-yl)propanoic acid 1-(4,5-dimethoxy-2-methylphenyl)ethanone 2-(2-chlorophenyl)-N-[3-methyl-5-[2-[4-(trifluoromethoxy)anilino]acetyl]indazol-1-yl]propanamide N-[4-(2,5-dimethylphenyl)pyrimidin-2-yl]nitramide 1-[3-[7-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]piperidin-1-yl]-2-methoxyethanone;2,2,2-trifluoroacetic acid (2R,4S)-5-amino-4-[(4-chlorophenyl)methoxy]pentane-1,2,3,4-tetrol 2-[2-hydroxyethyl-(1,3-thiazol-5-yl)amino]acetonitrile 4-(3,5-dimethylbenzoyl)piperazine-1-carboxylic acid 2-[2,2-dimethoxyethyl(1-phenylpropyl)amino]octanoic acid 5-ethoxycarbonyl-4-[3-oxo-1'-(pyridine-2-carbonyl)spiro[benzo[f]chromene-4,4'-piperidine]-2-yl]pentanoic acid 1-chloro-3-[2,4,6-trimethyl-N-(2-oxopropyl)anilino]butan-2-one 6-tert-butyl-3-hydroxy-2,4,5,7-tetramethylpyrrolo[2,3-c]pyridazine-1,3-dione 5-[5-(cyclohexyloxymethyl)pyridin-3-yl]-N-(6-fluoro-1,2,3,4-tetrahydronaphthalen-2-yl)-1H-indazole-3-carboxamide N-[2-(3,5-dichloropyridine-4-carbonyl)-1,3-dihydroisoindol-5-yl]-3-fluoropyridine-4-carboxamide N-[(2R,3S)-6-oxo-2-phenylpiperidin-3-yl]-5-[4-(trifluoromethoxy)phenyl]furan-2-carboxamide 3-[6-(1,2-dihydropyrimidin-5-yl)pyridin-3-yl]propanenitrile N-[6-(3,4-dimethoxyphenyl)isoquinolin-8-yl]formamide;2-ethoxyethanamine 3-fluoro-4-[2-[(3S)-3-methylpyrrolidine-1-carbonyl]thieno[3,2-b]pyridin-7-yl]oxybenzonitrile 1-(3-azidophenyl)-N-[4,5-bis(ethoxyphosphorylmethoxy)-2-fluorophenyl]methanesulfonamide 2-[(3,4-dichlorophenyl)methyl]-6-[4-[[ethyl-(3-methoxypropyl)amino]methyl]piperidin-1-yl]pyridazin-3-one 2-[(2E,4Z)-hepta-2,4-dien-3-yl]-N-methoxy-5-phenyl-1,2-oxazol-3-imine 1,2-difluorobenzene;1-[(4S)-4-ethylimidazolidine-1-carbonyl]pyrazole-3-carboxylic acid 1-(4,6-difluoroquinolin-3-yl)ethanethione [2-chloro-5-(trifluoromethyl)phenyl]boronic acid 5-fluoro-4,7-dimethyl-1H-indole;4-[3-(2-oxoethyl)pyrrolidin-1-yl]sulfonylbenzonitrile 5-(2,3-difluoro-4-methoxyphenyl)imidazolidine-2,4-dione 3-[5-[(dimethylamino)methyl]pyridin-2-yl]-N-propan-2-yl-1H-pyrrolo[3,4-c]pyridin-6-amine 1-(4,6-dimethylpyrimidin-2-yl)-5-phenylspiro[3H-1,2-oxazole-4,9'-xanthene] 3-[[5-methyl-7-(3-methylbut-2-enoxy)naphthalen-1-yl]oxymethyl]cyclopentan-1-ol ethane;1-[2-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)amino]ethoxy]-3H-2,1-benzoxaborole 3-(4,6-dimethylquinoline-2-carbonyl)oxypropane-1-sulfonate N-(4,6-dimethylpyrimidin-2-yl)-4-[1,3-thiazol-5-yl(pyridin-2-yl)amino]benzenesulfonamide 3-[2-(aminomethyl)-5-azidophenyl]-4,6-dichlorophenol 2-[[6-fluoro-3-(5H-imidazo[5,1-a]isoindol-5-yl)cyclohepta-1,4,6-trien-1-yl]methylamino]ethanol 2-(N-ethylsulfonyl-4-propan-2-ylanilino)acetamide 3-(4,6-diphenyl-1,2,3,5,6,7-hexahydropyrrolizin-8-yl)-N-[(3S)-pyrrolidin-3-yl]benzamide 1,2-dichlorobenzene;6-(4-methoxyphenyl)-5-N,5-N-dimethyl-2-N-[(E)-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]methylideneamino]pyrimidine-2,5-diamine 2-hydroxyimino-5-[(4S)-3,3,7-trimethyl-6,8-dihydro-5H-naphthalen-2-yl]benzoic acid 2-(4-methylpyrazol-1-yl)-N-[5-(trifluoromethyl)pyridin-2-yl]acetamide (4-cyclopropylphenyl)-[4-hydroxy-3-(1H-pyrazol-5-ylmethyl)piperazin-1-yl]methanone 2-bromo-6,7-dichloro-4H-[1]benzothiolo[3,2-d]pyrimidine 4-fluoro-5,6-dimethyl-3-phenylthieno[2,3-b]pyridine (3,4-dihydroxypiperidin-1-yl)-[4-[2-[6-(4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-5-ylidene]ethyl]piperazin-1-yl]methanone N-azido-5-ethylnaphthalene-2-sulfonamide 5-(2-methylsulfonylpyrimidin-4-yl)pyrrolo[3,2-b]pyridine 1-(2-cyclopropylethynyl)-3-(1,1,4,4,5,6-hexamethylpyridin-1-ium-2-yl)benzo[f]chromene 1-[7-azido-2,6-dichloro-4-(trifluoromethyl)benzimidazol-1-yl]propan-2-ol ethane;5-methylfuran-2-sulfonamide 1-azidooxy-3,4-dimethyl-9H-fluorene N-[1-(6,7-dimethoxyquinolin-4-yl)piperidin-3-yl]-N-(oxan-2-yloxy)formamide 2-[(4S)-3,3-difluoropiperidin-4-yl]oxy-5-[2-methyl-3-[8-methyl-7-(1-methylpiperidin-4-yl)pyrido[3,4-d]pyrimidin-2-yl]phenyl]benzonitrile 4-[(3,5-dimethylpiperidin-1-yl)amino]-6-[(E)-2-[5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]ethenyl]quinazolin-8-ol (2S,3R)-4-[2-[2-(3H-azepin-7-ylmethoxy)phenyl]imidazol-1-yl]-1-(4-chlorophenoxy)butan-2-ol 3-[1,2-difluoro-4-(7H-purin-6-ylamino)butan-2-yl]-N'-methylbenzenecarboximidamide ethane;3-(4-methylphenyl)sulfanyl-2H-thiochromene [4-[3-(2,5-dichloropyrimidin-4-yl)imidazo[1,2-a]pyrazin-6-yl]piperazin-1-yl]-[6-(trifluoromethyl)pyridin-3-yl]methanone 1-[(3,4-dichlorophenyl)methylamino]-3-decylthiourea (1-cyclobutylpiperidin-3-yl)-[6-hydroxy-2,5-bis(4-methoxyphenyl)imidazo[2,1-b][1,3]benzothiazol-7-yl]methanone 1-azido-3-(2,6-dimethylphenoxy)piperidine 6-chloro-3-[5-[(4-methylphenyl)diazenyl]furan-2-yl]chromen-2-one 2-cyclohexyloxy-5-[1-(7H-purin-6-ylamino)ethyl]-3-propan-2-ylbenzimidazole-4-carbonitrile 5-[3-hydroxy-4-(3,3,3-trifluoropropyl)pyrrolidine-1-carbonyl]pyridine-2-carboxylic acid 5-[1,2,3-trimethyl-4-[(6R)-6-(3-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-ium-4-yl]pyrrol-3-yl]thiophene-2-carbonitrile 4-[2-(6,7-dihydronaphthalen-1-yl)ethyl]phenol (3R,4S)-1-[2-(3-methylpyrazol-1-yl)ethyl]-4-[(5-propan-2-yl-1H-pyrazole-4-carbonyl)amino]pyrrolidine-3-carboxylic acid 2-[4-[[3-fluoro-5-(trifluoromethoxy)phenyl]carbamoylamino]phenoxy]acetamide 3-butyl-N-methylaniline;4-[2,5-di(propan-2-yl)pyrrol-1-id-3-yl]benzaldehyde 3-(3,4,5,6-tetrafluoropyridine-2-carbonyl)piperidine-1-carboxylic acid 5-azidooxy-1-bromoisoquinoline 6-[(E)-but-2-en-2-yl]-7-methoxy-3-[6-(trifluoromethyl)pyridin-3-yl]quinoline 2-[[(3R,4S)-1-methyl-3-phenylpiperidin-4-yl]amino]benzonitrile (2S)-4,7-difluoro-2-methyl-N-(1H-pyrrolo[3,2-c]pyridin-6-ylmethyl)heptanamide;hydrochloride 4-azido-5-chloro-2-(1,3-dioxolan-2-yl)pyrimidine (Z)-3-(1H-indol-4-ylmethylideneamino)-3-(4-nitrophenyl)prop-2-enenitrile 1-[2-chloro-4-(dimethylamino)phenyl]butane-1,3-dione 2-[(3-methylphenyl)methyl]-4,5-dihydroindazole 6-(2,3-dimethoxyphenyl)-8-[4-fluoro-5-(piperazin-1-ylmethyl)pyridin-3-yl]pyrido[3,4-d]pyrimidine N-[5-(5,6-dichloro-1H-indole-2-carbonyl)pyridin-2-yl]propanamide N-[(2S)-1-[amino-[(3S,4R)-1-benzylsulfonyl-4-methoxypyrrolidin-3-yl]amino]-1-oxopropan-2-yl]-5-chloro-4-(methylideneamino)thiophene-2-carboxamide 2-[(E)-4-methylpentylideneamino]isoindole-1,3-dione [2-[(3-ethylphenyl)methoxy]phenyl]hydrazine N-[(2S,3R)-4-[(5-ethylsulfonylpyridine-2-carbonyl)amino]-3-hydroxy-6-phenyl-1-[3-(trifluoromethoxy)anilino]hexan-2-yl]piperidine-2-carboxamide 2,3-dichloro-4-[6-(chloromethyl)pyridine-3-carbonyl]oxybenzoic acid 2-(cyclopentylmethoxy)benzenethiol 2-amino-N-[4-(3,5-dimethyl-1H-pyrazol-4-yl)phenyl]pyridine-4-carboxamide;hydrochloride [4-methoxycarbonyl-2,5-bis(trifluoromethyl)phenyl]boronic acid 1-[3,5-bis(4-fluorophenyl)-2-methylimidazol-4-yl]ethanone 3-[[2-fluoro-6-(trifluoromethyl)phenyl]carbamoylamino]naphthalene-1,7-disulfonic acid 3-azidooxy-7-bromo-6-methyl-5H-imidazo[1,2-b]pyrazole ethane;N-[(1R)-3-[4-hydroxy-5-methyl-6-oxo-2-(phenylsulfanylmethyl)pyran-3-yl]propyl]acetamide 5-amino-2-[(Z)-1,4-bis(sulfanylidene)but-2-en-2-yl]benzamide;ethane 2-(2,4-dichlorophenoxy)-N'-hydroxypyrimidine-4-carboximidamide 4-[(2E,4Z)-6-[5-fluoro-3-methyl-2-[[6-methyl-3-(2H-tetrazol-5-yl)pyridin-2-yl]amino]phenyl]hepta-2,4,6-trien-3-yl]oxybutanoic acid 4-[5-(2-amino-4,6-dichlorophenyl)pyridine-3-carbonyl]piperazin-2-one 2-[4-(5,5-dimethylhexan-3-yl)phenyl]pyridine 4-(2,6-dimethylphenoxy)-3-fluorobenzonitrile 1-[(3S)-7,7-difluoro-5-methyl-1-(4-propan-2-ylphenyl)sulfonyl-6,8-dihydro-5H-pyrrolizin-3-yl]-5-(1H-pyrazole-4-carbonylamino)pyridin-1-ium-3-carboxamide N-(2-methylpropoxy)-N-[1-[4-(trifluoromethoxy)phenyl]ethyl]butanamide [2-hydroxy-3-(propanoylamino)phenyl]phosphonic acid 3-[(1,2-dimethylcyclopropanecarbonyl)amino]-4-(3-fluorophenyl)benzoic acid N-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-2-oxochromene-3-carboxamide 1-(2,4-dichlorophenyl)-N-[3-[5-[4-fluoro-3-(4-methylpiperazine-1-carbonyl)phenoxy]pyrimidin-2-yl]oxypropyl]-2H-pyrimidin-6-amine 2-[[4-(2,6-dimethylphenoxy)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine 3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-6,7,8a,9,10,11-hexahydro-5aH-pyrido[2,3-c]azocin-4-one 2,3-bis(but-2-enyl)pyridine 2-[2,4,6-trimethyl-N-(3-morpholin-4-ylpropyl)anilino]decanoic acid 4-(2,6-dipyridin-4-yl-5H-1,3,4-thiadiazin-4-yl)benzene-1,2-diol 2-[(3-methoxyphenyl)methyl]-7-[4-(4-methylpiperazin-1-yl)anilino]-9H-pyrido[3,4-b]indole-3-carbonitrile N-[4-fluoro-2-(6-methyl-5-oxo-7,8-dihydroimidazo[1,2-a]pyrimidin-3-yl)phenyl]formamide 2-(2,5-diethylpyrazol-3-yl)-7-fluoro-6-methoxyquinoline N-[4-(2-acetamidophenyl)phenyl]-1-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide N-[1-(furan-2-ylmethyl)piperidin-4-yl]-3,5-dimethoxybenzamide 7-[(3R)-5,5-dimethylpyrrolidin-3-yl]oxy-2-(4-propan-2-ylpyridine-3-carbonyl)-9,10-dihydroanthracene-1-carboxamide 4-(2,2,6-trimethylpiperazin-1-ium-1-yl)benzamide ethane;3-[1-[(3E,5Z)-hepta-1,3,5-trien-4-yl]oxyethylideneamino]pyridine-2-carbonitrile 4-chloro-5-fluoro-3-[[2-(1H-pyrazol-5-yl)pyrrolidin-1-yl]methyl]-1,2-thiazole 1-methylspiro[2,4-dihydroquinoline-3,4'-piperidine] 1-[1,4-dimethyl-5-(trifluoromethoxy)pyrazol-3-yl]-3-[2-[6-(ethylamino)pyridin-3-yl]ethylamino]propan-2-ol 2-methyl-5-[(3S)-3-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)pyrrolidine-1-carbonyl]-3H-isoindol-1-one 3-[2,6-difluoro-N-(4-hydroxybutyl)anilino]propane-1,2-diol 1-[2-(4,5-dichlorocyclohexa-2,4-dien-1-yl)quinolin-3-yl]propan-1-ol 3-[4-(aminomethyl)phenyl]-5,7-diethyl-1H-pyrazolo[4,3-c]pyridine-6-carbonitrile 1,3-dichloro-5-[2-(3-methylsulfonylphenyl)ethynyl]benzene 2-amino-5-methylhexane;4-[(E)-3-(4-hydroxyphenyl)prop-1-enyl]phenol N-[1-(2,3-dimethoxyphenyl)ethyl]-4H-quinazoline-6-carboxamide 2,4-dinitro-1H-[1]benzothiolo[3,2-d]pyrimidine 6-[4-(1-azidocyclopropyl)phenoxy]-N,2,5-trimethylpyrimidin-4-amine 4-[azido(diphenyl)methyl]sulfanylphenol 3,5-dichloro-4-(3-methylbut-1-en-2-yl)phenol (5E)-3-benzyl-2-imino-4-oxo-N',5-diphenyl-5-propoxyiminocyclopentene-1-carboximidamide (3R)-5,6-dichloro-N-methyl-1-methylidene-3H-2-benzofuran-7-amine 1-[4-(2,6-dimethylphenyl)piperazin-1-yl]-3-piperidin-1-ylpropan-1-one 2-hydroxyethoxy(phenyl)phosphinate 2-methyl-3-[1-(oxan-4-yl)imidazol-2-yl]-7H-cyclohepta[b]pyran-6-one 4-[3,5-bis(trifluoromethyl)phenyl]-N,2-dimethyl-1H-pyrrole-3-carboxamide 1-(3,4-dimethyl-5H-pyrazolo[3,4-b]pyridin-7-yl)piperidin-2-one 3-[[4,5-dimethyl-1-(2-phenylethyl)imidazol-2-yl]sulfanylmethyl]-N'-hydroxypyridine-2-carboximidamide N-(6-propoxy-1,3-benzothiazol-2-yl)carbamate 2-bromo-4-[6-chloro-7-fluoro-8-(3,3,3-trifluoropropoxy)-1,5-naphthyridin-4-yl]piperazine-1-carboxylic acid ethane;5-[(3S)-1-phenylsulfanylpyrrolidin-3-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene 1-[(4-chlorophenyl)methyl]-3-[4-methoxy-7-(2-methylmorpholin-4-yl)-[1,3]thiazolo[5,4-c]pyridin-2-yl]urea 2-benzyl-6,7-dihydroxy-4H-pyrazolo[1,5-a]pyrimidin-5-one 5-[2-(3,4-dimethylphenyl)ethenyl]-6-hydroxy-1H-pyrimidine-2,4-dione [4-[1,1,2,3,3,3-hexafluoropropan-2-yl-[methyl(naphthalen-2-yl)amino]phosphoryl]oxyphenyl]azanium N-[(5Z)-3-chloro-4-oxo-5-phenacylidene-1,2-thiazolidin-2-yl]benzamide 7-bromo-N-[2-(dimethylamino)ethyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide N-cyclohexyl-2,4-difluoro-5-[1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]benzamide (2E,4Z)-3-[1-(1,1-difluoroethylsulfanylmethylamino)ethenyl]-N'-ethyl-2-methyl-4-phenylhepta-2,4-dienimidamide (E)-3-(4-fluorophenyl)-1,5-bis[2-nitro-6-(trifluoromethyl)pyridin-4-yl]pent-1-en-3-ol (2-methoxypyridin-4-yl)-[2-methyl-3-(5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl)piperidin-1-yl]methanone (4-fluorophenoxy)-[2-oxo-2-phenylmethoxyiminoethyl]phosphanium 5-(3-bromophenyl)-N'-hydroxypyridine-2-carboximidamide 4-[(4E)-5,6-dimethylidenedeca-4,8-dienyl]phenol;methanol 4-[4-[(3Z)-5-[cyclopentylmethyl(methyl)amino]-4-methylidenehexa-1,5-dien-2-yl]piperazin-1-yl]pyrimidine-2-carbonitrile N-(2,4-difluorophenyl)-7-(1H-indol-6-yl)-3,4-dihydro-2H-pyrido[2,3-b]pyrazine-1-carboxamide 1-(4-chlorophenyl)ethylphosphanylidenemethanethiol 1-[(3,5-dichlorophenyl)methyl]-4-(trifluoromethylsulfonyloxy)piperidine-4-carboxylate 2-[[4-(6-aminopyridin-3-yl)phenyl]methoxy]propanoic acid 4-[3,5-bis(trifluoromethyl)phenoxy]-N'-hydroxybenzenecarboximidamide (2R)-1-(3,5-difluorophenyl)-N-[1-[2-(4-ethylsulfonylphenyl)-2-methylpropyl]-7-methoxyimidazo[4,5-c]pyridin-6-yl]methanesulfonamide N-(4,5,6,7,8,9-hexahydro-[1]benzothiolo[2,3-d]azepin-3-ylmethylideneamino)aniline 2-[3,4-bis(difluoromethyl)pyrazol-1-yl]pyridine;N,6-dimethyl-2-thiophen-2-ylquinolin-7-amine 1-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)piperazin-1-yl]-2-pyridin-3-ylethanone;1-methyl-5-propan-2-yl-2H-pyrazine 2-[4-ethoxy-N-(3-methylbut-2-enyl)anilino]acetonitrile N-[4-(methylamino)-1-phenylbutyl]pyridine-3-carboxamide 4-(2,4-diaminopyrimidin-5-yl)-1-[(2R)-2-methoxy-2-phenylethyl]pyridin-2-one 2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfanylethanethiol 4-(1,3-dioxolan-2-yl)quinoline 1-[2,6-di(propan-2-yl)phenyl]ethenesulfinic acid N-(4-hydroxyphenyl)-4,5-dihydro-1H-imidazole-2-carboxamide (Z,2E)-5-methyl-N-[4-(3-methylidene-7H-pyrrolo[1,2-a]imidazol-6-ium-2-yl)phenyl]hex-2-en-1-imine N-(2,3,4,5,6-pentamethylphenyl)-1H-indol-3-amine 5-[4-amino-2-(6-aminopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-N-(3-ethoxypropyl)-2-methanimidoylaniline 6-[4-[3-(oxolan-2-ylmethoxy)propanoyl]piperazin-1-yl]-5-phenylpyridine-3-carbonitrile (4E)-5-amino-2-[2-(2,3-dihydro-1H-inden-2-yloxy)ethyl]-8,10-dioxobenzo[c]chromene-9-carboxamide 6-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidine;methane ethane;1-methyl-3,4-diphenylpyrazole 3-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)oxy-N'-hydroxyazetidine-1-carboximidamide (E)-1-(2,3-dihydro-1H-inden-5-yloxyamino)propan-2-ol 6-[(1S,2R)-2-(4-bromophenyl)cyclopropyl]pyridazine 2-(2,5-dibromophenyl)-4,6-dihydrazinyl-1,3,5-triazine-2-sulfonic acid 1-[4,5-bis(ethenyl)-2-methylidenehexa-3,5-dienoyl]-N'-hydroxy-N-propan-2-ylpyrazole-3-carbohydrazide 1-(2,3-dimethylphenyl)-5-[(E)-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-ylhydrazinylidene)methyl]-2,6-dihydropyrazolo[3,4-d]pyrimidin-4-one 2-[(1Z)-buta-1,3-dienyl]-4-methylidene-6-phenyl-1H-pyrimidine;ethane 3-[2,6-dichloro-4-(trifluoromethoxy)phenyl]-1,3-oxazolidine 2-(4-azidooxyphenyl)sulfonylnaphthalene (2Z,5E)-3-ethyl-2-[(4-methoxyphenyl)methylidene]-5-prop-2-enylidenethiolane 1-[3-(4-bromophenyl)-2,5-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl]-3-(oxolan-3-ylamino)-2-phenylpropan-1-one 1-[(4R,5S)-3-bromo-4-methyl-1,3-oxazolidin-5-yl]-N-[2-(6-oxocyclohexa-2,4-dien-1-ylidene)ethyl]naphthalene-2-carboxamide N-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-7-yl)pyridine-4-carboxamide 1-(8,9-difluoro-6H-isochromeno[4,3-b]chromen-2-yl)ethanone 4-[1-(difluoromethyl)pyrazole-3-carbonyl]-2,5,7,8-tetrahydropyrido[4,3-c]pyridazin-6-one 2-azido-4-fluoro-1,3-dihydroisoindole 4-[3,5-dimethoxy-N-(naphthalen-1-ylsulfanylamino)anilino]-N,N-dimethylbut-2-enamide (3R)-N-[2,4-difluoro-3-[5-methyl-7-(morpholin-4-ylmethyl)-2H-indazole-3-carbonyl]phenyl]pyrrolidine-3-carboxamide (2R,3S)-N-[(5-chloro-2-hydroxyphenyl)methyl]-1-(3-methylpyrazine-2-carbonyl)-2-(trifluoromethyl)pyrrolidine-3-carboxamide 7-[4-(2,4-dimethoxyphenyl)piperazine-1-carbonyl]-3H-[1,2,4]triazolo[4,3-a]pyridin-5-one N-[(Z)-1-pyridin-2-ylethylideneamino]quinoline-4-carboxamide 1-(3-ethyl-2H-pyran-5-yl)-3,4-dihydro-1H-isochromene N-[2,3-diamino-5-(oxan-4-yloxy)phenyl]furan-2-carboxamide 4-benzyl-2,6-dibromophenol 1-(4,6-dimethylpyridin-2-yl)propan-2-ylcarbamic acid 5-[(3R,5S)-1-(2,4-dichlorobenzoyl)-5-methylpyrrolidin-3-yl]-N,N-diethylpyridine-2-sulfonamide 2-[1-(1,3-benzodioxol-5-ylsulfonyl)pyrrolidin-2-yl]-N-cyclopentylacetamide 2-methylsulfanyl-1-phenyl-3,4-dihydroisoquinoline N-(1,3-benzodioxol-5-ylmethyl)-2-[4-[1-[(6E)-1-fluoro-6-hydrazinylidenepyridine-3-carbonyl]piperidin-4-yl]butyl]benzamide 4-(6,7-dimethoxy-2H-chromene-3-carbonyl)-3-methylpiperazin-2-one 1-[4-(2-chloro-3-fluoro-6-methoxyphenyl)-5-methylpyridin-2-yl]-4-[3-(difluoromethyl)-2H-triazol-1-yl]butan-1-one 2-[(3R,5S)-1-(3-fluorophenyl)sulfonylpyrrolidin-3-yl]-7-methoxy-8-propan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-amine 1-amino-N,2-dimethylpyrrole-3-carboxamide;5-(2-oxopyrrolidin-1-yl)-4H-1,4-benzothiazin-3-one 3,4-diaminophenol;N,2-diethylaniline 1-[[2-[6-[3-(trifluoromethyl)phenoxy]pyrazin-2-yl]phenyl]methylidene]guanidine 4-amino-2-(4-methylpyridin-3-yl)oxybenzamide 1-[(2S)-4-[bis(4-fluorophenyl)methyl]morpholin-2-yl]hexan-1-one 3-[(Z)-2-aminoethenyl]-5-[1-(3,4,5-trimethoxyphenyl)sulfonylpyrrolo[2,3-b]pyridin-2-yl]-1H-pyridin-4-one (2R,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-N-[3-[2-chloro-5-(morpholine-4-carbonyl)phenyl]prop-1-en-2-yl]-4-fluoropyrrolidine-2-carboxamide 1-azidooxy-2,3-dibromobenzene N-[(4S)-8-amino-2,7-dimethyl-3-oxoheptan-4-yl]-6-[2-methoxy-5-(trifluoromethyl)phenyl]pyridine-3-carboxamide 2-[1,3-dihydroxypropan-2-yl(methyl)amino]-N-(6-formamidopyrimidin-4-yl)acetamide N-(4-bromobutan-2-yl)-N-(5-bromopyridin-2-yl)benzenesulfonamide 4-chloro-2-(4-methylphenyl)sulfanylpyrimidine 1-azidosulfanyl-2,3,4-trimethoxybenzene 3-methyl-1-phenyl-5,6-dihydrotriazolo[4,5-d]pyridazine (2S)-2-[3-oxo-7-[(4R,6S)-1,6,8,9-tetrahydropyrano[2,3-g]quinolin-4-yl]-1H-isoindol-2-yl]cyclopentan-1-one N-[[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]methyl]-1-methoxypropan-2-amine 3-[(Z)-[7-cyclopropylimino-5-(methylideneamino)pyrazolo[1,5-a]pyrimidin-3-ylidene]methyl]-4H-1,2,4-oxadiazol-5-one N-azido-2,6-dinitroaniline 2-(1-cyclohexylethenylamino)oxycarbonylbenzoic acid N-[1-(4,4,5,5-tetramethyloxaborolan-2-yl)ethyl]quinoline-6-carboxamide 2-[(4S)-1,2-bis(3-fluorophenyl)-6-oxopiperidin-4-yl]propanamide N-(3,4-dihydro-1H-isoquinolin-2-yl)-4-propan-2-yloxy-6-pyridin-4-ylpyrimidin-5-amine ethane;(1-hydroxy-6,7-dihydronaphthalene-2-carbonyl)azanium N-(4-methoxyphenyl)-3,5-dimethyl-1-[5-[2-(methylamino)ethoxy]pyrimidine-2-carboximidoyl]-6,7-dihydroindol-6-amine N-(1,5-dimethylpyrazol-4-yl)sulfonyl-2-[3-(trifluoromethoxy)phenyl]propanamide 4-[1,3-bis(benzenesulfonyl)-5-methoxyindol-2-yl]-2-methoxyphenol 2-tert-butyl-3-chloro-5H-pyrrolo[1,2-b]pyridazine-4-carboxylic acid 3-[5-[4-(2,6-diphenylpyridine-4-carbonyl)piperazin-1-yl]sulfonyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione 3-(4-azidooxyphenoxy)propan-1-ol (2E)-5-[[1-(4,4,4-trifluorobutyl)pyrazol-3-yl]methylidene]imidazolidine-2,4-dione 1-(4-azidophenoxy)-3,6-dimethylnaphthalene N-(4,6-dimethylpyrimidin-2-yl)-4-[hexadecanoyl(1,3-thiazol-5-yl)amino]benzenesulfonamide 1-[3-[3-[(3,4-dimethoxyphenyl)methyl]azetidine-1-carbonyl]piperidin-1-yl]prop-2-en-1-one ethane;2-methyl-6-propanoylchromen-4-one 1-[4-bromo-2-(trifluoromethyl)phenyl]ethanone 2-[3,5-bis(trifluoromethyl)anilino]pyridine-4-carboxylic acid 1-[(3R)-4-(3,5-difluorophenyl)-2,3-dimethylbutanoyl]-N-[(2S)-1-hydroxypropan-2-yl]pyrrolidine-2-carboxamide 5-[2-methylsulfanyl-4-(trifluoromethyl)phenyl]imidazolidine-2,4-dione N-azido-2,5-difluoro-N-methyl-4-nitroaniline 2-(3,5-difluoroanilino)-6-[2-methyl-4-(4-methylpiperazin-1-yl)phenyl]pyrido[3,2-d]pyrimidine-8-carboxylic acid 4-(2,4-dichloropyrimidin-5-yl)oxy-3,5-dimethylbenzonitrile 2-(4,5-diphenylimidazol-1-yl)-6-[(3S)-pyrrolidin-3-yl]oxypyrimidine 6-(4-hexoxyphenyl)-5,7-dihydropyrrolo[3,4-b]pyridine 2-azido-1,4-diphenylbutane-1,3-dione 5-[(4-methoxyphenyl)methyl]-3,6-diphenylbenzene-1,2,4-triol 6,7-dimethyl-1,5-naphthyridine;2-methanimidoyl-4-(4-morpholin-4-ylphenyl)aniline (2E)-2-[(3,5-dibromophenyl)methylidene]-5-(4-fluorophenyl)-N,N-dimethylcyclohexan-1-amine 1-(4,5-dimethyl-2-phenylpiperazine-1-carbonyl)pyrazole-3-carboxylic acid 2-amino-6-(9H-fluoren-1-yl)-4-methylsulfonylphenol 2-[(1S)-1-azidoethyl]-5-fluoropyridine 5-[4-[(2S,3R)-4,4-difluoro-3-methylpiperidine-1-carbonyl]phenyl]-2H-isoquinolin-1-one 4-amino-2,6-dibromo-N'-(2,2,6,6-tetramethylpiperidin-4-ylidene)benzenecarboximidamide (3R)-4,6,6-trimethyl-8,9-dihydropurino[7,8-a]pyrazine 5-[2-azido-4-(trifluoromethyl)pyrimidin-5-yl]oxypentanoic acid 6-(2,3,4a,5,6,7,8,9,10,11,11a-decahydro-1H-pyrido[3,2-c]acridin-4-yl)-1H-pyridin-4-one N-methyl-1-[1-[4-(2,2,2-trifluoroethoxy)phenyl]piperidin-3-yl]methanesulfonamide 3-[4-amino-2-fluoro-5-(2,2,2-trifluoroethylsulfanyl)phenyl]-1-methylpyridin-2-one 2-[3-(4,5-diamino-1H-pyrrol-3-yl)propanoyl]-N-[4-[ethoxy(methyl)boramoyl]phenyl]-3-hydroxybutanediamide (3R)-N,5-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 3-[(2E)-1,7-dimethyl-4-phenylocta-2,6-dien-2-yl]-5-fluorobenzoic acid 5-[[4,6-bis(4-fluorophenyl)pyridine-2-carbonyl]amino]pentanoic acid 1-[6-[(2,4-dichlorophenoxy)methyl]-5-oxa-8-azaspiro[3.5]nonan-8-yl]ethanone;2,2,2-trifluoroacetic acid 1-(3-butyl-4,5,6,7,8,9-hexahydro-2H-cyclohepta[d]imidazol-1-yl)ethanone 2-[(3R)-1,1-dioxothiolan-3-yl]imino-5-methoxypyrrolo[3,4-f]isoindole-1,3,7-trione 6-(4,5-dichloro-2-methylsulfanylphenyl)-4H-[1,3]thiazolo[5,4-b]pyridine (1-aminocyclopentyl)-[2-[[5-(3,4-dimethoxyphenyl)pyridin-2-yl]amino]piperidin-1-yl]methanone;dihydrochloride 2-[[(1R)-4,6-bis(chloromethyl)cyclohexa-2,4-dien-1-yl]methoxy]-3H-pyrido[3,4-d]pyrimidin-4-one N-(3-hydroxypropyl)-2,2-dimethoxy-N'-[(E)-1-(6-nitronaphthalen-1-yl)ethylideneamino]ethanimidamide 2-[2-(3,5-dichlorophenyl)ethynyl]-6H-furo[2,3-b]pyrrole 2-(2,2-dimethylpropoxy)-N'-hydroxypyridine-4-carboximidamide 1-[4-[4-(4-cyclopropylbenzimidazol-1-yl)piperidine-1-carbonyl]phenyl]imidazolidine-2,4-dione N'-hydroxy-3,4-dimethylbenzenecarboximidamide 6-[[1-(4,5-dimethyl-2-phenyldiazenyl-N-prop-2-ynylanilino)-3-ethoxypropan-2-ylidene]amino]-N'-[1-(4-methoxyphenyl)ethenyl]pyridine-2-carboximidamide 2-[4-(5-azidopyridin-2-yl)piperazin-1-yl]ethanamine 4-[2,3-dihydroxypropyl(2,2-dimethoxyethyl)amino]benzenesulfonic acid 2-(dimethylamino)-6-nitrobenzamide 5-[(2R)-3,3-dimethylbutan-2-yl]sulfonyl-4-phenyl-1H-indazole (Z)-2-[2-chloro-4-fluoro-5-methyl-3-[6-(1,1,1-trifluoropropan-2-ylamino)pyridin-3-yl]phenyl]-3-cyclopentyl-N-ethenylbut-2-enamide ethane;3-[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]sulfonyl-4H-1,3-benzoxazin-2-one 3-chloro-N-[5-(furan-2-yl)-1H-pyrazol-3-yl]-5,6-dihydroimidazo[1,2-a]pyridine-7-carboxamide N-[4-chloro-3-(trifluoromethyl)phenyl]-2-(2-pyridin-3-yl-7H-purin-6-ylamino)acetamide;ethane ethane;(E)-3-[6-(methylideneamino)pyridazin-3-yl]hex-2-en-4-ynal 1-[(E)-(3-fluorophenyl)methylideneamino]-1,2,4-triazole-3-sulfonamide 5-methyl-N-(1,4-oxazepan-6-ylsulfonyl)pyridine-3-carboxamide 2-(1,3-dioxoisoindol-5-yl)imino-5-[(7-methoxyquinolin-4-yl)amino]pentanoic acid 2-[3,6-dimethyl-4-(1,2,3,3,5,6,7,8,9,10,11,12-dodecafluorophenanthren-9-yl)naphthalen-2-yl]naphthalene 4-[3-(2,5-dioxopyrrolidin-1-yl)phenoxy]benzonitrile 3-[4-(1H-indol-2-yl)phenyl]-1,2-oxazol-5-amine 2-N-[4-(4-hexylphenyl)butan-2-yl]benzene-1,2-diamine 4-N-ethyl-2-(methylamino)-1,3-thiazole-4,5-dicarboxamide N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-ylmethyl)aniline 2-(2,5-difluorobenzenecarbothioyl)-5-methylbenzaldehyde N-[3-chloro-4-(pyridine-2-carbonyl)phenyl]-5-fluoropyridine-2-sulfinamide;1,3-difluoro-5-methylbenzene 2,3-dibromo-4-methyl-6-(piperidine-1-carbonyl)benzaldehyde (2S)-1-[4-amino-3,5-bis(trifluoromethyl)phenyl]-2-fluorobutan-1-one;hydrochloride N-[(E)-but-2-enyl]-4-(ethylideneamino)benzenesulfonamide (3R)-1-[[3,5-bis(trifluoromethyl)phenyl]methyl]piperidine;5-chloro-6-(2-morpholin-4-ylethoxy)-N'-(1H-pyrazol-5-ylsulfamoyl)pyridine-3-carboximidamide 1-(2,6-dimethylphenyl)-3,5-dimethoxybenzene 2-aminopyrazolo[1,5-a]pyrimidine-3-carboxamide;8-ethyl-N-phenyl-1,6-naphthyridin-7-amine 1-[(6,6-dimethyloxan-3-yl)oxycarbonylamino]-2-phenylcyclopropane-1-carboxylic acid 1-(3-azidophenyl)indole (E)-1-[2-cyclobutylidene-7-methyl-4-(4-methylphenyl)-3H-1,5-benzodiazepin-8-yl]-3-(3,4,5-trifluorophenyl)prop-2-en-1-one N-[(E)-1-(4-hydroxyphenyl)ethylideneamino]-2-(7-methyl-2,3-dihydrochromen-4-ylidene)acetamide 1-azido-4-(2,5-difluorophenyl)piperidine 3-[4-chlorobutyl(pyridin-2-yl)amino]phenol 6-[(5-chloropyrrolo[2,3-b]pyridin-3-ylidene)methyl]-4H-1,4-benzoxazin-3-one N-(2,5-dichlorophenyl)-N'-(4,6-dimethylpyrimidin-2-yl)ethane-1,2-disulfonamide 2-[(4S)-6,8-dibromo-4-hydroxy-2-oxochromen-3-yl]oxyacetic acid N-(4-amino-3,5,6-trimethylpyridin-2-yl)-2-phenylacetamide 3-[6-chloro-5-(methoxymethyl)pyridazin-3-yl]sulfanylpyrrolidine-1-carboxylate 6-(2,3-difluorophenyl)-1-methyl-2-oxopyridine-3-carbonitrile 4-[(4,6-dimethoxy-1,3,5-triazin-2-yl)sulfanyl]benzene-1,2-dicarbonitrile N-[2-(4,5-dihydrothieno[3,2-d][1]benzazepine-10-carbonyl)-5-propan-2-ylthiophen-3-yl]pentanehydrazide 1-methyl-3,4-dihydroisochromen-4-ol (3S)-4-[(3R)-5,7-difluoro-2,3-dihydroindole-1-carbonyl]-N-[(3-fluoropyridin-4-yl)methyl]pyrrolidine-3-carboxamide N'-azido-N,2-dibenzylethane-1,2-diamine 2,5-bis(6-pyridin-3-ylpyridin-2-yl)pyrimidine 2-(1,5-dimethylpyrazol-4-yl)-7-[(2E,4Z)-hexa-2,4-dien-3-yl]-3H-imidazo[5,1-f][1,2,4]triazin-4-one (5Z)-1,3-bis[2-(1H-indol-2-yl)ethyl]-5-[(E)-pent-3-enylidene]imidazolidine-2,4-dione;chloromethane 1-[6-(6,8-dichloronaphthalen-2-yl)oxypyridin-3-yl]ethanone 2-[[(2E,4Z)-3-aminohepta-2,4,6-trienyl]sulfonylmethyl]benzoic acid N-[2-(3,4,5-trifluorophenyl)ethyl]quinazoline-7-carboxamide N-(4,6-dimethoxypyrimidin-2-yl)sulfanyl-1,3-benzoxazol-2-amine 6-[(4-chlorophenyl)methyl]-2,4a-dimethyl-8-propan-2-yloxy-3,5,11,13-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene;ethane 5-(5-aminopentyl)-3-propan-2-yl-1,6-dihydroindol-2-one;ethane N-[(5S)-5H-indeno[2,1-b]pyridin-8-yl]butanamide (5-chloro-1H-pyrrolo[2,3-b]pyridin-4-yl)boronic acid 2-(2,3-dihydroxyphenyl)-6H-pyrrolo[3,4-f]isoindole-1,3,5,7-tetrone 5-[2,6-difluoro-4-(4-methylphenyl)cyclohexa-1,3-dien-1-yl]pyridine-2-carbonitrile 2-[4-(3-aminopropyl)phenoxy]ethanamine;(6R)-7-butoxy-8-oxo-3,5-dioxabicyclo[4.1.0]heptane-2-carboxylic acid 3-methyl-4-[5-(6-phenylpyridine-2-carbonyl)spiro[1,3-dihydroisoquinoline-4,2'-piperidine]-1'-yl]benzamide (2S)-3-[4-[2-cyclopropyloxy-5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl]naphthalen-1-yl]oxy-N-(2,2-dimethylpentan-3-ylsulfamoyl)propanenitrilium 6-(3-chloropyridine-4-carbonyl)-7,8-dihydro-5H-pyrido[4,3-c]pyridazine-1,3-dione N-[6-(aminomethyl)cyclohexa-1,5-dien-3-yn-1-yl]-4-ethoxybenzamide (7-fluorospiro[chromene-2,4'-piperidine]-1'-yl)-pyridin-4-ylmethanone 2-methyl-4,9-dioxobenzo[f]chromene-6-carbonitrile 2-(3,5-dihydro-1H-pyrrolo[3,4-c]pyrazole-6-carbonyl)-N-methyl-2-azabicyclo[2.1.0]pentane-3-carboxamide;ethane 3-[(5Z)-3-(4,5-dihydro-1H-imidazol-2-yl)-2-ethylocta-2,5,7-trienoxy]benzonitrile 3-[(4-methoxyphenyl)-(3,5,6-triethyl-9H-carbazol-1-yl)sulfanyl]propane-1-sulfonate 1-(6-methylpyrimidine-4-carbonyl)-N,N-bis(2-methylpropyl)pyrrolidine-3-sulfonamide 2-(ethylcarbamothioylamino)oxy-N-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]acetamide 7,8-dichloro-3-(3,5-dichlorophenyl)-2-ethoxypyrido[2,3-e][1,4]oxazine N-[4,6-dimethoxy-5-(2-pyrrolidin-1-ylethyl)pyridin-3-yl]-2,5-difluorobenzenecarboximidate (1S,2R)-2-[4-[(3-fluoro-4-methoxyphenyl)carbamoyl]phenoxy]cyclopentane-1-carboxylic acid N-(3,4-dimethoxyphenyl)sulfonyl-6,7-diethoxyquinoline-2-carboxamide N-[(1R,2S)-3-methyl-1-(2-methylsulfanylpyrimidin-4-yl)oxybutan-2-yl]acetamide 4-ethyl-2-[1-(4-methoxyphenyl)-1,3,5-triazin-2-ylidene]pentanoate 6-fluoro-4-[(2R)-5-methylideneoxolan-2-yl]oxy-N-phenylpyridine-3-carboxamide 3-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-(1,2-oxazol-3-ylmethyl)pyrazole-1-carboxamide N-[3-(difluoromethyl)phenyl]-2-(4-oxoquinazolin-3-yl)acetamide 6-[(3E)-hexa-1,3,5-trien-3-yl]oxy-N-phenylpyridine-2-carboxamide 2-[(3S,4R)-1-ethylsulfonyl-4-hydroxypiperidin-3-yl]pyridine 3-[2,4,5-tris(sulfanyl)anilino]propanenitrile 7-fluoro-6,8-dimethoxy-N-[(2R)-1-methylpiperidin-3-yl]-4-oxo-1H-quinoline-3-carboxamide N-[3,5-bis(ethenyl)phenyl]-2-[2-chloro-1-(4-chlorophenoxy)ethoxy]-6-methylidenecyclohexa-1,3-diene-1-carboxamide 2-[2-(dimethylamino)ethoxy]benzaldehyde N-[2-amino-4-(1,3-dihydroisoindol-2-yl)phenyl]-5-(1H-benzimidazol-2-yl)thiophene-2-carboxamide 5-(2,3-difluoro-4-phenylmethoxyphenyl)sulfanyl-1H-pyrrolo[2,3-c]pyridine 4-[5-(3,5-dimethoxyphenyl)hexanoylamino]butanamide ethane;4-(2,5,7-trimethylcycloocta-1,3,6-trien-1-yl)oxy-4H-naphthalen-1-one 3-(4,5-dimethylthiophen-2-yl)-N-[(4-hydroxy-1,1-dioxothian-4-yl)methyl]-1H-pyrazole-5-carboxamide (2R)-N-[5,7-dimethyl-1-(4-phenylbutanoyl)pyrazol-3-yl]-6-oxopiperidine-2-carboxamide 2-[4-(5-fluoropyrimidin-4-yl)piperazin-1-yl]-N-methylacetamide 2-[1-(4,5-dimethylpyrimidin-2-yl)piperidin-3-yl]-6-[2-(trifluoromethoxy)phenyl]pyridazin-3-one (E)-4,8-dihydroxy-1,3-dihydroxyxanthene-9,10-dione 4-[2-methoxyethyl(pyridin-3-yl)amino]-6,7-dihydropyrrolo[1,2-a]pyrimidine-8-carboxamide 4-amino-6-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 4-chloro-6-(2-ethoxyphenyl)cyclohexa-2,4-dien-1-amine 5-[[4-[(E)-1,2-diphenylbut-1-enyl]phenyl]methyl]spiro[1H-indole-3,4'-piperidine]-2-one 3-[2-cyclopropyl-4-(2,5-dimethoxyphenyl)imidazol-1-yl]-1H-pyrazin-2-one [(3S)-1-[2-fluoro-4-(trifluoromethyl)phenyl]sulfonylpiperidin-3-yl]carbamic acid 4-[3-(2-methylpropoxy)phenyl]-2-sulfanylidene-1,3,4,6-tetrahydropyrimido[4,5-d]pyrimidin-5-one 5-[4-(2,4-dichlorophenyl)piperazin-1-yl]-3-propan-2-yl-1,2,4-thiadiazole N-[3-(2,5-dimethylphenyl)propyl]-2-(methylaminomethyl)cyclohexan-1-amine 4-(6-fluoroquinolin-3-yl)oxy-N,2-dimethylpentanamide;2-[3-(4-fluorophenyl)-5-hydroxy-1-benzofuran-7-yl]acetaldehyde N-[3-chloro-4-(1-methylpyrrolo[2,3-b]pyridin-4-yl)oxyphenyl]-5-(4-fluorophenyl)-1-methyl-6-oxopyridazine-3-carboxamide 1-[2,3-diamino-5-(trifluoromethyl)phenyl]ethanone 7-azidooxy-2,2-dimethylchromene 2-[(2,6-dichlorophenyl)carbamoylamino]cycloheptane-1-carboxylate 2-[(1,3-dimethylpyrazolo[4,3-b]pyridine-6-carbonyl)amino]-5-phenylpentanoic acid (Z)-N'-[1-[3,5-dimethyl-4-[4-(2,3,4,5-tetrafluorophenyl)piperazine-1-carbonyl]anilino]ethenyl]-N-ethylidenehex-2-enediamide 1,3-dibutyl-5-[2-[4-(5-carboxypentoxy)phenyl]propan-2-yl]-6-chloroindole-2-carboxylic acid 6-(2-bromo-5-chlorophenyl)-4-N,8-dimethylpyrimido[5,4-d]pyrimidine-2,4-diamine N-[2,6-dimethoxy-4-(5-methylimidazol-1-yl)phenyl]-N'-[(4S)-6-[1-(2-fluorophenyl)ethylsulfanyl]-1,2,3,4-tetrahydronaphthalene-1-carbonyl]-N-methylethanehydrazide 6,7-dimethoxy-2-[(E)-3-[4-(trifluoromethyl)phenyl]prop-1-enyl]quinoxaline 1,3-diamino-1-[2-[(E)-3-[4-[N'-(4-methoxyphenyl)carbamimidoyl]piperazin-1-yl]prop-1-enyl]sulfanyl-3-propan-2-yloxyphenyl]urea N-(2,5-dichlorophenyl)-1-[6-[3-(trifluoromethyl)phenyl]benzotriazol-1-yl]propan-2-imine 4-(1H-benzimidazol-2-ylmethoxy)benzenecarboximidamide 3-(4-azidooxybutyl)benzoic acid 3-[(2R)-1,4-dioxospiro[2H-pyrrolo[3,2-c]pyridine-3,4'-piperidine]-2-yl]propanamide;hydrochloride 2-[[5-chloro-4-(pyridine-3-carbonylamino)pyrimidin-2-yl]amino]acetic acid (5R)-2,2-dimethyl-7-oxo-N-[(1S)-1-phenylpropyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-5-carboxamide 2-(5-tert-butyl-3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclohexane-1-carboxylic acid 2-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethoxy]benzoic acid 2-(6,8-dichloro-2H-chromen-3-yl)-3,4-dimethylquinoline 1-N'-[(E)-2-phenylethenyl]-1-N'-(2,4,5-trifluoroanilino)cyclopropane-1,1-dicarboxamide 2-amino-5,6-difluoro-4-[3-hydroxy-3-(triazol-1-ylmethyl)piperidin-1-yl]quinoline-3-carbonitrile 7-[2,5-dichloro-6-(trifluoromethoxy)phenyl]-9H-pyrido[3,4-b]indole 4-(3,4-dihydro-2H-pyran-7-ylmethoxy)aniline 5-chloro-2,4-difluoro-N-[(4S)-3,8,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),4,10-tetraen-4-yl]benzenesulfonamide [1-hydroxy-2-(3-methoxyphenyl)ethylidene]azanium 1-methyl-4-propan-2-yloxypyrrolo[3,2-c]quinoline 2-[3-(cyclopropylmethyl)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl]-5-ethylbenzaldehyde 3-[(2E,5Z)-3-ethylocta-2,5-dienoxy]benzaldehyde 5-[4-(2-morpholin-4-ylethoxy)phenyl]imidazolidine-2,4-dione 3-[1-(2,6-dichlorophenyl)-5-[4-hydroxy-3-(trifluoromethyl)phenyl]pyrrol-2-yl]benzenesulfonamide 3-methyl-5-[4-(2-phenylethynyl)anilino]sulfanylbenzoic acid 1-(4,5-dimethyl-6-oxo-2,3-dihydro-1H-pyridin-3-yl)indole-3-carboxamide 2-methylbuta-1,3-diene;2-propan-2-yl-N,6-di(propan-2-yl)pyridin-4-amine 5-cyclohexyl-3-methyl-8-propan-2-yl-1,3,4,6,7,9-hexahydropyrazolo[4,3-b]quinoline (3-chlorophenyl)-[4-(7H-purin-2-yl)piperazin-1-yl]methanone (5R)-2,4,7-trimethyl-6-oxo-N-phenyl-1H-pteridine-8-carboxamide N-[2,4-dimethyl-5-(2-phenylacetyl)thiophen-3-yl]benzenesulfonamide 1,4-bis(3-butoxy-2-chlorophenoxy)isoquinoline 4-(4-nitropyrazol-1-yl)-N'-(pyridine-2-carbonylamino)piperidine-1-carboximidamide (Z)-3,4-dimethoxy-N-(1-methyl-2-oxo-5,6,7,8-tetrahydroquinolin-5-yl)but-2-enamide 4-(2,5-dimethylphenyl)benzoate N-methylsulfanyl-1,4-dioxoisoquinoline-5-carboxamide 3-[4-[2-(1,3-benzodioxol-5-yl)ethoxy]piperidine-1-carbonyl]-N-methylpyridine-4-carboxamide (5R)-3,9-diazaspiro[4.6]undecan-2-one;methylcyclohexane 1-ethenyl-2,3,4-trimethylindole [(1R)-2,3-dihydro-1H-inden-1-yl]carbamothioylcarbamic acid N-azido-3,5-dichlorothiophene-2-carboxamide 2-methylsulfonyloxy-4-phenylbenzoic acid 2-[4-[2-(dimethylamino)ethyl-methylcarbamoyl]phenoxy]acetic acid (6S)-8-benzyl-2-[4-chloro-3-(trifluoromethyl)anilino]-6,7-dihydropyrimido[5,4-d]pyrimidine-6-carboxylic acid 2-azido-5-[(4R)-6,8-difluoro-3-methyl-1-oxo-2H-isoquinolin-4-yl]benzonitrile (2S,6R)-4-[1-[5-chloro-2-fluoro-3-(trifluoromethyl)phenyl]ethoxy]-2,6-dimethylmorpholine N-[(4S,5Z)-4-methylocta-1,5-dien-2-yl]-5-(4-methylphenyl)pentanamide 2-amino-5,6-diethyl-3-[4-[1-[[(4S)-1-hexyl-4-propanoylpyrrolidine-3-carbonyl]amino]cyclobutyl]phenyl]benzimidazole-7-carboxylic acid 4-(2,6-dimethylphenyl)sulfanylmorpholine [3-(4-bromophenyl)morpholin-4-yl]-(1H-pyrazol-5-yl)methanone 5-[(5Z)-2,3-dihydroxyocta-1,5-dienyl]-6-propan-2-yloxybenzene-1,3-diol 1-[2,6-difluoro-3-methyl-5-[4-(trifluoromethoxy)phenyl]sulfanylphenyl]ethanethiol N'-hydroxy-1-benzofuran-5-carboximidamide 6-(8,9-dihydrodibenzofuran-2-yl)benzimidazolo[1,2-a]benzimidazole 4-methoxy-6-[5-(3-morpholin-4-ylpropoxy)pyrazin-2-yl]quinoline-7-carboxylic acid 2-[(3,5-dichloropyridin-4-yl)methylidene]propanedioic acid 4-N,5-dimethyl-3-N-[(1S)-2,2,2-trifluoro-1-phenylethyl]pyrazolo[1,5-a]pyrimidine-3,4-dicarboxamide 2-methyl-N-[4-[(5-nitro-1,3-benzoxazol-2-yl)amino]cyclohexylidene]pyridine-3-carboxamide 4-bromo-5-nitropyrimidine-2-carboxylate 3-[(4,6-dimethylpyridin-2-yl)oxymethyl]piperidin-1-amine 1-[4-(dimethylamino)piperidine-1-carbothioyl]pyrrole-2-carboxylic acid 6-amino-4-[2-[(3,5-dimethylphenoxy)methoxy]phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 4-[2,5-dimethyl-3-oxo-6-(thiophen-2-ylmethoxy)pyridazin-4-yl]benzonitrile 1-[2-(4-bromophenyl)sulfanylpropanoyl]-N',N'-dimethylpiperidine-3-carbohydrazide N-cyclopropylsulfanyl-1,1,1-trifluoro-5-(3-fluorophenyl)pent-4-en-2-amine 3-[2,6-diethyl-4-[(Z)-(5-methoxycarbonyl-1H-imidazol-4-yl)iminomethyl]phenoxy]propanoic acid N-[3-[2-(aminomethyl)-5-formylphenyl]-4,5-difluorophenyl]acetamide 2-[(3R,4S)-3-fluoro-1-phenylsulfonylpiperidin-4-yl]oxy-5-(4-methylimidazol-1-yl)pyridine (2R,3aS)-5-chloro-2-(dimethylamino)-1'-(pyridin-4-ylmethyl)spiro[indole-3,3'-pyrrolidine]-2'-one;2,2,2-trifluoroacetic acid 2-azido-N'-[6-(4,5-dimethylimidazol-1-yl)pyrimidin-4-yl]benzenecarboximidamide 3-[3-(5-methylthiophene-2-carbonyl)phenyl]-1-pyridazin-3-ylpropan-1-one N-[(2,4-dichlorophenyl)methyl]spiro[3,7a-dihydro-1H-imidazo[1,5-a]pyrazine-8,4'-piperidine]-1'-carboxamide 2,3-dimethyl-5-[2-oxo-2-(3H-1,2,4-triazol-5-yl)ethoxy]benzenesulfonamide (1R,2R)-N-(oxan-4-ylmethyl)-2-[3-oxo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-isoindol-2-yl]cyclohexane-1-carboxamide 2-methyl-N-(4-propan-2-ylphenyl)sulfanylcyclohexa-1,5-dien-3-yn-1-amine N-butan-2-yloxy-3,4,5-trimethoxyaniline 1,5-dichloro-2-methoxy-3-(methylsulfonylsulfanylmethyl)benzene N-[3,5-bis(trifluoromethyl)phenyl]-2,2,4,6,7,8-hexadeuterio-N'-(2,3,5-trifluorobenzoyl)-1-oxa-4-azaspiro[4.5]decane-9-carbohydrazide 3-[(2,5-dichlorophenoxy)methyl]cyclobutane-1-carboxylic acid N-[2-[(3R)-3-(4,6-dimethoxypyrimidin-2-yl)piperidin-1-yl]ethyl]propanamide 3-[(2S)-1-acetyl-2,3-dihydropyrido[2,3-b]pyrazin-4-yl]phenol (2-aminopyridin-3-yl)-[3-(5-phenyl-1,2,4-oxadiazol-3-yl)azetidin-1-yl]methanone 6-[(E)-2,3-dimethylbut-1-enyl]-7,8-dihydrocyclohepta[b]pyridine 5-hydroxy-1,6-dimethyl-4-oxopyridine-3-carboxylate 1-(dimethylamino)-2,2,6,6-tetrafluoro-N'-[5-(1H-indol-3-yl)pentanoyl]piperidine-4-carbohydrazide 7-chloro-8-cyclopropyl-5,6-dihydroxynaphthalene-1,4-dione N-[[1-(3,4-difluorophenyl)cyclopropyl]methyl]-5,6,7,8-tetrahydroquinazoline-2-carboxamide 5-(2,3,4,5-tetrahydroindol-1-yl)-N'-[7-(trifluoromethoxy)cyclohepta-1,6-dien-1-yl]pyridine-2-carboximidamide 1,3-dihydroisoindole;ethane;6-methylsulfonylpyridine-3-carbonitrile (2R,4S)-3-[[5-amino-6-(4-fluorophenyl)pyrazine-2-carbonyl]amino]-4-methylhexanoic acid (5R,7S)-N-[2-(dimethylamino)ethyl]-5,7-bis(4-methoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 3-[1-(7,8-dihydronaphthalen-2-yl)-5-ethynylpyrrol-2-yl]propanoic acid 2-[4-[[(3,5-dichloropyridine-2-carbonyl)amino]methyl]piperidine-1-carbothioyl]imidazo[1,2-a]pyridine-6-carboxylic acid 1-(5-bromo-3,4-difluorophenyl)-2-(4-methylpiperazin-1-yl)ethanone 1-N',2-N',7-N'-trimethyl-5-propan-2-yl-3-propan-2-ylidenebenzene-1,2,4,6,7-pentol 2-(4,5-dihydropyrrolo[1,2-a]quinoxaline-1-carbonyl)cyclohexan-1-one N-(4-chlorobutyl)-2,3-dihydroxybenzamide 5-[3-(4,6-diphenylpyridin-2-yl)phenoxy]pyrimidine 3-[[4,5-di(propanoyl)-1H-imidazol-2-yl]amino]-N-methoxybenzamide N-[6-methyl-2,4-dioxo-1-(3-propan-2-ylphenyl)pyrimidin-5-ylidene]propane-2-sulfinamide 2-[4-(aminomethyl)phenyl]pyridine-3,5-dicarboxamide 2-[azido(diphenyl)methyl]-1,3,5-trimethoxybenzene 2,6-dichloro-N-[2-(cyclohexylmethyl)phenyl]benzamide 7-[2-(3,4-difluorophenyl)morpholine-4-carbonyl]-6-methyl-1H-quinolin-2-one N-[(3S,5R)-1,7-dibenzyl-4-oxo-5-phenyl-8,9-dihydro-6H-imidazo[2,1-f]purin-3-ium-3-yl]-4-methylbenzenesulfonamide 5-amino-6-azido-2-chlorooxypyridine-3,4-dicarbonitrile 3-[[2,4-difluoro-N-(pyridin-2-ylmethoxy)anilino]methylideneamino]benzoic acid 3-[1,2-bis(4-chlorophenyl)ethyl]-7-[methoxy(methyl)amino]chromene-2,4-dione 1-[4,6-dibromo-2-(3,5-dimethylphenyl)quinoline-3-carbonyl]pyrrolidine-2-carboxylate 3-(4-tert-butylsulfonylphenyl)-2-(difluoromethoxy)propanoic acid 6-amino-4-[2,4-dimethyl-5-(trifluoromethoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide N-[1-(2,4-dichlorophenyl)ethyl]-5-fluorospiro[1H-indole-3,1'-cyclobutane]-2-carboxamide 2-[6-(2,4-difluorophenyl)pyridin-2-yl]ethanamine (5Z)-5-[(4-ethylthiophen-2-yl)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione 2-fluoro-N-[4-(4,4,5,5-tetramethyloxaborolan-1-ium-3-yl)phenyl]benzamide 2-[N-(4-hydroxybutyl)-4,5-dimethyl-2-phenyldiazenylanilino]acetonitrile 3-fluoro-5-methoxy-N-[1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonyl)piperidin-4-yl]benzamide 3-ethoxy-2-[4-(6-methyldodecan-5-yl)phenyl]pyridine 3-[4-[2-(trifluoromethoxy)phenyl]phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 2-azido-3-methylsulfanylbenzenesulfonate 4-bromo-2,5-dimethyl-N-(3-nitrophenyl)-N-[2-(trifluoromethyl)phenyl]aniline 5-[[2-(4,6-dimethylpyrimidin-5-yl)oxyethylamino]methyl]-N-phenylthiophene-3-carboxamide 2-[4-(5,6-dihydroxy-1H-benzimidazole-2-carbonyl)piperazin-1-yl]acetamide 1-azido-2,4,5-trimethylindazol-3-one 4-[2-(furan-3-ylmethylamino)ethoxy]cyclohexa-1,5-diene-1-carboxylic acid N-ethyl-3-iodonaphthalene-2-carboxamide 6-amino-7-[1-(dimethylamino)propan-2-ylamino]-3H-quinazolin-4-one;ethane 2-ethylimino-5-(4-methoxyphenyl)imidazolidin-4-one 3-[3,5-dimethoxy-4-(oxolane-2-carbonyl)anilino]-1-[(Z)-1H-indol-3-ylmethylideneamino]azetidine-2,5-dione 2-[3-cyano-4-ethyl-5,6-dimethoxy-N-[(4-phenylphenyl)methyl]anilino]acetic acid 3-[[(2S,4R)-4-hydroxy-1-methylpyrrolidin-2-yl]methoxy]benzenesulfonamide (6R,11S)-11-[[3-(trifluoromethyl)pyridine-2-carbonyl]amino]-1-azabicyclo[4.4.0]decan-6-olate 2-(azetidin-1-yl)-6-azidooxy-4-(oxolan-3-yloxy)quinazoline 3,3-dimethyl-1-[4-(6-methylpyridazine-4-carbonyl)piperidin-1-yl]butan-2-one N-azido-3,5-dichloro-N-(2-fluorobenzoyl)-6-hydroxypyridine-2-carboxamide N'-[1-[2-(2,4-dimethylphenyl)phenyl]ethenyl]propane-1,3-diamine 1-[2-ethoxy-5,6-difluoro-3-(trifluoromethyl)phenyl]tetrazolidine 2-azido-1,3,4,5,6,7,8,9,10-octafluoroanthracene [4-hydroxy-1-methyl-6-oxo-7-(2,3,5,6-tetrafluorophenoxy)pyrido[2,3-d]pyrimidin-8-yl]boronic acid 2-(N-benzoylanilino)benzenesulfonic acid N-[3-(azidomethyl)phenyl]-2,4,6-trifluorobenzenesulfonamide N-[5-(oxan-2-yloxy)pyridin-3-yl]formamide 3-(furan-2-ylmethoxy)-6,7-dihydro-5H-1-benzothiophen-4-one N-(2,5-dibromophenyl)sulfanyl-4-fluorobenzenesulfonamide [4-(2,6-dimethylphenyl)piperazin-1-yl]-(5,5-dimethyl-7H-pyrrolo[3,4-b]pyridin-3-yl)methanone 5-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl)quinolin-8-yl]-N-ethylsulfonyl-1H-imidazole-4-carboxamide 5-[[2,4-bis(trifluoromethyl)phenyl]carbamoylamino]-N-piperidin-3-ylnaphthalene-1-carboxamide 1-chloro-4-(2,3-difluorophenoxy)-5-hydroxy-9H-fluorene-2-carboxylic acid 1-(2,5-diethyl-4-nitrophenyl)ethanesulfonamide 1-(6-cyclopropylpyrimidin-4-yl)-2,3-dihydroindole-5-carboxylic acid 4-(9,10-dioxoanthracen-1-yl)oxybenzenesulfonic acid 5-cyclopropyl-2,4-difluoro-N-[(3S,4R)-1-methoxy-6-methylpiperidin-3-yl]benzamide N'-[2-(cyclopropylmethylamino)acetyl]benzenecarboximidamide 2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]pyridine;(E,4Z)-4-propylidenehept-6-enal 4-[6-(difluoromethyl)pyrimidine-4-carboximidoyl]pyridin-2-amine;N'-(1-hydroxyethylsulfonyl)ethanimidamide 1-[3-(ethylcarbamoylamino)phenyl]-N,N-dimethylcyclopropane-1-carboxamide 2-(4-chlorophenoxy)-N'-hydroxypyrimidine-4-carboximidamide 1-(2,6-dimethoxyphenyl)-N-[4-(3,5-dimethylpyrazol-1-yl)phenyl]pyrrolidine-3-carboxamide N-cyclohexyl-2,4-dimethoxy-5-[3-(2-methoxyethyl)imidazo[1,2-a]pyridin-6-yl]benzamide N-[1,2-difluoro-4-[6-(5-methyl-1H-pyrazol-3-yl)pyridin-3-yl]oxybutylidene]hydroxylamine 1,2-bis(3-methylbutyl)-4-nitroimidazole (3aR,7aS)-2-[5-(difluoromethyl)-1-methylpyrazole-4-carbonyl]-7a-(ethoxymethyl)-N-methyl-1,3,3a,6,7-hexahydropyrrolo[3,4-c]pyridine-5-carboxamide 4-(3,4-dimethylpentanoyl)-2,5-bis[5-methoxy-2-methyl-1-(4-methylphenyl)indole-3-carbonyl]benzoic acid (3R)-1-[2-bromo-4-[5-chloro-2,6-dimethyl-4-[(4-pyridin-2-ylpiperazine-1-carbonyl)amino]phenyl]sulfanylphenoxy]pyrrolidine-3-carboxylic acid N'-[(3E)-hepta-1,3-dien-4-yl]-2,6-dimethoxybenzenecarboximidamide 1-ethenyl-4-(6-methoxyhexyl)benzene (1S,2S)-N-[8-amino-6-(4-methoxypyridin-3-yl)isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide N-(4-methylphenyl)propanamide;2-piperidin-1-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidine 1-phenylmethoxycycloheptane;5,6,7,8-tetrahydronaphthalene-2-carboxylic acid 2-bromo-5,6-dichloro-N'-[(4-cyclohexylphenyl)methyl]benzenesulfonohydrazide 4-[(3Z)-3,4-difluorohexa-1,3,5-trien-2-yl]oxy-N-[[2-methoxy-6-(trifluoromethyl)phenyl]methyl]butanamide;ethane 2-[3-(5,6-difluorocyclohexa-1,5-dien-1-yl)oxyphenoxy]acetic acid (6S)-2,5-dimethyl-4-[1-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-phenyloxan-2-yl]oxybutyl]-6,7-dihydroisoindole-1,3-dione N-[4,6-bis(methylamino)pyridin-3-yl]-2-cyanoacetamide 2-[(5-bromo-1,3,4-thiadiazol-2-yl)amino]phenol 4-(2,5-diaminophenyl)naphthalene-1-sulfinate N-azidooxy-4-[(2,6-dichlorophenyl)methyl]aniline 7-methyl-N-(6-morpholin-4-ylpyridin-3-yl)imidazo[1,2-a]pyridine-8-carboxamide;N-(oxan-4-yloxy)formamide 1-[7,8-bis(sulfanyl)octyl]-3,4,5-trimethoxypyrrole N-(2,6-difluorophenyl)-5,7-dimethoxy-1H-indole-3-carboxamide 6-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[(4-methoxyphenyl)methylsulfanyl]-2,6-dihydro-[1,2,4]triazino[1,6-c]quinazolin-1-one 2-[5-carbamoyl-9-[[3-ethoxy-4-(7-oxo-1,6,8-triazatricyclo[8.2.0]tetradeca-3,5,10,12-tetraen-11-yl)phenyl]methyl]carbazol-4-yl]-2-hydroxyacetic acid (E)-N-[3-amino-1-oxo-2-phenylmethoxy-3-pyridin-4-ylpropan-2-yl]-5-[(1S)-1-ethoxyethyl]pent-2-enamide N-butyl-3,5-bis(2,4,6-trimethylphenyl)benzamide;ethane 3-(4-bromophenyl)-6-ethylsulfonyl-8-methoxycarbonylimidazo[1,2-b]pyridazine-7-carboxylic acid 1-[(2S)-1-[4-(aminomethyl)piperidin-1-yl]propan-2-yl]-3-[6-[5-(cyclopropanecarbonyl)pyridin-3-yl]pyrimidin-4-yl]urea N-(2,3-dimethyl-1H-indol-5-yl)-2-[4-(trifluoromethoxy)phenyl]quinoline-4-carboxamide 3-[[2,6-dimethyl-1-(pyridin-4-ylmethyl)piperidin-3-yl]oxymethyl]-5-propan-2-yl-1,2,4-oxadiazole;ethane 2-amino-6-(3,4-dichlorophenyl)-9-methyl-8H-pyrimido[5,4-b]pyrrolizine-7-carboxylic acid 1-chloro-3-(cyclopenta-2,4-dien-1-ylmethyl)isoquinoline N-[2,3-difluoro-4-(2-nitroethylamino)phenyl]benzamide 1,3-diamino-1-[2-[4-chloro-2-(trifluoromethyl)phenoxy]-5-methoxyphenyl]urea 3-(3,4-diethoxybenzoyl)cyclopentan-1-one (4S)-N'-[2,3-bis(ethenyl)phenyl]-1-cyclopentylspiro[5,7-dihydropyrazolo[3,4-b]pyridine-4,3'-indole]-2',6-diimine 4-[5-[6-(trifluoromethyl)pyridin-3-yl]-7H-cyclopenta[d]pyrimidin-4-yl]morpholine 2-(3,4-dibromophenyl)propanamide;ethane N-[(2S)-1-hydroxybutan-2-yl]-3,5-dinitrobenzamide N-[4,6-diamino-2-(diethylamino)pyrimidine-5-carboximidoyl]acetamide [2-(7,8-dichloroquinolin-4-yl)-6-phenylphenyl]azanide 2-[(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)methoxy]propanoic acid 3-methoxycarbonyl-1,4-dihydroquinoxaline-2-carboxylic acid 1-[4,6-dimethyl-2-(pyridine-3-carbonyl)pyrimidin-5-yl]ethanone [2-(2,4-dimethylphenyl)sulfonyl-1H-isoquinoline-3-carbonyl]carbamic acid N-(2-hydroxyethyl)-4-[5-[1-(4-methoxyphenyl)ethylidene]-2,3-dihydro-1H-pyrrol-4-yl]benzamide 3-(4,5-dichloropyrimidin-2-yl)oxy-1H-quinoxalin-2-one (2S,3R)-1-(1H-imidazole-5-carbonyl)-2-(phenylmethoxymethyl)pyrrolidine-3-carboxylic acid 3-[(4Z)-hepta-1,4,6-trien-2-yl]sulfanyl-6-methylpyridine 3-[(2R,4S)-2-[[1-(2,5-dimethoxyphenyl)piperidin-4-yl]carbamoyl]-4-hydroxypyrrolidine-1-carbonyl]piperidine-1-carboxylic acid 1-benzyl-3-methoxypyrazin-2-one 6-[3-(2,4-difluorophenyl)-1,2-oxazol-5-yl]-N-hydroxy-2-oxo-9-[4-(oxolan-3-ylaminomethyl)phenyl]nonanamide 1-(3,5-dimethylphenyl)-4-[1-[4-fluoro-2-[2-[4-[1-hydroxy-2-(methoxymethyl)-3-methylbutyl]phenoxy]ethyl]phenyl]ethenyl]piperidine 4-[[5-[3-(chloromethyl)anilino]pyridin-2-yl]amino]phenol 2-(4,5-dimethylcyclohexen-1-yl)oxyacetamide;ethane;3-[[2-(2-methylidene-6-propan-2-ylidenecyclohex-3-en-1-ylidene)hydrazinyl]methyl]benzenethiol 2-amino-5-cyclohexyl-3-[4-(1,2,4-triazol-1-yl)benzoyl]benzoic acid N-[(2S)-6,8-dimethoxy-1,2,3,4-tetrahydronaphthalen-2-yl]-N'-[1-(7-methylpyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]propanehydrazide 6-[2-(4-ethylphenyl)ethynyl]benzo[b][1,4]benzothiazepine 3-[4-[2-(cyclohexylamino)ethyl]piperazin-1-yl]phenol 1-[3,5-bis(trifluoromethyl)phenyl]-N-(4-butan-2-yloxyphenyl)sulfonylcyclopropane-1-carboxamide 4-methyl-N-[3-oxo-1-phenyl-3-[(3R)-4-prop-2-enoylpiperazin-1-yl]propylidene]-3H-benzimidazole-5-carboxamide 1-(3-fluorophenyl)-3-[[2-hydroxy-5-methyl-3,4-di[(Z)-prop-1-enyl]cyclohexa-1,3-diene-1-carbonyl]amino]urea 1-(6-ethyl-2-oxohexyl)-3-[4-[5-(propanoylamino)pyridine-2-carboximidoyl]phenyl]urea (3Z,4E)-1-ethyl-3-[1-(4-methoxyphenyl)ethenylidene]piperidin-2-one 4-[2-(3,5-dimethoxyphenyl)ethynyl]pyridine 7-cyclohexa-1,5-dien-1-yl-9,10,11-trioxotetracene-2-carboxamide 3-[2-chloro-3,4-bis(phenylmethoxy)phenyl]pentanoic acid 4-(difluoromethoxy)-N-[6-(1,3-thiazol-5-yl)cinnolin-3-yl]benzamide (6S)-2,8,11-trihydroxy-1,7-dimethyl-3,10-dioxoanthracene-9,10-dicarboxylic acid 3-(2,6-diphenylphenyl)benzamide 5-chloro-N-methyl-2-(1,3-thiazol-2-yl)pyrimidine-4-carboxamide 5-[2-(3,4-dimethylphenyl)ethynyl]pyrimidine 1-(3-methylbutyl)-2-[6-oxo-4-(trifluoromethoxy)-1H-pyrimidin-5-yl]benzimidazole-5-carbonitrile 6-(4-butylphenyl)-2,5-dimethoxypyridine-3-carbonitrile 1-azido-2-[3,5-bis(trifluoromethyl)phenyl]piperidine 2-[8-(6-methylpyridine-3-carbonyl)-3,8-diazabicyclo[4.2.0]octan-3-yl]-1-pyrrolidin-1-ylethanone N'-[5,6-bis(ethenyl)pyridin-3-yl]-1H-pyrazole-5-carboximidamide (1E,3Z)-N,N,5-trimethyl-2-propan-2-ylidenehexa-1,3-dien-1-amine;4-[3-oxo-3-[3-(trifluoromethoxy)anilino]prop-1-ynyl]thiophene-2-carboxylic acid 5-(6-cyclopropyl-2,3-difluorophenyl)-6-fluoro-4-[[1-(3-methoxypropyl)piperidin-4-ylidene]methylamino]pyridine-3-carboxylic acid 2-(2,3-dihydro-1H-inden-5-yloxy)-N-methylsulfonylacetamide 5-amino-2,4-dimethyl-N-(3-phenylsulfanylcyclobuta-1,4-dien-1-yl)benzamide N-[2-[4-[(3,5-dichlorophenyl)sulfamoyl]phenoxy]ethyl]-4-methoxybenzamide 4-[1-(2,3-dihydroindol-1-yl)-2-methylpropan-2-yl]oxy-N-ethylaniline 1-(4-chlorophenyl)sulfonyl-3,4-dihydro-2H-quinoline 5-amino-4,6-diphenylpyrimidine-2-carboxylic acid [4-(trifluoromethyl)phenyl]carbamodithioic acid 2-[4-[(2R)-3-(1H-indol-5-yloxy)propan-2-yl]sulfonylphenyl]acetic acid (4S)-4-[3-fluoro-2-methoxy-5-(trideuteriomethyl)phenyl]-1,3-dihydropyrrolo[2,3-b]pyridine (4S)-2,3,5,8-tetramethyl-1-oxo-N-(pyridin-4-ylmethyl)spiro[2H-pyrrolo[1,2-a]pyrazine-4,3'-pyrrolidine]-4'-carboxamide 1-azido-4,6-diphenyl-1,3,5-triazinane 2-[(4-chlorophenyl)methyl]-3-ethoxybenzoate 1-(5,6-dihydro-4H-pyrrolo[3,2-d]pyrimidine-7-carbonyl)-3-[1-(methoxymethyl)piperidin-4-yl]imidazolidin-4-one 4-N-(2,3,5-trichlorophenyl)pyrimidine-4,6-diamine (E)-3-[4-[2-cyclopropyl-1-(8-methoxy-1,2,3,4-tetrahydroquinolin-6-yl)ethyl]phenyl]-1-piperidin-4-yl-N-pyridin-3-ylprop-2-en-1-imine 6-fluoro-3,4a,5,10a-tetrahydro-2H-pyrano[3,2-c]quinoline 2-[1-(4,6-dioxocyclohexa-1,5-dien-1-yl)azetidin-3-yl]oxypyridine-3-carboxylic acid (3R)-4-[5-[2-(2-hydroxyethylamino)pyrimidin-4-yl]-1,3,4-oxadiazol-2-yl]-N,N-dimethylmorpholine-3-sulfonamide 4-[N-(2,3-dihydroxypropyl)-4-methoxycarbonylanilino]benzenesulfonic acid 3-ethylhexane;4,5,7-trinitro-2H-benzotriazole 3-[5-(4-aminophenyl)sulfanyl-1,3,4-thiadiazol-2-yl]propanoic acid 6-[2-(oxan-4-yl)ethynyl]quinoline 1-[4-(2,3-dihydroindole-1-carbonyl)phenyl]cyclopropane-1-sulfonamide 2-[(4R)-6,7-dimethoxy-4-(oxan-3-ylmethylamino)-3,4-dihydroisoquinolin-1-ylidene]acetic acid 4-(5,6-difluoro-2,3-dihydroindol-1-yl)pyrimidine-5-carboxylic acid 3-[(4-fluorophenyl)methyl]-1H-indole;N'-hydroxy-4-(piperidin-1-ylmethyl)pyridine-2-carboximidamide 1-[4-chloro-2-(trifluoromethyl)phenyl]-3-[3-methoxy-4-(1H-pyrazol-4-yl)phenyl]urea (6Z)-4,8-dimethyl-1-[2-oxo-2-(1H-pyrrol-3-yl)ethyl]-7,8,9,10-tetrahydroimidazo[4,5-a]azocine-5,10-dione;ethane (6-bromo-3,5-dimethylpyrazin-2-yl)carbamic acid (1S)-N',4-dimethyl-2-phenyl-3H-1,5-benzothiazepine-7-carbohydrazide 4-[5-fluoro-6-[2-(3,4,5-trifluorophenyl)ethynyl]naphthalen-2-yl]benzonitrile N-[(Z)-but-1-enyl]sulfanyl-5,8-difluoroquinoline-6-carboxamide;1-(1H-imidazol-2-ylmethyl)azepan-4-one 5-[8-chloro-7-[(4-hydroxycyclohexyl)amino]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-6,7-dimethoxyisoquinoline-3-carboxamide 2-amino-6-borono-1H-indole-5,7-dicarboxylic acid 3-[6-(4-hydroxyphenyl)-2H-thiopyran-5-yl]pentanoic acid N-[1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]-N'-methyl-2-(5-methylsulfanylthiophen-2-yl)acetohydrazide;ethane 2-tert-butyl-6-[[4-hydroxy-3,5-di(propan-2-yl)phenyl]methyl]-3-(3-methoxypropyl)phenol 2-[(3-butoxyphenyl)methylidene]-6-fluorocyclohexan-1-one 2-amino-6-(5-methyl-1,3,4-thiadiazol-2-yl)phenol 4-[(5R)-3-amino-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-5-carbonyl]benzonitrile 4-(1,3-benzodioxol-5-yl)-2-(cyclobutylmethylamino)quinazoline-6-carbonitrile 1-[4-(2,6-dioxopiperidin-3-yl)benzoyl]oxyethenylazanide 2-chloro-N-[4-[4-(3,5-dicyclopropylpyrazole-1-carbonyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl]benzamide 2-[1-(2,6-dioxopiperidin-3-yl)-2-methyl-4-(2-phenylethylamino)-3H-isoindol-5-yl]-N'-hydroxyethanimidamide [(3S)-3-aminopyrrolidin-1-yl]-[2,3-dimethyl-6-[4-[5-[4-(1H-pyrrol-2-yl)phenyl]pyrimidin-2-yl]piperazin-1-yl]pyridin-4-yl]methanone 2-(3,4-dimethoxyphenyl)-5,6-difluoro-1-benzofuran N-(3-chloro-4-fluorophenyl)-3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazole-2-carboxamide (3Z)-N'-tert-butyl-3-[(1,4-dimethoxynaphthalen-2-yl)methylidene]-2-oxoindole-5-carbohydrazide (4R)-2-[6-cyclopropyl-1-(2,5-dimethoxyphenyl)sulfonylindol-3-yl]-4-hydroxy-N,2-dimethylpentanamide N-cyclobutyl-1,4-dimethyl-3-methylidene-6,7-dihydropyrazolo[3,4-b]pyrazin-2-imine 4-(2,5-dimethylphenyl)-3-ethylaniline 4-[2,4-dioxo-3-[1-[5-(1H-pyrrol-2-ylmethylideneamino)pyridin-2-yl]piperidin-4-yl]cyclobuten-1-yl]oxy-N-phenylbenzamide 5-[4,6-bis(ethenyl)pyridin-2-yl]-3H-1,3,4-oxadiazol-2-one 2-[3-chloro-5-(trifluoromethyl)pyridin-4-yl]phenol N-[2,6-dimethyl-4-(2-phenoxyethoxy)phenyl]-2-fluoro-3-hydroxybenzamide 2-[3,5-dibromo-4-(7H-purin-6-ylamino)phenyl]propan-1-ol (1E,3Z)-5-(4-ethylphenyl)penta-1,3-dien-1-amine 2-[3,5-dichloro-4-(1H-indol-2-yl)phenyl]-6-methoxyoxan-4-ol (1-aminoethylideneamino)-[4-[3,5-difluoro-2-[(1R)-4-methylcyclohexa-2,4-dien-1-yl]oxyphenyl]phenyl]azanium 1-(2,2,3,3,4,5,4,5,5,6,7,8,8,9,10-heptadecafluorodecoxy)propane;(1R,2S)-2-phenylcyclopentan-1-ol 2-[[4-(3,5-dichlorophenyl)-6-ethoxy-1H-indole-2-carbonyl]amino]-2-phenylacetic acid 4-[4-fluoro-2-(trifluoromethyl)phenyl]-5-hydroxy-1H-pyrimidin-6-one 4-[1-(1,3-benzodioxol-5-yl)pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine (3R,4S)-1-benzyl-N-(2-methoxyethyl)-3-methylpiperidine-4-carboxamide N-[(1R)-3-aminocyclopentyl]-2,4-dimethylimidazo[1,5-a]pyrimidine-8-carboxamide;hydrochloride 2-amino-4,4-dimethoxy-6-(5-methylfuran-3-yl)-3-azabicyclo[3.1.0]hex-2-ene-1,5-disulfonic acid N-(3,4-dihydro-2H-chromen-6-ylsulfonyl)-5,6-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxamide;hydrochloride 3-[(E)-2-(6,7,8,9-tetrahydrodibenzofuran-1-yl)ethenyl]benzaldehyde (1Z)-3-[2,3-difluoro-5-(methylamino)phenyl]buta-1,3-dien-1-ol 2-(3-chloropyridin-4-yl)-N-methyl-5-[1-oxo-1-(oxan-4-ylamino)propan-2-yl]oxypyrazole-3-carboxamide 2-[(E)-2-phenylethenyl]-1H-quinoline-4,5-dione N-(2,5-dimethylphenyl)-5-oxo-1-[(3S)-1-propanoylpiperidin-3-yl]pyrrolidine-3-carboxamide N-azido-2-propoxybenzamide 2-[[5-chloro-1-(3,5-dimethylphenyl)pyrazole-4-carbonyl]amino]acetic acid [(2S)-1-methylpyrrolidin-2-yl]-[4-phenyl-5-(trifluoromethyl)thiophen-3-yl]methanone (4-methylsulfonylphenyl)-[1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]methanone N-[2-(cyclopropanecarbonylamino)imidazo[1,2-b]pyridazin-6-yl]-6-methoxypyridine-3-carboxamide 4-(N-methylanilino)pyridine-2-sulfonic acid 3-(2,6-difluorophenyl)-7-methyliodanuidylquinoline [(2S)-2-[[1,3-benzodioxol-4-ylmethylcarbamoyl-[6-(2-cyanophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]methyl]piperidine-1-carbonyl]oxidanium (5R)-2,3,5-trimethyl-8-(4-methylphenyl)-1-propan-2-ylidene-2H-imidazo[4,5-c]quinoline N-(3-bromopropyl)-N-butyl-4-nitrobenzamide 2-chloro-N,5-dimethyl-3H-1,4-benzodiazepine-8-carboxamide N-[2-chloro-4-(methoxyamino)phenyl]pyridine-3-carboxamide 2-[4-(dimethylamino)-1,3-dihydroisoindol-2-yl]-6-ethylpyridine-4-carboxylic acid 6-chloro-N-diazo-1H-indole-2-sulfonamide 4-(4,6-dimethylpyrimidin-2-yl)oxy-3-(2-ethyltriazol-4-yl)benzonitrile 3-[(1E,3Z)-1,4-diamino-5-methylpenta-1,3-dienoxy]aniline 2-[4-(azetidin-1-yl)phenyl]-N'-ethyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-6-carboximidamide 1-azidosulfanyl-2,3,5,6-tetramethyl-4-(2-nitrophenyl)benzene 5-[4-[4-(2,6-dioxopiperidin-3-yl)piperazin-1-yl]butylcarbamoylamino]pyridine-2-carboxamide N'-[3,5-bis(trifluoromethyl)benzoyl]-2,4-dichlorobenzenesulfonohydrazide (4R)-1-tert-butyl-3-methyl-4-pyridin-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 3-cyclopropyloxy-N-ethyl-5-(2H-tetrazol-5-yl)benzamide 2-methoxy-5,6-bis(phenylmethoxy)-3-[(2R)-oxan-2-yl]pyrimidin-4-one (1R,2R)-N-[8-amino-6-[4-(3-methylbutanoyl)piperazin-1-yl]isoquinolin-3-yl]-2-cyanocyclopropane-1-carboxamide 3-(azidomethyl)-1,5,8-trimethoxyanthracene [2,5-di(propan-2-yl)phenyl]-[3-methoxy-5-(1H-pyrazol-4-yl)piperidin-1-yl]methanone 2-methyl-5-[4-[5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl]phenyl]benzaldehyde 2-azido-4-methoxy-5,6,7,8-tetrahydro-3H-quinazolin-4-ol 5-[2-hydroxyethyl(3,3,3-trifluoropropyl)amino]sulfanylthiophene-2-carboxylic acid 2-[(3R,4S)-3-hydroxypiperidin-4-yl]oxybenzonitrile 4-[5-(methoxymethyl)furan-2-yl]-7-[1-[(6S,8R)-6,8,9-trifluoro-10-methoxy-5-oxo-1,2,3,4-tetrahydropyrano[3,4-c]isoquinolin-12-yl]ethyl]chromen-2-one 2-methyl-3,5-dihydropyridazino[4,5-b]quinoline N-(2-methylpropyl)spiro[1,4-dihydroquinoxaline-3,4'-piperidine]-2-imine (5E)-2-imino-5-[[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]thieno[3,2-d]pyrimidin-6-yl]methylidene]imidazolidin-4-one 3-(9H-fluoren-1-yl)-5,6-dimethoxypyridine-2-carboxylic acid 2-[1-amino-4-(3,4-difluorophenyl)sulfanylbutan-2-ylidene]guanidine 2-amino-4-[3-(3,5-ditert-butylphenyl)propanoyl]benzamide 3-[4-(1,2,3,4,5,6,7,8,9,10,10a-decahydropyren-2-yl)butyl]furan N-(4-fluorophenyl)sulfanyl-6-methoxypyrimidin-4-amine N-[5-[3,5-bis(trifluoromethyl)phenyl]-1H-imidazol-2-yl]butanamide 2,6-dimethoxy-4-(5-methyloctan-2-yl)aniline (Z)-3-[5-ethyl-4-hydroxy-2,6-dimethoxy-3-nitrophenyl]-2-(2H-tetrazol-5-yl)prop-2-enenitrile N-[5-[3,5-bis(trifluoromethyl)phenyl]-4-chloro-2-(4-hydroxypiperidin-1-yl)phenyl]benzamide 4-(chloromethyl)-3,5-difluorothiophene;[4-[2-(5-ethoxypyridin-2-yl)propan-2-yl]phenyl]sulfanium (Z,3Z)-N'-methoxy-3-[(2-methylphenyl)hydrazinylidene]prop-1-ene-1,2-diamine 1-(4,5-dihydrobenzo[g][2]benzoxepin-8-yl)pyrrole 1-[3-chloro-4-[(2S)-2,5-dimethylpiperazine-1-carbonyl]phenyl]piperidine-3-carboxylic acid 2-(4-phenylpiperidine-1-carbonyl)oxybenzenesulfonic acid 2-[2-amino-4-[3,5-bis(trifluoromethyl)phenyl]-1H-imidazol-5-yl]pyridine-4-carboxamide N-[1-[4-[(3R)-2,6-dioxopiperidin-3-yl]piperazine-1-carbonyl]piperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-carboxamide 2-[1-[4-chloro-3-(trifluoromethyl)phenyl]-5-methoxypyrazol-4-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide N-[5-(3,4-dichlorophenyl)-3H-1,2,4-oxadiazol-2-yl]-4-methoxyaniline 1-(4-azidooxyphenyl)-2,3-dihydronaphthalene (E)-3-(4-bromophenyl)-1-[2-(difluoromethoxy)phenyl]prop-2-en-1-one 6-[(4R)-2-amino-1,3-dioxospiro[2H-isoindole-5,2'-cyclopropane]-1'-yl]-N-isoquinolin-6-ylhexanamide 2-(N-butanoyl-4-hydroxyanilino)acetic acid 4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-2-hydroxybenzoic acid 1-[2,3-dichloro-6-(2,5-dimethoxyanilino)sulfanylpyridin-4-yl]piperidin-4-ol 7-benzyl-1-(5,6,7,8-tetrahydroquinazoline-2-carbonyl)-N-[[4-(trifluoromethoxy)phenyl]methyl]spiro[6,8-dihydropyrrolo[2,1-c][1,4]oxazine-9,4'-piperidine]-3-carboxamide 7-[(3,5-dichlorophenyl)methyl]-2-propan-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one 1-azido-6-(trifluoromethyl)indole 2-(3-fluoro-4-isothiocyanatophenyl)-5-heptylpyrazine 5-[4-chloro-6-[4-(2,3-dihydroindole-1-carbonyl)piperidin-1-yl]-1H-benzimidazole-2-carbonyl]pyrrolidin-2-one 1-(4-cyclobutylphenyl)-3,5-dimethoxybenzene;ethane (3S,4R)-1-[[4-fluoro-2-methyl-5-(2H-tetrazol-5-yl)phenyl]carbamoyl]-4-hydroxypiperidine-3-carboxylic acid 3-(2,4-difluorophenyl)sulfanyl-6-[1-(1H-pyrazol-5-ylmethyl)piperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-one 4-[(1E)-3-methylidenecycloocten-1-yl]benzonitrile 4-(3-bromophenyl)-8,13,15-triazatetracyclo[7.6.0.02,6.010,14]pentadeca-1(9),10,12,14-tetraene 4-[(4R)-1,3-dimethylpiperidin-4-yl]oxy-2-[(1Z)-1-(methylideneamino)buta-1,3-dienyl]aniline N-(3-chloropropyl)-4-methylaniline;ethane N-[(2S)-1-amino-3,4-dioxo-1-phenylbutan-2-yl]-2-hydroxypropane-1-sulfonamide;hydrochloride N-(4,6-dimethylpyrimidin-2-yl)-1H-pyrrolo[3,2-c]pyridine-2-carboxamide 3-[2-(1H-imidazol-2-yl)ethenyl]-N,N-dimethylpyridin-4-amine (2S)-1-[4-chloro-3-methyl-5-[3-(methylamino)phenoxy]phenyl]sulfonylpyrrolidine-2-carboxylic acid 4-hydroxy-6-[(2-methoxy-1H-indol-3-yl)diazenyl]naphthalene-1-sulfonic acid 5-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylsulfanyl)pyrimidine-2,4-diamine 3-[(E)-2-(5,6-diethoxy-1,3-benzoxazol-2-yl)ethenyl]benzene-1,2-disulfonic acid 1-[(2S)-4-[[8-amino-6-(5-methylpyridin-3-yl)isoquinolin-3-yl]amino]pyrrolidin-2-yl]propan-2-one 3-aminooxycarbonyl-5-(furan-2-yl)-7-oxo-6H-pyrazolo[4,3-d]pyrimidine-1-carboxylate 3-[4-(2,4-dichlorophenyl)-5H-pyrrolo[3,4-b]pyridin-7-yl]cyclobutan-1-amine 6-[(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)methoxy]pyridine-3-carboxamide 2-[5-methyl-4-(oxan-3-yl)cyclohexa-1,3-dien-1-yl]-N'-phenylbenzenecarboximidamide (E)-3-[2,5-dimethoxy-4-[3-[(1S)-3-methylidene-3a,7a-dihydro-1H-cyclopenta[b]naphthalen-2-yl]propoxy]phenyl]-N-ethoxy-2-methylprop-2-enamide 1-bromo-2-methyl-5,6,7,8-tetrahydroimidazo[4,5-c]azepine 4-azido-2,6-dimethyl-3,5-bis(trifluoromethyl)phenol N-(3,5-dimethylphenyl)-1-(6-fluorospiro[2H-indole-3,4'-oxane]-1-yl)methanesulfonamide N-[2-[1-(furan-3-yl)ethenyl]-5-methoxyphenyl]-3,4,6,7,8,9-hexahydro-1H-pyrimido[4,5-d]azepine-2-carboxamide (7-chloroquinoxalin-5-yl)thiourea;2,3-dihydroisoindol-1-one N-(3-cyanophenyl)-2-[4-[6-(dimethylamino)hexylcarbamoyl]piperazin-1-yl]acetamide 1-(4-bromophenyl)sulfonyl-N,3-dimethyl-6,7,8,9-tetrahydropyrrolo[2,1-c][1,4]oxazepine-5-carboxamide [3-(4,4-difluoropiperidine-1-carbonyl)-2-pyridin-2-ylphenyl]urea 4-[2,5-dichloro-N-(2-phenylethyl)anilino]benzenesulfonamide 7-amino-5-[3-fluoro-2-(methoxymethyl)phenyl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile N-(4-tert-butylphenyl)-3-methoxypropanamide;ethane 4-[(2R,3S)-2-ethenylpyrrolidin-1-ium-3-yl]oxy-6-(5-methoxypyridin-2-yl)thieno[2,3-d]pyrimidine (2S)-N-[(Z)-1H-indol-3-ylmethylideneamino]-2,4-dihydro-1H-pyrimido[1,2-a]benzimidazole-2-carboxamide 1-[[4-(8,11-dihydro-5H-pyrido[3,2-c][1,5]benzodiazepine-6-carbonyl)phenyl]methylamino]-3-ethoxyurea;(Z)-pent-2-ene 2-[(4S)-1,4-dimethyl-6-oxo-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-4-yl]-N-[(1S)-1-thiophen-2-ylethyl]acetamide 2-[4-(4-phenylquinazolin-3-ium-6-yl)carbazol-9-yl]isoindole N-cyclohexa-2,4-dien-1-yl-N,3-diphenylaniline 2-benzyl-7-bromo-5,8-dimethoxychromene (2Z,5E)-6-[3-ethylsulfanyl-4-(1H-indol-2-yl)phenyl]-4-(2-methoxyquinolin-3-yl)hexa-2,5-dienenitrile 2-(2,4-dichlorophenoxy)-N-[1-[3-(2-ethoxyphenyl)propyl]piperidin-4-yl]acetamide 6-[[2,4-difluoro-3-(trifluoromethyl)phenyl]methoxy]-N'-hydroxypyridine-2-carboximidamide 5-bromo-2-chloro-N'-hydroxypyridine-3-carboximidamide N-(4-methoxyphenyl)-N-([1,2,4]triazolo[4,3-a]pyrazin-5-yl)benzamide 5-bromo-4-(2-chloroethyl)pyrimidine (3R,4S)-1-[5-amino-2-[3-methylsulfonyl-6-[(3R)-oxolan-3-yl]oxypyrazolo[3,4-d]pyrimidin-1-yl]phenyl]pyrrolidine-3,4-diol 2-N-(2,3-dihydro-1H-inden-5-yl)-5-ethyl-4-N-[5-methoxy-6-[methyl-[1-(oxetan-3-yl)piperidin-4-yl]amino]pyridin-3-yl]pyrimidine-2,4-diamine N-[[5-chloro-2-(1,3-oxazol-4-yl)phenyl]methoxy]benzenesulfonamide 4-(2,6-dimethoxyphenyl)sulfanylbenzaldehyde 6-methyl-4-methylidene-1H-quinoline-2,3,5-trione N'-hydroxy-1,3-dimethyl-2,4-dioxoquinazoline-6-carboximidamide N-[(4,5-dimethoxyfuran-2-yl)methyl]-3-fluoropyridin-2-amine 5-azido-N,N-diethylpyrazolo[1,5-a]pyrimidine-3-sulfonamide 1-[3-[(5S)-2,3,4a,5,6,8,9,10,10a-octahydro-1H-benzo[h]isoquinolin-5-yl]propyl]piperidine;dihydrochloride 2-[4-[7-(3,5-dimethyl-1H-pyrazol-4-yl)quinolin-5-yl]phenyl]ethanamine 1-[4-(5,7,8,9-tetrahydro-[1,2]oxazolo[3,4-h][2,3]benzodiazin-4-yl)butoxymethyl]cyclopentan-1-amine 3-(2,6-diethylphenyl)-8-methoxypyrido[4,3-e][1,2,4]triazin-5-ium 2-[(3S)-1-cyclohexylpyrrolidin-3-yl]oxy-N'-hydroxypyridine-4-carboximidamide 3,5-bis(trifluoromethyl)-N-[4-[4-[1-[4-(trifluoromethoxy)phenyl]sulfonylpiperidin-2-yl]phenoxy]pyridin-2-yl]benzamide 2-[(5-bromo-1H-pyrrole-3-carbonyl)amino]propanoic acid (4R)-4-(3-chlorophenyl)-3-methyl-1-(6-oxo-1H-pyridazin-3-yl)-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one 3-azido-1H-benzo[e]indole 5-bromo-2-[(6,8-dimethoxy-4H-1,3-benzodioxin-7-yl)methylideneamino]phenol 1-[[4-[(2R)-2,5-diaminopentoxy]phenyl]methyl]pyrazolo[3,4-d]pyrimidine-4,6-diamine 1-[(5S,7R)-5,7-bis(4-chlorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]propan-2-one 1-(3,5-dimethylphenyl)-7-[(4-ethoxyphenyl)methyl]-8-(2-methoxyphenyl)-3-methylpurine-2,6-dione 4-[5-(3-bromophenyl)hexa-1,5-dien-2-yl]-N,N-dimethylaniline N'-[1-(4-fluorophenyl)sulfanylpiperidin-3-yl]-2,5-dimethoxybenzenecarboximidamide 2-[4-[4-(aminomethyl)piperidine-1-carbonyl]phenyl]benzonitrile (3-chloro-4-hydroxy-5-methylphenyl)urea 4-[(2S)-3-azido-1-oxo-1-phenylmethoxypropan-2-yl]benzenecarboximidamide 3-(1,3-benzodioxol-5-ylmethoxy)pyridine 5-(1,3-benzothiazol-6-yl)imidazolidine-2,4-dione 1-(2,5-dimethylpyrazol-3-yl)sulfonyl-N-[5-methyl-6-[4-(trifluoromethoxy)phenyl]pyridin-3-yl]piperidine-4-carboxamide (3R)-1-(2-cyclohexylethoxycarbonyl)piperidine-3-carboxylic acid;2-[4-[2-ethoxy-5-methyl-6-(6-methylpyridin-2-yl)pyrimidin-4-yl]piperazin-1-yl]acetic acid 6-chloro-2,3,4,5-tetrahydro-1H-1-benzazepine-8-carboxylic acid 7-[(3R)-1-(4,5-dihydroimidazol-1-ylmethyl)piperidin-3-yl]oxy-N-[6-[(2R)-2-methylmorpholine-4-carbonyl]pyridin-2-yl]-1H-indole-2-carboxamide ethane;[(5S)-3-[4-[4-(methylideneamino)-2,6-di(propan-2-yl)phenoxy]phenyl]-5-propoxy-1,5-oxazocan-5-yl]methanol 2-[3-[4-(5-hydroxypentyl)piperazin-1-yl]-6,7-dimethoxyquinoxalin-2-yl]phenol 3-methyl-2-[(6R,8S)-5,13-dioxo-17-oxa-4,8,10-triazatetracyclo[9.6.0.02,7.012,16]heptadeca-1(11),2,4,6,8,12(16)-hexaen-13-yl]butanoic acid 1-[(Z)-1,3-diaminoprop-2-enylidene]-3-methylsulfonyl-2H-indene-5-carbonitrile 3-[1-(2,4-dichlorophenyl)piperidin-4-yl]-5-iodophenol 2-(6,7-difluoronaphthalen-1-yl)oxypyridine (7-bromo-1,2,3,4-tetrahydronaphthalen-1-yl)methanamine;hydrochloride 1-[3-[4-(3-butan-2-ylphenyl)phenoxy]propylamino]ethenol;ethane 4-(2,4-dimethoxyphenyl)pyrimidine 1-[4-(5-aminopyrimidin-2-yl)phenyl]ethanone;4,5-dichloro-2-methoxy-N-[[4-(5-oxo-4H-1,3,4-oxadiazol-2-yl)phenyl]methyl]benzamide 1-[4-(2,6-dimethylphenyl)-3H-pyrrol-2-yl]ethanone 6-(3-bromophenyl)-8,9,10-trimethoxy-2-methylsulfanyl-1H-benzo[b][1,7]naphthyridine 1-cyclopropyl-5-[2-(trifluoromethoxy)phenyl]pyrazole 4-[(E)-3,7-dimethyloct-5-enoxy]benzoic acid 2-(1H-indol-6-ylmethoxy)pyridine-3-carboxamide N-[(1E)-4,5-dimethylhexa-1,3-dienyl]-2-(4-methoxyphenoxy)acetamide (2R)-2-[5-bromo-3,6-dideuterio-1-(4-cyanobenzoyl)-4-oxopyrrolo[3,2-c]pyridin-2-yl]propanoic acid 1-azidooxy-3-methylnaphthalene 6-azido-3,4-dimethyl-1-phenyltriazolo[4,5-c]pyridine 1-bromo-2-(3,4-dimethoxyphenyl)sulfanyl-3-ethenylbenzene 2-[(5-tert-butylthiophene-3-carbonyl)amino]octanoic acid 6-(2,4-difluorophenyl)-N-[1-(3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridazine-3-carboxamide 1-(4,6-dimethoxypyrimidin-2-yl)indazole 2-[4-chloro-3-[(2,4-difluorophenyl)methyl]phenoxy]-N-[3-[(E,3S)-3-hydroxy-5-oxopent-1-enyl]cyclobutyl]acetamide 3-[(2-cyanopyrimidin-5-yl)methylamino]-1-ethyl-N,4,5,6-tetrahydropyrazolo[3,4-b]pyrazine-7-carboxamide 1-amino-3-[5-fluoro-2,4-di(propan-2-yl)phenyl]urea 1-[2-(aminomethyl)phenyl]-N,3-dimethylpentan-1-amine;4-ethenylbenzaldehyde ethane;2-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-N-[(E)-(5-nitrothiophen-2-yl)methylideneamino]acetamide N-(2,3-dihydro-1H-inden-2-yl)-4-methylquinoline-2-carboxamide 3-[2-[(4,7-dimethyl-1H-indole-3-carbonyl)amino]ethylsulfanyl]-2,6-dihydropyrrol-1-ide;yttrium 4-(7-chloropyrazolo[1,5-a]pyridin-3-yl)-N-cyclopropyl-2-methoxy-6-morpholin-4-ylpyridine-3-carboxamide 6-[1-(aminomethyl)cyclopropyl]oxynaphthalene-2-carboxylic acid N-[6,7-dimethyl-3-(4-propanoylphenyl)thieno[2,3-c]pyridin-5-yl]acetamide;ethane N-(2-phenylpropyl)-N',N'-di(propan-2-yl)butanediamide [4-[6-(4,5-dimethylthiophen-2-yl)imidazo[1,2-a]pyridin-3-yl]phenyl]urea N-[3-(dimethylamino)propyl]-1-naphthalen-2-ylsulfonylpyrrole-3-carboxamide 2-[4-(benzenesulfonyl)phenyl]-N-hydroxyacetamide 1-(3,4-dimethylphenyl)-7,7a-dihydro-6H-benzimidazole 5-[(3R)-2,3-dihydro-1H-indene-5-carbonyl]-N-pyridin-4-yl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxamide 2-[2,5-difluoro-4-[3-[[4-(trifluoromethoxy)phenyl]carbamoylamino]phenyl]phenoxy]acetate 6-methyl-4H-indeno[1,2-c]pyridine 2-(3,5-dichlorophenyl)-4,5-dimethylpyrazolidin-3-one 5-(furan-2-yl)-N-propan-2-ylpyridine-3-carboxamide 4-tert-butyl-2-(5-tert-butylthiophen-2-yl)-5,6-dimethylpyridine;iridium 7-chloro-5-(4-chlorophenyl)-1-methyl-3H-1,4-benzodiazepin-2-one 3-(5-nitrofuran-2-yl)oxolane (3R)-1-[5-[4-chloro-2-fluoro-N-(2,2,2-trifluoroethyl)anilino]pyridin-2-yl]-N'-methanimidoylpyrrolidine-3-carboximidamide 4-(1,1-difluoroethyl)-2-[(3E,5Z)-hepta-1,3,5-trien-3-yl]quinoline N-[3,5-dichloro-4-(7-hydroxyquinolin-6-yl)oxyphenyl]-1-methyl-4-oxopyridine-3-carboxamide [(3S)-3-benzylpyrrolidin-1-yl]-(5-benzamidopyridin-2-yl)oxymethanolate 2-(ethylaminomethyl)-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one 1-(1,3-dioxolan-2-yl)-3-[4-[3-fluoro-5-methoxy-4-(4-propan-2-ylpiperazine-1-carbonyl)phenyl]phenyl]urea 1-(2,3,4a,5,7,8,8a-octahydropyrido[4,3-b][1,4]oxazin-6-yl)-3-[4-(benzenesulfonyl)phenyl]urea 2-[6-(3,4-dimethoxyphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridine-3-carboxylic acid 2-amino-6-(oxan-3-yloxy)benzaldehyde;2-phenyl-5,7-dihydrofuro[3,4-d]pyrimidine N-[(3R)-1,2-dimethylpyrrolidin-3-yl]-8-fluoroisoquinoline-3-carboxamide 1-[5-tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-diazourea N-(3-aminopropyl)-6-[6-(2,4-difluorophenyl)-5H-cyclopenta[b]pyridine-7-carbonyl]-4,4a,5,7,8,8a-hexahydropyrido[4,3-b][1,4]oxazin-3-amine;dihydrochloride N-[(3S,4R)-1-ethylsulfonylpiperidin-3-yl]pyrimidine-5-carboxamide 2-(6,7-dichloro-1H-indol-3-yl)-N-[1-(4-fluorocyclohexa-1,5-dien-1-yl)cyclopropyl]acetamide 1-methyl-3-[5-(2,4,6-trihydroxyphenyl)pentyl]thiourea 3-(2,6-dichlorophenyl)-7-[4-hydroxy-4-methyl-5-[(1R)-1-morpholin-4-ylethoxy]cyclohexa-1,5-dien-1-yl]-2H-1,3-benzoxazin-4-one 2,3-dihydro-1H-inden-4-yl(ethylidene)azanium [5-[(4-aminophenyl)sulfonylamino]-2-[(2,3-dichlorophenyl)sulfonylamino]phenoxy]boronic acid N-[2,3-bis(ethenyl)quinoxalin-6-yl]-4-methoxycyclohexane-1-carbothioamide 3-[5-[(2,4-dichlorophenyl)methyl]pyrimidin-1-ium-2-yl]pyrazolo[1,5-a]pyrimidine 4-[(2R)-3-methylbutan-2-yl]oxy-5,6,7,8-tetrahydropyrido[1,2-a]pyrimidine 1-(3,4-difluorophenyl)-7H-[1]benzofuro[2,3-c]carbazole 2-[3,5-dichloro-N-(4-hydroxybutyl)anilino]acetic acid 2-(5-fluoronaphthalen-1-yl)-3,4-dihydroisoquinolin-2-ium 4-N-[(E)-2-aminoethenyl]-5-chloro-2-N-[2-methoxy-3-(1,3-thiazol-2-ylcarbamoylsulfamoyl)phenyl]pyrimidine-2,4-diamine 4-bromo-2,6-ditert-butyl-3-ethoxyphenol 5-amino-6,7-dihydro-4H-[1,3]thiazolo[4,5-c]pyridine-2-carboxylic acid;3-(2-pyrrolidin-1-ylethoxy)naphthalene N-[1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethylideneamino]-2-methoxybenzamide 4-fluoro-N,N,5-trimethyl-2-[4-(trifluoromethyl)phenyl]cyclohexa-1,3-diene-1-carboxamide N-[1-[5-[2-[5-[5-(aminomethyl)pyridin-3-yl]-4H-pyrazolo[3,4-d]pyrimidin-3-yl]-2-cyanopropyl]pyridin-2-yl]piperidin-4-yl]formamide N-[4-fluoro-3-(2-pyrrolidin-1-ylethoxy)phenyl]-2,5-dimethyl-7-pyridin-4-ylpyrazolo[1,5-a]pyrimidine-6-carboxamide (6R,7S)-3-[2-acetamidoethyl(benzoyloxy)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid (2E,3Z)-6-(4-butylcyclohexa-1,5-dien-1-yl)oxy-2-ethylidene-8-oxoocta-3,7-dienenitrile;ethane [4-[5-(2,6-dichlorophenyl)-4,5-bis(ethylsulfanyl)-1H-imidazol-2-yl]piperidin-1-yl]-(furan-2-yl)methanone (1S)-2,2,2-trifluoro-1-(6-nitronaphthalen-2-yl)ethanamine (3S,4R)-1-[5-chloro-6-oxo-2-[[(2S,4R)-2-phenylpiperidin-4-yl]amino]pyrimidin-1-yl]-3-fluoropiperidine-4-carboxylic acid N-[5,6-dichloro-2-(3,4-dihydroxybutyl)-1H-indol-7-yl]-4-fluorobenzamide N-[5-(3,4-dichlorophenyl)sulfonyl-1H-indazol-3-yl]-2-piperidin-1-ylbenzamide 2-azido-1,3-difluoro-5-(1,1,2,2-tetrafluoroethoxy)benzene N-[4-[2-(oxan-4-yl)ethoxy]cyclohexa-1,3-dien-1-yl]-6-oxo-3-phenyl-1H-pyridazine-5-carboxamide 2-amino-3,3-dimethyl-N-[(E)-1-(2-oxoethoxy)but-2-en-2-yl]butanamide;N-[3-[4-[[2-hydroxyethyl(oxetan-3-yl)carbamoyl]amino]phenyl]propyl]formamide 4-[2,5-bis(trifluoromethyl)phenyl]-1-tert-butylpyrazole;ethane 2-cyclohepta-1,3,6-trien-1-yl-N'-phenylethanedithioamide (3R)-N',4-diphenyl-2-[(1S)-1-phenylethyl]butanediamide N-[(E)-3-cyclobutylprop-2-enyl]-5-[3-[7-[(1Z)-1-ethylideneamino]-5H-pyrazolo[4,3-b]pyridin-4-yl]-5-methoxyphenyl]pentanamide 6,7-dimethoxy-N'-[3-(4-methylpiperazin-1-yl)phenyl]quinazoline-2-carboximidamide (2R)-4-fluoro-N'-hydroxy-3-[[1-(5-methylpyrimidin-2-yl)piperidine-4-carbonyl]amino]-2-propan-2-yloxybutanehydrazide 6-chloro-N-(oxan-3-yl)-1H-pyrazolo[4,3-c]pyridine-3-carboxamide N-[(3,4-dichlorophenyl)methyl]-5-ethyl-6-[(2R)-1-(hydroxyamino)-1-oxopropan-2-yl]oxypyridine-3-carboxamide 5-(methoxymethyl)-3-[2-[5-(1H-pyrrolo[2,3-b]pyridin-4-ylamino)pentanoyl]phenyl]imidazolidine-2,4-dione N-[4-(3-cyano-1,2-oxazol-5-yl)pyridin-2-yl]-6-methoxy-N'-methanimidoyl-7H-cyclohepta[b]thiophene-2-carboximidamide 4-[5,8-difluoro-7-(3-hydroxypropyl)-2,3,4,9-tetrahydro-1H-carbazole-3-carbonyl]piperazine-1-sulfonamide N-butyl-2,3-dibromo-5,6-dimethoxybenzamide 5-ethyl-2,3-bis[2-(4-methoxyphenyl)ethynyl]-6-propan-2-ylidenecyclohexa-1,3-diene N-[3-(dimethylamino)-2,4-dioxocyclobutyl]benzenesulfonamide N-methyl-3-(propanoylamino)benzenesulfonamide 5-(methoxymethyl)-6,10-dioxapentacyclo[12.7.0.02,11.04,9.015,20]henicosa-1(14),2(11),3,8,12,15,17,19-octaene [(2R)-4-[3,5-difluoro-4-(trifluoromethyl)phenyl]oxan-2-yl]methanol 1-methyl-4-[(3Z)-3,6,7,11b-tetrahydro-2H-[1]benzothiolo[3,2-a]carbazol-12-yl]piperazine 6-bromo-N,N-dibutyl-1H-benzimidazole-2-sulfonamide 2-(2,5-dichloro-N-phenacylanilino)acetic acid 7-[4-fluoro-2-(4-methylphenyl)pyrrolidine-1-carbonyl]-8,9b-dihydrodibenzofuran-3-carboxylic acid (3S)-1-(5-chloropyridin-2-yl)pyrrolidine-3-carboxamide 3-(4-ethoxyphenyl)-6,7-dimethyl-2-[3-(trifluoromethyl)phenyl]imidazo[1,2-a]pyrimidine 5-azido-1-benzyl-2,3-dihydroindole 3-[4-[(1S)-2,3-dimethylcyclopentyl]phenyl]pyridine 7-(3,4-dichlorophenyl)-5-methyl-6-[2-oxo-2-(1,2,4-triazol-1-yl)acetyl]-N-(4-propanoylphenyl)imidazo[1,2-a]pyrimidine-3-carboxamide 1-N,3-N-bis[(Z)-(2,5-dimethyl-1H-pyrrol-3-yl)methylideneamino]benzene-1,3-disulfonamide 3-(2,4-dichlorophenyl)cyclohexan-1-one 3-[[2-amino-5-[[4-(azetidine-1-carbonyl)cyclohexylidene]methyl]-6H-1,3,4-thiadiazin-5-yl]oxy]-N'-ethylbenzenecarboximidamide 5-chloro-2-(1,6-dimethylpiperidin-3-yl)oxypyrimidine N-[(1S)-3-(4-cyanophenyl)cyclopentyl]cyclopropanecarboxamide 1-(4-bromophenyl)-4-(N'-ethylcarbamimidoyl)-3,5-dihydropyrido[2,3-e][1,4]thiazine-2-thione N-methyl-4-[(5-methylthiophene-2-carbonyl)amino]thiophene-3-carboxamide 2-methyl-N-[4-(2-methylimidazol-1-yl)butan-2-ylidene]propanethioamide 3-methyl-2,6,7,8-tetrahydrocyclohepta[d]pyrimidin-4-one 5-chloro-4-[(5S)-6,9-dimethyl-7-oxo-6,8-dihydropyrimido[4,5-b]indol-5-yl]-N-propan-2-ylpyridine-3-carboxamide N-ethyl-5-[(6-methoxynaphthalen-2-yl)sulfamoyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide 2-(7,8-dimethoxyquinazolin-4-yl)cyclohexan-1-ol 1-(1-cyclopropyltetrazol-5-yl)-1,3,4,9-tetrahydropyrido[3,4-b]indole N'-[(E)-1,2-diphenylpropylideneamino]-N-ethylpropane-1,3-diamine N-[(3,5-dimethoxyphenyl)methyl]-4-[4-ethoxy-2-(pyridin-4-ylamino)pyrimidin-5-yl]benzamide 3-(4-methoxyphenyl)-2,3-dihydropyrazolo[5,1-b]quinazoline 1-[2,5-dimethyl-4-(1,3-oxazol-2-yl)phenyl]ethanone 1-(3,4-dihydronaphthalene-1-carbonyl)piperidine-2-carboxylic acid 2-amino-4-(2,3,4,5,6-pentafluorophenyl)-1H-pyrimidin-6-one [(3S)-3-methyl-4-[2-methylsulfonyl-6-[(1R)-1,2,3,4-tetrahydroisoquinolin-1-yl]pyrimidin-4-yl]morpholin-2-ylidene]methanol 4-N-[1-(benzylamino)-3-(4,5-dichlorocyclohexa-1,5-dien-1-yl)propan-2-yl]quinazoline-2,4-diamine 6-[(4S)-2,7-dimethyl-3,4-dihydro-1H-isoquinolin-4-yl]-2H-triazolo[4,5-b]pyridin-5-amine N-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-5-phenylpentanamide (1S,2R)-2-[4-(azidomethyl)phenyl]cyclohexan-1-ol 1-N,3-N-diamino-5-cyclopropylsulfanylbenzene-1,2,3-triamine;ethane;(4R)-1,3,4,9-tetramethylfluorene 5-(5,7-dimethoxyquinazolin-4-yl)sulfanyl-1H-pyrazole-3-carboxylic acid 6-[2,5-dimethyl-1-(6-morpholin-4-ylpyridazine-3-carbonyl)pyrrol-3-yl]hexanoic acid 2-(N-cyclohexyl-2,6-difluoroanilino)acetamide N-(3-bromophenyl)-6-[4-[1-cyclohexylpropan-2-yl(methyl)amino]benzoyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-2-carboxamide 3,5-dimethyl-2-(9H-fluoren-1-yl)phenol 3-hydroxy-5-phenylmethoxycyclohexan-1-one 2-[[4-[[3,5-dimethyl-1-(2-oxo-3H-1,3,4-thiadiazol-5-yl)pyrazol-4-yl]diazenyl]benzoyl]amino]butanoic acid 4-fluoro-N-[1-(pyridine-2-carbonyl)cyclobutyl]benzamide N-[6-(hydroxymethyl)pyridin-2-yl]-3,5-bis[[4-[[methyl(2-oxoethylsulfanyl)amino]methoxymethyl]phenyl]methyl]benzamide 3-chloro-5,6-dihydrothieno[3,2-b]thiophene;ethane 4-[3-(ethoxymethyl)morpholine-4-carbonyl]benzoic acid 2-[3-(benzoylsulfamoyl)benzoyl]oxyacetate 2-bromo-N-(2,6-difluorophenyl)-N-(4-hydroxybutyl)benzamide [(2R,4S)-2-[5-[3,5-bis(trifluoromethyl)phenyl]-1H-imidazol-2-yl]-1-methylpiperidin-4-yl]carbamic acid;hydrochloride [4-(1,1,2,3,3,3-hexafluoropropyl)phenyl]boronic acid 2-(3,5-dichlorophenyl)sulfonyl-7-ethoxy-1H-quinazoline-2,4-diamine 2-[[(1R,3R)-2,2-difluorocyclopropyl]methoxy]-5-[5-(4-piperidin-4-ylphenyl)pyridin-3-yl]benzamide 5-(4,6-dimethylpyrimidin-2-yl)-2,7-dimethylimidazo[1,2-a]pyridine 2-[(6-oxo-4-propyl-1H-pyrimidin-2-yl)sulfanyl]pentanoic acid 6-[(3-chloro-2-fluorophenyl)methyl]-7H-pyrrolo[3,4-b]pyridine [5-(1,3-benzodioxol-4-ylmethoxy)-6-fluoronaphthalen-2-yl]methanimine 1-[2,6-di(propan-2-yl)phenyl]-3-ethyl-4-methylideneimidazolidine;4-methoxybenzene-5-ide;uranium(2+) (2Z,4E)-5-[2-amino-6-chloro-3-methyl-7-(propan-2-ylsulfanylmethyl)phenyl]penta-2,4-dienoic acid 2-methyl-3-phenyl-4H-chromeno[1,2-c]pyrazol-7-one 3-[2,5-dioxo-1-[4-(trifluoromethyl)phenyl]pyrrol-3-yl]-N-(5,6,7,8-tetrahydronaphthalen-2-ylsulfamoyl)propanamide 2-[N-(4-bromobutan-2-yl)anilino]ethanol 2-amino-4,4-diethoxy-3H-pyrano[3,2-g]chromene-5,10b-dione 4-[(E)-2-(4-bromophenyl)ethenyl]phenol 1-[4-(4,5,6,8,10-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-3-yl)piperidin-1-yl]prop-2-yn-1-one ethane;N-methylformamide;(3E,5Z)-4-(7-morpholin-4-ylquinazolin-4-yl)octa-1,3,5-trien-2-ol 2-(N-butyl-2,4,6-trichloroanilino)acetonitrile N-[(Z)-2-azidoethenyl]-5,6-dimethoxy-1H-benzimidazole-2-sulfonamide 2-[(2E,4Z)-hepta-2,4-dien-6-yn-3-yl]oxy-N-phenylacetamide 4-bromo-N'-[1-(3-hydroxyphenyl)ethyl]pyridine-2-carboximidamide (2Z)-N,3-bis(ethenyl)-5-methoxy-N-[1-(6-methylpyridin-3-yl)ethenyl]penta-2,4-dien-2-amine ethane;1-(3-hydroxyazetidin-1-yl)propan-1-one;2-[5-methoxy-8-methyl-7-(trifluoromethyl)quinolin-4-yl]acetic acid N-[[2,4-dimethyl-5-(trifluoromethyl)pyrazol-3-yl]methyl]spiro[1,2-dihydroindene-3,4'-oxane]-1'-carboxamide 4-[3-(2-hydroxyethyl)-1,2-dihydroimidazol-5-yl]benzonitrile 3-bromo-2,5,6-trimethylaniline;ethane N-(8,9-dihydropyrido[3,4-b]indol-1-ylmethyl)carbamate [5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]carbamoylazanide 3-[5-bromo-2-(4-fluorobenzoyl)phenyl]propanenitrile N'-[5-chloro-2-methyl-4-(3-oxomorpholin-4-yl)phenyl]oxamide 4-[[(5Z)-5-[[3,5-dibromo-2-(trifluoromethoxy)phenyl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoic acid 2-[4-(4-methoxy-7H-pyrrolo[3,2-d]pyrimidin-6-yl)phenyl]-N-(2,5,6-trifluoropyridin-3-yl)acetamide 2-[(3,5-dimethylphenyl)methylsulfanyl]-N-[(4,6-dioxocyclohexa-1,4-dien-1-yl)methyl]acetamide (3R)-N'-[2,6-dichloro-4-[1-[4-fluoro-3-(trifluoromethyl)phenyl]-5-oxo-4H-pyrazol-4-yl]phenyl]-2-hydroxy-3-propan-2-ylbutanediamide N-[(E)-(5-bromo-2,4-dihydroxyphenyl)methylideneamino]-3-cyanobenzamide 2-(3,5-dimethoxyphenyl)-6-[(4-hydroxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 6-[1,2-difluoro-2-(4-pentylphenyl)ethenyl]-2,3-dihydrothieno[3,4-b][1,4]dioxine [3-amino-5-(trifluoromethyl)phenyl]sulfonyl-methylideneazanium 3-methylsulfanyl-2-[4-(trifluoromethoxy)phenyl]prop-1-ene-1,1-diol (1E,4Z)-2-[5-bromo-2-oxo-3-[2-oxo-3-(2H-tetrazol-5-yl)butyl]sulfanylpyrimidin-6-yl]-N'-methoxyethenedithioamide (2R)-3-acetyl-4-[3-(4-hydroxyphenyl)propanoylamino]-N-(2H-tetrazol-5-yl)pyrrolidine-2-carboxamide 1-[(6-chloropyridine-3-carbonyl)amino]-N,4-dimethylpyrrolidine-2-carboxamide (2R)-4,4-difluoro-N-[5-fluoro-6-(5-methylpyrazolo[3,4-b]pyridin-1-yl)pyridin-3-yl]-2-phenylpiperidine-1-carboxamide (2S)-3,3-dimethyl-4-oxo-N-[(1R)-2-pyridin-3-ylcyclohexyl]pyrrolidine-2-carboxamide (2R)-3,6-dimethyl-4-[5-(1,8-naphthyridin-2-ylamino)pentanoyl]piperazine-2-carboxylic acid 2-[(2-fluorophenyl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-quinazolin-4-one [(Z)-5-amino-2,4-dimethylpent-4-enoyl]-phenylcyanamide 3-[(5S)-5-(2,4-dichlorophenyl)-5-(3-methylphenyl)-6H-1,2,4-triazin-3-yl]cyclobutan-1-one 3-(6,11-dihydrobenzo[c][1]benzoxepine-2-carbonyl)thiophene-2-carboxylic acid 1-cyclohexa-2,4-dien-1-yl-3-[2,6-difluoro-4-(1H-pyrazol-5-yl)phenyl]urea 4-(2,6-dimethylphenyl)-N'-hydroxypyridine-3-carboximidamide N-[1-(1H-indole-2-carbonyl)piperidin-3-yl]benzamide N-benzyl-2,2-dimethyl-7-[(1S)-2-oxocyclobutyl]-4,5,6,8-tetrahydro-3H-pyrido[3,4-d]pyrimidine-5-carboxamide 2-(azepan-1-yl)benzenecarbothioamide N-[(3,4-difluorophenyl)methyl]-8-hydroxy-7,9,12-trioxo-1,10-diazatricyclo[6.2.0.04,11]deca-2,4,6,8-tetraene-3-carboxamide 5-[(6-cyclopropylsulfonylpyridin-3-yl)methoxy]-3,4-dihydro-2H-chromene-8-carboxylic acid 1,2-bis[(E)-3,5-dimethylhex-2-enoxy]benzene (2Z,3Z)-N-[1-phenylethenyl]-N-propan-2-ylidenehexa-2,5-dienamide 2-[[4-(1,1,1,3,3,3-hexafluoropropan-2-yl)phenoxy]methyl]quinoline 6-(9-azido-4-methylfluoren-3-yl)pyridine-3-carbonitrile 4-[3-fluoro-5-(hydroxymethyl)phenyl]iminobutanoic acid 2-(2,3-dihydropyridin-4-yl)-1-[(E)-3-methoxyprop-1-enyl]-5H-thieno[3,2-d]pyrimidine-2,4-diamine N-[4-(2,3-dihydro-1H-inden-5-yl)-1,3-thiazol-2-yl]-4-methylsulfonylbenzamide 1-[3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)phenyl]pyrrolidine-2,5-dione 1-azidooxy-2,3-dimethyl-4-(trifluoromethoxy)benzene [(5Z)-2,3-bis(ethenyl)hepta-1,5-dienoxy]benzene [(3R)-4-[bis(4-methoxyphenyl)methyl]piperidin-3-yl]methanol 2-(3,6-dihydro-2H-pyridin-1-ylsulfonyl)-N-methoxy-1H-indole-7-carboxamide 3-(benzenesulfonyl)-4-methoxybenzonitrile 2-(3,5-dimethylphenyl)-1H-indole N-benzyl-2-ethoxy-4,6-dimethyl-3,5-dinitroaniline N-[4-(2-aminopyrimidin-5-yl)-1,3-thiazol-2-yl]-4-azidobutanamide N-[(Z)-1H-indol-3-ylmethylideneamino]-2-(naphthalen-2-ylamino)acetamide ethene;2-ethenyl-4,7-dimethoxy-1H-indole 2-[1,3-dimethyl-5-(4-propan-2-ylpiperazin-1-yl)indol-7-yl]acetamide (Z)-2,3-diamino-1-[7-bromo-6-methylidene-4-[(Z)-propan-2-yloxyiminomethyl]phthalazin-1-yl]but-2-en-1-one 2-[3-(2,4-difluorophenyl)-1H-pyrazole-5-carbonyl]-N,N,7-trimethyl-3,4,6,7,8,9a-hexahydro-1H-pyrrolo[1,2-a]pyrazine-6-carboxamide 2,6-dimethyl-5-[(3-phenylpyrrolidin-1-yl)methyl]pyrazine 4-(1H-indol-5-yl)-3,8-dihydropyrimido[4,5-d]pyrimidine-2,5,7-trithione 5-azido-2-(4-methylphenoxy)pyrimidine (5S)-2-(4-carbamoylpiperidin-1-yl)-N-(4-chlorophenyl)-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide 4-[[1-(5-chloropyridine-2-carbonyl)piperidin-3-yl]methoxy]-2-fluoro-N-(4,4,4-trifluorobutanoyl)benzamide N-[(2,3-dimethoxyphenyl)methyl]-N-(2-methylpropyl)but-2-ynamide 1-azidosulfonyloxy-2,3-dihydroindole (3R)-N-[2-(2,4-difluorophenyl)ethyl]-9-[(E)-5-hydroxypent-2-enoyl]-6-methoxy-1,2,3,4-tetrahydrocarbazole-3-carboxamide 1-(4-azidophenyl)sulfanyl-N,N-dimethylpropan-2-amine (5-fluoro-2,3-dimethylindol-1-yl)-[4-[6-[(2E,4Z)-hepta-2,4-dien-6-yn-3-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone 1-benzylpiperidin-2-one;N,N-dimethylethanamine N-[2,3-bis(ethenyl)phenyl]formamide N-benzyl-2-fluoro-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide;ethane 3-methyl-4-(5-piperidin-1-ylpentoxy)aniline 4-[4-(N-(2,5-dichlorophenyl)-3-nitroanilino)phenyl]-N-(oxolan-2-ylmethyl)-1,3-thiazol-2-amine 2-[4-(6,7-dimethoxyquinazolin-4-yl)piperazin-1-yl]-N-[(Z)-propylideneamino]pyrimidine-5-carboxamide N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide N'-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(2,5-difluorophenyl)pyridine-2-carboximidamide 1-[(3R)-3-[2,6-dimethyl-4-[5-methylsulfonyl-1-[[4-(trifluoromethyl)phenyl]methyl]indazol-7-yl]phenoxy]butanoyl]-N-hydroxypiperidine-3-carboxamide 3-[1-amino-2-(4-tert-butylphenyl)ethenoxy]cyclohexa-2,5-diene-1,4-dione 1-[2,4-bis(trifluoromethyl)phenyl]-N-ethylpentan-3-imine (5Z)-5-[[3,5-dibromo-4-[2-nitro-4-(trifluoromethoxy)phenoxy]phenyl]methylidene]imidazolidine-2,4-dione 5-(2,3-dimethylbutanoylamino)-N-[(4S,5R)-3-methyl-6-oxo-1-phenyl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-5-yl]thiophene-2-carboxamide 2-[2,4-bis(ethenyl)phenyl]-3H-pyrido[4,3-d]pyrimidin-4-one 2-[3,5-bis(trifluoromethyl)phenyl]-2-cyanopropanamide 5-tert-butyl-2-[2-(2,6-difluorophenyl)-1H-inden-4-yl]oxan-4-ol 4-amino-6-[(3,5-dibromo-2-propoxyphenyl)methyl]-3-sulfanylidene-2H-1,2,4-triazin-5-one 1-methyl-3-[[4-(trifluoromethyl)anilino]methyl]pyrrolidine-2,5-dione 6-[6-(dimethylamino)pyridin-3-yl]-2-N,4-N,4-triethyl-5H-1,3-diazepine-2,4-diamine 2-[1,1-di(carbazol-9-yl)ethenyl]benzonitrile 3-[4-chloro-2-(5-methylbenzotriazol-2-yl)phenoxy]-N,N-dimethylpropan-1-amine 4-tert-butyl-2,6-bis(4-propan-2-ylphenoxy)aniline 5-(3,4-dichlorophenyl)sulfinyl-N'-hydroxypyridine-2-carboximidamide 4-(5-bromopyridin-2-yl)but-3-ynamide (2S)-N'-hydroxy-3-[4-(2-morpholin-4-ylethoxymethyl)phenyl]sulfonylspiro[1,4-dihydroquinoxaline-2,4'-piperidine]-5-carboximidamide;hydrochloride (5-chloro-1,2-benzoxazol-3-yl)-[4-[5-(methoxymethoxy)-7H-cyclopenta[b]pyridin-6-yl]phenyl]methanone N-[2,6-dichloro-4-(trifluoromethyl)phenyl]-1H-indole-3-carboxamide 4-[(3,3-dimethyl-1-propanoylpiperidin-4-ylidene)amino]benzonitrile 4-[2-(diethylamino)ethoxy]quinoline-3-carboxamide 6-[(E)-2-(4-chlorophenyl)ethenyl]sulfonyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 4-(3,5-dimethylphenyl)benzoate 5-(3,3a,4,6,7,7a-hexahydro-1H-pyrano[4,3-c]pyrrol-2-yl)sulfonylpyridine-2-carbonitrile 4-[1-(3,4-dimethoxyphenyl)ethyl]-2-ethylmorpholine;ethane 1-(2,3-dihydroindol-1-yl)pentan-3-one;ethane N-(3,4-dimethoxyphenyl)-6-ethoxy-2-[2-(furan-2-ylmethylsulfanyl)ethylamino]pyrimidine-5-carboxamide 3-[5-[6-(difluoromethyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]iminobutanamide 2-[3,5-difluoro-4-[1-(4-methylphenyl)ethoxy]phenyl]-6-ethoxy-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 4-[(6-oxocyclohexa-2,4-dien-1-yl)amino]-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile 5-tert-butyl-N'-[2-(dimethylamino)ethyl]-1,3,4-oxadiazol-2-amine (5Z)-5-[[1-[2,4-bis(trifluoromethyl)phenyl]cyclopropyl]methylidene]imidazolidine-2,4-dione 2-cyclohexylacetate;3,4,5-trimethoxybenzoate 2,3-ditert-butyl-4-methoxyphenol 2-chloro-N-(5-methylpyridin-3-yl)propanamide 3-hydroxy-1',1'-dimethylspiro[4H-quinoxaline-2,4'-piperidine] N-[6-[4-(dimethylamino)piperidine-1-carbonyl]-3,5-dihydro-2H-pyrrolo[3,2-f]quinazolin-1-ylidene]benzenesulfonamide 4-[6-[2,5-difluoro-4-(trifluoromethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-sulfonamide 3-[(2R)-3,4-dimethylpentan-2-yl]oxy-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 2-chloro-4-[1-(3,5-dichlorophenyl)ethyl]-6-methoxyaniline 5-(2,6-difluoro-3,5-dimethoxyphenyl)-N-[4-[ethyl-[2-[methyl(pent-1-en-3-ylamino)amino]ethyl]amino]pyridin-3-yl]-8-oxopyrido[2,3-d]pyrimidine-7-carboxamide 5-(4-bromo-2,5-dimethylphenyl)-3H-1,3,4-oxadiazol-2-one 5-[2,3-dihydroxypropyl(1,1,1,2,3,3,3-heptafluoropropan-2-yl)amino]naphthalene-2-sulfonic acid 1-(2,5-dimethylphenyl)-3,4-dihydroisoquinoline;hydrochloride (5Z)-2-(4-chlorophenyl)imino-5-[(3-hydroxynaphthalen-2-yl)methylidene]-1,3-thiazolidin-4-one 2-[[4,5-bis(ethenyl)-6-methylidenepyran-2-carbonyl]amino]acetic acid;1H-imidazole (5R)-2-(4-ethylphenyl)imino-5-[(3-methoxynaphthalen-2-yl)methyl]-1,3-thiazolidin-4-one 2-[3,5-diamino-6-(4-methoxyphenyl)pyridazin-4-yl]phenol (2E)-N'-[(E,3R)-4-cyclohexyl-5-phenylpent-1-en-3-yl]-2-hydrazinylideneethanimidamide N-[6-(1H-indol-4-yl)imidazo[1,2-a]pyrazin-8-yl]methanimine 2-(4,5-dimethylthiophene-3-carbonyl)-9H-fluoren-1-ol 2-(4-bromophenyl)-1,5-di(propanoyl)piperazine 2-[(2S)-1-benzylsulfonylpyrrolidin-2-yl]-N,N-diethyl-3H-benzimidazole-5-carboxamide 2-amino-5-[4-methyl-3-[(1E,3Z)-penta-1,3-dienoxy]phenyl]pyridine-3-carboxamide 3-methyl-7-(4,4,5,5-tetramethyloxaborolan-2-yl)dibenzofuran N-[(1S)-6-chloro-5,7-difluoro-2,3-dihydro-1H-inden-1-yl]-1-methylpyrazole-4-carboxamide [6-(triazolo[1,5-a]pyridin-7-ylmethoxy)-3,4-dihydro-2H-chromen-4-yl]urea 5-[[(5S)-2-oxo-5-phenylcyclopentyl]amino]pentanoic acid 4-amino-N'-(4,4,4-trifluorobutyl)pyridine-3-carboximidamide (E)-2,4-dimethylhept-3-enal;ethane;N-methoxy-N,5-dipropyl-1H-pyrrolo[2,3-c]pyridine-2-carboxamide 1-(3,4-difluorophenyl)-N-[(2R)-2-methoxybutyl]-5-[5-(1H-pyrazol-4-yl)thiophen-2-yl]pyrazole-3-carboxamide 4-[2-(1,3-dioxolan-2-yl)ethoxymethyl]benzamide 4-[(3R,5S)-5-methylpiperidin-3-yl]sulfonylbenzoic acid 2,3-bis(methoxycarbonyl)-4-oxo-1H-quinoline-7-carboxylic acid 5-[4-(3-azido-1,2-oxazol-5-yl)phenyl]-2-methoxyaniline 3-[4-fluoro-N-(2-oxopropyl)anilino]propanoic acid 4-(1,3-dioxol-2-yl)benzenesulfinate 2-(3,4-difluorophenyl)-7-pentylphenanthrene 6-(3,4-dimethylcyclohexa-2,4-dien-1-ylidene)-7H-benzo[c]carbazole 5-(2,3-difluorophenyl)-4-iminocyclohexan-1-amine 2-amino-4-[4-(cyclopropylmethoxy)phenyl]-6-ethoxy-4H-pyran-3,5-dicarbonitrile N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4,5-dihydro-1,3-thiazole-4-carboxamide 1-[3,5-dichloro-4-(1H-pyrrol-2-yl)phenyl]pyrrole [(Z)-2,3,5,6-tetraethylhept-1-enoxy]methylbenzene (2E,5S)-2-[(Z)-1-naphthalen-2-ylethylidenehydrazinylidene]-5-phenacyl-1,3-thiazolidin-4-one 2-[[1-(3,4-dichlorophenyl)-5-methylpyrazol-3-yl]amino]ethanol;hydrochloride 7-tert-butyl-2,5-dimethoxybenzenesulfonic acid 3,5-dichloro-N-[(2S)-1-hydroxybutan-2-yl]pyridine-4-carboxamide (Z)-N',N'-diphenylbut-2-enediamide 3-(2-oxoazepan-1-yl)-N-[[4-(trifluoromethoxy)phenyl]methylideneamino]benzamide 4-azido-2,5-dichloro-N,N,3,6-tetramethylaniline 3-[1-(1,2,4-triazol-1-yl)ethyl]cyclopentan-1-one N-[2-(dimethylamino)ethyl]-3-(trifluoromethoxy)benzamide 4-N,4-N-bis(difluoromethyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 1-(3,5-dichlorophenyl)-6-ethyl-7-methoxy-N-(2H-tetrazol-5-ylmethyl)benzimidazole-2-carboxamide;ethane 2-[5-(3,4,6,7,8,9-hexahydropyrido[1,2-a]pyrazine-1-carbonyl)-1H-indol-2-yl]-2-oxoacetamide (4R)-1,3-dimethyl-4-thiophen-2-yl-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one [2-(1,3-dimethylpyrazol-4-yl)piperidin-1-yl]-[5-methoxy-4-(2-pyrrolidin-1-ylethoxy)pyridin-2-yl]methanone N-[3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carbonyl)phenyl]acetamide 2-(diethylamino)-1,3-diethylbenzimidazol-3-ium-5-sulfonic acid N-[2,5-difluoro-4-(1,1,3,3-tetramethyl-2H-inden-5-yl)phenyl]acetamide (2E)-1-cyano-3,3-dimethyl-2-[[4-[6-(trifluoromethyl)pyrimidin-4-yl]sulfanylphenyl]hydrazinylidene]butan-1-olate (3S,4S)-2-[(4-methoxyphenyl)sulfonylamino]-N-(5-methylpyrazin-2-yl)oxane-3-carboxamide 4-(benzylideneamino)-1-ethenylpiperidine-4,5-diamine 2-[1,3-dihydroisoindole-2-carbonyl(propyl)amino]-N-pyridin-3-ylacetamide 2,2-dimethylpentane;[3-fluoro-4-(2-methylsulfanylpropan-2-yl)phenyl]methanol (4S)-3,7,9-trihydroxy-6-methyl-2-(1H-pyrrolo[3,2-b]pyridin-5-yloxycarbonylamino)-1,8-naphthyridine-4-carboxylic acid (E)-N-[2-cyclopropyl-5-fluoro-4-[4-[1-[(2R,5S)-5-methyloxolan-2-yl]ethoxy]phenyl]sulfonylphenyl]hexanamide (2S,3S)-3-ethyl-N-[[4-(1H-imidazol-5-ylmethoxy)phenyl]methyl]oxolan-2-amine 4-(4,7-dimethylundecan-4-yl)phenol 4-azidosulfanyl-6,7,8-trimethoxyquinazoline 4-ethyl-2,5-diiodo-N'-(4-nitrophenyl)benzenecarboximidamide 2-(methylsulfonylamino)-6-[4-[1-(piperidine-3-carbonyl)piperidin-4-yl]oxyphenyl]pyridine-3-carboxamide;hydrochloride N-ethyl-4-methoxy-3-[[(1S,2S)-1-phenylpropan-2-yl]sulfamoylmethyl]benzamide N-(2,3,4,5,6-pentadeuteriophenyl)-2-piperazin-1-ylethanimine 5-(3,4-dichlorophenyl)sulfanyl-2-pyridin-3-yl-1,3-dihydro-1,2,4-triazole 4-[(Z)-(2,3-dihydroxyphenyl)methylideneamino]piperazine-1-carboxamide 6-[2-(4-fluorophenyl)acetyl]-N-(pyridin-3-ylmethyl)-6-azaspiro[3.4]octane-8-carboxamide 1-(2,3-dihydro-1H-indene-4-carbonyl)-4-hydroxypiperidine-2-carboxylic acid (3E,5Z)-2,3-dimethylhepta-1,3,5-triene;[4-[2-[[(1R)-2-ethoxycyclohexa-2,4-dien-1-yl]amino]pyrimidin-5-yl]phenyl]-morpholin-4-ylmethanone 3-bromo-5,7-dichlorochromen-4-one 5-[4-[6-(2,6-difluorophenyl)pyridine-3-carbonyl]piperazin-1-yl]-6H-phenanthridin-7-one 2-[3,5-dibromo-4-[(3-oxocyclobutyl)amino]phenyl]acetonitrile 4-(N-hexadecyl-2,4-dinitroanilino)butan-1-ol 1-[(2R,3S)-3-hydroxy-2-phenyloxiran-2-yl]pentan-2-one 2-(4-chlorophenyl)-1-[3-[4,5-dimethyl-6-[(Z)-prop-1-enyl]pyridin-3-yl]pyrrolidin-1-yl]ethanone 6-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4,5,7-tetrahydrothieno[2,3-c]pyridin-6-ium-2-one 6-(4-fluorophenyl)-5,6-dihydro-1H-pyrimidine-2,4-dione 4-(1,3-benzodioxol-5-ylmethyl)-N-cyclobutyl-1,3-thiazolidin-2-imine 5-ethyl-3,4-dinitro-1H-pyrrole-2-carboxylic acid 4-N-methylsulfanyl-1-N-[(E)-2-methylpropylideneamino]benzene-1,3-diamine 4-[3-[(dimethylamino)methyl]phenyl]-N-(1,2-oxazol-5-ylsulfonyl)butanamide 4-(4-azidopiperidin-1-yl)sulfonyl-N-(1,3-benzodioxol-5-ylmethyl)aniline 4-[4-methoxycarbonyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperazine-1-carboxylic acid 2,3-dimethyl-1H-indole;formaldehyde;methane 1-(4-aminophenyl)-6,7-dihydro-5H-cyclopenta[c]pyridine-4-carboxamide 4-[(Z)-(3,5-dichlorophenyl)methylideneamino]oxybenzonitrile (3-azido-2H-1,4-benzodioxin-5-yl)-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)methanone 2-[4-(4,4-dimethylpiperidin-1-yl)-5-[3-fluoro-5-(trifluoromethoxy)phenyl]-2-methylpyridin-3-yl]-6-(hydroxymethyl)oxan-4-ol 1-(cyclopropylmethylamino)-3-[3-[4-(trifluoromethoxy)phenoxy]propyl]thiourea 1-[[3-(2,6-difluorophenyl)pyrazol-1-yl]methoxy]propan-2-ol N-(6,7-dihydro-4H-pyrano[3,4-d][1,2]oxazol-3-ylmethyl)formamide;N'-hydroxy-1,2-benzothiazole-3-carboximidamide N-(2,6-dimethylphenyl)-3-(2-ethoxy-4-methoxyphenyl)sulfanylpropanamide N-(4-chlorophenyl)-2,4-dihydroxybenzenecarbothioamide N-(2,4-difluorophenyl)-5-methyl-1-[[2-oxo-8-[(1-phenylpyrazole-3-carbonyl)amino]-3H-imidazo[1,2-a]pyridin-3-yl]methyl]pyrazole-4-carboxamide (2S)-3-[2-[4-[3,5-difluoro-2-(3-methyl-1H-indol-2-yl)phenoxy]butoxy]phenyl]-2-ethoxypropanoic acid 4-N-cyclopropyl-2,5-difluorobenzene-1,4-disulfonamide N-[4,7-dichloro-2-[5-chloro-3-[(3S)-3-ethylpyrrolidine-1-carbonyl]indol-1-yl]quinolin-6-yl]methanesulfonamide N-[1-(6-chloropyridine-3-carbonyl)piperidin-4-yl]-1,2-dimethoxybenzimidazole-5-carboxamide N-[(2-hydroxyphenyl)methylideneamino]-7-oxoheptanamide [(4-chlorophenyl)methylamino]-diphenoxyphosphanium N-[5-(2,6-dichlorophenyl)pyridin-2-yl]-3-(ethylideneamino)-4-imino-1-methanimidoylpyridine-2-carboxamide N-butyl-2,3,4,5,6-pentadeuterio-7-[3-(trifluoromethoxy)phenyl]-8H-carbazole-1-carboxamide 3-[(3R)-7,10-difluoro-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-4-[2-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole-5-thione 1-[3,5-bis(trifluoromethyl)phenyl]-N-[(E)-3-methoxyprop-1-enyl]ethanimine 2-[4-chloro-N-(3,5-dichlorophenyl)anilino]acetamide 5-bromo-N-methyl-1H-indole-2-carboxamide 2-[(E)-2-aminoethenyl]-N-(3,5-dimethoxyphenyl)-1H-pyrimidin-6-imine 6-[3,4-difluoro-2-(trifluoromethyl)phenyl]-5H-imidazo[1,2-a]purine 2-[4-chloro-N-(1,3-thiazol-5-yl)anilino]acetonitrile 1-[(2S,3R)-5-(8-cyanoquinolin-4-yl)-1-methylpiperidin-3-yl]-3-ethyl-1-[(1R)-1-phenylethyl]urea 2-[1-hydroxy-3,4-bis(phenylmethoxy)butyl]piperidine-1,6-dicarboxylic acid 4-azidosulfanyl-2-(trifluoromethoxy)pyrimidine 3-[4,5-bis(ethenyl)-1H-pyrrol-3-yl]-6-bromoindole 4-[(3,5-dimethoxyphenyl)sulfonylamino]butanoic acid ethane;2-fluoro-4-methyl-3,5-bis(trifluoromethyl)pyridine N-[(2S)-3-(4,5-dihydrobenzotriazol-1-yl)propyl]-2-methylbutanamide 2-[4,5-bis(trifluoromethyl)pyridin-3-yl]sulfanyl-6-ethoxy-1H-indole 4-[[1-(oxolane-3-carbonyl)piperidin-4-yl]amino]-1H-pyrrolo[2,3-b]pyridine-5-carbonitrile 3-benzylsulfanyl-5,6,7,8-tetrahydro-[1,2]oxazolo[4,5-b]quinoline (3S,4R)-1-[[1-(2-aminoethyl)cyclopropyl]methyl]-4-benzylpyrrolidin-3-ol;dihydrochloride 2-(3-methoxyphenyl)ethanimidamide;2-phenylbenzenecarboximidamide 2,6-dibutyl-4-(5-methoxypentyl)phenol 6-(5-bromopyridin-2-yl)pyridine-3-carbonitrile 2,4-dimethoxy-6-(trifluoromethyl)benzenecarboximidate 1-[4-(azidomethyl)phenyl]-3-(cyclopenten-1-yl)urea 1-[2-(5-ethylfuran-3-yl)phenyl]-N-methoxypropan-1-imine 3-[2,4,6-tris(trifluoromethyl)phenyl]benzonitrile (7R)-2-(3,5-dimethoxyphenyl)-5-oxo-N-(4-propan-2-ylphenyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrimidine-7-carboxamide 2-azidooxy-N,N-dimethylbenzamide (2S)-2-amino-3-[4-(2,6-dimethoxyphenoxy)phenyl]propanoic acid [(2S,4R)-1-(cyclopropylmethylsulfonyl)-4-hydroxypyrrolidin-2-yl]-[6-phenyl-3-(trifluoromethyl)pyridin-2-yl]methanone [4-(2,3-difluorophenyl)piperazin-1-yl]-[5-(4-methoxyphenyl)-6-oxo-4H-thieno[2,3-c]pyrrol-2-yl]methanone N-[4-(3,5-dimethylpyrazol-1-yl)phenyl]propanamide (2S)-5-methyl-N-[(Z)-3,4,6-trimethylhept-2-en-2-yl]-1-azapentacyclo[10.7.1.02,7.08,20.013,18]icosa-2(7),3,5,8(20),9,11,13,15,17-nonaen-9-amine 3-bromo-4-(cyclohexylmethoxy)pyridine 1-[(Z)-1-ethenylsulfanylbut-2-enyl]-4-(trifluoromethoxy)benzene 2-[(4-phenyltriazol-1-yl)methoxy]oxolane N-[2-amino-1-(4,6-dimethoxypyridin-3-yl)ethylidene]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide (4R,5S)-4-phenyl-3,7,7-triazabicyclo[4.1.0]heptane 5-bromo-3-methoxy-4-(trifluoromethyl)benzonitrile 3-chloro-5-[(2R,6S)-4-[(Z)-1-(furan-2-ylmethylamino)prop-1-enoxy]-2,6-dimethylpiperazine-1-carbonyl]benzenesulfonamide 5-bromo-3-(1H-imidazol-2-yl)-N-methylidenethiophene-2-carboxamide 2,3-difluoro-4-[2-(8-propyl-1,2,3,4-tetrahydronaphthalen-2-yl)ethynyl]phenol 2-[(2,4-dichlorophenyl)methyl]-N,N,7-trimethylimidazo[1,2-a]pyridine-6-carboxamide 3-[(Z)-(4-chlorophenyl)methylideneamino]-6-methyl-1H-pyrimidine-2,4-dione (4-butan-2-yloxyphenyl)-(6,7-dihydroxy-1,3,8-trimethylnaphthalen-2-yl)methanone (2R)-2-[4-[1-(4,5-dihydro-1H-imidazol-2-ylmethoxy)ethenyl]phenyl]butanoic acid 2-[3-(cyclohexylamino)-5-oxo-7,8-dihydrophenazin-1-yl]propanamide 1-azidosulfanyloxy-2,3,4-triethoxybenzene 2-[1,6-dimethyl-3-(3-methyl-4-phenylmethoxyphenoxy)-5-oxocyclohexa-1,3-dien-1-yl]acetic acid 5-amino-4-[7-fluoro-6-(3,5,5,8,8-pentamethylnaphthalene-2-carbonyl)-1H-benzimidazol-2-yl]pentanoic acid 3-[3,5-bis(trifluoromethyl)phenyl]-N-[4-chloro-2-(5-oxo-1H-tetrazol-4-yl)phenyl]propanamide N-[(3R)-3-[5-(2,4-difluorophenyl)-1H-imidazol-2-yl]cyclohexyl]-3-methoxybenzamide 4-azido-2-chlorobenzenesulfonic acid 2-[(Z)-1,3-bis(4-chlorophenyl)prop-2-enyl]sulfanyl-5-methyl-6H-[1,3]thiazolo[5,4-d]pyrimidin-7-one N-(2-hydroxyethyl)-3-[4-methoxy-1-(pyridine-2-carbonyl)piperidin-4-yl]propanamide 3-[(1E)-buta-1,3-dienyl]-2-(4-ethoxyphenyl)-7-methoxychromene 3-azidooxy-7,8,9,10-tetrahydrobenzo[h]chromen-2-one 4-methyl-2,3,5-tri(propan-2-yl)furan 5-[2,3-dihydro-1H-inden-4-yl(methoxycarbonylamino)carbamoyl]-2,6-dimethylpyrimidine-4-carboxylic acid 2-[4-chlorobutyl([1,3]thiazolo[5,4-c]pyridin-2-yl)amino]ethanol 6-chloro-4-methylquinoline;propane 3-methyl-5-[3-(4-pyridin-2-yl-1H-indol-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl]phenol 5-fluoro-2-(4-phenylmethoxypiperazin-1-yl)pyrimidine 4-cyclopropyl-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]butanenitrile 1-(4,5,6,7-tetrahydrobenzo[d][2]benzazepin-10-yl)ethanone 2-[(5R)-4-oxo-3,5-dihydro-2H-1,5-benzoxazepine-5-carbonyl]cyclopentane-1-carboxylic acid 2-cyclopentyl-5-[2-[(3R)-oxolan-3-yl]oxy-4,7-dihydro-[1,3]thiazolo[5,4-d]pyrimidin-6-yl]phenol 2-[4-(trifluoromethyl)phenyl]spiro[1,3-dihydroisoquinoline-4,1'-cyclopropane] (2S)-3-(4,5-dichloro-1H-pyrrol-3-yl)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoic acid 1-(4,4-dimethylcyclohexen-1-yl)-3-(N'-ethylcarbamimidoyl)-2,6-dimethyl-2H-quinoline-7-carboxylic acid N-[2-(dimethylamino)ethyl]-1,2-dihydroquinoline-8-carboxamide 6-methyl-3-(2,2,2-trifluoroethoxy)pyridine-2-carbonitrile N-azido-4-methyl-6-(trifluoromethoxy)pyrimidin-2-amine 2-bromo-N-(4,5-dimethyl-2-phenyldiazenylphenyl)-N-pyridin-3-ylbenzamide 5-chloro-N-(3,5-dimethylpyridin-4-yl)furan-2-carboxamide 2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrole;ethane 2-[4-[1-(cyclopropylmethyl)pyrazol-3-yl]phenoxy]ethanol 1-(4,6-dimethylpyrimidin-2-yl)-N-ethyl-3-phenyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamide 4-[(3,5-dimethylpiperidin-1-yl)methyl]-N'-hydroxypyridine-2-carboximidamide 5-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(octyl)amino]naphthalene-2-sulfonic acid [3-(cyclopropylmethoxy)-5-(4-hydroxybut-2-ynoxy)phenyl]methanesulfonic acid 5-[[(3S,4R)-2,2-dimethyl-1-oxo-6-(4-phenylpiperidine-1-carbonyl)heptan-4-yl]amino]-1H-pyrrole-3-carbonitrile (2R)-1,4-dioxaspiro[4.5]decane;6-methoxy-4-N-methyl-3-nitropyridine-2,4-diamine 2-[(2R,5S)-3,4-dihydroxy-5-methoxypyrrolidin-2-yl]-5-(1H-indazol-5-ylamino)-1-methylpyrimidin-4-one N-[1-(4,6-dimethoxypyrimidine-5-carbonyl)piperidin-3-yl]-N-(pyridin-2-ylmethyl)cyclopropanecarboxamide 2-methoxy-4-phenylmethoxypyrimidine N'-[(4R)-2,5-diphenyl-3,4-bis(phenylmethoxy)pentan-2-yl]-N,N'-dimethyloxamide (E)-2,4-dimethylpent-3-ene;(Z)-6-ethylidene-4-phenyloct-1-en-5-yne 3-[1-(2,4-dimethoxyphenyl)sulfonylpiperidine-3-carbonyl]-5H-pyrrolo[3,4-b]pyridin-7-one N-[1-(2-fluoro-6-propoxyphenyl)ethyl]-7H-purin-2-amine 3,6-bis(methylamino)anthracene-9,10-dione;ethane 5-(methylsulfanylamino)-4-phenylmethoxypentan-2-ol (2R)-2,4,5-trimethyl-3-N,6-diphenylhexane-3,3-diamine 3-[(1R,2S)-3-(2H-triazolo[4,5-b]pyridine-3-carbonyl)cyclopentyl]propanamide N-[(1R)-1-[5-fluoro-2-(hydroxymethyl)phenyl]ethyl]-3-iodopyrazolo[1,5-a]pyrimidine-5-carboxamide 1-[5-(2,4-difluorophenyl)pyrimidin-2-yl]ethanethiol;3,8-dimethyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-d][1,4]diazepine N-[(4-ethoxyphenyl)methyl]-2-[5-(oxolan-3-ylmethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-7-yl]acetamide;2,2,2-trifluoroacetic acid 4-[(3Z)-3-[amino(propyl)amino]hepta-1,3-dien-2-yl]-N-methoxy-N-methylbenzamide 2-chloro-5,6-dideuterio-N-[1-(1H-indol-3-yl)-3-methylidenepentan-2-yl]pyrimidin-4-amine 3-(3,5-dichlorophenyl)sulfonyl-1H-indole [6-(1-cyclohexyl-4,5,7,8-tetrahydrooxepino[4,5-c]pyrazol-3-yl)pyridin-2-yl]-methoxyazanide 1-[(2R)-3,5-dihydroxy-6-oxo-8-(trifluoromethyl)-9H-xanthen-2-yl]azepane-4-carboxylic acid 6-methylsulfanyl-4H-imidazo[1,2-a]benzimidazole N-butyl-2,4,6-trimethyl-N-(1-phenylpropyl)benzenesulfonamide N-[4-(2,3-dihydroindole-1-carbonyl)phenyl]quinoxaline-6-carboxamide 5-amino-4-(3,5-dichlorophenyl)-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidine-2-thione N-[1-(6,7-dihydropyrrolo[2,3-c]pyridine-1-carbonyl)cyclohexyl]propane-2-sulfonamide 2-[(3aR)-5-hydroxy-1,3,3a,4,6,6a-hexahydrocyclopenta[c]pyrrol-2-yl]-N-[(7S)-8-oxo-6-phenyl-9-propanoyl-5,6-dihydrobenzo[b][1,4]benzoxazepin-7-yl]acetamide 2-hydroxy-N,3,6,7-tetramethylphenazine-1-carboxamide 3-(4-fluorophenyl)sulfonyl-2-[[3-(1H-indole-3-carbonylamino)propanoyl-methylamino]methoxy]propanoic acid 3-(2,6-difluorophenyl)sulfanyl-N'-[4-methyl-3-(5-oxo-1H-1,2,4-triazol-4-yl)phenyl]propanehydrazide (5R,7S)-N-[2-methylsulfanyl-5-(trifluoromethoxy)phenyl]-5-(4-propan-2-ylphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 5-azido-4-phenyl-2H-triazole N-(3,5-dimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine;hydrochloride (4E)-2-(3,5-dimethoxyphenyl)-4-[(4-fluorophenyl)methylidene]-1H-imidazol-5-one 5-ethyl-1,3-difluorobenzene;methanamine;2-[(4-naphthalen-2-ylphenyl)sulfanylamino]acetic acid 2-[1-[(4-methoxyphenyl)methyl]triazol-4-yl]propanoic acid 3-[2,6-dimethyl-4-(8-methylquinolin-5-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 2-(3,5-dimethylphenyl)-6-[4-hydroxy-3-(trifluoromethoxy)phenyl]-8H-imidazo[1,2-a]pyrimidin-7-one 3-(2,4-dihydroxyphenyl)-N-[(4-methylphenyl)-naphthalen-1-ylmethyl]propanamide (5R)-5,6-diethoxy-2-[4-methyl-3-[[5-methylidene-7-propan-2-yl-1,2,4-triazolo[1,5-a]pyrimidin-8-yl]methoxy]phenyl]-5H-isoindole N-[(1R,2S)-4-bromocyclohexa-2,4-dien-1-yl]-5-chloro-6-methoxyquinazolin-4-amine (3S)-4-[(3S,5R)-3,5-dimethyl-1-[8-(trifluoromethylsulfanylamino)quinolin-5-yl]piperidin-4-yl]-3-phenylpiperazine-1-carboxylic acid 3-methyl-4-(6-methylimidazo[1,2-a]pyrimidine-3-carbonyl)piperazine-1-carboxylic acid 2-(4-tert-butylphenyl)-N,7-dimethylimidazo[1,2-a]pyridine-6-carboxamide 1,2-diamino-4-(3-ethoxy-5-iodophenyl)-6-oxopyridine-3,5-dicarbonitrile 6-bromo-1-(2,5-dimethoxyphenyl)cyclohexa-3,5-diene-1,3-dicarboxylic acid 2-chloro-4-(1,3-dimethylpyrazolo[3,4-d]pyrimidin-6-yl)phenol 5-[3-(4-butylphenyl)pentan-3-yl]-2H-tetrazole 1-[4-(3,5-difluorophenyl)-2-methylbutan-2-yl]-3-[[(Z)-hydroxyiminomethyl]amino]thiourea 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N-[2-(1-methylpyrazol-4-yl)ethyl]acetamide (Z)-3-(4-chlorophenyl)-3-hydroxy-N-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)-2-pyridin-1-ium-1-ylprop-2-enethioamide (5Z)-2-phenylimino-5-[[4-(3,4,5-trimethoxybenzoyl)oxyphenyl]methylidene]-1,3-thiazolidine-4-carboxylic acid 5-(6,7-dimethoxyquinazolin-4-yl)oxy-N-[3-fluoro-2-hydroxy-5-(trifluoromethyl)phenyl]-1-benzofuran-2-carboxamide N-benzyl-6-(5,5-dioxo-1,3,2-oxathiazolidin-2-yl)naphthalene-2-carboxamide 3-(dimethylamino)-1-(7,8-dimethylimidazo[1,2-a]pyridine-2-carbonyl)piperidine-3-carboxylic acid 1-[2-azido-4-(trifluoromethyl)phenyl]piperidine N-(3,4-dihydro-2H-pyran-7-ylmethyl)-8-ethylnaphthalene-1-sulfonamide 5-azidooxy-2,6-diphenylpyrimidine 4-[(Z)-aminomethylidenehydrazinylidene]-2-imino-5,7,8-trimethyl-N-[4-(1H-pyrazol-4-yl)phenyl]thieno[3,2-c]quinoline-6-carboxamide 2-N,4-N,5-triphenylpyrimidine-2,4-diamine [2-(1,3-benzodioxol-5-yloxy)cyclopentyl]-(4-cyclopropylpiperazin-1-yl)methanone 4-hydroxy-2,7-dioxoazecine-3-carbonitrile 1-[(4,5-dichlorothiophen-2-yl)methyl]-3-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]urea 6-[2-(3,5-difluorophenyl)ethylamino]-1-propyl-5H-pyrazolo[3,4-d]pyrimidin-4-one 5-[5-(2-cyclopropylpyrazol-3-yl)pyridin-3-yl]-1,3-thiazol-2-amine;ethane 1-[6-(3,5-difluorophenyl)-2-methylpyrimidin-4-yl]piperidine-3-carboxylic acid (3-azido-5-propylsulfonylphenyl)methanamine N-[3-(4,5-dimethyl-6-oxo-1H-pyrimidin-2-yl)-4-propoxyphenyl]cyclopropanecarboxamide 3-(4,5-diphenylfuran-2-yl)-N-hydroxy-1H-indole-6-carboxamide (4R)-4-ethenyl-1,3,4-trimethyl-7-[(Z)-prop-1-enyl]quinoxaline-2,6-dione 1-[(5S,7R)-5-phenyl-7-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]pyrrolidine-3-carboxylic acid 4-(2,6-dimethylmorpholine-4-carbonyl)-3H-1,3-thiazol-2-one 5-[5-[(2S,3R)-1-amino-3-methylpentan-2-yl]thiophen-2-yl]-N'-hydrazinylpyridine-2-carboximidamide N-[2-[(4,6-dimethylpyrimidin-5-yl)sulfonylamino]ethyl]-4-nitrobenzenesulfonamide 4-[(3-fluorophenyl)methyl]-1-piperidin-3-ylpyrazolo[3,4-d]pyrimidine;hydrochloride 4-[4-(1,3-benzothiazol-2-yloxy)-3-methoxyphenyl]morpholine 3-[4-[[1,2,5]oxadiazolo[3,4-b]pyridin-7-ylmethyl(methyl)amino]phenyl]cyclopropane-1,1,2,2-tetracarbonitrile 2-[5-bromo-6,7-dichloro-3-oxo-1-(2,4,6-trimethylphenyl)sulfonylindol-2-ylidene]propanedinitrile 1-(3,4-dimethylphenyl)ethanol;2-[6-ethoxy-5-fluoro-3-(2-propoxyethoxy)pyridin-2-yl]acetaldehyde 4-methyl-N-(3,4,5-trifluorophenyl)sulfanylbenzenesulfonamide 3-(5-azidopyrazol-1-yl)-4-cyclopropylpyridine 4-azido-5-methylpyrrolo[3,2-d]pyrimidine N-[5,6-dichloro-1-(2,4-dimethylphenyl)sulfonylbenzimidazol-2-yl]acetamide 3-(2,2-dimethylpropylamino)-5,11,12-triazatetracyclo[7.6.0.02,6.010,14]pentadeca-1(9),2(6),4,7,15-pentaene-13-carboxamide 2-[6-amino-3-(cyclopropylmethoxy)cyclohepta-1,4,6-trien-1-yl]-N-(4,5-difluoropyridin-3-yl)acetamide 2-chloro-4-fluoro-N-[(Z)-1H-indol-3-ylmethylideneamino]benzamide (7R)-1,7-diethyl-8-methoxy-6,9-dihydro-5H-triazolo[4,5-c]quinolin-4-one 2-(1H-indole-3-carbonyl)-N-[3-methyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolidine-1-carboxamide 2-[(3S)-1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carbonyl)pyrrolidin-3-yl]-5,6,7,8-tetrahydro-3H-quinazolin-4-one 4-[[2,3-difluoro-5-methyl-6-(trifluoromethyl)phenyl]carbamoylamino]benzoic acid (1R,2S)-2-azido-4-(7H-purin-6-ylmethylamino)cyclopentan-1-ol 2-[3,5-bis(trifluoromethyl)phenyl]cyclohepta-1,3,6-trien-1-ol 1-[3-(3,4-difluorophenyl)cyclobutyl]-2H-pyridine 7-cyclohexylimino-2-(furan-3-yl)-5-[2-(6-methoxypyridin-3-yl)pyridin-4-yl]pyrazolo[1,5-a]pyrimidine-3,6-dicarbonitrile 3-(5,6-difluoro-2-methoxypyridin-3-yl)-4,5,6,7-tetrahydro-1H-indazole;fluorobenzene N-(3,4-dichlorophenyl)-2-[4-hydroxybutyl-methylsulfonylamino]acetamide 3-benzyl-2,2,4H-1,4-benzothiadiazin-7-amine 5-[2,4-difluoro-6-(hydroxymethyl)phenyl]-3-(4-thiophen-3-ylthiophen-2-yl)-1H-pyridin-2-one N-[3-(diaminomethylidene)cyclopentyl]-3,4,5-trifluorobenzamide 4-[[2-(azidooxymethyl)phenyl]methylideneamino]phenol 5-(2,4-difluorophenoxy)-1H-pyrrolo[2,3-b]pyridine (5S,6R)-3-ethylsulfanyl-2,4-dioxo-N-phenyl-1,3-thiazolidine-5-carboxamide [(2S)-1-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-4,4-dimethylpentan-2-yl]azanide;2-ethylthiophene;iridium(3+) 6-fluoro-3-methyl-4-phenyl-1H-quinoline-2,7-dione 4-methyl-2-[[(Z)-1,3,3-trihydroxyprop-1-en-2-yl]diazenyl]isoindole-1,3-dione 2-[4,5-bis(3-chlorophenyl)furan-2-yl]-N-[2-hydroxy-5-(2H-tetrazol-5-ylmethoxy)phenyl]acetamide 3-[4-[4-[6-ethyl-7-methoxy-2-(2,4,6-trifluorophenyl)-5H-pyrrolo[1,2-a]imidazole-3-carbonyl]pyrazol-1-yl]butyl]-1,3-oxazolidin-2-one 3-hydroxy-1,2-dimethylindolizine-6-carboxamide 1-[4-[(3,5-difluorophenyl)methyl]piperazine-1-carbonyl]pyrazole-3-carboxylic acid ethane;1-[4-(7-hydroxyquinoxalin-5-yl)oxypiperidin-1-yl]-2-pyridin-3-ylethanone N-[4-(4-fluorophenoxy)phenyl]-6,7-dimethoxyquinazolin-4-amine;2-methylphenol [3-amino-6-(2,4-difluorophenyl)thieno[2,3-b]pyridin-2-yl]-[2-fluoro-6-(1H-indole-3-carbonyl)phenyl]methanone 1-azido-2,4-diphenyl-3-(trichloromethyl)benzene 5-[2-(4-chlorophenyl)piperidin-1-yl]sulfonyl-N-methoxypyrazin-2-amine 7-chloro-2,9-dimethylindeno[1,2-b]pyrazine 4-[2-(1,3-benzodioxol-5-yl)propanoylamino]-N-cyclopentylpyrazole-1-carboxamide 3-[(4-chlorophenyl)methyl]-N'-hydroxybenzenecarboximidamide 5-(4-chlorophenyl)-2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrole 1-azidooxy-4-ethyl-2,3-diphenylbenzene 2-(1H-benzimidazol-2-yl)-4-(trifluoromethoxycarbonylamino)benzoic acid 6-(4-ethylphenoxy)pyridine-2-carboxamide 1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]indole 2-[5,6-bis(trifluoromethyl)pyridin-3-yl]-N-methylacetamide 2-(3,5-difluoro-4-hydroxyphenyl)-6-methylcyclohexan-1-one N-[(2S)-1-[4-[(3S,5R)-3-amino-5-methylpiperidin-1-yl]-6-fluoroquinolin-3-yl]propan-2-yl]benzamide 4-(6,7-dihydrodibenzofuran-4-yl)-2-methylbutan-2-ol 2-(1,3-benzothiazol-2-yl)-4-[(E)-4-methoxybut-2-en-2-yl]phenol 2-(3,4-dihydro-1H-isoquinolin-2-yl)-5-methanimidoylphenol 1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)azetidin-2-one 5-azidosulfanyl-3-[2,6-dimethoxy-4-(trifluoromethyl)phenyl]-1,2,4-thiadiazole [4-azido-2,3-dimethoxy-6-[3-(trifluoromethyl)phenyl]phenyl]phosphane 2-amino-6-ethoxy-4-[3-(methylamino)phenyl]-4H-pyran-3,5-dicarbonitrile 1-(2,3,4a,5,6,7,8,9,9a-octahydrobenzo[b][1]benzoxepin-10-yl)ethanimine 1-[4-(5-nitrothiophen-2-yl)phenyl]ethanone (E)-N-[1-[2,6-dichloro-4-(trifluoromethyl)phenyl]ethylideneamino]butanamide (6S)-6,7-dimethyl-3-[[4-(oxan-2-yloxy)phenyl]sulfonylmethyl]heptan-1-ol N-cyclohexyl-6-[[3,5-difluoro-4-(trifluoromethoxy)phenyl]methyl]-1-formamido-2H-pyridine-3-carboxamide 2-[4-(diethylamino)phenyl]-4,6-bis(2-pyridin-2-ylethynyl)pyrimidine-5-carbonitrile 4-[(6,8-dimethylimidazo[1,2-a]pyridin-2-yl)sulfonyl]-3,5-dimethoxybenzenecarboximidamide 4-hydroxy-3,7-dimethyl-1-[(2R)-5,6,6-trimethyloct-7-enoxy]quinolin-2-one 1-(2,5-dimethyl-1,3-thiazol-4-yl)-3-[6-(trifluoromethyl)pyrimidin-4-yl]urea 2-azidooxy-4,5-dichloro-N-[1-(5-methylsulfanylpyridin-3-yl)ethyl]benzamide 3-(methanesulfonamido)-N-[1-[4-[2-[1-(2,2,2-trifluoroethylamino)ethenyl]phenyl]piperidine-1-carbonyl]cyclopentyl]propanamide N-methyl-1-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carbonyl)piperidine-2-carboxamide N-(6-chloropyridin-3-yl)-2-methoxy-N-(1,3-thiazol-5-yl)acetamide 5-methoxy-N-[4-(trifluoromethyl)pyridin-2-yl]benzenesulfonamide [1-amino-2-[4-[(2R)-3-azidobutan-2-yl]oxyphenyl]ethylidene]azanium 1-N,4,6-trimethylisoquinoline-1,8-diamine 2-[3-(methylcarbamoyl)anilino]-4-oxobut-2-enoate 1-(2,2,2-trifluoroethyl)naphthalene 5-methoxy-2-(1,2-oxazol-3-yl)benzenesulfonic acid N-(2,3-dihydro-1H-inden-5-yl)-N'-[1-(3-ethoxypropyl)-7-fluorobenzimidazol-2-yl]ethane-1,2-diamine 3-[(4-methoxyphenyl)sulfonylamino]-N,N-dipropylbenzamide 3-(2-aminopyridin-4-yl)-1,1-bis[1-(cyclopropylmethoxy)naphthalen-2-yl]urea [4-[2,6-difluoro-3-(trifluoromethyl)phenyl]piperazin-1-yl]-[5-(hydroxyiminomethyl)thiophen-2-yl]methanone 2-(5,7-dibromo-1H-indole-3-carbonyl)propanedioic acid N-[4-(1,3-dioxoisoindol-2-yl)sulfonylphenyl]-5-hydroxy-N'-methyl-1H-indole-7-carboximidamide 2-[3-(1,5-dimethylpyrazol-4-yl)morpholine-4-carbonyl]-4H-isoquinoline-1,3-dione (2S)-N-[2-[4-cyano-3-(trifluoromethyl)phenyl]ethyl]piperidine-2-carboxamide 2-methyl-N,4-diphenylpiperazine-1-carboxamide N-(2,3-dihydro-1H-inden-2-yl)-6-methoxy-8,11,11-trioxo-5-azaspiro[3.9]tetradecane-7-carboxamide;2-ethylthiophene 1-[4-(2,3-dichlorophenyl)piperazin-1-yl]propan-1-one N-[2-(4-methoxyphenyl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide;2-[(5S,6S)-6-methylpiperidin-3-yl]guanidine 2-azido-6-bromoisoquinolin-1-one 1-[2,4-bis(trifluoromethyl)phenyl]-3-methoxypropan-2-one 4-[[(2S)-1-acetylpyrrolidin-2-yl]methylamino]-6,7,8,9-tetrahydropyrido[3,2-a]indolizine-5,10-dione 1-azidooxy-2,4,5-trimethyl-3-propan-2-ylbenzene 1-[(3S)-3-hydroxypyrrolidin-1-yl]-2,4-diphenylbutan-1-one 5-[6-(4,5-dimethoxycyclohepta-1,3,6-trien-1-yl)hexyl]imidazole-2,4-dione 6-(3,4,5-trifluorophenyl)-2H-benzotriazol-4-ol (E)-4-[(Z,3R)-6-aminohex-2-en-3-yl]oxy-N-methylidene-5-phenylpent-4-enamide 1-(2,4-difluorophenyl)sulfonylspiro[2H-indole-3,7'-6H-furo[2,3-f][1]benzofuran] 3-(4-chlorophenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidine 1-cyclohexa-2,4-dien-1-ylnaphthalene;ethane 4-methyl-2-[3-nitro-N-(1,3-thiazol-5-yl)anilino]pentanoic acid 6-[(1S)-1-ethoxypropyl]naphthalene-2-carboxylate 4-(chloromethyl)-1,3-diphenyl-5H-imidazo[4,5-c]pyridine 2-N,3-N-bis(4-chlorobutyl)benzene-1,2,3-triamine (2R)-2-methoxy-N-[2-(2,4,5-trifluorobenzenecarbothioyl)phenyl]butanamide 3-(2,6-dichlorophenyl)-7-[4-ethyl-4-(1-hydroxyethyl)piperidin-1-yl]-1-methylquinoxalin-2-one;hydrochloride 2-[2-(aminomethyl)phenyl]sulfanyl-4-methyl-1H-pyrimidin-6-one N-[4-(2-azidoethoxy)phenyl]methanesulfonamide 2-[(1R)-5-chloro-2,3-dihydro-1H-inden-1-yl]acetamide N-(cyclohexa-1,5-dien-1-ylmethyl)-3-[4-[2-[(E)-hydroxyiminomethyl]phenyl]sulfanylphenoxy]propanamide N-[4-hydroxy-3,5-bis(methoxycarbonyl)-1H-pyrrol-2-yl]butanimidate 6-tert-butyl-7,11-dihydrobenzo[c]carbazole N-[2-(3,4-dimethylphenyl)ethylidene]hydroxylamine 5-[5-(4,6-diphenylpyridin-2-yl)pyridin-3-yl]-2H-triazole 1-[(3R)-5,6-dimethyl-2,3-dihydro-1H-inden-1-yl]pyrrole-2,5-dione 2-(5-fluoropyridin-3-yl)-8-methyl-7H-purine 1-[(3R)-3,4-dimethylhexan-2-ylidene]-6-phenylbenzimidazol-5-ol 2-azidooxy-6,7,8,9-tetrahydro-5H-acridine 4-(1H-pyrrolo[2,3-b]pyridin-4-ylmethyl)benzamide 2-[4-(2,3,5,6-tetramethylphenyl)pyrazol-1-yl]phenol 5-[2-(1H-indol-3-yl)ethyl-methylsulfonylamino]naphthalene-2-sulfonic acid [(2R)-5-butoxy-1,1-dioxo-4H-thieno[3,4-d]triazin-2-yl]methanesulfonic acid N-[(Z)-3-aminoprop-2-enimidoyl]-6-chloro-7-formamido-2,4-dimethylindole-1-carboxamide (3E)-1-methyl-3-[[2-methyl-5-propoxy-4-(thiophen-2-yldiazenyl)phenyl]hydrazinylidene]indol-2-one 3-(4-chlorophenyl)-5-[3-[4-hydroxy-2-(propan-2-yloxymethyl)phenoxy]propoxy]-1,4-dihydroquinazolin-2-one 4-[1-(2,5-difluorophenyl)ethyl]-3-methoxyaniline 2-[4,6-bis(4-fluorophenyl)pyrimidin-1-ium-2-yl]oxyethanamine N-[4-amino-3,4-dioxo-1-(1H-pyrrol-2-yl)butan-2-yl]-5-pyridin-2-yl-1,2-thiazole-4-carboxamide 2-[(5,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)amino]butanedioic acid (5S)-2,2-diethylsulfanyl-N-phenyl-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide N-[(E)-but-2-enyl]-4-(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)piperazine-1-carboxamide 3-[6-(azepane-1-carbonyl)naphthalen-2-yl]propanoic acid 6-chloro-2,4,4a,9a-tetrahydroindeno[1,2-a]indene N-[1-(1H-imidazol-5-ylmethyl)piperidin-4-yl]formamide 3-[(1S)-2,6-dimethylcyclohexa-2,4-dien-1-yl]-6-pyridin-4-yl-9H-carbazole 6-methoxy-4,7-dinitrofluoren-9-one 2-ethylsulfanyl-3,4-dimethoxypyridine (4-benzylpiperidin-1-yl)-(1H-pyrrol-2-yl)methanone 5-[3-[(1R,5S)-8-chloro-8-phenyl-9-azatricyclo[6.2.02,7]dodeca-2(7),3,5-trien-4-yl]propanoylamino]pyridine-2-carboxylic acid 2-amino-6-(4-hydroxy-3-methylbutanoyl)-3H-pteridin-4-one 3-[[4-(2,1,3-benzoxadiazol-5-yl)piperazin-1-yl]methyl]benzoic acid;hydrochloride 4-[5-(2-amino-1,3-thiazol-4-yl)pyridin-3-yl]phenol [4-(1H-indol-2-yl)phenyl]methanamine;hydrochloride 2-bromo-4-[(Z)-[[5-chloro-6-(2,3-dihydro-1H-isoindol-5-ylamino)pyrimidin-4-yl]hydrazinylidene]methyl]phenol (2R)-2-[amino-(4,5-dimethylbenzimidazole-1-carbonyl)oxymethylidene]pyrrolidine-3-carboxylic acid 1-[(3R)-4,5-bis(benzenesulfonyl)-6-(2-bromophenyl)-3-methyl-2-oxo-1H-pyridin-3-yl]ethanone 1-ethenyl-4-fluorobenzene;(2S)-2-[(Z)-6-methoxyhex-2-en-3-yl]-N,N-dipropylcyclopentan-1-amine N-[5-cyano-6-(triazol-2-yl)pyridin-3-yl]-1-[5-cyano-4-methoxy-6-(trifluoromethyl)pyridin-3-yl]-5-(trifluoromethyl)pyrazole-4-carboxamide 2-(1-chlorocyclohexyl)sulfanyl-N'-hydroxypyrimidine-4-carboximidamide 1-(2,4-difluorophenyl)sulfonyl-6-(2-methylbenzimidazol-1-yl)-5-propan-2-yloxyindole 4-(6,7-difluoro-2H-chromene-3-carbonyl)piperazine-1-carboxylic acid 3-(1,3-benzothiazol-2-yl)-5-methoxychromen-4-one (E)-1-[4-(cyclopropylmethoxy)-3-fluorophenyl]-N-ethenyl-3,3-dimethylbut-1-en-2-amine;ethene N-[[4-chloro-3,5-bis(trifluoromethyl)phenyl]methoxy]-2-(5-fluoro-6-oxopyrimidin-1-yl)acetamide 4-[2-(9H-fluoren-1-yl)piperidine-1-carbonyl]-2,5,6-trimethoxybenzenesulfonamide 2-(azetidin-1-yl)-4,5-dichlorobenzaldehyde (4R,5S)-2,8-dimethyl-4-propan-2-yl-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-1-one;2,2,2-trifluoroacetic acid 2-(3,4-difluorophenyl)-6-[4-(3-methylpentan-3-yloxy)piperidin-1-yl]pyrimidine 2-(5,8-dibromonaphthalen-2-yl)cyclohexane-1,3-dione 4-[(3-azidophenyl)methyl]morpholine 5-benzylsulfanyl-3,4,6-triphenylbenzene-1,2-diol 5-(2,4-dihydroxy-6-methylphenyl)-N-ethyl-4-[4-(pyridine-3-carbonyl)piperazine-1-carbonyl]-1,2-oxazole-3-carboxamide N-[4-(4,6-dimethoxypyrimidin-2-yl)sulfanylphenyl]formamide 5-[3-bromo-2,6-dihydroxy-4-(trifluoromethyl)phenyl]thiophene-2-carboxylic acid 2-[3-cyano-4-ethyl-5-isocyano-6-(4-pyridin-4-ylphenyl)pyridin-2-yl]sulfanyl-N,N-dimethylbenzenecarboximidamide 4-[(3R)-5-[2-[1-hydroxy-6-imino-2,7-dimethyl-3-(2-thiophen-2-ylethylcarbamoyl)piperidin-4-ylidene]hydrazinyl]-3-methyl-9-oxoxanthen-9-yl]benzoic acid 4-N-[2-(dimethylamino)ethyl]-1-N,2-diethylbenzene-1,4-diamine N-[(Z)-1-(4-hydroxyphenyl)ethylideneamino]-1,3-benzothiazole-2-carboxamide 2,4-difluoro-N-[(1S)-2,2,3,3,3-pentafluoro-1-[4-[5-(trifluoromethyl)pyridin-2-yl]oxyphenyl]propyl]benzamide 2-[(3R)-4-[benzyl(methyl)amino]-2,2,7,7-tetrafluoroheptanoyl]sulfanylacetic acid 4-[3-hydroxy-5-(trifluoromethyl)phenyl]sulfonylmorpholine 2-[3,5-bis(trifluoromethyl)anilino]-1-(4-methoxyphenyl)pentan-3-one 2-[[4-(hydroxymethyl)-3,5-dimethoxyphenyl]methylideneamino]-N-[4-(1-methylpyrazol-4-yl)phenyl]acetamide (1R)-2,3-dihydro-1H-inden-1-amine;6-[(4-methoxyphenyl)sulfonylamino]hexanamide 4-(2,5-dimethylphenyl)-1-[2-(hydroxyamino)-2-oxoethoxy]-7-(4-piperidin-4-ylbutyl)isoquinoline-3-carboxamide 2-[3-[(E)-[4-(4-chlorophenyl)-5-oxo-1,3,4-oxadiazol-2-ylidene]methyl]-2-methylindol-1-yl]propanoic acid N-(3,4-dichlorophenyl)-2-[(6S)-5-oxo-7-thiophen-2-yl-4,6-dihydrotetrazolo[1,5-a]pyrimidin-6-yl]acetamide 1-[4-(3-amino-5-nitrophenyl)piperazin-1-yl]-2,2-dimethylpropan-1-one 2,6-dipyridin-3-ylpyridine;methanol 4-[6-amino-5-(methyliminomethyl)pyrimidin-4-yl]oxypiperidine-1-carboxylic acid 2-[5-aminosulfanyl-4-(benzenesulfonyl)thiophen-3-yl]-N-[3,5-dibromo-1-(3,4-dimethoxyphenyl)penta-1,4-dien-2-yl]acetamide;ethane 2-tert-butyl-4-(cyclohexylmethoxy)-3-nitrobenzenesulfonic acid 3-[2-(4-ethylsulfanylphenyl)-1H-indol-5-yl]propanoic acid 6-amino-5-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-N'-hydroxypyridine-2-carboximidamide 2,6-bis(4-chlorophenyl)-3-methylbenzonitrile 2-[[2-(4-chlorophenyl)morpholin-4-yl]methyl]-3H-quinazolin-4-one 2-[5-(4-bromophenyl)sulfonyl-2-methoxyphenyl]benzoic acid 3-amino-4-ethyl-N-(2-methoxyphenyl)thieno[2,3-b]pyridine-2-carboxamide N-[5-(cyclopropylcarbamoyl)pyridin-2-yl]formamide;(2S,3R)-3-methylhexan-2-one N-cyclohexyl-4-[5-(4-hydroxyphenyl)-1,2,3,3a,4,5,6,7,7a-octahydropentalen-2-yl]benzenesulfonamide 6-bromo-5-(dimethoxymethyl)triazolo[1,5-a]pyridine 5-methoxy-N,3-dimethylpyrazine-2-carboxamide (3R)-2,2,4-trimethyl-7-N-(1-methylpiperidin-4-yl)-1H-1,5-benzodiazepine-3,7-dicarboxamide 5-[[1-(cyclopropylmethoxy)isoquinoline-3-carbonyl]amino]-2,4-difluorobenzoic acid 2-methoxy-4,6-dinitrobenzenecarboximidamide [(E)-[3-[(4-chlorophenyl)methyl]-2H-1,5,6-oxadiazin-4-yl]methylideneamino]thiourea 6-chloro-4-phenylsulfanyl-1,2-dihydroanthracene N-[4-(4-oxo-3H-quinazolin-2-yl)phenyl]-N,3-dipropylbutanamide 1-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)piperidine-4-thiol (5-aminotetrazol-1-yl)oxymethylphosphonic acid 1,2-bis(2-methoxyphenyl)ethane-1,2-diamine (2S)-1-[3,5-dichloro-4-[[7-fluoro-6-(1H-pyrazol-4-yl)quinazolin-4-yl]amino]benzoyl]pyrrolidine-2-carboxylic acid 3-[4-(2-bromophenyl)butyl]dithiole 1-(4-bromophenyl)-3-[2-(1,5-naphthyridin-2-ylamino)ethyl]thiourea 1-[5-bromo-2,6-dichloro-4-(trifluoromethyl)pyridin-3-yl]ethanone 4-fluoro-3,5-di(nonyl)benzoic acid N-[(1,4-dimethylpyrazol-3-yl)methyl]-2,8-bis(trifluoromethyl)pyrazolo[1,5-a][1,3,5]triazin-4-amine 1-azido-2,4-dibromo-3-phenoxybenzene N-[2,6-difluoro-4-(1-methylsulfonylpiperidin-4-yl)oxyphenyl]quinoxaline-5-carboxamide 6-[4-[(2,4-dichlorophenyl)methyl]piperazin-1-yl]-1H-benzimidazole [1-(5,7-dimethylthieno[3,2-b]pyridine-6-carbonyl)piperidin-3-yl]carbamic acid 5-(bromomethyl)-4-butan-2-yloxy-N'-hydroxypyridine-2-carboximidamide 3-[[2-[(1R)-1-methoxyethyl]phenyl]sulfonylamino]azetidine-1-carboxylic acid 3-[4-(2-methylpropoxy)phenyl]sulfanylpropanenitrile (2R,4S)-1-(1H-pyrrole-3-carbonyl)-4-[3-[5-(trifluoromethyl)pyridin-2-yl]oxypyrrolidine-1-carbonyl]pyrrolidine-2-carbonitrile (2R)-N-[2-(dimethylamino)ethyl]-2-[1,3-thiazol-4-ylsulfonyl(trifluoromethylsulfinyl)amino]-4-(trifluoromethyl)butanamide 2,3-dichloro-4,6-dicyclopentylaniline 4-[2-(4,4-dimethylcyclohexen-1-yl)ethenyl]-N,3-bis(ethoxycarbonyl)-5-(hydroxyiminomethyl)benzamide 3-[3-chloro-4-[1-[2-(oxan-4-yl)ethyl]-2,6-dioxopiperidin-3-yl]phenyl]benzonitrile 1,2-dimethyl-5-[4-(oxiran-2-ylmethoxy)phenyl]-3H-pyrazole N-azido-2,4-dihydroxybenzamide N-[3,4-bis(trifluoromethyl)phenyl]acetamide;ethane (2S,4S)-2-[(1R)-1-[2-chloro-4-(trifluoromethyl)phenoxy]ethyl]piperidine-4-carboxylic acid (5E)-3-cyclohepta-1,4,6-trien-1-yl-N-[(Z)-1H-indol-3-ylmethylideneamino]-5-[(E)-2-phenylethenyl]-1,2-dihydroimidazole-4-carboxamide N-[[(2S,4S)-4-[[(1R)-1-phenylethyl]amino]pyrrolidin-2-yl]methyl]-1H-pyrazole-5-carboxamide N-(3,4-dimethoxyphenyl)-2-[5-(1H-indol-3-yl)-4-(thiophen-2-ylmethylidene)-1,2,4-triazol-3-ium-3-yl]acetamide 2-(3,4-dimethoxyphenyl)-5-[(1E)-2-ethylbuta-1,3-dienyl]pyridine (1S,2R)-N-[(Z)-2-amino-3-[(6-methoxypyridin-3-yl)amino]prop-2-enyl]-2-phenylcyclopropane-1-carboxamide 3-azidooxy-1-(3,4,5-trifluorophenyl)propan-1-one 1-chloro-3-methoxybenzene;N'-[4-(3,3-dihydroxypropoxy)naphthalen-1-yl]sulfonyl-2-(methylamino)ethanimidamide 3-amino-4-oxo-5,6,7,8-tetrahydropyrrolo[1,2-a]quinazoline-9-carboxylate 4-(3-cyanophenyl)sulfonyl-2,3,5,6-tetrafluorobenzoic acid (1R,3S)-6-[2-ethyl-4-[2-methoxy-3-[1-(7H-purin-6-ylamino)propyl]phenyl]phenoxy]-2,2-difluorocyclohexane-1-carboxylic acid 3-azido-6,7-dimethoxy-2H-isoquinolin-1-one N-(2,6-difluorophenyl)-5-methyl-4-piperidin-3-ylpyrimidine-2-carboxamide;dihydrochloride 2-[2,3-dihydroindole-1-carbonyl(methyl)amino]acetic acid 3-(3,4-dihydropyridin-3-yl)-9H-pyrido[2,3-b]indole 4-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]-8-pyrrolidin-1-ylpyrido[2,3-d]pyrimidin-7-one 1-(4-acetylpiperazin-1-yl)-2-[7-[2-(trifluoromethoxy)phenyl]-1,2,3,4-tetrahydronaphthalen-2-yl]ethanone (2S,4R)-N-[1-(2,6-dichloro-3-fluorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide;hydrochloride 2-[(4-hydroxypiperidin-1-yl)methyl]-3H-thieno[3,2-d]pyrimidin-4-one 2-[5-amino-3-(fluoromethyl)pyrazol-1-yl]-N'-hydroxyethanimidamide 2-[3,5-bis(trifluoromethyl)anilino]benzenesulfonic acid N-(4-chlorobutyl)-6,11-dioxobenzo[a]quinolizine-3-carboxamide 4-[7-methoxy-3-(4,5,6-triethoxypyridin-2-yl)-1H-indol-5-yl]phenol 5-[(3,5-difluorophenoxy)methyl]-2-ethoxypyridine (3R)-1-[2-amino-5-fluoro-4-(propanoylamino)benzoyl]-N-cyclohexylpiperidine-3-carboxamide 4-(5,6-dimethoxy-1H-benzimidazol-2-yl)phenol 2-[(2,4-difluorophenyl)methyl]-5-nitrofuran 7-[3-(2-hydroxypropan-2-yl)phenyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 2-methyl-7-phenyl-3H-quinazolin-4-one 4-methylbenzenesulfonic acid;5-nitroquinolin-8-ol 2-[2-(2,5-dihydroxyphenyl)propan-2-yl]benzene-1,3-diol 6-(2-diazohydrazinyl)-3,4-dihydro-1H-quinolin-2-one 3-[(7S)-2-fluoro-8-methyl-6,7-dihydropyrido[1,2-a]indol-10-yl]-N-methylaniline 2-[[4-[6-[(4-cyano-2,3-difluorophenyl)methoxy]pyridin-2-yl]piperazin-1-yl]methyl]-3-[[(1R,2S)-2-hydroxycyclopentyl]methyl]benzimidazole-5-carboxylic acid 2-[(3R,4S)-4-hydroxy-1-methylpyrrolidin-3-yl]oxy-5-pyridin-3-ylbenzonitrile 1-(1-acetylpiperidin-4-yl)-3-[7-hydroxy-8-(2-methoxyethylamino)-2,5-dioxopyrano[2,3-d]pyrimidin-6-yl]urea 7-(6,8-dichloro-2-methyl-3,4-dihydro-1H-isoquinolin-4-yl)-5,11-dioxo-[1,2]thiazolo[4,5-b][2]benzazepine-1-carboxylic acid N-[6-(azetidine-1-carbonyl)pyridin-3-yl]morpholine-4-carboxamide (5R)-2-benzylsulfanyl-8,8-dimethyl-5-phenyl-5,7,9,10-tetrahydro-3H-pyrimido[4,5-b]quinoline-4,6-dione 2-[(E)-2-[4-[bis[2-(cyclopropylmethoxy)ethyl]amino]phenyl]ethenyl]-1,3-benzothiazol-6-ol 1-(2,3-dihydro-1H-inden-4-yloxy)pyrazole 4-[(3E)-hexa-1,3,5-trien-3-yl]-N-methyl-2H-benzotriazol-5-amine 1-[2,4-dichloro-3-(ethylaminomethyl)phenyl]ethanone 7-(2,6-difluorophenyl)-N-[1-(4-methylpiperazine-1-carbonyl)pyrazol-3-yl]-5-oxo-4H-pyrazolo[1,5-a]pyrimidine-2-carboxamide 3-(azidomethyl)benzenesulfonic acid 3-cyclobutyloxy-4,6-dimethylpyridine-2-carboxylic acid 3-(1H-imidazol-2-ylmethyl)-7-nitroquinazolin-4-one 5-[4-[3-(4-amino-3,6-dihydro-2H-pyridin-1-yl)propoxy]phenyl]-N-(pyridin-2-ylmethyl)furan-2-carboxamide 6-(2,3-difluorophenyl)-4-[3-[5-(3,5-dimethylpyridin-1-ium-2-yl)oxypentoxy]-2-methylphenyl]-5H-pyrrolo[3,4-b]pyridin-7-one 4-N,6-N-dimethylquinazoline-4,6-diamine 2-[4-[(Z)-(2,5-dioxoimidazolidin-1-ium-4-ylidene)methyl]phenyl]isoindole-1,3-dione 4-bromo-2-[[5-(3,6-dimethylquinoxalin-2-yl)cyclohexa-1,5-dien-1-yl]methoxy]benzonitrile 2-[4,5-dihydroxy-6-(morpholine-4-carbonyl)naphthalen-1-yl]-3-methoxy-8a-methylnaphthalene-1,4-dione 2-(3,4-difluorophenyl)-1,5-dimethylimidazole (2R,3S)-2-methyl-5-oxo-6-phenyl-N-[(4-oxo-3H-thieno[3,2-d]pyrimidin-2-yl)methoxy]hexanamide 2-(1,3-benzothiazol-6-ylmethylideneamino)-5-propan-2-ylphenol (2S)-1-[[3,5-difluoro-4-(4-fluorophenyl)benzoyl]amino]-N-[(2R)-2-(hydroxymethyl)cyclohexyl]pyrrolidine-2-carboxamide 1-[5-chloro-2,4-dihydroxy-3-(3-morpholin-4-ylpropyl)phenyl]ethanone 3-[1-(dimethylamino)ethenyl]-5-[2-oxo-2-[(4R,6S)-8-azaspiro[4.5]decan-4-yl]ethoxy]benzonitrile 5-[4-fluoro-3-[7-(5-methylthiophen-2-yl)-1H-imidazo[4,5-b]pyridin-2-yl]-2H-pyrazolo[3,4-b]pyridin-5-yl]-N,N-dimethylpyridin-3-amine 2-[(2Z,5S)-2-[(Z)-1-(4-bromophenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazolidin-5-yl]acetic acid 4-[2,5-dimethyl-3-[(2R)-1-(6-pyridin-2-ylpyridazin-3-yl)propan-2-yl]oxyphenoxy]benzonitrile 1-[2,4-dimethoxy-6-(1H-pyrazol-5-yl)phenyl]-3-[4-(triazol-1-ylmethyl)-3-(trifluoromethyl)phenyl]urea 2-[6-(2-diazohydrazinyl)pyridin-3-yl]ethanol 2-methylsulfonyloxy-3,4-dihydrochromene-6-carboxylic acid 2,3-dichloro-5H-benzo[b]phenanthridine 4-[1-[6-[5-(aminomethyl)oxolan-2-yl]pyridine-3-carbonyl]piperidin-3-yl]oxybenzonitrile 4-amino-2-[(3S)-pyrrolidin-3-yl]oxybenzonitrile 2-[3,5-dichloro-4-(4-methylsulfonylphenoxy)phenyl]-6-(ethoxymethyl)-1H-pyridazine (4R)-N'-[5-amino-2-(benzylsulfanylmethyl)phenyl]-N,1-dimethylpiperidine-4-carboximidamide 2-[1,4-diphenyl-5-(trifluoromethyl)pyrrol-3-yl]-1H-benzimidazole [1-[2-(4,4-dimethyl-5H-1,3-oxazol-2-yl)-6-fluorophenyl]piperidin-3-ylidene]methanolate 5-(2-hydroxyethyl)-4-methoxy-1H-imidazole-2-sulfonic acid 1-[(3R)-4-benzylpiperidine-3-carbonyl]azetidin-2-one;hydrochloride (2S)-N-methyl-1-[4-(trifluoromethoxy)phenyl]pyrrolidine-2-carboxamide 5-[(2R)-3,3-dimethylbutan-2-yl]-2H-triazole-4-carboxylic acid 4-(2,6-dibromophenoxy)-N'-hydroxypyridine-2-carboximidamide 2-[4,5-dimethyl-1-(1-phenyl-4H-pyridazine-3-carbonyl)pyrazol-3-yl]-N-ethoxy-N-formamidoacetamide 2-bromo-5-[[(E)-3-(4,6-dichloropyridin-3-yl)prop-2-enoyl]amino]benzoic acid 2-[azido(furan-3-yl)methyl]-1H-imidazole 2-[3,5-dibromo-4-(9H-fluoren-1-yloxy)phenyl]acetaldehyde 2,4-difluoro-N-[[6-[[5-(trifluoromethyl)pyridin-3-yl]amino]pyridine-3-carbonyl]carbamoyl]benzamide 2-[(3R)-4-[(E)-2-quinolin-6-ylethenyl]sulfonyloxolan-3-yl]acetic acid 4-[[3,5-bis(trifluoromethyl)benzoyl]amino]-N-cyclohexa-1,5-dien-3-yn-1-ylpiperidine-1-carboxamide 2,6-difluoro-N-(4-methoxyphenyl)-N,3-dimethylaniline 2-[4-(5,6-dimethyl-1H-benzimidazol-2-yl)cyclohexa-2,4-dien-1-ylidene]propanedinitrile 3-[6-ethoxy-5-fluoro-2-(4-hydroxyphenyl)indol-1-yl]-N,N-dipropylbenzamide N-[6-cyano-4-[1,3-dioxo-4-(2,2,2-trifluoroethyl)isoindol-2-yl]quinolin-7-yl]oxyacetamide N-[4-methoxy-2,6-di(propan-2-yl)phenyl]formamide 2-[1,3-dihydroxypropan-2-yl(ethyl)amino]-6-nitro-3H-quinazolin-4-one N-[3-(4-chlorophenyl)propyl]-2,5-dimethyl-6-pyrimidin-5-ylpyrimidin-4-amine N-(3,4-dimethylphenyl)-1-[(E)-pent-2-enoxy]methanimine 3-[2,4-dimethoxy-5-(2-oxoimidazolidin-1-yl)phenyl]cyclopropane-1,1,2,2-tetracarbonitrile (4S)-5,7,8-trihydroxy-2-(2-methylpropanoyl)chromen-4-one 4-N,6-dimethylpyrimidine-2,4-diamine;(E)-3-(7-nitroindol-1-yl)prop-2-enal 1-[4-[(4,6-dimethoxypyrimidin-2-yl)sulfamoyl]phenyl]-3-(1-ethylpyrrolidin-3-yl)urea (7R)-7-[4-fluoro-3-(trifluoromethoxy)phenyl]-N,2-dimethyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 6-(3-methylphenyl)imino-1,3-benzothiazole-2-thiol 4-[2,6-bis(ethenyl)-3,6-dioxohexanoyl]benzene-1,3-disulfonic acid 2-(4,5-dimethyl-3H-pyrrol-2-yl)-3,4,7,8-tetrahydro-1H-quinolin-4-amine 3-[1,1,1,2,3,3,3-heptafluoropropan-2-yl(pyridin-3-yl)amino]phenol N-[2,4-difluoro-3-(hydroxymethyl)phenyl]propane-1-sulfonamide 1-[4-(2,3,5,6-tetrafluorophenyl)piperazin-1-yl]propan-2-one 4-N,2-dimethyl-1-N,3-diphenylbenzene-1,4-disulfonamide N-[3,5-bis(trifluoromethyl)phenyl]-2-[3-chloro-4-(trifluoromethoxy)phenoxy]ethanimidate N-[5-[[(3R)-5,7-difluoro-2,3-dihydro-1H-inden-4-yl]oxy]pyridin-2-yl]cyclopropanesulfonamide 4-chloro-1,2-bis(3,5-diphenylbenzoyl)piperazine-2-carboxamide 1-[3,3-dimethyl-4-(oxan-2-yloxy)butyl]pyrazole-4-carboxylic acid 6-[(3S)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]oxy-2,3-dihydroisoindol-1-one 3-(6-azidohexyl)-5,8-dichlorotriazolo[4,5-d]pyrimidine (Z)-5-chloro-1-[4-[3-methyl-2,6-dioxo-4-(trifluoromethoxy)pyrimidine-1-carbonyl]piperazin-1-yl]-5-naphthalen-1-ylpent-3-en-2-one;2,2,2-trifluoroacetic acid 2-amino-4,8-dioxo-6-(2,3,5,6-tetrafluorophenyl)-1,3,7,9-tetrahydropyrimido[2,1-c][1,4]oxazine-10-carbonitrile 1-[3-(azidomethyl)-5-fluorophenyl]pyrrole N-[3-(trifluoromethoxy)phenyl]-2,4,5-triazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),5,7,9,11,15,17-heptaen-3-amine 3-[N-(benzenesulfonyl)-2,4-difluoroanilino]propanoic acid 4-chloro-N-[(4-chlorophenyl)methyl]aniline;1,3-dihydroindol-2-one 3-[[2,6-di(propan-2-yl)phenyl]iminomethyl]-N-(pyridin-3-ylmethyl)benzenesulfonamide;iron(2+);dichloride 5-bromo-N-[1-(2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]-3-methoxypyridine-2-carboxamide 2-(4-aminophenyl)-6,7-diethyl-3H-pyrrolo[3,4-f]benzimidazole-5,6-diol 3-[5-methyl-4-[(1Z)-1-pyridin-3-ylbuta-1,3-dienyl]-1H-pyrrol-2-yl]-5-pyrimidin-5-yl-2H-pyrazolo[3,4-b]pyridine 3-[1-(4-fluorophenyl)pyrazol-3-yl]piperidine;hydrochloride 3-[2-(4-iodo-1H-indol-2-yl)ethoxy]pyrrolidine-1-carboxylic acid 3-methylimino-N-(4-methylphenyl)-9-oxotriazole-4-carboxamide 4-[(3E)-6-methyl-4-oxohexa-1,3,5-trien-3-yl]benzonitrile N-[(4S)-3,3-difluoropiperidin-4-yl]-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide 4-(2,5-dimethylphenoxy)benzenecarboximidamide ethane;3-[(2Z,4E)-hexa-2,4-dien-3-yl]-6-methoxy-1H-benzimidazol-3-ium N-(6,7-dimethoxyquinazolin-4-yl)piperidine-3-carboxamide 1-(4,6-dimethylthieno[2,3-b]pyridine-5-carbonyl)-N'-hydroxypiperidine-3-carboximidamide 4-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[4-(2-ethoxyphenoxy)phenyl]pyridin-2-amine 1-azido-4-(3,5-dichlorophenyl)sulfanylpiperidine 5-[[4-(methoxymethyl)piperidin-1-yl]methyl]-4H-furo[3,2-b]pyrrole 6-[(5R,7S)-1,4,5,7-tetramethyl-8-oxo-9,10-dihydroacridin-2-yl]hexanoic acid 4-[5-[3,5-bis(4-hydroxyphenyl)phenyl]-1,2-oxazol-4-yl]phenol 2-[[6,7-dimethoxy-4-[(E)-3-(1H-pyrazol-5-ylamino)but-1-enyl]quinazolin-2-yl]amino]ethanol 4-hydroxy-2,7,7-trimethylbenzo[g]pteridine-6-thione 5-(2,6-dimethylphenyl)-N-[5-fluoro-4-[1-hydroxyethyl(propanoyl)amino]pyrimidin-2-yl]furan-2-carboxamide (2R,3S)-N-[5-chloro-4-fluoro-6-(triazol-2-yl)pyridin-2-yl]-1-methyl-2-(2-methylpropanoylamino)cyclohexane-1-carboxamide [4-[3-[2-(4-methoxyphenyl)pyrrolidine-1-carbonyl]piperidin-1-yl]piperidin-4-yl]carbamic acid 7-(3,4-dimethylphenyl)heptanenitrile (4R,5S)-2-(5-tert-butylthiophen-2-yl)imino-3-methyl-7-oxo-N-phenyl-1,4,6,8-tetrahydropyrido[1,2-a]pyrimidine-4-carboxamide 6-[3-(2,6-dichlorophenoxy)piperidine-1-carbonyl]pyridine-2-carboxamide 3-(2,6-difluorophenyl)sulfanyl-N'-hydroxypyridine-4-carboximidamide 4-N,4-N-ditert-butylbenzene-1,2,3-triamine 4-[3,5-dimethyl-2-(oxan-4-ylideneamino)cyclohexa-1,3-dien-1-yl]aniline 6-methyl-N-[(3S)-4-phenylpyrrolidin-3-yl]pyridine-2-carboxamide (3R,4S)-1-[2-fluoro-6-methyl-4-(trifluoromethyl)phenyl]-N-hydroxy-4-[2-(2H-pyrazolo[3,4-b]pyridin-3-yl)ethynyl]pyrrolidine-3-carboxamide N-[2-(4-hydroxyphenyl)ethyl]-7-phenylmethoxyquinoline-3-carboxamide (3R)-3-[4,5,7-trifluoro-6-(2-methylindazol-5-yl)naphthalen-2-yl]oxypyrrolidine 6-methoxy-1-(2,4,5-trifluorophenyl)indole 5-(1,1-difluoroethyl)-3-[2-[4-[hydroxy(pyridin-4-ylmethoxy)methyl]-4-phenylpiperidin-1-yl]-2-oxoethyl]pyrimidin-4-one 4-(1-aminocyclopropyl)-6-[5-chloro-2-(propan-2-ylsulfamoyl)phenyl]pyridine-3-carboxamide 1-(2,6-dimethylphenyl)-3-[1-[4-(1H-pyrrol-2-yl)piperidin-1-yl]ethenyl]urea 1-[2,6-di(propan-2-yl)phenyl]-3-iodo-2-[5-[1-[(1-methylpyrazol-4-yl)amino]ethyl]pyridin-2-yl]guanidine 2-(4,5-dichloro-1H-imidazole-2-carbonyl)cyclopentane-1-carboxylic acid 2-benzylsulfanyl-N-(3,4,5-trimethoxyphenyl)acetamide (6R)-7-[[2-fluoro-5-[(6-methoxypyridin-3-yl)amino]sulfanylbenzoyl]amino]-3,9-dimethylidene-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 2-fluoro-4-methyl-6-(triazolo[1,5-a]pyridin-3-yl)phenol 1-[[2,4-dichloro-3-(2H-tetrazol-5-yl)phenyl]methyl]piperidine 1-[[3-[4-[(2,4-difluorophenyl)methyl]piperazine-1-carbonyl]-5-phenylpyridin-2-yl]amino]ethenamine N-[2,6-di(propan-2-yl)phenyl]-3-methoxy-1,4,5,7-tetrahydropyrazolo[3,4-c]pyridine-6-carboxamide 2-[(E)-2-methoxyethenyl]-1,4-bis[(Z)-prop-1-enyl]benzene 1-(2-bromophenyl)-5,6-dichlorobenzimidazole 4-chloro-2,6-dinitrophenol (5E)-2,4-dimethyl-5-[(3-propan-2-yloxyphenyl)methylidene]pyrazole 2-(3-amino-5,6-dihydrobenzo[b][1]benzazepin-11-yl)acetamide (5E)-2-cyclopentylimino-5-[(3,4-dimethoxyphenyl)methylidene]-1,3-thiazolidin-4-one 1-chloro-6-[2-chloro-4-(difluoromethyl)phenyl]-5-methyl-3H-imidazo[4,5-b]pyrazine-2-thione 6-(3,5-dimethoxyphenyl)-N-[(1R)-2-hydroxycyclohexyl]-4H-imidazo[1,2-a][1,8]naphthyridine-3-carboxamide 4-[(5R,7S)-2-chloro-6-(methoxymethyl)-5,7-dihydropyrrolo[3,4-d]pyrimidine-5-carbonyl]piperazin-2-one (5E)-2-[4-[[4-(diethylamino)phenyl]methylidene]-3,5,10-triazatetracyclo[7.6.0.02,6.011,15]pentadeca-1(9),2(6),7,11,13-pentaen-12-ium-12-ylidene]-N-(3,5-dimethoxyphenyl)-3-oxobutanamide 2-[(4-chlorophenyl)sulfonylamino]-3-hydroxy-N,2-dimethylpropanamide 1-(2-azidoethynyl)-4-[2,5-bis(trifluoromethyl)phenyl]piperazine N-[5-[3-(1H-benzimidazol-2-yl)-1H-indazol-5-yl]pyridin-3-yl]cyclopentanecarboxamide (2E)-2-[5-amino-1-[3-[4-[2-fluoro-3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]piperidin-2-ylidene]acetic acid 2-(7,8-dimethylnona-3,6,10-trienyl)benzamide 4-[3,5-bis(trifluoromethyl)phenyl]piperidine 2-[3,5-difluoro-4-(trifluoromethoxy)phenyl]-6-ethyl-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalene 7-[2,6-dichloro-4-(trifluoromethyl)phenyl]quinazolin-8-ol 1-(3,5-dimethoxyphenyl)-N-[4-[2-[5-(methylideneamino)penta-1,4-dien-2-yl]pyridin-4-yl]oxyphenyl]cyclopropane-1-carboxamide 2-N-(5-fluoro-4-morpholin-4-ylpyrimidin-2-yl)-3-methoxy-5-(triazol-1-yl)benzene-1,2-diamine 2-[1-(4-ethylcyclohexanecarbonyl)piperidin-3-yl]-6-propanoyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one [(2S,4R)-1-acetyl-4-fluoropyrrolidin-2-yl]-methylidyneazanium;6-[4-(trifluoromethoxy)phenoxy]-1H-benzimidazole (7S)-5-[2-fluoro-4-(6-fluoroquinolin-3-yl)phenyl]-1-propan-2-yl-3,4,4a,5,7a-hexahydro-2H-pyrrolo[3,4-b]pyridin-6-one 5-amino-3-(4-methylsulfanylphenyl)pyrazine-2,6-dicarbonitrile N-[2-(2-butoxyethyl)-5-oxopyrrolidin-3-yl]-5-methylpyridine-2-carboxamide 3-azido-2,6-ditert-butyl-4-methoxyphenol 1-amino-3-methylsulfonyl-4-propanoylquinolin-2-one 2-(7-bromo-4-methoxyimidazo[1,5-a]quinoxalin-5-yl)acetonitrile 7-[(2,6-dichlorophenyl)methoxy]-N,N-diethyl-1H-indole-3-carboxamide 2-(4-methylcyclohexyl)oxy-5-nitropyridine 2-methoxy-1,4-di(pyrimidine-5-carbonyl)pyrrole-3-carboxylic acid 2-(3-fluorophenyl)-5,7-dimethylimidazo[4,5-b]pyridine 1-[2,6-difluoro-4-(2-methylbutanoyl)phenyl]-3-[5-ethynyl-4-[6-morpholin-4-yl-4-(trifluoromethoxy)cyclohepta-1,4,6-trien-1-yl]pyridin-2-yl]urea 3-amino-2-[5-[1-(2,4-dihydroxyphenyl)-4-ethylhexan-2-yl]-2-propylphenyl]benzoic acid N-(1,3-benzodioxol-5-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamide;hydrochloride 1-ethyl-N'-hydroxyindazole-3-carboximidamide 3-(N-naphthalen-2-yl-4-propylanilino)propane-1,2-diol (6S)-N-[2-(dimethylamino)ethyl]-6-(2,4-dimethyl-1,3-thiazol-5-yl)-4-oxo-6,7-dihydro-5H-triazolo[1,5-a]pyrazine-3-carboxamide (2S)-N-ethyl-2-[[1-methoxy-3-(4-phenylmethoxyphenyl)propan-2-ylidene]amino]-3-naphthalen-2-ylpropanamide 3-(2-chlorocyclohexa-1,5-dien-1-yl)-N-[(1R)-4-[6-(trifluoromethoxy)pyridin-3-yl]-1H-2,1]benzoxaborol-6-yl]propanamide 2-[5-(1,3,4-oxadiazol-2-yl)pentoxy]benzoic acid (3E)-1,2-dihydropyrrolo[2,3-b]acridine-3-carboxamide 2-[[3-hydroxy-3-(5-methyl-1,4-oxazepane-4-carbonyl)piperidin-1-yl]methyl]benzoic acid 6-[5-chloro-2,4-dimethyl-1-(oxetan-3-yl)pyrrole-3-carbonyl]-2-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one 5-(7-morpholin-4-ylquinazolin-3-ium-2-yl)cyclohepta-1,4,6-trien-1-amine 2-[5-[5-methyl-4-(5,6,7,8-tetrahydronaphthalen-2-yl)-1H-imidazol-2-yl]pyridin-3-yl]oxyethanamine 2-(4-fluorophenyl)-N-[3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]pyrrolidine-1-carboxamide 1-(2,4-dimethoxyphenyl)-N'-[(Z)-(3-ethoxy-4-hydroxyphenyl)methylideneamino]-5-oxopyrrolidine-3-carbohydrazide N-[3-[[1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carbonyl]amino]propyl]thiophene-2-carboxamide 2,6-ditert-butyl-4-[5-methoxy-3-(pyridin-4-ylcarbamoyl)indol-1-yl]sulfonylphenolate N-[(5S)-3-[4-fluoro-2-(2-methoxyethoxy)phenyl]-2,6-dioxo-1-(trideuteriomethyl)-4H-pyrido[2,3-d]pyrimidin-5-id-7-yl]-2,3,3,3-tetramethylbutanamide N-[(E)-3-(1-benzyl-7,9-dihydro-6H-imidazo[4,5-h]quinolin-8-yl)prop-2-enyl]but-1-en-2-amine 1-(4-chlorophenyl)propan-2-one;ethane;N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)cyclobutyl]formamide 3-(2,5-dimethylphenyl)-4-hydroxy-8-nitrochromen-2-one 2-[(3,4-dichlorophenyl)methyl]-6H-imidazo[1,5-a]imidazole 2-fluoro-N,1,3,9-tetramethyl-6H-pyrrolo[3,4-f]quinolin-7-imine 3-[2-[4-(2,3-difluorophenoxy)piperidine-1-carbonyl]indol-1-yl]piperidine-2,6-dione 3-(3,5-dimethylanilino)-2-hydroxypropanethioamide;1-[(E)-3-methoxybut-1-enyl]pyrrolidine 2-(4-chlorophenyl)-1,3-diphenylpropane-1,3-dione 3-amino-2,6-dimethylbenzenesulfonic acid;N-[(E)-1-(methylideneamino)prop-1-en-2-yl]-4-(trifluoromethoxy)aniline 1-[(3,5-dimethylphenyl)methyl]-3,6-dihydropyrrolo[3,4-c]pyrrole-2-carboxylate 2-[3,5-bis(trifluoromethyl)phenyl]sulfanylethanamine 1,3-bis[2,6-di(propan-2-yl)phenyl]imidazolidine N-[2-(N'-hydroxycarbamimidoyl)phenyl]formamide 4-[4-(2,6-difluorophenoxy)piperidine-1-carbonyl]-1H-pyrrole-2-carboxylic acid 1-ethyl-4-(1,1,2,2,3,3,4,4,5,5-decafluorohexyl)benzene 1-(2,3-dimethyloxan-4-yl)sulfonyl-7H-purine-6,8-dione 3-[4-chloro-5,8-dimethyl-7-(naphthalen-2-ylsulfanylamino)pyrido[3,4-b]pyrazin-6-yl]-N',2-difluorobenzenecarboximidamide [5-chloro-4-(2-ethyl-1,3-oxazol-5-yl)pyridin-2-yl]hydrazine (5S)-6-hydroxy-5-[3-methyl-7-oxo-4-[4-(2,4,4-trimethylpentan-2-yl)phenyl]-1H-pyrazolo[4,3-c]pyridin-6-yl]hexanamide 2-[8-(4-chlorophenyl)-6-ethyl-7-methyl-2,3-dihydro-1H-pyrrolo[3,2-e]indol-5-yl]-N'-hydroxyethanimidamide;ethane 2-[[3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]carbamoylamino]-5H-thieno[3,2-b]pyridine-7-carboxylic acid N-benzyl-4,7-dimethylquinolin-8-amine;ethane 4-(2,5-dichlorothiophen-3-yl)-N'-methanimidoyl-1H-pyrrole-2-carboximidamide (5-azido-4,6-dimethylpyrimidin-2-yl)-phenyl-thiomorpholin-4-ylmethanone (4Z)-4-[(2,6-dichlorophenyl)methylidene]-2-ethylsulfanyl-1H-imidazol-5-one 4-[[2-fluoro-6-(trifluoromethyl)phenyl]methoxy]benzaldehyde 2-[4-[(2,6-difluorophenyl)methoxy]phenyl]benzoic acid 2-chloro-N-(3-chloro-4-fluorophenyl)-11-oxopyrido[1,2-b]isoquinoline-6-carboxamide (E)-2-[2,3-bis(trifluoromethyl)phenyl]-1,4,5,6,7-pentahydroxyhept-2-en-3-one 1-[4-(4,5-dihydroimidazol-1-ylmethoxy)phenyl]-N,2-dimethylpropan-1-imine 2,3-dimethyl-7-[(3R)-3-phenylpyrrolidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one 3-[4-(9H-fluoren-2-yl)phenoxy]propanoate 5-(trifluoromethyl)indole-1,3-dicarboxylate N-(4-benzylsulfanylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide [4-(1,5,7,10-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-12-yl)piperidin-1-yl]-pyrrolidin-1-ylmethanone 3,6-dimethyl-N-[1-(2-oxo-1H-pyridine-4-carbonyl)piperidin-3-yl]pyrazine-2-carboxamide 3-[(2S,3R)-1-azido-5-oxopyrrolidine-2-carbonyl]chromen-2-one 1-(7,8-difluoroquinolin-4-yl)ethanol ethane;1-phenyl-4,5-dihydroimidazole;propane 5-(2,3-dimethylphenyl)iminopentanamide 5-[2,3-dihydroxypropyl(naphthalen-1-yl)amino]-1H-pyrimidine-2,4-dione 2-[(Z)-[amino-[4-methyl-3-(trifluoromethyl)phenyl]methylidene]amino]guanidine;N'-methoxy-5,6-dihydronaphthalene-2-carboximidamide 4-[[2,6-difluoro-4-(4-methylphenyl)phenyl]-hydroxyphosphanyl]-N-ethoxy-1,5-dimethylpyrazole-3-carboxamide N-[1-[6,7-dimethoxy-5-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]piperidin-4-ylidene]hydroxylamine 5-hydroxy-8,10-dihydrothieno[2,3-c]acridine-7,9-dione 3-[2-[(6R)-6-methyl-1,4,5,7-tetrahydropyrazolo[3,4-c]pyridin-3-yl]ethynyl]benzonitrile (2-amino-4,6-dimethoxyphenyl)-(7-fluoroimidazo[1,2-a]pyridin-3-yl)methanone 2-[(1R)-1-azidoethyl]-6,7-dimethoxynaphthalene N-(cyclopropylmethoxy)-2-(3,4-difluorophenyl)-3-[5-fluoro-6-(1,1,1-trifluorobutan-2-ylamino)pyridin-3-yl]imidazo[1,2-b]pyridazin-8-amine 3-[1,3-benzodioxol-5-ylmethoxy(pyridin-2-yl)carbamoyl]cyclohexane-1-carboxylic acid 4-[2-methylpropyl(1,3-thiazol-5-yl)amino]butan-1-ol 6-amino-4-(2,3-difluoro-5-nitrophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamide 2-(3,4,5-trimethoxyphenyl)imino-1H-benzo[g]pteridin-6-one 5-[(3,5-difluorophenyl)methyl]-N-[4-(3,3-dipropylcyclohexa-1,5-dien-1-yl)oxyphenyl]pyridine-2-carboxamide (1-azido-2,4-dimethylpiperazin-1-yl)-[3-[6-(2-ethoxyphenyl)imidazo[1,2-a]pyridin-7-yl]phenyl]methanone 5-[1-(4,4-difluorocyclohexyl)imidazol-2-yl]-2-methoxybenzoic acid 1-[4-(2-chlorophenyl)-5-methoxypyrimidin-2-yl]-3-ethylurea N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1H-pyrrole-2-carboxamide 2-(3,5-dimethylpyrazol-1-yl)-N-[4-[(6R)-7-oxo-4,6-dihydrotriazolo[1,5-a]pyrazin-5-yl]phenyl]acetamide (2R)-N-[1-cyclohexyl-3-[5-[(Z,4E)-2-fluoro-4-hydroxyimino-6-methoxyhept-4-en-2-yl]-1,3,4-oxadiazol-2-yl]propan-2-yl]-2-phenylpentanamide [(2S,3R)-1-amino-4-methyl-5-oxo-7-pyridin-3-ylsulfonylazepan-3-yl]carbamic acid 3-(2-ethoxybenzoyl)-7,8-dimethoxychromen-4-one N-[4-(2-bromophenyl)oxan-4-yl]-6,7-dimethoxy-1H-indole-2-carboxamide N-azido-6-chloro-5-[2-(1,1-difluoroethyl)phenyl]pyridine-3-sulfonamide 5-[(2,4-dichlorophenyl)methylsulfanyl]-3H-1,3,4-thiadiazol-2-one (7R)-2,2-dimethyl-3-(3-methylpyridine-4-carbonyl)cyclopropan-1-one N-butyl-6,6-dimethyl-2-(4-phenylphenyl)octanamide N-(2,3-dihydro-1H-inden-5-yl)-5-methoxynaphthalene-2-carboxamide N-(4-methoxyphenyl)-4-[(3Z,6E,8S)-5-methylsulfanylnona-1,3,6,8-tetraen-2-yl]aniline 2-tert-butylsulfanyl-1,4-difluoronaphthalene 4-(3-methylpyridin-4-yl)-1,2-thiazol-5-amine 6-azidooxy-2,3-dichloropyridine 4-[2-(3,5-dimethylpyrazol-1-yl)propanoyl]-8-phenyl-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-9-one (2R,3S)-1-[[(2E,4Z)-6-[4-methoxycarbonyl-N-methylanilino]hexa-2,4-dienoyl]amino]-3-methylpyrrolidine-2-carboxylic acid 1-[4-methoxy-7-(3-piperidin-1-ylpropoxy)naphthalen-2-yl]ethanone 3-[(E)-1,2-diamino-2-(3-chlorophenyl)ethenyl]sulfanylpropanenitrile (2R,3S)-1-methyl-5-oxo-N-[(5-thiophen-2-yl-1H-pyrazol-4-yl)methylideneamino]pyrrolidine-2-carboxamide 2-(4-chlorophenyl)-1-methyl-6,7-dihydropyrrolo[3,2-c]pyridine (5R,7S)-N-[(3-methylphenyl)methyl]-2-[(4-methylphenyl)methylsulfanyl]-5,7-dihydrofuro[3,4-d]pyrimidine-5-carboxamide 3-(3,5-dimethylphenyl)-6-hydroxyiminopiperidine-2,4-dione 2,4-dimethyl-6-(phenylsulfanylamino)phenol;ethane 2-(N-butyl-4-methoxyanilino)ethanol 1-(3,5-ditert-butylphenyl)-2-[(Z)-(4-hydroxycyclohexyl)methylideneamino]guanidine 2-cyclohepta-1,3,6-trien-1-yl-5-methyl-4H-indeno[1,2-d]pyrimidine;ethane N-[6-(2-iodoethyl)pyridin-3-yl]acetamide 4-[3,5-bis(trifluoromethyl)phenyl]piperidine-2-carboxylic acid N'-ethyl-N-[6-(3-hydroxyphenyl)-1H-indazol-5-yl]-2,4-dioxopyrimidine-1-carboximidamide 4-[1-(cyclohexylmethoxy)ethenyl]-5-methyl-3,4-dihydro-2H-chromene 2-(3,4-dichlorophenyl)-5,6-diethyl-7-methyl-1H-imidazo[1,2-a]pyrimidine;ethane 2-(cyclobutylmethylamino)-N-[3-hydroxy-4-[6-(2-methoxyphenyl)-7H-pyrrolo[3,2-d]pyrimidin-4-yl]phenyl]acetamide [2-fluoro-3-(methylamino)pyridin-4-yl]-[3-methoxy-4-(1,3-thiazol-5-yl)pyrrolidin-1-yl]methanone 4-[(3Z)-2,6-dimethylhepta-1,3,5-trien-4-yl]-2-fluoro-N,5-bis(2-hydroxyethoxy)benzamide N-methoxy-N,3-dimethyl-2-propanoylbenzamide N-[(2R,3S)-5-[(4-chlorophenyl)sulfonylamino]-3-hydroxy-1-methyl-6-oxo-8-pyrimidin-4-yloctan-2-yl]carbamate 1,4-dibromo-6,6-bis(methoxysulfanyl)cyclohexa-2,4-dien-1-amine 2,4-dimethyl-1'-(6-phenylpyridin-3-yl)spiro[5H-pyrazolo[3,4-d]pyrimidine-7,4'-piperidine] 2-[5-chloro-4-(2,4-difluorophenyl)-1H-pyrazol-3-yl]piperidine-1-carboxylic acid (2S)-2-[(6-aminopyridine-3-carbonyl)-methylamino]-N-[(1R,3S)-3-[4-cyano-3-(trifluoromethyl)phenyl]cyclopentyl]butanamide;2,2,2-trifluoroacetic acid 2-[3-(6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonyl)phenyl]acetic acid 7-(4-chlorophenyl)-2,5-dimethyl-N-[2-[methyl-[[4-[methyl(2,2,2-trifluoroethanimidoyloxy)amino]phenyl]methyl]amino]-2-oxoethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 1-azidooxy-3,4,5-tris(phenylmethoxy)cyclohexa-2,4-diene 2-(2-methyl-6-oxopyridin-1-yl)-N-[(5S,7R)-3,4,5,6-tetrahydroimidazo[1,2-a]azocin-9-yl]propanamide (3E)-4-amino-3-[[1-(2,6-dichlorophenyl)pyrazol-4-yl]methylidene]azete-2-thione (2-propan-2-ylsulfanylphenyl)-[4-(6H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]methanone N-ethyl-2-methoxy-4-(5,6,7,8-tetrahydro-1,6-naphthyridin-3-yl)aniline 1-(2,4-dimethoxyphenyl)-2-[4-[1-(5-methylsulfanylpyrimidin-2-yl)piperidin-3-yl]butyl]hydrazine 4-[(2-aminobenzoyl)amino]benzenesulfonate (6R,11bR)-9,10-dimethoxy-3-(4-nitrobenzoyl)-6-phenylmethoxy-2,6,7,11b-tetrahydro-[1]benzofuro[2,3-a]quinolizin-12-one 2-(azetidin-1-yl)-5,6,7,8-tetrahydroquinoline 6-fluoro-4-[2-(oxan-3-yl)ethoxy]quinazoline (5Z)-2-(3,4-dimethylphenyl)imino-5-[[1-[(4-nitrophenyl)methyl]indol-3-yl]methylidene]-1,3-thiazolidin-4-one 5-[4-(6,7-dimethoxyquinazolin-4-yl)phenyl]-N-(2-fluorophenyl)-1H-pyrrole-3-carboxamide 3-[5,7-difluoro-2-(4-fluorophenyl)quinolin-6-yl]-1-methoxycarbonylpyrrolidine-3-carboxylic acid 3-chloro-N'-hydroxy-2-(4-methoxyphenyl)quinoline-4-carboximidamide 2-[azido(fluoro)methyl]-4-bromobenzenesulfonic acid 5-methyliodanuidyl-N-[4-(trifluoromethoxy)phenyl]pyridine-3-carboxamide N-(4,6-dimethylpyrimidin-2-yl)-5-[ethyl(3-phenoxypropyl)amino]pentanamide N-[(5S)-4,8,9-trioxo-1H-furo[2,3-h]chromen-7-yl]pyrrolidine-2-carboxamide 5-cyclobutyl-N'-[2-(4-fluorophenyl)-1H-pyrrolo[3,2-b]pyridine-6-carbonyl]pyrazine-2-carbohydrazide 2-[3-ethylsulfonyl-5-(trifluoromethyl)pyridin-2-yl]-1-fluoro-6-nitrophthalazine 2-(2,2-dimethylpropanoyloxy)naphthalene-1,4-disulfonic acid 1-(1-azido-9H-fluoren-2-yl)piperidine (2Z)-1,3-diphenylbuta-2,4-dien-1-one 6-[(E)-2-(1,3-dioxan-2-yl)ethenyl]-5H-[1]benzothiepino[4,5-b]pyridine 2-[(E)-3-azidobut-1-enyl]-6-methoxynaphthalene 2-[(2Z)-3-methylpenta-2,4-dienylidene]-3H-inden-1-one (E)-1-[4-(4-aminophenyl)sulfanyl-6-methoxyquinolin-3-yl]but-1-en-1-ol 2-(7-amino-3,4-dihydronaphthalen-1-yl)oxyethanol 4-amino-5-(2-methylpropanoyl)-1H-imidazole-2-carbohydrazide N-methyl-1-[6-(1H-pyrrole-2-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]pyrrolidine-2-carboxamide 2-[(4S)-4-(benzylamino)-6,8-dichlorospiro[1,3-dihydroisoquinoline-4,3'-pyrrolidine]-2'-yl]-N,N-dimethylacetamide;cyclohexanamine 1-[2-(2-butan-2-ylphenoxy)ethoxy]-4-ethoxy-5,6,7,8-tetrahydronaphthalene 1-(5-aminoisoquinolin-3-yl)propan-1-one 2-(3,5-dimethylpiperazin-1-ium-1-ylidene)pyrido[4,3-d]pyrimidine 4-[3-(6,7-difluoroquinolin-5-yl)-1H-pyrazole-5-carbonyl]-2,6-dimethoxycyclohexane-1-carboxylic acid 5-azidooxy-3-ethylsulfonylpyridine 2-[N'-(3-nitrophenyl)carbamimidoyl]benzamide;hydrate N-[4-(cyclohexylmethyl)pyrimidin-2-yl]-5,6-difluoro-1H-indole-3-sulfonamide [2-hydroxy-4-(2,2,2-trifluoroethyl)-6-azaspiro[2.5]octan-6-yl]-(3-methoxyphenyl)methanone (E)-N-methylsulfonyl-3-[5-oxo-4H-1,2,4]triazin-6-yl-N-(thietan-2-ylmethyl)prop-2-enamide 4-amino-1-[1,3]thiazolo[5,4-h]quinoline-2-thione;ethane 4-[2,5-bis(trifluoromethyl)phenyl]sulfonyl-3-(1-ethoxyethenyl)-1,1,2,2,6,6-hexafluoropiperidine 2-(4-bromo-N-cyclohexyl-3,5-dimethylanilino)decanoic acid 2-[(4R)-3,9,10,12-tetrahydroperylen-4-yl]benzamide 4-[5-(1,3-benzodioxol-5-yl)pyrazol-1-yl]phenol 2-azidosulfanyl-5-tert-butylsulfinylthiophene N-cyclopropylformamide;2-[2-hydroxyethyl(methyl)amino]acetaldehyde;4-(3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,3,6,8,11-pentaen-4-ylmethoxy)phenol 1-(2,3-dihydro-1H-indene-5-carbonyl)-3,7-dimethyl-4,6,8,9-tetrahydropyrazolo[3,4-c]isoquinolin-5-one N-[[5-chloro-2,3-dimethoxy-6-[(E)-2-(4-methylphenyl)ethenyl]phenyl]methyl]formamide;ethane (5S)-1-(4-fluoro-3-morpholin-4-ylphenyl)-2,7-dimethyl-N-[5-(trifluoromethoxy)pyridin-3-yl]-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-3-carboxamide 4-[(E)-3-(2,5-dimethoxyphenyl)prop-2-enoyl]-N'-hydroxy-1H-pyrrole-2-carboximidamide 3-(1-benzylpiperidin-4-yl)-N-cyclopropylpyridine-2-carboxamide 2-[1-(2,4,6-trimethylphenyl)imidazol-4-yl]pyridine;platinum 4-[2-(7,8-dihydronaphthalen-1-yl)propanoyloxy]butanoic acid N-[3-[(2S)-4,5-dihydroxy-2-methoxy-6-(3-methylbut-3-enyl)oxan-2-yl]phenyl]-3,5-diethoxybenzamide 2-(4-ethenylsulfonylphenyl)ethanesulfonic acid 6-[3-(azepan-1-yl)propoxy]pyridine-2,4-diamine 4-[5-[[1,3-dioxo-2-(4,4,4-trifluorobutyl)isoindol-5-yl]amino]-3-[2-methoxyethyl(methyl)amino]pyridine-2-carbonyl]piperazine-2-carboxylic acid 6-(3-hydroxypropoxy)naphthalene-2-carbonitrile N'-[2,4,6-trimethyl-3-(pyridine-2-carbonyl)phenyl]carbamimidate 4-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]benzonitrile N-(2,5-dimethoxyphenyl)sulfanyl-6-nitro-1H-indol-7-amine 2-[N-(carboxymethyl)-3,5-bis(trifluoromethyl)anilino]acetic acid 4-(3-chloro-2,6-difluorophenyl)-1H-pyrazole 1-(3,5-difluoro-2-methylphenyl)butane-1,3-dione 3-[3-(7-bromo-4-methoxyindol-1-yl)propyl]cyclopentane-1-carboxylic acid 7-azidooxy-N,3-dimethyl-1H-indole-2-carboxamide (2S,5R)-4-[1-(3-chlorophenyl)triazole-4-carbonyl]oxy-5-methylmorpholine-2-carboxylic acid 1-(2,5-dimethoxyphenyl)-N'-methylsulfanylsulfonylcyclobutane-1-carbohydrazide 2-cyclopentyloxy-6-fluorobenzaldehyde 4-[(2-azidobenzoyl)amino]butanamide (2S)-N',2-bis[3,5-dichloro-4-(dimethylcarbamoyloxy)phenyl]pyrrolidine-1-carboximidamide 2-amino-3-(1,1,2,2,2-pentafluoroethyl)-6-[4-(trifluoromethoxy)phenyl]-5H-pyrido[2,3-d]pyrimidine-4,7-dione 1-[2-azidooxy-5-(3,4,5-trimethoxyphenyl)pentyl]-4-(trifluoromethylsulfonyl)benzene 5-(furan-2-yl)-N-[3-[1-[1-(hydroxymethyl)cyclopentanecarbonyl]pyrrolidin-3-yl]oxyphenyl]pyridine-3-carboxamide 2-[2-(3-methylbutoxy)ethyl]terephthalic acid 1-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridine-7-carbonyl)piperidine-2-carboxylic acid N-[2-[3-(1H-indol-2-yl)phenyl]propan-2-yloxy]benzenesulfonamide 4-[(3S)-1-[(2,5-dimethylpyrazol-3-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-6-one 5-[(5E)-5,6-dimethylhepta-1,3,5-trien-2-yl]sulfonyl-N-[(4-fluorophenyl)methyl]-2,4-dihydroxybenzamide 1-azido-3-propylnaphthalene 4-[2-[5,7-bis(cyclopropylmethoxy)-1H-indol-3-yl]propan-2-ylamino]-N'-hydroxypyridine-2-carboximidamide N-(1,3-benzodioxol-5-ylmethyl)-2-(5-iodo-3-methoxypyridine-4-carbonyl)-9-oxa-2-azaspiro[5.5]undecane-4-carboxamide ethane;2-methoxy-4,6-bis(2-phenylpropan-2-yl)phenol 2-azidooxy-1,3,4-tris(trifluoromethyl)benzene 4-[[(1S)-1-cyclopropylethyl]amino]-2-methoxypyrimidine-5-carboxamide 2-[[4-(3,5-diaminophenyl)sulfanylbenzoyl]amino]benzoic acid 1-[(Z)-3-(2,5-dioxopyrrol-1-yl)-5-phenylpent-4-enoxy]-N,N'-diethylethanimidamide 2-hydroxy-N-[3-(methanesulfonamido)cyclobutyl]pyrimidine-5-carboxamide 4-[(3,5-dimethylpyridin-2-yl)amino]-N-(1,4,6,7-tetrahydropyrano[4,3-c]pyrazol-3-ylmethyl)benzamide 5-(4,7-difluoronaphthalen-1-yl)-N-piperidin-3-ylpyrazine-2-carboxamide 4-hydroxy-2,3-bis(sulfanyl)benzoic acid (2E,4Z)-N-[4-amino-3-(1H-indole-2-carboximidoyl)phenyl]-3-(cyclohexylmethoxy)-2-methylhepta-2,4,6-trienenitrilium 3-bromo-4,7-dimethoxynaphthalene-1-sulfonic acid 4-[[2-(1H-indole-3-carbonylamino)acetyl]amino]butanoic acid N-(furan-2-ylmethyl)-3-(4-methoxyphenyl)sulfanyl-N-[[1-[[5-(trifluoromethyl)pyridin-2-yl]methyl]pyrazol-4-yl]methyl]propanamide 3-[(2R)-butan-2-yl]oxy-N'-hydroxypyridine-4-carboximidamide N-[3-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)propyl]-1-(pyridine-4-carbonyl)piperidine-3-carboxamide 1-[3,6-bis(4-tert-butylphenyl)-2H-pyrazin-5-ylidene]-3-dibenzofuran-4-ylthiourea 4-(4-azidophenyl)-N,N-dimethylaniline N-[3-fluoro-4-[[7-(2-fluoro-6-methoxyphenyl)-1,5-naphthyridin-4-yl]oxy]phenyl]-3-oxo-4H-naphthalene-1-carboxamide N-(5-chlorothiophen-2-yl)sulfonyl-3-methoxy-1H-pyrazole-5-carboxamide [6-(4-methylpiperidin-1-yl)pyridine-3-carbonyl]oxyboronic acid 3-(1,2,2a,8b-tetrahydrocyclopropa[a]naphthalene-5-carbonylamino)pyridine-4-carboxylic acid 4-[2-(3,3a,4,5,6,7,7a-octahydroisoindol-1-yl)ethoxy]benzamide N-(5-tert-butylpyridin-2-yl)cyclopentanecarboxamide;dihydrochloride 5-[4-(2,2,2-trifluoroethoxy)phenyl]pyrimidine 5-[(2E,4Z)-hepta-2,4,6-trienyl]-3-(1H-pyrrolo[3,2-b]pyridin-2-ylmethylideneamino)thiophene-2-carboxylic acid 3,7-ditert-butyl-1,2,4,5,6-pentamethylbenzimidazol-1-ium 3-[3,5-difluoro-4-(7-oxononyl)phenyl]propanoic acid 4-(2,6-difluoro-3-methoxyphenyl)-1H-tetrazol-5-one (NE)-N-[2-(3,5-dichlorophenyl)-1-[3-[4-(2H-tetrazol-5-ylmethoxyimino)piperidine-1-carbonyl]phenyl]ethylidene]methanesulfonamide 4-[(2R)-1,3-bis(4-fluorophenyl)propan-2-yl]oxy-N-(5-fluoropyrimidin-2-yl)-3-methylbenzamide 3-amino-2,6-dichlorobenzenesulfonic acid N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-(methoxymethyl)-6-oxo-2-propan-2-yl-1H-pyrimidine-5-carboxamide 4-hydroxy-5,7,11-trioxa-13-azatricyclo[8.4.0.02,6]tetradeca-1(10),9,12-triene-8,14-dione (1R,2S)-2-[5-amino-4-methyl-3-(trifluoromethyl)pyrazol-1-yl]cyclohexan-1-ol;hydrochloride (3R,4R)-3-azido-4-phenylpiperidine 1-[2,4-di(butan-2-yl)phenyl]-N-methoxyethanethioamide 4-[5-(2-cyano-3-methylphenoxy)-6-propanoyl-1,3-dihydroisoindol-2-yl]butanamide (5R)-3,3-bis[3-fluoro-4-(trifluoromethyl)phenyl]-5-methyl-1,2-oxazolidine 1-[4-(5,6-dimethoxy-2,3-dihydro-1H-indene-2-carbonyl)piperazin-1-yl]-2,2,2-trifluoroethanone;2,2,2-trifluoroacetic acid 3-[(4R)-2-oxopiperidine-4-carbonyl]benzoic acid N-[4-[3-(oxolan-2-ylmethoxy)propanoyl]phenyl]butanamide (2R)-2-[(4-bromophenyl)sulfonylamino]-3-hydroxypropanoic acid N-[3-(5-azidooxythiophen-2-yl)-1,7-naphthyridin-6-yl]propanamide 2-[(Z)-1-hydroxypentan-3-yl]-5,6,7-trimethoxy-4H-1,3-benzodioxin-8-ol [[5-(4-chlorophenyl)furan-2-yl]methylideneamino]thiourea N-[6-(1H-indole-2-carbonyl)pyridin-3-yl]-5-methoxypyridine-3-carboxamide 4-methoxy-3-[[4-(4-propan-2-ylphenyl)cyclohexyl]methylamino]benzaldehyde ethane;4-(3-methoxyphenyl)-1-piperidin-4-ylbutan-2-one 4-[2,2-dimethylpropanoyl(pent-1-en-3-yn-2-yl)amino]thiophene-2-carboxylic acid 2-[8-chloro-1,3-dimethyl-6-(1H-pyrrol-2-yl)-4,9b-dihydro-1aH-cyclopropa[c]quinolin-7-yl]acetamide 4-[2,5-dimethyl-1-(naphthalen-1-ylmethyl)pyrrol-3-yl]-N,N-bis(2-phenylethyl)cyclohexa-2,4-diene-1-carboxamide 5-butyl-2,3-dihydrothiophene-4-carboxylic acid 3-[(2E,4Z)-hepta-2,4,6-trien-3-yl]-5-methyl-1H-pyrrolo[2,3-b]pyridine [(E)-2,3-bis(4-methoxyphenyl)but-1-enyl]benzene 4-[2,3-bis(trifluoromethyl)phenyl]-N,1-dimethylpiperidin-4-amine 4-methoxy-3-(6-methyl-1H-benzimidazol-2-yl)benzenesulfonamide 1-(1H-benzimidazol-2-yl)azepane;1-methylpiperazine 2-amino-1,3-bis(benzenesulfonyl)propan-1-ol 2-[3-[(Z)-2-aminoethenyl]-5,6-dimethoxyindazol-1-yl]-N-cyclopropyl-6-azaspiro[2.5]octane-6-carboxamide 4-[1-azidooxy-2-(trifluoromethyl)dec-9-enyl]phenol 4-[3-(methoxymethyl)piperidin-1-yl]-6-methylpyridine-2,3-dicarbonitrile 2-[(4R)-6,7-dimethoxy-1-[4-(4-methylpiperazin-1-yl)phenyl]sulfonyl-3,4-dihydro-2H-isoquinolin-4-yl]acetic acid 2-amino-3-[4-(2,4-difluorophenyl)phenyl]propanoic acid;hydrochloride 1-(2-azidooxy-4,5-difluorophenyl)ethanamine 1-(4-bromophenyl)-3,5-dichloro-2H-pyridine 2-[3-(methylsulfanylmethoxy)phenyl]sulfonylpropanedinitrile 2-methyl-5,7-dioxobenzo[b]phosphindole-6,9-dicarboxylic acid 6-[2-[(4-butan-2-yloxy-3-methoxyphenyl)methylidene]hydrazinyl]pyridine-3,5-dicarbonitrile N-[2-(4-cyanophenyl)-3-(6-fluoro-1H-indol-3-yl)propyl]-N-methylmethanesulfonamide [4-(1,3-benzothiazol-2-yl)phenyl]boronic acid 2-[(5R)-4,7-dioxo-2-propylsulfanyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidin-5-yl]-N-[(3,4-dimethoxyphenyl)methyl]acetamide N-[3,5-dimethyl-4-(4-oxopentanoyl)phenyl]acetamide 2-[4-[[3,5-dichloro-4-(cyclopropylcarbamoyl)phenyl]methylamino]phenoxy]acetic acid;ethane 4-(aminomethyl)-1-(2,2-diphenylacetyl)-5-[3-fluoro-5-(2-methoxypyridin-4-yl)phenyl]pyrrolidine-2-carboxylic acid 2-[(7,8-dimethoxy-2-oxochromene-3-carbonyl)amino]acetic acid 6-(2-chlorophenyl)-3-methylsulfanylhexanoic acid 1-(5,6-dimethylimidazo[2,1-b][1,3]thiazol-3-yl)cyclopentan-1-amine 4-(2-aminoethyl)-6-(benzenesulfonylmethoxy)pyridine-3,5-dicarboxylic acid 2-chloro-5-[(3E)-4,5-dimethylhepta-1,3,5-trien-3-yl]benzenecarboximidamide 1-[4-[(7R,8aS)-7-[2-[4-(2-hydroxyethoxymethyl)phenyl]acetyl]-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-1-yl]piperidin-1-yl]propan-1-one 5-(3,4-dihydroxyphenyl)-2,3-bis[[1-ethyl-6-(trifluoromethoxy)benzimidazol-2-yl]methylideneamino]cyclohexa-2,4-dien-1-one N-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)piperidine-4-carboxamide 3-[2-(3-bromo-4,5-difluorophenyl)ethynyl]-6-[3-(trifluoromethyl)phenyl]pyridazine (2S)-1-[4-(3,4-dichlorophenyl)piperidin-1-yl]propan-2-ol 1-methoxy-4-[3-(trifluoromethyl)phenyl]sulfanylpiperazine N-(5-chloropyridin-2-yl)-3-methoxy-4,9-dihydroacridine-1-carboxamide;ethane N-[2,3-difluoro-4-(5-pyridin-3-yl-1H-pyrazolo[4,3-b]pyridine-3-carbonyl)phenyl]-2-morpholin-4-ylethanesulfonamide 1-[2-chloro-3-(trifluoromethyl)phenyl]-2-[6-methoxy-7-(piperidin-4-ylamino)quinolin-3-yl]ethanone 3-[4-[6-[[(2S)-1,4-dioxan-2-yl]methoxy]-5-fluoropyridin-3-yl]-2-fluorophenyl]-5-fluorophenol N-[1-[2,6-dimethoxy-4-(4-propan-2-ylpiperazine-1-carbonyl)phenyl]ethyl]formamide 2-(4,6-dimethylquinolin-3-yl)oxy-5-(trifluoromethyl)aniline 2,6-dichloro-N-[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]benzamide (6R)-7,8-diamino-10-oxo-2,3,5,6-tetrahydro-1H-pyrido[3,4-f]quinoline-4-carbonitrile N-[(2S,3R)-1-hydroxy-5-oxo-4-propan-2-ylpyrrolidin-3-yl]-5-methoxypyridine-2-carboxamide (2S,3R)-3-acetyloxy-5-azido-N-[4-(3-chlorophenyl)butanoyl]azetidine-1-carboxamide 6-[2-(3,4-dichlorophenyl)ethyl]-N-methoxybenzotriazol-1-amine (1S,5R)-3-[[5-chloro-6-(oxolan-2-ylmethoxy)pyridin-3-yl]methyl]-7-pyrimidin-4-yl-8-azabicyclo[3.2.0]heptan-6-one N-[5,6-dimethyl-3-(2H-pyridin-1-id-4-yl)pyridin-2-yl]formamide;yttrium N-(4,4-dichlorocyclohexyl)-1H-pyrrolo[3,2-c]pyridine-2-carboxamide 4-(1H-benzimidazol-2-yl)-N-[3,5-dichloro-4-[(3R)-3-methoxypyrrolidin-1-yl]phenyl]benzamide 5-[2,3-dichloro-4-(propanoylamino)phenyl]pentanoic acid 1,5-dimethyl-3-(2-methylphenyl)isoquinoline 1-cyclopentyl-7-[(3,4-dichlorophenyl)methyl]-3-methoxypyrrolo[2,3-c]pyridine 2-azido-1-[4-(trifluoromethoxy)phenyl]piperazine 4-azido-6-butylquinoline 2,6-difluoro-3-[4-[(4-pentylcyclohexyl)methoxy]phenyl]phenol N-[[5-(2-oxoimidazolidin-1-yl)thiophen-3-yl]methyl]piperidine-4-carboxamide 4-methyl-5-[2-[[(3S)-pyrrolidine-3-carbonyl]amino]thieno[3,2-b]pyridin-7-yl]oxyindole-1-carboxylic acid (3S)-7-[3-cyclopropyl-5-fluoro-4-(oxetan-2-ylmethoxy)phenyl]-5-oxo-3-pyridin-4-ylheptanal 7-(3,5-dichlorophenyl)pyrido[2,3-d]pyrimidine 5-[(3,4,6-trimethylquinolin-8-yl)amino]pentanoic acid [3-(furan-2-ylmethylamino)phenyl]-piperidin-1-ylmethanone 1-[(3S,4R)-2-oxooxolan-3-yl]-7H-purin-6-one 5-[3,6-diamino-2,4-dicyano-5-(3,4-dimethoxyphenyl)pyridin-1-ium-1-yl]pentanenitrile;chloride 2-benzylsulfanyl-N'-hydroxypyrimidine-4-carboximidamide N-azido-3,6-dichloropyridine-2-carboxamide N-(1,3-benzodioxol-5-ylmethyl)-2-[4-(4-fluorophenyl)-3-hydroxy-6-methyl-7-(trifluoromethyl)pyrazolo[3,4-b]pyridin-1-yl]acetamide 2-(1,3-benzodioxol-5-ylmethyl)-3-phenylisoindol-1-one 2-bromo-N-[1-(4-ethylphenyl)sulfonylpiperidin-4-ylidene]benzamide (6-amino-2-methylpyridin-3-yl)oxy-[4,5-bis(4-chlorophenyl)-4-methoxypentyl]phosphinic acid;ethane 1-benzyl-3-[6-(4-hydroxyphenyl)pyrido[2,3-b]pyrazin-3-yl]urea 5-chloro-3-methyl-2,4-diphenylphenol 4-[(3S,5R)-1-(4-cyclopropyl-2,6-dimethoxybenzoyl)-5-(hydroxymethyl)pyrrolidin-3-yl]oxybenzoic acid 2-[4-[5-[(2,4-difluorophenyl)methyl]nonanoylamino]-3-hydroxypiperidine-1-carbonyl]-4-propan-2-yloxypyridine-3-carboxamide 2-(4-fluorophenyl)propane-1,3-diol;N'-hydroxy-6-[methyl(thiophen-3-ylsulfonyl)amino]hexanimidamide 2-(3,4-dimethylbenzoyl)oxypropanoate 6-bromo-3-(3-chlorophenyl)iminospiro[1,4-dihydroquinoxaline-2,4'-piperidine]-5-carboxamide 2-[(2Z)-4-oxo-2-[(3-phenoxyphenyl)methylidene]-1,3-thiazolidin-5-yl]acetamide 4-(1,3-thiazol-2-yl)benzenecarboximidamide 2-azido-N',6-diphenylbenzenecarboximidamide 5-azidooxy-2,3-dimethyl-4H-pyrazolo[1,5-a]pyrimidine ethane;1-methylnaphthalene;8-[(3Z,5E)-5-methylidenehepta-1,3,6-trien-2-yl]dibenzofuran 2-(5-aminopentyliminomethyl)benzene-1,4-diol 2-azido-5-(6,8-dihydro-5H-[1,2,4]triazolo[3,4-c][1,4]oxazin-3-yl)pyridine-4-carbonitrile N-[2-(3,5-dimethylpiperidin-1-yl)ethyl]-4-oxo-3H-quinazoline-7-carboxamide N-[(E)-2,5-dimethylhex-3-enyl]propanamide;6-fluoro-7-N,1-bis(4-fluorophenyl)quinazoline-4,7-diamine N-[4-(5-amino-2,3-dihydro-1H-pyrazol-3-yl)phenyl]-2-methoxybenzamide (2R)-1-[4-(5-fluoroquinolin-7-yl)phenyl]propan-2-amine 3-[[1-(4,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]amino]propanoic acid 1-[5-(difluoromethyl)-2,3-bis(triazol-1-yl)phenyl]-N-methylmethanamine 4-[3-(3,4-dichlorophenyl)propyl]-2-phenyl-1H-imidazole N-[(1E,3Z)-2-methylpenta-1,3-dienyl]-4-(3H-pyrrol-2-ylmethylideneamino)benzamide (4S)-3-[2,6-difluoro-4-(methoxycarbonylamino)benzoyl]-4-phenyl-1,3-oxazolidine-5-carboxylic acid 6-[(E)-3,3-dimethylbutanoyl]pyridine-2-carboxylate 1-(2,5-dimethylfuran-3-carbonyl)-N-[4-(hydroxyamino)phenyl]-N-methylpyrrolidine-2-carboxamide 4-[(5-methylpyridin-3-yl)oxymethyl]-1,2-oxazole 2-[(E)-3-hydroxyprop-1-enyl]-5-methylpyridine-4-carboxylic acid 2-[2-methylbutyl(phenacyl)amino]decanoic acid 1-[(5S)-7-bromo-3,4-dihydro-2H-chromen-5-yl]ethanamine 1-[4-(3,5-dimethylpyridine-2-carbonyl)phenyl]-N-methylcyclopropane-1-carboxamide 2-(5-tert-butylfuran-2-yl)-4,7,8-trimethyl-3H-quinoline 4-[(2S)-5,8-dichloro-6-phenylmethoxy-1,2,3,4-tetrahydronaphthalen-2-yl]-N,N-diethylbutanamide ethane;N'-methyl-4-(2,3,5,6-tetrafluorophenoxy)benzenecarboximidamide N-(2,2-diethoxyethyl)-N-[4-(quinoxalin-2-ylsulfamoyl)phenyl]butanamide 1-(3,5-difluorophenyl)sulfonyl-6-methoxyindole 7-methoxy-N-[(4S,5R)-4-methylazepan-3-yl]quinolin-2-amine;dihydrochloride N-(4,5-dimethyl-2-phenyldiazenylphenyl)-2-methoxy-N-phenacylacetamide 3-(4-methoxyphenyl)-6-methyl-1H-pyrrolo[2,3-b]pyridine 1-azido-2,3-dipropylbenzimidazole (7R)-3-chloro-N-[(2,4-difluorophenyl)methyl]-9-hydroxy-5,6,10,11,15-pentazatetracyclo[8.7.0.02,7.012,17]heptadeca-1(17),2(7),10,12,14,16-hexaene-13-carboxamide 2-azido-3-ethoxy-6,7,8,9-tetrahydropyrido[1,2-a]indole 5-amino-6-[(3,4-difluorophenyl)methylsulfanyl]pyridine-3-carboxylic acid 1-(3,4-dichlorophenyl)-5-imino-4-[4-(3-methylphenyl)-1,3-thiazol-2-yl]-2H-pyrrol-3-amine 2-(1H-indol-3-yl)-N-[(1S,2R,5S)-4-methoxy-6-bicyclo[3.2.0]heptanyl]acetamide N-[1-methylsulfonyl-3-(trifluoromethyl)piperidin-4-yl]-3,7a-dihydroindole-1-carboxamide 3-amino-N,6,6-trimethyl-1-phenylheptan-2-amine N-(3,5-dichlorophenyl)-2-[6-methyl-7-oxo-4-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridin-5-ylidene]acetamide 4-[(1S,2R)-2-azidocyclopropyl]benzenesulfonamide 2-[(5S)-5,6-dimethyl-1H-indol-3-yl]-N-[5-methyl-4-(trifluoromethoxy)thiophen-3-yl]acetamide (3R)-4,5-diamino-1-[2-fluoro-6-methoxy-4-(trifluoromethyl)phenyl]pentan-3-ol 3-(2,6-dimethylphenyl)-8,11,13,15,16-pentazatetracyclo[8.7.0.02,7.012,17]heptadeca-1(10),2,4,6,12(17),13,15-heptaene N-[3-(2,4-difluorophenyl)sulfonylphenyl]carbamate 1-(2,4-dimethylphenyl)sulfanyloctane N-[3-(4-ethylphenoxy)prop-1-en-2-yl]cyclohexanamine 3-[6-(2-aminopropanoyl)oxy-4-methyl-1-phenylcyclohexa-2,4-dien-1-yl]propanoic acid 2-[5-(methylideneamino)pyridin-3-yl]-N-(5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-ylmethyl)aniline 2-[(4R)-6-methylsulfonylspiro[1,3-dihydroisochromene-4,3'-pyrrolidine]-2'-carbonyl]cyclohexane-1-carboxylic acid N-[3-chloro-5-[2-(4-formylpiperazin-1-yl)ethoxy]phenyl]-6,7-dimethoxyquinazoline-4-carboxamide;propane 2,5-dichloro-4-[(Z)-3-[5-methyl-1-(2,2,6,6-tetramethylpiperidin-4-yl)triazol-4-yl]-3-oxoprop-1-enyl]benzaldehyde 2-[(3,4-dichlorophenyl)methyl]-5-propan-2-ylphenol (2S)-N',2-diphenyloctanehydrazide N-[4-(3,6-dimethylimidazo[1,2-b]pyridazin-8-yl)oxyphenyl]-2-thiophen-2-ylacetamide 5-[(2,5-difluoro-4-methylphenyl)methoxy]-1H-indazole 2-[(4-cyclopropylsulfonylphenyl)methoxy]pyridine 2-[2,3-dichloro-4-(1H-imidazol-5-yl)phenyl]acetic acid 2-[1-[4-(dimethylamino)phenyl]ethylamino]benzenecarboximidamide;1,3-xylene 2-(2,4-dioxopyrimidin-1-yl)-N-methoxy-N-phenylacetamide 2-[(3E,5Z)-hepta-1,3,5-trien-4-yl]-N-methoxy-6-methylpyridine-4-carboxamide 4-[3,5-bis(trifluoromethyl)phenyl]-N,6-dimethylpyrimidin-2-amine 7-azido-N-(2-chlorophenyl)quinazolin-4-amine (Z)-N'-hydroxy-4-[6-(methylamino)purin-9-yl]but-2-enimidamide N-[5-(2,4-dioxopyrrolidin-1-yl)pentyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-3-carboxamide (Z)-4-amino-2,7-dimethyl-3-phenyl-6-[1-phenylethyl(pyridine-2-carbonyl)amino]oct-4-enoic acid (1-azidocyclopropyl)methoxymethylbenzene 1,5-bis(2-hydroxynaphthalen-1-yl)naphthalene-2,7,9-trisulfonic acid 2-fluoro-N-[3-[1-(6-methylpyrazin-2-yl)piperidine-4-carbonyl]-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl]benzamide 2-[[6-[3-fluoro-4-(trifluoromethoxy)phenyl]pyrazolo[4,3-b]pyridin-1-yl]methylamino]ethanol 2-[5-methoxycarbonyl-4-oxo-7-[(Z)-2-thiophen-3-ylethenyl]-1,3-benzothiazin-2-yl]acetic acid 7-[3-(aminomethyl)-2H-pyridin-1-yl]quinazolin-4-amine (1E,3Z)-2-cyclopropyl-4-fluorohexa-1,3,5-triene;[(3E)-6-methoxy-5-methylidenehepta-3,6-dien-1-yn-4-yl]benzene N-(1H-benzimidazol-2-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide